10gs A 2.2 BS01 VWW A 1 F8 V10 R13 W38 K44 Q51 L52 Q64 S65 Y108 G205 F7 V9 R12 W37 K43 Q50 L51 Q63 S64 Y107 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=0.4uM remove_due_to_license_issue Ki=420nM P09211 9398518 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 10gs B 2.2 BS01 VWW B 1 F8 V10 R13 W38 K44 Q51 L52 Q64 S65 Y108 G205 F7 V9 R12 W37 K43 Q50 L51 Q63 S64 Y107 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=0.4uM remove_due_to_license_issue Ki=420nM P09211 9398518 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 11gs A 2.3 BS01 GSH A 1 Y7 R13 W38 K44 Q51 L52 Q64 S65 Y6 R12 W37 K43 Q50 L51 Q63 S64 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 9426214 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 11gs A 2.3 BS02 EAA A 1 F8 I104 Y108 G205 F7 I103 Y107 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue IC50=2.6e+4nM P09211 9426214 211 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 11gs B 2.3 BS01 GSH B 1 Y7 R13 W38 K44 Q51 L52 Q64 S65 Y6 R12 W37 K43 Q50 L51 Q63 S64 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 9426214 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 11gs B 2.3 BS02 EAA B 1 F8 I104 Y108 G205 F7 I103 Y107 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue IC50=2.6e+4nM P09211 9426214 211 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 13gs A 1.9 BS02 SAS A 1 F8 P9 V10 R13 V35 I104 Y108 P202 G205 F9 P10 V11 R14 V36 I105 Y109 P203 G206 Y7 R13 Y8 R14 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=24uM remove_due_to_license_issue P09211 10452896 211 MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 16pk A 1.6 BS01 BIS A 1 G217 A218 K223 A242 Y245 L315 P340 G342 V343 E345 G397 G398 G399 G213 A214 K219 A238 Y241 L311 P336 G338 V339 E341 G393 G394 G395 R39 K219 G376 G399 R35 K215 G372 G395 2.7.2.3 0004618,0005524,0005829,0006094,0006096,0016301,0020015,0043531 remove_due_to_license_issue P07378 9642090 499 EKKSINECDLKGKKVLIRVDFNVPVKNGKITNDYRIRSALPTLKKVLTEGGSCVLMSHLGRPKGIPMAQAGKIRSTGGVPGFQQKATLKPVAKRLSELLLRPVTFAPDCLNAADVVSKMSPGDVVLLENVRFYKEEGSKKAKDREAMAKILASYGDVYISDAFGTAHRDSATMTGIPKILGNGAAGYLMEKEISYFAKVLGNPPRPLVAIVGGAKVSDKIQLLDNMLQRIDYLLIGGAMAYTFLKAQGYSIGKSKCEESKLEFARSLLKKAEDRKVQVILPIDHVCHTEFKAVDSPLITEDQNIPEGHMALDIGPKTIEKYVQTIGKCKSAIWNGPMGVFEMVPYSKGTFAIAKAMGRGTHEHGLMSIIGGGDSASAAELSGEAKRMSHVSTGGGASLELLEGKTLPGVTVLDDK 184l A 1.8 BS01 I4B A 1 A99 L118 A99 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Ka=51000M^-1 remove_due_to_license_issue P00720 7612599 401 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 185l A 1.8 BS01 IND A 1 A99 L118 L121 F153 A99 L118 L121 F153 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=289uM remove_due_to_license_issue P00720 7612599 400 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 186l A 1.8 BS01 N4B A 1 A99 V111 L118 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=14uM remove_due_to_license_issue P00720 7612599 400 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 187l A 1.8 BS01 PXY A 1 A99 V111 L118 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=422uM remove_due_to_license_issue Kd=151000nM P00720 7612599 400 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 188l A 1.8 BS01 OXE A 1 A99 V111 L118 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=469uM remove_due_to_license_issue P00720 7612599 400 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 1a0q H 2.3 BS02 HEP H 1 H35 K93 Y96 Y97 H34 K96 Y99 Y100 ? Ki=27nM remove_due_to_license_issue P01869 9753552 214 VQLQESDAELVKPGASVKISCKASGYTFTDHVIHWVKQKPEQGLEWIGYISPGNGDIKYNEKFKGKATLTADKSSSTAYMQLNSLTSEDSAVYLCKRGYYVDYWGQGTTLTVSSAKTTPPSVYPLAPSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIE 1a0q L 2.3 BS02 HEP H 1 Y36 L89 Y91 R96 Y35 L88 Y90 R94 ? 0005576,0005886,0030183 remove_due_to_license_issue P01837 9753552 214 IELTQSPSSLSASLGGKVTITCKASQDIKKYIGWYQHKPGKQPRLLIHYTSTLLPGIPSRFRGSGSGRDYSFSISNLEPEDIATYYCLQYYNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYSKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1a28 A 1.8 BS01 STR A 1 L718 N719 Q725 M759 L797 Y890 C891 L37 N38 Q44 M78 L116 Y209 C210 ? Ki=5.1nM remove_due_to_license_issue Ki=3.5nM, EC50=2.9nM, IC50=>10000nM P06401 9620806 1 QLIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 1a42 A 2.25 BS02 BZU A 1 H94 H96 H119 V121 F131 L198 T199 T200 H91 H93 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 9541386 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1a46 H 2.12 BS03 00K H 1 H57 Y60A W60D L99 E192 G193 S195 W215 G216 G219 H43 Y47 W50 L96 E194 G195 S197 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10212123 372 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1a4g A 2.2 BS02 ZMR A 1 R115 E116 D148 R149 W176 A244 E274 R291 R373 Y408 R40 E41 D73 R74 W101 A169 E199 R216 R298 Y333 D148 E275 R291 R373 Y408 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.004uM remove_due_to_license_issue P27907 9526556 466 EPEWTYPRLSCQGSTFQKALLISPHRFGEARGNSAPLIIREPFIACGPKECKHFALTHYAAQPGGYYNGTREDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDSNALIKIKYGEAYTDTYHSYANNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEIFPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTETYLDTPRPDDGSITGPCESNGDKGRGGIKGGFVHQRMASKIGRWYSRTMSKTERMGMELYVRYDGDPWTDSDALAHSGVMVSMKEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKKTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1a4h A 2.5 BS01 GDM A 1 N37 D40 A41 K44 D79 N92 K98 G121 V122 F124 N37 D40 A41 K44 D79 N92 K98 G121 V122 F124 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 9230303 300 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 1a4k B 2.4 BS01 FRA B 1 N31 G33 N35 W50 A95 E96 R97 N31 G33 N35 W50 A99 E100 R101 Kd=0.01uM remove_due_to_license_issue 9506942 3083 QVQLLESGPELKKPGETVKISCKASGYTFTNYGMNWVKQAPGKGLKWMGWINTYTGEPTYADDFKGRFAFSLETSASTAYLQINNLKNEDTATYFCVQAERLRRTFDYWGAGTTVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 1a4m A 1.95 BS02 PRH A 1 H17 D19 F61 L62 F65 M155 G184 H214 E217 D295 D296 H14 D16 F58 L59 F62 M152 G181 H211 E214 D292 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0000255,0001666,0001701,0001829,0001889,0001890,0002314,0002467,0002636,0002686,0002901,0002906,0004000,0005737,0005764,0005829,0005886,0006154,0006157,0006196,0006915,0006939,0007155,0008270,0009117,0009168,0009897,0009986,0010460,0014074,0016020,0016787,0019239,0019722,0030217,0030324,0030890,0031410,0032261,0032263,0032264,0033077,0033089,0033632,0042100,0042110,0043066,0043084,0043605,0044209,0045580,0045582,0045987,0046059,0046061,0046085,0046101,0046103,0046111,0046632,0046638,0046872,0046936,0048286,0048541,0048566,0050728,0050850,0050852,0050862,0050870,0050900,0060169,0060205,0060407,0070161,0070242,0070244,0070254,0070256,0140928 Ki~0.1pM remove_due_to_license_issue P03958 9622483 354 TPAFNKPKVELHVHLDGAIKPETILYFGKKRGIALPADTVEELRNIIGMDKPLSLPGFLAKFDYYMPVIAGCREAIKRIAYEFVEMKAKEGVVYVEVRYSPHLLANSKVDPMPWNQTEGDVTPDDVVDLVNQGLQEGEQAFGIKVRSILCCMRHQPSWSLEVLELCKKYNQKTVVAMDLAGDETIEGSSLFPGHVEAYEGAVKNGIHRTVHAGEVGSPEVVREAVDILKTERVGHGYHTIEDEALYNRLLKENMHFEVCPWSSYLTGAWDPKTTHAVVRFKNDKANYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEEEKKELLERLYREYQ 1a4q A 1.9 BS02 DPC A 1 R115 E116 D148 W176 I220 R222 A244 E274 E275 R291 N293 R373 Y408 R40 E41 D73 W101 I145 R147 A169 E199 E200 R216 N218 R298 Y333 D148 E275 R291 R373 Y408 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=3.6uM remove_due_to_license_issue P27907 9526556 466 EPEWTYPRLSCQGSTFQKALLISPHRFGEARGNSAPLIIREPFIACGPKECKHFALTHYAAQPGGYYNGTREDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDSNALIKIKYGEAYTDTYHSYANNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEIFPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTETYLDTPRPDDGSITGPCESNGDKGRGGIKGGFVHQRMASKIGRWYSRTMSKTERMGMELYVRYDGDPWTDSDALAHSGVMVSMKEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKKTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1a4r B 2.5 BS01 GNH B 1 A213 G215 K216 T217 C218 F228 Q316 D318 L319 S358 A359 L360 A13 G15 K16 T17 C18 F28 Q116 D118 L119 S158 A159 L160 3.6.5.2 0000139,0000322,0002040,0003015,0003161,0003253,0003924,0003925,0005515,0005525,0005737,0005789,0005813,0005819,0005829,0005856,0005886,0005911,0005925,0006897,0006911,0007015,0007030,0007088,0007097,0007163,0007229,0007264,0007399,0008104,0009653,0010591,0010592,0016020,0016787,0017119,0019901,0021762,0030010,0030036,0030141,0030154,0030175,0030225,0030307,0030335,0030425,0030496,0030742,0031252,0031256,0031274,0031333,0031435,0031996,0032427,0032467,0032488,0032956,0032991,0034191,0034329,0034332,0035050,0035088,0036336,0036464,0038189,0042802,0042995,0043005,0043025,0043197,0043410,0043525,0044788,0045177,0045198,0045335,0045740,0046330,0046847,0048549,0048664,0051130,0051233,0051489,0051491,0051492,0051496,0051647,0051649,0051683,0051835,0051897,0051988,0060047,0060071,0060501,0060661,0060997,0061630,0070062,0071346,0071944,0072384,0072686,0086101,0090135,0090316,0098685,0098794,0098978,0099159,0099175,1900026,1990606 Kd=0.22uM remove_due_to_license_issue P60953 10211824 400 MQTIKCVVVGDVAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAGQEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLRDDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPPEPKKSRRCVL 1a4w H 1.8 BS03 QWE H 1 Y60A W60D K60F L99 D189 A190 C191 W215 G216 G219 Y47 W50 K52 L96 D191 A192 C193 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 Ki=1.2uM remove_due_to_license_issue P00734 8913620 373 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 1a50 A 2.3 BS01 FIP A 1 F22 D60 L100 Y175 T183 F212 G213 G234 S235 F21 D59 L99 Y174 T182 F205 G206 G227 S228 E49 D60 Y102 Y173 Y175 T183 S233 G234 S235 E48 D59 Y101 Y172 Y174 T182 S226 G227 S228 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 Kd=0.35uM remove_due_to_license_issue P00929 9548921 270 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1a52 A 2.8 BS01 EST A 1 E353 L387 M388 L391 F404 H524 L525 E48 L82 M83 L86 F99 H219 L220 ? remove_due_to_license_issue IC50=1.3nM, Kd=0.2nM, EC50=0.75nM, Ki=0.21nM P03372 9600906 1 LALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHERLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEML 1a5g H 2.06 BS03 00L H 1 L41 H57 Y60A W60D I174 D189 A190 E192 G193 S195 W215 G216 L27 H43 Y47 W50 I171 D191 A192 E194 G195 S197 W219 G220 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10212123 372 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1a5h A 2.9 BS02 BBA A 1 D97 T98 Y99 D189 A190 Q192 I213 W215 G216 G219 D91 T92 Y93 D197 A198 Q200 I221 W223 G224 G226 H57 D102 G193 S195 H47 D96 G201 S203 3.4.21.68 0004252,0006508 remove_due_to_license_issue P00750 9268299 250 IKGGLFADIASHPWQAAIFAKHRRSPGERFLCGGILISSCWILSAAHCFQERFPPHHLTVILGRTYRVVPGEEEQKFEVEKYIVHKEFDDDTYDNDIALLQLKSDSSRCAQESSVVRTVCLPPADLQLPDWTECELSGYGKHEALSPFYSERLKEAHVRLYPSSRCTSQHLLNRTVTDNMLCAGDTRSGGPQANLHDACQGDSGGPLVCLNDGRMTLVGIISWGLGCGQKDVPGVYTKVTNYLDWIRDNMRP 1a5v A 1.9 BS02 Y3 A 1 Q62 A154 M155 Q9 A101 M102 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0015074 ic50=800uM remove_due_to_license_issue O92956 9560188 1 GLGPLQIWQTDFTLEPRMAPRSWLAVTVDTASSAIVVTQHGRVTSVAAQHHWATAIAVLGRPKAIKTDNGSCFTSKSTREWLARWGIAHTTGIPGNSQGQAMVERANRLLKDKIRVLAEGDGFMKRIPTSKQGELLAKAMYALNHF 1a61 H 2.2 BS03 00N H 1 H57 Y60A W60D D189 G193 D194 S195 W215 G216 H43 Y47 W50 D191 G195 D196 S197 W219 G220 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10212123 372 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1a69 A 2.1 BS01 FMB A 1 M64 S90 C91 G92 F159 V178 E179 M180 E181 D204 M64 S90 C91 G92 F159 V178 E179 M180 E181 D204 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0006974,0009116,0009164,0016020,0016757,0016763,0019686,0042278,0042802,0047975 Ki=5uM remove_due_to_license_issue P0ABP8 9653038 240 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHIRTHEQTTAAERQTTFNDMIKIALESVLLGDK 1a69 C 2.1 BS01 FMB C 1 S90 C91 G92 F159 V178 M180 E181 D204 S90 C91 G92 F159 V178 M180 E181 D204 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R213 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0006974,0009116,0009164,0016020,0016757,0016763,0019686,0042278,0042802,0047975 Ki=5uM remove_due_to_license_issue P0ABP8 9653038 240 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHIRTTAAERQTTFNDMIKIALESVLLGDK 1a7x A 2.0 BS01 FKA B 1 E54 D79 A81 Y82 E54 D79 A81 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 remove_due_to_license_issue P62942 9871618 201 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1a7x B 2.0 BS01 FKA B 1 Y26 D37 F46 Q53 E54 V55 I56 W59 Y82 F99 Y26 D37 F46 Q53 E54 V55 I56 W59 Y82 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Kd=0.2nM remove_due_to_license_issue P62942 9871618 201 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1a85 A 2.0 BS05 0DY A 1 I159 L160 A161 L193 H197 E198 H201 H207 L214 Y216 N218 Y219 I75 L76 A77 L109 H113 E114 H117 H123 L130 Y132 N134 Y135 H197 E198 H201 H207 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=26000nM P22894 9655333 1 NPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1a86 A 2.0 BS01 0ZB A 1 I159 L160 A161 H197 E198 H201 H207 L214 Y216 N218 Y219 I75 L76 A77 H113 E114 H117 H123 L130 Y132 N134 Y135 H197 E198 H201 H207 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=88000nM P22894 9655333 1 NPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1a8i A 1.78 BS01 GLS A 1 G135 L136 N284 H377 V455 N484 E672 S674 G675 G129 L130 N268 H355 V433 N462 E650 S652 G653 H377 K568 R569 K574 T676 K680 H355 K546 R547 K552 T654 K658 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=3uM remove_due_to_license_issue Ki=3100nM, IC50=3100nM P00489 9568898 998 QEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 1a8t A 2.55 BS03 061 A 1 I29 W32 V35 H145 C164 D168 N176 H206 G207 I29 W32 V35 H145 C164 D168 N176 H206 G207 H82 H84 D86 H145 C164 K167 N176 H206 H82 H84 D86 H145 C164 K167 N176 H206 3.5.2.6 0008270,0008800,0017001 remove_due_to_license_issue P25910 9545432 250 AQKSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTS 1a94 A 2.0 BS01 0Q4 A 1 R8 G27 A28 D29 D30 I47 G48 P81 R8 G27 A28 D29 D30 I47 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=14nM remove_due_to_license_issue P03367 9521772 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWEPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1a94 B 2.0 BS01 0Q4 A 1 D25 G27 A28 D29 G48 V82 I84 D25 G27 A28 D29 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 9521772 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWEPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1a99 A 2.2 BS01 PUT A 1 W37 S38 Y40 W244 D247 F276 D278 Y314 W9 S10 Y12 W216 D219 F248 D250 Y286 ? 0015846,0015847,0016020,0019808,0019810,0030288,0042597,0055052 Kd=2uM remove_due_to_license_issue P31133 9651355 371 QKTLHIYNWSDYIAPDTVANFEKETGIKVVYDVFDSNEVLEGKLMAGSTGFDLVVPSASFLERQLTAGVFQPLDKSKLPEWKNLDPELLKLVAKHDPDNKFAMPYMWATTGIGYNVDKVKAVLGENAPVDSWDLILKPENLEKLKSCGVSFLDAPEEVFATVLNYLGKDPNSTKADDYTGPATDLLLKLRPNIRYFHSSQYINDLANGDICVAIGWAGDVWQASNRAKEAKNGVNVSFSIPKEGAMAFFDVFAMPADAKNKDEAYQFLNYLLRPDVVAHISDHVFYANANKAATPLVSAEVRENPGIYPPADVRAKLFTLKVQDPKIDRVRTRAWTKVKSG 1a9m A 2.3 BS01 U0E B 1 R8 D25 G49 I84 R8 D25 G49 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9450540 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIHGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1a9m B 2.3 BS01 U0E B 1 D25 G27 A28 D29 D30 I47 H48 I50 V82 D25 G27 A28 D29 D30 I47 H48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=119nM remove_due_to_license_issue P03366 9450540 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIHGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1a9q A 2.0 BS01 HPA A 1 A117 G118 F200 E201 M219 N243 A117 G118 F200 E201 M219 N243 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 remove_due_to_license_issue Kd=680nM P55859 9585525 290 MQNGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGENPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDTESQGKANHEEVLEAGKQAAQKLEQFVSLLMASI 1a9u A 2.5 BS01 SB2 A 1 Y35 A51 K53 L104 V105 T106 M109 R173 Y32 A48 K50 L101 V102 T103 M106 R170 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 9753691 800 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1aaq A 2.5 BS01 PSI B 1 R8 D25 G27 A28 D29 G48 R8 D25 G27 A28 D29 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 1637805 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1aaq B 2.5 BS01 PSI B 1 D25 G27 A28 D29 I47 G48 P81 V82 D25 G27 A28 D29 I47 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3nM remove_due_to_license_issue P03367 1637805 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1abf A 1.9 BS01 FCA A 1 K10 E14 W16 D90 R151 M204 N205 N232 K9 E13 W15 D89 R150 M203 N204 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=3.8uM remove_due_to_license_issue P02924 2818726 307 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMMAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 1acj A 2.8 BS01 THA A 1 W84 G118 E199 F330 W432 H440 W81 G115 E196 F327 W429 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue IC50=29nM, Ki=40nM P04058 8415649 999 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1ad8 H 2.0 BS03 MDL H 1 H57 Y60A I174 A190 C191 E192 G193 S195 W215 G216 G226 H43 Y47 I172 A193 C194 E195 G196 S198 W220 G221 G231 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 9033393 250 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1add A 2.4 BS02 1DA A 1 H17 D19 F61 F65 M155 G184 E217 D296 H14 D16 F58 F62 M152 G181 E214 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0000255,0001666,0001701,0001829,0001889,0001890,0002314,0002467,0002636,0002686,0002901,0002906,0004000,0005737,0005764,0005829,0005886,0006154,0006157,0006196,0006915,0006939,0007155,0008270,0009117,0009168,0009897,0009986,0010460,0014074,0016020,0016787,0019239,0019722,0030217,0030324,0030890,0031410,0032261,0032263,0032264,0033077,0033089,0033632,0042100,0042110,0043066,0043084,0043605,0044209,0045580,0045582,0045987,0046059,0046061,0046085,0046101,0046103,0046111,0046632,0046638,0046872,0046936,0048286,0048541,0048566,0050728,0050850,0050852,0050862,0050870,0050900,0060169,0060205,0060407,0070161,0070242,0070244,0070254,0070256,0140928 Ki=0.18uM remove_due_to_license_issue P03958 8439534 353 TPAFNKPKVELHVHLDGAIKPETILYFGKKRGIALPADTVEELRNIIGMDKPLSLPGFLAKFDYYMPVIAGCREAIKRIAYEFVEMKAKEGVVYVEVRYSPHLLANSKVDPMPWNQTEGDVTPDDVVDLVNQGLQEGEQAFGIKVRSILCCMRHQPSWSLEVLELCKKYNQKTVVAMDLAGDETIEGSSLFPGHVEAYEGAVKNGIHRTVHAGEVGSPEVVREAVDILKTERVGHGYHTIEDEALYNRLLKENMHFEVCPWSSYLTGAWDPKTTHAVVRFKNDKANYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEEEKKELLERLYREYQ 1adl A 1.6 BS01 ACD A 1 T29 A33 D76 R126 Y128 T29 A33 D76 R126 Y128 ? 0005324,0005634,0005654,0005737,0008289,0009617,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0071285,0071356,0120162 Kd=4.4uM remove_due_to_license_issue P04117 7929228 135 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDLVTIRSESTFKNTEISFKLGVEFDEITADDRKVKSIITLDGGALVQVQKWDGKSTTIKRKRDGDKLVVECVMKGVTSTRVYERA 1af2 A 2.3 BS02 U A 1 N89 E91 H102 E104 P128 C129 N89 E91 H102 E104 P128 C129 H102 E104 C129 C132 H102 E104 C129 C132 3.5.4.5 0001884,0003824,0004126,0005737,0005829,0006217,0008270,0009972,0015949,0016787,0042802,0042803,0046872,0055086,0072527,1901135 remove_due_to_license_issue P0ABF6 9125497 295 MHPRFQTAFAQLADNLQSALEPILADKYFPALLTGEQVSSLKSATGLDEDALAFALLPLAAACARTPLSNFNVGAIARGVSGTWYFGANMEFIGATMQQTVHAEQSAISHAWLSGEKALAAITVNYTPCGHCRQFMNELNSGLDLRIHLPGREAHALRDYLPDAFGPKDLEIKTLLMDEQDHGYALTGDALSQAAIAAANRSHMPYSKSPSGVALECKDGRIFSGSYAENAAFNPTLPPLQGALILLNLKGYDYPDIQRAVLAEKADAPLIQWDATSATLKALGCHSIDRVLLA 1af6 A 2.4 BS01 GLC D 1 R8 Y41 E43 R82 R109 D116 Y118 R8 Y41 E43 R82 R109 D116 Y118 ? 0001618,0005363,0005515,0006811,0006974,0009279,0015144,0015288,0015768,0015774,0016020,0034219,0042956,0042958,0046718,0046930,0106234,1904981 remove_due_to_license_issue P02943 9299337 1 VDFHGYARSGIGWTGSGGEQQCFQTTGAQSKYRLGNECETYAELKLGQEVWKEGDKSFYFDTNVAYSVAQQNDWEATDPAFREANVQGKNLIEWLPGSTIWAGKRFYQRHDVHMIDFYYWDISGPGAGLENIDVGFGKLSLAATRSSEAGGSSSFASNNIYDYTNETANDVFDVRLAQMEINPGGTLELGVDYGRANLRDNYRLVDGASKDGWLFTAEHTQSVLKGFNKFVVQYATDSMTSQGKGLSQGSGVAFDNEKFAYNINNNGHMLRILDHGAISMGDNWDMMYVGMYQDINWDNDNGTKWWTVGIRPMYKWTPIMSTVMEIGYDNVESQRTGDKNNQYKITLAQQWQAGDSIWSRPAIRVFATYAKWDEKWGYDYTGNADNNANFGKAVPADFNGGSFGRGDSDEWTFGAQMEIWW 1af6 B 2.4 BS01 GLC E 1 R8 Y41 E43 R109 D116 Y118 R8 Y41 E43 R109 D116 Y118 ? 0001618,0005363,0005515,0006811,0006974,0009279,0015144,0015288,0015768,0015774,0016020,0034219,0042956,0042958,0046718,0046930,0106234,1904981 remove_due_to_license_issue P02943 9299337 1 VDFHGYARSGIGWTGSGGEQQCFQTTGAQSKYRLGNECETYAELKLGQEVWKEGDKSFYFDTNVAYSVAQQNDWEATDPAFREANVQGKNLIEWLPGSTIWAGKRFYQRHDVHMIDFYYWDISGPGAGLENIDVGFGKLSLAATRSSEAGGSSSFASNNIYDYTNETANDVFDVRLAQMEINPGGTLELGVDYGRANLRDNYRLVDGASKDGWLFTAEHTQSVLKGFNKFVVQYATDSMTSQGKGLSQGSGVAFDNEKFAYNINNNGHMLRILDHGAISMGDNWDMMYVGMYQDINWDNDNGTKWWTVGIRPMYKWTPIMSTVMEIGYDNVESQRTGDKNNQYKITLAQQWQAGDSIWSRPAIRVFATYAKWDEKWGYDYTGNADNNANFGKAVPADFNGGSFGRGDSDEWTFGAQMEIWW 1afk A 1.7 BS01 PAP A 1 K7 Q11 H12 C65 N67 Q69 N71 A109 E111 V118 H119 K7 Q11 H12 C65 N67 Q69 N71 A109 E111 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=240nM remove_due_to_license_issue P61823 9154942 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1afl A 1.7 BS01 ATR A 1 K7 H12 C65 N67 Q69 N71 A109 E111 V118 H119 K7 H12 C65 N67 Q69 N71 A109 E111 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=520nM remove_due_to_license_issue P61823 9154942 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1ag9 A 1.8 BS02 FMN A 1 S10 D11 T12 N14 T15 P55 T56 W57 Y58 Y59 C88 G89 D90 Y94 Y97 F98 D147 S9 D10 T11 N13 T14 P54 T55 W56 Y57 Y58 C87 G88 D89 Y93 Y96 F97 D146 ? 0000166,0005515,0005737,0005829,0009055,0010181 Kd=1nM remove_due_to_license_issue P61949 9416602 177 AITGIFFGSDTGNTENIAKMIQKQLGKDVADVHDIAKSSKEDLEAYDILLLGIPTWYYGEAQCDWDDFFPTLEEIDFNGKLVALFGCGDQEDYAEYFCDALGTIRDIIEPRGATIVGHWPTAGYHFEASKGLADDDHFVGLAIDEDRQPELTAERVEKWVKQISEELHLDEILNA 1ag9 B 1.8 BS02 FMN B 1 S10 D11 T12 G13 N14 T15 P55 T56 W57 Y58 Y59 C88 G89 D90 Y94 Y97 F98 D147 S9 D10 T11 G12 N13 T14 P54 T55 W56 Y57 Y58 C87 G88 D89 Y93 Y96 F97 D146 ? 0000166,0005515,0005737,0005829,0009055,0010181 Kd=1nM remove_due_to_license_issue P61949 9416602 177 AITGIFFGSDTGNTENIAKMIQKQLGKDVADVHDIAKSSKEDLEAYDILLLGIPTWYYGEAQCDWDDFFPTLEEIDFNGKLVALFGCGDQEDYAEYFCDALGTIRDIIEPRGATIVGHWPTAGYHFEASKGLADDDHFVGLAIDEDRQPELTAERVEKWVKQISEELHLDEILNA 1agw A 2.4 BS01 SU2 A 1 L484 A512 V561 E562 Y563 A564 S565 K566 G567 L630 L21 A40 V89 E90 Y91 A92 S93 K94 G95 L146 D623 A625 R627 N628 D641 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 9139660 1001 ELPEDPRWELPRDRLVLGKPLGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS 1aht H 1.6 BS03 APA H 1 H57 D189 A190 C191 E192 G193 S195 V213 W215 H43 D192 A193 C194 E195 G196 S198 V218 W220 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 7574675 401 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1ahx A 2.0 BS02 HCI A 1 I17 L18 G38 W140 K258 R386 I13 L14 G34 W130 K246 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=120uM remove_due_to_license_issue P00509 7664122 411 MFENITAAPADPILGLADLFRADERPGKINLGIGLYYDETGKIPVLTSVKKAEQYLLENETTKLYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFGLYNERVGACTLVAADSETVDRAFSQMKAAIRANYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1ahx B 2.0 BS02 HCI B 1 I17 L18 I37 G38 W140 K258 R386 I13 L14 I33 G34 W130 K246 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=120uM remove_due_to_license_issue P00509 7664122 411 MFENITAAPADPILGLADLFRADERPGKINLGIGLYYDETGKIPVLTSVKKAEQYLLENETTKLYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFGLYNERVGACTLVAADSETVDRAFSQMKAAIRANYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1ai4 B 2.35 BS02 DHY B 1 S1 F24 S67 A69 S1 F24 S67 A69 S1 Q23 A69 F71 N241 S1 Q23 A69 F71 N241 3.5.1.11 0016787,0017000 Ki=3.13mM remove_due_to_license_issue P06875 9813130 559 SNMWVIGKSKAQDAKAIMVNGPQFGWYAPAYTYGIGLHGAGYDVTGNTPFAYPGLVFGHNGVISWGSTAGFGDDVDIFAERLSAEKPGYYLHNGKWVKMLSREETITVKNGQAETFTVWRTVHGNILQTDQTTQTAYAKSRAWDGKEVASLLAWTHQMKAKNWQQWTQQAAKQALTINWYYADVNGNIGYVHTGAYPDRQSGHDPRLPVPGTGKWDWKGLLPFEMNPKVYNPQSGYIANWNNSPQKDYPASDLFAFLWGGADRVTEIDRLLEQKPRLTADQAWDVIRQTSRQDLNLRLFLPTLQAATSGLTQSDPRRQLVETLTRWDGINLLNDDGKTWQQPGSAILNVWLTSMLKRTVVAAVPMPFDKWYSASGYETTQDGPTGSLNISVGAKILYEAVQGDKSPIPQAVDLFAGKPQQEVVLAALEDTWETLSKRYGNNVSNWKTPAMALTFRANNFFGVPQAAAEETRHQAEYQNRGTENDMIVFSPTTSDRPVLAWDVVAPGQSGFIAPDGTVDKHYEDQLKMYENFGRKSLWLTKQDVEAHKESQEVLHVQR 1ai5 B 2.36 BS02 MNP B 1 S1 P22 F24 S67 A69 S1 P22 F24 S67 A69 S1 Q23 A69 F71 N241 S1 Q23 A69 F71 N241 3.5.1.11 0016787,0017000 Ki=0.189mM remove_due_to_license_issue P06875 9813130 559 SNMWVIGKSKAQDAKAIMVNGPQFGWYAPAYTYGIGLHGAGYDVTGNTPFAYPGLVFGHNGVISWGSTAGFGDDVDIFAERLSAEKPGYYLHNGKWVKMLSREETITVKNGQAETFTVWRTVHGNILQTDQTTQTAYAKSRAWDGKEVASLLAWTHQMKAKNWQQWTQQAAKQALTINWYYADVNGNIGYVHTGAYPDRQSGHDPRLPVPGTGKWDWKGLLPFEMNPKVYNPQSGYIANWNNSPQKDYPASDLFAFLWGGADRVTEIDRLLEQKPRLTADQAWDVIRQTSRQDLNLRLFLPTLQAATSGLTQSDPRRQLVETLTRWDGINLLNDDGKTWQQPGSAILNVWLTSMLKRTVVAAVPMPFDKWYSASGYETTQDGPTGSLNISVGAKILYEAVQGDKSPIPQAVDLFAGKPQQEVVLAALEDTWETLSKRYGNNVSNWKTPAMALTFRANNFFGVPQAAAEETRHQAEYQNRGTENDMIVFSPTTSDRPVLAWDVVAPGQSGFIAPDGTVDKHYEDQLKMYENFGRKSLWLTKQDVEAHKESQEVLHVQR 1ai6 B 2.55 BS02 4HP B 1 S1 F24 S67 T68 A69 S1 F24 S67 T68 A69 S1 Q23 A69 F71 N241 S1 Q23 A69 F71 N241 3.5.1.11 0016787,0017000 remove_due_to_license_issue P06875 9813130 559 SNMWVIGKSKAQDAKAIMVNGPQFGWYAPAYTYGIGLHGAGYDVTGNTPFAYPGLVFGHNGVISWGSTAGFGDDVDIFAERLSAEKPGYYLHNGKWVKMLSREETITVKNGQAETFTVWRTVHGNILQTDQTTQTAYAKSRAWDGKEVASLLAWTHQMKAKNWQQWTQQAAKQALTINWYYADVNGNIGYVHTGAYPDRQSGHDPRLPVPGTGKWDWKGLLPFEMNPKVYNPQSGYIANWNNSPQKDYPASDLFAFLWGGADRVTEIDRLLEQKPRLTADQAWDVIRQTSRQDLNLRLFLPTLQAATSGLTQSDPRRQLVETLTRWDGINLLNDDGKTWQQPGSAILNVWLTSMLKRTVVAAVPMPFDKWYSASGYETTQDGPTGSLNISVGAKILYEAVQGDKSPIPQAVDLFAGKPQQEVVLAALEDTWETLSKRYGNNVSNWKTPAMALTFRANNFFGVPQAAAEETRHQAEYQNRGTENDMIVFSPTTSDRPVLAWDVVAPGQSGFIAPDGTVDKHYEDQLKMYENFGRKSLWLTKQDVEAHKESQEVLHVQR 1aid A 2.2 BS01 THK B 1 D30 V32 I47 T80 I84 D30 V32 I47 T80 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 8340363 201 PQITLWQRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1aid B 2.2 BS01 THK B 1 I47 I50 T80 I47 I50 T80 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=15uM remove_due_to_license_issue P03369 8340363 201 PQITLWQRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1aj6 A 2.3 BS01 NOV A 1 N46 R76 I78 P79 I94 N35 R65 I67 P68 I78 5.6.2.2 0003677,0003918,0005524,0006265 Kd=1.2uM remove_due_to_license_issue IC50=170nM, Kd=7.0nM, Ki=7.0nM P0AES6 9245398 1 VLKGLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIVSAAEVIMTVLHAGGKFSGGLHGVGVSVVNALSQKLELVIQHEGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFH 1aj7 H 2.1 BS01 NPE H 1 Y33 H35 Y99 G100 W103 Y33 H35 Y100 G101 W104 ? Kd=135uM remove_due_to_license_issue P01857 9180069 217 QVQLQQSGAELVKPGASVKLSCTASGFNIKDTYMHWVKQRPEQGLEWIGRIDPANGNTKYDPKFQGKATITADTSSNTAYLQLSSLTSEDTAVYYCASYYGIYWGQGTTLTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 1aj7 L 2.1 BS01 NPE H 1 L89 Y94 R96 F98 L89 Y94 R96 F98 remove_due_to_license_issue 9180069 217 DIQMTQSPSSLSASLGERVSLTCRASQEISGYLSWLQQKPDGTIKRLIYAASTLDSGVPKRFSGSRSGSDYSLTISSLESEDFADYYCLQYASYPRTFGGGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 1ajn B 2.36 BS02 AAN B 1 S1 F24 S67 A69 S1 F24 S67 A69 S1 Q23 A69 F71 N241 S1 Q23 A69 F71 N241 3.5.1.11 0016787,0017000 Ki=2.32mM remove_due_to_license_issue P06875 9813130 559 SNMWVIGKSKAQDAKAIMVNGPQFGWYAPAYTYGIGLHGAGYDVTGNTPFAYPGLVFGHNGVISWGSTAGFGDDVDIFAERLSAEKPGYYLHNGKWVKMLSREETITVKNGQAETFTVWRTVHGNILQTDQTTQTAYAKSRAWDGKEVASLLAWTHQMKAKNWQQWTQQAAKQALTINWYYADVNGNIGYVHTGAYPDRQSGHDPRLPVPGTGKWDWKGLLPFEMNPKVYNPQSGYIANWNNSPQKDYPASDLFAFLWGGADRVTEIDRLLEQKPRLTADQAWDVIRQTSRQDLNLRLFLPTLQAATSGLTQSDPRRQLVETLTRWDGINLLNDDGKTWQQPGSAILNVWLTSMLKRTVVAAVPMPFDKWYSASGYETTQDGPTGSLNISVGAKILYEAVQGDKSPIPQAVDLFAGKPQQEVVLAALEDTWETLSKRYGNNVSNWKTPAMALTFRANNFFGVPQAAAEETRHQAEYQNRGTENDMIVFSPTTSDRPVLAWDVVAPGQSGFIAPDGTVDKHYEDQLKMYENFGRKSLWLTKQDVEAHKESQEVLHVQR 1ajp B 2.31 BS01 OMD A 1 S1 P22 S67 T68 A69 S1 P22 S67 T68 A69 S1 Q23 A69 F71 N241 S1 Q23 A69 F71 N241 3.5.1.11 0016787,0017000 remove_due_to_license_issue P06875 9813130 210 SNMWVIGKSKAQDAKAIMVNGPQFGWYAPAYTYGIGLHGAGYDVTGNTPFAYPGLVFGHNGVISWGSTAGFGDDVDIFAERLSAEKPGYYLHNGKWVKMLSREETITVKNGQAETFTVWRTVHGNILQTDQTTQTAYAKSRAWDGKEVASLLAWTHQMKAKNWQQWTQQAAKQALTINWYYADVNGNIGYVHTGAYPDRQSGHDPRLPVPGTGKWDWKGLLPFEMNPKVYNPQSGYIANWNNSPQKDYPASDLFAFLWGGADRVTEIDRLLEQKPRLTADQAWDVIRQTSRQDLNLRLFLPTLQAATSGLTQSDPRRQLVETLTRWDGINLLNDDGKTWQQPGSAILNVWLTSMLKRTVVAAVPMPFDKWYSASGYETTQDGPTGSLNISVGAKILYEAVQGDKSPIPQAVDLFAGKPQQEVVLAALEDTWETLSKRYGNNVSNWKTPAMALTFRANNFFGVPQAAAEETRHQAEYQNRGTENDMIVFSPTTSDRPVLAWDVVAPGQSGFIAPDGTVDKHYEDQLKMYENFGRKSLWLTKQDVEAHKESQEVLHVQR 1ajq B 2.05 BS02 SPA B 1 S1 F24 S67 A69 S1 F24 S67 A69 S1 Q23 A69 F71 N241 S1 Q23 A69 F71 N241 3.5.1.11 0016787,0017000 Ki=0.049mM remove_due_to_license_issue P06875 9813130 559 SNMWVIGKSKAQDAKAIMVNGPQFGWYAPAYTYGIGLHGAGYDVTGNTPFAYPGLVFGHNGVISWGSTAGFGDDVDIFAERLSAEKPGYYLHNGKWVKMLSREETITVKNGQAETFTVWRTVHGNILQTDQTTQTAYAKSRAWDGKEVASLLAWTHQMKAKNWQQWTQQAAKQALTINWYYADVNGNIGYVHTGAYPDRQSGHDPRLPVPGTGKWDWKGLLPFEMNPKVYNPQSGYIANWNNSPQKDYPASDLFAFLWGGADRVTEIDRLLEQKPRLTADQAWDVIRQTSRQDLNLRLFLPTLQAATSGLTQSDPRRQLVETLTRWDGINLLNDDGKTWQQPGSAILNVWLTSMLKRTVVAAVPMPFDKWYSASGYETTQDGPTGSLNISVGAKILYEAVQGDKSPIPQAVDLFAGKPQQEVVLAALEDTWETLSKRYGNNVSNWKTPAMALTFRANNFFGVPQAAAEETRHQAEYQNRGTENDMIVFSPTTSDRPVLAWDVVAPGQSGFIAPDGTVDKHYEDQLKMYENFGRKSLWLTKQDVEAHKESQEVLHVQR 1ajv A 2.0 BS01 NMB A 1 L23 D25 G27 A28 G49 I50 V82 I84 L23 D25 G27 A28 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=19.1nM remove_due_to_license_issue P03366 9083478 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ajv B 2.0 BS01 NMB A 1 D25 G27 A28 D30 V32 G49 I50 P81 D25 G27 A28 D30 V32 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9083478 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ajx A 2.0 BS01 AH1 A 1 D25 G27 A28 I50 P81 V82 D25 G27 A28 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=12.2nM remove_due_to_license_issue P03366 9083478 500 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ajx B 2.0 BS01 AH1 A 1 R8 L23 D25 G27 A28 G49 I50 R8 L23 D25 G27 A28 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9083478 500 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1akq A 1.9 BS01 FMN A 1 S10 T11 T12 N14 T15 S58 T59 W60 D62 C93 G94 A95 Y98 Y100 F101 S9 T10 T11 N13 T14 S57 T58 W59 D61 C92 G93 A94 Y97 Y99 F100 ? 0009055,0010181 Kd=0.79nM remove_due_to_license_issue P00323 12206666 149 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWGDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGASSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1akr A 1.58 BS01 FMN A 1 S10 T11 T12 G13 N14 T15 S58 T59 W60 A61 C93 G94 D95 Y98 F101 S9 T10 T11 G12 N13 T14 S57 T58 W59 A60 C92 G93 D94 Y97 F100 ? 0009055,0010181 Kd=0.82nM remove_due_to_license_issue P00323 9622492 149 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWADDSIELQDDFIPLFDSLEETGAQGRKVACFGCGDSSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1akt A 1.8 BS01 FMN A 1 S10 T11 T12 G13 N14 T15 S58 T59 W60 N61 C93 G94 D95 Y98 Y100 F101 S9 T10 T11 G12 N13 T14 S57 T58 W59 N60 C92 G93 D94 Y97 Y99 F100 ? 0009055,0010181 Kd=3.2nM remove_due_to_license_issue P00323 9622492 149 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWNDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGDSSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1aku A 1.9 BS01 FMN A 1 S10 T11 T12 N14 T15 S58 T59 W60 G61 C93 G94 A95 Y98 Y100 F101 S9 T10 T11 N13 T14 S57 T58 W59 G60 C92 G93 A94 Y97 Y99 F100 ? 0009055,0010181 Kd=746nM remove_due_to_license_issue P00323 12206666 150 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWGDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGASSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1akv A 2.0 BS01 FMN A 1 S10 T11 T12 N14 T15 S58 T59 W60 G61 C93 G94 A95 Y98 Y100 F101 C102 S9 T10 T11 N13 T14 S57 T58 W59 G60 C92 G93 A94 Y97 Y99 F100 C101 ? 0009055,0010181 Kd=0.0026nM remove_due_to_license_issue P00323 12206666 152 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWGDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGASSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1akw A 1.75 BS01 FMN A 1 S10 T11 T12 N14 T15 S58 T59 W60 L61 G94 D95 Y98 F101 S9 T10 T11 N13 T14 S57 T58 W59 L60 G93 D94 Y97 F100 ? 0009055,0010181 Kd=2.6nM remove_due_to_license_issue P00323 9622492 149 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWLDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGDSSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1al7 A 2.6 BS02 HST A 1 Y24 W108 Y129 R164 F172 I207 H254 R257 Y24 W108 Y129 R164 F172 I198 H245 R248 S106 Y129 T155 D157 K230 H254 S106 Y129 T155 D157 K221 H245 1.1.3.15 0003973,0005777,0009853,0009854,0010181,0016491,0051707 remove_due_to_license_issue P05414 9144771 361 MEITNVNEYEAIAKQKLPKMVYDYYASGAEDQWTLAENRNAFSRILFRPRILIDVTNIDMTTTILGFKISMPIMIAPTAMQKMAHPEGEYATARAASAAGTIMTLSSWATSSVEEVASTGPGIRFFQLYVYKDRNVVAQLVRRAERAGFKAIALTVDTPRLGRREADIKNRFVLPPFLTLKNFEGIDLGLSSYVAGQIDRSLSWKDVAWLQTITSLPILVKGVITAEDARLAVQHGAAGIIVSNHGARQLDYVPATIMALEEVVKAAQGRIPVFLDGGVRRGTDVFKALALGAAGVFIGRPVVFSLAAEGEAGVKKVLQMMRDEFELTMALSGCRSLKEISRSHIAADWD 1al8 A 2.2 BS02 DHP A 1 Y24 W108 Y129 F172 H254 R257 Y24 W108 Y129 F166 H239 R242 S106 Y129 T155 D157 K230 H254 S106 Y129 T155 D157 K215 H239 1.1.3.15 0003973,0005777,0009853,0009854,0010181,0016491,0051707 Ki=4.8uM remove_due_to_license_issue P05414 9144771 361 MEITNVNEYEAIAKQKLPKMVYDYYASGAEDQWTLAENRNAFSRILFRPRILIDVTNIDMTTTILGFKISMPIMIAPTAMQKMAHPEGEYATARAASAAGTIMTLSSWATSSVEEVASTGPGIRFFQLYVYKDRNVVAQLVRRAERAGFKAIALTVDTPRLIKNRFVLPPFLTLKNFEGIDLGLSSYVAGQIDRSLSWKDVAWLQTITSLPILVKGVITAEDARLAVQHGAAGIIVSNHGARQLDYVPATIMALEEVVKAAQGRIPVFLDGGVRRGTDVFKALALGAAGVFIGRPVVFSLAAEGEAGVKKVLQMMRDEFELTMALSGCRSLKEISRSHIAADWD 1alw A 2.03 BS05 ISA A 1 H129 Q173 H36 Q80 F162 G185 I187 F69 G92 I94 ? 0005509 Ki=0.3uM remove_due_to_license_issue P04574 9228946 11 EEVRQFRRLFAQLAGDDMEVSATELMNILNKVVTRHPDLKTDGFGIDTCRSMVAVMDSDTTGKLGFEEFKYLWNNIKKWQAIYKQFDVDRSGTIGSSELPGAFEAAGFHLNEHLYSMIIRRYSDEGGNMDFDNFISCLVRLDAMFRAFKSLDKDGTGQIQVNIQEWLQLTMYS 1amk A 1.83 BS01 PGA A 1 K13 H95 E167 I172 G173 G212 S213 G234 G235 K13 H95 E167 I172 G173 G212 S213 G234 G235 N11 K13 H95 E97 E167 G173 S213 N11 K13 H95 E97 E167 G173 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=0.05mM remove_due_to_license_issue P48499 10235625 600 SAKPQPIAAANWKCNGTTASIEKLVQVFNEHTISHDVQCVVAPTFVHIPLVQAKLRNPKYVISAENAIAKSGAFTGEVSMPILKDIGVHWVILGHSERRTYYGETDEIVAQKVSEACKQGFMVIACIGETLQQREANQTAKVVLSQTSAIAAKLTKDAWNQVVLAYEPVWAIGTGKVATPEQAQEVHLLLRKWVSENIGTDVAAKLRILYGGSVNAANAATLYAKPDINGFLVGGASLKPEFRDIIDATR 1amn A 2.8 BS01 NAF A 1 W84 G118 G119 S200 W233 F288 F290 F331 H440 W81 G115 G116 S197 W230 F285 F287 F328 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 594 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNA 1amw A 1.85 BS01 ADP A 1 N37 A41 M84 N92 G121 V122 F124 N36 A40 M83 N91 G120 V121 F123 ? 0005524,0006457,0016887,0051082,0140662 Kd=29uM remove_due_to_license_issue P02829 9230303 300 ASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 1ao0 A 2.8 BS04 ADP A 1 H25 Y242 S244 R245 P246 P281 D282 S283 K305 H25 Y238 S240 R241 P242 P277 D278 S279 K301 C1 G27 N102 G103 Y242 E300 K305 Q315 K423 C1 G27 N98 G99 Y238 E296 K301 Q311 K419 2.4.2.14 0000287,0004044,0006164,0006189,0009113,0016757,0046872,0051536,0051539 remove_due_to_license_issue P00497 9271502 468 CGVFGIWGHEEAPQITYYGLHSLQHRGQEGAGIVATDGEKLTAHKGQGLITEVFQNGELSKVKGKGAIGHVRYATGYENVQPLLFRSQNNGSLALAHNGNLVNATQLKQQLENQGSIFQTSSDTEVLAHLIKRSGHFTLKDQIKNSLSMLKGAYAFLIMTETEMIVALDPNGLRPLSIGMMGDAYVVASETCAFDVVGATYLREVEPGEMLIINDEGMKSERFSMNINRSICSMEYIYFSRPDSNIDGINVHSARKNLGKMLAQESAVEADVVTGVPDSSISAAIGYAEATGIPYELGLIKNRYVGRTFIQPSQALREQGVRMKLSAVRGVVEGKRVVMVDDSIVRGTTSRRIVTMLREAGATEVHVKISSPPIAHPCFYGIDTSTHEELIASSHSVEEIRQEIGADTLSFLSVEGLLKGIGRKYDDSNCGQCLACFTGKYPTEIYQDTVLPHVK 1ao0 A 2.8 BS05 ADP B 1 I304 K305 R307 I300 K301 R303 C1 G27 N102 G103 Y242 E300 K305 Q315 K423 C1 G27 N98 G99 Y238 E296 K301 Q311 K419 2.4.2.14 0000287,0004044,0006164,0006189,0009113,0016757,0046872,0051536,0051539 remove_due_to_license_issue P00497 9271502 468 CGVFGIWGHEEAPQITYYGLHSLQHRGQEGAGIVATDGEKLTAHKGQGLITEVFQNGELSKVKGKGAIGHVRYATGYENVQPLLFRSQNNGSLALAHNGNLVNATQLKQQLENQGSIFQTSSDTEVLAHLIKRSGHFTLKDQIKNSLSMLKGAYAFLIMTETEMIVALDPNGLRPLSIGMMGDAYVVASETCAFDVVGATYLREVEPGEMLIINDEGMKSERFSMNINRSICSMEYIYFSRPDSNIDGINVHSARKNLGKMLAQESAVEADVVTGVPDSSISAAIGYAEATGIPYELGLIKNRYVGRTFIQPSQALREQGVRMKLSAVRGVVEGKRVVMVDDSIVRGTTSRRIVTMLREAGATEVHVKISSPPIAHPCFYGIDTSTHEELIASSHSVEEIRQEIGADTLSFLSVEGLLKGIGRKYDDSNCGQCLACFTGKYPTEIYQDTVLPHVK 1ao0 B 2.8 BS01 ADP A 1 I304 K305 R307 I300 K301 R303 C1 G27 N102 G103 Y242 E300 K305 Q315 K423 C1 G27 N98 G99 Y238 E296 K301 Q311 K419 2.4.2.14 0000287,0004044,0006164,0006189,0009113,0016757,0046872,0051536,0051539 remove_due_to_license_issue P00497 9271502 468 CGVFGIWGHEEAPQITYYGLHSLQHRGQEGAGIVATDGEKLTAHKGQGLITEVFQNGELSKVKGKGAIGHVRYATGYENVQPLLFRSQNNGSLALAHNGNLVNATQLKQQLENQGSIFQTSSDTEVLAHLIKRSGHFTLKDQIKNSLSMLKGAYAFLIMTETEMIVALDPNGLRPLSIGMMGDAYVVASETCAFDVVGATYLREVEPGEMLIINDEGMKSERFSMNINRSICSMEYIYFSRPDSNIDGINVHSARKNLGKMLAQESAVEADVVTGVPDSSISAAIGYAEATGIPYELGLIKNRYVGRTFIQPSQALREQGVRMKLSAVRGVVEGKRVVMVDDSIVRGTTSRRIVTMLREAGATEVHVKISSPPIAHPCFYGIDTSTHEELIASSHSVEEIRQEIGADTLSFLSVEGLLKGIGRKYDDSNCGQCLACFTGKYPTEIYQDTVLPHVK 1ao0 B 2.8 BS05 ADP B 1 Y242 S244 R245 P246 P281 D282 S283 K305 Y238 S240 R241 P242 P277 D278 S279 K301 C1 G27 N102 G103 Y242 E300 K305 Q315 K423 C1 G27 N98 G99 Y238 E296 K301 Q311 K419 2.4.2.14 0000287,0004044,0006164,0006189,0009113,0016757,0046872,0051536,0051539 remove_due_to_license_issue P00497 9271502 468 CGVFGIWGHEEAPQITYYGLHSLQHRGQEGAGIVATDGEKLTAHKGQGLITEVFQNGELSKVKGKGAIGHVRYATGYENVQPLLFRSQNNGSLALAHNGNLVNATQLKQQLENQGSIFQTSSDTEVLAHLIKRSGHFTLKDQIKNSLSMLKGAYAFLIMTETEMIVALDPNGLRPLSIGMMGDAYVVASETCAFDVVGATYLREVEPGEMLIINDEGMKSERFSMNINRSICSMEYIYFSRPDSNIDGINVHSARKNLGKMLAQESAVEADVVTGVPDSSISAAIGYAEATGIPYELGLIKNRYVGRTFIQPSQALREQGVRMKLSAVRGVVEGKRVVMVDDSIVRGTTSRRIVTMLREAGATEVHVKISSPPIAHPCFYGIDTSTHEELIASSHSVEEIRQEIGADTLSFLSVEGLLKGIGRKYDDSNCGQCLACFTGKYPTEIYQDTVLPHVK 1ao8 A -1.00 BS01 MTX A 1 L4 A6 D26 L27 F30 R31 F49 R57 L4 A6 D26 L27 F30 R31 F49 R57 L4 L19 W21 D26 L27 F30 L54 L94 T116 L4 L19 W21 D26 L27 F30 L54 L94 T116 1.5.1.3 0004146,0005829,0006730,0016491,0031427,0046452,0046654,0046655,0046677,0050661 remove_due_to_license_issue IC50=16nM, Ki=0.004000nM P00381 9514736 170 TAFLWAQDRDGLIGKDGHLPWHLPDDLHYFRAQTVGKIMVVGRRTYESFPKRPLPERTNVVLTHQEDYQAQGAVVVHDVAAVFAYAKQHPDQELVIAGGAQIFTAFKDDVDTLLVTRLAGSFEGDTKMIPLNWDDFTKVSSRTVEDTNPALTHTYEVWQKKA 1apb A 1.76 BS02 FCB A 1 K10 E14 W16 D90 R151 N232 K9 E13 W15 D89 R150 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=1.51uM remove_due_to_license_issue P02924 2204627 308 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMMAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLGSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 1aq1 A 2.0 BS01 STU A 1 I10 G13 A31 E81 F82 L83 H84 Q85 D86 Q131 L134 D145 I10 G13 A31 E73 F74 L75 H76 Q77 D78 Q123 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 9334743 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1aqi A 2.6 BS01 SAH A 1 V21 A47 E71 I72 D89 F90 N105 P107 Y108 V1 A27 E51 I52 D69 F70 N85 P87 Y88 N105 P106 Y108 F196 N85 P86 Y88 F165 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 8995524 500 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTGYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSTLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 1aqj A 2.6 BS01 SFG A 1 V21 A47 E71 F90 N105 P106 P107 Y108 F146 V1 A27 E51 F70 N85 P86 P87 Y88 F114 N105 P106 Y108 F196 N85 P86 Y88 F164 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 8995524 500 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTGYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 1atr A 2.34 BS02 ADP A 1 G12 T14 Y15 G201 G202 E268 K271 R272 S275 G339 G11 T13 Y14 G200 G201 E267 K270 R271 S274 G338 D10 K71 E175 D199 D9 K70 E174 D198 3.6.4.10 0005524,0140662 remove_due_to_license_issue P19120 8226982 486 SKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGVFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILSGDK 1au0 A 2.6 BS01 SDK A 1 N18 Q19 G20 G23 C25 G65 G66 Y67 L160 N161 H162 N18 Q19 G20 G23 C25 G65 G66 Y67 L160 N161 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue Ki=22nM P43235 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1au2 A 2.6 BS01 POS A 1 N18 Q19 G20 G23 C25 G66 Y67 M68 L160 N161 H162 W184 N18 Q19 G20 G23 C25 G66 Y67 M68 L160 N161 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1auj A 2.1 BS01 PPB A 1 H57 N97 S190 C191 Q192 G193 S195 S214 W215 G216 G219 H40 N79 S172 C173 Q174 G175 S177 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 9341205 247 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1avd A 2.7 BS01 BTN A 1 L14 S16 Y33 T35 V37 A39 T40 W70 S73 S75 T77 W97 L12 S14 Y31 T33 V35 A37 T38 W68 S71 S73 T75 W95 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 8515446 400 KCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYTTAVTATSNEIKESPLHGTENTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRLRT 1avn A 2.0 BS03 HSM A 1 N62 H64 N67 Q92 N59 H61 N64 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.125mM remove_due_to_license_issue P00918 9265618 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1aw1 A 2.7 BS01 PGA A 1 K11 H97 E169 L233 G235 G236 K10 H96 E168 L232 G234 G235 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 remove_due_to_license_issue P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAKA 1aw1 B 2.7 BS01 PGA B 1 K11 H97 E169 I174 G175 G213 S214 L233 G235 K10 H96 E168 I173 G174 G212 S213 L232 G234 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 remove_due_to_license_issue P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAK 1awf H 2.2 BS03 GR4 H 1 H57 W60D W148 A190 C191 E192 G193 S195 W215 G216 H43 W50 W148 A200 C201 E202 G203 S205 W227 G228 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 9578548 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1awh D 3.0 BS01 GR3 D 1 H57 W60D A190 C191 E192 G193 D194 S195 S214 W215 H43 W50 A200 C201 E202 G203 D204 S205 S226 W227 H57 D102 E192 G193 D194 S195 G196 H43 D99 E202 G203 D204 S205 G206 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 9578548 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1axr A 2.3 BS02 HTP A 1 L136 L139 N284 H377 N484 E672 S674 G675 L123 L126 N271 H364 N471 E659 S661 G662 H377 K568 R569 K574 T676 K680 H364 K555 R556 K561 T663 K667 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=540uM remove_due_to_license_issue P00489 998 SVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1axs H 2.6 BS01 HOP H 1 E35 G95 H96 Y1001 D101 W103 E35 G99 H100 Y105 D108 W110 ? remove_due_to_license_issue P01857 9305839 1006 QVQLLESGAELMKPGASVKISCKATGYTFSSFWIEWVKQRPGHGLEWIGEILPGSGGTHYNEKFKGKATFTADKSSNTAYMQLSSLTSEDSAVYYCARGHSYYFYDGDYWGQGTSVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 1axs L 2.6 BS01 HOP H 1 F36 L89 Y91 F36 L89 Y91 ? 0005576 remove_due_to_license_issue Q7Z3Y4 9305839 1006 ELVLTQSPSSMYASLGERVTITCKASQDINSYLNWFQQKPGKSPKTLIYRTNRLVDGVPSRFSGSGSGQDYSLTISSLEYEDMGIYYCLQYDEFPYTFGSGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNR 1axz A 1.95 BS02 GAL A 1 D89 G107 F131 N133 G217 A218 Q219 D89 G107 F131 N133 G217 A218 Q219 ? 0030246 Ka=1570M^-1 remove_due_to_license_issue P16404 9545381 402 VETISFSFSEFEPGNDNLTLQGAALITQSGVLQLTKINQNGMPAWDSTGRTLYAKPVHIWDMTTGTVASFETRFSFSIEQPYTRPLPADGLVFFMGPTKSKPAQGYGYLGIFNNSKQDNSYQTLGVEFDTFSNPWDPPQVPHIGIDVNSIRSIKTQPFQLDNGQVANVVIKYDASSKILHAVLVYPSSGAIYTIAEIVDVKQVLPEWVDVGLSGATGAQRDAAETHDVYSWSFQASLPE 1ayu A 2.2 BS01 INA A 1 Q19 G20 Q21 C22 G23 C25 W26 D61 G65 G66 Y67 H162 W184 Q19 G20 Q21 C22 G23 C25 W26 D61 G65 G66 Y67 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue Ki=0.7nM P43235 9405598 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1ayv A 2.3 BS01 IN6 A 1 Q19 G20 Q21 G23 C25 W26 D61 G64 G65 G66 Y67 H162 W184 Q19 G20 Q21 G23 C25 W26 D61 G64 G65 G66 Y67 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue Ki=10.0nM P43235 9405598 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1azl A 1.8 BS01 FMN A 1 S10 T11 T12 N14 T15 S58 T59 W60 V61 C93 G94 D95 Y98 F101 S9 T10 T11 N13 T14 S57 T58 W59 V60 C92 G93 D94 Y97 F100 ? 0009055,0010181 Kd=2.4nM remove_due_to_license_issue P00323 9622492 149 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWVDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGDSSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1azm A 2.0 BS02 AZM A 1 F91 H94 L198 T199 H200 F89 H92 L196 T197 H198 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T197 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 remove_due_to_license_issue Ki=250nM, Kd=1400nM, IC50=5.8nM P00915 7932756 262 PDWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 1b0f A 3.0 BS02 SEI A 1 H57 R177 C191 F192 G193 D194 S195 S214 F215 V216 R217 H41 R153 C169 F170 G171 D172 S173 S188 F189 V190 R191 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G167 C169 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 remove_due_to_license_issue Ki=25nM P08246 9651152 300 IVGGRRARPHAWPFMVSLQLAGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFEDGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 1b11 A 1.9 BS01 3TL A 1 G32 D34 M56 I57 G58 G29 D31 M53 I54 G55 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 Ki=41nM remove_due_to_license_issue P16088 10651036 201 VGTTTTLEKRPEILIFVNGYPIKFLLDTGADITILNRRDFQVKNSIENGRQNMIGVGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLIQPLLGRDNMIKFNIRLVM 1b2i A -1.00 BS01 AMH A 1 Y36 D55 E57 W62 R71 W72 Y39 D58 E60 W64 R73 W74 3.4.21.7 remove_due_to_license_issue Kd=1100nM, IC50=3100nM, Ki=25000000nM P00747 10625440 84 TSEECMHGSGENYDGKISKTMSGLECQAWDSQSPHAHGYIPSKFPNKNLKKNYCRNPDRELRPWCFTTDPNKRWELCDIPRCT 1b38 A 2.0 BS02 ATP A 1 I10 G13 T14 V18 A31 K33 F82 L83 D86 K129 Q131 N132 L134 D145 I10 G13 T14 V18 A31 K33 F74 L75 D78 K121 Q123 N124 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=0.254uM remove_due_to_license_issue P24941 10085115 381 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1b39 A 2.1 BS02 ATP A 1 I10 G13 T14 V18 A31 K33 F82 L83 D86 K129 Q131 N132 L134 D145 I10 G13 T14 V18 A31 K33 F74 L75 D78 K121 Q123 N124 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=0.12uM remove_due_to_license_issue P24941 10085115 381 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1b42 A 2.2 BS02 M1A A 1 Y22 F180 E233 Y22 F174 E227 2.1.1.57 0003746,0004483,0006370,0031440 Kd=97.9uM remove_due_to_license_issue P07617 10377383 600 MDVVSLDKPFMYFEEIDNELDYEPESANEVAKKLPYQGQLKLLLGELFFLSKLQRHGILDGATVVYIGSAPGTHIRYLRDHFYNLGVIIKWMLIDGRHHDPILNGLRDVTLVTRFVDEEYLRSIKKQLHPSKIILISDVRSPSTADLLSNYALQNVMISILNPVASSLKWRCPFPDQWIKDFYIPHGNKMLQPFAPSYSAEMRLLSIYTGENMRLTRVTKSDAVNYEKKMYYLNKIVRNKVVVNFDYPNQEYDYFHMYFMLRTVYCNKTFPTTKAKVLFLQQSIFRFLNIP 1b4d A 2.0 BS01 CRA A 1 G135 L136 N284 H377 T378 N484 E672 S674 G675 G123 L124 N262 H346 T347 N453 E641 S643 G644 H377 K568 R569 K574 T676 K680 H346 K537 R538 K543 T645 K649 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=15.6uM remove_due_to_license_issue Ki=16000nM P00489 10211820 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 1b55 A 2.4 BS02 4IP A 1 K12 S14 Q15 Q16 K17 K18 S21 N24 R28 Y39 K53 K11 S13 Q14 Q15 K16 K17 S20 N23 R27 Y38 K52 2.7.10.2 0035556 Kd=40nM remove_due_to_license_issue Q06187 10196129 171 AAVILESIFLKRSQQKKKTSPLNFKKRLFLLTVHKLSYYEYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIPRRMEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQILEN 1b55 B 2.4 BS02 4IP B 1 K12 S14 Q15 Q16 K17 K18 S21 N24 R28 Y39 K53 K11 S13 Q14 Q15 K16 K17 S20 N23 R27 Y38 K52 2.7.10.2 0035556 Kd=40nM remove_due_to_license_issue Q06187 10196129 172 AAVILESIFLKRSQQKKKTSPLNFKKRLFLLTVHKLSYYEYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQISEMEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQILEN 1b57 A 2.0 BS04 PGH A 1 D109 H110 H226 G227 H264 G265 S267 N286 I287 D288 T289 D109 H110 H214 G215 H252 G253 S255 N274 I275 D276 T277 D109 H110 E182 H226 H264 N286 D109 H110 E182 H214 H252 N274 4.1.2.13 0004332,0005515,0005829,0005975,0006094,0006096,0008270,0016829,0016832,0042802,0042803,0046872 remove_due_to_license_issue P0AB71 10080900 359 SKIFDFVKPGVITGDDVQKVFQVAKENNFALPAVNCVGTDSINAVLETAAKVKAPVIVQFSNGGASFIAGKGVKSDVPQGAAILGAISGAHHVHQMAEHYGVPVILHTDHCAKKLLPWIDGLLDAGEKHFAATGKPLFSSHMIDLSEESLQENIEICSKYLERMSKIGMTLEIELGCTGGEELYTQPEDVDYAYTELSKISPRFTIAASFGNVHGVYKPGNVVLTPTILRDSQEYVSKKHNLPHNSLNFVFHGGSGSTAQEIKDSVSYGVVKMNIDTDTQWATWEGVLNYYKANEAYLQGQLGNPKGEDQPNKKYYDPRVWLRAGQTSMIARLEKAFQELNAIDVL 1b57 B 2.0 BS04 PGH B 1 D109 H110 H226 G227 H264 G265 S267 N286 I287 D288 T289 D109 H110 H214 G215 H252 G253 S255 N274 I275 D276 T277 D109 H110 E182 H226 H264 N286 D109 H110 E182 H214 H252 N274 4.1.2.13 0004332,0005515,0005829,0005975,0006094,0006096,0008270,0016829,0016832,0042802,0042803,0046872 remove_due_to_license_issue P0AB71 10080900 359 SKIFDFVKPGVITGDDVQKVFQVAKENNFALPAVNCVGTDSINAVLETAAKVKAPVIVQFSNGGASFIAGKGVKSDVPQGAAILGAISGAHHVHQMAEHYGVPVILHTDHCAKKLLPWIDGLLDAGEKHFAATGKPLFSSHMIDLSEESLQENIEICSKYLERMSKIGMTLEIELGCTGGEELYTQPEDVDYAYTELSKISPRFTIAASFGNVHGVYKPGNVVLTPTILRDSQEYVSKKHNLPHNSLNFVFHGGSGSTAQEIKDSVSYGVVKMNIDTDTQWATWEGVLNYYKANEAYLQGQLGNPKGEDQPNKKYYDPRVWLRAGQTSMIARLEKAFQELNAIDVL 1b5g H 2.07 BS03 0ZE H 1 H57 Y60A W60D D189 A190 E192 G193 S195 S214 W215 G216 G219 H43 Y47 W50 D191 A192 E194 G195 S197 S218 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10212123 372 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1b69 A -1.00 BS01 dna B 0 R5 T15 G16 E17 S18 R20 K21 K28 I30 R55 R3 T13 G14 E15 S16 R18 K19 K26 I28 R53 ? 0003677,0008907,0015074 remove_due_to_license_issue P22886 10201406 101 ~ 113 EKRRDNRGRILKTGESQRKDGRYLYKYIDSFGEPQFVYSWKLVATDRVPAGKRDAISLREKIAELQKDI 1b69 A -1.00 BS02 dna C 0 R24 K28 F38 Y40 R22 K26 F36 Y38 ? 0003677,0008907,0015074 remove_due_to_license_issue P22886 10201406 114 ~ 126 EKRRDNRGRILKTGESQRKDGRYLYKYIDSFGEPQFVYSWKLVATDRVPAGKRDAISLREKIAELQKDI 1b6k A 1.85 BS01 PI5 A 1 D25 G27 A28 D29 G48 G49 P81 V82 D25 G27 A28 D29 G48 G49 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.8nM remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6k B 1.85 BS01 PI5 A 1 D125 G127 A128 D129 G148 V182 D25 G27 A28 D29 G48 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6l A 1.75 BS01 PI4 A 1 D25 G27 A28 D29 D30 G48 V82 D25 G27 A28 D29 D30 G48 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=5nM remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6l B 1.75 BS01 PI4 A 1 D125 G127 V182 I184 D25 G27 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6m A 1.85 BS01 PI6 B 1 R8 D25 G27 G48 G49 I50 P81 V82 R8 D25 G27 G48 G49 I50 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6m B 1.85 BS01 PI6 B 1 D125 G127 A128 D129 G148 G149 I184 D25 G27 A28 D29 G48 G49 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4nM remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6p A 2.0 BS01 PI7 A 1 D25 G27 D29 G48 P81 V82 D25 G27 D29 G48 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3nM remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b6p B 2.0 BS01 PI7 A 1 D125 G127 D129 G148 G149 I184 D25 G27 D29 G48 G49 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1b74 A 2.3 BS01 DGN A 1 C70 N71 G177 C178 C70 N71 G177 C178 D7 S8 C70 T72 T114 E147 C178 H180 D7 S8 C70 T72 T114 E147 C178 H180 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0071555 Ki=50mM remove_due_to_license_issue P56868 10331867 538 MKIGIFDSGVGGLTVLKAIRNRYRKVDIVYLGDTARVPYGIRSKDTIIRYSLECAGFLKDKGVDIIVVACNTASAYALERLKKEINVPVFGVIEPGVKEALKKSRNKKIGVIGTPATVKSGAYQRKLEEGGADVFAKACPLFAPLAEEGLLEGEITRKVVEHYLKEFKGKIDTLILGCTHYPLLKKEIKKFLGDAEVVDSSEALSLSLHNFIKDDGSSSLELFFTDLSPNLQFLIKLILGRDYPVKLAEGVF 1b8n A 2.0 BS01 IMG A 1 H86 Y88 A116 G118 F200 E201 V217 G218 M219 N243 H257 V260 H85 Y87 A115 G117 F199 E200 V216 G217 M218 N242 H256 V259 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S32 H63 H85 Y87 E88 A115 M218 S219 N242 V244 H256 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Ki=30pM remove_due_to_license_issue Ki=0.030000nM P55859 12463747 600 QNGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGENPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESQGKANHEEVLEAGKQAAQKLEQFVSLLM 1b8o A 1.5 BS02 IMH A 1 H86 Y88 A116 G118 F200 E201 M219 N243 H257 V260 H84 Y86 A114 G116 F198 E199 M217 N241 H255 V258 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S31 H62 H84 Y86 E87 A114 M217 S218 N241 V243 H255 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Ki=23pM remove_due_to_license_issue P55859 11170405 600 NGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGENPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESQGKANHEEVLEAGKQAAQKLEQFVSLLMASI 1b8y A 2.0 BS06 IN7 A 1 L164 A165 L197 H201 E202 H211 L218 P221 L222 Y223 H224 L82 A83 L115 H119 E120 H129 L136 P139 L140 Y141 H142 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=14nM remove_due_to_license_issue P08254 10422833 502 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPP 1b9s A 2.5 BS02 FDI A 1 R116 D149 R223 R292 R374 Y409 R40 D73 R147 R216 R298 Y333 D149 E276 R292 R374 Y409 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50>667uM remove_due_to_license_issue IC50=670000nM P03474 10547289 468 EPEWTYPRLSCQGSTFQKALLISPHRFGEIKGNSAPLIIREPFVACGPKECRHFALTHYAAQPGGYYNGTRKDRNKLRHLVSVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDNDALVKIKYGEAYTDTYHSYAHNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEILPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTKTYLDTPRPDDGSIAGPCESNGDKWLGGIKGGFVHQRMASKIGRWYSRTMSKTNRMGMELYVRYDGDPWTDSDALTLSGVMVSIEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKDTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1b9t A 2.4 BS02 RAI A 1 R116 E117 D149 R150 E226 E275 E276 R292 R374 Y409 R40 E41 D73 R74 E150 E199 E200 R216 R298 Y333 D149 E276 R292 R374 Y409 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=8uM remove_due_to_license_issue IC50=8000nM P03474 10547289 468 EPEWTYPRLSCQGSTFQKALLISPHRFGEIKGNSAPLIIREPFVACGPKECRHFALTHYAAQPGGYYNGTRKDRNKLRHLVSVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDNDALVKIKYGEAYTDTYHSYAHNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEILPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTKTYLDTPRPDDGSIAGPCESNGDKWLGGIKGGFVHQRMASKIGRWYSRTMSKTNRMGMELYVRYDGDPWTDSDALTLSGVMVSIEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKDTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1b9v A 2.35 BS02 RA2 A 1 R116 E117 D149 R150 W177 R223 E226 E275 E276 R292 N294 R374 Y409 R40 E41 D73 R74 W101 R147 E150 E199 E200 R216 N218 R298 Y333 D149 E276 R292 R374 Y409 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=224uM remove_due_to_license_issue IC50=271000nM P03474 10547289 468 EPEWTYPRLSCQGSTFQKALLISPHRFGEIKGNSAPLIIREPFVACGPKECRHFALTHYAAQPGGYYNGTRKDRNKLRHLVSVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDNDALVKIKYGEAYTDTYHSYAHNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEILPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTKTYLDTPRPDDGSIAGPCESNGDKWLGGIKGGFVHQRMASKIGRWYSRTMSKTNRMGMELYVRYDGDPWTDSDALTLSGVMVSIEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKDTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1ba8 B 1.8 BS02 0IT B 1 H57 Y60A W60D E97A L99 I174 D189 A190 S195 S214 W215 G216 H43 Y47 W50 E94 L96 I172 D192 A193 S198 S219 W220 G221 H57 D102 E192 G193 D194 S195 G196 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 9724521 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1bai A 2.4 BS01 0Q4 A 1 D37 G39 D42 N61 I64 H65 P105 V106 D37 G39 D42 N61 I64 H65 P105 V106 D37 T38 G39 D37 T38 G39 3.4.23.- 0004190,0006508 Ki=20nM remove_due_to_license_issue P03322 9521772 125 LAMTMEHKDRPLVRVILTNTGSHPVKQRSVYITALLDTGADDTVISEEDWPTDWPVMEAANPQIHGIGGGIPVRKSRDMIELGVINRDGSLERPLLLFPLVAMTPVNILGRDCLQGLGLRLTNL 1bai B 2.4 BS01 0Q4 A 1 L35 A40 Q63 V106 L35 A40 Q63 V106 D37 T38 G39 D37 T38 G39 3.4.23.- 0004190,0006508 remove_due_to_license_issue P03322 9521772 125 LAMTMEHKDRPLVRVILTNTGSHPVKQRSVYITALLDTGADDTVISEEDWPTDWPVMEAANPQIHGIGGGIPVRKSRDMIELGVINRDGSLERPLLLFPLVAMTPVNILGRDCLQGLGLRLTNL 1bap A 1.75 BS02 ARB A 1 K10 E14 D90 R151 M204 N232 K9 E13 D89 R150 M203 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.14uM remove_due_to_license_issue P02924 2204627 308 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMMAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLGSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 1bb0 B 2.1 BS03 0IV B 1 H57 Y60A W60D I174 D189 C191 S195 S214 W215 G216 G219 H42 Y46 W49 I170 D190 C192 S196 S217 W218 G219 G221 H57 D102 E192 G193 D194 S195 G196 H42 D98 E193 G194 D195 S196 G197 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=28.8nM P00734 9724521 1 IVEGSDAEIGMSPWQVMLFRKPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1bcd A 1.9 BS02 FMS A 1 H94 H119 L198 T199 T200 W209 H92 H117 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=2nM remove_due_to_license_issue Kd=130nM, IC50=13nM P00918 8070585 500 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bcu H 2.0 BS03 PRL H 1 D189 A190 W215 G216 G219 C220 D191 A192 W219 G220 G222 C223 3.4.21.5 0004252,0005509,0006508,0007596 Kd=0.53mM remove_due_to_license_issue IC50=12000nM P00734 9559654 280 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1bdh A 2.7 BS01 dna B 0 S14 T16 T17 R26 V28 A29 T32 L54 A55 S12 T14 T15 R24 V26 A27 T30 L52 A53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLAVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1bdi A 3.0 BS01 dna B 0 V13 S14 T16 T17 R26 V28 A29 T32 L54 K55 V11 S12 T14 T15 R24 V26 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1bdl A 2.8 BS01 IM1 A 1 G27 D29 D30 K45 M46 I47 G48 G27 D29 D30 K45 M46 I47 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9692985 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDSIVAGIELPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1bdl B 2.8 BS01 IM1 B 1 G27 A28 D29 D30 I47 G48 I50 G27 A28 D29 D30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9692985 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDSIVAGIELPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1bdq A 2.5 BS01 IM1 B 1 R8 G27 A28 D30 G48 G49 I50 I82 R8 G27 A28 D30 G48 G49 I50 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9692985 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDSIVAGIELPGRWKPKMVGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 1bdq B 2.5 BS01 IM1 B 1 D25 G27 A28 D29 G48 I50 I82 D25 G27 A28 D29 G48 I50 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=460nM remove_due_to_license_issue P04587 9692985 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDSIVAGIELPGRWKPKMVGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 1bdr A 2.8 BS01 IM1 B 1 D25 G27 G48 G49 V82 D25 G27 G48 G49 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9692985 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDSVVAGIELPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1bdr B 2.8 BS01 IM1 B 1 D25 G27 A28 D29 G48 G49 I50 V82 D25 G27 A28 D29 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9692985 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDSVVAGIELPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1bdt A 2.5 BS01 dna E 0 M1 M4 R23 S32 V33 M1 M4 R23 S32 V33 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIG 1bdt A 2.5 BS02 dna F 0 Q9 F10 N11 R13 Q9 F10 N11 R13 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIG 1bdt B 2.5 BS01 dna E 0 Q9 F10 N11 R13 Q9 F10 N11 R13 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIGA 1bdt B 2.5 BS02 dna F 0 M1 G3 M4 S5 R23 S32 V33 N34 M1 G3 M4 S5 R23 S32 V33 N34 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIGA 1bdt C 2.5 BS01 dna E 0 Q9 F10 N11 R13 Q9 F10 N11 R13 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGR 1bdt C 2.5 BS02 dna F 0 M1 K2 G3 M4 S5 R23 S32 V33 N34 M1 K2 G3 M4 S5 R23 S32 V33 N34 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGR 1bdt D 2.5 BS01 dna E 0 M1 G3 M4 S5 N11 S32 V33 N34 M1 G3 M4 S5 N11 S32 V33 N34 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGR 1bdt D 2.5 BS02 dna F 0 Q9 F10 N11 Q9 F10 N11 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQFNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGR 1bdv A 2.8 BS01 dna E 0 R13 R23 S32 R7 R17 S26 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIG 1bdv A 2.8 BS02 dna F 0 N11 R13 N5 R7 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIG 1bdv B 2.8 BS01 dna E 0 Q9 N11 Q9 N11 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIGA 1bdv B 2.8 BS02 dna F 0 M1 G3 M4 S5 S32 V33 N34 M1 G3 M4 S5 S32 V33 N34 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGRIGA 1bdv C 2.8 BS01 dna E 0 Q9 N11 Q3 N5 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEG 1bdv C 2.8 BS02 dna F 0 N11 R23 S32 V33 N5 R17 S26 V27 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEG 1bdv D 2.8 BS01 dna E 0 M1 G3 M4 S5 N11 S32 V33 N34 M1 G3 M4 S5 N11 S32 V33 N34 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGR 1bdv D 2.8 BS02 dna F 0 Q9 N11 Q9 N11 ? 0003677,0006355 remove_due_to_license_issue P03050 9927650 1 ~ 22 MKGMSKMPQVNLRWPREVLDLVRKVAEENGRSVNSEIYQRVMESFKKEGR 1bgo A 2.3 BS01 I10 A 1 Q19 G23 C25 D61 G65 G66 Y67 A137 N161 H162 W184 Q19 G23 C25 D61 G65 G66 Y67 A137 N161 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1bgq A 2.5 BS01 RDC A 1 N37 D40 K44 D79 M84 F124 L173 N37 D40 K44 D79 M84 F124 L173 ? 0005524,0006457,0016887,0051082,0140662 Kd=2.7nM remove_due_to_license_issue IC50=2e+2nM P02829 9925731 300 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 1bhx B 2.3 BS02 R56 F 1 H57 Y60A E97A H43 Y47 E94 H57 D102 H43 D99 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=145nM P00734 9733491 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKET 1bhx F 2.3 BS01 R56 F 1 D189 A190 C191 S195 S214 W215 G216 E217 D45 A46 C47 S51 S72 W73 G74 E75 3.4.21.5 0004252,0006508 Ki=0.145uM remove_due_to_license_issue Ki=145nM P00734 9733491 1 GQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1bil A 2.4 BS01 0IU A 1 D32 Y75 S76 T77 P111 F117 D215 G217 A218 S219 Y220 S222 M289 A300 D35 Y80 S81 T82 P115 F121 D220 G222 A223 S224 Y225 S227 M297 A308 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D220 A223 3.4.23.15 0004190,0006508 ic50=0.5nM remove_due_to_license_issue P00797 7493993 391 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSESLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 1bim A 2.8 BS01 0QB A 1 D32 G34 Y75 S76 T77 P111 F117 D215 G217 A218 S219 Y220 S222 M289 I291 A300 D35 G37 Y80 S81 T82 P115 F121 D220 G222 A223 S224 Y225 S227 M297 I299 A308 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D220 A223 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 7493993 391 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSESLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 1bio A 1.5 BS01 SOA A 1 C191 K192 S195 S215 R218 C179 K180 S183 S199 R202 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 remove_due_to_license_issue P00746 9753554 244 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 1biw B 2.5 BS06 S80 B 1 N162 V163 L164 V198 H201 E202 H205 H211 P221 L222 Y223 N80 V81 L82 V116 H119 E120 H123 H129 P139 L140 Y141 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=104nM remove_due_to_license_issue IC50=104nM P08254 9873489 401 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1bji A 2.0 BS02 DPC A 1 R118 E119 D151 I222 R224 A246 E276 E277 R292 N294 R371 Y406 R37 E38 D70 I142 R144 A166 E196 E197 R212 N214 R290 Y324 D151 E277 R292 R371 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.002uM remove_due_to_license_issue P03472 9526556 479G RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1bju A 1.8 BS03 GP6 A 1 H57 L99 D189 S190 Q192 W215 G216 G219 H40 L81 D171 S172 Q174 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=6.2uM remove_due_to_license_issue P00760 9836602 910 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1bjv A 1.8 BS04 GP8 A 1 H57 L99 D189 S190 W215 G216 G219 H40 L81 D171 S172 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=13uM remove_due_to_license_issue P00760 9836602 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1bkj A 1.8 BS01 FMN A 1 H11 R12 S13 R15 Q67 V127 Y128 I129 G130 R169 H10 R11 S12 R14 Q66 V126 Y127 I128 G129 R168 1.5.1.38 0008218,0008752,0016491,0052873 Kd=0.17uM remove_due_to_license_issue Q56691 8885832 241 NNTIETILAHRSIRKFTAVPITDEQRQTIIQAGLAASSSSMLQVVSIVRVTDSEKRNELAQFAGNQAYVESAAEFLVFCIDYQRHATINPDVQADFTELTLIGAVDSGIMAQNCLLAAESMGLGGVYIGGLRNSAAQVDELLGLPENSAVLFGMCLGHPDQNPEVKPRLPAHVVVHENQYQELNLDDIQSYDQTMQAYYSTWSQEVTGKLAGESRPHILPYLNSKGLAKR 1bkj A 1.8 BS02 FMN B 1 S38 S39 S40 S37 S38 S39 1.5.1.38 0008218,0008752,0016491,0052873 Kd=0.17uM remove_due_to_license_issue Q56691 8885832 241 NNTIETILAHRSIRKFTAVPITDEQRQTIIQAGLAASSSSMLQVVSIVRVTDSEKRNELAQFAGNQAYVESAAEFLVFCIDYQRHATINPDVQADFTELTLIGAVDSGIMAQNCLLAAESMGLGGVYIGGLRNSAAQVDELLGLPENSAVLFGMCLGHPDQNPEVKPRLPAHVVVHENQYQELNLDDIQSYDQTMQAYYSTWSQEVTGKLAGESRPHILPYLNSKGLAKR 1bkj B 1.8 BS01 FMN A 1 S38 S39 S40 S37 S38 S39 1.5.1.38 0008218,0008752,0016491,0052873 Kd=0.17uM remove_due_to_license_issue Q56691 8885832 241 NNTIETILAHRSIRKFTAVPITDEQRQTIIQAGLAASSSSMLQVVSIVRVTDSEKRNELAQFAGNQAYVESAAEFLVFCIDYQRHATINPDVQADFTELTLIGAVDSGIMAQNCLLAAESMGLGGVYIGGLRNSAAQVDELLGLPENSAVLFGMCLGHPDQNPEVKPRLPAHVVVHENQYQELNLDDIQSYDQTMQAYYSTWSQEVTGKLAGESRPHILPYLNSKGLAKR 1bkj B 1.8 BS02 FMN B 1 H11 R12 S13 R15 Q67 Y128 I129 G130 R169 H10 R11 S12 R14 Q66 Y127 I128 G129 R168 1.5.1.38 0008218,0008752,0016491,0052873 Kd=0.17uM remove_due_to_license_issue Q56691 8885832 241 NNTIETILAHRSIRKFTAVPITDEQRQTIIQAGLAASSSSMLQVVSIVRVTDSEKRNELAQFAGNQAYVESAAEFLVFCIDYQRHATINPDVQADFTELTLIGAVDSGIMAQNCLLAAESMGLGGVYIGGLRNSAAQVDELLGLPENSAVLFGMCLGHPDQNPEVKPRLPAHVVVHENQYQELNLDDIQSYDQTMQAYYSTWSQEVTGKLAGESRPHILPYLNSKGLAKR 1bkm A 2.0 BS01 1C5 A 1 R12 R32 S34 E35 T36 H58 Y59 K60 T72 G93 R10 R30 S32 E33 T34 H56 Y57 K58 T70 G91 2.7.10.2 remove_due_to_license_issue P00524 113 EEWYFGKITRRESEALLLNPENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFSSLQQLVAYYSKHADGLCHRLTNVCPT 1bky A 2.0 BS02 1MC A 1 Y22 F180 Y22 F174 2.1.1.57 0003723,0003746,0004483,0006370,0008168,0031440,0032259,0044423 Kd=144uM remove_due_to_license_issue P07617 10377383 600 MDVVSLDKPFMYFEEIDNELDYEPESANEVAKKLPYQGQLKLLLGELFFLSKLQRHGILDGATVVYIGSAPGTHIRYLRDHFYNLGVIIKWMLIDGRHHDPILNGLRDVTLVTRFVDEEYLRSIKKQLHPSKIILISDVRSPSTADLLSNYALQNVMISILNPVASSLKWRCPFPDQWIKDFYIPHGNKMLQPFAPSYSAEMRLLSIYTGENMRLTRVTKSDAVNYEKKMYYLNKIVRNKVVVNFDYPNQEYDYFHMYFMLRTVYCNKTFPTTKAKVLFLQQSIFRFLNIP 1bl4 A 1.9 BS01 AP1 A 1 Y26 V36 F46 Q53 E54 V55 I56 W59 Y82 H87 F99 Y26 V36 F46 Q53 E54 V55 I56 W59 Y82 H87 F99 Y26 V36 D37 I56 Y82 F99 Y26 V36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 ic50=1.8nM remove_due_to_license_issue IC50=8.2nM P62942 9724721 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKVDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1bl4 B 1.9 BS01 AP1 B 1 Y26 V36 F46 E54 V55 I56 W59 Y82 H87 F99 Y26 V36 F46 E54 V55 I56 W59 Y82 H87 F99 Y26 V36 D37 I56 Y82 F99 Y26 V36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 ic50=1.8nM remove_due_to_license_issue IC50=8.2nM P62942 9724721 109 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKVDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1bl6 A 2.5 BS01 SB6 A 1 Y35 A51 K53 I84 L104 V105 T106 M109 Y32 A48 K50 I81 L101 V102 T103 M106 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=160nM Q16539 9753691 800 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1bl7 A 2.5 BS01 SB4 A 1 A51 K53 I84 L104 V105 T106 M109 D168 A48 K50 I81 L101 V102 T103 M106 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=19nM Q16539 9753691 800 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1bm6 A -1.00 BS05 HAV A 1 V163 A165 H201 H205 V81 A83 H119 H123 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P08254 9760240 1 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1bm6 A -1.00 BS06 MSB A 1 N162 L164 V198 H201 L218 M219 P221 L222 N80 L82 V116 H119 L136 M137 P139 L140 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P08254 9760240 3 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1bm7 A 2.0 BS01 FLF A 1 K15 A108 S117 T119 K6 A99 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=30nM remove_due_to_license_issue IC50=2900nM P02766 9789022 501 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVT 1bm7 B 2.0 BS01 FLF B 1 K15 A108 S117 T119 K6 A99 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=30nM remove_due_to_license_issue IC50=2900nM P02766 9789022 502 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVT 1bma A 1.8 BS02 0QH A 1 H60 V103 C199 Q200 S203 S222 F223 V224 S225 R226 G228 C229 H45 V88 C184 Q185 S188 S207 F208 V209 S210 R211 G213 C214 H60 D108 Q200 G201 D202 S203 G204 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 Ki=26uM remove_due_to_license_issue P00772 7604279 256 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1bmk A 2.4 BS01 SB5 A 1 V30 G31 S32 Y35 V38 A51 K53 L104 V105 T106 L108 M109 V27 G28 S29 Y32 V35 A48 K50 L101 V102 T103 L105 M106 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=25nM Q16539 9753691 800 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1bmm H 2.6 BS03 BM2 H 1 H57 Y60A W60D L99 E192 S195 W215 G216 E217 G219 H43 Y47 W50 L96 E202 S205 W227 G228 E229 G230 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=390nM P00734 8745399 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1bmn H 2.8 BS03 BM9 H 1 H57 Y60A W60D L99 C191 E192 V213 S214 W215 G216 E217 G219 C220 H43 Y47 W50 L96 C201 E202 V225 S226 W227 G228 E229 G230 C231 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=16nM, Ki=3.6nM P00734 8745399 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1bmq A 2.5 BS01 MNO A 1 R179 H237 C285 R49 H107 C155 P177 R178 H237 G238 C285 R286 P47 R48 H107 G108 C155 R156 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 9987822 601 GNVKLCSLEEAQRIWKQKSAEIYPIMDKSSRTRLALIICNEEFDSIPRRTGAEVDITGMTMLLQNLGYSVDVKKNLTASDMTTELEAFAHRPEHKTSDSTFLVFMSHGIREGICGKKHSEQVPDILQLNAIFNMLNTKNCPSLKDKPKVIIIQACRGDSPGVVWFKD 1bmq B 2.5 BS01 MNO A 1 S339 W340 R341 R383 S23 W24 R25 R67 E390 E74 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 9987822 601 AIKKAHIEKDFIAFCSSTPDNVSWRHPTMGSVFIGRLIEHMQEYACSCDVEEIFRKVRFSFEQPDGRAQMPTTERVTLTRCFYLFPGH 1bn1 A 2.1 BS02 AL5 A 1 H94 H96 H119 L198 T199 T200 P202 H91 H93 H116 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.46nM remove_due_to_license_issue Kd=0.46nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bn3 A 2.2 BS02 AL6 A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.13nM remove_due_to_license_issue Kd=0.13nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bn4 A 2.1 BS02 AL9 A 1 H94 H96 H119 L198 T199 T200 P202 H91 H93 H116 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.49nM remove_due_to_license_issue Kd=0.49nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bnm A 2.6 BS02 AL8 A 1 H94 H119 V121 F131 L198 T199 T200 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=0.1nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bnn A 2.3 BS02 AL1 A 1 H94 H96 H119 F131 L198 T199 T200 L204 H91 H93 H116 F127 L194 T195 T196 L200 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.1nM remove_due_to_license_issue Kd=0.1nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bnq A 2.4 BS02 AL4 A 1 W5 H94 V121 F131 L198 T199 T200 W2 H91 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.32nM remove_due_to_license_issue Kd=0.32nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1bnt A 2.15 BS02 AL2 A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.16nM remove_due_to_license_issue Kd=0.16nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1bnu A 2.15 BS02 AL3 A 1 H94 H119 V121 F131 L198 T199 T200 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.2nM remove_due_to_license_issue Kd=0.2nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1bnv A 2.4 BS02 AL7 A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.7nM remove_due_to_license_issue Kd=1.7nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1bnw A 2.25 BS02 TPD A 1 H94 H96 H119 F131 L198 T199 T200 P202 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.83nM remove_due_to_license_issue Kd=0.83nM P00918 9865942 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1bo5 O 3.2 BS01 FBP O 1 G233 G234 R236 G232 G233 R235 2.7.1.30 0004370,0005515,0005524,0005829,0005975,0006071,0006072,0006974,0008270,0016301,0016773,0019563,0042802,0046872 remove_due_to_license_issue P0A6F3 9843423 502 EKKYIVALDQGTTSSRAVVMDHDANIISVSQREFEQIYPKPGWVEHDPMEIWATQSSTLVEVLAKADISSDQIAAIGITNQRETTIVWEKETGKPIYNAIVWQCRRTAEICEHLKRDGLEDYIRSNTGLVIDPYFSGTKVKWILDHVEGSRERARRGELLFGTVDTWLIWKMTQGRVHVTDYTNASRTMLFNIHTLDWDDKMLEVLDIPREMLPEVRRSSEVYGQTNIGGKGGTRIPISGIAGDQQAALFGQLCVKEGMAKNTYGTGCFMLMNTGEKAVKSENGLLTTIACGPTGEVNYALEGAVFMAGASIQWLRDEMKLINDAYDSEYFATKVQNTNGVYVVPAFTGLGAPYWDPYARGAIFGLTRGVNANHIIRATLESIAYQTRDVLEAMQADSGIRLHALRVDGGAVANNFLMQFQSDILGTRVERPEVREVTALGAAYLAGLAVGFWQNLDELQEKAVIEREFRPGIETTERNYRYAGWKKAVKRAMAWEEH 1bp0 A 2.4 BS01 UMP A 1 C198 H199 R218 S219 A220 D221 N229 H259 Y261 C198 H199 R218 S219 A220 D221 N229 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=4uM remove_due_to_license_issue P00469 10653645 317 MLEQPYLDLAKKVLDEGHFKPDITHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1bq3 D 2.7 BS01 IHP D 1 R7 S11 W13 N14 L18 F19 T20 K97 R113 R7 S11 W13 N14 L18 F19 T20 K97 R113 H8 R59 E86 H181 H8 R59 E86 H181 5.4.2.11 0003824,0004619,0005737,0005739,0005741,0005758,0005829,0006094,0006096,0016853,0016868,0046538 remove_due_to_license_issue P00950 10369755 350 PKLVLVRHGQSEWNEKNLFTGWVDVKLSAKGQQEAARAGELLKEKKVYPDVLYTSKLSRAIQTANIALEKADRLWIPVNRSWRLNERHYGDLQGKDKAETLKKFGEEKFNTYRRSFDVPPPPIDASSPFSQKGDERYKYVDPNVLPETESLALVIDRLLPYWQDVIAKDLLSGKTVMIAAHGNSLRGLVKHLEGISDADIAKLNIPTGIPLVFELDENLKPSKPSYYLDPEAAA 1bq4 A 2.5 BS01 BHC A 1 Y89 R113 R114 N183 N204 Y89 R113 R114 N183 N204 H8 R59 E86 H181 H8 R59 E86 H181 5.4.2.11 0003824,0004619,0005737,0005739,0005741,0005758,0005829,0006094,0006096,0016853,0016868,0046538 Ki=6uM remove_due_to_license_issue P00950 10369755 302 PKLVLVRHGQSEWNEKNLFTGWVDVKLSAKGQQEAARAGELLKEKKVYPDVLYTSKLSRAIQTANIALEKADRLWIPVNRSWRLNERHYGDLQGKDKAETLKKFGEEKFNTYRRSFDVPPPPIDASSPFSQKGDERYKYVDPNVLPETESLALVIDRLLPYWQDVIAKDLLSGKTVMIAAHGNSLRGLVKHLEGISDADIAKLNIPTGIPLVFELDENLKPSKPSYYLDPEAAA 1bqm A 3.1 BS01 HBY A 1 L100 K101 Y188 V189 G190 F227 W229 L234 Y318 L100 K101 Y188 V189 G190 F227 W229 L234 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 9813120 557 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGI 1bqn A 3.3 BS01 HBY A 1 L100 K101 V106 Y181 L188 V189 G190 W229 L234 H235 Y318 L100 K101 V106 Y181 L188 V189 G190 W229 L234 H235 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 9813120 559 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLLVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPQKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNQQVDKLVSAGIRK 1bqo B 2.3 BS06 N25 B 1 V163 L164 A165 H166 H201 E202 H205 H211 V81 L82 A83 H84 H119 E120 H123 H129 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=18.4nM remove_due_to_license_issue IC50=18nM, Ki=18nM P08254 9733482 401 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1br5 A 2.5 BS01 NEO A 1 Y80 V81 G121 Y123 I172 E177 R180 Y80 V81 G121 Y123 I172 E177 R180 V81 E177 R180 V81 E177 R180 3.2.2.22 0017148,0030598 Ki>2mM remove_due_to_license_issue P02879 9086280 500 IFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 1br6 A 2.3 BS01 PT1 A 1 N78 Y80 V81 G121 Y123 I172 S176 E177 R180 N79 Y81 V82 G122 Y124 I173 S177 E178 R181 V81 E177 R180 V82 E178 R181 3.2.2.22 0017148,0030598 Ki=0.6mM remove_due_to_license_issue P02879 9086280 301 MIFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 1bra A 2.2 BS02 BEN A 1 S190 Q192 S195 V213 G216 G219 S172 Q174 S177 V191 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=15000uM remove_due_to_license_issue P00763 8478942 246 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRKTLNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASYPGKITDNMVCVGFLEGGKGSCQGDSGGPVVCNGELQGIVSWGYGCALPDNPDVYTKVCNYVDWIQDTIAAN 1bsk A 3.0 BS02 MLN A 1 G43 I44 G45 Q50 E88 G89 L91 H132 E133 H136 G43 I44 G45 Q50 E88 G89 L91 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 3.5.1.88 0005515,0005829,0006412,0008198,0008270,0016787,0042586,0043022,0043686,0046872 remove_due_to_license_issue P0A6K3 10200158 171 SVLQVLHIPDERLRKVAKPVEEVNAEIQRIVDDMFETMYAEEGIGLAATQVDIHQRIIVIDVSENRDERLVLINPELLEKSGETGIEEGCLSIPEQRALVPRAEKVKIRALDRDGKPFELEADGLLAICIQHEMDHLVGKLFMDYLSPLKQQRIRQKVEKLDRLKA 1bsu A 2.0 BS01 dna C 0 T37 N70 K92 T93 T94 Y95 T106 G109 T111 S112 K119 S183 T186 N188 T36 N69 K91 T92 T93 Y94 T105 G108 T110 S111 K118 S175 T178 N180 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 902 ~ 911 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKENEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bsu A 2.0 BS02 dna D 0 Q69 N70 S183 G184 N185 S223 Q68 N69 S175 G176 N177 S215 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 801 ~ 811 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKENEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bsu B 2.0 BS01 dna C 0 Q69 N70 S183 G184 N185 S223 R226 Q64 N65 S168 G169 N170 S208 R211 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 902 ~ 911 SLRSDLINALYDEDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bsu B 2.0 BS02 dna D 0 T37 N70 K92 T93 T94 Y95 T106 G109 T111 S112 S183 T186 N188 T32 N65 K87 T88 T89 Y90 T96 G99 T101 S102 S168 T171 N173 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 801 ~ 811 SLRSDLINALYDEDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1btn A 2.0 BS01 I3P A 1 K8 R21 S22 W23 Y69 K71 K8 R21 S22 W23 Y69 K71 ? 0005543 Kd=40uM remove_due_to_license_issue Q62261 7588597 107 MEGFLNRKHEWEAHNKKASSRSWHNVYCVINNQEMGFYKDAKSAASGIPYHSEVPVSLKEAICEVALDYKKKKHVFKLRLSDGNEYLFQAKDDEEMNTWIQAISSA 1bua A 2.15 BS01 dna C 0 N70 K92 T93 T94 Y95 T106 T111 S112 K119 N120 S183 T186 N188 N68 K90 T91 T92 Y93 T100 T105 S106 K113 N114 S170 T173 N175 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 901 ~ 911 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPQQNHYPDFTLYKPSEPNKKIAIDIKTTYTEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bua A 2.15 BS02 dna D 0 Q69 S183 G184 N185 S223 Q67 S170 G171 N172 S210 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 801 ~ 811 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPQQNHYPDFTLYKPSEPNKKIAIDIKTTYTEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bua B 2.15 BS01 dna C 0 N70 S183 G184 N185 S223 N65 S168 G169 N170 S208 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 901 ~ 911 SLRSDLINALYDEDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bua B 2.15 BS02 dna D 0 N70 K92 T93 T94 Y95 T106 T111 S112 K119 S183 T186 N188 N65 K87 T88 T89 Y90 T97 T102 S103 K110 S168 T171 N173 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 10074946 801 ~ 811 SLRSDLINALYDEDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGR 1bug A 2.7 BS03 URS A 1 H88 H109 H240 H244 M258 N260 F261 H274 H88 H109 H240 H244 M258 N260 F261 H274 H88 H109 H118 H240 H244 F261 H274 H88 H109 H118 H240 H244 F261 H274 1.10.3.1 0004097,0016491 remove_due_to_license_issue Q9ZP19 9846879 1002 APIQAPEISKCVVPPADLPPGAVVDNCCPPVASNIVDYKLPAVTTMKVRPAAHTMDKDAIAKFAKAVELMKALPADDPRNFYQQALVHCAYCNGGYDQVNFPDQEIQVHNSWLFFPFHRWYLYFYERILGKLIGDPSFGLPFWNWDNPGGMVLPDFLNDSTSSLYDSNRNQSHLPPVVVDLGYNGADTDVTDQQRITDNLALMYKQMVTNAGTAELFLGKAYRAGDAPSPGAGSIETSPHIPIHRWVGDPRNTNNEDMGNFYSAGRDIAFYCHHSNVDRMWTIWQQLARDYTDSDWLNATFLFYDENGQAVKVRIGDSLDNQKMGYKYAKTPLPWL 1bux A 2.8 BS01 PPS A 1 K16 Y56 R62 F64 L68 T98 H122 K11 Y51 R57 F59 L63 T93 H117 K16 Y56 N119 H122 E133 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 9786875 160 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIHGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1bux B 2.8 BS01 PPS B 1 Y56 H59 F64 L68 T98 V116 N119 H122 Y51 H54 F59 L63 T93 V111 N114 H117 K16 Y56 N119 H122 E133 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 9786875 160 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIHGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1bv7 A 2.0 BS01 XV6 A 1 D25 G27 A28 D30 I47 G48 G49 I50 P81 F82 I84 D25 G27 A28 D30 I47 G48 G49 I50 P81 F82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.5nM remove_due_to_license_issue P04585 9790666 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNIIGRNLLTQIGCTLNF 1bv7 B 2.0 BS01 XV6 A 1 D25 G27 A28 D30 V32 I47 G48 G49 I50 F82 D25 G27 A28 D30 V32 I47 G48 G49 I50 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9790666 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNIIGRNLLTQIGCTLNF 1bv9 A 2.0 BS01 XV6 A 1 D25 G27 A28 D30 I47 G48 G49 I50 P81 V82 D25 G27 A28 D30 I47 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.1nM remove_due_to_license_issue P04585 9790666 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 1bv9 B 2.0 BS01 XV6 A 1 D25 G27 A28 D30 I47 G48 G49 I50 V82 D25 G27 A28 D30 I47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9790666 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 1bwa A 1.9 BS01 XV6 B 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9790666 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1bwa B 1.9 BS01 XV6 B 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 D25 G27 A28 D29 D30 V32 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2.5nM remove_due_to_license_issue P04585 9790666 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1bwb A 1.8 BS01 146 B 1 D25 G27 A28 D30 V32 K45 I47 G48 I50 P81 D25 G27 A28 D30 V32 K45 I47 G48 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9790666 641 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1bwb B 1.8 BS01 146 B 1 D25 G27 A28 D30 V32 M46 I47 G48 G49 I50 D25 G27 A28 D30 V32 M46 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.8nM remove_due_to_license_issue P04585 9790666 641 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1bwn A 2.1 BS02 4IP A 1 K12 S14 Q15 Q16 K17 K18 S21 P22 N24 K26 R28 Y39 K53 K11 S13 Q14 Q15 K16 K17 S20 P21 N23 K25 R27 Y38 K52 2.7.10.2 0035556 Kd=87nM remove_due_to_license_issue Q06187 10196129 1 AAVILESIFLKRSQQKKKTSPLNFKKRLFLLTVHKLSYYKYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIPRRGSEMEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQILEN 1bwn A 2.1 BS03 4IP A 2 K41 K53 K40 K52 2.7.10.2 0035556 Kd=87nM remove_due_to_license_issue Q06187 10196129 172 AAVILESIFLKRSQQKKKTSPLNFKKRLFLLTVHKLSYYKYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIPRRGSEMEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQILEN 1bwn B 2.1 BS02 4IP B 1 K12 S14 Q15 Q16 K17 K18 S21 N24 R28 Y39 K11 S13 Q14 Q15 K16 K17 S20 N23 R27 Y38 2.7.10.2 0035556 Kd=87nM remove_due_to_license_issue Q06187 10196129 1 AAVILESIFLKRSQQKKKTSPLNFKKRLFLLTVHKLSYYKYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIEMEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQILEN 1bwn B 2.1 BS03 4IP B 2 K41 K53 K40 K52 2.7.10.2 0035556 Kd=87nM remove_due_to_license_issue Q06187 10196129 172 AAVILESIFLKRSQQKKKTSPLNFKKRLFLLTVHKLSYYKYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIEMEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQILEN 1bxo A 0.95 BS02 PP7 A 1 E15 D33 G35 Y75 G76 D77 D213 G215 T216 T217 I297 E15 D33 G35 Y75 G76 D77 D213 G215 T216 T217 I297 D33 S36 D38 W40 Y75 D213 T216 D33 S36 D38 W40 Y75 D213 T216 3.4.23.20 0004190,0005576,0006508 Ki=0.1nM remove_due_to_license_issue P00798 9836576 324 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 1bxq A 1.41 BS01 PP8 A 1 E15 D33 Y75 G76 D77 I211 D213 G215 T216 T217 Y274 I293 I297 E15 D33 Y75 G76 D77 I211 D213 G215 T216 T217 Y274 I293 I297 D33 S36 D38 W40 Y75 D213 T216 D33 S36 D38 W40 Y75 D213 T216 3.4.23.20 0004190,0005576,0006508 Ki=42nM remove_due_to_license_issue P00798 9836576 324 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 1bxr A 2.1 BS04 ANP A 1 R129 I167 R169 M174 G175 G176 L210 I211 E215 M240 G241 H243 T244 Q285 E299 R306 T376 R129 I167 R169 M174 G175 G176 L210 I211 E215 M240 G241 H243 T244 Q285 E299 R306 T376 R129 R169 M174 G176 K202 E215 H243 N283 Q285 E299 N301 R303 S307 D338 G507 K634 R715 G721 G722 S745 E761 D769 Q829 E841 N843 R848 P901 R129 R169 M174 G176 K202 E215 H243 N283 Q285 E299 N301 R303 S307 D338 G507 K634 R715 G721 G722 S745 E761 D769 Q829 E841 N843 R848 P901 6.3.4.16,6.3.5.5 0000166,0004087,0004088,0005515,0005524,0005737,0005829,0005951,0006221,0006526,0006541,0008652,0016597,0016874,0019856,0044205,0046872 remove_due_to_license_issue P00968 10029528 1083 MPKRTDIKSILILGAGPIVIGQACEFDYSGAQACKALREEGYRVILVNSNPATIMTDPEMADATYIEPIHWEVVRKIIEKERPDAVLPTMGGQTALNCALELERQGVLEEFGVTMIGATADAIDKAEDRRRFDVAMKKIGLETARSGIAHTMEEALAVAADVGFPCIIRPSFTMGGSGGGIAYNREEFEEICARGLDLSPTKELLIDESLIGWKEYEMEVVRDKNDNCIIVCSIENFDAMGIHTGDSITVAPAQTLTDKEYQIMRNASMAVLREIGVETGGSNVQFAVNPKNGRLIVIEMNPRVSRSSALASKATGFPIAKVAAKLAVGYTLDELMNDITGGRTPASFEPSIDYVVTKIPRFNFEKFAGANDRLTTQMKSVGEVMAIGRTQQESLQKALRGLEVGATGFDPKVSLDDPEALTKIRRELKDAGADRIWYIADAFRAGLSVDGVFNLTNIDRWFLVQIEELVRLEEKVAEVGITGLNADFLRQLKRKGFADARLAKLAGVREAEIRKLRDQYDLHPVYKRVDTCAAEFATDTAYMYSTYEEECEANPSTDREKIMVLGGGPNRIGQGIEFDYCCVHASLALREDGYETIMVNCNPETVSTDYDTSDRLYFEPVTLEDVLEIVRIEKPKGVIVQYGGQTPLKLARALEAAGVPVIGTSPDAIDRAEDRERFQHAVERLKLKQPANATVTAIEMAVEKAKEIGYPLVVRPSYVLGGRAMEIVYDEADLRRYFQTAVSVSNDAPVLLDHFLDDAVEVDVDAICDGEMVLIGGIMEHIEQAGVHSGDSACSLPAYTLSQEIQDVMRQQVQKLAFELQVRGLMNVQFAVKNNEVYLIEVNPRAARTVPFVSKATGVPLAKVAARVMAGKSLAEQGVTKEVIPPYYSVKEVVLPFNKFPGVDPLLGPEMRSTGEVMGVGRTFAEAFAKAQLGSNSTMKKHGRALLSVREGDKERVVDLAAKLLKQGFELDATHGTAIVLGEAGINPRLVNKVHEGRPHIQDRIKNGEYTYIINTTSGRRAIEDSRVIRRSALQYKVHYDTTLNGGFATAMALNADATEKVISVQEMHAQIK 1bxr A 2.1 BS05 ANP A 2 R675 V713 R715 L720 G721 G722 M725 D753 F755 L756 E761 A785 G786 V787 H788 Q829 E841 N843 R848 R675 V713 R715 L720 G721 G722 M725 D753 F755 L756 E761 A785 G786 V787 H788 Q829 E841 N843 R848 R129 R169 M174 G176 K202 E215 H243 N283 Q285 E299 N301 R303 S307 D338 G507 K634 R715 G721 G722 S745 E761 D769 Q829 E841 N843 R848 P901 R129 R169 M174 G176 K202 E215 H243 N283 Q285 E299 N301 R303 S307 D338 G507 K634 R715 G721 G722 S745 E761 D769 Q829 E841 N843 R848 P901 6.3.4.16,6.3.5.5 0000166,0004087,0004088,0005515,0005524,0005737,0005829,0005951,0006221,0006526,0006541,0008652,0016597,0016874,0019856,0044205,0046872 remove_due_to_license_issue P00968 10029528 1084 MPKRTDIKSILILGAGPIVIGQACEFDYSGAQACKALREEGYRVILVNSNPATIMTDPEMADATYIEPIHWEVVRKIIEKERPDAVLPTMGGQTALNCALELERQGVLEEFGVTMIGATADAIDKAEDRRRFDVAMKKIGLETARSGIAHTMEEALAVAADVGFPCIIRPSFTMGGSGGGIAYNREEFEEICARGLDLSPTKELLIDESLIGWKEYEMEVVRDKNDNCIIVCSIENFDAMGIHTGDSITVAPAQTLTDKEYQIMRNASMAVLREIGVETGGSNVQFAVNPKNGRLIVIEMNPRVSRSSALASKATGFPIAKVAAKLAVGYTLDELMNDITGGRTPASFEPSIDYVVTKIPRFNFEKFAGANDRLTTQMKSVGEVMAIGRTQQESLQKALRGLEVGATGFDPKVSLDDPEALTKIRRELKDAGADRIWYIADAFRAGLSVDGVFNLTNIDRWFLVQIEELVRLEEKVAEVGITGLNADFLRQLKRKGFADARLAKLAGVREAEIRKLRDQYDLHPVYKRVDTCAAEFATDTAYMYSTYEEECEANPSTDREKIMVLGGGPNRIGQGIEFDYCCVHASLALREDGYETIMVNCNPETVSTDYDTSDRLYFEPVTLEDVLEIVRIEKPKGVIVQYGGQTPLKLARALEAAGVPVIGTSPDAIDRAEDRERFQHAVERLKLKQPANATVTAIEMAVEKAKEIGYPLVVRPSYVLGGRAMEIVYDEADLRRYFQTAVSVSNDAPVLLDHFLDDAVEVDVDAICDGEMVLIGGIMEHIEQAGVHSGDSACSLPAYTLSQEIQDVMRQQVQKLAFELQVRGLMNVQFAVKNNEVYLIEVNPRAARTVPFVSKATGVPLAKVAARVMAGKSLAEQGVTKEVIPPYYSVKEVVLPFNKFPGVDPLLGPEMRSTGEVMGVGRTFAEAFAKAQLGSNSTMKKHGRALLSVREGDKERVVDLAAKLLKQGFELDATHGTAIVLGEAGINPRLVNKVHEGRPHIQDRIKNGEYTYIINTTSGRRAIEDSRVIRRSALQYKVHYDTTLNGGFATAMALNADATEKVISVQEMHAQIK 1by4 A 2.1 BS01 dna E 0 K1145 H1146 K1160 R1209 K15 H16 K30 R79 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 1495 ~ 1509 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 A 2.1 BS02 dna F 0 E1153 R1161 N1185 Q1188 R1191 E23 R31 N55 Q58 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 1531 ~ 1545 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 B 2.1 BS01 dna E 0 K1245 H1246 R1264 Q1306 R1309 K18 H19 R37 Q79 R82 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 1495 ~ 1509 GSFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 B 2.1 BS02 dna F 0 E1253 G1254 R1261 R1284 N1285 R1291 E26 G27 R34 R57 N58 R64 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 1531 ~ 1545 GSFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 B 2.1 BS03 dna G 0 N1285 R1286 N58 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 2494 ~ 2509 GSFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 C 2.1 BS01 dna G 0 K2145 H2146 K2156 K14 H15 K25 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 2494 ~ 2509 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 C 2.1 BS02 dna H 0 E2153 F2158 R2161 R2184 N2185 Q2188 R2191 E22 F27 R30 R53 N54 Q57 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 2531 ~ 2545 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 1by4 D 2.1 BS01 dna G 0 K2245 H2246 Y2247 R2264 V2305 Q2306 K17 H18 Y19 R36 V77 Q78 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 2494 ~ 2509 SFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEE 1by4 D 2.1 BS02 dna H 0 E2253 G2254 F2258 R2261 R2284 N2285 Q2288 R2291 E25 G26 F30 R33 R56 N57 Q60 R63 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 10669605 2531 ~ 2545 SFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEE 1bzc A 2.35 BS01 TPI A 1 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 Y45 D47 D180 F181 C214 S215 A216 I218 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=12uM remove_due_to_license_issue P18031 9922143 902 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTAEQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1bzf A -1.00 BS01 TMQ A 1 L4 L19 D26 L27 F30 F49 A97 L4 L19 D26 L27 F30 F49 A97 L4 L19 W21 D26 L27 F30 L54 L94 T116 L4 L19 W21 D26 L27 F30 L54 L94 T116 1.5.1.3 0004146,0005829,0006730,0016491,0031427,0046452,0046654,0046655,0046677,0050661 remove_due_to_license_issue P00381 10091649 170 TAFLWAQDRDGLIGKDGHLPWHLPDDLHYFRAQTVGKIMVVGRRTYESFPKRPLPERTNVVLTHQEDYQAQGAVVVHDVAAVFAYAKQHPDQELVIAGGAQIFTAFKDDVDTLLVTRLAGSFEGDTKMIPLNWDDFTKVSSRTVEDTNPALTHTYEVWQKKA 1bzj A 2.25 BS01 PIC A 1 Y46 V49 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 V48 D180 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=22uM remove_due_to_license_issue Ki=22000nM P18031 9922143 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1bzs A 1.7 BS05 BSI A 1 I159 L160 A161 H197 E198 H201 H207 L214 P217 N218 Y219 I81 L82 A83 H119 E120 H123 H129 L136 P139 N140 Y141 H197 E198 H201 H207 H119 E120 H123 H129 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=10nM remove_due_to_license_issue P22894 10354399 250 FMLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYGD 1bzy A 2.0 BS01 IMU A 1 Y104 E133 D134 I135 D137 T138 G139 K140 T141 K165 F186 V187 L192 D193 Y101 E130 D131 I132 D134 T135 G136 K137 T138 K162 F183 V184 L189 D190 E133 D134 D137 F186 R199 E130 D131 D134 F183 R196 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Kd=4.6nM remove_due_to_license_issue Ki=4.6nM P00492 10360366 300 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSYCNDQSTGDIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 1c12 A 2.6 BS01 TRZ A 1 V89 Y91L F96L F98L V89 Y91 F96 F98 ? 0005576,0005886,0030183 remove_due_to_license_issue P01837 10525411 215 DIELTQSPSSMSVSLGDTVSITCHASQGISSNIGWLQQKPGKSFKGLIYHGTNLEDGVPSRFSGSGSGADYSLTISSLESEDFADYYCVQYVQFPFTFGSGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEA 1c12 B 2.6 BS01 TRZ A 1 N35H V393 L96H N36 V97 L100 ? remove_due_to_license_issue P01869 10525411 215 QVQLQESGPGLVKPSQSLSLTCTVTGYSITSDYAWNWIRQFPGNKLEWMGYISYSGSTSYSPSLKSRISLTRDTSKNQFFLQLNSVTTEDTATYYCVTSLTWLLRRKRSYWGQGTTVTVSSASTKGPSVYPLAPGSKAAASMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPE 1c1r A 1.37 BS04 BAI A 1 D189 S190 V213 G219 C220 D171 S172 V191 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.0235uM remove_due_to_license_issue P00760 9468142 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1c1u H 1.75 BS03 BAI H 1 K60F D195 A196 E198 S201 G222 K52 D192 A193 E195 S198 G221 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 9468142 410 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1c1v H 1.98 BS03 BAB H 1 K60F D195 A196 E198 W221 G222 G225 K52 D192 A193 E195 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.023uM remove_due_to_license_issue P00734 9468142 410 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1c29 A 2.3 BS01 HE1 A 1 F22 D60 L100 Y175 T183 G184 F212 G213 G234 S235 F21 D59 L99 Y174 T182 G183 F209 G210 G231 S232 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 ic50=472nM remove_due_to_license_issue P00929 10504236 270 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1c2t B 2.1 BS01 NHS B 1 R64 F88 M89 R90 I91 L92 N106 H108 L118 V139 T140 D141 L143 D144 R64 F88 M89 R90 I91 L92 N106 H108 L118 V139 T140 D141 L143 D144 N106 H108 S135 D144 N106 H108 S135 D144 2.1.2.2 0003824,0004644,0005737,0005829,0006164,0006189,0006974,0009058,0016740 Ki=260nM remove_due_to_license_issue P08179 10606510 220 MNIVVLISGNGSNLQAIIDACKTNKIKGTVRAVFSNKADAFGLERARQAGIATHTLIASAFDSREAYDRELIHEIDMYAPDVVVLAGFMRILSPAFVSHYAGRLLNIHPSLLPKYPGLHTHRQALENGDEEHGTSVHFVTDELDGGPVILQAKVPVFAGDSEDDITARVQTQEHAIYPLVISWFADGRLKMHENAAWLDGQRLPPQGYA 1c3b A 2.25 BS01 BZB A 1 S64 Y150 N152 Y221 G317 A318 S61 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue IC50=200nM, Ki=27nM P00811 10595535 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1c3e A 2.1 BS01 NHR A 1 R64 F88 M89 R90 I91 L92 N106 H108 L118 V139 T140 L143 D144 R64 F88 M89 R90 I91 L92 N106 H108 L118 V139 T140 L143 D144 N106 H108 S135 D144 N106 H108 S135 D144 2.1.2.2 0003824,0004644,0005737,0005829,0006164,0006189,0006974,0009058,0016740 remove_due_to_license_issue P08179 10606510 220 MNIVVLISGNGSNLQAIIDACKTNKIKGTVRAVFSNKADAFGLERARQAGIATHTLIASAFDSREAYDRELIHEIDMYAPDVVVLAGFMRILSPAFVSHYAGRLLNIHPSLLPKYPGLHTHRQALENGDEEHGTSVHFVTDELDGGPVILQAKVPVFAGDSEDDITARVQTQEHAIYPLVISWFADGRLKMHENAAWLDGQRLPPQGYA 1c3i B 1.83 BS06 TR1 B 1 N162 V163 L164 A165 V198 H201 E202 H205 H211 L218 Y220 P221 L222 Y223 N80 V81 L82 A83 V116 H119 E120 H123 H129 L136 Y138 P139 L140 Y141 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P08254 10877850 1 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1c3r A 2.0 BS02 TSN A 1 P22 H131 H132 F141 D168 H170 Y297 P21 H130 H131 F140 D167 H169 Y296 ? 0004407,0040029,0045149,0045150,0046872 remove_due_to_license_issue O67135 10490031 502 KKVKLIGTLDYGKYRYPKNHPLKIPRVSLLLRFKDAMNLIDEKELIKSRPATKEELLLFHTEDYINTLMEAERSQSVPKGAREKYNIGGYENPVSYAMFTGSSLATGSTVQAIEEFLKGNVAFNPAGGMHHAFKSRANGFCYINNPAVGIEYLRKKGFKRILYIDLDAHHCDGVQEAFYDTDQVFVLSLHQSPEYAFPFEKGFLEEIGEGKGKGYNLNIPLPKGLNDNEFLFALEKSLEIVKEVFEPEVYLLQLGTDPLLEDYLSKFNLSNVAFLKAFNIVREVFGEGVYLGGGGYHPYALARAWTLIWCELSGREVPEKLNNKAKELLKSIDFEEFDDEVDRSYMLETLKDPWRGGEVRKEVKDTLEKAKA 1c3r B 2.0 BS02 TSN B 1 P22 H131 H132 F141 D168 H170 Y297 P21 H130 H131 F140 D167 H169 Y296 ? 0004407,0040029,0045149,0045150,0046872 remove_due_to_license_issue O67135 10490031 504 KKVKLIGTLDYGKYRYPKNHPLKIPRVSLLLRFKDAMNLIDEKELIKSRPATKEELLLFHTEDYINTLMEAERSQSVPKGAREKYNIGGYENPVSYAMFTGSSLATGSTVQAIEEFLKGNVAFNPAGGMHHAFKSRANGFCYINNPAVGIEYLRKKGFKRILYIDLDAHHCDGVQEAFYDTDQVFVLSLHQSPEYAFPFEKGFLEEIGEGKGKGYNLNIPLPKGLNDNEFLFALEKSLEIVKEVFEPEVYLLQLGTDPLLEDYLSKFNLSNVAFLKAFNIVREVFGEGVYLGGGGYHPYALARAWTLIWCELSGREVPEKLNNKAKELLKSIDFEEFDDEVDRSYMLETLKDPWRGGEVRKEVKDTLEKAKA 1c3x A 2.4 BS02 8IG A 1 G135 C136 G137 Y203 E204 G221 M222 T245 G119 C120 G121 Y187 E188 G205 M206 T229 S46 R83 H105 Y107 E108 G135 M222 S223 N246 H258 S38 R67 H89 Y91 E92 G119 M206 S207 N230 H242 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0016763 remove_due_to_license_issue P81989 10600382 306 PPLDDPATDPFLVARAAADHIAQATGVEGHDMALVLGSGWGGAAELLGEVVAEVPTHEIPGFSSVTRSIRVERADGSVRHALVLGSRTHLYEGKGVRAVVHGVRTAAATGAETLILTNGCGGLNQEWGAGTPVLLSDHINLTARSPLEGPTFVDLTDVYSPRLRELAHRVDPTLPEGVYAQFPGPHYETPAEVRMAGILGADLVGMSTTLEAIAARHCGLEVLGVSLVTNLAAGISPTPLSHAEVIEAGQAAGPRISALLADIAKR 1c3x B 2.4 BS03 8IG B 1 G135 C136 G137 Y203 E204 G221 M222 T245 G119 C120 G121 Y187 E188 G205 M206 T229 S46 R83 H105 Y107 E108 G135 M222 S223 N246 H258 S38 R67 H89 Y91 E92 G119 M206 S207 N230 H242 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0016763 remove_due_to_license_issue P81989 10600382 305 PPLDDPATDPFLVARAAADHIAQATGVEGHDMALVLGSGWGGAAELLGEVVAEVPTHEIPGFSSVTRSIRVERADGSVRHALVLGSRTHLYEGKGVRAVVHGVRTAAATGAETLILTNGCGGLNQEWGAGTPVLLSDHINLTARSPLEGPTFVDLTDVYSPRLRELAHRVDPTLPEGVYAQFPGPHYETPAEVRMAGILGADLVGMSTTLEAIAARHCGLEVLGVSLVTNLAAGISPTPLSHAEVIEAGQAAGPRISALLADIAKR 1c4u 2 2.1 BS02 IH1 2 1 H57 Y60A W60D E97A N98 L99 D189 A190 S214 W215 G216 G219 H43 Y47 W50 E94 N95 L96 D192 A193 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.043nM remove_due_to_license_issue P00734 10713516 370 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1c4v 2 2.1 BS02 IH2 2 1 H57 Y60A W60D N98 I174 D189 A190 S195 V213 S214 W215 G216 E217 H43 Y47 W50 N95 I172 D192 A193 S198 V218 S219 W220 G221 E222 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.016nM remove_due_to_license_issue P00734 10713516 370 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1c4y 2 2.7 BS03 IH3 2 1 H57 Y60A W60D L99 R173 I174 D189 A190 V213 W215 G216 E217 H43 Y47 W50 L96 R174 I175 D195 A196 V221 W223 G224 E225 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10713516 370 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTAGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1c50 A 2.3 BS02 CHI A 1 R60 V64 W67 W189 E190 K191 P229 R48 V52 W55 W177 E178 K179 P217 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=334nM remove_due_to_license_issue P00489 10873856 920 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1c5c H 1.61 BS01 TK4 L 1 H35 I95 A101 H35 I99 A100 remove_due_to_license_issue 11183784 1001 QVQLLEPGTELVKPGASVKLSCRASGYSFTSYWMHWVKQRPGQGLEWIGLIDPSNGRTNFNDKFKSRATLTVDTSSSTAYMQLSSLTSEDSAVYYCVRIAYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 1c5c L 1.61 BS01 TK4 L 1 S34 R46 L89 Y91 R96 S34 R46 L89 Y91 R96 Kd=110nM remove_due_to_license_issue 11183784 1001 EIQLTQSPSSLSASLGERVSLTCRTSQEISGYLSWLQQKPDGTIKRLIYDATKLDSGAPKRFSGSRSGSDYSLTISSLESEDFADYYCLQYASFPRTFGGGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 1c5n H 1.5 BS03 ESI H 1 D189 S195 G216 G219 D192 S198 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=20uM remove_due_to_license_issue Ki=20000nM P00734 10779411 522 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1c5q A 1.43 BS02 ESI A 1 D189 S190 S195 W215 G216 G219 C220 D171 S172 S177 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.44uM remove_due_to_license_issue Ki=440nM P00760 10779411 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1c5s A 1.36 BS02 ESX A 1 D189 S190 C191 Q192 S195 W215 G216 G219 D171 S172 C173 Q174 S177 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1uM remove_due_to_license_issue Ki=1000nM P00760 10779411 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1c5t A 1.37 BS02 ESP A 1 D189 S190 Q192 S195 W215 D171 S172 Q174 S177 W193 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=80uM remove_due_to_license_issue Ki=80000nM P00760 10779411 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1c5x B 1.75 BS02 ESI B 1 D189 S190 Q192 S195 W215 G216 G219 C220 G226 D192 S193 Q195 S198 W218 G219 G221 C222 G229 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.21uM remove_due_to_license_issue Ki=210nM P00749 10779411 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEE 1c5y B 1.65 BS02 ESP B 1 D189 S190 Q192 S195 W215 G216 G219 C220 D192 S193 Q195 S198 W218 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=63uM remove_due_to_license_issue Ki=63000nM P00749 10779411 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEE 1c6y A 2.5 BS01 MK1 B 1 D25 G48 G49 I50 T82 D25 G48 G49 I50 T82 3.4.24.- 0004190,0006508 remove_due_to_license_issue O09893 10739910 524 PQITLWQRPVVTIKIGGQLMEALIDTGADDTVLEEMDLPGRWKPKIIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPTNIIGRNLLTQIGCTLNF 1c6y B 2.5 BS01 MK1 B 1 D225 G227 A228 D229 D230 V232 G248 P281 I284 D25 G27 A28 D29 D30 V32 G48 P81 I84 D225 T226 G227 D25 T26 G27 3.4.24.- 0004190,0006508 Ki=0.31nM remove_due_to_license_issue O09893 10739910 524 PQITLWQRPVVTIKIGGQLMEALIDTGADDTVLEEMDLPGRWKPKIIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPTNIIGRNLLTQIGCTLNF 1c70 A 2.5 BS01 L75 B 1 R8 D25 G27 G49 I50 V82 R8 D25 G27 G49 I50 V82 3.4.23.- 0004190,0006508 remove_due_to_license_issue O92103 10739910 423 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1c70 B 2.5 BS01 L75 B 1 D225 G227 A228 D229 D230 V232 G248 G249 T280 P281 D25 G27 A28 D29 D30 V32 G48 G49 T80 P81 D225 T226 G227 D25 T26 G27 3.4.23.- 0004190,0006508 Ki=0.05nM remove_due_to_license_issue O92103 10739910 423 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1c7f A 2.0 BS01 FMN A 1 S10 T11 T12 N14 T15 S58 T59 W60 G94 E95 Y98 F101 S9 T10 T11 N13 T14 S57 T58 W59 G93 E94 Y97 F100 ? 0009055,0010181 Kd=0.3nM remove_due_to_license_issue P00323 12206666 1149 PKALIVYGSTTGNTEYTAETIARELADAGYEVDSRDAASVEAGGLFEGFDLVLLGCSTWGDDSIELQDDFIPLFDSLEETGAQGRKVACFGCGESSYEYFCGAVDAIEEKLKNLGAEIVQDGLRIDGDPRAARDDIVGWAHDVRGAI 1c83 A 1.8 BS01 OAI A 1 Y46 V49 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 V48 K119 D180 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=14uM remove_due_to_license_issue Ki=7943.28nM P18031 10702277 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1c84 A 2.35 BS01 761 A 1 Y46 V49 D181 F182 C215 S216 A217 I219 G220 R221 Y45 V48 D180 F181 C214 S215 A216 I218 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=9.9uM remove_due_to_license_issue Ki=10000nM P18031 10702277 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1c85 A 2.72 BS01 OBA A 1 Y46 D181 F182 C215 S216 A217 G220 R221 Y45 D180 F181 C214 S215 A216 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=22908.68nM P18031 10702277 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1c86 A 2.3 BS01 OPA A 1 Y46 N48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y44 N46 K118 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 Ki=20uM remove_due_to_license_issue Ki=71449632607551nM P18031 10744717 301 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYVNVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1c87 A 2.1 BS01 OPA A 1 Y46 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 K119 D180 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=63uM remove_due_to_license_issue Ki=71449632607551nM P18031 10744717 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1c88 A 1.8 BS01 OTA A 1 Y46 D48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 D47 K119 D180 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=5.1uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 10744717 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1c8k A 1.76 BS02 CPB A 1 F285 E382 A610 G612 Y613 F273 E370 A598 G600 Y601 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=1uM remove_due_to_license_issue IC50=1200nM P00489 10924512 940 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1c8l A 2.3 BS02 BIN A 1 I68 Q71 Q72 Y75 R193 F196 R309 R310 I64 Q67 Q68 Y71 R189 F192 R296 R297 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=6.9nM remove_due_to_license_issue P00489 11368311 930 SDQEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 1c8v A 2.2 BS01 HE1 A 1 F22 D60 L100 Y175 T183 G184 F212 G234 S235 F21 D59 L99 Y174 T182 G183 F209 G231 S232 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 ic50=472nM remove_due_to_license_issue P00929 10504236 270 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1c9d A 2.3 BS01 HF1 A 1 D60 L100 Y175 T183 G184 F212 G234 S235 D59 L99 Y174 T182 G183 F209 G231 S232 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 ic50=499nM remove_due_to_license_issue P00929 10504236 270 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1ca8 B 2.1 BS03 0KV B 1 H57 Y60A W60D I174 D189 C191 S195 S214 W215 G216 G219 H42 Y46 W49 I170 D190 C192 S196 S217 W218 G219 G221 H57 D102 E192 G193 D194 S195 G196 H42 D98 E193 G194 D195 S196 G197 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=0.67nM P00734 9724521 248 IVEGSDAEIGMSPWQVMLFRKPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1caq A 1.8 BS06 DPS A 1 L164 A165 H201 E202 H205 H211 P221 L222 Y223 H224 L226 L82 A83 H119 E120 H123 H129 P139 L140 Y141 H142 L144 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=19nM remove_due_to_license_issue P08254 10422833 502 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPP 1cbr A 2.9 BS01 REA A 1 L120 R131 Y133 L120 R131 Y133 ? 0005501,0005737,0008289,0016918,0019841 remove_due_to_license_issue Kd=>200nM P62965 7704533 200 PNFAGTWKMRSSENFDELLKALGVNAMLRKVAVAAASKPHVEIRQDGDQFYIKTSTTVRTTEINFKVGEGFEEETVDGRKCRSLPTWENENKIHCTQTLLEGDGPKTYWTRELANDELILTFGADDVVCTRIYVRE 1cbr B 2.9 BS01 REA B 1 L120 R131 Y133 L120 R131 Y133 ? 0005501,0005737,0008289,0016918,0019841 remove_due_to_license_issue Kd=>200nM P62965 7704533 200 PNFAGTWKMRSSENFDELLKALGVNAMLRKVAVAAASKPHVEIRQDGDQFYIKTSTTVRTTEINFKVGEGFEEETVDGRKCRSLPTWENENKIHCTQTLLEGDGPKTYWTRELANDELILTFGADDVVCTRIYVRE 1cbx A 2.0 BS02 BZS A 1 H69 R127 N144 R145 H196 I243 Y248 E270 H69 R127 N144 R145 H196 I243 Y248 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=0.45uM remove_due_to_license_issue Ki=500nM P00730 1738164 500 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 1ce5 A 1.9 BS02 BEN A 1 D189 S190 Q192 S195 V213 G219 D171 S172 Q174 S177 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=18.4uM remove_due_to_license_issue P00760 10651279 703 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1cea A 2.06 BS01 ACA A 1 D54 D56 W61 Y63 R70 Y71 D55 D57 W62 Y64 R71 Y72 3.4.21.7 Kd~11uM remove_due_to_license_issue Ki=53000000nM, Kd=9000nM, IC50=105000nM P00747 8611560 90 ECKTGNGKNYRGTMSKTKNGITCQKWSSTSPHRPRFSPATHPSEGLEENYCRNPDNDPQGPWCYTTDPEKRYDYCDILEC 1cea B 2.06 BS01 ACA B 1 R34 F35 D54 D56 W61 Y63 R70 Y71 R35 F36 D55 D57 W62 Y64 R71 Y72 3.4.21.7 Kd~11uM remove_due_to_license_issue Ki=53000000nM, Kd=9000nM, IC50=105000nM P00747 8611560 90 ECKTGNGKNYRGTMSKTKNGITCQKWSSTSPHRPRFSPATHPSEGLEENYCRNPDNDPQGPWCYTTDPEKRYDYCDILEC 1ceb A 2.07 BS01 AMH A 1 R34 D54 D56 W61 Y63 R70 Y71 R35 D55 D57 W62 Y64 R71 Y72 3.4.21.7 Kd~1uM remove_due_to_license_issue Kd=1100nM, IC50=3100nM, Ki=25000000nM P00747 8611560 90 ECKTGNGKNYRGTMSKTKNGITCQKWSSTSPHRPRFSPATHPSEGLEENYCRNPDNDPQGPWCYTTDPEKRYDYCDILEC 1cet A 2.05 BS01 CLQ A 1 V26 G27 F52 D53 I54 Y85 A98 I119 E122 V9 G10 F33 D34 I35 Y66 A79 I94 E97 R109 D168 R171 H195 R84 D144 R147 H171 1.1.1.27 0003824,0004459,0006089,0006090,0016491,0016616,0019752 Ki=1.3mM remove_due_to_license_issue Q27743 10187806 1001 APKAKIVLVGSGMIGGVMATLIVQKNLGDVVLFDIVKNMPHGKALDTSHTNVMAYSNCKVSGSNTYDDLAGSDVVIVTAGFTNRLDLLPLNNKIMIEIGGHIKKNCPNAFIIVVTNPVDVMVQLLHQHSGVPKNKIIGLGGVLDTSRLKYYISQKLNVCPRDVNAHIVGAHGNKMVLLKRYITVGGIPLQEFINNKLISDAELEAIFDRTVNTALEIVNLHASPYVAPAAAIIEMAESYLKDLKKVLICSTLLEGQYGHSDIFGGTPVVLGANGVEQVIELQLNSEEKAKFDEAIAETKRMKALA 1cgl A 2.4 BS04 0ED A 1 G179 N180 L181 A182 H183 Y210 H218 E219 H228 P238 S239 Y240 G79 N80 L81 A82 H83 Y110 H118 E119 H128 P138 S139 Y140 H218 E219 H222 H228 H118 E119 H122 H128 3.4.24.7 0004222,0006508,0008237,0008270,0031012 Ki=135nM remove_due_to_license_issue P03956 8278810 1 VLTEGNPRWEQTHLRYRIENYTPDLPRADVDHAIEKAFQLWSDVTPLTFTKVSEGQADIMISFVRGDHRDNSPFDGPGGNLAHAFDPGPGIGGDAHFDEDERWTNNFREYNLHRVAAHELGHSLGLSHSTDIGALMYPSYTFSGDVQLAQDDIDGIQAIYGRSQNPVQ 1cgl A 2.4 BS05 0ED B 1 G179 T230 P238 S239 G79 T130 P138 S139 H218 E219 H222 H228 H118 E119 H122 H128 3.4.24.7 0004222,0006508,0008237,0008270,0031012 Ki=135nM remove_due_to_license_issue P03956 8278810 1 VLTEGNPRWEQTHLRYRIENYTPDLPRADVDHAIEKAFQLWSDVTPLTFTKVSEGQADIMISFVRGDHRDNSPFDGPGGNLAHAFDPGPGIGGDAHFDEDERWTNNFREYNLHRVAAHELGHSLGLSHSTDIGALMYPSYTFSGDVQLAQDDIDGIQAIYGRSQNPVQ 1ch8 A 2.5 BS02 GPX A 1 D13 G15 K16 G17 G40 H41 T42 K49 R305 K331 D333 S414 G416 P417 D13 G15 K16 G17 G40 H41 T42 K49 R305 K331 D333 S414 G416 P417 D13 K16 G40 H41 Q224 D13 K16 G40 H41 Q224 6.3.4.4 0000166,0000287,0004019,0005515,0005525,0005737,0005829,0006164,0006974,0015949,0016020,0016874,0044208,0046040,0046086,0046872,0097216 remove_due_to_license_issue P0A7D4 10364182 432 GNNVVVLGTQWGDEGKGKIVDLLTERAKYVVRYQGGHNAGHTLVINGEKTVLHLIPSGILRENVTSIIGNGVVLSPAALMKEMKELEDRGIPVRERLLLSEACPLILDYHVALDNAREKARGAKAIGTTGRGIGPAYEDKVARRGLRVGDLFDKETFAEKLKEVMEYHNFQLVNYYKAEAVDYQKVLDDTMAVADILTSMVVDVSDLLDQARQRGDFVMFEGAQGTLLDIDHGTYPYVTSSNTTAGGVATGSGLGPRYVDYVLGILKAYSTRVGAGPFPTELFDETGEFLCKQGNEFGATTGRRRRTGWLDTVAVRRAVQLNSLSGFCLTKLDVLDGLKEVKLCVAYRMPDGREVTTTPLAADDWKGVEPIYETMPGWSESTFGVKDRSGLPQAALNYIKRIEELTGVPIDIISTGPDRTETMILRDPFDA 1cil A 1.6 BS02 ETS A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.372nM remove_due_to_license_issue Ki=9nM, IC50=26.61nM, Kd=0.043000nM P00918 8142888 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1cim A 2.1 BS02 PTS A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.52nM remove_due_to_license_issue Ki=1.5nM P00918 8142888 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1cin A 2.1 BS02 MTS A 1 H64 H94 H96 H119 F131 L198 T199 T200 H61 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.88nM remove_due_to_license_issue Ki=1.9nM P00918 8142888 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1cit A 2.7 BS01 dna B 0 Q242 H243 Y244 K253 V302 R303 G309 R310 R311 G312 R313 Q13 H14 Y15 K24 V73 R74 G80 R81 R82 G83 R84 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22829 10331876 402 ~ 417 GRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKSAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKP 1cit A 2.7 BS02 dna C 0 E250 G251 F255 R258 R281 N282 R288 R310 R311 G312 R313 P315 S316 K317 E21 G22 F26 R29 R52 N53 R59 R81 R82 G83 R84 P86 S87 K88 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22829 10331876 419 ~ 434 GRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKSAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKP 1ciz A 1.64 BS06 DPS A 1 L164 A165 L197 H201 E202 H205 H211 P221 L222 Y223 H224 F232 L82 A83 L115 H119 E120 H123 H129 P139 L140 Y141 H142 F150 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=36nM remove_due_to_license_issue P08254 10422833 307 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPP 1cj1 A 3.0 BS01 C78 A 1 R67 R86 S88 S90 S96 Q106 H107 F108 K109 L120 W121 R11 R30 S32 S34 S40 Q50 H51 F52 K53 L64 W65 ? remove_due_to_license_issue P62993 10395476 155 PHPWFFGKIPRAKAEEMLSKQRHDGAFLIRESESAPGDFSLSVKFGNDVQHFKVLRDGAGKYFLWVVKFNSLNELVDYHRSTSVSRNQQIFLRDIE 1clu A 1.7 BS01 DBG A 1 P12 G13 G15 K16 S17 A18 F28 V29 D30 N116 K117 D119 S145 A146 P12 G13 G15 K16 S17 A18 F28 V29 D30 N110 K111 D113 S139 A140 3.6.5.2 0003924,0005525,0007165,0016020 Kd=5.4nM remove_due_to_license_issue P01112 10359839 167 MTEYKLVVVGAPGVGKSALTIQLIQNHFVDEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHQYREQIKRVKDSDDVPMVLVGNKCDLAARTVESRQAQDLARSYGIPYIETSAKTRQGVEDAFYTLVREIRQH 1cnw A 2.0 BS02 EG1 A 1 H94 H119 V121 V135 L198 T199 T200 P202 H91 H116 V118 V131 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=19nM remove_due_to_license_issue P00918 7608893 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1cnx A 1.9 BS02 EG2 A 1 H94 H119 V121 V135 L198 T199 T200 H91 H116 V118 V131 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=43nM remove_due_to_license_issue P00918 7608893 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1cny A 2.3 BS02 EG3 A 1 H94 H119 V135 L198 T199 T200 P202 W209 H91 H116 V131 L194 T195 T196 P198 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=14nM remove_due_to_license_issue P00918 7608893 555 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1cp6 A 1.9 BS03 BUB A 1 E151 Y225 C227 E151 Y225 C227 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=10uM remove_due_to_license_issue Q01693 10413478 601 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 1cps A 2.25 BS02 CPM A 1 N144 R145 H196 I243 T268 E270 N144 R145 H196 I243 T268 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=0.22uM remove_due_to_license_issue P00730 1527041 588 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 1cqp A 2.6 BS02 803 A 1 L132 I235 Y257 L298 L302 L5 I108 Y130 L171 L175 ? remove_due_to_license_issue Kd=12900nM, IC50=2400nM P20701 10493852 311 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 1cqp A 2.6 BS03 803 B 1 V308 I309 V181 I182 ? remove_due_to_license_issue Kd=12900nM, IC50=2400nM P20701 10493852 311 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 1cr6 A 2.8 BS01 CPU A 1 D333 W334 V337 M361 I416 Y465 D276 W277 V280 M304 I359 Y408 F265 D333 W334 N357 I376 Y381 Y465 D495 H523 F208 D276 W277 N300 I319 Y324 Y408 D438 H466 3.1.3.76,3.3.2.10 0000287,0003824,0004301,0005737,0005777,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0090181,0097176 remove_due_to_license_issue P34914 10485878 1100 RVAAFDLDGVLALPSIGPTEQLMKGKITFSQWQIFSQAMAARSINRPMLQAAIALKKKGFTTCIVTNNWLDDGDKRDSLAQMMCELSQHFDFLIESCQVGMIKPEPQIYNFLLDTLKAKPNEVVFLDDFGSNLKPARDMGMVTILVHNTASALRELEKVTGTQFPEAPLPVPCNPNDVSHGYVTVKPGIRLHFVEMGSGPALCLCHGFPESWFSWRYQIPALAQAGFRVLAIDMKGYGDSSSPPEIEEYAMELLCKEMVTFLDKLGIPQAVFIGHDWAGVMVWNMALFYPERVRAVASLNTPFMPPDPDVSPMKVIRSIPVFNYQLYFQEPGVAEAELEKNMSRTFKSFFRASDETGFIAVHKATEIGGILVNTPEDPNLSKITTEEEIEFYIQQFKKTGFRGPLNWYRNTERNWKWSCKGLGRKILVPALMVTAEKDIVLRPEMSKNMEKWIPFLKRGHIEDCGHWTQIEKPTEVNQILIKWLQTE 1cs4 A 2.5 BS04 101 B 1 T401 L438 D440 T25 L62 D64 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P30803 11087399 1082 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1cs4 B 2.5 BS03 101 B 1 K938 D1018 N1025 S1028 K61 D131 N138 S141 S891 I892 S942 R1029 K1065 S14 I15 S65 R142 K178 4.6.1.1 0009190,0016849,0035556 ic50=2.7uM remove_due_to_license_issue P26769 11087399 1082 YHQSYDCVCVMFASIPDFKEFYTESDVNKEGLECLRLLNEIIADFDDLLSKPKFSGVEKIKTIGSTYMAATGLSAIRQYMHIGTMVEFAYALVGKLDAINKHSFNDFKLRVGINHGPVIAGVIGAQKPQYDIWGNTVNVASRMDSTGVLDKIQVTEETSLILQTLGYTCTCRGIINVKGKGDLKTYFVNT 1csh A 1.65 BS02 AMX A 1 R46 L273 H274 A277 V314 V315 G317 Y318 G319 H320 A321 K366 A367 K368 N373 D375 R44 L271 H272 A275 V312 V313 G315 Y316 G317 H318 A319 K364 A365 K366 N371 D373 S244 H274 H320 R329 D375 S242 H272 H318 R327 D373 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 Ki=28nM remove_due_to_license_issue P23007 8011640 700 STNLKDVLASLIPKEQARIKTFRQQHGNTAVGQITVDMSYGGMRGMKGLIYETSVLDPDEGIRFRGFSIPECQKLLPKAGGGEEPLPEGLFWLLVTGQIPTPEQVSWVSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGINRTKYWEFVYEDAMDLIAKLPCVAAKIYRNLYRAGSSIGAIDSKLDWSHNFTNMLGYTDPQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLLWLSQLQKDLGADASDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPSDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTAGLEKLSAGG 1csi A 1.7 BS02 CMX A 1 R46 L273 H274 A277 V314 V315 G317 Y318 G319 H320 A321 K366 A367 K368 N373 D375 R44 L271 H272 A275 V312 V313 G315 Y316 G317 H318 A319 K364 A365 K366 N371 D373 S244 H274 H320 R329 D375 S242 H272 H318 R327 D373 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 Ki=1.6nM remove_due_to_license_issue P23007 8011640 700 STNLKDVLASLIPKEQARIKTFRQQHGNTAVGQITVDMSYGGMRGMKGLIYETSVLDPDEGIRFRGFSIPECQKLLPKAGGGEEPLPEGLFWLLVTGQIPTPEQVSWVSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGINRTKYWEFVYEDAMDLIAKLPCVAAKIYRNLYRAGSSIGAIDSKLDWSHNFTNMLGYTDPQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLLWLSQLQKDLGADASDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPSDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTAGLEKLSAGG 1csr A 1.7 BS02 FAM A 1 R46 L273 H274 A277 V314 V315 G317 Y318 G319 H320 A321 K366 A367 K368 N373 D375 F397 R44 L271 H272 A275 V312 V313 G315 Y316 G317 H318 A319 K364 A365 K366 N371 D373 F395 S244 H274 H320 R329 D375 S242 H272 H318 R327 D373 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 Ki=42nM remove_due_to_license_issue P23007 7492547 700 STNLKDVLASLIPKEQARIKTFRQQHGNTAVGQITVDMSYGGMRGMKGLIYETSVLDPDEGIRFRGFSIPECQKLLPKAGGGEEPLPEGLFWLLVTGQIPTPEQVSWVSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGINRTKYWEFVYEDAMDLIAKLPCVAAKIYRNLYRAGSSIGAIDSKLDWSHNFTNMLGYTDPQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLLWLSQLQKDLGADASDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPSDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTAGLEKLSAGG 1css A 1.7 BS02 FCX A 1 R46 L273 H274 A277 V314 V315 G317 Y318 G319 H320 A321 K366 A367 K368 N373 D375 R44 L271 H272 A275 V312 V313 G315 Y316 G317 H318 A319 K364 A365 K366 N371 D373 S244 H274 H320 R329 D375 S242 H272 H318 R327 D373 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 Ki=0.8uM remove_due_to_license_issue P23007 7492547 700 STNLKDVLASLIPKEQARIKTFRQQHGNTAVGQITVDMSYGGMRGMKGLIYETSVLDPDEGIRFRGFSIPECQKLLPKAGGGEEPLPEGLFWLLVTGQIPTPEQVSWVSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGINRTKYWEFVYEDAMDLIAKLPCVAAKIYRNLYRAGSSIGAIDSKLDWSHNFTNMLGYTDPQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLLWLSQLQKDLGADASDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPSDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTAGLEKLSAGG 1ct8 A 2.2 BS01 TAA B 1 H92 R94 L96 H92 R94 L96 ? 0005576,0005886,0030183 remove_due_to_license_issue P01837 10574796 550 ELVMTQTPATLSVTPGDSVSLSCRASQSVSNKLHWYQQKSHESPRLLIKFASQSIPGIPSRFSGSGSGSDFTLSINSVETEDFGIYFCHQTHGRPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 1ct8 B 2.2 BS01 TAA B 1 Y33 N35 W50 Y95 Y97 F100A Y33 N35 W50 Y99 Y101 F105 ? Kd=0.3uM remove_due_to_license_issue P01868 10574796 550 QVKLLESGAVLVKPGASVKLSCKTSGFTFSSSYINWLKQKPGQSLEWIAWIYAGSGGTVYNQHFTDKARLTVDTSSSTAYMQFSSLTTEDSAIYYCARYRYDEGFAYWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRDC 1ct8 B 2.2 BS02 TAA D 1 S54 G56 S55 G57 ? Kd=0.3uM remove_due_to_license_issue P01868 10574796 551 QVKLLESGAVLVKPGASVKLSCKTSGFTFSSSYINWLKQKPGQSLEWIAWIYAGSGGTVYNQHFTDKARLTVDTSSSTAYMQFSSLTTEDSAIYYCARYRYDEGFAYWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRDC 1ct8 C 2.2 BS01 TAA D 1 H92 R94 L96 H92 R94 L96 ? 0005576,0005886,0030183 remove_due_to_license_issue P01837 10574796 551 ELVMTQTPATLSVTPGDSVSLSCRASQSVSNKLHWYQQKSHESPRLLIKFASQSIPGIPSRFSGSGSGSDFTLSINSVETEDFGIYFCHQTHGRPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 1ct8 D 2.2 BS01 TAA B 1 S54 G56 S55 G57 ? Kd=0.3uM remove_due_to_license_issue P01868 10574796 550 QVKLLESGAVLVKPGASVKLSCKTSGFTFSSSYINWLKQKPGQSLEWIAWIYAGSGGTVYNQHFTDKARLTVDTSSSTAYMQFSSLTTEDSAIYYCARYRYDEGFAYWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRDC 1ct8 D 2.2 BS02 TAA D 1 Y33 N35 W50 Y95 Y97 F100A Y33 N35 W50 Y99 Y101 F105 ? Kd=0.3uM remove_due_to_license_issue P01868 10574796 551 QVKLLESGAVLVKPGASVKLSCKTSGFTFSSSYINWLKQKPGQSLEWIAWIYAGSGGTVYNQHFTDKARLTVDTSSSTAYMQFSSLTTEDSAIYYCARYRYDEGFAYWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRDC 1ctr A 2.45 BS05 TFP A 1 M124 E127 A128 V136 M144 M118 E121 A122 V130 M138 V35 V35 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 remove_due_to_license_issue Kd=1000nM P0DP23 7803388 153 ADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTA 1ctt A 2.2 BS02 DHZ A 1 F71 N89 E91 H102 E104 F71 N89 E91 H102 E104 H102 E104 C129 C132 H102 E104 C129 C132 3.5.4.5 0001884,0003824,0004126,0005737,0005829,0006217,0008270,0009972,0015949,0016787,0042802,0042803,0046872,0055086,0072527,1901135 Ki=30uM remove_due_to_license_issue P0ABF6 7718553 295 MHPRFQTAFAQLADNLQSALEPILADKYFPALLTGEQVSSLKSATGLDEDALAFALLPLAAACARTPLSNFNVGAIARGVSGTWYFGANMEFIGATMQQTVHAEQSAISHAWLSGEKALAAITVNYTPCGHCRQFMNELNSGLDLRIHLPGREAHALRDYLPDAFGPKDLEIKTLLMDEQDHGYALTGDALSQAAIAAANRSHMPYSKSPSGVALECKDGRIFSGSYAENAAFNPTLPPLQGALILLNLKGYDYPDIQRAVLAEKADAPLIQWDATSATLKALGCHSIDRVLLA 1ctu A 2.3 BS02 ZEB A 1 N89 E91 H102 E104 P128 C129 C132 N89 E91 H102 E104 P128 C129 C132 H102 E104 C129 C132 H102 E104 C129 C132 3.5.4.5 0001884,0003824,0004126,0005737,0005829,0006217,0008270,0009972,0015949,0016787,0042802,0042803,0046872,0055086,0072527,1901135 Ki=1.2pM remove_due_to_license_issue P0ABF6 7718553 295 MHPRFQTAFAQLADNLQSALEPILADKYFPALLTGEQVSSLKSATGLDEDALAFALLPLAAACARTPLSNFNVGAIARGVSGTWYFGANMEFIGATMQQTVHAEQSAISHAWLSGEKALAAITVNYTPCGHCRQFMNELNSGLDLRIHLPGREAHALRDYLPDAFGPKDLEIKTLLMDEQDHGYALTGDALSQAAIAAANRSHMPYSKSPSGVALECKDGRIFSGSYAENAAFNPTLPPLQGALILLNLKGYDYPDIQRAVLAEKADAPLIQWDATSATLKALGCHSIDRVLLA 1cw2 A 2.0 BS01 HSP A 1 F22 D60 L100 Y175 T183 G184 F212 G234 S235 F21 D59 L99 Y174 T182 G183 F209 G231 S232 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 ic50=715nM remove_due_to_license_issue P00929 10504236 270 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1cx9 A 2.3 BS01 NHP A 1 L100 Y175 T183 G184 F212 G234 S235 L99 Y174 T182 G183 F209 G231 S232 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 ic50=178nM remove_due_to_license_issue P00929 10504236 270 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1czc A 2.5 BS02 GUA A 1 I17 W140 N194 R386 I13 W130 N183 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=1.5mM remove_due_to_license_issue P00509 10731702 414 MFENITTAPADPILGLADLLRADERPGKIDLGMGVYNDETGKTPVLTSVKKAEQYLLENETTKNYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGTGALRVAADFLAKNTSVRRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFGLYNERVGTCTLVAADSETVDRAFSQMKAAIRVNYSSPPAHGASVVATILGNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFTIKQNGMFFFGGLTKEQVLRLREEFGVYAVASGRLNVAGMTPDNLAPLCEAIVAVL 1czk A 1.9 BS01 FMN A 1 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 V59 A88 G89 D90 Y94 F98 D146 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 V59 A88 G89 D90 Y94 F98 D146 ? 0009055,0010181 Kd=1.5nM remove_due_to_license_issue P10340 10610792 170 AKIGLFYGTQTGVTQTIAESIQQEFGGESIVDLNDIANADASDLNAYDYLIIGCPTWNVGELQSDWEGIYDDLDSVNFQGKKVAYFGAGDQVGYSDNFQNAMGILEEKISSLGSQTVGYWPIEGYDFNESKAVRNNQFVGLAIDEDNQPDLTKNRIKTWVSQLKSEFGL 1czl A 1.8 BS01 FMN A 1 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 G60 A88 G89 D90 Y94 N97 F98 D146 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 G60 A88 G89 D90 Y94 N97 F98 D146 ? 0009055,0010181 Ka=1400000000M^-1 remove_due_to_license_issue P10340 10610792 170 AKIGLFYGTQTGVTQTIAESIQQEFGGESIVDLNDIANADASDLNAYDYLIIGCPTWNVGELQSDWEGIYDDLDSVNFQGKKVAYFGAGDQVGYSDNFQDAMGILEEKISSLGSQTVGYWPIEGYDFNESKAVRNNQFVGLAIDEDNQPDLTKNRIKTWVSQLKSEFGL 1czo A 1.85 BS01 FMN A 1 T9 Q10 T11 V13 T14 P55 T56 W57 G58 G60 A88 G89 D90 Y94 N97 F98 D146 T9 Q10 T11 V13 T14 P55 T56 W57 G58 G60 A88 G89 D90 Y94 N97 F98 D146 ? 0009055,0010181 Ka=35000M^-1 remove_due_to_license_issue P10340 10610792 170 AKIGLFYGTQTGVTQTIAESIQQEFGGESIVDLNDIANADASDLNAYDYLIIGCPTWGVGELQSDWEGIYDDLDSVNFQGKKVAYFGAGDQVGYSDNFQDAMGILEEKISSLGSQTVGYWPIEGYDFNESKAVRNNQFVGLAIDEDNQPDLTKNRIKTWVSQLKSEFGL 1czr A 1.9 BS01 FMN A 1 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 V59 A88 G89 N90 Y94 N97 F98 D146 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 V59 A88 G89 N90 Y94 N97 F98 D146 ? 0009055,0010181 Kd=1nM remove_due_to_license_issue P10340 10610792 170 AKIGLFYGTQTGVTQTIAESIQQEFGGESIVDLNDIANADASDLNAYDYLIIGCPTWNVGELQSDWEGIYDDLDSVNFQGKKVAYFGAGNQVGYSDNFQDAMGILEEKISSLGSQTVGYWPIEGYDFNESKAVRNNQFVGLAIDEDNQPDLTKNRIKTWVSQLKSEFGL 1d04 A 1.85 BS01 FMN A 1 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 V59 A88 G89 D90 Y94 N97 F98 D146 T9 Q10 T11 G12 V13 T14 P55 T56 W57 N58 V59 A88 G89 D90 Y94 N97 F98 D146 ? 0009055,0010181 Ka=38000M^-1 remove_due_to_license_issue P10340 10610792 170 AKIGLFYGTQTGVTQTIAESIQQEFGGESIVDLNDIANADASDLNAYDYLIIGCPTWNVGELQSDWEGIYDDLDSVNFQGKKVAYFGAGDQVGYSDNFQDAMGILEEKISSLGSQTVGYWPIEGYDFNESKAVRNNQFVGLAIDEDNQPDLTKNRIKTWVSQLKSEFGL 1d09 A 2.1 BS01 PAL A 1 S52 T53 R54 T55 R105 H134 R167 R229 L267 S52 T53 R54 T55 R105 H134 R167 R229 L267 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=27nM remove_due_to_license_issue P0A786 10651286 1311 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQQTQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPEYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 1d1p A 2.2 BS01 EPE A 1 C13 L14 G15 F17 C18 R19 H52 D132 W134 C9 L10 G11 F13 C14 R15 H48 D128 W130 C13 N16 C18 R19 S20 D132 C9 N12 C14 R15 S16 D128 3.1.3.2,3.1.3.48 0003993,0004721,0004725,0004726,0005634,0005737,0006338,0006470,0030946,0140793 remove_due_to_license_issue P40347 10684639 201 PKISVAFICLGNFCRSPMAEAIFKHEVEKANLENRFNKIDSFGTSNYHVGESPDHRTVSICKQHGVKINHKGKQIKTKHFDEYDYIIGMDESNINNLKKIQPEGSKAKVCLFGDWNTNDGTVQTIIEDPWYGDIQDFEYNFKQITYFSKQFLKKEL 1d2e A 1.94 BS01 GDP A 1 D67 G69 K70 T71 T72 Y92 N181 K182 D184 S219 L221 D13 G15 K16 T17 T18 Y38 N127 K128 D130 S165 L167 D67 K70 T71 T107 H130 D13 K16 T17 T53 H76 ? 0003746,0003924,0005525,0006414 Kd=1uM remove_due_to_license_issue P49410 10715211 1301 KPHVNVGTIGHVDHGKTTLTAAITKILAEGGGAKFKKYEEIDNAPEERARGITINAAHVEYSTAARHYAHTDCPGHADYVKNMITGTAPLDGCILVVAANDGPMPQTREHLLLARQIGVEHVVVYVNKADAVQDSEMVELVELEIRELLTEFGYKGEETPIIVGSALCALEQRDPELGLKSVQKLLDAVDTYIPVPTRDLEKPFLLPVESVYSIPGRGTVVTGTLERGILKKGDECEFLGHSKNIRTVVTGIEMFHKSLDRAEAGDNLGALVRGLKREDLRRGLVMAKPGSIQPHQKVEAQVYILTKEEGGRHKPFVSHFMPVMFSLTWDMACRIILPPGKELAMPGEDLKLTLILRQPMILEKGQRFTLRDGNRTIGTGLVTDTPAMTEEDKNIKW 1d2s A 1.55 BS02 DHT A 1 S41 S42 D65 F67 N82 L171 S29 S30 D53 F55 N70 L153 ? remove_due_to_license_issue IC50=3.8nM, Kd=0.182000nM P04278 10675319 301 PPAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAEISASAPTSLRSC 1d3d B 2.04 BS03 BZT B 1 H79 Y83 W86 L132 D235 A236 C237 E238 V261 S262 W263 G264 H43 Y47 W50 L96 D192 A193 C194 E195 V218 S219 W220 G221 H79 D135 E238 G239 D240 S241 G242 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ka=1240000000M^-1 remove_due_to_license_issue Ki=2.1nM P00734 10739244 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1d3p B 2.1 BS03 BT3 B 1 H79 W86 N131 L132 D235 A236 C237 E238 V261 S262 W263 G264 H43 W50 N95 L96 D192 A193 C194 E195 V218 S219 W220 G221 H79 D135 E238 G239 D240 S241 G242 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ka=24300000M^-1 remove_due_to_license_issue P00734 10739244 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1d3q B 2.9 BS03 BT2 B 1 Y83 W86 E130 N131 L132 I215 A236 C237 E238 S262 W263 G264 C267 Y47 W50 E94 N95 L96 I172 A193 C194 E195 S219 W220 G221 C224 H79 D135 E238 G239 D240 S241 G242 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10739244 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1d3v A 1.7 BS03 ABH A 1 H101 D124 H126 D128 N130 S137 H141 D232 H96 D119 H121 D123 N125 S132 H136 D227 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 Kd=0.11uM remove_due_to_license_issue P07824 10542097 551 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTTSSGNLHGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHK 1d4h A 1.81 BS01 BEH B 1 R8 D25 G27 A28 D30 G49 V82 R8 D25 G27 A28 D30 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4h B 1.81 BS01 BEH B 1 R108 L123 D125 G127 A128 D129 D130 G148 P181 V182 R8 L23 D25 G27 A28 D29 D30 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.1nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4i A 1.81 BS01 BEG A 1 R8 D25 G27 A28 D29 D30 G48 G49 V82 R8 D25 G27 A28 D29 D30 G48 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.4nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4i B 1.81 BS01 BEG A 1 R108 D125 G127 A128 D129 D130 G148 P181 V182 R8 D25 G27 A28 D29 D30 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4j A 1.81 BS01 MSC B 1 R8 D25 G27 D30 G48 G49 V82 I84 R8 D25 G27 D30 G48 G49 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4j B 1.81 BS01 MSC B 1 R108 D125 G127 A128 D129 D130 I147 G148 P181 V182 R8 D25 G27 A28 D29 D30 I47 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.4nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4k A 1.85 BS01 PI8 A 1 R8 D25 G27 A28 D29 D30 G48 P81 V82 R8 D25 G27 A28 D29 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P03369 11000004 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1d4k B 1.85 BS01 PI8 A 1 R8 D25 G27 A28 D29 G48 V82 I84 R8 D25 G27 A28 D29 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 11000004 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1d4l A 1.75 BS01 PI9 A 1 D25 G27 A28 D29 G48 I50 V82 I84 D25 G27 A28 D29 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.7nM remove_due_to_license_issue P03369 11000004 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1d4l B 1.75 BS01 PI9 A 1 D25 A28 D30 I50 P81 V82 I84 D25 A28 D30 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 11000004 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1d4p B 2.07 BS03 BPP B 1 Y83 W86 L132 D235 A236 W263 G264 G266 Y47 W50 L96 D192 A193 W220 G221 G223 H79 D135 E238 G239 D240 S241 G242 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ka=2000000M^-1 remove_due_to_license_issue P00734 9232642 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1d4y A 1.97 BS01 TPV A 1 D25 D29 D30 G48 V82 D25 D29 D30 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.008nM remove_due_to_license_issue P03367 8893827 501 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d4y B 1.97 BS01 TPV A 1 R8 L23 D25 G49 I50 R8 L23 D25 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 8893827 501 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1d5j A 2.6 BS06 MM3 A 1 V163 L164 A165 V198 H201 E202 H205 H211 P221 L222 Y223 V81 L82 A83 V116 H119 E120 H123 H129 P139 L140 Y141 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P08254 10579818 401 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPD 1d6n A 2.7 BS02 PPO A 1 I135 D137 K165 F186 V187 I132 D134 K162 F183 V184 E133 D134 D137 F186 R199 E130 D131 D134 F183 R196 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 10338013 300 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLAGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLGSYCNDQSTGDIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 1d6s A 2.3 BS02 PLP A 1 N71 G176 T177 G178 T180 G228 S272 P299 N71 G176 T177 G178 T180 G228 S272 P299 A41 G228 A41 G228 2.5.1.47 0004124,0005737,0006535,0016740,0016765,0019344,0080146 remove_due_to_license_issue P0A1E3 10452898 501 SKIYEDNSLTIGHTPLVRLNRIGNGRILAKVESRNPSFSVACRIGANMIWDAEKRGVLKPGVELVEPTNGNTGIALAYVAAARGYKLTLTMPETMSIERRKLLKALGANLVLTEGAKGMKGAIQKAEEIVASDPQKYLLLQQFSNPANPEIHEKTTGPEIWEDTDGQVDVFISGVGTGGTLTGVTRYIKGTKGKTDLITVAVEPTDSPVIAQALAGEEIKPGPHKIQGIGAGFIPGNLDLKLIDKVVGITNEEAISTARRLMEEEGILAGISSGAAVAAALKLQEDESFTNKNIVVILPSSGERYLSTALFADLFTEKELQQ 1d6v H 2.0 BS01 HOP H 1 E35 G95 H96 Y100A D101 W103 E35 G99 H100 Y105 D108 W110 ? Kd=670nM remove_due_to_license_issue P01857 10651626 401 QVQLQQSGAELMKPGASVKISCKATGYTFSSYWIEWVKQRPGHGLEWIGEILPGSGSTNYNEKFKGKATFTADTSSNTAYMQLSSLTSEDSAVYYCARGHSYYFYDGDYWGQGTSVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 1d6v L 2.0 BS01 HOP H 1 F36 L89 Y91 F36 L89 Y91 ? 0002250,0003823,0005576,0005615,0005886,0006955,0016064,0019814,0050853,0070062,0071735,0071738,0071742,0071745,0071753,0072562 remove_due_to_license_issue P01834 10651626 401 DIKMTQSPSSMYASLGERVTITCKASQDINSYLSWFQQKPGKSPKTLIYRANRLVDGVPSRFSGSGSGQDYSLTISSLEYEDMGIYYCLQYDEFPYTFGSGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNR 1d6w A 2.0 BS02 00R A 1 H57 Y60A W60D N98 L99 I174 D189 S195 W215 G216 G219 G226 H71 Y75 W78 N123 L124 I200 D220 S226 W248 G249 G251 G259 H57 D102 E192 G193 D194 S195 G196 H71 D127 E223 G224 D225 S226 G227 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=1100nM remove_due_to_license_issue P00734 10713516 380 ADCGLRPLFEKKSLEDKTERELLESYIDIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1d7i A 1.9 BS01 DSS A 1 Y26 F46 V55 I56 Y26 F46 V55 I56 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Kd=250uM remove_due_to_license_issue P62942 10656803 301 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1d7j A 1.85 BS01 BUQ A 1 V55 I56 W59 F99 V55 I56 W59 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Kd=500uM remove_due_to_license_issue P62942 10656803 311 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1d7x A 2.0 BS06 SPC A 1 V163 L164 A165 H201 E202 H205 H211 L222 Y223 V81 L82 A83 H119 E120 H123 H129 L140 Y141 H201 H205 H211 H119 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=19nM P08254 10639284 401 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPD 1d7x B 2.0 BS06 SPC B 1 V663 L664 A665 H701 E702 H705 H711 L722 Y723 V81 L82 A83 H119 E120 H123 H129 L140 Y141 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=19nM P08254 10639284 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1d8f B 2.4 BS06 SPI B 1 L664 A665 V698 H701 E702 H705 H711 P721 Y723 L82 A83 V116 H119 E120 H123 H129 P139 Y141 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=18nM remove_due_to_license_issue IC50=18nM P08254 10669564 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1d8m B 2.44 BS06 BBH B 1 L664 A665 H701 E702 H705 H711 Y723 L82 A83 H119 E120 H123 H129 Y141 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=3.1nM P08254 11327577 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1d9i A 2.3 BS02 00P A 1 H57 Y60A W60D I174 C191 E192 S214 W215 G216 E217 G219 H71 Y75 W78 I200 C222 E223 S247 W248 G249 E250 G251 H57 D102 E192 G193 D194 S195 G196 H71 D127 E223 G224 D225 S226 G227 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=0.78nM remove_due_to_license_issue P00734 10713516 380 ADCGLRPLFEKKSLEDKTERELLESYIDIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1dar A 2.4 BS01 GDP A 1 D22 G24 K25 T26 T27 N137 K138 D140 S262 L264 D22 G24 K25 T26 T27 N109 K110 D112 S234 L236 D22 D22 ? 0003746,0003924,0005525,0005737,0006412,0006414,0032790 Kd=11uM remove_due_to_license_issue Q5SHN5 8736554 692 MAVKVEYDLKRLRNIGIAAHIDAGKTTTTERILYYTGRAAVTTCFWKDHRINIIDTPGHVDFTIEVERSMRVLDGAIVVFDSSQGVEPQSETVWRQAEKYKVPRIAFANKMDKTGADLWLVIRTMQERLGARPVVMQLPIGREDTFSGIIDVLRMKAYTYGNDLGTDIREIPIPEEYLDQAREYHEKLVEVAADFDENIMLKYLEGEEPTEEELVAAIRKGTIDLKITPVFLGSALKNKGVQLLLDAVVDYLPSPLDIPPIKGTTPEGEVVEIHPDPNGPLAALAFKIMADPYVGRLTFIRVYSGTLTSGSYVYNTTKGRKERVARLLRMHANHREEVEELKAGDLGAVVGLKETITGDTLVGEDAPRVILEEEDPTFRVSTQTIISGMGELKREFKVDANVGKPQVAYRETITKPVDVEGKFIRQTGGRGQYGHVKIKVEPLPRGSGFEFVNAIVGGVIPKEYIPAVQKGIEEAMQSGPLIGFPVVDIKVTLYDGSYHEVDSSEMAFKIAGSMAIKEAVQKGDPVILEPIMRVEVTTPEEYMGDVIGDLNARRGQILGMEPRGNAQVIRAFVPLAEMFGYATDLRSKTQGRGSFVMFFDHYQEVPKQVQEKLIK 1db1 A 1.8 BS01 VDX A 1 Y143 L233 S237 R274 S275 S278 W286 H305 Y24 L63 S67 R104 S105 S108 W116 H135 ? 0003677,0004879,0006355 Kd=0.55nM remove_due_to_license_issue EC50=10nM, IC50=1.1nM, Kd=0.065nM P11473 10678179 428 LRPKLSEEQQRIIAILLDAHHKTYDPTYSDFCQFRPPVRVNDGGGSVTLELSQLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSEDQIVLLKSSAIEVIMLRSNESFTMDDMSWTCGNQDYKYRVSDVTKAGHSLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAALIEAIQDRLSNTLQTYIRCRHPPPLLYAKMIQKLADLRSLNEEHSKQYRCLSFQPECSMKLTPLVLEVFG 1db4 A 2.2 BS03 8IN A 1 L2 F5 H6 Y21 C28 G29 V30 G31 H47 D48 Y51 K62 L2 F5 H6 Y21 C28 G29 V30 G31 H47 D48 Y51 K62 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 remove_due_to_license_issue IC50=57.0nM P14555 7664108 200 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 1db5 A 2.8 BS03 6IN A 1 F5 Y21 G29 V30 G31 C44 H47 D48 Y51 F5 Y21 G29 V30 G31 C44 H47 D48 Y51 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 remove_due_to_license_issue IC50=69000nM P14555 7664108 200 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 1dbb H 2.7 BS01 STR H 1 W50 G95 D96 Y97 W50 G99 D100 Y101 ? remove_due_to_license_issue P01868 8496956 229 QIQLVQSGPELKKPGETVKISCKASGYAFTNYGVNWVKEAPGKELKWMGWINIYTGEPTYVDDFKGRFAFSLETSASTAYLEINNLKNEDTATYFCTRGDYVNWYFDVWGAGTTVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPR 1dbb L 2.7 BS01 STR H 1 H27D S91 V94 H31 S96 V99 remove_due_to_license_issue 8496956 229 DVVMTQIPLSLPVNLGDQASISCRSSQSLIHSNGNTYLHWYLQKPGQSPKLLMYKVSNRFYGVPDRFSGSGSGTDFTLKISRVEAEDLGIYFCSQSSHVPPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 1dbj H 2.7 BS01 AE2 H 1 N35 W50 G95 W100 N35 W50 G99 W104 ? remove_due_to_license_issue P01868 8413674 229 QIQLVQSGPELKKPGETVKISCKASGYAFTNYGVNWVKEAPGKELKWMGWINIYTGEPTYVDDFKGRFAFSLETSASTAYLEINNLKNEDTATYFCTRGDYVNWYFDVWGAGTTVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPR 1dbk H 3.0 BS01 ANO H 1 N35 W50 G95 Y97 N35 W50 G99 Y101 ? remove_due_to_license_issue P01868 8413674 229 QIQLVQSGPELKKPGETVKISCKASGYAFTNYGVNWVKEAPGKELKWMGWINIYTGEPTYVDDFKGRFAFSLETSASTAYLEINNLKNEDTATYFCTRGDYVNWYFDVWGAGTTVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPR 1det A 1.8 BS01 2GP A 1 Y42 N43 N44 Y45 E46 X58 Y42 N43 N44 Y45 E46 X58 Y38 H40 E58 D76 R77 T91 H92 F100 Y38 H40 E58 D76 R77 T91 H92 F100 4.6.1.24 0001411,0003723,0004519,0004521,0004540,0008150,0016829,0030428,0046589 Kd=50uM remove_due_to_license_issue P00651 8679590 105 ACDYTCGSNCYSSSDVSTAQAAGYQLHEDGETVGSNSYPHKYNNYEGFDFSVSSPYYEWPILSSGDVYSGGSPGADRVVFNENNQLAGVITHTGASGNNFVECT 1df8 A 1.51 BS01 BTN A 1 N23 L25 S27 Y43 V47 N49 W79 S88 T90 W108 D128 N8 L10 S12 Y28 V32 N34 W64 S73 T75 W93 D113 ? 0009374 Kd=0.2nM remove_due_to_license_issue Kd=1.000000nM P22629 10850797 201 GITGTWYNQLGSTFIVTAGADGALTGTYEAAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1dfo A 2.4 BS02 FFO A 1 L121 G125 H126 L127 S175 N347 S355 P356 F357 L120 G124 H125 L126 S174 N346 S354 P355 F356 Y55 E57 D200 T226 K229 R235 Y54 E56 D199 T225 K228 R234 2.1.2.1 0003824,0004372,0005515,0005737,0005829,0006545,0006546,0006564,0006565,0006730,0008270,0008652,0008732,0016020,0016740,0019264,0030170,0035999,0042802,0042803,0046653 remove_due_to_license_issue P0A825 10656824 1002 LKREMNIADYDAELWQAMEQEKVRQEEHIELIASENYTSPRVMQAQGSQLTNKYAEGYPGKRYYGGCEYVDIVEQLAIDRAKELFGADYANVQPHSGSQANFAVYTALLEPGDTVLGMNLAHGGHLTHGSPVNFSGKLYNIVPYGIDATGHIDYADLEKQAKEHKPKMIIGGFSAYSGVVDWAKMREIADSIGAYLFVDMAHVAGLVAAGVYPNPVPHAHVVTTTTHKTLAGPRGGLILAKGGSEELYKKLNSAVFPGGQGGPLMHVIAGKAVALKEAMEPEFKTYQQQVAKNAKAMVEVFLERGYKVVSGGTDNHLFLVDLVDKNLTGKEADAALGRANITVNKNSVPNDPKSPFVTSGIRVGTPAITRRGFKEAEAKELAGWMCDVLDSINDEAVIERIKGKVLDICARYPVYA 1dfo A 2.4 BS04 FFO B 1 E57 Y64 Y65 E56 Y63 Y64 Y55 E57 D200 T226 K229 R235 Y54 E56 D199 T225 K228 R234 2.1.2.1 0003824,0004372,0005515,0005737,0005829,0006545,0006546,0006564,0006565,0006730,0008270,0008652,0008732,0016020,0016740,0019264,0030170,0035999,0042802,0042803,0046653 remove_due_to_license_issue P0A825 10656824 2002 LKREMNIADYDAELWQAMEQEKVRQEEHIELIASENYTSPRVMQAQGSQLTNKYAEGYPGKRYYGGCEYVDIVEQLAIDRAKELFGADYANVQPHSGSQANFAVYTALLEPGDTVLGMNLAHGGHLTHGSPVNFSGKLYNIVPYGIDATGHIDYADLEKQAKEHKPKMIIGGFSAYSGVVDWAKMREIADSIGAYLFVDMAHVAGLVAAGVYPNPVPHAHVVTTTTHKTLAGPRGGLILAKGGSEELYKKLNSAVFPGGQGGPLMHVIAGKAVALKEAMEPEFKTYQQQVAKNAKAMVEVFLERGYKVVSGGTDNHLFLVDLVDKNLTGKEADAALGRANITVNKNSVPNDPKSPFVTSGIRVGTPAITRRGFKEAEAKELAGWMCDVLDSINDEAVIERIKGKVLDICARYPVYA 1dfo B 2.4 BS02 FFO A 1 E57 Y64 Y65 E57 Y64 Y65 Y55 E57 D200 T226 K229 R235 Y55 E57 D200 T226 K229 R235 2.1.2.1 0003824,0004372,0005515,0005737,0005829,0006545,0006546,0006564,0006565,0006730,0008270,0008652,0008732,0016020,0016740,0019264,0030170,0035999,0042802,0042803,0046653 remove_due_to_license_issue P0A825 10656824 1002 MLKREMNIADYDAELWQAMEQEKVRQEEHIELIASENYTSPRVMQAQGSQLTNKYAEGYPGKRYYGGCEYVDIVEQLAIDRAKELFGADYANVQPHSGSQANFAVYTALLEPGDTVLGMNLAHGGHLTHGSPVNFSGKLYNIVPYGIDATGHIDYADLEKQAKEHKPKMIIGGFSAYSGVVDWAKMREIADSIGAYLFVDMAHVAGLVAAGVYPNPVPHAHVVTTTTHKTLAGPRGGLILAKGGSEELYKKLNSAVFPGGQGGPLMHVIAGKAVALKEAMEPEFKTYQQQVAKNAKAMVEVFLERGYKVVSGGTDNHLFLVDLVDKNLTGKEADAALGRANITVNKNSVPNDPKSPFVTSGIRVGTPAITRRGFKEAEAKELAGWMCDVLDSINDEAVIERIKGKVLDICARYPVYA 1dfo B 2.4 BS04 FFO B 1 L121 G125 H126 L127 S175 N347 S355 P356 F357 L121 G125 H126 L127 S175 N347 S355 P356 F357 Y55 E57 D200 T226 K229 R235 Y55 E57 D200 T226 K229 R235 2.1.2.1 0003824,0004372,0005515,0005737,0005829,0006545,0006546,0006564,0006565,0006730,0008270,0008652,0008732,0016020,0016740,0019264,0030170,0035999,0042802,0042803,0046653 remove_due_to_license_issue P0A825 10656824 2002 MLKREMNIADYDAELWQAMEQEKVRQEEHIELIASENYTSPRVMQAQGSQLTNKYAEGYPGKRYYGGCEYVDIVEQLAIDRAKELFGADYANVQPHSGSQANFAVYTALLEPGDTVLGMNLAHGGHLTHGSPVNFSGKLYNIVPYGIDATGHIDYADLEKQAKEHKPKMIIGGFSAYSGVVDWAKMREIADSIGAYLFVDMAHVAGLVAAGVYPNPVPHAHVVTTTTHKTLAGPRGGLILAKGGSEELYKKLNSAVFPGGQGGPLMHVIAGKAVALKEAMEPEFKTYQQQVAKNAKAMVEVFLERGYKVVSGGTDNHLFLVDLVDKNLTGKEADAALGRANITVNKNSVPNDPKSPFVTSGIRVGTPAITRRGFKEAEAKELAGWMCDVLDSINDEAVIERIKGKVLDICARYPVYA 1dfo B 2.4 BS05 FFO C 1 S245 E247 S245 E247 Y55 E57 D200 T226 K229 R235 Y55 E57 D200 T226 K229 R235 2.1.2.1 0003824,0004372,0005515,0005737,0005829,0006545,0006546,0006564,0006565,0006730,0008270,0008652,0008732,0016020,0016740,0019264,0030170,0035999,0042802,0042803,0046653 remove_due_to_license_issue P0A825 10656824 3002 MLKREMNIADYDAELWQAMEQEKVRQEEHIELIASENYTSPRVMQAQGSQLTNKYAEGYPGKRYYGGCEYVDIVEQLAIDRAKELFGADYANVQPHSGSQANFAVYTALLEPGDTVLGMNLAHGGHLTHGSPVNFSGKLYNIVPYGIDATGHIDYADLEKQAKEHKPKMIIGGFSAYSGVVDWAKMREIADSIGAYLFVDMAHVAGLVAAGVYPNPVPHAHVVTTTTHKTLAGPRGGLILAKGGSEELYKKLNSAVFPGGQGGPLMHVIAGKAVALKEAMEPEFKTYQQQVAKNAKAMVEVFLERGYKVVSGGTDNHLFLVDLVDKNLTGKEADAALGRANITVNKNSVPNDPKSPFVTSGIRVGTPAITRRGFKEAEAKELAGWMCDVLDSINDEAVIERIKGKVLDICARYPVYA 1dgm A 1.8 BS02 ADN A 1 N20 D24 G69 S70 Y169 D318 N11 D15 G60 S61 Y160 D301 R136 G315 A316 G317 D318 R127 G298 A299 G300 D301 2.7.1.20 0004001,0005524,0005634,0005829,0006144,0006166,0016301,0034654,0044209,0046872,0055086 remove_due_to_license_issue Ki=8900nM Q9TVW2 10794412 375 TGPMRVFAIGNPILDLVAEVPSSFLDEFFLKRGDATLATPEQMRIYSTLDQFNPTSLPGGSALNSVRVVQKLLRKPGSAGYMGAIGDDPRGQVLKELCDKEGLATRFMVAPGQSTGVCAVLINEKERTLCTHLGACGSFRLPEDWTTFASGALIFYATAYTLTATPKNAFEVAGYAHGIPNAIFTLNLSAPFCVELYKDAMQSLLLHTNILFGNEEEFAHLAKVHNLVTANKEHAVEVCTGALRLLTAGQNTGATKLVVMTRGHNPVIAAEQTADGTVVVHEVGVPVVAAEKIVDTNGAGDAFVGGFLYALSQGKTVKQCIMCGNACAQDVIQHVGFSLSFTSLPC 1dh3 A 3.0 BS01 dna B 0 N293 R294 R298 R301 N9 R10 R14 R17 ? 0003677,0003700,0005634,0006355 remove_due_to_license_issue Q01147 10952992 -11 ~ 10 KREVRLMKNREAARESRRKKKEYVKSLENRVAVLENQNKTLIEELKALKDLYSHK 1dh3 C 3.0 BS01 dna D 0 R286 N293 R294 R298 K305 R2 N9 R10 R14 K21 ? 0003677,0003700,0005634,0006355 remove_due_to_license_issue Q01147 10952992 -11 ~ 10 KREVRLMKNREAARESRRKKKEYVKSLENRVAVLENQNKTLIEELKALKDLYSHK 1dhi A 1.9 BS01 MTX A 1 I5 A6 F31 K32 I50 R57 I94 I5 A6 F31 K32 I50 R57 I94 I5 M20 W22 S27 L28 F31 L54 I91 T113 I5 M20 W22 S27 L28 F31 L54 I91 T113 1.5.1.3 0004146,0005515,0005542,0005829,0006730,0009257,0009410,0016491,0031427,0046452,0046654,0046655,0046656,0046677,0050661,0051870,0051871,0070401,0070402 Kd=55nM remove_due_to_license_issue IC50=8.8nM, EC50=1nM P0ABQ4 8265622 161 MISLIAALAVDRVIGMENAMPWNLPASLAWFKRNTLDKPVIMGRHTWESIGRPLPGRKNIILSSQPGTDDRVTWVKSVDEAIAACGDVPEIMVIGGGRVYEQFLPKAQKLYLTHIDAEVEGDTHFPDYEPDDWESVFSEFHDADAQNSHSYCFEILERR 1dhi B 1.9 BS01 MTX B 1 A6 F31 K32 I50 R57 I94 A6 F31 K32 I50 R57 I94 I5 M20 W22 S27 L28 F31 L54 I91 T113 I5 M20 W22 S27 L28 F31 L54 I91 T113 1.5.1.3 0004146,0005515,0005542,0005829,0006730,0009257,0009410,0016491,0031427,0046452,0046654,0046655,0046656,0046677,0050661,0051870,0051871,0070401,0070402 Kd=55nM remove_due_to_license_issue IC50=8.8nM, EC50=1nM P0ABQ4 8265622 361 MISLIAALAVDRVIGMENAMPWNLPASLAWFKRNTLDKPVIMGRHTWESIGRPLPGRKNIILSSQPGTDDRVTWVKSVDEAIAACGDVPEIMVIGGGRVYEQFLPKAQKLYLTHIDAEVEGDTHFPDYEPDDWESVFSEFHDADAQNSHSYCFEILERR 1dhj A 1.8 BS01 MTX A 1 I5 A6 L28 F31 K32 I50 R52 R57 I94 I5 A6 L28 F31 K32 I50 R52 R57 I94 I5 M20 W22 S27 L28 F31 L54 I91 T113 I5 M20 W22 S27 L28 F31 L54 I91 T113 1.5.1.3 0004146,0005515,0005542,0005829,0006730,0009257,0009410,0016491,0031427,0046452,0046654,0046655,0046656,0046677,0050661,0051870,0051871,0070401,0070402 Kd=281nM remove_due_to_license_issue IC50=8.8nM, EC50=1nM P0ABQ4 8265622 161 MISLIAALAVDRVIGMENAMPWNLPASLAWFKRNTLDKPVIMGRHTWESIGRPLPGRKNIILSSQPGTDDRVTWVKSVDEAIAACGDVPEIMVIGGGRVYEQFLPKAQKLYLTHIDAEVEGDTHFPDYEPDDWESVSSEFHDADAQNSHSYCFEILERR 1dhj B 1.8 BS01 MTX B 1 I5 A6 A7 L28 F31 K32 I50 R52 R57 I94 I5 A6 A7 L28 F31 K32 I50 R52 R57 I94 I5 M20 W22 S27 L28 F31 L54 I91 T113 I5 M20 W22 S27 L28 F31 L54 I91 T113 1.5.1.3 0004146,0005515,0005542,0005829,0006730,0009257,0009410,0016491,0031427,0046452,0046654,0046655,0046656,0046677,0050661,0051870,0051871,0070401,0070402 Kd=281nM remove_due_to_license_issue IC50=8.8nM, EC50=1nM P0ABQ4 8265622 361 MISLIAALAVDRVIGMENAMPWNLPASLAWFKRNTLDKPVIMGRHTWESIGRPLPGRKNIILSSQPGTDDRVTWVKSVDEAIAACGDVPEIMVIGGGRVYEQFLPKAQKLYLTHIDAEVEGDTHFPDYEPDDWESVSSEFHDADAQNSHSYCFEILERR 1di8 A 2.2 BS01 DTQ A 1 I10 A31 K33 F80 F82 L83 H84 L134 D145 I10 A31 K33 F74 F76 L77 H78 L128 D139 D127 K129 Q131 N132 D145 T165 D121 K123 Q125 N126 D139 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1uM remove_due_to_license_issue IC50=1000nM P24941 10633045 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1di9 A 2.6 BS01 MSQ A 1 V30 A51 K53 L104 T106 L108 M109 V27 A48 K50 L101 T103 L105 M106 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 10633045 500 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 1dif A 1.7 BS01 A85 B 1 R8 D25 G27 A28 D29 G48 G49 V82 I84 R8 D25 G27 A28 D29 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 8551523 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1dif B 1.7 BS01 A85 B 1 R8 D25 G27 A28 D29 G48 G49 I50 I84 R8 D25 G27 A28 D29 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=22pM remove_due_to_license_issue P03367 8551523 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1dis A -1.00 BS01 BDM A 1 W5 A6 L19 D26 L27 H28 F30 R31 S48 F49 P50 W5 A6 L19 D26 L27 H28 F30 R31 S48 F49 P50 L4 L19 W21 D26 L27 F30 L54 L94 T116 L4 L19 W21 D26 L27 F30 L54 L94 T116 1.5.1.3 0004146,0005829,0006730,0016491,0031427,0046452,0046654,0046655,0046677,0050661 remove_due_to_license_issue P00381 7547901 163 TAFLWAQDRDGLIGKDGHLPWHLPDDLHYFRAQTVGKIMVVGRRTYESFPKRPLPERTNVVLTHQEDYQAQGAVVVHDVAAVFAYAKQHPDQELVIAGGAQIFTAFKDDVDTLLVTRLAGSFEGDTKMIPLNWDDFTKVSSRTVEDTNPALTHTYEVWQKKA 1dl7 H 2.35 BS01 NCH L 1 W52 Y99 W52 Y99 ? 0002250,0003823,0005576,0016064,0019814 remove_due_to_license_issue P01820 10859335 999 QVQLKESGPGLVAPSQSLSITCTVSGFSLTGYGVNWVRQPPGKGLEWLGMIWGDGSTDYNSALKSRLNISKDKSKSQVFLRMYSLQTDDTARYYCARDYGPYWGQGTLVTVS 1dl7 L 2.35 BS01 NCH L 1 Y34 G52 H55 W93 Y34 G52 H55 W93 ? 0002250,0006955,0019814 Kd=0.32uM remove_due_to_license_issue P01724 10859335 999 QAVVTQESALTTSPGETVTLTCRSSTGAVTTSNYANWVQEKPDHLFTGLIGGTKHRTPGAPARFSGSLIGDKAALTITGAQTEDEAIYFCALWYSNHWVFGGGTKLTVL 1dm2 A 2.1 BS01 HMD A 1 A31 F80 E81 F82 L83 L134 D145 A31 F71 E72 F73 L74 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T141 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 10662688 400 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1dmp A 2.0 BS01 DMQ B 1 D25 G27 A28 D30 G49 I50 V82 D25 G27 A28 D30 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 8807858 450 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1dmp B 2.0 BS01 DMQ B 1 D25 G27 A28 D30 G49 I50 I84 D25 G27 A28 D30 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.28nM remove_due_to_license_issue P04585 8807858 450 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1dmt A 2.1 BS02 RDF A 1 R102 F106 R110 N542 A543 F544 V580 E584 H587 E646 H711 R717 R49 F53 R57 N489 A490 F491 V527 E531 H534 E593 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 remove_due_to_license_issue IC50=30nM P08473 10669592 750 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 1doj A 1.7 BS02 1Z0 A 1 H57 Y60A W60D K60F L99 D189 A190 E192 G193 S195 S214 W215 G216 H77 Y81 W84 K86 L130 D233 A234 E236 G237 S239 S260 W261 G262 H57 D102 E192 G193 D194 S195 G196 H77 D133 E236 G237 D238 S239 G240 3.4.21.5 0004252,0005509,0005576,0006508,0007596 remove_due_to_license_issue P00734 11053836 401 TFGSGEADCGLRPLFEKKSLEDKTERELLESYIDIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1dqn A 1.75 BS02 IMU A 1 D125 E126 Y127 D129 S130 G131 T133 W180 L181 D125 E126 Y127 D129 S130 G131 T133 W180 L181 2.4.2.8 0000166,0000287,0004422,0005829,0006178,0016757,0032263,0032264,0046100,0046872 Ki=10nM remove_due_to_license_issue Q24973 10841757 300 MICSVTGKPVKDVLSTFFKDRNDVLESEVKKFHLLATFEECKALAADTARRMNEYYKDVAEPVTLVALLTGAYLYASLLTVHLTFPYTLHFVKVSSYKGTRQESVVFDEEDLKQLKEKREVVLIDEYVDSGHTIFSIQEQIKHAKICSCFVKDVDAIKKHSALADTKMFYGYTPMPKGSWLIGFGLDDNGLRRGWAHLFDINLSESEVTEFRRRLTEHIKGLNINGVNRY 1dqx A 2.4 BS01 BMP A 1 S35 D37 K59 H61 D91 K93 L153 S154 P202 Q215 Y217 G234 R235 S35 D37 K59 H61 D91 K93 L153 S154 P202 Q215 Y217 G234 R235 4.1.1.23 0004590,0005829,0006207,0006221,0006222,0016831,0044205,0055086,0072528 Ki=9pM remove_due_to_license_issue Ki=0.0090nM P03962 10681417 601 MHKATYKERAATHPSPVAAKLFNIMHEKQTNLCASLDVRTTKELLELVEALGPKICLLKTHVDILTDFSMEGTVKPLKALSAKYNFLLFEDRKFADIGNTVKLQYSAGVYRIAEWADITNAHGVVGPGIVSGLKQAAEEVTKEPRGLLMLAELSCKGSLSTGEYTKGTVDIAKSDKDFVIGFIAQRDMGGRDEGYDWLIMTPGVGLDDKGDALGQQYRTVDDVVSTGSDIIIVGRGLFAKGRDAKVEGERYRKAGWEAYLRRCGQQD 1dqx A 2.4 BS02 BMP B 1 D96 I97 T100 D96 I97 T100 4.1.1.23 0004590,0005829,0006207,0006221,0006222,0016831,0044205,0055086,0072528 Ki=9pM remove_due_to_license_issue Ki=0.0090nM P03962 10681417 602 MHKATYKERAATHPSPVAAKLFNIMHEKQTNLCASLDVRTTKELLELVEALGPKICLLKTHVDILTDFSMEGTVKPLKALSAKYNFLLFEDRKFADIGNTVKLQYSAGVYRIAEWADITNAHGVVGPGIVSGLKQAAEEVTKEPRGLLMLAELSCKGSLSTGEYTKGTVDIAKSDKDFVIGFIAQRDMGGRDEGYDWLIMTPGVGLDDKGDALGQQYRTVDDVVSTGSDIIIVGRGLFAKGRDAKVEGERYRKAGWEAYLRRCGQQD 1dqx B 2.4 BS01 BMP A 1 D96 I97 T100 D96 I97 T100 4.1.1.23 0004590,0005829,0006207,0006221,0006222,0016831,0044205,0055086,0072528 Ki=9pM remove_due_to_license_issue Ki=0.0090nM P03962 10681417 601 MHKATYKERAATHPSPVAAKLFNIMHEKQTNLCASLDVRTTKELLELVEALGPKICLLKTHVDILTDFSMEGTVKPLKALSAKYNFLLFEDRKFADIGNTVKLQYSAGVYRIAEWADITNAHGVVGPGIVSGLKQAAEEVTKEPRGLLMLAELSCKGSLSTGEYTKGTVDIAKSDKDFVIGFIAQRDMGGRDEGYDWLIMTPGVGLDDKGDALGQQYRTVDDVVSTGSDIIIVGRGLFAKGRDAKVEGERYRKAGWEAYLRRCGQQD 1dqx B 2.4 BS02 BMP B 1 S35 D37 K59 H61 D91 K93 L153 S154 P202 Q215 Y217 G234 R235 S35 D37 K59 H61 D91 K93 L153 S154 P202 Q215 Y217 G234 R235 4.1.1.23 0004590,0005829,0006207,0006221,0006222,0016831,0044205,0055086,0072528 Ki=9pM remove_due_to_license_issue Ki=0.0090nM P03962 10681417 602 MHKATYKERAATHPSPVAAKLFNIMHEKQTNLCASLDVRTTKELLELVEALGPKICLLKTHVDILTDFSMEGTVKPLKALSAKYNFLLFEDRKFADIGNTVKLQYSAGVYRIAEWADITNAHGVVGPGIVSGLKQAAEEVTKEPRGLLMLAELSCKGSLSTGEYTKGTVDIAKSDKDFVIGFIAQRDMGGRDEGYDWLIMTPGVGLDDKGDALGQQYRTVDDVVSTGSDIIIVGRGLFAKGRDAKVEGERYRKAGWEAYLRRCGQQD 1drj A 2.5 BS01 RIP A 1 N13 F15 D89 R90 R141 F164 N190 D215 N13 F15 D89 R90 R141 F164 N190 D215 ? 0005515,0006935,0015752,0016020,0030246,0030288,0042597,0048029,0050918,0055052,0055085 Kd=0.04uM remove_due_to_license_issue P02925 7982928 272 KDTIALVVSTLNNPFFVSLKDGAQKEADKLGYNLVVLDSQNNPAKELANVQDLTVRGTKILLINPTDSDAVGNAVKMANQANIPVITLDRQATKGEVVSHIASDNVLGGKIAGDYIAKKAGEGAKVIELQGIARTSAARERGEGFQQAVAAHKFNVLASQPADFDRIKGLNVMQNLLTAHPDVQAVFAQNDEMALGALRALQTAGKSDVMVVGFDGTPDGEKAVNDGKLAATIAQLPDQIGAKGVETADKVLKGEKVQAKYPVDLKLVVKQ 1drk A 2.0 BS01 RIP A 1 N13 F15 F16 D89 R90 R141 F164 N190 D215 Q235 N13 F15 F16 D89 R90 R141 F164 N190 D215 Q235 ? 0005515,0006935,0015752,0016020,0030246,0030288,0042597,0048029,0050918,0055052,0055085 Kd=0.15uM remove_due_to_license_issue P02925 7982928 272 KDTIALVVSTLNNPFFVSLKDGAQKEADKLGYNLVVLDSQNNPAKELANVQDLTVRGTKILLINPTDSDAVGNAVKMANQANIPVITLDRQATKGEVVSHIASDNVLGGKIAGDYIAKKAGEGAKVIELQGTAATSAARERGEGFQQAVAAHKFNVLASQPADFDRIKGLNVMQNLLTAHPDVQAVFAQNDEMALGALRALQTAGKSDVMVVGFDGTPDGEKAVNDGKLAATIAQLPDQIGAKGVETADKVLKGEKVQAKYPVDLKLVVKQ 1drv A 2.2 BS01 A3D A 1 G12 G15 R16 M17 E38 F79 T80 R81 G84 G102 A127 F129 R240 G9 G12 R13 M14 E35 F76 T77 R78 G81 G99 A124 F126 R237 H159 K163 H156 K160 1.17.1.8 0005737,0005829,0008652,0008839,0009085,0009089,0016491,0016726,0019877,0042802,0050661,0051287 Kd=0.29uM remove_due_to_license_issue P04036 8873595 301 ANIRVAIAGAGGRMGRQLIQAALALEGVQLGAALEREGSSLLGSDAGELAGAGKTGVTVQSSLDAVKDDFDVFIDFTRPEGTLNHLAFCRQHGKGMVIGTTGFDEAGKQAIRDAAADIAIVFAANFSVGVNVMLKLLEKAAKVMGDYTDIEIIEAHHRHKVDAPSGTALAMGEAIAHALDKDLKDCAVYSREGHTGERVPGTIGFATVRAGDIVGEHTAMFADIGERLEITHKASSRMTFANGAVRSALWLSGKESGLFDMRDVLDLNNL 1dth A 2.0 BS03 BAT A 1 L108 G109 L110 T139 H142 E143 H152 C164 I165 R167 P168 G169 L170 T171 Y176 L108 G109 L110 T139 H142 E143 H152 C164 I165 R167 P168 G169 L170 T171 Y176 3.4.24.42 0004222,0006508,0008237 ic50=6nM remove_due_to_license_issue P15167 8610113 972 QNLPQRYIELVVVADHRVFMKYNSDLNTIRTRVHEIVNFINGFYRSLNIHVSLTDLEIWSNEDQINIQSASSDTLNAFAEWRETDLLNRKSHDNAQLLTAIELDEETLGLAPLGTMCDPKLSIGIVQDHSPINLLMGVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTKGRSYEFSDDSMHYYERFLKQYKPQCILNKP 1dtq A 2.8 BS01 FPT A 1 K101 K103 V179 Y181 Y188 W229 L234 H235 P236 Y318 K98 K100 V176 Y178 Y185 W226 L231 H232 P233 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 10681546 999 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAH 1dtt A 3.0 BS01 FTC A 1 L100 K101 V106 V179 Y181 Y188 F227 L234 H235 Y318 L100 K101 V106 V177 Y179 Y186 F225 L232 H233 Y316 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 10681546 999 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIG 1du0 A 2.0 BS01 dna C 0 F8 Q44 I47 N51 F2 Q38 I41 N45 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 10889025 201 ~ 221 AFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFANKRAKIKKS 1du0 A 2.0 BS02 dna D 0 Y25 R53 K57 Y19 R47 K51 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 10889025 301 ~ 321 AFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFANKRAKIKKS 1du0 B 2.0 BS01 dna C 0 Y125 E128 R131 R153 K157 Y23 E26 R29 R51 K55 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 10889025 201 ~ 221 RPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFANKRAKIKK 1du0 B 2.0 BS02 dna D 0 R103 I147 N151 R1 I45 N49 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 10889025 301 ~ 321 RPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFANKRAKIKK 1dub A 2.5 BS01 CAA A 1 K56 A57 L58 A60 A96 A98 D99 I100 Y137 G140 G141 E144 P163 E164 L167 G172 K26 A27 L28 A30 A66 A68 D69 I70 Y107 G110 G111 E114 P133 E134 L137 G142 A98 M103 S113 L117 G141 E144 P163 E164 T169 P171 G172 K257 F267 A68 M73 S83 L87 G111 E114 P133 E134 T139 P141 G142 K227 F237 4.2.1.17,5.3.3.8 0003824,0004165,0004300,0005739,0005759,0006631,0006635,0016829,0016836,0016853,0043956,0120092 Ki=1.6uM remove_due_to_license_issue P14604 8895557 300 ANFQYIITEKKGKNSSVGLIQLNRPKALNALCNGLIEELNQALETFEEDPAVGAIVLTGGEKAFAAGADIKEMQNRTFQDCYSGKFLSHWDHITRIKKPVIAAVNGYALGGGCELAMMCDIIYAGEKAQFGQPEILLGTIPGAGGTQRLTRAVGKSLAMEMVLTGDRISAQDAKQAGLVSKIFPVETLVEEAIQCAEKIANNSKIIVAMAKESVNAAFEMTLTEGNKLEKKLFYSTFATDDRREGMSAFVEKRKANFKDH 1dub A 2.5 BS02 CAA C 1 F263 F279 F233 F249 A98 M103 S113 L117 G141 E144 P163 E164 T169 P171 G172 K257 F267 A68 M73 S83 L87 G111 E114 P133 E134 T139 P141 G142 K227 F237 4.2.1.17,5.3.3.8 0003824,0004165,0004300,0005739,0005759,0006631,0006635,0016829,0016836,0016853,0043956,0120092 Ki=1.6uM remove_due_to_license_issue P14604 8895557 300 ANFQYIITEKKGKNSSVGLIQLNRPKALNALCNGLIEELNQALETFEEDPAVGAIVLTGGEKAFAAGADIKEMQNRTFQDCYSGKFLSHWDHITRIKKPVIAAVNGYALGGGCELAMMCDIIYAGEKAQFGQPEILLGTIPGAGGTQRLTRAVGKSLAMEMVLTGDRISAQDAKQAGLVSKIFPVETLVEEAIQCAEKIANNSKIIVAMAKESVNAAFEMTLTEGNKLEKKLFYSTFATDDRREGMSAFVEKRKANFKDH 1dub B 2.5 BS01 CAA A 1 F279 K282 F248 K251 A98 M103 S113 L117 G141 E144 P163 E164 T169 P171 G172 K257 F267 A67 M72 S82 L86 G110 E113 P132 E133 T138 P140 G141 K226 F236 4.2.1.17,5.3.3.8 0003824,0004165,0004300,0005739,0005759,0006631,0006635,0016829,0016836,0016853,0043956,0120092 Ki=1.6uM remove_due_to_license_issue P14604 8895557 300 NFQYIITEKKGKNSSVGLIQLNRPKALNALCNGLIEELNQALETFEEDPAVGAIVLTGGEKAFAAGADIKEMQNRTFQDCYSGKFLSHWDHITRIKKPVIAAVNGYALGGGCELAMMCDIIYAGEKAQFGQPEILLGTIPGAGGTQRLTRAVGKSLAMEMVLTGDRISAQDAKQAGLVSKIFPVETLVEEAIQCAEKIANNSKIIVAMAKESVNAAFEMTLTEGNKLEKKLFYSTFATDDRREGMSAFVEKRKANFKDH 1dub B 2.5 BS02 CAA B 1 K56 A57 L58 A60 A96 A98 D99 I100 M103 G140 G141 E144 P163 E164 L167 G172 K25 A26 L27 A29 A65 A67 D68 I69 M72 G109 G110 E113 P132 E133 L136 G141 A98 M103 S113 L117 G141 E144 P163 E164 T169 P171 G172 K257 F267 A67 M72 S82 L86 G110 E113 P132 E133 T138 P140 G141 K226 F236 4.2.1.17,5.3.3.8 0003824,0004165,0004300,0005739,0005759,0006631,0006635,0016829,0016836,0016853,0043956,0120092 Ki=1.6uM remove_due_to_license_issue P14604 8895557 300 NFQYIITEKKGKNSSVGLIQLNRPKALNALCNGLIEELNQALETFEEDPAVGAIVLTGGEKAFAAGADIKEMQNRTFQDCYSGKFLSHWDHITRIKKPVIAAVNGYALGGGCELAMMCDIIYAGEKAQFGQPEILLGTIPGAGGTQRLTRAVGKSLAMEMVLTGDRISAQDAKQAGLVSKIFPVETLVEEAIQCAEKIANNSKIIVAMAKESVNAAFEMTLTEGNKLEKKLFYSTFATDDRREGMSAFVEKRKANFKDH 1duv G 1.7 BS01 PSQ G 1 S55 T56 R57 T58 R106 L128 H133 N167 D231 S235 M236 C273 L274 R319 S55 T56 R57 T58 R106 L128 H133 N167 D231 S235 M236 C273 L274 R319 2.1.3.3 0004585,0005737,0006520,0006526,0006591,0016597,0016740,0016743,0019240,0042450,0046872 Kd=1.6pM remove_due_to_license_issue P04391 10747936 401 SGFYHKHFLKLLDFTPAELNSLLQLAAKLKADKKSGKEEAKLTGKNIALIFEKDSTRTRCSFEVAAYDQGARVTYLGPSGSQIGHKESIKDTARVLGRMYDGIQYRGYGQEIVETLAEYASVPVWNGLTNEFHPTQLLADLLTMQEHLPGKAFNEMTLVYAGDARNNMGNSMLEAAALTGLDLRLVAPQACWPEAALVTECRALAQQNGGNITLTEDVAKGVEGADFIYTDVWVSMGEAKEKWAERIALLREYQVNSKMMQLTGNPEVKFLHCLPAFHDDQTTLGKKMAEEFGLHGGMEVTDEVFESAASIVFDQAENRMHTIKAVMVATLSK 1duv I 1.7 BS01 PSQ I 1 S55 T56 R57 T58 R106 L128 H133 Q136 N167 D231 S235 M236 C273 L274 R319 S55 T56 R57 T58 R106 L128 H133 Q136 N167 D231 S235 M236 C273 L274 R319 2.1.3.3 0004585,0005737,0006520,0006526,0006591,0016597,0016740,0016743,0019240,0042450,0046872 Kd=1.6pM remove_due_to_license_issue P04391 10747936 403 SGFYHKHFLKLLDFTPAELNSLLQLAAKLKADKKSGKEEAKLTGKNIALIFEKDSTRTRCSFEVAAYDQGARVTYLGPSGSQIGHKESIKDTARVLGRMYDGIQYRGYGQEIVETLAEYASVPVWNGLTNEFHPTQLLADLLTMQEHLPGKAFNEMTLVYAGDARNNMGNSMLEAAALTGLDLRLVAPQACWPEAALVTECRALAQQNGGNITLTEDVAKGVEGADFIYTDVWVSMGEAKEKWAERIALLREYQVNSKMMQLTGNPEVKFLHCLPAFHDDQTTLGKKMAEEFGLHGGMEVTDEVFESAASIVFDQAENRMHTIKAVMVATLSK 1dwc H 3.0 BS03 MIT H 1 H57 Y60A W60D D189 A190 S195 W215 G216 H43 Y47 W50 D199 A200 S205 W227 G228 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 1939071 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1dwd H 3.0 BS03 MID H 1 H57 Y60A W60D N98 L99 I174 D189 A190 W215 G216 H43 Y47 W50 N95 L96 I179 D199 A200 W227 G228 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=6nM, IC50=690nM, EC50=750nM P00734 1939071 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1dx6 A 2.3 BS01 GNT A 1 W84 G117 G118 G119 Y121 E199 S200 F290 F331 H440 W81 G114 G115 G116 Y118 E196 S197 F287 F328 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 ic50=652nM remove_due_to_license_issue IC50=1069nM, Ki=1.9e+2nM P04058 10606746 602 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1dy4 A 1.9 BS01 SNP A 1 Y145 Q175 E212 E217 T246 D369 Y371 W376 Y145 Q175 E212 E217 T246 D369 Y371 W376 E212 D214 E217 H228 E212 D214 E217 H228 3.2.1.91 0004553,0005975 Ki=44uM remove_due_to_license_issue P62694 11114249 437 ESACTLQSETHPPLTWQKCSSGGTCTQQTGSVVIDANWRWTHATNSSTNCYDGNTWSSTLCPDNETCAKNCCLDGAAYASTYGVTTSGNSLSIGFVTQSAQKNVGARLYLMASDTTYQEFTLLGNEFSFDVDVSQLPCGLNGALYFVSMDADGGVSKYPTNTAGAKYGTGYCDSQCPRDLKFINGQANVEGWEPSSNNANTGIGGHGSCCSEMDIWEANSISEALTPHPCTTVGQEICEGDGCGGTYSDNRYGGTCDPDGCDWNPYRLGNTSFYGPGSSFTLDTTKKLTVVTQFETSGAINRYYVQNGVTFQQPNAELGSYSGNELNDDYCTAEEAEFGGSSFSDKGGLTQFKKATSGGMVLVMSLWDDYYANMLWLDSTYPTNETSSTPGAVRGSCSTSSGVPAQVESQSPNAKVTFSNIKFGPIGSTGNPSG 1dzj A 2.0 BS01 SES A 1 L53 Y82 F88 I100 L44 Y73 F79 I91 ? 0005549,0005576,0005615,0007608,0036094 ic50=1.3uM remove_due_to_license_issue P81245 10864504 700 FELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1dzk A 1.48 BS01 PRZ A 1 F35 M39 M114 F26 M30 M105 ? 0005549,0005576,0005615,0007608,0036094 Kd=0.8uM remove_due_to_license_issue P81245 10864504 700 FELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1dzm A 1.93 BS01 BZM A 1 M39 V80 N102 M114 T115 G116 M31 V72 N94 M106 T107 G108 ? 0005549,0005576,0005615,0007608,0036094 ic50=3.9uM remove_due_to_license_issue P81245 10864504 600 PFELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1dzp B 1.83 BS01 BZQ B 1 I21 V80 F88 N102 G116 I11 V70 F78 N92 G106 ? 0005549,0005576,0005615,0007608,0036094 ic50=3.6uM remove_due_to_license_issue P81245 10864504 600 ELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1e00 A 1.83 BS01 DHM A 1 F88 N102 M114 T115 F80 N94 M106 T107 ? 0005549,0005576,0005615,0007608,0036094 ic50=0.8uM remove_due_to_license_issue P81245 10864504 600 PFELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1e02 A 2.15 BS01 UNA A 1 V37 M39 L53 L118 V29 M31 L45 L110 ? 0005549,0005576,0005615,0007608,0036094 ic50=0.7uM remove_due_to_license_issue P81245 10864504 600 PFELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1e06 A 2.12 BS01 IPB A 1 V37 N86 N102 V29 N78 N94 ? 0005549,0005576,0005615,0007608,0036094 ic50=2.5uM remove_due_to_license_issue P81245 10864504 600 PFELSGKWITSYIGSSDLEKIGENAPFQVFMRSIEFDDKESKVYLNFFSKENGICEEFSLIGTKQEGNTYDVNYAGNNKFVVSYASETALIISNINVDEEGDKTIMTGLLGKGTDIEDQDLEKFKEVTRENGIPEENIVNIIERDDCPA 1e1v A 1.95 BS01 CMG A 1 A31 K33 E81 F82 L83 L134 A31 K33 E73 F74 L75 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=12uM remove_due_to_license_issue IC50=17000nM P24941 10956187 401 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1e1x A 1.85 BS01 NW1 A 1 K33 E81 F82 L83 L134 K33 E73 F74 L75 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=1.3uM remove_due_to_license_issue IC50=2200nM, Ki=1300nM P24941 10956187 401 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1e1y A 2.23 BS01 CPB A 1 N284 F285 L380 E382 A610 G612 Y613 N270 F271 L355 E357 A585 G587 Y588 H377 K568 R569 K574 T676 K680 H352 K543 R544 K549 T651 K655 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=2.5uM remove_due_to_license_issue IC50=1200nM P00489 10924512 940 SDQEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPD 1e2k A 1.7 BS01 TMC A 1 H58 E83 I97 Q125 M128 R163 A168 Y172 R222 H13 E34 I48 Q76 M79 R110 A115 Y119 R169 K62 E83 D162 R163 R220 E225 K17 E34 D109 R110 R167 E172 2.7.1.21 0004797,0005524,0006230 Ki=11.4uM remove_due_to_license_issue P0DTH5 10924157 500 MPTLLRVYIDGPHGMGKTTTTQLLVADDIVYVPEPMTYWRVLGASETIANIYTTQHRLDQGEISAGDAAVVMTSAQITMGMPYAVTDAVLAPHIGGEAGPPPALTLIFDRHPIAALLCYPAARYLMGSMTPQAVLAFVALIPPTLPGTNIVLGALPEDRHIDRLAKRQRPGERLDLAMLAAIRRVYGLLANTVRYLQCGGSWREDWGQLSGTGPRPHIGDTLFTLFRAPELLAPNGDLYNVFAWALDVLAKRLRSMHVFILDYDQSPAGCRDALLQLTSGMVQTHVTTPGSIPTICDLARTFAREMGE 1e2l A 2.4 BS01 TMC A 1 H58 I97 Q125 M128 R163 Y172 R222 H13 I45 Q73 M76 R108 Y117 R167 K62 E83 D162 R163 K17 E31 D107 R108 2.7.1.21 0004797,0005524,0006230 Ki=51.5uM remove_due_to_license_issue P0DTH5 10924157 500 MPTLLRVYIDGPHGMGKTTTTQLLDIVYVPEPMTYWRVLGASETIANIFTTQHRLDQGEISAGDAAVVMTSAQITMGMPYAVTDAVLAPHIGGEAGSPPPALTLIFDRHPIAALLCYPAARYLMGSMTPQAVLAFVALIPPTLPGTNIVLGALPEDRHIDRLAKRQRPGERLDLAMLAAIRRVYGLLANTVRYLQCGGSWREDWGQLSGPRPHIGDTLFTLFRAPELLAPNGDLYNVFAWALDVLAKRLRSMHVFILDYDQSPAGCRDALLQLTSGMVQTHVTTPGSIPTICDLARTFAREMGE 1e34 B 1.8 BS02 TPX B 1 H57 R61 C191 Q192 S195 F215 V216 H45 R49 C184 Q185 S188 F208 V209 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 11023818 280 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1e37 B 1.75 BS02 TPY B 1 C42 H57 C58 R61 C191 Q192 G193 S195 F215 V216 C30 H45 C46 R49 C184 Q185 G186 S188 F208 V209 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 11023818 280 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1e3g A 2.4 BS01 R18 A 1 L704 N705 Q711 M745 M749 F764 T877 M895 L36 N37 Q43 M77 M81 F96 T209 M227 ? remove_due_to_license_issue Kd=0.99nM, IC50=0.302000nM, EC50=0.013000nM, Ki=0.400000nM P10275 10840043 1000 CQPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 1e3v A 2.0 BS01 DXC A 1 Y16 D40 Y57 G60 L99 D103 M116 Y15 D39 Y56 G59 L98 D102 M115 Y16 D40 D100 D103 Y15 D39 D99 D102 5.3.3.1 0004769,0008202,0016853 Kd=45.74uM remove_due_to_license_issue P07445 11007792 801 NLPTAQEVQGLMARYIELVDVGDIEAIVQMYADDATVEDPFGQPPIHGREQIAAFYRQGLGGGKVRACLTGPVRASHNGCGAMPFRVEMVWNGQPCALDVIDVMRFDEHGRIQTMQAYWSEVNLSVRE 1e4h A 1.8 BS01 PBR B 1 K15 L17 A108 T119 K6 L8 A99 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.9nM remove_due_to_license_issue P02766 10957627 999 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 1e4h B 1.8 BS01 PBR A 1 K15 L17 A108 T119 K6 L8 A99 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.9nM remove_due_to_license_issue P02766 10957627 998 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 1e55 A 2.0 BS01 BGC A 1 D191 Y333 E406 W457 E464 Y473 D182 Y324 E397 W448 E455 Y464 R96 H142 D191 T194 N331 Y333 E406 R87 H133 D182 T185 N322 Y324 E397 3.2.1.182,3.2.1.21 0004553,0005975,0008422,0009507,0009736,0015923,0015925,0015928,0016162,0016798,0097599,0102726 remove_due_to_license_issue P49235 11106394 513 VQMLSPSEIPQRDWFPSDFTFGAATSAYQIEGAWNEDGKGESNWDHFCHNHPERILDGSNSDIGANSYHMYKTDVRLLKEMGMDAYRFSISWPRILPKGTKEGGINPDGIKYYRNLINLLLENGIEPYVTIFHWDVPQALEEKYGGFLDKSHKSIVEDYTYFAKVCFDNFGDKVKNWLTFNDPQTFTSFSYGTGVFAPGRCSPGLDCAYPTGNSLVEPYTAGHNILLAHAEAVDLYNKHYKRDDTRIGLAFDVMGRVPYGTSFLDKQAEERSWDINLGWFLEPVVRGDYPFSMRSLARERLPFFKDEQKEKLAGSYNMLGLNYYTSRFSKNIDISPNYSPVLNTDDAYASQEVNGPDGKPIGPPMGNPWIYMYPEGLKDLLMIMKNKYGNPPIYITENGIGDVDTKETPLPMEAALNDYKRLDYIQRHIATLKESIDLGSNVQGYFAWSLLDNFEWFAGFTERYGIVYVDRNNNCTRYMKESAKWLKEFNTA 1e55 A 2.0 BS02 DHR A 1 F198 F466 F189 F457 R96 H142 D191 T194 N331 Y333 E406 R87 H133 D182 T185 N322 Y324 E397 3.2.1.182,3.2.1.21 0004553,0005975,0008422,0009507,0009736,0015923,0015925,0015928,0016162,0016798,0097599,0102726 Ki=76uM remove_due_to_license_issue P49235 11106394 514 VQMLSPSEIPQRDWFPSDFTFGAATSAYQIEGAWNEDGKGESNWDHFCHNHPERILDGSNSDIGANSYHMYKTDVRLLKEMGMDAYRFSISWPRILPKGTKEGGINPDGIKYYRNLINLLLENGIEPYVTIFHWDVPQALEEKYGGFLDKSHKSIVEDYTYFAKVCFDNFGDKVKNWLTFNDPQTFTSFSYGTGVFAPGRCSPGLDCAYPTGNSLVEPYTAGHNILLAHAEAVDLYNKHYKRDDTRIGLAFDVMGRVPYGTSFLDKQAEERSWDINLGWFLEPVVRGDYPFSMRSLARERLPFFKDEQKEKLAGSYNMLGLNYYTSRFSKNIDISPNYSPVLNTDDAYASQEVNGPDGKPIGPPMGNPWIYMYPEGLKDLLMIMKNKYGNPPIYITENGIGDVDTKETPLPMEAALNDYKRLDYIQRHIATLKESIDLGSNVQGYFAWSLLDNFEWFAGFTERYGIVYVDRNNNCTRYMKESAKWLKEFNTA 1e5a A 1.8 BS01 TBP A 1 K15 L17 K6 L8 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=23nM remove_due_to_license_issue P02766 10957627 999 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 1e5a B 1.8 BS01 TBP B 1 K15 A108 K6 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=23nM remove_due_to_license_issue P02766 10957627 999 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 1e5j A 1.85 BS01 SGC B 1 E139 Y202 E136 Y199 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11828460 2 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESAS 1e5j A 1.85 BS02 SGC B 2 H35 Y66 W262 K267 E269 H32 Y63 W259 K264 E266 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11828460 3 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESAS 1e5j A 1.85 BS03 GLC B 1 W39 K267 W36 K264 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11828460 4 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESAS 1e66 A 2.1 BS01 HUX A 1 W84 G118 G119 Y121 F330 F331 W432 I439 H440 W81 G115 G116 Y118 F327 F328 W429 I436 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=0.13nM remove_due_to_license_issue P04058 11863435 803 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1e6q M 1.35 BS01 NTZ M 1 Q39 H141 Q187 Y330 E409 W457 E464 F465 F473 Q37 H139 Q185 Y328 E407 W455 E462 F463 F471 3.2.1.147 0004553,0005773,0005975,0008422,0016798,0019137,0046872 Ki=0.7mM remove_due_to_license_issue P29736 10978344 999 EITCQENLPFTCGNTDALNSSSFSSDFIFGVASSAYQIEGTIGRGLNIWDGFTHRYPNKSGPDHGNGDTTCDSFSYWQKDIDVLDELNATGYRFSIAWSRIIPRGKRSRGVNEKGIDYYHGLISGLIKKGITPFVTLFHWDLPQTLQDEYEGFLDPQIIDDFKDYADLCFEEFGDSVKYWLTINQLYSVPTRGYGSALDAPGRCSPTVDPSCYAGNSSTEPYIVAHHQLLAHAKVVDLYRKNYTHQGGKIGPTMITRWFLPYNDTDRHSIAATERMKEFFLGWFMGPLTNGTYPQIMIDTVGERLPSFSPEESNLVKGSYDFLGLNYYFTQYAQPSPNPVNSTNHTAMMDAGAKLTYINASGHYIGPLFEKDKADSTDNIYYYPKGIYSVMDYFKNKYYNPLIYVTENGISTPGDENRNQSMLDYTRIDYLCSHLCFLNKVIKEKDVNVKGYLAWALGDNYEFNKGFTVRFGLSYIDWNNVTDRDLKKSGQWYQSFISP 1e6s M 1.35 BS01 GOX M 1 Q39 H141 Q187 Y330 E409 W457 E464 F465 F473 Q37 H139 Q185 Y328 E407 W455 E462 F463 F471 3.2.1.147 0004553,0005773,0005975,0008422,0016798,0019137,0046872 Ki=0.6mM remove_due_to_license_issue P29736 10978344 921 EITCQENLPFTCGNTDALNSSSFSSDFIFGVASSAYQIEGTIGRGLNIWDGFTHRYPNKSGPDHGNGDTTCDSFSYWQKDIDVLDELNATGYRFSIAWSRIIPRGKRSRGVNEKGIDYYHGLISGLIKKGITPFVTLFHWDLPQTLQDEYEGFLDPQIIDDFKDYADLCFEEFGDSVKYWLTINQLYSVPTRGYGSALDAPGRCSPTVDPSCYAGNSSTEPYIVAHHQLLAHAKVVDLYRKNYTHQGGKIGPTMITRWFLPYNDTDRHSIAATERMKEFFLGWFMGPLTNGTYPQIMIDTVGERLPSFSPEESNLVKGSYDFLGLNYYFTQYAQPSPNPVNSTNHTAMMDAGAKLTYINASGHYIGPLFEKDKADSTDNIYYYPKGIYSVMDYFKNKYYNPLIYVTENGISTPGDENRNQSMLDYTRIDYLCSHLCFLNKVIKEKDVNVKGYLAWALGDNYEFNKGFTVRFGLSYIDWNNVTDRDLKKSGQWYQSFISP 1e72 M 1.6 BS02 GOX M 1 Q39 H141 N186 Q187 Y330 E409 W457 E464 F465 F473 Q37 H139 N184 Q185 Y328 E407 W455 E462 F463 F471 3.2.1.147 0004553,0005773,0005975,0008422,0016798,0019137,0046872 Ki=0.6mM remove_due_to_license_issue P29736 10978344 999 EITCQENLPFTCGNTDALNSSSFSSDFIFGVASSAYQIEGTIGRGLNIWDGFTHRYPNKSGPDHGNGDTTCDSFSYWQKDIDVLDELNATGYRFSIAWSRIIPRGKRSRGVNEKGIDYYHGLISGLIKKGITPFVTLFHWDLPQTLQDEYEGFLDPQIIDDFKDYADLCFEEFGDSVKYWLTINQLYSVPTRGYGSALDAPGRCSPTVDPSCYAGNSSTEPYIVAHHQLLAHAKVVDLYRKNYTHQGGKIGPTMITRWFLPYNDTDRHSIAATERMKEFFLGWFMGPLTNGTYPQIMIDTVGERLPSFSPEESNLVKGSYDFLGLNYYFTQYAQPSPNPVNSTNHTAMMDAGAKLTYINASGHYIGPLFEKDKADSTDNIYYYPKGIYSVMDYFKNKYYNPLIYVTENGISTPGDENRNQSMLDYTRIDYLCSHLCFLNKVIKEKDVNVKGYLAWALGDNYEFNKGFTVRFGLSYIDWNNVTDRDLKKSGQWYQSFISP 1e7j A BS01 dna B 0 R7 P8 L9 M13 V32 R7 P8 L9 M13 V32 ? remove_due_to_license_issue 1 ~ 14 MSDKPKRPLSAYMLWLNSARESIKRENPGIKVTEVAKRGGELWRAMKDKSEWEAKAAKAKDDYDRAVKEFEANG 1e7j A BS02 dna C 0 Y12 W43 Y12 W43 ? remove_due_to_license_issue 15 ~ 26 MSDKPKRPLSAYMLWLNSARESIKRENPGIKVTEVAKRGGELWRAMKDKSEWEAKAAKAKDDYDRAVKEFEANG 1e8h A 2.6 BS01 ADP A 1 P99 S101 I102 G103 R104 S175 E182 I261 V262 K545 P84 S86 I87 G88 R89 S160 E167 I246 V247 K530 Y108 D170 E182 D192 D317 V397 E410 I414 H422 H466 Y503 R504 K545 Y93 D155 E167 D177 D302 V382 E395 I399 H407 H451 Y488 R489 K530 1.1.3.38 0003824,0004458,0005737,0005739,0005777,0008720,0015945,0016491,0018465,0050660,0071949,1903457 remove_due_to_license_issue P56216 10984479 600 EFRPLTLPPKLSLSDFNEFIQDIIRIVGSENVEVISMKPTHTHDPTHVMDQDYFLASAIVAPRNVADVQSIVGLANKFSFPLWPISIGRNSGYGGAAPRVSGSVVLDMGKNMNRVLEVNVEGAYCVVEPGVTYHDLHNYLEANNLRDKLWLDVPDLGGGSVLGNAVERGVGYTPYGDHWMMHSGMEVVLANGELLRTGMGALPDPKRPETMGLKPEDQPWSKIAHLFPYGFGPYIDGLFSQSNMGIVTKIGIWLMPNPGGYQSYLITLPKDGDLKQAVDIIRPLRLGMALQNVPTIRHILLDAAVLGDKRSYSSRTEPLSDEELDKIAKQLNLGRWNFYGALYGPEPIRRVLWETIKDAFSAIPGVKFYFPEDTPENSVLRVRDKTMQGIPTYDELKWIDWLPNGAHLFFSPIAKVSGEDAMMQYAVTKKRCQEAGLDFIGTFTVGMREMHHIVCIVFNKKDLIQKRKVQWLMRTLIDDCAANGWGEYRTHLAFMDQIMETYNWNNSSFLRFNEVLKNAVDPNGIIAPGKSGVWPSQYSHVTWKL 1e9h A 2.5 BS01 INR A 1 I10 A31 K33 F80 F82 L83 H84 Q85 K89 L134 D145 I10 A31 K33 F80 F82 L83 H84 Q85 K89 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=35nM remove_due_to_license_issue IC50=3e+2nM P24941 11377199 1298 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1eas A 1.8 BS01 TFK A 1 H57 C191 Q192 G193 S195 S214 F215 V216 R217A H45 C184 Q185 G186 S188 S207 F208 V209 R211 H57 D102 Q192 G193 D194 S195 G196 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 7932559 1 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1eat A 2.0 BS01 TFI A 1 H57 C191 Q192 G193 S195 S214 F215 V216 R217A H45 C184 Q185 G186 S188 S207 F208 V209 R211 H57 D102 Q192 G193 D194 S195 G196 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 7837246 1 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1eb2 A 2.0 BS02 BPO A 1 N97 T98 D189 S190 C191 Q192 V213 W215 G216 S217 G219 C220 N79 T80 D171 S172 C173 Q174 V191 W193 G194 S195 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=16nM remove_due_to_license_issue Ki=980nM P00760 11881991 1248 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1ebg A 2.1 BS02 PAH A 1 G37 A38 S39 H159 Q167 E168 D246 D320 K345 R374 S375 K396 G37 A38 S39 H159 Q167 E168 D246 D320 K345 R374 S375 K396 S39 H159 E168 E211 D246 E295 D320 K345 H373 K396 S39 H159 E168 E211 D246 E295 D320 K345 H373 K396 4.2.1.11 0000015,0000287,0000324,0004634,0005737,0005739,0005829,0005886,0006096,0016829,0032889,0046872,1904408 Ki=15pM remove_due_to_license_issue P00924 8049235 440 AVSKVYARSVYDSRGNPTVEVELTTEKGVFRSIVPSGASTGVHEALEMRDGDKSKWMGKGVLHAVKNVNDVIAPAFVKANIDVKDQKAVDDFLISLDGTANKSKLGANAILGVSLAASRAAAAEKNVPLYKHLADLSKSKTSPYVLPVPFLNVLNGGSHAGGALALQEFMIAPTGAKTFAEALRIGSEVYHNLKSLTKKRYGASAGNVGDEGGVAPNIQTAEEALDLIVDAIKAAGHDGKVKIGLDCASSEFFKDGKYDLDFKNPNSDKSKWLTGPQLADLYHSLMKRYPIVSIEDPFAEDDWEAWSHFFKTAGIQIVADDLTVTNPKRIATAIEKKAADALLLKVNQIGTLSESIKAAQDSFAAGWGVMVSHRSGETEDTFIADLVVGLRTGQIKTGAPARSERLAKLNQLLRIEEELGDNAVFAGENFHHGDKL 1ebw A 1.81 BS01 BEI A 1 D25 G27 A28 D29 G48 G49 I50 V82 I84 D25 G27 A28 D29 G48 G49 I50 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.9nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ebw B 1.81 BS01 BEI A 1 D125 G127 A128 D129 G148 P181 V182 D25 G27 A28 D29 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1eby A 2.294 BS01 BEB B 1 R8 D25 G27 A28 D29 G48 G49 V82 R8 D25 G27 A28 D29 G48 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1eby B 2.294 BS01 BEB B 1 D125 G127 A128 D129 D130 V132 G148 P181 V182 D25 G27 A28 D29 D30 V32 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.2nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ebz A 2.01 BS01 BEC B 1 R8 D25 G27 A28 D29 G48 G49 V82 R8 D25 G27 A28 D29 G48 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ebz B 2.01 BS01 BEC B 1 D125 G127 A128 D129 D130 V132 G148 V182 D25 G27 A28 D29 D30 V32 G48 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.4nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec0 A 1.79 BS01 BED A 1 R8 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 R8 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.2nM remove_due_to_license_issue P03366 15560801 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec0 B 1.79 BS01 BED A 1 R108 D125 G127 A128 D129 D130 V132 G148 G149 I150 V182 R8 D25 G27 A28 D29 D30 V32 G48 G49 I50 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15560801 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec1 A 2.1 BS01 BEE A 1 D25 G27 A28 D29 G48 G49 P81 V82 D25 G27 A28 D29 G48 G49 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.2nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec1 B 2.1 BS01 BEE A 1 D125 G127 A128 D129 G148 G149 P181 V182 I184 D25 G27 A28 D29 G48 G49 P81 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec2 A 2.0 BS01 BEJ B 1 D25 G27 A28 D29 G48 G49 V82 D25 G27 A28 D29 G48 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec2 B 2.0 BS01 BEJ B 1 L123 D125 G127 A128 D129 G148 G149 P181 V182 L23 D25 G27 A28 D29 G48 G49 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.1nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec3 A 1.8 BS01 MS3 A 1 R8 D25 G27 A28 D29 G48 G49 P81 V82 I84 R8 D25 G27 A28 D29 G48 G49 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.92nM remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec3 B 1.8 BS01 MS3 A 1 R108 D125 G127 A128 D129 G148 G149 I150 P181 V182 R8 D25 G27 A28 D29 G48 G49 I50 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12694187 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ec9 A 2.0 BS02 XYH A 1 H32 T103 Y150 K207 D235 N237 N289 H339 S340 N341 H368 R422 H29 T100 Y147 K204 D232 N234 N286 H336 S337 N338 H365 R419 K205 K207 D235 N237 E260 N289 M290 D313 H339 N341 I365 K202 K204 D232 N234 E257 N286 M287 D310 H336 N338 I362 4.2.1.40 0000287,0008872,0016829,0019394,0042838,0046872 Ki=0.8mM remove_due_to_license_issue P0AES2 10769114 499 QFTTPVVTEMQVIPVAGHDSMLMNLSGAHAPFFTRNIVIIKDNSGHTGVGEIPGGEKIRKTLEDAIPLVVGKTLGEYKNVLTLVRNTFADRDAGGRGLQTFDLRTTIHVVTGIEAAMLDLLGQHLGVNVASLLGDGQQRSEVEMLGYLFFVGNRKATPLPYQSQPDDSCDWYRLRHEEAMTPDAVVRLAEAAYEKYGFNDFKLKGGVLAGEEEAESIVALAQRFPQARITLDPNGAWSLNEAIKIGKYLKGSLAYAEDPCGAEQGFSGREVMAEFRRATGLPTATNMIATDWRQMGHTLSLQSVDIPLADPHFWTMQGSVRVAQMCHEFGLTWGSHSNNHFDISLAMFTHVAAAAPGKITAIDTHWIWQEGNQRLTKEPFEIKGGLVQVPEKPGLGVEIDMDQVMKAHELYQKHGLGARDDAMGMQYLIPGWTFDNKRPCMVR 1ecq A 2.0 BS01 DXG A 1 N27 H32 T103 Y150 F152 K207 D235 N237 N289 H339 S340 N341 H368 R422 N25 H30 T101 Y148 F150 K205 D233 N235 N287 H337 S338 N339 H366 R420 K205 K207 D235 N237 E260 N289 M290 D313 H339 N341 I365 K203 K205 D233 N235 E258 N287 M288 D311 H337 N339 I363 4.2.1.40 0000287,0008872,0016829,0019394,0042838,0046872 Ki=1mM remove_due_to_license_issue P0AES2 10769114 499 SQFTTPVVTEMQVIPVAGHDSMLMNLSGAHAPFFTRNIVIIKDNSGHTGVGEIPGGEKIRKTLEDAIPLVVGKTLGEYKNVLTLVRNTFADRDAGGRGLQTFDLRTTIHVVTGIEAAMLDLLGQHLGVNVASLLGDGQQRSEVEMLGYLFFVGNRKATPLPYQSQPDDSCDWYRLRHEEAMTPDAVVRLAEAAYEKYGFNDFKLKGGVLAGEEEAESIVALAQRFPQARITLDPNGAWSLNEAIKIGKYLKGSLAYAEDPCGAEQGFSGREVMAEFRRATGLPTATNMIATDWRQMGHTLSLQSVDIPLADPHFWTMQGSVRVAQMCHEFGLTWGSHSNNHFDISLAMFTHVAAAAPGKITAIDTHWIWQEGNQRLTKEPFEIKGGLVQVPEKPGLGVEIDMDQVMKAHELYQKHGLGARDDAMGMQYLIPGWTFDNKRPCMVR 1ecv A 1.95 BS01 878 A 1 Y46 V49 K120 D181 F182 C215 S216 A217 I219 G220 R221 Y45 V48 K119 D180 F181 C214 S215 A216 I218 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=14uM remove_due_to_license_issue Ki=71449632607551nM P18031 10702277 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1eed P 2.0 BS01 0EO P 1 I7 D30 D32 G34 S74 Y75 G76 D77 D215 G217 T218 T219 I10 D33 D35 G37 S78 Y79 G80 D81 D219 G221 T222 T223 3.4.23.22 0004190,0006508 Ki=16.2uM remove_due_to_license_issue P11838 1525155 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 1eef G 1.8 BS01 GLA G 1 E51 Q56 Q61 W88 N90 K91 E51 Q56 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 remove_due_to_license_issue P32890 11173465 107 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef G 1.8 BS02 I06 G 1 Y12 I58 Y12 I58 ? 0005576,0031640,0035821,0090729 remove_due_to_license_issue P32890 11173465 108 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef H 1.8 BS01 GLA H 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 remove_due_to_license_issue P32890 11173465 109 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef H 1.8 BS02 I06 H 1 Y12 I58 Y12 I58 ? 0005576,0031640,0035821,0090729 remove_due_to_license_issue P32890 11173465 110 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eei D 2.0 BS01 GAA D 1 Y12 E51 Q56 H57 Q61 W88 N90 K91 Y12 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0046872 ic50=0.7mM remove_due_to_license_issue Q57193 11173465 504 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 1eei E 2.0 BS01 GAA E 1 Y12 E51 Q56 W88 N90 K91 Y12 E51 Q56 W88 N90 K91 ? 0005576,0046872 ic50=0.7mM remove_due_to_license_issue Q57193 11173465 505 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 1efi D 1.6 BS01 GAT D 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=12mM remove_due_to_license_issue P32890 11173465 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1efi E 1.6 BS01 GAT E 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=12mM remove_due_to_license_issue P32890 11173465 105 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1efy A 2.2 BS01 BZC A 1 Q763 H862 G863 Y896 F897 S904 Y907 E988 Q102 H201 G202 Y235 F236 S243 Y246 E327 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 Ki=6nM remove_due_to_license_issue P26446 11063605 201 KSKLAKPIQDLIKMIFDVESMKKAMVEFEIDLQKMPLGKLSKRQIQSAYSILNEVQQAVSDGGSESQILDLSNRFYTLIPHDFGMKKPPLLSNLEYIQAKVQMLDNLLDIEVAYSLLRGGNEDGDKDPIDINYEKLRTDIKVVDKDSEEAKIIKQYVKNTHAATHNAYDLKVVEIFRIEREGESQRYKPFKQLHNRQLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQADPIGLILLGEVALGNMYELKNASHITKLPKGKHSVKGLGKTAPDPTATTTLDGVEVPLGNGISTGINDTCLLYNEYIVYDVAQVNLKYLLKLKFNYKT 1egh A 2.0 BS01 PGA A 1 V17 K23 T45 T47 T48 S65 G66 D71 H98 V17 K23 T45 T47 T48 S65 G66 D71 H98 H19 G66 D71 D91 H98 D101 R107 H19 G66 D71 D91 H98 D101 R107 4.2.3.3 0005737,0005829,0008929,0016829,0019242,0034214,0042802 Ki=2uM remove_due_to_license_issue P0A731 10715115 201 MELTTRTLPARKHIALVAHDHCKQMLMSWVERHQPLLEQHVLYATGTTGNLISRATGMNVNAMLSGPMGGDQQVGALISEGKIDVLIFFWDPLNAVPHDPDVKALLRLATVWNIPVATNVATADFIIQSPHFNDAVDILIPDYQRYLADRLK 1egh F 2.0 BS01 PGA F 1 V17 K23 T45 T47 T48 S65 G66 D71 H98 V17 K23 T45 T47 T48 S65 G66 D71 H98 H19 G66 D71 D91 H98 D101 R107 H19 G66 D71 D91 H98 D101 R107 4.2.3.3 0005737,0005829,0008929,0016829,0019242,0034214,0042802 Ki=2uM remove_due_to_license_issue P0A731 10715115 251 MELTTRTLPARKHIALVAHDHCKQMLMSWVERHQPLLEQHVLYATGTTGNLISRATGMNVNAMLSGPMGGDQQVGALISEGKIDVLIFFWDPLNAVPHDPDVKALLRLATVWNIPVATNVATADFIIQSPHFNDAVDILIPDYQRYLADRL 1eix A 2.5 BS01 BMQ A 1 A20 D22 K44 K73 L130 T131 P189 R192 Q201 G221 R222 A9 D11 K33 K62 L119 T120 P178 R181 Q190 G210 R211 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 Ki=8.8pM remove_due_to_license_issue P08244 10757968 1301 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1eix A 2.5 BS02 BMQ B 1 D76 I77 T80 D65 I66 T69 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 Ki=8.8pM remove_due_to_license_issue P08244 10757968 1302 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1eix B 2.5 BS01 BMQ A 1 D76 I77 T80 D65 I66 T69 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 Ki=8.8pM remove_due_to_license_issue P08244 10757968 1301 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1eix B 2.5 BS02 BMQ B 1 A20 D22 K44 K73 L130 T131 P189 R192 Q201 G221 R222 A9 D11 K33 K62 L119 T120 P178 R181 Q190 G210 R211 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 Ki=8.8pM remove_due_to_license_issue P08244 10757968 1302 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1ejn A 1.8 BS01 AGB A 1 C42 D189 S190 C191 Q192 G193 S195 S214 W215 G216 G219 G226 C31 D192 S193 C194 Q195 G196 S198 S217 W218 G219 G221 G229 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=2.4uM remove_due_to_license_issue P00749 10805774 800 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1ek1 A 3.1 BS01 CIU A 1 F265 D333 W334 Y381 Q382 F406 Y465 F211 D279 W280 Y327 Q328 F352 Y411 F265 D333 W334 N357 I376 Y381 Y465 D495 H523 F211 D279 W280 N303 I322 Y327 Y411 D441 H469 3.1.3.76,3.3.2.10 0000287,0003824,0004301,0005737,0005777,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0090181,0097176 remove_due_to_license_issue P34914 10747889 1100 RVAAFDLDGVLALPSIGPTEQLMKGKITFSQWVPLQIFSQAMAARSINRPMLQAAIALKKKGFTTCIVTNNWLDDGDKRDSLAQMMCELSQHFDFLIESCQVGMIKPEPQIYNFLLDTLKAKPNEVVFLDDFGSNLKPARDMGMVTILVHNTASALRELEKVTGTQFPEAPLPVPCNPNDVSHGYVTVKPGIRLHFVEMGSGPALCLCHGFPESWFSWRYQIPALAQAGFRVLAIDMKGYGDSSSPPEIEEYAMELLCKEMVTFLDKLGIPQAVFIGHDWAGVMVWNMALFYPERVRAVASLNTPFMPPDPDVSPMKVIRSIPVFNYQLYFQEPGVAEAELEKNMSRTFKSFFRASDETGFIAVHKATEIGGILVNTPEDPNLSKITTEEEIEFYIQQFKKTGFRGPLNWYRNTERNWKWSCKGLGRKILVPALMVTAEKDIVLRPEMSKNMEKWIPFLKRGHIEDCGHWTQIEKPTEVNQILIKWLQTE 1ek2 A 3.0 BS01 CDU A 1 F265 D333 Y381 Q382 F406 Y465 H523 W524 F208 D276 Y324 Q325 F349 Y408 H466 W467 F265 D333 W334 N357 I376 Y381 Y465 D495 H523 F208 D276 W277 N300 I319 Y324 Y408 D438 H466 3.1.3.76,3.3.2.10 0000287,0003824,0004301,0005737,0005777,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0090181,0097176 remove_due_to_license_issue IC50=50nM P34914 10747889 1100 RVAAFDLDGVLALPSIGPTEQLMKGKITFSQWQIFSQAMAARSINRPMLQAAIALKKKGFTTCIVTNNWLDDGDKRDSLAQMMCELSQHFDFLIESCQVGMIKPEPQIYNFLLDTLKAKPNEVVFLDDFGSNLKPARDMGMVTILVHNTASALRELEKVTGTQFPEAPLPVPCNPNDVSHGYVTVKPGIRLHFVEMGSGPALCLCHGFPESWFSWRYQIPALAQAGFRVLAIDMKGYGDSSSPPEIEEYAMELLCKEMVTFLDKLGIPQAVFIGHDWAGVMVWNMALFYPERVRAVASLNTPFMPPDPDVSPMKVIRSIPVFNYQLYFQEPGVAEAELEKNMSRTFKSFFRASDETGFIAVHKATEIGGILVNTPEDPNLSKITTEEEIEFYIQQFKKTGFRGPLNWYRNTERNWKWSCKGLGRKILVPALMVTAEKDIVLRPEMSKNMEKWIPFLKRGHIEDCGHWTQIEKPTEVNQILIKWLQTE 1ela A 2.0 BS01 0Z1 A 1 H60 V103 A104 C199 Q200 S203 S222 F223 V224 H45 V88 A89 C184 Q185 S188 S207 F208 V209 H60 D108 Q200 G201 D202 S203 G204 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 Ki=0.44uM remove_due_to_license_issue P00772 7656008 256 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1elb A 2.1 BS01 0Z4 A 1 H60 C199 Q200 S203 S222 F223 V224 R226 H45 C184 Q185 S188 S207 F208 V209 R211 H60 D108 Q200 G201 D202 S203 G204 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 Ki=70nM remove_due_to_license_issue P00772 7656008 256 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1elc A 1.75 BS01 0Z3 A 1 H60 T100 C199 Q200 S203 T221 S222 F223 V224 S225 R226 L227 G228 H45 T85 C184 Q185 S188 T206 S207 F208 V209 S210 R211 L212 G213 H60 D108 Q200 G201 D202 S203 G204 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 7656008 256 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1eld E 2.0 BS01 0Z0 E 1 H60 V103 C199 Q200 S203 S222 F223 V224 H45 V88 C184 Q185 S188 S207 F208 V209 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 Ki=0.2uM remove_due_to_license_issue P00772 7880814 256 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1ele E 2.0 BS01 0QN E 1 H60 C199 Q200 S203 S222 F223 V224 R226 H45 C184 Q185 S188 S207 F208 V209 R211 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 Ki=0.14uM remove_due_to_license_issue P00772 7880814 256 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1els A 2.4 BS03 PAH A 1 S39 E168 D246 D320 K345 R374 S375 K396 S39 E168 D246 D320 K345 R374 S375 K396 S39 H159 E168 E211 D246 E295 D320 K345 H373 K396 S39 H159 E168 E211 D246 E295 D320 K345 H373 K396 4.2.1.11 0000015,0000287,0000324,0004634,0005737,0005739,0005829,0005886,0006096,0016829,0032889,0046872,1904408 Ki=15pM remove_due_to_license_issue P00924 8193144 439 AVSKVYARSVYDSRGNPTVEVELTTEKGVFRSIVPSGASTGVHEALEMRDGDKSKWMGKGVLHAVKNVNDVIAPAFVKANIDVSDQKAVDDFLISLDGTANKSKLGANAILGVSLAASRAAAAEKNVPLYKHLADLSKSKTSPYVLPVPFLNVLNGGSHAGGALALQEFMIAPTGAKTFAEALRIGSEVYHNLKSLTKKRYGASAGNVGDEGGVAPNIQTAEEALDLIVDAIKAAGHDGKVKIGLDCASSEFFKDGKYDLDFKNPNSDKSKWLTGPQLADLYHSLMKRYPIVSIEDPFAEDDWEAWSHFFKTAGIQIVADDLTVTNPKRIATAIEKKAADALLLKVNQIGTLSESIKAAQDSFAAGWGVMVSHRSGETEDTFIADLVVGLRTGQIKTGAPARSERLAKLNQLLRIEEELGDNAVFAGENFHHGDKL 1em6 A 2.2 BS02 CP4 A 1 T38 V40 R60 W67 P188 E190 K191 P229 T17 V19 R39 W46 P167 E169 K170 P208 H377 K568 R569 K574 T676 K680 H337 K528 R529 K534 T633 K637 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 ic50=6nM remove_due_to_license_issue IC50=6.0nM P06737 10980448 862 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASTVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1em6 B 2.2 BS01 CP4 A 1 T38 V40 R60 W67 E190 K191 P229 T17 V19 R39 W46 E169 K170 P208 H377 K568 R569 K574 T676 K680 H337 K528 R529 K534 T633 K637 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 remove_due_to_license_issue IC50=6.0nM P06737 10980448 862 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASTVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1ent E 1.9 BS01 0EM E 1 D12 D32 Y75 G76 D77 F189 D215 G217 T218 T219 I297 D15 D35 Y79 G80 D81 F194 D219 G221 T222 T223 I300 3.4.23.22 0004190,0006508 Ki=110nM remove_due_to_license_issue P11838 2179568 822 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 1enu A 1.95 BS02 APZ A 1 Y106 D156 C158 G229 G230 M260 Y96 D146 C148 G219 G220 M250 D102 D280 C318 C320 C323 H349 D92 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=8.3uM remove_due_to_license_issue P28720 11178905 400 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1eoc B 2.25 BS02 4NC B 1 Y324 Y408 W449 R457 H460 H462 I491 Y22 Y106 W147 R155 H158 H160 I189 Y408 Y447 R457 H460 H462 Y106 Y145 R155 H158 H160 1.13.11.3 0003824,0005506,0005515,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=0.9uM remove_due_to_license_issue P20372 10891075 999 IIWGAYAQRNTEDHPPAYAPGYKTSVLRSPKNALISIAETLSEVTAPHFSADKFGPKDNDLILNYAKDGLPIGERVIVHGYVRDQFGRPVKNALVEVWQANASGRYRHPNDQYIGAMDPNFGGCGRMLTDDNGYYVFRTIKPGPYPWRNRINEWRPAHIHFSLIADGWAQRLISQFYFEGDTLIDSCPILKTIPSEQQRRALIALEDKSNFIEADSRCYRFDITLRGRRATYFENDLT 1eou A 2.1 BS02 SMS A 1 N67 Q92 H94 F130 L197 T198 T199 N65 Q90 H92 F128 L195 T196 T197 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=36nM remove_due_to_license_issue IC50=36nM, Kd=10nM, Ki=12nM P00918 11802772 301 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1epo E 2.0 BS01 2Z3 E 1 D12 D32 G34 Y75 G76 D77 F111 D215 G217 T218 T219 D15 D35 G37 Y79 G80 D81 F116 D219 G221 T222 T223 3.4.23.22 0004190,0006508 Ki=11nM remove_due_to_license_issue P11838 1304340 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 1epp E 1.9 BS01 1Z1 E 1 D12 D32 G34 Y75 G76 D77 F189 D215 G217 T218 T219 D15 D35 G37 Y79 G80 D81 F194 D219 G221 T222 T223 3.4.23.22 0004190,0006508 Ki=69nM remove_due_to_license_issue P11838 8254610 333 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 1epq E 1.9 BS01 0QF E 1 D32 Y75 G76 D77 F111 F189 D215 G217 T218 T219 I297 D35 Y79 G80 D81 F116 F194 D219 G221 T222 T223 I300 3.4.23.22 0004190,0006508 Ki=6.5nM remove_due_to_license_issue P11838 8254610 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 1erb A 1.9 BS01 ETR A 1 V61 M73 M88 Q98 C174 V60 M72 M87 Q97 C173 ? 0005501,0005576,0005615,0016918,0019841,0034632,0034633 Kd=8nM remove_due_to_license_issue P18902 8227049 184 RDCRVSSFRVKENFDKARFAGTWYAMAKKDPEGLFLQDNIVAEFSVDENGHMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIIDTDYETFAVQYSCRLLNLDGTCADSYSFVFARDPSGFSPEVQKIVRQRQEELCLARQYRLIPHNGYC 1ero A 2.1 BS01 BJP A 1 M69 S70 K73 Y105 S130 N132 E166 N170 S235 G236 A237 M44 S45 K48 Y80 S105 N107 E141 N145 S210 G211 A212 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 10820001 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTMPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1erq A 1.9 BS01 BJH A 1 M69 S70 K73 Y105 S130 N132 E166 N170 S235 G236 A237 R243 M44 S45 K48 Y80 S105 N107 E141 N145 S210 G211 A212 R218 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 10820001 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTMPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1err A 2.6 BS01 RAL A 1 L346 T347 A350 D351 E353 L354 W383 L387 F404 M421 I424 H524 L525 L40 T41 A44 D45 E47 L48 W77 L81 F98 M115 I118 H208 L209 ? remove_due_to_license_issue IC50=1.8nM, EC50=2.4nM, Ki=0.37nM P03372 9338790 600 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMPLYDLLLEMLDAH 1esz A 2.0 BS01 CPO A 1 E42 W68 R84 S103 Y106 I183 W217 W273 F274 Y275 E10 W36 R52 S71 Y74 I151 W185 W241 F242 Y243 ? 0005515,0006826,0015687,0030288,0042597,0055052,0098711,1901678 Kd=0.3uM remove_due_to_license_issue P07822 11805094 500 IDPNRIVALEWLPVELLLALGIVPYGVADTINYRLWVSEPPLPDSVIDVGLRTEPNLELLTEMKPSFMVWSAGYGPSPEMLARIAPGRGFNFSDGKQPLAMARKSLTEMADLLNLQSAAETHLAQYEDFIRSMKPRFVKRGARPLLLTTLIDPRHMLVFGPNSLFQEILDEYGIPNAWQGETNFWGSTAVSIDRLAAYKDVDVLCFDHDNSKDMDALMATPLWQAMPFVRAGRFQRVPAVWFYGATLSAMHFVRVLDNAI 1ets H 2.3 BS01 MID H 1 H57 W60D N98 L99 D189 A190 E192 S195 W215 G216 E217 G219 C220 H43 W50 N95 L96 D199 A200 E202 S205 W227 G228 E229 G230 C231 3.4.21.5 0004252,0005509,0006508,0007596 Ki=6nM remove_due_to_license_issue Ki=6nM P00735 1518046 1 IVEGQDAEVGLSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTVDDLLVRIGKHSRTRYERKVEKISMLDKIYIHPRYNWKENLDRDIALLKLKRPIELSDYIHPVCLPDKQTAAKLLHAGFKGRVTGWGNRRETWTTSVAEVQPSVLQVVNLPLVERPVCKASTRIRITDNMFCAGYKPGEGKRGDACEGDSGGPFVMKSPYNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDRLGS 1ett H 2.5 BS01 4QQ H 1 H57 Y60A W60D D189 A190 W215 G216 G219 H43 Y47 W50 D199 A200 W227 G228 G230 3.4.21.5 0004252,0005509,0006508,0007596 Ki=1.3uM remove_due_to_license_issue P00735 1518046 301 IVEGQDAEVGLSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTVDDLLVRIGKHSRTRYERKVEKISMLDKIYIHPRYNWKENLDRDIALLKLKRPIELSDYIHPVCLPDKQTAAKLLHAGFKGRVTGWGNRRETWTTSVAEVQPSVLQVVNLPLVERPVCKASTRIRITDNMFCAGYKPGEGKRGDACEGDSGGPFVMKSPYNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDRLGS 1etz H 2.6 BS01 GAS H 1 K58 Y60 R100 F102 Y104 Y111 K58 Y60 R100 F102 Y104 Y111 ? remove_due_to_license_issue P01867 10993728 229 QVTLKESGPGILQPSQTLSLTCSFSGFSLSTSGMGVGWIRQPSGEGLEWLADIWWNDKKYYNPSLKSRLTVSKDTSSNQVFLKITSVDTSDTATYHCARRTFSYYYGSSFYYFDNWGQGTTLTVSSAKTTPPSVYPLAPGCGDTTGSSVTLGCLVKGYFPESVTVTWNSGSLSSSVHTFPALLQSGLYTMSSSVTVPSSTWPSQTVTCSVAHPASSTTVDKKLEPSGP 1etz L 2.6 BS01 GAS H 1 W93 W98 W93 W98 ? remove_due_to_license_issue G0YP42 10993728 229 FAVVTQESALTTSPGETVTLTCRSSTGAVTTSNYAIWVQEKPDHLFSGLIGGTNNRVPGVPARFSGSLIGDKAALTVTGAQTEDEAIYFCALWYSNHWVFGGGTKLTVLGQPKSSPSVTLFTPSSEELETNKATLVCTITDFYPGVVTVDWKVDGTPVTQGMETTQPSKQSNNKYMASSYLTLTARAWERHSSYSCQVTHEGHTVEKSLSRAECS 1eub A -1.00 BS05 HAV A 1 L184 A186 H222 E223 H226 H232 L81 A83 H119 E120 H123 H129 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P45452 10926524 1 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDEDPN 1eub A -1.00 BS06 3MP A 1 G183 P242 G80 P139 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P45452 10926524 2 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDEDPN 1eub A -1.00 BS07 MSB A 1 L185 A186 L218 H222 F241 P242 I243 Y244 L82 A83 L115 H119 F138 P139 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P45452 10926524 3 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDEDPN 1eve A 2.5 BS01 E20 A 1 W84 Y121 E199 W279 F330 F331 H440 W83 Y120 E198 W278 F329 F330 H439 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G117 G118 G150 S199 A200 A238 F289 F291 E326 H439 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 ic50=5.7nM remove_due_to_license_issue IC50=23nM, Ki=3.3nM P04058 10368299 2001 DHSELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1evw A 3.1 BS01 dna E 0 A48 G53 K56 N57 K65 A47 G52 K55 N56 K64 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 2 ~ 13 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw A 3.1 BS02 dna O 0 R61 Q63 R74 T79 T95 A96 H98 N119 R60 Q62 R73 T78 T94 A95 H97 N118 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 13 ~ 20 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw B 3.1 BS01 dna M 0 N57 R61 Q63 R74 T79 T95 A96 S97 H98 N119 N56 R60 Q62 R73 T78 T94 A95 S96 H97 N118 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 14 ~ 21 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw B 3.1 BS02 dna F 0 G53 K56 N57 K65 G52 K55 N56 K64 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 1 ~ 12 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw C 3.1 BS01 dna G 0 A48 P49 G51 V52 G53 K56 N57 K65 R66 A47 P48 G50 V51 G52 K55 N56 K64 R65 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 2 ~ 13 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw C 3.1 BS02 dna P 0 R61 Q63 R74 T79 T95 A96 H98 N119 R60 Q62 R73 T78 T94 A95 H97 N118 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 13 ~ 20 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw D 3.1 BS01 dna N 0 N57 R61 Q63 R74 A96 S97 H98 N119 N56 R60 Q62 R73 A95 S96 H97 N118 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 14 ~ 21 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1evw D 3.1 BS02 dna H 0 P49 V52 G53 N57 K65 P48 V51 G52 N56 K64 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 10891275 1 ~ 12 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASHLCHNTRCHNPLHLCWESADDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 1ew8 A 2.2 BS06 PAE A 1 D51 D101 S102 R166 D327 H412 D51 D101 S102 R166 D327 H412 D51 S102 D153 T155 R166 E322 D327 K328 H331 D369 H370 H412 D51 S102 D153 T155 R166 E322 D327 K328 H331 D369 H370 H412 3.1.3.1 0000287,0004035,0004721,0005515,0006470,0008270,0016787,0016791,0030288,0030613,0033748,0042597,0046872 Ki=5.5mM remove_due_to_license_issue P00634 10850800 556 TPEMPVLENRAAQGDITAPGGARRLTGDQTAALRDSLSDKPAKNIILLIGDGMGDSEITAARNYAEGAGGFFKGIDALPLTGQYTHYALNKKTGKPDYVTDSAASATAWSTGVKTYNGALGVDIHEKDHPTILEMAKAAGLATGNVSTAELQDATPAALVAHVTSRKCYGPSATSEKCPGNALEKGGKGSITEQLLNARADVTLGGGAKTFAETATAGEWQGKTLREQAQARGYQLVSDAASLNSVTEANQQKPLLGLFADGNMPVRWLGPKATYHGNIDKPAVTCTPNPQRNDSVPTLAQMTDKAIELLSKNEKGFFLQVEGASIDKQDHAANPCGQIGETVDLDEAVQRALEFAKKEGNTLVIVTADHAHASQIVAPDTKAPGLTQALNTKDGAVMVMSYGNSEEDSQEHTGSQLRIAAYGPHAANVVGLTDQTDLFYTMKAALGLK 1ew9 A 2.0 BS05 MMQ A 1 S102 R166 D327 H331 H412 S102 R166 D327 H331 H412 D51 S102 D153 T155 R166 E322 D327 K328 H331 D369 H370 H412 D51 S102 D153 T155 R166 E322 D327 K328 H331 D369 H370 H412 3.1.3.1 0000287,0004035,0004721,0005515,0006470,0008270,0016787,0016791,0030288,0030613,0033748,0042597,0046872 Ki=0.6mM remove_due_to_license_issue P00634 10850800 559 TPEMPVLENRAAQGDITAPGGARRLTGDQTAALRDSLSDKPAKNIILLIGDGMGDSEITAARNYAEGAGGFFKGIDALPLTGQYTHYALNKKTGKPDYVTDSAASATAWSTGVKTYNGALGVDIHEKDHPTILEMAKAAGLATGNVSTAELQDATPAALVAHVTSRKCYGPSATSEKCPGNALEKGGKGSITEQLLNARADVTLGGGAKTFAETATAGEWQGKTLREQAQARGYQLVSDAASLNSVTEANQQKPLLGLFADGNMPVRWLGPKATYHGNIDKPAVTCTPNPQRNDSVPTLAQMTDKAIELLSKNEKGFFLQVEGASIDKQDHAANPCGQIGETVDLDEAVQRALEFAKKEGNTLVIVTADHAHASQIVAPDTKAPGLTQALNTKDGAVMVMSYGNSEEDSQEHTGSQLRIAAYGPHAANVVGLTDQTDLFYTMKAALGLK 1ew9 B 2.0 BS05 MMQ B 1 S102 R166 D327 H331 H412 S102 R166 D327 H331 H412 D51 S102 D153 T155 R166 E322 D327 K328 H331 D369 H370 H412 D51 S102 D153 T155 R166 E322 D327 K328 H331 D369 H370 H412 3.1.3.1 0000287,0004035,0004721,0005515,0006470,0008270,0016787,0016791,0030288,0030613,0033748,0042597,0046872 Ki=0.6mM remove_due_to_license_issue P00634 10850800 559 TPEMPVLENRAAQGDITAPGGARRLTGDQTAALRDSLSDKPAKNIILLIGDGMGDSEITAARNYAEGAGGFFKGIDALPLTGQYTHYALNKKTGKPDYVTDSAASATAWSTGVKTYNGALGVDIHEKDHPTILEMAKAAGLATGNVSTAELQDATPAALVAHVTSRKCYGPSATSEKCPGNALEKGGKGSITEQLLNARADVTLGGGAKTFAETATAGEWQGKTLREQAQARGYQLVSDAASLNSVTEANQQKPLLGLFADGNMPVRWLGPKATYHGNIDKPAVTCTPNPQRNDSVPTLAQMTDKAIELLSKNEKGFFLQVEGASIDKQDHAANPCGQIGETVDLDEAVQRALEFAKKEGNTLVIVTADHAHASQIVAPDTKAPGLTQALNTKDGAVMVMSYGNSEEDSQEHTGSQLRIAAYGPHAANVVGLTDQTDLFYTMKAALGLK 1ewj A 2.5 BS01 BLM A 1 L56 A57 S58 W59 R65 S86 G87 R90 W99 G111 L113 R115 N119 L55 A56 S57 W58 R64 S85 G86 R89 W98 G110 L112 R114 N118 ? 0046677 remove_due_to_license_issue P13081 11134052 1001 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj A 2.5 BS02 BLM B 1 F30 W35 I37 F29 W34 I36 ? 0046677 remove_due_to_license_issue P13081 11134052 1002 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj B 2.5 BS01 BLM A 1 F30 W35 F29 W34 ? 0046677 remove_due_to_license_issue P13081 11134052 1001 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj B 2.5 BS02 BLM B 1 L56 A57 S58 W59 S61 R65 G87 R90 W99 G111 R115 N119 L55 A56 S57 W58 S60 R64 G86 R89 W98 G110 R114 N118 ? 0046677 remove_due_to_license_issue P13081 11134052 1002 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ex8 A 1.85 BS01 A4P A 1 T42 P43 L45 Y53 N55 Q74 R82 R84 R88 W89 R92 D97 I98 R110 L111 T112 H115 F123 T42 P43 L45 Y53 N55 Q74 R82 R84 R88 W89 R92 D97 I98 R110 L111 T112 H115 F123 R82 R92 D95 D97 R82 R92 D95 D97 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=0.47uM remove_due_to_license_issue P26281 11311059 171 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 1exd A 2.7 BS01 rna B 0 E34 D66 T68 N69 P126 R130 R133 L136 T137 G168 P181 F182 I183 V189 R192 K194 M210 Y211 F233 Q234 D235 I313 T316 K317 Q318 D319 N320 T321 E323 A325 S326 S329 N336 R341 P369 Q399 K401 R402 R410 R412 N413 V455 Q517 E519 R520 L544 R545 E27 D59 T61 N62 P119 R123 R126 L129 T130 G161 P174 F175 I176 V182 R185 K187 M203 Y204 F226 Q227 D228 I306 T309 K310 Q311 D312 N313 T314 E316 A318 S319 S322 N329 R334 P362 Q392 K394 R395 R403 R405 N406 V437 Q499 E501 R502 L526 R527 E34 R260 K270 E27 R253 K263 6.1.1.18 0000166,0004812,0004819,0005524,0005737,0005829,0006412,0006418,0006424,0006425,0043039 remove_due_to_license_issue P00962 10881199 902 ~ 976 TNFIRQIIDEDLASGKHTTVHTRFPPEPNGYLHIGHAKSICLNFGIAQDYKGQCNLRFDDTNPVKEDIEYVESIKNDVEWLGFHWSGNVRYSSDYFDQLHAYAIELINKGLAYVDELTPEQIREYRGTLTQPGKNSPYRDRSVEENLALFEKMRAGGFEEGKACLRAKIDMASPFIVMRDPVLYRIKFAEHHQTGNKWCIYPMYDFTHCISDALEGITHSLCTLEFQDNRRLYDWVLDNITIPVHPRQYEFSRLNLEYTVMSKRKLNLLVTDKHVEGWDDPRMPTISGLRRRGYTAASIREFCKRIGVTKQDNTIEMASLESCIREDLNENAPRAMAVIDPVKLVIENYQGEGEMVTMPNHPNKPEMGSRQVPFSGEIWIDRADFREEANKQYKRLVLGKEVRLRNAYVIKAERVEKDAEGNITTIFCTYDADTLGVIHWVSAAHALPVEIRLYDRLFSVPNPGAADDFLSVINPESLVIKQGFAEPSLKDAVAGKAFQFEREGYFCLDSRHSTAEKPVFNRTVGLRDT 1exv A 2.4 BS03 700 A 1 R60 W67 P188 E190 K191 R38 W45 P166 E168 K169 H377 K568 R569 K574 T676 K680 H333 K524 R525 K530 T632 K636 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 ic50=45nM remove_due_to_license_issue IC50=45nM P06737 10980448 862 NVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKAFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1exv A 2.4 BS04 700 B 1 T38 V40 F53 H57 P188 T16 V18 F31 H35 P166 H377 K568 R569 K574 T676 K680 H333 K524 R525 K530 T632 K636 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 ic50=45nM remove_due_to_license_issue IC50=45nM P06737 10980448 1862 NVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKAFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1exv B 2.4 BS01 700 A 1 T38 V40 F53 H57 P188 T16 V18 F31 H35 P166 H377 K568 R569 K574 T676 K680 H333 K524 R525 K530 T632 K636 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 ic50=45nM remove_due_to_license_issue IC50=45nM P06737 10980448 862 NVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKAFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1exv B 2.4 BS04 700 B 1 R60 W67 P188 E190 K191 P229 R38 W45 P166 E168 K169 P207 H377 K568 R569 K574 T676 K680 H333 K524 R525 K530 T632 K636 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 ic50=45nM remove_due_to_license_issue IC50=45nM P06737 10980448 1862 NVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKAFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1exw A 2.4 BS01 HDS A 1 M41 S115 Q116 Q142 A171 W186 M14 S88 Q89 Q115 A144 W159 M41 S115 Q116 D233 H289 E294 M14 S88 Q89 D206 H262 E267 3.1.2.22 0002084,0005576,0005634,0005764,0005794,0005829,0006897,0006898,0006907,0007042,0007399,0007420,0008021,0008474,0015031,0016042,0016787,0030308,0030424,0031579,0043066,0043524,0045121,0048260,0048549,0052816,0098599,0120146 remove_due_to_license_issue P45478 10801859 430 DPPAPLPLVIWHGMGDSCCNPLSMGAIKKMVEKKIPGIHVLSLEIGKTLREDVENSFFLNVNSQVTTVCQILAKDPKLQQGYNAMGFSQGGQFLRAVAQRCPSPPMVNLISVGGQHQGVFGLPRCPGESSHICDFIRKTLNAGAYNKAIQERLVQAEYWHDPIREDIYRNHSIFLADINQERGVNESYKKNLMALKKFVMVKFLNDTIVDPVDSEWFGFYRSGQAKETIPLQESTLYTQDRLGLKAMDKAGQLVFLALEGDHLQLSEEWFYAHIIPFLE 1ez9 A 1.9 BS01 GLC C 1 E111 Y155 W230 E111 Y155 W230 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9 11790091 2 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTRITK 1ez9 A 1.9 BS02 GLC C 2 D65 E153 P154 Y155 W340 D65 E153 P154 Y155 W340 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9 11790091 3 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTRITK 1ez9 A 1.9 BS03 GLC C 3 E153 W340 Y341 R344 E153 W340 Y341 R344 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9 11790091 4 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTRITK 1ezf A 2.15 BS01 IN0 A 1 R52 F54 Y73 G180 L183 G208 L211 P292 R15 F17 Y36 G143 L146 G171 L174 P255 Y171 R218 R228 F288 Y134 R181 R191 F251 2.5.1.21 0008610,0009058,0016765,0045338,0051996 remove_due_to_license_issue P37268 10896663 991 NSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVKIDATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQN 1ezq A 2.2 BS02 RPR A 1 E97 Y99 E147 F174 D189 A190 C191 Q192 S195 W215 G216 E217 G219 C220 E83 Y85 E135 F162 D179 A180 C181 Q182 S185 W205 G206 E207 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.9nM remove_due_to_license_issue Ki=0.9nM P00742 10966741 265 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1f0q A 2.63 BS01 EMO A 1 V53 K68 F113 M163 I174 D175 V48 K63 F108 M158 I169 D170 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue Ki=1850nM P28523 10882732 400 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENSR 1f0r A 2.1 BS02 815 A 1 Y99 F174 S195 V213 W215 G216 E217 G219 C220 Y85 F162 S185 V203 W205 G206 E207 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=22nM remove_due_to_license_issue Ki=22nM P00742 10966741 401 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1f0s A 2.1 BS02 PR2 A 1 Y99 F174 C191 Q192 W215 G216 E217 G219 C220 Y85 F162 C181 Q182 W205 G206 E207 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=18nM remove_due_to_license_issue Ki=18nM P00742 10966741 401 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1f0t A 1.8 BS02 PR1 A 1 T98 L99 D189 S190 C191 Q192 W215 G216 G219 T80 L81 D171 S172 C173 Q174 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Ki=1000nM remove_due_to_license_issue Ki=1000nM P00760 10966741 304 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1f0u A 1.9 BS02 RPR A 1 N97 D189 S190 C191 Q192 W215 G216 G219 C220 N79 D171 S172 C173 Q174 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Ki=69nM remove_due_to_license_issue Ki=69nM P00760 10966741 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1f28 A 1.9 BS02 F89 A 1 F58 G61 E65 H85 I86 W87 D202 G206 F209 S296 F56 G59 E63 H83 I84 W85 D200 G204 F207 S294 E65 W87 Y113 C173 R199 D202 E63 W85 Y111 C171 R197 D200 2.1.1.45 0004633,0004799,0004864,0005739,0005829,0006231,0006235,0008168,0009165,0010181,0016741,0032259,0034399 Ki=16nM remove_due_to_license_issue P13100 11358692 401 NAEEQQYLNLVQYIINHGEDRPDRTGTGTLSVFAPSPLKFSLRNKTFPLLTTKRVFIRGVIEELLWFIRGETDSLKLREKNIHIWDANGSREYLDSIGLTKRQEGDLGPIYGFQWRHFGAEYIDCKTNYIGQGVDQLANIIQKIRTSPYDRRLILSAWNPADLEKMALPPCHMFCQFYVHIPSNNHRPELSCQLYQRSCDMGLGVPFNIASYALLTCMIAHVCDLDPGDFIHVMGDCHIYKDHIEALQQQLTRSPRPFPTLSLNRSITDIEDFTLDDFNIQNYHPYETIKMKMSI 1f28 B 1.9 BS03 F89 B 1 F58 E65 I86 W87 D202 G206 F209 Y242 M295 F56 E63 I84 W85 D200 G204 F207 Y240 M293 E65 W87 Y113 C173 R199 D202 E63 W85 Y111 C171 R197 D200 2.1.1.45 0004633,0004799,0004864,0005739,0005829,0006231,0006235,0008168,0009165,0010181,0016741,0032259,0034399 Ki=16nM remove_due_to_license_issue P13100 11358692 402 NAEEQQYLNLVQYIINHGEDRPDRTGTGTLSVFAPSPLKFSLRNKTFPLLTTKRVFIRGVIEELLWFIRGETDSLKLREKNIHIWDANGSREYLDSIGLTKRQEGDLGPIYGFQWRHFGAEYIDCKTNYIGQGVDQLANIIQKIRTSPYDRRLILSAWNPADLEKMALPPCHMFCQFYVHIPSNNHRPELSCQLYQRSCDMGLGVPFNIASYALLTCMIAHVCDLDPGDFIHVMGDCHIYKDHIEALQQQLTRSPRPFPTLSLNRSITDIEDFTLDDFNIQNYHPYETIKMKMSI 1f2o A 1.7 BS04 LEU A 1 D97 E131 E132 D160 R202 Y246 H247 D97 E131 E132 D160 R202 Y246 H247 N77 D97 E131 E132 D160 N77 D97 E131 E132 D160 3.4.11.24 0004177,0006508,0008235 Ki=12.4mM remove_due_to_license_issue P80561 11484227 903 APDIPLANVKAHLTQLSTIAANNGGNRAHGRPGYKASVDYVKAKLDAAGYTTTLQQFTSGGATGYNLIANWPGGDPNKVLMAGAHLDSVSSGAGINDNGSGSAAVLETALAVSRAGYQPDKHLRFAWWGAEELGLIGSKFYVNNLPSADRSKLAGYLNFDMIGSPNPGYFVYDDDPVIEKTFKNYFAGLNVPTEIETEGDGRSDHAPFKNVGVPVGGLFTGAGYTKSAAQAQKWGGTAGQAFDRCYHSSCDSLSNINDTALDRNSDAAAHAIWTLSS 1f2p A 1.8 BS04 PHE A 1 E131 E132 D160 R202 F219 Y246 E131 E132 D160 R199 F216 Y243 N77 D97 E131 E132 D160 N77 D97 E131 E132 D160 3.4.11.24 0004177,0006508,0008235 Ki=12.7mM remove_due_to_license_issue P80561 11484227 903 APDIPLANVKAHLTQLSTIAANNGGNRAHGRPGYKASVDYVKAKLDAAGYTTTLQQFTSGGATGYNLIANWPGGDPNKVLMAGAHLDSVSSGAGINDNGSGSAAVLETALAVSRAGYQPDKHLRFAWWGAEELGLIGSKFYVNNLPSADRSKLAGYLNFDMIGSPNPGYFVYDDDPVIEKTFKNYFAGLNVPTEIETERSDHAPFKNVGVPVGGLFTGAGYTKSAAQAQKWGGTAGQAFDRCYHSSCDSLSNINDTALDRNSDAAAHAIWTLSS 1f3e A 1.85 BS02 DPZ A 1 Y106 D156 C158 Q203 G229 G230 M260 Y96 D146 C148 Q193 G219 G220 M250 D102 D280 C318 C320 C323 H349 D92 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=0.2uM remove_due_to_license_issue P28720 11178905 400 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1f40 A -1.00 BS01 GPI A 1 Y26 F46 V55 I56 Y82 H87 Y26 F46 V55 I56 Y82 H87 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 remove_due_to_license_issue Ki=7.5nM, IC50=1240nM P62942 10951192 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1f4e A 1.9 BS01 TPR A 1 W80 Y94 H147 F176 W80 Y94 H147 F176 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.1mM remove_due_to_license_issue P0A884 10944209 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1f4e A 1.9 BS02 TPR A 2 Q64 G65 D66 Q64 G65 D66 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.1mM remove_due_to_license_issue P0A884 10944209 302 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1f4f A 2.0 BS01 TP3 A 1 I79 W80 L143 L172 F176 I79 W80 L143 L172 F176 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=24uM remove_due_to_license_issue P0A884 10944209 701 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPV 1f4f B 2.0 BS01 TP3 B 1 S54 W80 L143 C146 L172 F176 S54 W80 L143 C146 L172 F176 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=24uM remove_due_to_license_issue P0A884 10944209 702 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAP 1f4g A 1.75 BS01 TP4 A 1 S54 I79 W80 L143 C146 S167 D169 L172 F176 H207 Y209 S54 I79 W80 L143 C146 S167 D169 L172 F176 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=330nM remove_due_to_license_issue P0A884 10944209 601 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPV 1f4g B 1.75 BS01 TP4 B 1 S54 I79 W80 L143 C146 S167 D169 L172 F176 H207 Y209 S54 I79 W80 L143 C146 S167 D169 L172 F176 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=330nM remove_due_to_license_issue P0A884 10944209 602 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAP 1f4k A 2.5 BS01 dna D 0 K14 Q15 R16 N53 T55 R59 K7 Q8 R9 N46 T48 R52 ? 0003677,0006274 remove_due_to_license_issue P0CI76 11224562 1 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 1f4k A 2.5 BS02 dna E 0 T9 Y33 G34 L35 H54 Y58 H62 Q83 T2 Y26 G27 L28 H47 Y51 H55 Q76 ? 0003677,0006274 remove_due_to_license_issue P0CI76 11224562 1 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 1f4k B 2.5 BS01 dna D 0 T9 Y33 G34 L35 H54 Y58 H62 Q72 V85 T2 Y26 G27 L28 H47 Y51 H55 Q65 V78 ? 0003677,0006274 remove_due_to_license_issue P0CI76 11224562 1 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 1f4k B 2.5 BS02 dna E 0 K14 Q15 R16 N53 T55 R59 E84 K7 Q8 R9 N46 T48 R52 E77 ? 0003677,0006274 remove_due_to_license_issue P0CI76 11224562 1 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 1f4x H 2.3 BS01 MGS H 1 T31 Y32 D33 H99 Y101 A102 T31 Y32 D33 H99 Y101 A102 Kd=2.6uM remove_due_to_license_issue 10880560 301 EVQLEESGGGLVTPGGSLRLSCAASGYVFSTYDMSWVRQTPEKRLEWVAFISSGGGRTSYPDTVKGRFTISRDDAKNTLYLQMSSLQSEDTAMYYCTRHFYAVLDYWGRGTTLTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVP 1f57 A 1.75 BS02 DCY A 1 H69 R127 R145 H196 E270 H69 R127 R145 H196 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=2.3uM remove_due_to_license_issue Ki=2300nM P00730 10955996 308 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 1f5l A 2.1 BS01 AMR A 1 D189 S190 Q192 S195 G219 G226 D192 S193 Q195 S198 G221 G229 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=5.3uM remove_due_to_license_issue IC50=7000nM, Ki=7000nM P00749 10926521 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1f5t A 3.0 BS01 dna E 0 R1027 A1028 R1029 S1042 R1060 R26 A27 R28 S41 R59 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 295 ~ 337 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t A 3.0 BS02 dna F 0 K1002 T1007 Q1036 S1037 P1039 T1040 Q1043 R1047 R1050 K1 T6 Q35 S36 P38 T39 Q42 R46 R49 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 396 ~ 438 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t B 3.0 BS01 dna E 0 T2007 Q2036 S2037 P2039 T2040 Q2043 R2047 R2050 T6 Q35 S36 P38 T39 Q42 R46 R49 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 295 ~ 337 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t B 3.0 BS02 dna F 0 K2002 R2027 A2028 R2029 S2042 R2060 K1 R26 A27 R28 S41 R59 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 396 ~ 438 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t C 3.0 BS01 dna E 0 T3007 Q3036 S3037 P3039 T3040 Q3043 R3047 R3050 T6 Q35 S36 P38 T39 Q42 R46 R49 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 295 ~ 337 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t C 3.0 BS02 dna F 0 R3027 A3028 R3029 S3042 R26 A27 R28 S41 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 396 ~ 438 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t D 3.0 BS01 dna E 0 R4027 A4028 S4042 R4060 R26 A27 S41 R59 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 295 ~ 337 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f5t D 3.0 BS02 dna F 0 K4002 T4007 Q4036 S4037 P4039 T4040 Q4043 R4047 R4050 K1 T6 Q35 S36 P38 T39 Q42 R46 R49 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P0DJL7 10956029 396 ~ 438 KDLVDTTEMYLRTIYELEEEGVTPLRARIAERLEQSGPTVSQTVARMERDGLVVVASDRSLQMTPTGRTLATAVMRKHRLAERLLTDIIGLDINKVHDEADRWEHVMSDEVERRLVKVLK 1f6u A -1.00 BS01 rna B 0 K3 Q9 K14 F16 I24 A25 K26 N27 R32 G35 C36 W37 Q45 M46 K3 Q9 K14 F16 I24 A25 K26 N27 R32 G35 C36 W37 Q45 M46 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0008270 remove_due_to_license_issue P35963 10926523 201 ~ 219 MQKGNFRNQRKTVKCFNCGKEGHIAKNCRAPRKKGCWKCGKEGHQMKDCTERQAN 1f73 A 1.95 BS01 HMN A 1 A10 G46 S47 T48 K164 G188 D190 E191 G206 S207 A10 G46 S47 T48 K159 G183 D185 E186 G201 S202 S47 Y110 Y136 K164 I205 S47 Y110 Y136 K159 I200 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262 Ki=4.1mM remove_due_to_license_issue P44539 11031117 700 MRDLKGIFSALLVSFNEDGTINEKGLRQIIRHNIDKMKVDGLYVGGSTGENFMLSTEEKKEIFRIAKDEAKDQIALIAQVGSVNLKEAVELGKYATELGYDCLSAVTPFYYKFSFPEIKHYYDTIIAETGSNMIVYSIPNMGIEQFGELYKNPKVLGVKFTAGDFYLLERLKKAYPNHLIWAGFDEMMLPAASLGVDGAIGSTFNVNGVRARQIFELTKAGKLKEALEIQHVTNDLIEGILANGLYLTIKELLKLEGVDAGYCREPMTSKATAEQVAKAKDLKAKFLS 1f73 C 1.95 BS01 HMN C 1 A10 G46 S47 T48 K164 G188 D190 E191 G206 S207 L250 A10 G46 S47 T48 K159 G183 D185 E186 G201 S202 L245 S47 Y110 Y136 K164 I205 S47 Y110 Y136 K159 I200 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262 Ki=4.1mM remove_due_to_license_issue P44539 11031117 702 MRDLKGIFSALLVSFNEDGTINEKGLRQIIRHNIDKMKVDGLYVGGSTGENFMLSTEEKKEIFRIAKDEAKDQIALIAQVGSVNLKEAVELGKYATELGYDCLSAVTPFYYKFSFPEIKHYYDTIIAETGSNMIVYSIPNMGIEQFGELYKNPKVLGVKFTAGDFYLLERLKKAYPNHLIWAGFDEMMLPAASLGVDGAIGSTFNVNGVRARQIFELTKAGKLKEALEIQHVTNDLIEGILANGLYLTIKELLKLEGVDAGYCREPMTSKATAEQVAKAKDLKAKFLS 1f73 D 1.95 BS01 HMN D 1 A10 G46 S47 T48 K164 G188 D190 E191 G206 S207 A10 G46 S47 T48 K159 G183 D185 E186 G201 S202 S47 Y110 Y136 K164 I205 S47 Y110 Y136 K159 I200 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262 Ki=4.1mM remove_due_to_license_issue P44539 11031117 703 MRDLKGIFSALLVSFNEDGTINEKGLRQIIRHNIDKMKVDGLYVGGSTGENFMLSTEEKKEIFRIAKDEAKDQIALIAQVGSVNLKEAVELGKYATELGYDCLSAVTPFYYKFSFPEIKHYYDTIIAETGSNMIVYSIPNMGIEQFGELYKNPKVLGVKFTAGDFYLLERLKKAYPNHLIWAGFDEMMLPAASLGVDGAIGSTFNVNGVRARQIFELTKAGKLKEALEIQHVTNDLIEGILANGLYLTIKELLKLEGVDAGYCREPMTSKATAEQVAKAKDLKAKFLS 1f74 A 1.6 BS01 NAY A 1 A10 S47 T48 K164 F189 D190 E191 G206 S207 A10 S47 T48 K164 F189 D190 E191 G206 S207 S47 Y110 Y136 L141 K164 I205 S47 Y110 Y136 L141 K164 I205 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262 Ki=0.9mM remove_due_to_license_issue P44539 11031117 950 MRDLKGIFSALLVSFNEDGTINEKGLRQIIRHNIDKMKVDGLYVGGSTGENFMLSTEEKKEIFRIAKDEAKDQIALIAQVGSVNLKEAVELGKYATELGYDCLSAVTPFYYKFSFPEIKHYYDTIIAETGSNMIVYSIPFLTGVNMGIEQFGELYKNPKVLGVKFTAGDFYLLERLKKAYPNHLIWAGFDEMMLPAASLGVDGAIGSTFNVNGVRARQIFELTKAGKLKEALEIQHVTNDLIEGILANGLYLTIKELLKLEGVDAGYCREPMTSKATAEQVAKAKDLKAKFLS 1f74 C 1.6 BS01 NAY C 1 A10 S47 T48 K164 G188 F189 D190 E191 I205 G206 S207 A10 S47 T48 K164 G188 F189 D190 E191 I205 G206 S207 S47 Y110 L141 S47 Y110 L141 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262 Ki=0.9mM remove_due_to_license_issue P44539 11031117 951 MRDLKGIFSALLVSFNEDGTINEKGLRQIIRHNIDKMKVDGLYVGGSTGENFMLSTEEKKEIFRIAKDEAKDQIALIAQVGSVNLKEAVELGKYATELGYDCLSAVTPFYYKFSFPEIKHYYDTIIAETGSNMIVYSIPFLTGVNMGIEQFGELYKNPKVLGVKFTAGDFYLLERLKKAYPNHLIWAGFDEMMLPAASLGVDGAIGSTFNVNGVRARQIFELTKAGKLKEALEIQHVTNDLIEGILANGLYLTIKELLKLEGVDAGYCREPMTSKATAEQVAKAKDLKAKFLS 1f7b C 1.8 BS01 NAV C 1 Y43 G46 S47 T48 K164 G188 F189 D190 E191 G206 S207 L250 Y43 G46 S47 T48 K156 G180 F181 D182 E183 G198 S199 L242 S47 Y110 S47 Y110 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262 remove_due_to_license_issue P44539 11031117 902 MRDLKGIFSALLVSFNEDGTINEKGLRQIIRHNIDKMKVDGLYVGGSTGENFMLSTEEKKEIFRIAKDEAKDQIALIAQVGSVNLKEAVELGKYATELGYDCLSAVTPFYYKFSFPEIKHYYDTIIAETGSNMIVYSMGIEQFGELYKNPKVLGVKFTAGDFYLLERLKKAYPNHLIWAGFDEMMLPAASLGVDGAIGSTFNVNGVRARQIFELTKAGKLKEALEIQHVTNDLIEGILANGLYLTIKELLKLEGVDAGYCREPMTSKATAEQVAKAKDLKAKFLS 1f8b A 1.8 BS02 DAN A 1 R118 E119 D151 R152 W178 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W98 A166 E196 R212 R290 Y324 D151 E277 R292 R371 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=4uM remove_due_to_license_issue IC50=13000nM P03472 11274459 0 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1f8c A 1.7 BS02 4AM A 1 R118 E119 D151 R152 W178 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W98 A166 E196 R212 R290 Y324 D151 E277 R292 R371 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=0.04uM remove_due_to_license_issue P03472 11274459 4 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1f8d A 1.4 BS02 9AM A 1 R118 E119 D151 R152 W178 E276 R292 R371 Y406 R37 E38 D70 R71 W98 E196 R212 R290 Y324 D151 E277 R292 R371 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=400uM remove_due_to_license_issue P03472 11274459 0 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1f8e A 1.4 BS02 49A A 1 R118 E119 D151 R152 W178 E276 R292 R371 Y406 R37 E38 D70 R71 W98 E196 R212 R290 Y324 D151 E277 R292 R371 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=15uM remove_due_to_license_issue P03472 11274459 0 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1f92 A 2.6 BS01 UKP A 1 H57 L97B H99 D189 S190 C191 Q192 V213 W215 G216 G219 H46 L92 H94 D192 S193 C194 Q195 V216 W218 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue Ki=640nM P00749 10926521 300 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1f9g A 2.0 BS01 ASC A 1 W292 R462 W123 R293 N349 H399 Y408 R462 E577 N180 H230 Y239 R293 E408 4.2.2.1 0003824,0005576,0005975,0016829,0030246 Ki=53mM remove_due_to_license_issue Q54873 11278838 950 VKDTYTDRLDDWNGIIAGNQYYDSKNDQMAKLNQELEGKVADSLSSISSQADRIYLWEKFSNYKTSANLTATYRKLEEMAKQVTNPSSRYYQDETVVRTVRDSMEWMHKHVYNSEKSIVGNWWDYEIGTPRAINNTLSLMKEYFSDEEIKKYTDVIEKFVPDPEHFRKTTDNPFKALGGNLVDMGRVKVIAGLLRKDDQEISSTIRSIEQVFKLVDQGEGFYQDGSYIDHTNVAYTGAYGNVLIDGLSQLLPVIQKTKNPIDKDKMQTMYHWIDKSFAPLLVNGELMDMSRGRSISRANSEGHVAAVEVLRGIHRIADMSEGETKQRLQSLVKTIVQSDSYYDVFKNLKTYKDISLMQSLLSDAGVASVPRTSYLSAFNKMDKTAMYNAEKGFGFGLSLFSSRTLNYEHMNKENKRGWYTSDGMFYLYNGDLSHYSDGYWPTVNPYKMPGTTETDAKRADSDTGKVLPSAFVGTSKLDDANATATMDFTNWNQTLTAHKSWFMLKDKIAFLGSNIQNTSTDTAATTIDQRKLESSNPYKVYVNDKEASLTEQEKDYPETQSVFLESSDSKKNIGYFFFKKSSISMSKALQKGAWKDINEGQSDKEVENEFLTISQAHKQNGDSYGYMLIPNVDRATFNQMIKELESSLIENNETLQSVYDAKQGVWGIVKYDDSVSTISNQFQVLKRGVYTIRKEGDEYKIAYYNPETQESAPDQEVFKKL 1fao A 1.8 BS01 4IP A 1 K173 G175 G176 L177 V178 T180 R184 Y195 I205 R235 K12 G14 G15 L16 V17 T19 R23 Y34 I44 R74 ? Kd=0.043uM remove_due_to_license_issue Q9UN19 10983984 274 PSLGTKEGYLTKQGGLVKTWKTRWFTLHRNELKYFKDQMSPEPIRILDLTECSAVQFDYSQERVNCFCLVFPFRTFYLCAKTGVEADEWIKILRWKLSQI 1fax A 3.0 BS02 DX9 A 1 E97 D189 A190 C191 Q192 W215 G216 G218 E83 D179 A180 C181 Q182 W205 G206 G208 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=41nM, IC50=70nM P00742 8939944 265 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTAAEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTR 1fbm A 2.7 BS01 RTL B 1 L44 L51 L18 L25 ? remove_due_to_license_issue P35444 9736606 951 MDLAPQMLRELQETNAALQDVRELLRQQVKEITFLKNTVMECDACG 1fbm B 2.7 BS01 RTL B 1 L44 L51 L18 L25 ? remove_due_to_license_issue P35444 9736606 951 MDLAPQMLRELQETNAALQDVRELLRQQVKEITFLKNTVMECDACG 1fbm D 2.7 BS01 RTL B 1 L44 L51 L18 L25 ? remove_due_to_license_issue P35444 9736606 951 MDLAPQMLRELQETNAALQDVRELLRQQVKEITFLKNTVMECDACG 1fbm E 2.7 BS01 RTL B 1 L44 V47 L51 L18 V21 L25 ? remove_due_to_license_issue P35444 9736606 951 MDLAPQMLRELQETNAALQDVRELLRQQVKEITFLKNTVMECDACG 1fcx A 1.47 BS01 184 A 1 F230 A234 C237 L271 M272 I275 F288 S289 G303 F304 F48 A52 C55 L89 M90 I93 F106 S107 G121 F122 ? 0003677,0004879,0005634,0006355,0048384 Kd=64nM remove_due_to_license_issue Kd=64nM P13631 10964567 450 SPQLEELITKVSKAHQETFPSLCQLGKYTTNSSADHRVQLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLSIADQITLLKAACLDILMLRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFAFAGQLLPLEMDDTETGLLSAICLICGDRMDLEEPEKVDKLQEPLLEALRLYARRRRPSQPYMFPRMLMKITDLRGISTKGAERAITLKMEIPGPMPPLIREMLE 1fcy A 1.3 BS01 564 A 1 W227 F230 A234 C237 L271 M272 I275 F288 S289 G303 F304 G393 W46 F49 A53 C56 L90 M91 I94 F107 S108 G122 F123 G212 ? 0003677,0004879,0005634,0006355,0048384 Kd=3nM remove_due_to_license_issue Kd=3nM P13631 10964567 450 ASPQLEELITKVSKAHQETFPSLCQLGKYTTNSSADHRVQLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLSIADQITLLKAACLDILMLRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFAFAGQLLPLEMDDTETGLLSAICLICGDRMDLEEPEKVDKLQEPLLEALRLYARRRRPSQPYMFPRMLMKITDLRGISTKGAERAITLKMEIPGPMPPLIREMLE 1fcz A 1.38 BS01 156 A 1 F230 A234 C237 L268 L271 M272 I275 F288 S289 F304 F48 A52 C55 L86 L89 M90 I93 F106 S107 F122 ? 0003677,0004879,0005634,0006355,0048384 Kd=0.6nM remove_due_to_license_issue P13631 10964567 450 SPQLEELITKVSKAHQETFPSLCQLGKYTTNSSADHRVQLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLSIADQITLLKAACLDILMLRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFAFAGQLLPLEMDDTETGLLSAICLICGDRMDLEEPEKVDKLQEPLLEALRLYARRRRPSQPYMFPRMLMKITDLRGISTKGAERAITLKMEIPGPMPPLIREMLE 1fd0 A 1.38 BS01 254 A 1 F230 A234 C237 L271 M272 I275 F288 S289 G303 F304 I412 F48 A52 C55 L89 M90 I93 F106 S107 G121 F122 I230 ? 0003677,0004879,0005634,0006355,0048384 Kd~4nM remove_due_to_license_issue P13631 12220491 450 SPQLEELITKVSKAHQETFPSLCQLGKYTTNSSADHRVQLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLSIADQITLLKAACLDILMLRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFAFAGQLLPLEMDDTETGLLSAICLICGDRMDLEEPEKVDKLQEPLLEALRLYARRRRPSQPYMFPRMLMKITDLRGISTKGAERAITLKMEIPGPMPPLIREMLE 1fd7 D 1.8 BS01 AI1 D 1 Y12 E51 Q56 H57 Q61 W88 N90 K91 Y12 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=14mM remove_due_to_license_issue P32890 11173465 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1fd7 E 1.8 BS01 AI1 E 1 E11 Y12 E51 Q56 H57 Q61 W88 N90 K91 E11 Y12 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=14mM remove_due_to_license_issue P32890 11173465 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1fdq A 2.1 BS01 HXA A 1 V40 T60 E72 T74 A75 D76 M115 R126 Y128 V40 T60 E72 T74 A75 D76 M115 R126 Y128 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 Kd=53.4nM remove_due_to_license_issue O15540 10854433 133 VEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA 1fe3 A 2.8 BS01 OLA A 1 G33 K58 D76 Y128 G33 K58 D76 Y128 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 remove_due_to_license_issue O15540 10854433 133 VEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA 1fgi A 2.5 BS01 SU1 A 1 G485 F489 A512 E562 Y563 A564 G567 L630 G22 F26 A45 E95 Y96 A97 G100 L151 D623 A625 R627 N628 D641 D144 A146 R148 N149 D162 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue IC50=30nM P11362 9139660 1001 ELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS 1fh7 A 1.82 BS01 XYP A 1 E43 N44 K47 Q87 W273 W281 E43 N44 K47 Q87 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 601 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fh7 A 1.82 BS02 XDN A 1 K47 H80 W84 N126 Q203 E233 W273 W281 K47 H80 W84 N126 Q203 E233 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 602 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fh8 A 1.95 BS01 XYP A 1 E43 N44 K47 Q87 W273 W281 E43 N44 K47 Q87 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 601 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fh8 A 1.95 BS02 XIF A 1 K47 H80 W84 E127 Q203 E233 W273 W281 K47 H80 W84 E127 Q203 E233 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 602 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fh9 A 1.72 BS01 LOX B 1 K47 H80 W84 E127 Q203 H205 E233 W273 W281 K47 H80 W84 E127 Q203 H205 E233 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 1 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fh9 A 1.72 BS02 XYP B 1 E43 N44 K47 Q87 W273 W281 E43 N44 K47 Q87 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 2 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fhd A 1.9 BS01 XYP A 1 E43 N44 K47 Q87 W273 E43 N44 K47 Q87 W273 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 601 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fhd A 1.9 BS02 XIM A 1 K47 H80 W84 E127 Q203 H205 E233 W273 W281 K47 H80 W84 E127 Q203 H205 E233 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 remove_due_to_license_issue P07986 10995222 602 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1fig H 3.0 BS01 TSA H 1 N33 R94 R95 Y100 F100B N33 R98 R99 Y104 F106 remove_due_to_license_issue 8303271 224 DVQLQQSGPELEKPGASVKISCKASGFSLPGHNINWIVQRNGKSLEWIGNIDPYYGGTNFNPKFKGKATLTVDKSSSTLYMHLTSLQSEDSAVYYCARRRDGNYGFTYWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKI 1fj4 A 2.35 BS01 TLM A 1 C163 F229 V270 A271 P272 H298 T300 H333 F390 G391 F392 G394 C162 F228 V269 A270 P271 H297 T299 H332 F389 G390 F391 G393 C163 H298 E309 K328 H333 F390 F392 C162 H297 E308 K327 H332 F389 F391 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 Kd=26uM remove_due_to_license_issue IC50=12000nM P0A953 11050088 500 KRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 1fj4 B 2.35 BS01 TLM B 1 C163 F229 V270 A271 H298 T300 H333 F390 G391 F392 G394 C162 F228 V269 A270 H297 T299 H332 F389 G390 F391 G393 C163 H298 E309 K328 H333 F390 F392 C162 H297 E308 K327 H332 F389 F391 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 Kd=26uM remove_due_to_license_issue IC50=12000nM P0A953 11050088 501 KRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 1fje B -1.00 BS01 rna A 0 F17 V27 R49 T52 R54 F56 Y58 K89 G90 S93 K94 K95 L103 K105 R127 L128 V129 I138 Y140 F17 V27 R49 T52 R54 F56 Y58 K89 G90 S93 K94 K95 L103 K105 R127 L128 V129 I138 Y140 ? 0003676,0003723 remove_due_to_license_issue P08199 11118222 1 ~ 22 GSHMVEGSESTTPFNLFIGNLNPNKSVAELKVAISELFAKNDLAVVDVRTGTNRKFGYVDFESAEDLEKALELTGLKVFGNEIKLEKPKGRDSKKVRAARTLLAKNLSFNITEDELKEVFEDALEIRLVSQDGKSKGIAYIEFKSEADAEKNLEEKQGAEIDGRSVSLYYTGEKG 1fjs A 1.92 BS02 Z34 A 1 E97 T98 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G218 C220 E83 T84 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.11nM remove_due_to_license_issue Ki=0.11nM P00742 11027132 500 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1fjx A 2.26 BS01 dna C 0 D42 K43 Y44 I86 K234 G236 Q237 G256 G257 I258 S294 Q297 D42 K43 Y44 I86 K234 G236 Q237 G256 G257 I258 S294 Q297 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 11102456 401 ~ 413 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNFASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAIGLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 1fjx A 2.26 BS02 dna D 0 F79 C81 S85 I86 S87 K89 E119 V121 K162 R165 T226 R228 Q237 R240 Y242 G250 S252 A253 Y254 G303 N304 F79 C81 S85 I86 S87 K89 E119 V121 K162 R165 T226 R228 Q237 R240 Y242 G250 S252 A253 Y254 G303 N304 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 11102456 421 ~ 433 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNFASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAIGLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 1fkb A 1.7 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 F99 Y26 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Kd=0.2nM remove_due_to_license_issue IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fkf A 1.7 BS01 FK5 A 1 Y26 D37 F46 E54 V55 I56 W59 Y82 H87 F99 Y26 D37 F46 E54 V55 I56 W59 Y82 H87 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Kd=0.4nM remove_due_to_license_issue Kd=0.200000nM, EC50=0.900000nM, Ki=0.40nM, IC50=2.3nM P62942 1709302 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fkg A 2.0 BS01 SB3 A 1 Y26 D37 F46 V55 I56 W59 Y82 Y26 D37 F46 V55 I56 W59 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Ki=10nM remove_due_to_license_issue Ki=17nM P62942 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fkh A 1.95 BS01 SBX A 1 Y26 F36 D37 V55 I56 W59 Y82 H87 Y26 F36 D37 V55 I56 W59 Y82 H87 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Ki=7nM remove_due_to_license_issue P62942 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fki A 2.2 BS01 SB1 A 1 Y26 D37 R42 F46 V55 W59 Y82 Y26 D37 R42 F46 V55 W59 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Ki=100nM remove_due_to_license_issue P62942 109 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fkw A 2.4 BS02 PUR A 1 H17 D19 F61 F65 Y102 G184 E295 D296 H14 D16 F58 F62 Y99 G181 E292 D293 H15 H17 H214 E217 H238 E295 H12 H14 H211 E214 H235 E292 3.5.4.4 0000255,0001666,0001701,0001829,0001889,0001890,0002314,0002467,0002636,0002686,0002901,0002906,0004000,0005737,0005764,0005829,0005886,0006154,0006157,0006196,0006915,0006939,0007155,0008270,0009117,0009168,0009897,0009986,0010460,0014074,0016020,0016787,0019239,0019722,0030217,0030324,0030890,0031410,0032261,0032263,0032264,0033077,0033089,0033632,0042100,0042110,0043066,0043084,0043605,0044209,0045580,0045582,0045987,0046059,0046061,0046085,0046101,0046103,0046111,0046632,0046638,0046872,0046936,0048286,0048541,0048566,0050728,0050850,0050852,0050862,0050870,0050900,0060169,0060205,0060407,0070161,0070242,0070244,0070254,0070256,0140928 Ki=9uM remove_due_to_license_issue P03958 8672487 353 TPAFNKPKVELHVHLDGAIKPETILYFGKKRGIALPADTVEELRNIIGMDKPLSLPGFLAKFDYYMPVIAGCREAIKRIAYEFVEMKAKEGVVYVEVRYSPHLLANSKVDPMPWNQTEGDVTPDDVVDLVNQGLQEGEQAFGIKVRSILCCMRHQPSWSLEVLELCKKYNQKTVVAMDLAGDETIEGSSLFPGHVEAYEGAVKNGIHRTVHAGEVGSPEVVREAVDILKTERVGHGYHTIEDEALYNRLLKENMHFEVCPWSSYLTGAWDPKTTHAVVRFKNDKANYSLNTEDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEEEKKELLERLYREYQ 1fl3 H 2.45 BS01 SPB L 1 G100 W106 G97 W103 ? remove_due_to_license_issue P01867 11030644 225 AALLESGGGLVKPGGSLKLSCTASGITFSRYIMSWVRQIPEKRLEWVASISSGGITYYPDSVAGRFTISRDNVRNILYLQMSSLRSEDTALYYCARGQGRPYWGQGTSVTVSAAKTTPPSVYPAAPGCGDTTGSSVTLGCLVKGYFPEPVTVTWNSGGSSVHTFPALLQSGLYTMSSSVTVPSSTWPSTVTCSVAHPASSTTVDKKLE 1fl3 L 2.45 BS01 SPB L 1 Y39 P49 N96 L97 E98 P101 Y38 P48 N95 L96 E97 P100 ? 0005576,0005886,0030183 Kd=0.16uM remove_due_to_license_issue P01837 11030644 225 AALTQSPVSNPVTLGTSASISCRSTKSLLHSNGITYLYWYLQKPGQSPQLLIYQMSNLASGVPNRFSSSGSGTDFTLRINTVEAEDVGVYYCAQNLELPPTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNGYTCEATHKTSTSPIVKSFN 1fl6 H 2.8 BS01 AAH H 1 Y33 R52 D95 G96 A99 Y33 R52 D101 G102 A105 remove_due_to_license_issue 11535051 824 QVQLVESGGGLVQPGGSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKANGYTTEYSASVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDGSYAMDYWGQGTSVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 1fl6 L 2.8 BS01 AAH H 1 E34 R96 E39 R101 remove_due_to_license_issue 11535051 824 ELVMTQTPLSLPVSLGDQASISCRSSQSIVHSNGNTYLEWYLQKPGQSPKLLIYKVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFQGSHVPRTFGGGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRG 1flm A 1.3 BS01 FMN A 1 H27 V29 N30 T31 W32 P47 G49 G50 M51 H52 K53 T54 H27 V29 N30 T31 W32 P47 G49 G50 M51 H52 K53 T54 ? 0005737 Kd=0.43nM remove_due_to_license_issue Q46604 10713530 123 MLPGTFFEVLKNEGVVAIATQGEDGPHLVNTWNSYLKVLDGNRIVVPVGGMHKTEANVARDERVLMTLGSRKVAGRNGPGTGFLIRGSAAFRTDGPEFEAIARFKWARAALVITVVSAEQTL 1flm A 1.3 BS02 FMN B 1 G82 T121 L122 G82 T121 L122 ? 0005737 Kd=0.43nM remove_due_to_license_issue Q46604 10713530 123 MLPGTFFEVLKNEGVVAIATQGEDGPHLVNTWNSYLKVLDGNRIVVPVGGMHKTEANVARDERVLMTLGSRKVAGRNGPGTGFLIRGSAAFRTDGPEFEAIARFKWARAALVITVVSAEQTL 1flm B 1.3 BS01 FMN A 1 G82 T121 L122 G82 T121 L122 ? 0005737 Kd=0.43nM remove_due_to_license_issue Q46604 10713530 123 MLPGTFFEVLKNEGVVAIATQGEDGPHLVNTWNSYLKVLDGNRIVVPVGGMHKTEANVARDERVLMTLGSRKVAGRNGPGTGFLIRGSAAFRTDGPEFEAIARFKWARAALVITVVSAEQTL 1flm B 1.3 BS02 FMN B 1 H27 V29 N30 T31 W32 P47 G49 G50 M51 K53 T54 H27 V29 N30 T31 W32 P47 G49 G50 M51 K53 T54 ? 0005737 Kd=0.43nM remove_due_to_license_issue Q46604 10713530 123 MLPGTFFEVLKNEGVVAIATQGEDGPHLVNTWNSYLKVLDGNRIVVPVGGMHKTEANVARDERVLMTLGSRKVAGRNGPGTGFLIRGSAAFRTDGPEFEAIARFKWARAALVITVVSAEQTL 1flr H 1.85 BS01 FLU L 1 W33 Y56 Y102 Y103 G104 W33 Y56 Y100 Y101 G102 ? remove_due_to_license_issue P01865 8637844 600 EVKLDETGGGLVQPGRPMKLSCVASGFTFSDYWMNWVRQSPEKGLEWVAQIRNKPYNYETYYSDSVKGRFTISRDDSSVYLQMNNLRVEDMGIYYCTGSYYGMDYWGQGTSVTVSSAKTTAPSVYPLAPVCGDTTGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEPR 1flr L 1.85 BS01 FLU L 1 H31 Y37 R39 S96 W101 H31 Y37 R39 S96 W101 Kd=0.1nM remove_due_to_license_issue 8637844 600 DVVMTQTPLSLPVSLGDQASISCRSSQSLVHSNGNTYLRWYLQKPGQSPKVLIYKVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYFCSQSTHVPWTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 1fls A -1.00 BS04 WAY A 1 L81 H119 H123 H129 P139 Y141 L75 H113 H117 H123 P133 Y135 H119 E120 H123 H129 H113 E114 H117 H123 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=8nM P45452 10986126 169 TLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYG 1fm9 D 2.1 BS02 570 D 1 I281 F282 G284 C285 Q286 S289 H323 Y327 L330 I341 F360 F363 M364 H449 L465 L469 Y473 I76 F77 G79 C80 Q81 S84 H118 Y122 L125 I136 F155 F158 M159 H244 L260 L264 Y268 ? 0003677,0004879,0005634,0006355 Ki=1nM remove_due_to_license_issue Ki=1.1nM, EC50=0.338844nM, IC50=25nM P37231 10882139 200 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 1fmb A 1.8 BS01 HYB A 1 G27 A28 D29 I53 G54 G55 V56 G27 A28 D29 I53 G54 G55 V56 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.- 0004190,0006508 Ki=0.1nM remove_due_to_license_issue P32542 8844837 201 VTYNLEKRPTTIVLINDTPLNVLLDTGADTSVLTTAHYNRLKYRGRKYQGTGIGGVGGNVETFSTPVTIKKKGRHIKTRMLVADIPVTILGRDILQDLGAKLVL 1fo2 A 2.38 BS01 DMJ A 1 R597 P598 E599 F659 E663 T688 E689 R356 P357 E358 F418 E422 T447 E448 E330 R334 D463 E599 E91 R95 D222 E358 3.2.1.113 0004571,0005509,0005975,0016020 ic50=20uM remove_due_to_license_issue Q9UKM7 10995765 704 TQGPVHLNYRQKGVIDVFLHAWKGYRKFAWGHDELKPVSRSFSEWFGLGLTLIDALDTMWILGLRKEFEEARKWVSKKLHFEKDVDVNLFESTIRILGGLLSAYHLSGDSLFLRKAEDFGNRLMPAFRTPSKIPYSDVNIGTGVAHPPRSDSTVAEVTSIQLEFRELSRLTGDKKFQEAVEKVTQHIHGLSGKKDGLVPMFINTHSGLFTHLGVFTLGARADSYYEYLLKQWIQGGKQETQLLEDYVEAIEGVRTHLLRHSEPSKLTFVGELAHGRFSAKMDHLVCFLPGTLALGVYHGLPASHMELAQELMETCYQMNRQMETGLSPEIVHFNLYPQPGRRDVEVKPADRHNLLRPETVESLFYLYRVTGDRKYQDWGWEILQSFSRFTRVPSGGYSSINNVQDPQKPEPRDKMESFFLGETLKYLFLLFSDDPNLLSLDAYVFNTEAHPLPIWT 1fo3 A 1.75 BS01 KIF A 1 L525 R597 E599 F659 E663 T688 E689 L283 R355 E357 F417 E421 T446 E447 E330 R334 D463 E599 E90 R94 D221 E357 3.2.1.113 0004571,0005509,0005975,0016020 ic50=0.2uM remove_due_to_license_issue Q9UKM7 10995765 704 QGPVHLNYRQKGVIDVFLHAWKGYRKFAWGHDELKPVSRSFSEWFGLGLTLIDALDTMWILGLRKEFEEARKWVSKKLHFEKDVDVNLFESTIRILGGLLSAYHLSGDSLFLRKAEDFGNRLMPAFRTPSKIPYSDVNIGTGVAHPPRSDSTVAEVTSIQLEFRELSRLTGDKKFQEAVEKVTQHIHGLSGKKDGLVPMFINTHSGLFTHLGVFTLGARADSYYEYLLKQWIQGGKQETQLLEDYVEAIEGVRTHLLRHSEPSKLTFVGELAHGRFSAKMDHLVCFLPGTLALGVYHGLPASHMELAQELMETCYQMNRQMETGLSPEIVHFNLYPQPGRRDVEVKPADRHNLLRPETVESLFYLYRVTGDRKYQDWGWEILQSFSRFTRVPSGGYSSINNVQDPQKPEPRDKMESFFLGETLKYLFLLFSDDPNLLSLDAYVFNTEAHPLPIWT 1fpc H 2.3 BS03 0ZI H 1 H57 Y60A W60D L99 D189 A190 C191 E192 W215 G216 G219 C220 H43 Y47 W50 L96 D191 A192 C193 E194 W219 G220 G222 C223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.1uM remove_due_to_license_issue P00734 15299843 371 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 1fpi A 2.3 BS04 AMP A 1 V17 Q20 G21 G26 T27 E29 M30 Y113 R140 V9 Q12 G13 G18 T19 E21 M22 Y95 R122 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 remove_due_to_license_issue IC50=1300nM P00636 7568043 339 NIVTLTRFVMEQGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGKLDVLSNDLVINVLKSSFATCVLVTEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRNVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1fpp B 2.75 BS02 FPP B 1 W102 W106 R202 G250 W303 Y361 W81 W85 R181 G229 W282 Y340 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H227 R270 K273 D276 C278 Y279 D331 D338 H341 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 9609683 440 PLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVP 1fpy A 2.89 BS04 PPQ A 1 E131 E212 G265 H269 R321 E327 R359 E131 E212 G265 H269 R321 E327 R359 6.3.1.2 0003824,0004356,0005524,0005737,0006542,0016020,0016874,0016879,0019740,0030145,0046872,0051260 remove_due_to_license_issue P0A1P6 11329256 5900 SAEHVLTMLNEHEVKFVDLRFTDTKGKEQHVTIPAHQVNAEFFEEGKMFDGSSIGGWKGINESDMVLMPDASTAVIDPFFADSTLIIRCDILEPGTLQGYDRDPRSIAKRAEDYLRATGIADTVLFGPEPEFFLFDDIRFGASISGSHVAIDDIEGAWNSSTKYEGGNKGHRPGVKGGYFPVPPVDSAQDIRSEMCLVMEQMGLVVEAHHHEVATAGQNEVATRFNTMTKKADEIQIYKYVVHNVAHRFGKTATFMPKPMFGDNGSGMHCHMSLAKNGTNLFSGDKYAGLSEQALYYIGGVIKHAKAINALANPTTNSYKRLVPGYEAPVMLAYSARNRSASIRIPVVASPKARRIEVRFPDPAANPYLCFAALLMAGLDGIKNKIHPGEPMDKNLYDLPPEEAKEIPQVAGSLEEALNALDLDREFLKAGGVFTDEAIDAYIALRREEDDRVRMTPHPVEFELYYSV 1fpy B 2.89 BS04 PPQ B 1 E131 E212 G265 H269 R321 E327 R359 E131 E212 G265 H269 R321 E327 R359 6.3.1.2 0003824,0004356,0005524,0005737,0006542,0016020,0016874,0016879,0019740,0030145,0046872,0051260 remove_due_to_license_issue P0A1P6 11329256 5901 SAEHVLTMLNEHEVKFVDLRFTDTKGKEQHVTIPAHQVNAEFFEEGKMFDGSSIGGWKGINESDMVLMPDASTAVIDPFFADSTLIIRCDILEPGTLQGYDRDPRSIAKRAEDYLRATGIADTVLFGPEPEFFLFDDIRFGASISGSHVAIDDIEGAWNSSTKYEGGNKGHRPGVKGGYFPVPPVDSAQDIRSEMCLVMEQMGLVVEAHHHEVATAGQNEVATRFNTMTKKADEIQIYKYVVHNVAHRFGKTATFMPKPMFGDNGSGMHCHMSLAKNGTNLFSGDKYAGLSEQALYYIGGVIKHAKAINALANPTTNSYKRLVPGYEAPVMLAYSARNRSASIRIPVVASPKARRIEVRFPDPAANPYLCFAALLMAGLDGIKNKIHPGEPMDKNLYDLPPEEAKEIPQVAGSLEEALNALDLDREFLKAGGVFTDEAIDAYIALRREEDDRVRMTPHPVEFELYYSV 1fq4 A 2.7 BS02 2Y2 A 1 Q13 D32 G34 Y75 G76 T77 I128 Y189 D215 G217 T218 S219 Q14 D33 G35 Y76 G77 T78 I129 Y193 D218 G220 T221 S222 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D218 T221 3.4.23.25 0000324,0004190,0006508 remove_due_to_license_issue P07267 11061973 338 GGHDVPLTNYLNAQYYTDITLGTPPQNFKVILDTGSSNLWVPSNECGSLACFLHSKYDHEASSSYKANGTEFAIQYGTGSLEGYISQDTLSIGDLTIPKQDFAEATSEPGLTFAFGKFDGILGLGYDTISVDKVVPPFYNAIQQDLLDEKRFAFYLGDTSKDTENGGEATFGGIDESKFKGDITWLPVRRKAYWEVKFEGIGLGDEYAELESHGAAIDTGTSLITLPSGLAEMINAEIGAKKGWTGQYTLDCNTRDNLPDLIFNFNGYNFTIGPYDYTLEVSGSCISAITPMDFPEPVGPLAIVGDAFLRKYYSIYDIGNNAVGLAKAI 1fq5 A 2.4 BS01 0GM A 1 Q13 D32 Q74 Y75 G76 T77 T111 G115 F117 I120 I128 D215 G217 T218 S219 F291 Q14 D33 Q75 Y76 G77 T78 T112 G116 F118 I121 I129 D218 G220 T221 S222 F294 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D218 T221 3.4.23.25 0000324,0004190,0006508 Ki=4nM remove_due_to_license_issue P07267 11061973 338 GGHDVPLTNYLNAQYYTDITLGTPPQNFKVILDTGSSNLWVPSNECGSLACFLHSKYDHEASSSYKANGTEFAIQYGTGSLEGYISQDTLSIGDLTIPKQDFAEATSEPGLTFAFGKFDGILGLGYDTISVDKVVPPFYNAIQQDLLDEKRFAFYLGDTSKDTENGGEATFGGIDESKFKGDITWLPVRRKAYWEVKFEGIGLGDEYAELESHGAAIDTGTSLITLPSGLAEMINAEIGAKKGWTGQYTLDCNTRDNLPDLIFNFNGYNFTIGPYDYTLEVSGSCISAITPMDFPEPVGPLAIVGDAFLRKYYSIYDIGNNAVGLAKAI 1fq6 A 2.7 BS01 0QF A 1 Q13 I30 D32 Y75 G76 T77 T111 I120 Y189 D215 G217 T218 S219 I300 Q14 I31 D33 Y76 G77 T78 T112 I121 Y193 D218 G220 T221 S222 I303 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D218 T221 3.4.23.25 0000324,0004190,0006508 remove_due_to_license_issue P07267 11061973 400 GGHDVPLTNYLNAQYYTDITLGTPPQNFKVILDTGSSNLWVPSNECGSLACFLHSKYDHEASSSYKANGTEFAIQYGTGSLEGYISQDTLSIGDLTIPKQDFAEATSEPGLTFAFGKFDGILGLGYDTISVDKVVPPFYNAIQQDLLDEKRFAFYLGDTSKDTENGGEATFGGIDESKFKGDITWLPVRRKAYWEVKFEGIGLGDEYAELESHGAAIDTGTSLITLPSGLAEMINAEIGAKKGWTGQYTLDCNTRDNLPDLIFNFNGYNFTIGPYDYTLEVSGSCISAITPMDFPEPVGPLAIVGDAFLRKYYSIYDIGNNAVGLAKAI 1fq7 A 2.8 BS02 2Y3 A 1 Q13 I30 D32 G34 Y75 G76 T77 T111 F117 Y189 D215 G217 T218 S219 Q14 I31 D33 G35 Y76 G77 T78 T112 F118 Y193 D218 G220 T221 S222 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D218 T221 3.4.23.25 0000324,0004190,0006508 remove_due_to_license_issue P07267 11061973 400 GGHDVPLTNYLNAQYYTDITLGTPPQNFKVILDTGSSNLWVPSNECGSLACFLHSKYDHEASSSYKANGTEFAIQYGTGSLEGYISQDTLSIGDLTIPKQDFAEATSEPGLTFAFGKFDGILGLGYDTISVDKVVPPFYNAIQQDLLDEKRFAFYLGDTSKDTENGGEATFGGIDESKFKGDITWLPVRRKAYWEVKFEGIGLGDEYAELESHGAAIDTGTSLITLPSGLAEMINAEIGAKKGWTGQYTLDCNTRDNLPDLIFNFNGYNFTIGPYDYTLEVSGSCISAITPMDFPEPVGPLAIVGDAFLRKYYSIYDIGNNAVGLAKAI 1fq8 A 2.8 BS01 2Y4 A 1 Q13 I30 D32 Y75 G76 T77 F117 D215 G217 T218 S219 Q14 I31 D33 Y76 G77 T78 F118 D218 G220 T221 S222 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D218 T221 3.4.23.25 0000324,0004190,0006508 remove_due_to_license_issue P07267 11061973 400 GGHDVPLTNYLNAQYYTDITLGTPPQNFKVILDTGSSNLWVPSNECGSLACFLHSKYDHEASSSYKANGTEFAIQYGTGSLEGYISQDTLSIGDLTIPKQDFAEATSEPGLTFAFGKFDGILGLGYDTISVDKVVPPFYNAIQQDLLDEKRFAFYLGDTSKDTENGGEATFGGIDESKFKGDITWLPVRRKAYWEVKFEGIGLGDEYAELESHGAAIDTGTSLITLPSGLAEMINAEIGAKKGWTGQYTLDCNTRDNLPDLIFNFNGYNFTIGPYDYTLEVSGSCISAITPMDFPEPVGPLAIVGDAFLRKYYSIYDIGNNAVGLAKAI 1fsg A 1.05 BS02 9DG A 1 Y118 D150 K178 W199 I200 Y205 D206 Y121 D153 K181 W202 I203 Y208 D209 E146 D147 D150 W199 R212 E149 D150 D153 W202 R215 2.4.2.22,2.4.2.8 0000166,0000287,0000310,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032265,0046100,0046872,0052657 ic50=9.5uM remove_due_to_license_issue Q26997 11188695 304 GSHMASKPIEDYGKGKGRIEPMYIPDNTFYNADDFLVPPHCKPYIDKILLPGGLVKDRVEKLAYDIHRTYFGEELHIICILKGSRGFFNLLIDYLATIQKYSGRESSVPPFFEHYVRLKSYQNDNSTGQLTVLSDDLSIFRDKHVLIVEDIVDTGFTLTEFGERLKAVGPKSMRIATLVEKRTDRSNSLKGDFVGFSIEDVWIVGCCYDFNEMFRDFDHVAVLSDAARKKFEK 1fsw A 1.9 BS01 CTB A 1 S64 K67 Q120 Y150 N152 A318 T319 S61 K64 Q117 Y147 N149 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=3.2e+2nM P00811 11182316 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALA 1fsy A 1.75 BS01 105 A 1 S64 Q120 Y150 N152 Y221 A318 S61 Q117 Y147 N149 Y218 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=150nM P00811 11182316 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALA 1ft4 A 2.9 BS01 703 A 1 T61 A62 L67 L71 T51 A52 L57 L61 ? 0005031,0006693,0006954,0033209 remove_due_to_license_issue P19438 11592999 962 MDSVCPQGKYIHPQNNSICCTKCHKGTYLYNDCPGPGQDTDCRECESGSFTASENHLRHCLSCSKCRKEMGQVEISSCTVDRDTVCGCRKNQYRHYWSENLFQCFNCSLCLNGTVHLSCQEKQNTVCTCHAGFFLRENEC 1ft7 A 2.2 BS03 PLU A 1 H97 D117 E151 E152 D179 C227 H97 D117 E151 E152 D179 C227 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=6.6uM remove_due_to_license_issue Q01693 11401547 500 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 1fta A 2.3 BS01 AMP A 1 V17 E20 G21 A24 G26 T27 G28 E29 L30 T31 K112 Y113 V9 E12 G13 A16 G18 T19 G20 E21 L22 T23 K96 Y97 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=3200nM P09467 7961695 338 DVVTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEAYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPIILGSPDDVLEFLKVYEKHS 1fta C 2.3 BS01 AMP C 1 V17 E20 G21 A24 G26 T27 G28 E29 L30 K112 Y113 R140 M177 V9 E12 G13 A16 G18 T19 G20 E21 L22 K94 Y95 R122 M159 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=3200nM P09467 7961695 338 DVVTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEAYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPIILGSPDDVLEFLKVYEKHS 1ftj A 1.9 BS02 GLU A 1 Y61 L90 T91 R96 G141 S142 T143 E193 Y58 L87 T88 R93 G138 S139 T140 E190 ? 0015276,0016020 ic50=821nM remove_due_to_license_issue P19491 11086992 274 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1ftk A 1.6 BS01 KAI A 1 Y73 P101 T103 R108 L154 S158 T159 E209 M212 Y55 P83 T85 R90 L127 S131 T132 E182 M185 ? 0015276,0016020 ic50=14.5uM remove_due_to_license_issue EC50=380000nM, Ki=3690nM P19491 11086992 999 KTVVVTTILESPYVMMKKMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1ftm A 1.7 BS02 AMQ A 1 Y61 T91 R96 G141 S142 T143 L192 E193 M196 Y220 Y58 T88 R93 G138 S139 T140 L189 E190 M193 Y217 ? 0015276,0016020 Kd=24.8nM remove_due_to_license_issue Ki=17nM P19491 11086992 428 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1fv0 A 1.7 BS01 9AR A 1 L2 A18 I19 Y22 G30 W31 C45 H48 D49 L2 A17 I18 Y21 G29 W30 C44 H47 D48 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 Ki=1.18uM remove_due_to_license_issue P59071 12206661 401 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 1fv9 A 3.0 BS01 172 A 1 D191 S192 C193 G218 G220 D192 S193 C194 G219 G221 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 11052791 246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1fvt A 2.2 BS01 106 A 1 I10 A31 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F73 E74 F75 L76 H77 Q78 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=60nM P24941 11141566 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1fvv A 2.8 BS01 107 A 1 K9 I10 A31 K33 F80 F82 L83 H84 Q85 D86 K89 L134 D145 K9 I10 A31 K33 F80 F82 L83 H84 Q85 D86 K89 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 11141566 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1fw0 A 1.9 BS01 KAI A 1 E13 Y61 P89 T91 R96 L138 G141 S142 T143 E193 M196 E10 Y58 P86 T88 R93 L135 G138 S139 T140 E190 M193 ? 0015276,0016020 remove_due_to_license_issue EC50=380000nM, Ki=3690nM P19491 11086992 999 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1fwe C 2.0 BS03 HAE C 1 H134 K217 H246 G277 D360 A363 H133 K216 H245 G276 D345 A348 H134 H136 K217 H219 D221 H246 H272 R336 D360 H133 H135 K216 H218 D220 H245 H271 R321 D345 3.5.1.5 0005515,0005737,0009039,0016151,0016787,0016810,0043419,0046872 remove_due_to_license_issue P18314 9201965 989 SNISRQAYADMFGPTVGDKVRLADTELWIEVEDDLTTYGEEVKFGGGKVIRDGMGQGQMLAADCVDLVLTNALIVDHWGIVKADIGVKDGRIFAIGKAGNPDIQPNVTIPIGAATEVIAAEGKIVTAGGIDTHIHWICPQQAEEALVSGVTTMVGGGTGPAAGTHATTCTPGPWYISRMLQAADSLPVNIGLLGKGNVSQPDALREQVAAGVIGLKIHEDWGATPAAIDCALTVADEMDIQVALHSDTLNESGFVEDTLAAIGGRTIHTFHTEGAGGGHAPDIITACAHPNILPSSTNPTLPYTLNTIDEHLDMLMFAESRIRRETIAAEDVLHDLGAFSLTSSDSQAMGRVGEVILRTWQVAHRMKVQRGALAEETGDNDNFRVKRYIAKYTINPALTHGIAHEVGSIEVGKLADLVVWSPAFFGVKPATVIKGGMIAIAPMGDINASIPTPQPVHYRPMFGALGSARHHCRLTFLSQAAAANGVAERLNLRSAIAVVKGCRTVQKADMVHNSLQPNITVDAQTYEVRVDGELITSEPADVLPMAQRYFLF 1fwu A 1.9 BS01 SGA B 1 N102 Y111 G113 G115 W117 N101 Y110 G112 G114 W116 ? remove_due_to_license_issue Q61830 11152606 3 DARQFLIYNEDHKRCVDALSAISVQTATCNPEAESQKFRWVSDSQIMSVAFKLCLGVPSKTDWASVTLYACDSKSEYQKWECKNDTLFGIKGTELYFNYGNRQEKNIKLYKGSGLWSRWKVYGTTDDLCSRGYE 1fwv A 2.2 BS01 SGA B 1 N102 Y111 G113 G115 W117 N101 Y110 G112 G114 W116 ? remove_due_to_license_issue Q61830 11152606 2 DARQFLIYNEDHKRCVDALSAISVQTATCNPEAESQKFRWVSDSQIMSVAFKLCLGVPSKTDWASVTLYACDSKSEYQKWECKNDTLFGIKGTELYFNYGNRQEKNIKLYKGSGLWSRWKVYGTTDDLCSRGYE 1fzq A 1.7 BS01 GDP A 1 N27 G29 K30 T31 T32 N126 K127 D129 L130 S159 A160 L161 N26 G28 K29 T30 T31 N125 K126 D128 L129 S158 A159 L160 Q71 Q70 ? 0000139,0000281,0000287,0001822,0003924,0005515,0005525,0005634,0005654,0005737,0005794,0005813,0005819,0005856,0005876,0005881,0005929,0005930,0006892,0006893,0007224,0007264,0008017,0015031,0016020,0019003,0030496,0032391,0035869,0036064,0042073,0042461,0042995,0046872,0051301,0060271,0061512,1903441 Kd=24nM remove_due_to_license_issue Q9WUL7 11188688 301 GLLSILRKLKSAPDQEVRILLLGLDNAGKTTLLKQLASEDISHITPTQGFNIKSVQSQGFKLNVWDIGGQRKIRPYWRSYFENTDILIYVIDSADRKRFEETGQELTELLEEEKLSCVPVLIFANKQDLLTAAPASEIAEGLNLHTIRDRVWQIQSCSALTGEGVQDGMNWVCKNV 1g05 B 2.45 BS06 BBH B 1 N662 L664 A665 H701 E702 H705 H711 N80 L82 A83 H119 E120 H123 H129 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=3.1nM remove_due_to_license_issue IC50=3.1nM P08254 11327577 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET 1g1d A 2.04 BS02 FSB A 1 H94 H96 H119 L198 T199 T200 H92 H94 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.36nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g27 A 2.1 BS01 BB1 A 1 G43 I44 G45 Q50 G89 C90 L91 C129 H132 E133 H136 G43 I44 G45 Q50 G89 C90 L91 C129 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 3.5.1.88 0005515,0005829,0006412,0008198,0008270,0016787,0042586,0043022,0043686,0046872 ic50=7nM remove_due_to_license_issue P0A6K3 11158755 1001 SVLQVLHIPDERLRKVAKPVEEVNAEIQRIVDDMFETMYAEEGIGLAATQVDIHQRIIVIDVSENRDERLVLINPELLEKSGETGIEEGCLSIPEQRALVPRAEKVKIRALDRDGKPFELEADGLLAICIQHEMDHLVGKLFMDYLSPLKQQRIRQKVEKLDRL 1g2a A 1.75 BS01 BB2 A 1 G43 I44 G45 Q50 E87 G89 C90 R97 C129 H132 E133 H136 G43 I44 G45 Q50 E87 G89 C90 R97 C129 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 3.5.1.88 0005515,0005829,0006412,0008198,0008270,0016787,0042586,0043022,0043686,0046872 ic50=10nM remove_due_to_license_issue P0A6K3 11158755 1001 SVLQVLHIPDERLRKVAKPVEEVNAEIQRIVDDMFETMYAEEGIGLAATQVDIHQRIIVIDVSENRDERLVLINPELLEKSGETGIEEGCLSIPEQRALVPRAEKVKIRALDRDGKPFELEADGLLAICIQHEMDHLVGKLFMDYLSPLKQQRIRQKVEKLDRL 1g2k A 1.95 BS01 NM1 B 1 D25 G27 A28 D29 D30 I50 V82 D25 G27 A28 D29 D30 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 11170625 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1g2k B 1.95 BS01 NM1 B 1 R8 D25 G27 A28 D30 V32 G49 I50 R8 D25 G27 A28 D30 V32 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=11nM remove_due_to_license_issue P04587 11170625 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1g2l A 1.9 BS02 T87 A 1 H57 T99 Y100 F177 D194 A195 C196 Q197 S200 V218 W220 G223 H42 T84 Y85 F162 D179 A180 C181 Q182 S185 V203 W205 G208 H57 D103 Q197 G198 D199 S200 G201 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=57nM remove_due_to_license_issue Ki=57nM P00742 11342132 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTR 1g2m A 3.02 BS02 R11 A 1 H57 T98 Y99 F174 D189 A190 C191 V213 W215 G216 G218 C220 H42 T84 Y85 F162 D179 A180 C181 V203 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=40nM P00742 11342132 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTR 1g2o A 1.75 BS02 IMH A 1 Y92 A120 G122 Y188 E189 V205 G206 M207 N231 H243 Y86 A114 G116 Y182 E183 V199 G200 M201 N225 H237 S36 H68 H90 Y92 E93 A120 M207 S208 N231 A233 H243 S30 H62 H84 Y86 E87 A114 M201 S202 N225 A227 H237 2.4.2.1 0003824,0004731,0005737,0006139,0006154,0006161,0009116,0016757,0016763 Ki=28pM remove_due_to_license_issue P9WP01 11444966 351 DPDELARRAAQVIADRTGIGEHDVAVVLGSGWLPAVAALGSPTTVLPQAELPGFVPPTAAGHAGELLSVPIGAHRVLVLAGRIHAYEGHDLRYVVHPVRAARAAGAQIMVLTNAAGGLRADLQVGQPVLISDHLNLTARSPLVGGEFVDLTDAYSPRLRELARQSDPQLAEGVYAGLPGPHYETPAEIRMLQTLGADLVGMSTVHETIAARAAGAEVLGVSLVTNLAAGITGEPLSHAEVLAAGAASATRMGALLADVIARF 1g2o B 1.75 BS02 IMH B 1 Y92 A120 G122 Y188 E189 G206 M207 N231 H243 Y86 A114 G116 Y182 E183 G200 M201 N225 H237 S36 H68 H90 Y92 E93 A120 M207 S208 N231 A233 H243 S30 H62 H84 Y86 E87 A114 M201 S202 N225 A227 H237 2.4.2.1 0003824,0004731,0005737,0006139,0006154,0006161,0009116,0016757,0016763 Ki=28pM remove_due_to_license_issue P9WP01 11444966 352 DPDELARRAAQVIADRTGIGEHDVAVVLGSGWLPAVAALGSPTTVLPQAELPGFVPPTAAGHAGELLSVPIGAHRVLVLAGRIHAYEGHDLRYVVHPVRAARAAGAQIMVLTNAAGGLRADLQVGQPVLISDHLNLTARSPLVGGEFVDLTDAYSPRLRELARQSDPQLAEGVYAGLPGPHYETPAEIRMLQTLGADLVGMSTVHETIAARAAGAEVLGVSLVTNLAAGITGEPLSHAEVLAAGAASATRMGALLADVIARF 1g30 B 2.0 BS03 T87 B 1 H57 Y60A W60D N98 L99 I174 D189 A190 S195 V213 S214 W215 G216 H43 Y47 W50 N95 L96 I172 D192 A193 S198 V218 S219 W220 G221 H57 D102 E192 G193 D194 S195 G196 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=140nM remove_due_to_license_issue Ki=140nM P00734 11342132 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1g32 B 1.9 BS03 R11 B 1 H57 Y60A W60D N98 L99 I174 D189 A190 S195 S214 W215 G216 H43 Y47 W50 N95 L96 I172 D192 A193 S198 S219 W220 G221 H57 D102 E192 G193 D194 S195 G196 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=780nM remove_due_to_license_issue Ki=780nM P00734 11342132 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1g35 A 1.8 BS01 AHF B 1 R8 D25 G27 A28 D30 G48 P81 R8 D25 G27 A28 D30 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 11170625 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1g35 B 1.8 BS01 AHF B 1 R8 L23 D25 G27 A28 D30 V32 G49 I50 P81 R8 L23 D25 G27 A28 D30 V32 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=7.3nM remove_due_to_license_issue P03366 11170625 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1g36 A 1.9 BS02 R11 A 1 H57 N97 L99 Q175 D189 S190 S195 W215 G216 G219 H40 N79 L81 Q155 D171 S172 S177 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=67nM remove_due_to_license_issue Ki=67nM P00760 11342132 990 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1g37 A 2.0 BS02 110 A 1 L40 L41 H57 W60D E97A N98 L99 I174 A190 E192 G193 S195 W215 G216 G219 L53 L54 H70 W77 E121 N122 L123 I199 A220 E222 G223 S225 W247 G248 G250 H57 D102 E192 G193 D194 S195 G196 H70 D126 E222 G223 D224 S225 G226 3.4.21.5 0004252,0005509,0005576,0006508,0007596 remove_due_to_license_issue P00734 11212093 900 ADCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1g3b A 1.8 BS02 108 A 1 D189 S190 C191 Q192 V213 W215 G216 G219 D171 S172 C173 Q174 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.8uM remove_due_to_license_issue P00760 11152605 601 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1g3c A 1.8 BS02 109 A 1 H57 D189 S190 Q192 S214 W215 G216 C220 H40 D171 S172 Q174 S192 W193 G194 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 11152605 601 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1g3c A 1.8 BS03 109 A 2 Q192 W215 Q174 W193 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 11152605 602 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1g3d A 1.8 BS02 108 A 1 D189 S190 S195 V213 W215 D171 S172 S177 V191 W193 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=2.8uM remove_due_to_license_issue P00760 11152605 601 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1g3e A 1.8 BS02 109 A 1 D189 S190 S214 W215 G216 G219 D171 S172 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=4.2uM remove_due_to_license_issue P00760 11152605 601 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1g3m B 1.7 BS02 PCQ B 1 Y20 F80 K105 H107 F141 V145 A146 Y239 I246 Y18 F78 K98 H100 F134 V138 A139 Y232 I239 K47 H107 S137 K45 H100 S130 2.8.2.4 0004062,0004304,0005496,0005515,0005737,0005829,0006068,0006629,0006711,0008146,0008202,0008210,0016740,0031965,0045600,0047894,0050294,0050427,0051923 ic50~0.15nM remove_due_to_license_issue P49888 12782487 711 SELDYYEKFEEVHGILMYKDFVKYWDNVEAFQARPDDLVIATYPKSGTTWVSEIVYMIYKEGDVEKCKEDVIFNRIPFLECRNGVKQLDEMNSPRIVKTHLPPELLPASFWEKDCKIIYLCRNAKDVAVSFYYFFLMVAGHPNPGSFPEFVEKFMQGQVPYGSWYKHVKSWWEKGKSPRVLFLFYEDLKEDIRKEVIKLIHFLERKPSEELVDRIIHHTSFQEMKNNPSTNYTTLPDEIMNQKLSPFMRKGITGDWKNHFTVALNEKFDKHYEQQMKESTLKFRT 1g45 A 1.83 BS02 FSB A 1 H94 H96 H119 L198 T199 T200 P202 H92 H94 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=2.3nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g46 A 1.84 BS02 F2B A 1 H94 H96 H119 L198 T199 T200 H92 H94 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.6nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g48 A 1.86 BS02 F6B A 1 H94 H96 H119 L198 T199 T200 P202 H92 H94 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.9nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g49 B 1.9 BS06 111 B 1 L664 A665 L697 H701 E702 H705 H711 L718 P721 L722 L82 A83 L115 H119 E120 H123 H129 L136 P139 L140 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=16nM remove_due_to_license_issue IC50=16nM P08254 11150165 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1g4j A 1.84 BS02 FFB A 1 H94 H96 H119 L198 T199 T200 H92 H94 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=2nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g4j A 1.84 BS03 FFB A 2 E69 F70 D72 I91 Q92 V131 V135 E67 F68 D70 I89 Q90 V128 V132 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=2nM remove_due_to_license_issue P00918 666 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g4k A 2.0 BS06 HQQ A 1 L164 A165 H201 E202 H205 H211 L218 Y220 P221 L222 Y223 H224 L82 A83 H119 E120 H123 H129 L136 Y138 P139 L140 Y141 H142 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=2000nM P08254 11316871 306 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPP 1g4o A 1.96 BS02 BSB A 1 H94 H96 H119 L198 T199 T200 P202 H92 H94 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=5.6nM remove_due_to_license_issue Kd=1.1nM P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g50 A 2.9 BS01 EST A 1 E353 L387 R394 F404 H524 L525 E50 L84 R91 F101 H221 L222 ? remove_due_to_license_issue IC50=1.3nM, Kd=0.2nM, EC50=0.75nM, Ki=0.21nM P03372 11437591 600 NSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLH 1g52 A 1.8 BS02 F2B A 1 H94 H96 H119 L198 T199 T200 P202 H92 H94 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.29nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g53 A 1.94 BS02 F6B A 1 H94 H96 H119 F131 L198 T199 T200 P202 H92 H94 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.91nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g54 A 1.86 BS02 FFB A 1 H94 H96 H119 F131 V135 L198 T199 T200 H92 H94 H117 F128 V132 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.5nM remove_due_to_license_issue P00918 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1g59 A 2.4 BS01 rna B 0 D44 R45 A46 R47 P109 V145 R163 V166 E172 V177 K180 S181 D182 E207 E208 R237 K241 T242 K243 M273 G274 E282 S299 L300 P303 V304 K309 W312 R319 P357 R358 R417 K426 L427 Q432 R435 L442 E443 T444 P445 G446 L447 F448 D44 R45 A46 R47 P109 V145 R163 V166 E172 V177 K180 S181 D182 E207 E208 R237 K241 T242 K243 M273 G274 E282 S299 L300 P303 V304 K309 W312 R319 P357 R358 R417 K426 L427 Q432 R435 L442 E443 T444 P445 G446 L447 F448 6.1.1.17 0000049,0000166,0004812,0004818,0005524,0005737,0005829,0006412,0006418,0006424,0008270,0043039 remove_due_to_license_issue P27000 11224561 501 ~ 576 MVVTRIAPSPTGDPHVGTAYIALFNYAWARRNGGRFIVRIEDTDRARYVPGAEERILAALKWLGLSYDEGPDVAAPTGPYRQSERLPLYQKYAEELLKRGWAYRAFETPEELEQIRKEKGGYDGRARNIPPEEAEERARRGEPHVIRLKVPRPGTTEVKDELRGVVVYDNQEIPDVVLLKSDGYPTYHLANVVDDHLMGVTDVIRAEEWLVSTPIHVLLYRAFGWEAPRFYHMPLLRNPDKTKISKRKSHTSLDWYKAEGFLPEALRNYLCLMGFSMPDGREIFTLEEFIQAFTWERVSLGGPVFDLEKLRWMNGKYIREVLSLEEVAERVKPFLREAGLSWESEAYLRRAVELMRPRFDTLKEFPEKARYLFTEDYPVSEKAQRKLEEGLPLLKELYPRLRAQEEWTEAALEALLRGFAAEKGVKLGQVAQPLRAALTGSLETPGLFEILALLGKERALRRLERALA 1g59 C 2.4 BS01 rna D 0 D44 R45 A46 R116 V145 R163 V166 E172 V177 K180 S181 D182 E207 L235 R237 K241 K243 G274 E282 R297 S299 P303 V304 K309 W312 P357 R358 R417 L427 Q432 R435 L442 E443 T444 P445 G446 L447 F448 D44 R45 A46 R116 V145 R163 V166 E172 V177 K180 S181 D182 E207 L235 R237 K241 K243 G274 E282 R297 S299 P303 V304 K309 W312 P357 R358 R417 L427 Q432 R435 L442 E443 T444 P445 G446 L447 F448 K246 K246 6.1.1.17 0000049,0000166,0004812,0004818,0005524,0005737,0005829,0006412,0006418,0006424,0008270,0043039 remove_due_to_license_issue P27000 11224561 501 ~ 576 MVVTRIAPSPTGDPHVGTAYIALFNYAWARRNGGRFIVRIEDTDRARYVPGAEERILAALKWLGLSYDEGPDVAAPTGPYRQSERLPLYQKYAEELLKRGWAYRAFETPEELEQIRKEKGGYDGRARNIPPEEAEERARRGEPHVIRLKVPRPGTTEVKDELRGVVVYDNQEIPDVVLLKSDGYPTYHLANVVDDHLMGVTDVIRAEEWLVSTPIHVLLYRAFGWEAPRFYHMPLLRNPDKTKISKRKSHTSLDWYKAEGFLPEALRNYLCLMGFSMPDGREIFTLEEFIQAFTWERVSLGGPVFDLEKLRWMNGKYIREVLSLEEVAERVKPFLREAGLSWESEAYLRRAVELMRPRFDTLKEFPEKARYLFTEDYPVSEKAQRKLEEGLPLLKELYPRLRAQEEWTEAALEALLRGFAAEKGVKLGQVAQPLRAALTGSLETPGLFEILALLGKERALRRLERALA 1g5s A 2.61 BS01 I17 A 1 I10 E12 A31 F80 F82 L83 H84 N132 L134 D145 I10 E12 A31 F71 F73 L74 H75 N123 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T142 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=48nM P24941 11170642 400 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1g6s A 1.5 BS01 S3P A 1 K22 S23 R27 T97 S169 S170 Q171 S197 Y200 D313 N336 K340 K22 S23 R27 T97 S169 S170 Q171 S197 Y200 D313 N336 K340 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 remove_due_to_license_issue Kd=7000nM P0A6D3 11171958 601 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 1g74 A 1.7 BS01 OLA A 1 F16 M20 P38 S53 S55 V75 D76 V115 C117 R126 Y128 F16 M20 P38 S53 S55 V75 D76 V115 C117 R126 Y128 ? 0005324,0005634,0005654,0005737,0008289,0009617,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0071285,0071356,0120162 Kd=0.3uM remove_due_to_license_issue P04117 14594993 132 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDLVTIRSESTFKNTEISFKLGVEFDEETVDGRKVKSIITLDGGALVQVQKWDGKSTTIKRKRDGDKLVVECVMKGVTSTRVYERA 1g7f A 1.8 BS01 INZ A 1 Y46 R47 D48 S216 A217 I219 G220 R221 Q262 Q266 Y45 R46 D47 S215 A216 I218 G219 R220 Q261 Q265 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=3.4uM remove_due_to_license_issue P18031 11341829 500 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1g7g A 2.2 BS01 INX A 1 Y46 R47 D48 K120 D181 F182 A217 R221 Y45 R46 D47 K119 D180 F181 A216 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.25uM remove_due_to_license_issue P18031 11341829 600 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1g7v A 2.4 BS01 PAI A 1 N62 R63 F117 R168 H202 Q205 A247 G251 P252 N62 R63 F117 R168 H202 Q205 A247 G251 P252 N26 K60 D250 N26 K60 D250 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0032991,0042802 Kd=0.4uM remove_due_to_license_issue P0A715 11371194 300 MKQKVVSIGDINVANDLPFVLFGGMNVLESRDLAMRICEHYVTVTQKLGIPYVFKASFDKANRSSIHSYRGPGLEEGMKIFQELKQTFGVKIITDVHEPSQAQPVADVVDVIQLPAFLARQTDLVEAMAKTGAVINVKKPQFVSPGQMGNIVDKFKEGGNEKVILCDRGANFGYDNLVVDMLGFSIMKKVSGNSPVIFDVTHALQCRDPFGAASGGRRAQVAELARAGMAVGLAGLFIEAHPDPEHAKCDGPSALPLAKLEPFLKQMKAIDDLVKGFEELDTSK 1g85 A 1.8 BS01 3OL A 1 F36 F56 F36 F56 ? 0005549,0005576,0005615,0007608,0036094 Kd=3.3uM remove_due_to_license_issue P07435 11114310 1001 AQEEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTGLFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPHPE 1g85 A 1.8 BS02 3OL A 2 T38 F56 T116 T38 F56 T116 ? 0005549,0005576,0005615,0007608,0036094 Kd=3.3uM remove_due_to_license_issue P07435 11114310 1002 AQEEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTGLFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPHPE 1g85 B 1.8 BS01 3OL B 1 N87 F89 N103 N85 F87 N101 ? 0005549,0005576,0005615,0007608,0036094 Kd=3.3uM remove_due_to_license_issue P07435 11114310 1004 EEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTGLFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPH 1g98 A 1.9 BS01 PA5 A 1 I156 G158 S209 K210 T211 T214 E357 K518 I156 G158 S209 K210 T211 T214 E357 K518 K210 E216 G271 R272 E357 H388 K518 K210 E216 G271 R272 E357 H388 K518 5.3.1.9 0004347,0005125,0005576,0005615,0005737,0005829,0006094,0006096,0007165,0016853,0048029,0051156,0097367,1901135 Ki=2uM remove_due_to_license_issue Q9N1E2 11327814 558 AALTRNPQFQKLQQWHREHGSELNLRHLFDTDKERFNHFSLTLNTNHGHILLDYSKNLVTEEVMHMLLDLAKSRGVEAARESMFNGEKINSTEDRAVLHVALRNRSNTPIVVDGKDVMPEVNKVLDKMKAFCQRVRSGDWKGYTGKTITDVINIGIGGSDLGPLMVTEALKPYSSGGPRVWFVSNIDGTHIAKTLACLNPESSLFIIASKTFTTQETITNAKTAKDWFLLSAKDPSTVAKHFVALSTNTAKVKEFGIDPQNMFEFWDWVGGRYSLWSAIGLSIALHVGFDNFEQLLSGAHWMDQHFRTTPLEKNAPVLLAMLGIWYINCFGCETQAVLPYDQYLHRFAAYFQQGDMESNGKYITKSGARVDHQTGPIVWGEPGTNGQHAFYQLIHQGTKMIPCDFLIPVQTQHPIRKGLHHKILLANFLAQTEALMKGKSTEEARKELQAAGKSPEDLMKLLPHKVFEGNRPTNSIVFTKLTPFILGALIAMYEHKIFVQGVVWDINSFDQWGVELGKQLAKKIEPELDGSSPVTSHDSSTNGLINFIKQQREAK 1g98 B 1.9 BS01 PA5 B 1 I156 G158 S209 K210 T211 T214 E357 K518 I156 G158 S209 K210 T211 T214 E357 K518 K210 E216 G271 R272 E357 H388 K518 K210 E216 G271 R272 E357 H388 K518 5.3.1.9 0004347,0005125,0005576,0005615,0005737,0005829,0006094,0006096,0007165,0016853,0048029,0051156,0097367,1901135 Ki=2uM remove_due_to_license_issue Q9N1E2 11327814 558 AALTRNPQFQKLQQWHREHGSELNLRHLFDTDKERFNHFSLTLNTNHGHILLDYSKNLVTEEVMHMLLDLAKSRGVEAARESMFNGEKINSTEDRAVLHVALRNRSNTPIVVDGKDVMPEVNKVLDKMKAFCQRVRSGDWKGYTGKTITDVINIGIGGSDLGPLMVTEALKPYSSGGPRVWFVSNIDGTHIAKTLACLNPESSLFIIASKTFTTQETITNAKTAKDWFLLSAKDPSTVAKHFVALSTNTAKVKEFGIDPQNMFEFWDWVGGRYSLWSAIGLSIALHVGFDNFEQLLSGAHWMDQHFRTTPLEKNAPVLLAMLGIWYINCFGCETQAVLPYDQYLHRFAAYFQQGDMESNGKYITKSGARVDHQTGPIVWGEPGTNGQHAFYQLIHQGTKMIPCDFLIPVQTQHPIRKGLHHKILLANFLAQTEALMKGKSTEEARKELQAAGKSPEDLMKLLPHKVFEGNRPTNSIVFTKLTPFILGALIAMYEHKIFVQGVVWDINSFDQWGVELGKQLAKKIEPELDGSSPVTSHDSSTNGLINFIKQQREAK 1g9a A 2.1 BS02 BAB A 1 D68 Q258 R369 Y372 F373 S374 D375 S376 E451 L453 F454 F455 T709 Y712 T713 D68 Q258 R369 Y372 F373 S374 D375 S376 E448 L450 F451 F452 T706 Y709 T710 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 ic50~7.5uM remove_due_to_license_issue P10844 12146945 1292 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1g9a A 2.1 BS03 BAB A 2 N203 R217 D375 L377 D452 F537 L540 E716 K720 Y724 N203 R217 D375 L377 D449 F534 L537 E713 K717 Y721 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 ic50~7.5uM remove_due_to_license_issue P10844 12146945 1293 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1g9b A 2.0 BS02 BAB A 1 D68 Q258 R369 Y372 F373 S374 D375 S376 E451 L453 F454 F455 T709 Q710 Y712 T713 D68 Q258 R369 Y372 F373 S374 D375 S376 E448 L450 F451 F452 T706 Q707 Y709 T710 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 ic50~7.5uM remove_due_to_license_issue P10844 12146945 1292 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1g9b A 2.0 BS03 BAB A 2 N203 R217 D375 L377 D452 F537 L540 E716 K720 Y724 N203 R217 D375 L377 D449 F534 L537 E713 K717 Y721 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 ic50~7.5uM remove_due_to_license_issue P10844 12146945 1293 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1g9c A 2.35 BS02 BAB A 1 D68 Q258 R369 Y372 F373 S374 D375 S376 E451 F455 T709 Q710 T713 D68 Q258 R369 Y372 F373 S374 D375 S376 E448 F452 T706 Q707 T710 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 ic50~7.5uM remove_due_to_license_issue P10844 12146945 1292 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1g9c A 2.35 BS03 BAB A 2 N203 R217 D375 L377 D452 F537 L540 E716 K720 N203 R217 D375 L377 D449 F534 L537 E713 K717 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 ic50~7.5uM remove_due_to_license_issue P10844 12146945 1293 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1g9r A 2.0 BS02 UPF A 1 A6 A7 D8 Y11 H78 I79 S80 T83 R86 D103 I104 D105 N153 A154 Q187 D188 Q189 H244 C246 G247 K250 A6 A7 D8 Y11 H78 I79 S80 T83 R86 D103 I104 D105 N153 A154 Q187 D188 Q189 H240 C242 G243 K246 H78 D103 D105 D130 D188 Q189 H244 K250 H78 D103 D105 D130 D188 Q189 H240 K246 2.4.1.- 0016757,0046872 Ki=2uM remove_due_to_license_issue Q93EK7 11175908 401 MDIVFAADDNYAAYLCVAAKSVEAAHPDTEIRFHVLDAGISEANRAAVAANLRGGGGNIRFIDVNPEDFAGFPLNIRHISITTYARLKLGEYIADCDKVLYLDIDVLVRDSLTPLWDTDLGDNWLGASIDLFVERQEGYKQKIGMADGEYYFNAGVLLINLKKWRRHDIFKMSSEWVEQYKDVMQYQDQDILNGLFKGGVCYANSRFNFMPTNYAFMASRHTDPLYRDRTNTVMPVAVSHYCGPAKPWHRDCTAWGAERFTELAGSLTTVPEEWRGKL 1g9s A 2.8 BS01 IMP A 1 E103 I105 D107 S108 G109 N110 T111 L112 F156 E91 I93 D95 S96 G97 N98 T99 L100 F144 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 12070315 190 MKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSRDLKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILLD 1g9t A 2.8 BS01 5GP A 1 E103 D107 S108 G109 T111 L112 F156 V157 I162 E90 D94 S95 G96 T98 L99 F143 V144 I149 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 12070315 190 MKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASRDLKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILL 1ga9 A 2.1 BS01 ETP A 1 S64 Y150 N152 Y221 G317 A318 T319 N343 S61 Y147 N149 Y218 G314 A315 T316 N340 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=80nM P00811 11410378 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1gaf H 1.95 BS01 NPE H 1 Y33 H35 Y100 G101 Y33 H35 Y100 G101 ? Kd=10nM remove_due_to_license_issue P01857 8599084 218 QVQLQQSGAELVKPGASVKLSCTASGFNIKDTYMHWVKQRPKQGLEWIGRIDPANVDTKYDPKFQDKATITADTSSKTTYLQLSSLTSEDTAVYYCASYYGIYWGQGTTLTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 1gaf L 1.95 BS01 NPE H 1 R46 Y91 R96 R46 Y91 R96 ? 0002250,0003823,0005576,0005615,0005886,0006955,0016064,0019814,0050853,0070062,0071735,0071738,0071742,0071745,0071753,0072562 remove_due_to_license_issue P01834 8599084 218 DIQMTQSPSSLSASLGERVSLTCRASQEINGYLGWLQQKPDGTIKRLIYAASTLHSGVPKRFSGSRSGSDYSLTISSLESEDFADYYCLQYASYPRTFGGGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 1gar A 1.96 BS01 U89 A 1 N10 G11 S12 N13 R64 G87 M89 R90 I91 L92 N106 I107 H108 P109 L143 D144 E173 N10 G11 S12 N13 R64 G87 M89 R90 I91 L92 N106 I107 H108 P109 L138 D139 E168 N106 H108 S135 D144 N106 H108 S130 D139 2.1.2.2 0003824,0004644,0005737,0005829,0006164,0006189,0006974,0009058,0016740 Ki=100pM remove_due_to_license_issue P08179 7776369 213 MNIVVLISGNGSNLQAIIDACKTNKIKGTVRAVFSNKADAFGLERARQAGIATHTLIASAFDSREAYDRELIHEIDMYAPDVVVLAGFMRILSPAFVSHYAGRLLNIHPSLLPKYPGLHTHNGDEEHGTSVHFVTDELDGGPVILQAKVPVFAGDSEDDITARVQTQEHAIYPLVISWFADGRLKMHENAAWLDGQRLPPQGYA 1gbt A 2.0 BS02 GBS A 1 D189 S190 C191 Q192 S195 S214 W215 G216 G219 D171 S172 C173 Q174 S177 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 2252895 704 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1gca A 1.7 BS01 GAL A 1 D14 F16 N91 K92 H152 D154 R158 N211 D236 N256 D14 F16 N91 K92 H152 D154 R158 N211 D236 N256 ? 0006935,0030246,0030288,0042597,0046872 Kd=0.2uM remove_due_to_license_issue P23905 8240551 350 ADTRIGVTIYKYDDNFMSVVRKAIEKDGKSAPDVQLLMNDSQNDQSKQNDQIDVLLAKGVKALAINLVDPAAAGTVIEKARGQNVPVVFFNKEPSRKALDSYDKAYYVGTDSKESGVIQGDLIAKHWQANQGWDLNKDGKIQYVLLKGEPGHPDAEARTTYVVKELNDKGIQTEQLALDTAMWDTAQAKDKMDAWLSGPNANKIEVVIANNDAMAMGAVEALKAHNKSSIPVFGVDALPEALALVKSGAMAGTVLNDANNQAKATFDLAKNLAEGKGAADGTSWKIENKIVRVPYVGVDKDNLSEFTQK 1gcz A 1.9 BS01 YZ9 A 1 P1 K32 Y36 H62 S63 I64 V106 P1 K32 Y36 H62 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=7.4uM remove_due_to_license_issue Ki=7400nM P14174 11170644 900 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFALEHH 1gcz A 1.9 BS02 YZ9 B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=7.4uM remove_due_to_license_issue Ki=7400nM P14174 11170644 902 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFALEHH 1gcz C 1.9 BS01 YZ9 A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=7.4uM remove_due_to_license_issue Ki=7400nM P14174 11170644 900 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFALEHH 1gcz C 1.9 BS02 YZ9 C 1 P1 M2 K32 H62 S63 I64 V106 F113 P1 M2 K32 H62 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=7.4uM remove_due_to_license_issue Ki=7400nM P14174 11170644 901 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFALEHH 1gfw A 2.8 BS01 MSI A 1 M61 H121 G122 C163 M33 H93 G94 C135 T62 S63 H121 G122 C163 R164 T34 S35 H93 G94 C135 R136 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue Ki=15nM, IC50=114nM, EC50=7670nM P42574 10821855 1 SGISLDNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 1gfw B 2.8 BS01 MSI A 1 Y204 W206 R207 F256 Y20 W22 R23 F72 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue Ki=15nM, IC50=114nM, EC50=7670nM P42574 10821855 1 HKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH 1gfy A 2.13 BS01 COL A 1 Y46 N48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y44 N46 K118 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=8317.64nM P18031 10748206 301 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYVNVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRCQLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1gfz A 2.3 BS03 CFF A 1 F285 H571 G612 Y613 F269 H548 G589 Y590 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki~0.15mM remove_due_to_license_issue IC50=114000nM P00489 10924512 940 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1ggd B 1.5 BS02 FAF C 1 H57 I99 H42 I84 H57 D102 H42 D87 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 11327865 301 IVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGVTTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKYNSLTINNDITLLKLSTAASFSQTVSAVCLPSASDDFAAGTTCVTTGWGLTRY 1ggd C 1.5 BS02 FAF C 1 S190 C191 M192 S195 S214 W215 G216 S217 S40 C41 M42 S45 S64 W65 G66 S67 M192 G193 D194 S195 G196 M42 G43 D44 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 11327865 301 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 1ggn A 2.36 BS01 GLS A 1 G135 L136 N284 H377 N484 E672 G675 G123 L124 N272 H365 N472 E660 G663 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=3.1uM remove_due_to_license_issue Ki=3100nM, IC50=3100nM P00489 11741774 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1ghv H 1.85 BS02 120 H 1 H57 D189 A190 E192 S195 V213 H43 D192 A193 E195 S198 V218 3.4.21.5 0004252,0005509,0006508,0007596 Ki=45uM remove_due_to_license_issue P00734 11292354 246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1ghw H 1.75 BS02 BMZ H 1 H57 W60D D189 A190 E192 S195 V213 H43 W50 D192 A193 E195 S198 V218 3.4.21.5 0004252,0005509,0006508,0007596 Ki=4uM remove_due_to_license_issue P00734 11292354 246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1ghy H 1.85 BS03 121 H 1 H57 W60D D189 A190 C191 E192 S195 S214 G216 G219 H43 W50 D192 A193 C194 E195 S198 S219 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.008uM remove_due_to_license_issue P00734 11292354 246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1ghz A 1.39 BS03 120 A 1 H57 D189 S190 S195 V213 G219 H40 D171 S172 S177 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=16uM remove_due_to_license_issue P00760 11292354 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1gi1 A 1.42 BS02 BMZ A 1 H57 D189 S190 C191 S195 V213 G216 H40 D171 S172 C173 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=3.6uM remove_due_to_license_issue P00760 11292354 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1gi4 A 1.37 BS03 122 A 1 H57 D189 S190 C191 Q192 S195 V213 S214 W215 G219 H40 D171 S172 C173 Q174 S177 V191 S192 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.065uM remove_due_to_license_issue Ki=3600nM P00760 11292354 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1gi6 A 1.49 BS02 124 A 1 H57 D189 S190 C191 Q192 S195 V213 H40 D171 S172 C173 Q174 S177 V191 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.7uM remove_due_to_license_issue Ki=1700nM P00760 11292354 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1gi7 B 1.79 BS02 120 B 1 D189 S190 C191 Q192 G219 D192 S193 C194 Q195 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=31uM remove_due_to_license_issue P00749 11292354 246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1gi8 B 1.75 BS02 BMZ B 1 H57 S190 C191 Q192 S195 V213 W215 G216 H46 S193 C194 Q195 S198 V216 W218 G219 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 11292354 246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1gi9 B 1.8 BS02 123 B 1 H57 S190 C191 Q192 S195 V213 W215 G216 H46 S193 C194 Q195 S198 V216 W218 G219 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=1.1uM remove_due_to_license_issue P00749 11292354 246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1gj4 H 1.81 BS03 132 H 1 H57 W60D K60F D189 A190 E192 S195 V213 W215 G219 H43 W50 K52 D192 A193 E195 S198 V218 W220 G223 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=60000nM P00734 11731301 410 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1gj5 H 1.73 BS02 130 H 1 C42 H57 C58 W60D D189 A190 E192 S195 V213 C28 H43 C44 W50 D192 A193 E195 S198 V218 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 11731301 410 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1gj6 A 1.5 BS02 132 A 1 H57 D189 S190 Q192 S195 V213 S214 W215 G219 G226 V227 Y228 H40 D171 S172 Q174 S177 V191 S192 W193 G196 G204 V205 Y206 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.23uM remove_due_to_license_issue Ki=100nM P00760 11731301 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1gj7 B 1.5 BS02 132 B 1 H57 D189 S190 Q192 S195 V213 S214 W215 G219 C220 G226 V227 H46 D192 S193 Q195 S198 V216 S217 W218 G221 C222 G229 V230 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.009uM remove_due_to_license_issue Ki=14nM P00749 11731301 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 1gj8 B 1.64 BS02 133 B 1 V41 H57 C58 S190 C191 Q192 S195 V213 G219 V30 H46 C47 S193 C194 Q195 S198 V216 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.11uM remove_due_to_license_issue P00749 11731301 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1gja B 1.56 BS02 135 B 1 H57 D189 S190 C191 Q192 G193 S195 G219 C220 H46 D192 S193 C194 Q195 G196 S198 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=3.8uM remove_due_to_license_issue Ki=2700nM P00749 11731301 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1gjb B 1.9 BS02 130 B 1 H57 S190 C191 Q192 S195 V213 W215 H46 S193 C194 Q195 S198 V216 W218 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.45uM remove_due_to_license_issue P00749 11731301 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 1gjc B 1.73 BS02 130 B 1 H57 S190 C191 Q192 S195 V213 W215 G219 H46 S193 C194 Q195 S198 V216 W218 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.45uM remove_due_to_license_issue P00749 11731301 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 1gjd B 1.75 BS02 136 B 1 D189 S190 C191 Q192 G193 S195 W215 G216 G219 C220 G226 D192 S193 C194 Q195 G196 S198 W218 G219 G221 C222 G229 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=6uM remove_due_to_license_issue Ki=6000nM P00749 11731301 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1gji A 2.85 BS01 dna C 0 Y24 C26 K110 K111 R178 P180 Q211 K212 Q238 Y18 C20 K104 K105 R172 P174 Q205 K206 Q232 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P16236 11587641 1 ~ 20 PYIEIFEQPRQRGMRFRYKCEGRSAGSIPGEHSTDNNKTFPSIQILNYFGKVKIRTTLVTKNEPYKPHPHDLVGKDCRDGYYEAEFGPERRVLSFQNLGIQCVKKKDLKESISLRISKKINPFNVPEEQLHNIDEYDLNVVRLCFQAFLPDEHGNYTLALPPLISNPIYDNRAPNTAELRICRVNKNCGSVKGGDEIFILCDKVQKDDIEVRFVLDNWEAKGSFSQADVHRQVAIVFRTPPFLRDITEPITVKMQLRRPSDQEVSEPMDFRYLPD 1gji A 2.85 BS02 dna D 0 R21 R23 S30 R15 R17 S24 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P16236 11587641 301 ~ 320 PYIEIFEQPRQRGMRFRYKCEGRSAGSIPGEHSTDNNKTFPSIQILNYFGKVKIRTTLVTKNEPYKPHPHDLVGKDCRDGYYEAEFGPERRVLSFQNLGIQCVKKKDLKESISLRISKKINPFNVPEEQLHNIDEYDLNVVRLCFQAFLPDEHGNYTLALPPLISNPIYDNRAPNTAELRICRVNKNCGSVKGGDEIFILCDKVQKDDIEVRFVLDNWEAKGSFSQADVHRQVAIVFRTPPFLRDITEPITVKMQLRRPSDQEVSEPMDFRYLPD 1gji B 2.85 BS01 dna C 0 R21 S30 G32 R15 S24 G26 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P16236 11587641 1 ~ 20 PYIEIFEQPRQRGMRFRYKCEGRSAGSIPGEHSTDNNKTFPSIQILNYFGKVKIRTTLVTKNEPYKPHPHDLVGKDCRDGYYEAEFGPERRVLSFQNLGIQCVKKKDLKESISLRISKKINPFNVPEEQLHNIDEYDLNVVRLCFQAFLPDEHGNYTLALPPLISNPIYDNRAPNTAELRICRVNKNCGSVKGGDEIFILCDKVQKDDIEVRFVLDNWEAKGSFSQADVHRQVAIVFRTPPFLRDITEPITVKMQLRRPSDQEVSEPMDFRYLPD 1gji B 2.85 BS02 dna D 0 Y24 C26 E27 K110 K111 K212 R237 Q238 Y18 C20 E21 K104 K105 K206 R231 Q232 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P16236 11587641 301 ~ 320 PYIEIFEQPRQRGMRFRYKCEGRSAGSIPGEHSTDNNKTFPSIQILNYFGKVKIRTTLVTKNEPYKPHPHDLVGKDCRDGYYEAEFGPERRVLSFQNLGIQCVKKKDLKESISLRISKKINPFNVPEEQLHNIDEYDLNVVRLCFQAFLPDEHGNYTLALPPLISNPIYDNRAPNTAELRICRVNKNCGSVKGGDEIFILCDKVQKDDIEVRFVLDNWEAKGSFSQADVHRQVAIVFRTPPFLRDITEPITVKMQLRRPSDQEVSEPMDFRYLPD 1gni A 2.4 BS01 OLA A 1 R117 Y138 F157 A158 Y161 G189 R115 Y136 F155 A156 Y159 G187 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=8.5nM remove_due_to_license_issue P02768 11743713 1001 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gni A 2.4 BS02 OLA A 2 V46 Y150 A254 R257 S287 V44 Y148 A252 R255 S285 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=8.5nM remove_due_to_license_issue P02768 11743713 1002 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gni A 2.4 BS03 OLA A 3 S342 R348 I388 C392 G434 R485 S340 R346 I386 C390 G432 R483 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=8.5nM remove_due_to_license_issue P02768 11743713 1003 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gni A 2.4 BS04 OLA A 4 Y411 V418 S419 T422 L460 L463 F488 S489 Y409 V416 S417 T420 L458 L461 F486 S487 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=8.5nM remove_due_to_license_issue P02768 11743713 1004 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gni A 2.4 BS05 OLA A 5 Y401 K525 H535 M548 F551 Q580 Y399 K523 H533 M546 F549 Q578 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=8.5nM remove_due_to_license_issue P02768 11743713 1005 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS01 ACD A 1 R117 M123 Y138 F157 Y161 R115 M121 Y136 F155 Y159 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1001 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS02 ACD A 2 V46 F70 Y150 L251 A254 R257 L283 S287 V44 F68 Y148 L249 A252 R255 L281 S285 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1002 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS03 ACD A 3 V344 R348 L387 I388 N391 Y411 R485 V342 R346 L385 I386 N389 Y409 R483 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1003 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS04 ACD A 4 Y411 V415 V418 L430 L457 H464 F488 S489 Y409 V413 V416 L428 L455 H462 F486 S487 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1004 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS05 ACD A 5 Y401 F507 K525 A528 H535 M548 F551 S579 Q580 Y399 F505 K523 A526 H533 M546 F549 S577 Q578 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1005 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS06 ACD A 6 A213 D324 A211 D322 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1006 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS07 ACD A 7 L260 I290 L258 I288 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1007 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnj A 2.6 BS08 ACD A 8 S419 T422 T467 S417 T420 T465 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 11743713 1008 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1gnm A 2.3 BS01 U0E A 1 R8 D25 G27 D82 I84 R8 D25 G27 D82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=560nM remove_due_to_license_issue P03366 8718851 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPDNIIGRNLLTQIGCTLNF 1gnm A 2.3 BS02 U0E A 2 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 I84 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=560nM remove_due_to_license_issue P03366 8718851 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPDNIIGRNLLTQIGCTLNF 1gnm B 2.3 BS01 U0E A 1 D25 G27 A28 D29 D30 I47 G48 I50 P81 D82 D25 G27 A28 D29 D30 I47 G48 I50 P81 D82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8718851 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPDNIIGRNLLTQIGCTLNF 1gnm B 2.3 BS02 U0E A 2 D25 G27 I50 D25 G27 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8718851 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPDNIIGRNLLTQIGCTLNF 1gnn A 2.3 BS01 U0E A 1 R8 D25 G27 G49 I50 N82 I84 R8 D25 G27 G49 I50 N82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2100nM remove_due_to_license_issue P03366 8718851 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPNNIIGRNLLTQIGCTLNF 1gnn A 2.3 BS02 U0E A 2 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 N82 I84 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 N82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2100nM remove_due_to_license_issue P03366 8718851 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPNNIIGRNLLTQIGCTLNF 1gnn B 2.3 BS01 U0E A 1 D25 G27 A28 D29 D30 I47 G48 I50 P81 N82 D25 G27 A28 D29 D30 I47 G48 I50 P81 N82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8718851 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPNNIIGRNLLTQIGCTLNF 1gnn B 2.3 BS02 U0E A 2 D25 G27 G49 D25 G27 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8718851 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPNNIIGRNLLTQIGCTLNF 1gno A 2.3 BS01 U0E B 1 R8 D25 G27 G49 R8 D25 G27 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8718851 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1gno A 2.3 BS02 U0E B 2 D25 G27 A28 D29 D30 I47 G48 G49 P81 V82 D25 G27 A28 D29 D30 I47 G48 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8718851 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1gno B 2.3 BS01 U0E B 1 D25 G27 A28 D29 D30 I47 G48 P81 V82 D25 G27 A28 D29 D30 I47 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P03366 8718851 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1gno B 2.3 BS02 U0E B 2 D25 G27 D25 G27 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P03366 8718851 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1gpk A 2.1 BS01 HUP A 1 W84 G118 S122 G123 Y130 F330 F331 H440 W81 G115 S119 G120 Y127 F327 F328 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=4.3uM remove_due_to_license_issue IC50=11.4nM P04058 12196020 1540 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1gpn A 2.35 BS01 HUB A 1 W84 G117 G118 G119 Y121 Y130 H440 W81 G114 G115 G116 Y118 Y127 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=0.334uM remove_due_to_license_issue Ki=334nM P04058 12196020 1538 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1gpy A 2.4 BS01 G6P A 1 I68 R193 D227 R242 R309 R310 I55 R180 D214 R229 R296 R297 H377 K568 R569 K574 T676 K680 H364 K555 R556 K561 T663 K667 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Kd~25uM remove_due_to_license_issue P00489 8331662 998 SVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKI 1gqs A 3.0 BS01 SAF A 1 W84 G118 G119 E199 F290 F331 W81 G115 G116 E196 F287 F328 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue Ki=700nM P04058 11888271 603 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1gsf A 2.7 BS01 EAA A 1 Y9 F10 R15 V55 L107 V111 M208 F220 F222 Y8 F9 R14 V54 L106 V110 M207 F219 F221 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 remove_due_to_license_issue IC50=5000nM P08263 8591048 223 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1gsz A 2.8 BS01 R71 A 1 W169 A170 I261 P263 W312 F365 D376 W489 F601 F605 W160 A161 I252 P254 W303 F356 D367 W480 F592 F596 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12031670 1630 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1gt1 A 1.71 BS02 ANC A 1 T38 F56 N103 T116 T37 F55 N102 T115 ? 0005549,0005576,0005615,0007608,0036094 Kd=1uM remove_due_to_license_issue P07435 15373829 1161 QEEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPHPE 1gt1 B 1.71 BS01 ANC B 1 F89 N103 T116 E117 F119 F87 N101 T114 E115 F117 ? 0005549,0005576,0005615,0007608,0036094 Kd=1uM remove_due_to_license_issue P07435 15373829 1158 EEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPH 1gt3 A 1.8 BS01 DHM A 1 F54 V69 N87 F54 V69 N87 ? 0005549,0005576,0005615,0007608,0036094 Kd=0.35uM remove_due_to_license_issue P07435 15373829 1160 AQEEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPHPE 1gt3 B 1.8 BS01 DHM B 1 N87 N103 N85 N101 ? 0005549,0005576,0005615,0007608,0036094 Kd=0.35uM remove_due_to_license_issue P07435 15373829 1159 EEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPH 1gt4 A 2.1 BS01 UNA A 1 F36 F56 V69 Y83 N87 N103 F36 F56 V69 Y83 N87 N103 ? 0005549,0005576,0005615,0007608,0036094 Kd=0.3uM remove_due_to_license_issue P07435 15373829 1160 AQEEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPHPE 1gt4 B 2.1 BS01 UNA B 1 N87 F89 N103 N85 F87 N101 ? 0005549,0005576,0005615,0007608,0036094 Kd=0.3uM remove_due_to_license_issue P07435 15373829 1158 EEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPH 1gt5 B 2.08 BS01 BZQ B 1 F36 F89 N103 T116 E117 F34 F87 N101 T114 E115 ? 0005549,0005576,0005615,0007608,0036094 Kd=0.8uM remove_due_to_license_issue P07435 15373829 1158 EEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPH 1gu1 A 1.8 BS01 FA1 A 1 Y28 N79 A81 A82 H85 H106 I107 S108 R117 Y27 N78 A80 A81 H84 H105 I106 S107 R116 P15 N16 R23 Y28 N79 A82 E104 H106 R113 P14 N15 R22 Y27 N78 A81 E103 H105 R112 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=30uM remove_due_to_license_issue Kd=30000nM P15474 11937054 201 RSLANAPIMILNGPNLNLLGQRQPEIYGSDTLADVEALCVKAAAAHGGTVDFRQSNHEGELVDWIHEARLNHCGIVINPAAYSHTSVAILDALNTCDGLPVVEVHISNIHQREPFRHHSYVSQRADGVVAGCGVQGYVFGVERIAALAG 1gu1 B 1.8 BS01 FA1 B 1 Y28 N79 A81 A82 H85 H106 I107 S108 R117 Y27 N78 A80 A81 H84 H105 I106 S107 R116 P15 N16 R23 Y28 N79 A82 E104 H106 R113 P14 N15 R22 Y27 N78 A81 E103 H105 R112 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=30uM remove_due_to_license_issue Kd=30000nM P15474 11937054 201 RSLANAPIMILNGPNLNLLGQRQPEIYGSDTLADVEALCVKAAAAHGGTVDFRQSNHEGELVDWIHEARLNHCGIVINPAAYSHTSVAILDALNTCDGLPVVEVHISNIHQREPFRHHSYVSQRADGVVAGCGVQGYVFGVERIAALAG 1gvw A 1.0 BS01 0EM A 1 D15 D35 Y79 G80 D81 F194 D219 G221 T222 T223 F280 I304 D15 D35 Y77 G78 D79 F192 D217 G219 T220 T221 F278 I302 D35 S38 D40 W42 G80 T220 T223 D35 S38 D40 W42 G78 T218 T221 3.4.23.22 0004190,0006508 Ki=110nM remove_due_to_license_issue P11838 12083527 401 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 1gww A 1.8 BS01 UDP A 1 F134 A135 V136 Y139 I198 R202 D225 V226 D227 K359 Y361 R365 F53 A54 V55 Y58 I117 R121 D144 V145 D146 K278 Y280 R284 Q247 H280 W314 E317 W356 R365 Q166 H199 W233 E236 W275 R284 2.4.1.87 0005975,0016020,0016758 remove_due_to_license_issue P14769 12011052 1369 KLKLSDWFNPFKRPEVVTMTKWKAPVVWEGTYNRAVLDNYYAKQKITVGLTVFAVGRYIEHYLEEFLTSANKHFMVGHPVIFYIMVDDVSRMPLIELGPLRSFKVFKIKPEKRWQDISMMRMKTIGEHIVAHIQHEVDFLFCMDVDQVFQDKFGVETLGESVAQLQAWWYKADPNDFTYERRKESAAYIPFGEGDFYYHAAIFGGTPTQVLNITQECFKGILKDKKNDIEAQWHDESHLNKYFLLNKPTKILSPEYCWDYHIGLPADIKLVKMSWQTKEYNVVRNNV 1gx0 A 1.8 BS01 UDP A 1 F134 A135 V136 Y139 I198 R202 D225 V226 D227 K359 Y361 R365 F53 A54 V55 Y58 I117 R121 D144 V145 D146 K278 Y280 R284 Q247 H280 W314 E317 W356 R365 Q166 H199 W233 E236 W275 R284 2.4.1.87 0005975,0016020,0016758 remove_due_to_license_issue P14769 12011052 1369 KLKLSDWFNPFKRPEVVTMTKWKAPVVWEGTYNRAVLDNYYAKQKITVGLTVFAVGRYIEHYLEEFLTSANKHFMVGHPVIFYIMVDDVSRMPLIELGPLRSFKVFKIKPEKRWQDISMMRMKTIGEHIVAHIQHEVDFLFCMDVDQVFQDKFGVETLGESVAQLQAWWYKADPNDFTYERRKESAAYIPFGEGDFYYHAAIFGGTPTQVLNITQECFKGILKDKKNDIEAQWHDESHLNKYFLLNKPTKILSPEYCWDYHIGLPADIKLVKMSWQTKEYNVVRNNV 1gx4 A 1.46 BS02 UDP A 1 F134 A135 V136 Y139 I198 R202 D225 V226 D227 K359 Y361 R365 F53 A54 V55 Y58 I117 R121 D144 V145 D146 K278 Y280 R284 Q247 H280 W314 E317 W356 R365 Q166 H199 W233 E236 W275 R284 2.4.1.87 0005975,0016020,0016758 Kd=0.053mM remove_due_to_license_issue P14769 12011052 401 KLKLSDWFNPFKRPEVVTMTKWKAPVVWEGTYNRAVLDNYYAKQKITVGLTVFAVGRYIEHYLEEFLTSANKHFMVGHPVIFYIMVDDVSRMPLIELGPLRSFKVFKIKPEKRWQDISMMRMKTIGEHIVAHIQHEVDFLFCMDVDQVFQDKFGVETLGESVAQLQAWWYKADPNDFTYERRKESAAYIPFGEGDFYYHAAIFGGTPTQVLNITQECFKGILKDKKNDIEAQWHDESHLNKYFLLNKPTKILSPEYCWDYHIGLPADIKLVKMSWQTKEYNVVRNNV 1gx8 A 2.4 BS01 RTL A 1 L39 E62 K69 I71 F105 M107 L38 E61 K68 I70 F104 M106 ? 0005515,0005576,0019841,0036041,0036094,0042802 remove_due_to_license_issue Kd=36nM P02754 12054801 1163 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 1gym A 2.2 BS01 MYG A 1 H32 R69 K115 R163 D198 Y200 H32 R69 K115 R163 D198 Y200 H32 D33 R69 H82 D274 H32 D33 R69 H82 D274 4.6.1.13 0004436,0005576,0006629,0008081,0016042,0016829 ic50=2mM remove_due_to_license_issue P14262 8755729 702 ASSVNELENWSKWMQPIPDSIPLARISIPGTHDSGTFKLQNPIKQVWGMTQEYDFRYQMDHGARIFDIRGRLTDDNTIVLHHGPLYLYVTLHEFINEAKQFLKDNPSETIIMSLKKEYEDMKGAEDSFSSTFEKKYFVDPIFLKTEGNIKLGDARGKIVLLKRYSGSNEPGGYNNFYWPDNETFTTTVNQNANVTVQDKYKVSYDEKVKSIKDTMDETMNNSEDLNHLYINFTSLSSGGTAWNSPYYYASYINPEIANYIKQKNPARVGWVIQDYINEKWSPLLYQEVIRANKSLI 1gyy A 1.35 BS01 FHC A 1 P1 S38 P1 S38 5.3.2.- 0005737,0016853,0016862,0042803 Ki=230uM remove_due_to_license_issue P31992 12356301 500 PHIDIKCFPRELDEQQKAALAADITDVIIRHLNSKDSSISIALQQIQPESWQAIWDAEIAPQMEALIKKPGYSMNA 1gyy A 1.35 BS02 FHC B 1 C7 F8 W51 Y72 C7 F8 W51 Y72 5.3.2.- 0005737,0016853,0016862,0042803 Ki=230uM remove_due_to_license_issue P31992 12356301 500 PHIDIKCFPRELDEQQKAALAADITDVIIRHLNSKDSSISIALQQIQPESWQAIWDAEIAPQMEALIKKPGYSMNA 1gyy B 1.35 BS01 FHC A 1 C7 F8 W51 Y72 C7 F8 W51 Y72 5.3.2.- 0005737,0016853,0016862,0042803 Ki=230uM remove_due_to_license_issue P31992 12356301 500 PHIDIKCFPRELDEQQKAALAADITDVIIRHLNSKDSSISIALQQIQPESWQAIWDAEIAPQMEALIKKPGYSMNA 1gyy B 1.35 BS02 FHC B 1 P1 S38 P1 S38 5.3.2.- 0005737,0016853,0016862,0042803 Ki=230uM remove_due_to_license_issue P31992 12356301 500 PHIDIKCFPRELDEQQKAALAADITDVIIRHLNSKDSSISIALQQIQPESWQAIWDAEIAPQMEALIKKPGYSMNA 1gz3 A 2.3 BS01 ATP A 1 R165 N259 A312 G313 E314 A315 D345 K346 V392 A393 G394 L398 R146 N240 A293 G294 E295 A296 D326 K327 V373 A374 G375 L379 Y112 R165 K183 E255 D256 D278 D279 N421 Y93 R146 K164 E236 D237 D259 D260 N402 1.1.1.38 0004470,0004471,0004473,0005739,0005759,0006090,0006108,0008948,0009055,0016491,0016616,0043231,0046872,0051287,1902031 Ki=0.2mM remove_due_to_license_issue P23368 12121650 601 HIKEKGKPLMLNPRTNKGMAFTLQERQMLGLQGLLPPKIETQDIQALRFHRNLKKMTSPLEKYIYIMGIQERNEKLFYRILQDDIESLMPIVYTPTVGLACSQYGHIFRRPKGLFISISDRGHVRSIVDNWPENHVKAVVVTDGERILGLGDLGVYGMGIPVGKLCLYTACAGIRPDQCLPVCIDVGTDNIALLKDPFYMGLYQKRDRTQQYDDLIDEFMKAITDRYGRNTLIQFEDFGNHNAFRFLRKYREKYCTFNDDIQGTAAVALAGLLAAQKVISKPISEHKILFLGAGEAALGIANLIVMSMVENGLSEQEAQKKIWMFDKYGLLVKGRKAKIDSYQEPFTHSAPESIPDTFEDAVNILKPSTIIGVAGAGRLFTPDVIRAMASINERPVIFALSNPTAQAECTAEEAYTLTEGRCLFASGSPFGPVKLTDGRVFTPGQGNNVYIFPGVALAVILCNTRHISDSVFLEAAKALTSQLTDEELAQGRLYPPLANIQEVSINIAIKVTEYLYANKMAFVYPEPEDKAKYVKEQTWRSEYDSLLPDVYEWP 1gz4 A 2.2 BS01 ATP A 1 R165 N259 G311 A312 G313 E314 A315 D345 K346 V392 A393 R143 N237 G289 A290 G291 E292 A293 D323 K324 V370 A371 Y112 R165 K183 E255 D256 D278 D279 N421 Y90 R143 K161 E233 D234 D256 D257 N399 1.1.1.38 0004470,0004471,0004473,0005739,0005759,0006090,0006108,0008948,0009055,0016491,0016616,0043231,0046872,0051287,1902031 Ki=0.2mM remove_due_to_license_issue P23368 12121650 601 EKGKPLMLNPRTNKGMAFTLQERQMLGLQGLLPPKIETQDIQALRFHRNLKKMTSPLEKYIYIMGIQERNEKLFYRILQDDIESLMPIVYTPTVGLACSQYGHIFRRPKGLFISISDRGHVRSIVDNWPENHVKAVVVTDGERILGLGDLGVYGMGIPVGKLCLYTACAGIRPDRCLPVCIDVGTDNIALLKDPFYMGLYQKRDRTQQYDDLIDEFMKAITDRYGRNTLIQFEDFGNHNAFRFLRKYREKYCTFNDDIQGTAAVALAGLLAAQKVISKPISEHKILFLGAGEAALGIANLIVMSMVENGLSEQEAQKKIWMFDKYGLLVKGRKAKIDSYQEPFTHSAPESIPDTFEDAVNILKPSTIIGVAGAGRLFTPDVIRAMASINERPVIFALSNPTAQAECTAEEAYTLTEGRCLFASGSPFGPVKLTDGRVFTPGQGNNVYIFPGVALAVILCNTRHISDSVFLEAAKALTSQLTDEELAQGRLYPPLANIQEVSINIAIKVTEYLYANKMAFRYPEPEDKAKYVKERTWRSEYDSLLPDVYEWP 1gz4 A 2.2 BS02 ATP A 2 H154 I193 R194 R197 I479 L480 R542 Y552 R556 H132 I171 R172 R175 I457 L458 R520 Y530 R534 Y112 R165 K183 E255 D256 D278 D279 N421 Y90 R143 K161 E233 D234 D256 D257 N399 1.1.1.38 0004470,0004471,0004473,0005739,0005759,0006090,0006108,0008948,0009055,0016491,0016616,0043231,0046872,0051287,1902031 Ki=0.2mM remove_due_to_license_issue P23368 12121650 602 EKGKPLMLNPRTNKGMAFTLQERQMLGLQGLLPPKIETQDIQALRFHRNLKKMTSPLEKYIYIMGIQERNEKLFYRILQDDIESLMPIVYTPTVGLACSQYGHIFRRPKGLFISISDRGHVRSIVDNWPENHVKAVVVTDGERILGLGDLGVYGMGIPVGKLCLYTACAGIRPDRCLPVCIDVGTDNIALLKDPFYMGLYQKRDRTQQYDDLIDEFMKAITDRYGRNTLIQFEDFGNHNAFRFLRKYREKYCTFNDDIQGTAAVALAGLLAAQKVISKPISEHKILFLGAGEAALGIANLIVMSMVENGLSEQEAQKKIWMFDKYGLLVKGRKAKIDSYQEPFTHSAPESIPDTFEDAVNILKPSTIIGVAGAGRLFTPDVIRAMASINERPVIFALSNPTAQAECTAEEAYTLTEGRCLFASGSPFGPVKLTDGRVFTPGQGNNVYIFPGVALAVILCNTRHISDSVFLEAAKALTSQLTDEELAQGRLYPPLANIQEVSINIAIKVTEYLYANKMAFRYPEPEDKAKYVKERTWRSEYDSLLPDVYEWP 1gzg B 1.66 BS01 LAF B 1 S175 K205 R215 K229 Q233 S171 K201 R211 K217 Q221 K205 K260 K201 K248 4.2.1.24 0004655,0005829,0006779,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue Q59643 12079382 1338 PANRAYPYTRLRRNRRDDFSRRLVRENVLTVDDLILPVFVLDGVNQRESIPSMPGVERLSIDQLLIEAEEWVALGIPALALFPVTPVEKKSLDAAEAYNPEGIAQRATRALRERFPELGIITDVALDPFTTHGQNGILDDDGYVLNDVSIDVLVRQALSHAEAGAQVVAPSDMMDGRIGAIREALESAGHTNVRVMAYSAKYASAYYGPFRDAVGSKATYQMDPANSDEALHEVAADLAEGADMVMVKPGMPYLDIVRRVKDEFRAPTFVYQVSGEYAMHMGAIQNGWLAESVILESLTAFKRAGADGILTYFAKQAAEQLRR 1gzg B 1.66 BS02 LAF B 2 Y211 F214 K260 Y283 V285 S286 Y324 Y207 F210 K248 Y271 V273 S274 Y312 K205 K260 K201 K248 4.2.1.24 0004655,0005829,0006779,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue Q59643 12079382 1337 PANRAYPYTRLRRNRRDDFSRRLVRENVLTVDDLILPVFVLDGVNQRESIPSMPGVERLSIDQLLIEAEEWVALGIPALALFPVTPVEKKSLDAAEAYNPEGIAQRATRALRERFPELGIITDVALDPFTTHGQNGILDDDGYVLNDVSIDVLVRQALSHAEAGAQVVAPSDMMDGRIGAIREALESAGHTNVRVMAYSAKYASAYYGPFRDAVGSKATYQMDPANSDEALHEVAADLAEGADMVMVKPGMPYLDIVRRVKDEFRAPTFVYQVSGEYAMHMGAIQNGWLAESVILESLTAFKRAGADGILTYFAKQAAEQLRR 1gzv A 3.51 BS01 PA5 A 1 I156 G157 G158 S209 K210 T211 T214 Q353 E357 K518 I156 G157 G158 S209 K210 T211 T214 Q353 E357 K518 K210 E216 G271 R272 E357 H388 K518 K210 E216 G271 R272 E357 H388 K518 5.3.1.9 0001701,0001707,0002639,0004347,0005125,0005576,0005615,0005737,0005829,0005886,0006002,0006094,0006096,0007165,0010595,0016853,0031625,0034101,0042593,0048029,0051156,0060170,0097367,0141199,1901135 remove_due_to_license_issue P08059 12402366 600 AALTQNPQFKKLQTWYHEHRSDLNLRRLFEGDKDRFNHFSLNLNTNHGRILLDYSKNLVTEAVMQMLVDLAKSRGVEAARERMFNGEKINFTEDRAVLHVALRNRSNTPILVDGKDVMPEVNRVLEKMKSFCKRVRSGEWKGYSGKSITDVINIGIGGSDLGPLMVTEALKPYSAEGPRVWFVSNIDGTHIAKTLATLNPESSLFIIASKTFTTQETITNAETAKEWFLQSAKDPSAVAKHFVALSTNTTKVKEFGIDPQNMFEFWDWVGGRYSLWSAIGLSIALHVGFDNFEQLLSGAHWMDQHFRTTPLEKNAPVLLALLGIWYINFFGCETHAMLPYDQYLHRFAAYFQQGDMESNGKYITKSGTRVDHQTGPIVWGEPGTNGQHAFYQLIHQGTKMIPCDFLIPVQTQHPIRKGLHHKILLANFLAQTEALMKGKSTEEARKELQAAGKSPEDFEKLLPHKVFEGNRPTNSIVFTKLTPFILGALIAMYEHKIFVQGVIWDINSFDQWGVELGKQLAKKIEPELDGSSPVTSHDSSTNGLINFIKQEREA 1h00 A 1.6 BS01 FAP A 1 I10 V18 A31 E81 F82 L83 K89 L134 D145 I10 V16 A29 E71 F72 L73 K79 L124 D135 D127 K129 Q131 N132 D145 T165 D117 K119 Q121 N122 D135 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=38uM remove_due_to_license_issue IC50=38000nM P24941 12941311 1300 MENFQKVEKIGEYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1h01 A 1.79 BS01 FAL A 1 I10 G11 V18 A31 L83 H84 L134 D145 I10 G11 V18 A31 L74 H75 L125 D136 D127 K129 Q131 N132 D145 T158 T165 D118 K120 Q122 N123 D136 T149 T156 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=22uM remove_due_to_license_issue IC50=1000nM P24941 12941311 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1h07 A 1.85 BS01 MFP A 1 I10 V18 A31 F80 E81 F82 L83 D86 K88 Q131 N132 L134 A144 D145 I10 V18 A31 F73 E74 F75 L76 D79 K81 Q124 N125 L127 A137 D138 D127 K129 Q131 N132 D145 T158 T165 D120 K122 Q124 N125 D138 T147 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=3uM remove_due_to_license_issue IC50=3000nM P24941 12941311 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1h08 A 1.8 BS01 BYP A 1 I10 V18 A31 F80 L83 D86 K89 L134 I10 V18 A31 F72 L75 D78 K81 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 12941311 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1h0a A 1.7 BS01 I3P A 1 R7 R8 K11 S29 N30 R63 K69 H73 R7 R8 K11 S29 N30 R63 K69 H73 ? Kd=3.6uM remove_due_to_license_issue O88339 12353027 1164 MSTSSLRRQMKNIVHNYSEAEIKVREATSNDPWGPSSSLMSEIADLTYNVVAFSEIMSMIWKRLNDHGKNWRHVYKAMTLMEYLIKTGSERVSQQCKENMYAVQTLKDFQYVDRDGKDQGVNVREKAKQLVALLRDEDRLREERAHALKTKEKLAQTA 1h0r A 2.1 BS01 FA1 A 1 Y24 N75 G77 G78 H81 H101 I102 S103 R112 Y19 N70 G72 G73 H76 H96 I97 S98 R107 P11 N12 Y24 N75 G78 E99 H101 R108 P10 N11 Y19 N70 G73 E94 H96 R103 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=200uM remove_due_to_license_issue Kd=200000nM, Ki=200000nM P9WPX7 200 ELIVNVINGPNLGRLGRVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEHV 1h0w A 2.1 BS01 207 A 1 I10 G11 A31 F82 L83 Q131 L134 I10 G11 A31 F75 L76 Q124 L127 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 12139449 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1h1b A 2.0 BS02 151 A 1 H57 L99B C191 F192 S195 S214 F215 V216 H41 L85 C169 F170 S173 S188 F189 V190 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G167 C169 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 remove_due_to_license_issue P08246 12190311 400 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 1h1b B 2.0 BS02 151 B 1 L99B C191 F192 S195 S214 F215 V216 L85 C169 F170 S173 S188 F189 V190 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G167 C169 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 remove_due_to_license_issue P08246 12190311 400 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 1h1d A 2.0 BS03 BIA A 1 W38 W143 K144 N170 P174 E199 W36 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=6nM remove_due_to_license_issue P22734 12237326 335 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 1h1h A 2.0 BS01 A2P A 1 Q14 K38 H128 Q15 K39 H129 K38 H128 L129 D130 K39 H129 L130 D131 3.1.27.- 0001530,0002227,0003676,0004519,0004540,0005576,0005615,0006401,0006935,0019731,0035578,0042742,0043152,0045087,0050829,0050830,0061844 Ki~6.5uM remove_due_to_license_issue P12724 12356310 1134 MRPPQFTRAQWFAIQHISLNPPRCTIAMRAINNYRWRCKNQNTFLRTTFANVVNVCGNQSIRCPHNRTLNNCHRSRFRVPLLHCDLINPGAQNISNCRYADRPGRRFYVVACDNRDPRDSPRYPVVPVHLDTTI 1h1p A 2.1 BS01 CMG A 1 E12 A31 E81 F82 L83 L134 E13 A32 E82 F83 L84 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=12uM remove_due_to_license_issue IC50=17000nM P24941 12244298 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1h1q A 2.5 BS01 2A6 A 1 I10 E12 A31 F80 E81 F82 L83 H84 Q85 Q131 L134 I11 E13 A32 F81 E82 F83 L84 H85 Q86 Q132 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1uM remove_due_to_license_issue IC50=2300nM P24941 12244298 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1h1r A 2.0 BS01 6CP A 1 I10 E12 A31 V64 F80 E81 F82 L83 H84 Q85 L134 I11 E13 A32 V65 F81 E82 F83 L84 H85 Q86 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=2.3uM remove_due_to_license_issue IC50=2300nM P24941 12244298 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1h1s A 2.0 BS01 4SP A 1 I10 E12 A31 V64 F80 E81 L83 H84 Q85 D86 K89 L134 I11 E13 A32 V65 F81 E82 L84 H85 Q86 D87 K90 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=6nM remove_due_to_license_issue IC50=6.0nM, Ki=6.0nM, Kd=1310nM P24941 12244298 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1h22 A 2.15 BS01 E10 A 1 Y70 W84 G118 G123 Y130 W279 I287 F288 F330 F331 Y334 G335 T535 Y67 W81 G115 G120 Y127 W276 I284 F285 F327 F328 Y331 G332 T528 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=0.8nM remove_due_to_license_issue Ki=0.8nM, IC50=2.4nM P04058 12517147 1536 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1h23 A 2.15 BS01 E12 A 1 Y70 W84 G117 G118 Y121 Y130 E199 W279 I287 F288 F330 F331 Y334 G335 Y67 W81 G114 G115 Y118 Y127 E196 W276 I284 F285 F327 F328 Y331 G332 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=4.5nM remove_due_to_license_issue Ki=4.5nM, IC50=16.0nM P04058 12517147 1536 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1h2t Z 2.1 BS01 GDP Z 1 Y20 R127 V134 Y138 Y16 R123 V130 Y134 ? 0000184,0000339,0000340,0000380,0000398,0002191,0003676,0003677,0003723,0003729,0005515,0005634,0005654,0005737,0005829,0005846,0006397,0006406,0006408,0006417,0006446,0008334,0008380,0016071,0017069,0031047,0031053,0031124,0031442,0032968,0034518,0035194,0035195,0042789,0045292,0046833,0051028 remove_due_to_license_issue P52298 12374755 1151 LLKALRSDSYVELSQYRDQHFRGDNEEQEKLLKKSCTLYVGNLSFYTTEEQIYELFSKSGDIKKIIMGLDKMKKTACGFCFVEYYSRADAENAMRYINGTRLDDRIIRTDWDAGFKEGRQYGRGRSGGQVRDEYRQDYDAGRGGYG 1h2t Z 2.1 BS02 7MG Z 1 Y20 D22 Y43 F83 R112 D114 R123 R127 Q133 V134 Y16 D18 Y39 F79 R108 D110 R119 R123 Q129 V130 ? 0000184,0000339,0000340,0000380,0000398,0002191,0003676,0003677,0003723,0003729,0005515,0005634,0005654,0005737,0005829,0005846,0006397,0006406,0006408,0006417,0006446,0008334,0008380,0016071,0017069,0031047,0031053,0031124,0031442,0032968,0034518,0035194,0035195,0042789,0045292,0046833,0051028 remove_due_to_license_issue P52298 12374755 1152 LLKALRSDSYVELSQYRDQHFRGDNEEQEKLLKKSCTLYVGNLSFYTTEEQIYELFSKSGDIKKIIMGLDKMKKTACGFCFVEYYSRADAENAMRYINGTRLDDRIIRTDWDAGFKEGRQYGRGRSGGQVRDEYRQDYDAGRGGYG 1h2u X 2.4 BS01 GDP X 1 Y20 R127 V134 Y17 R124 V131 ? 0000184,0000339,0000340,0000380,0000398,0002191,0003676,0003677,0003723,0003729,0005515,0005634,0005654,0005737,0005829,0005846,0006397,0006406,0006408,0006417,0006446,0008334,0008380,0016071,0017069,0031047,0031053,0031124,0031442,0032968,0034518,0035194,0035195,0042789,0045292,0046833,0051028 remove_due_to_license_issue P52298 12374755 1153 GLLKALRSDSYVELSQYRDQHFRGDNEEQEKLLKKSCTLYVGNLSFYTTEEQIYELFSKSGDIKKIIMGLDKMKKTACGFCFVEYYSRADAENAMRYINGTRLDDRIIRTDWDAGFKEGRQYGRGRSGGQVRDEYRQDYDAGRGGYGKL 1h2u X 2.4 BS02 7MG X 1 Y20 Y43 F83 D114 R123 G126 R127 Q133 V134 Y17 Y40 F80 D111 R120 G123 R124 Q130 V131 ? 0000184,0000339,0000340,0000380,0000398,0002191,0003676,0003677,0003723,0003729,0005515,0005634,0005654,0005737,0005829,0005846,0006397,0006406,0006408,0006417,0006446,0008334,0008380,0016071,0017069,0031047,0031053,0031124,0031442,0032968,0034518,0035194,0035195,0042789,0045292,0046833,0051028 remove_due_to_license_issue P52298 12374755 1154 GLLKALRSDSYVELSQYRDQHFRGDNEEQEKLLKKSCTLYVGNLSFYTTEEQIYELFSKSGDIKKIIMGLDKMKKTACGFCFVEYYSRADAENAMRYINGTRLDDRIIRTDWDAGFKEGRQYGRGRSGGQVRDEYRQDYDAGRGGYGKL 1h35 A 2.8 BS02 R01 A 1 F129 I261 P263 W312 F365 Y420 F601 F605 F120 I252 P254 W303 F356 Y411 F592 F596 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h36 A 2.8 BS02 R88 A 1 P263 A306 W312 F365 D374 D376 F437 W489 F605 L607 P254 A297 W303 F356 D365 D367 F428 W480 F596 L598 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h37 A 2.8 BS02 R02 A 1 F129 W169 P263 W312 F365 D374 W489 F601 F120 W160 P254 W303 F356 D365 W480 F592 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h39 A 2.8 BS02 R03 A 1 F129 T173 P263 F365 D374 F601 F605 F120 T164 P254 F356 D365 F592 F596 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h3a A 2.85 BS02 R04 A 1 W169 I261 P263 S307 W312 F365 D374 D376 F437 W489 F601 F605 L607 W160 I252 P254 S298 W303 F356 D365 D367 F428 W480 F592 F596 L598 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h3b A 2.8 BS02 R46 A 1 R127 F129 W169 P263 S307 W312 F365 D374 D376 D377 F437 W489 F601 R118 F120 W160 P254 S298 W303 F356 D365 D367 D368 F428 W480 F592 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h3c A 2.9 BS02 R79 A 1 A170 T173 P263 W312 D374 D376 W489 F601 F605 A161 T164 P254 W303 D365 D367 W480 F592 F596 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1h46 X 1.52 BS01 RNP X 1 Y142 D170 Q172 E207 D209 E212 R240 A369 W373 Y378 Y142 D170 Q172 E207 D209 E212 R240 A369 W373 Y378 3.2.1.-,3.2.1.4 0004553,0005975 Ki=270uM remove_due_to_license_issue Q7LHI2 12657782 1433 EQAGTNTAENHPQLQSQQCTTSGGCKPLSTKVVLDSNWRWVHSTSGYTNCYTGNEWDTSLCPDGKTCAANCALDGADYSGTYGITSTGTALTLKFVTGSNVGSRVYLMADDTHYQLLKLLNQEFTFDVDMSNLPCGLNGALYLSAMDADGGMSKYPGNKAGAKYGTGYCDSQCPKDIKFINGEANVGNWTETGSNTGTGSYGTCCSEMDIWEANNDAAAFTPHPCTTTGQTRCSGDDCARNTGLCDGDGCDFNSFRMGDKTFLGKGMTVDTSKPFTVVTQFLTNDNTSTGTLSEIRRIYIQNGKVIQNSVANIPGVDPVNSITDNFCAQQKTAFGDTNWFAQKGGLKQMGEALGNGMVLALSIWDDHAANMLWLDSDYPTDKDPSAPGVARGTCATTSGVPSDVESQVPNSQVVFSNIKFGDIGSTFSGTS 1h4w A 1.7 BS01 BEN A 1 D189 S190 C191 Q192 S195 G219 D171 S172 C173 Q174 S177 G196 H57 D102 Q192 R193 D194 S195 G196 H40 D84 Q174 R175 D176 S177 G178 3.4.21.4 0004252,0006508 Ki=22uM remove_due_to_license_issue P35030 11827488 250 IVGGYTCEENSLPYQVSLNSGSHFCGGSLISEQWVVSAAHCYKTRIQVRLGEHNIKVLEGNEQFINAVKIIRHPKYNRDTLDNDIMLIKLSSPAVINARVSTISLPTAPPAAGTECLISGWGNTLSFGADYPDELKCLDAPVLTQAECKASYPGKITNSMFCVGFLEGGKDSCQRDSGGPVVCNGQLQGVVSWGHGCAWKNRPGVYTKVYNYVDWIKDTIAANS 1h5u A 1.76 BS01 CHI A 1 R60 V64 W67 W189 E190 K191 R48 V52 W55 W177 E178 K179 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=178nM remove_due_to_license_issue P00489 11886794 920 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1h5v A 1.1 BS01 MA3 B 1 Q180 H206 Q177 H203 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11679762 1 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESA 1h5v A 1.1 BS02 SGC B 1 E139 Y202 W262 E136 Y199 W259 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11679762 3 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESA 1h5v A 1.1 BS03 SSG B 1 H35 Y66 K267 E269 H32 Y63 K264 E266 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11679762 4 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESA 1h5v A 1.1 BS04 GLC B 1 W39 Y40 K267 W36 Y37 K264 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 11679762 5 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRESA 1h60 A 1.6 BS02 STR A 1 T26 R142 H181 H184 Y186 Q241 Y351 T26 R142 H181 H184 Y186 Q241 Y351 T26 H181 H184 Y186 R233 Q241 T26 H181 H184 Y186 R233 Q241 ? 0000166,0005829,0010181,0016491 Kd=20uM remove_due_to_license_issue P71278 11428899 500 SAEKLFTPLKVGAVTAPNRVFMAPLTRLRSIEPGDIPTPLMGEYYRQRASAGLIISEATQISAQAKGYAGAPGLHSPEQIAAWKKITAGVHAEDGRIAVQLWHTGRISHSSIQPGGQAPVSASALNANTRTSLRDENGNAIRVDTTTPRALELDEIPGIVNDFRQAVANAREAGFDLVELHSAHGYLLHQFLSPSSNQRTDQYGGSVENRARLVLEVVDAVCNEWSADRIGIRVSPIGTFQNVDNGPNEEADALYLIEELAKRGIAYLHMSETDLAGGKPYSEAFRQKVRERFHGVIIGAGAYTAEKAEDLIGKGLIDAVAFGRDYIANPDLVARLQKKAELNPQRPESFYGGGAEGYTDYPSL 1h61 A 1.4 BS02 PDN A 1 T26 R130 H184 Y186 Q241 Y351 T26 R130 H184 Y186 Q241 Y351 T26 H181 H184 Y186 R233 Q241 T26 H181 H184 Y186 R233 Q241 ? 0000166,0005829,0010181,0016491 Kd=13uM remove_due_to_license_issue P71278 11428899 1366 SAEKLFTPLKVGAVTAPNRVFMAPLTRLRSIEPGDIPTPLMGEYYRQRASAGLIISEATQISAQAKGYAGAPGLHSPEQIAAWKKITAGVHAEDGRIAVQLWHTGRISHSSIQPGGQAPVSASALNANTRTSLRDENGNAIRVDTTTPRALELDEIPGIVNDFRQAVANAREAGFDLVELHSAHGYLLHQFLSPSSNQRTDQYGGSVENRARLVLEVVDAVCNEWSADRIGIRVSPIGTFQNVDNGPNEEADALYLIEELAKRGIAYLHMSETDLAGGKPYSEAFRQKVRERFHGVIIGAGAYTAEKAEDLIGKGLIDAVAFGRDYIANPDLVARLQKKAELNPQRPESFYGGGAEGYTDYPSL 1h62 A 1.9 BS01 ANB A 1 T26 Y68 S132 R142 H181 H184 Y186 Q241 Y351 T26 Y68 S132 R142 H181 H184 Y186 Q241 Y351 T26 H181 H184 Y186 R233 Q241 T26 H181 H184 Y186 R233 Q241 ? 0000166,0005829,0010181,0016491 Kd=17uM remove_due_to_license_issue P71278 11428899 501 SAEKLFTPLKVGAVTAPNRVFMAPLTRLRSIEPGDIPTPLMGEYYRQRASAGLIISEATQISAQAKGYAGAPGLHSPEQIAAWKKITAGVHAEDGRIAVQLWHTGRISHSSIQPGGQAPVSASALNANTRTSLRDENGNAIRVDTTTPRALELDEIPGIVNDFRQAVANAREAGFDLVELHSAHGYLLHQFLSPSSNQRTDQYGGSVENRARLVLEVVDAVCNEWSADRIGIRVSPIGTFQNVDNGPNEEADALYLIEELAKRGIAYLHMSETDLAGGKPYSEAFRQKVRERFHGVIIGAGAYTAEKAEDLIGKGLIDAVAFGRDYIANPDLVARLQKKAELNPQRPESFYGGGAEGYTDYPSL 1h6h A 1.7 BS01 PIB A 1 R58 Y59 R60 K92 V93 Y94 R105 R57 Y58 R59 K91 V92 Y93 R104 ? 0006909,0016176,0035091,0043020,0045730 Kd=5uM remove_due_to_license_issue Q15080 11684018 150 AVAQQLRAESDFEQLPDDVAISANIADIEEKRGFTSHFVFVIEVKTKGGSKYLIYRRYRQFHALQSKLEERFGPDSKSSALACTLPTLPAKVYVGVKQEIAEMRIPALNAYMKSLLSLPVWVLMDEDVRIFFYQSPYDSEQVP 1h79 A 2.9 BS01 TTP A 1 I99 E100 K103 V107 I111 Q114 I73 E74 K77 V81 I85 Q88 N78 C79 M288 C290 S292 N311 Y441 E446 A580 N52 C53 M262 C264 S266 N285 Y415 E420 A554 1.1.98.6 0003824,0004748,0006260,0008998,0009265,0016491,0046872 remove_due_to_license_issue P07071 11587648 1586 SRVFPTQRDLMAGIVSKHIAKNMVPSFIMKAHESGIIHVHDIDYSPALPFTNCCLVDLKGMLENGFKLGNAQIETPKSIGVATAIMAQITAQVASHQYGGTTFANVDKVLSPYVKRTYAKHIEDAEKWQIADALNYAQSKTEKDVYDAFQAYEYEVNTLFSSNGQTPFVTITFGTGTDWTERMIQKAILKNRIKGLGRDGITPIFPKLVMFVEEGVNLYKDDPNYDIKQLALECASKRMYPDIISAKNNKAITGSSVPVSPMGCRSFLSVWKDSTGNEILDGRNNLGVVTLNLPRIALDSYIGTQFNEQKFVELFNERMDLCFEALMCRISSLKGVKATVAPILYQEGAFGVRLKPDDDIIELFKNGRSSVSLGYIGIHELNILVGRDIGREILTKMNAHLKQWTERTGFAFSLYSTPAENLCYRFCKLDTEKYGSVKDVTDKGWYTNSFHVSVEENITPFEKISREAPYHFIATGGHISYVELPDMKNNLKGLEAVWDYAAQHLDYFGVNMPVDKCFTCGSTHEMTPTENGFVCSICGETDPKKMNTIRRTCAYLGNP 1h79 A 2.9 BS03 TTP A 2 H64 H66 Q191 A445 E446 N447 L448 R451 H38 H40 Q165 A419 E420 N421 L422 R425 N78 C79 M288 C290 S292 N311 Y441 E446 A580 N52 C53 M262 C264 S266 N285 Y415 E420 A554 1.1.98.6 0003824,0004748,0006260,0008998,0009265,0016491,0046872 remove_due_to_license_issue P07071 11587648 1589 SRVFPTQRDLMAGIVSKHIAKNMVPSFIMKAHESGIIHVHDIDYSPALPFTNCCLVDLKGMLENGFKLGNAQIETPKSIGVATAIMAQITAQVASHQYGGTTFANVDKVLSPYVKRTYAKHIEDAEKWQIADALNYAQSKTEKDVYDAFQAYEYEVNTLFSSNGQTPFVTITFGTGTDWTERMIQKAILKNRIKGLGRDGITPIFPKLVMFVEEGVNLYKDDPNYDIKQLALECASKRMYPDIISAKNNKAITGSSVPVSPMGCRSFLSVWKDSTGNEILDGRNNLGVVTLNLPRIALDSYIGTQFNEQKFVELFNERMDLCFEALMCRISSLKGVKATVAPILYQEGAFGVRLKPDDDIIELFKNGRSSVSLGYIGIHELNILVGRDIGREILTKMNAHLKQWTERTGFAFSLYSTPAENLCYRFCKLDTEKYGSVKDVTDKGWYTNSFHVSVEENITPFEKISREAPYHFIATGGHISYVELPDMKNNLKGLEAVWDYAAQHLDYFGVNMPVDKCFTCGSTHEMTPTENGFVCSICGETDPKKMNTIRRTCAYLGNP 1h7a A 2.75 BS01 DTP A 1 I99 E100 K103 V107 I111 Q114 K146 I73 E74 K77 V81 I85 Q88 K120 N78 C79 M288 C290 S292 N311 Y441 E446 A580 N52 C53 M262 C264 S266 N285 Y415 E420 A554 1.1.98.6 0003824,0004748,0006260,0008998,0009265,0016491,0046872 remove_due_to_license_issue P07071 11587648 1590 SRVFPTQRDLMAGIVSKHIAKNMVPSFIMKAHESGIIHVHDIDYSPALPFTNCCLVDLKGMLENGFKLGNAQIETPKSIGVATAIMAQITAQVASHQYGGTTFANVDKVLSPYVKRTYAKHIEDAEKWQIADALNYAQSKTEKDVYDAFQAYEYEVNTLFSSNGQTPFVTITFGTGTDWTERMIQKAILKNRIKGLGRDGITPIFPKLVMFVEEGVNLYKDDPNYDIKQLALECASKRMYPDIISAKNNKAITGSSVPVSPMGCRSFLSVWKDSTGNEILDGRNNLGVVTLNLPRIALDSYIGTQFNEQKFVELFNERMDLCFEALMCRISSLKGVKATVAPILYQEGAFGVRLKPDDDIIELFKNGRSSVSLGYIGIHELNILVGRDIGREILTKMNAHLKQWTERTGFAFSLYSTPAENLCYRFCKLDTEKYGSVKDVTDKGWYTNSFHVSVEENITPFEKISREAPYHFIATGGHISYVELPDMKNNLKGLEAVWDYAAQHLDYFGVNMPVDKCFTCGSTHEMTPTENGFVCSICGETDPKKMNTIRRTCAYLGNPNERG 1h88 A 2.8 BS01 dna D 0 K269 Y274 R278 N281 N282 R286 R289 K3 Y8 R12 N15 N16 R20 R23 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 VDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h88 A 2.8 BS02 dna E 0 K287 S288 R289 K21 S22 R23 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 VDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h88 B 2.8 BS01 dna D 0 V285 S288 R289 V20 S23 R24 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 TVDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h88 B 2.8 BS02 dna E 0 Y274 R278 N281 N282 R289 Y9 R13 N16 N17 R24 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 TVDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h88 C 2.8 BS01 dna D 0 K92 K128 Q129 E132 R133 H137 N179 N183 S187 K54 K90 Q91 E94 R95 H99 N141 N145 S149 ? remove_due_to_license_issue P06876 11792321 1 ~ 26 GKTRWTREEDEKLKKLVEQNGTDDWKVIANYLPNRTDVQCQHRWQKVLNPELIKGPWTKEEDQRVIKLVQKYGPKRWSVIAKHLKGRIGKQCRERWHNHLNPEVKKTSWTEEEDRIIYQAHKRLGNRWAEIAKLLPGRTDNAIKNHWNSTMR 1h88 C 2.8 BS02 dna E 0 K113 R114 W115 R131 N164 R165 W166 A167 K182 K75 R76 W77 R93 N126 R127 W128 A129 K144 ? remove_due_to_license_issue P06876 11792321 1 ~ 26 GKTRWTREEDEKLKKLVEQNGTDDWKVIANYLPNRTDVQCQHRWQKVLNPELIKGPWTKEEDQRVIKLVQKYGPKRWSVIAKHLKGRIGKQCRERWHNHLNPEVKKTSWTEEEDRIIYQAHKRLGNRWAEIAKLLPGRTDNAIKNHWNSTMR 1h89 A 2.45 BS01 dna D 0 Y274 R278 N281 N282 R286 R289 K293 Y2 R6 N9 N10 R14 R17 K21 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 EYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h89 A 2.45 BS02 dna E 0 R280 V285 K287 S288 R8 V13 K15 S16 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 EYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h89 B 2.45 BS01 dna D 0 V285 K287 S288 R289 V13 K15 S16 R17 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 EYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h89 B 2.45 BS02 dna E 0 Y274 R278 N281 N282 R286 R289 Y2 R6 N9 N10 R14 R17 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 EYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 1h89 C 2.45 BS01 dna D 0 K92 K128 Q129 E132 R133 H137 N179 N183 S187 T188 K16 K52 Q53 E56 R57 H61 N103 N107 S111 T112 ? remove_due_to_license_issue P06876 11792321 1 ~ 26 QCQHRWQKVLNPELIKGPWTKEEDQRVIKLVQKYGPKRWSVIAKHLKGRIGKQCRERWHNHLNPEVKKTSWTEEEDRIIYQAHKRLGNRWAEIAKLLPGRTDNAIKNHWNSTMRR 1h89 C 2.45 BS02 dna E 0 K113 R114 W115 K128 R131 N164 W166 A167 K182 K37 R38 W39 K52 R55 N88 W90 A91 K106 ? remove_due_to_license_issue P06876 11792321 1 ~ 26 QCQHRWQKVLNPELIKGPWTKEEDQRVIKLVQKYGPKRWSVIAKHLKGRIGKQCRERWHNHLNPEVKKTSWTEEEDRIIYQAHKRLGNRWAEIAKLLPGRTDNAIKNHWNSTMRR 1h8a A 2.23 BS01 dna D 0 K269 Y274 R278 N281 N282 R286 R289 K3 Y8 R12 N15 N16 R20 R23 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 VDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQL 1h8a A 2.23 BS02 dna E 0 R280 K287 S288 K291 R14 K21 S22 K25 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 VDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQL 1h8a B 2.23 BS01 dna D 0 A284 V285 K287 S288 R289 A17 V18 K20 S21 R22 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 DKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQL 1h8a B 2.23 BS02 dna E 0 K269 Y274 R278 N282 R289 K2 Y7 R11 N15 R22 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11792321 1 ~ 26 DKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQL 1h8a C 2.23 BS01 dna D 0 K92 K128 Q129 E132 N179 N183 S187 R191 K6 K42 Q43 E46 N93 N97 S101 R105 ? remove_due_to_license_issue P01104 11792321 1 ~ 26 NPELNKGPWTKEEDQRVIEHVQKYGPKRWSDIAKHLKGRIGKQCRERWHNHLNPEVKKTSWTEEEDRIIYQAHKRLGNRWAEIAKLLPGRTDNAVKNHWNSTMRR 1h8a C 2.23 BS02 dna E 0 R131 N164 W166 A167 K182 R45 N78 W80 A81 K96 ? remove_due_to_license_issue P01104 11792321 1 ~ 26 NPELNKGPWTKEEDQRVIEHVQKYGPKRWSDIAKHLKGRIGKQCRERWHNHLNPEVKKTSWTEEEDRIIYQAHKRLGNRWAEIAKLLPGRTDNAVKNHWNSTMRR 1h8l A 2.6 BS01 GEM A 1 H74 E77 R135 N144 R145 H181 N188 D192 G246 Y250 V252 E272 H71 E74 R132 N141 R142 H178 N185 D189 G243 Y247 V249 E269 3.4.17.22 0004180,0004181,0005615,0006508,0006518,0008237,0008270,0016020,0016485,0046872 remove_due_to_license_issue P83852 11278909 801 QAVQPVDFRHHHFSDMEIFLRRYANEYPSITRLYSVGKSVELRELYVMEISDNPGIHEAGEPEFKYIGNMHGNEVVGRELLLNLIEYLCKNFGTDPEVTDLVQSTRIHIMPSMNPDGYEKSQEGDRGGTVGRNNSNNYDLNRNFPDQFFQVTDPPQPETLAVMSWLKTYPFVLSANLHGGSLVVNYPFDDDEQGIAIYSKSPDDAVFQQLALSYSKENKKMYQGSPCKDLYPTEYFPHGITNGAQWYNVPGGMQDWNYLNTNCFEVTIELGCVKYPKAEELPKYWEQNRRSLLQFIKQVHRGIWGFVLDATDGRGILNATISVADINHPVTTYKDGDYWRLLVQGTYKVTASARGYDPVTKTVEVDSKGGVQVNFTLSRT 1h8s A 2.4 BS01 AIC A 1 Q92 Y97 L99 W164 N166 W230 W233 Q89 Y94 L96 W140 N142 W206 W209 Kd=1.54uM remove_due_to_license_issue 11397088 1000 DIVLTQSHKFMSTSVGDRVSITCKASQDVGTAVAWYQQKPGQSPKLLIYWASTRHTGVPDRFTGSGSGTDFTLTISNVQSEDLADYFCQQYSSYPLTFGAGTKLELKQVQLQEPGGELVRPGASVKLSCKASGYTFTSYWINWVKQRPGQGLEWIGNIYPSDSYTNYNQKFKDKATLTVDKSSSTAYMQLSSLTSEDSAVYFCARWGYWGQGTLVTVS 1h8y A 2.0 BS01 MER A 1 S67 T206 G207 F208 L247 R250 S48 T187 G188 F189 L228 R231 S67 K70 S115 F120 W154 F208 S48 K51 S96 F101 W135 F189 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0071555 remove_due_to_license_issue Q51400 11453693 300 SSITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNNLARASKEYLPASTFKIPSAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLSLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLFLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKGTEVYFFAFNMDIDNENKLPLRKSIPTKIMASEGIIGG 1h8y B 2.0 BS01 MER B 1 S67 V117 T206 G207 F208 E244 L247 R250 S48 V98 T187 G188 F189 E225 L228 R231 S67 K70 S115 F120 W154 F208 S48 K51 S96 F101 W135 F189 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0071555 remove_due_to_license_issue Q51400 11453693 300 SSITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNNLARASKEYLPASTFKIPSAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLSLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLFLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKGTEVYFFAFNMDIDNENKLPLRKSIPTKIMASEGIIGG 1h9d A 2.6 BS01 dna E 0 R80 R135 R142 R174 R177 R27 R82 R89 R121 R124 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q01196 11276260 1 ~ 10 VLADHPGELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPRR 1h9d A 2.6 BS02 dna F 0 R142 G143 K167 T169 V170 D171 R89 G90 K114 T116 V117 D118 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q01196 11276260 1 ~ 10 VLADHPGELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPRR 1h9d C 2.6 BS01 dna G 0 R80 R135 R174 R27 R82 R121 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q01196 11276260 1 ~ 10 VLADHPGELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPRR 1h9d C 2.6 BS02 dna H 0 R139 R142 G143 K167 T169 V170 D171 R86 R89 G90 K114 T116 V117 D118 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q01196 11276260 1 ~ 10 VLADHPGELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPRR 1h9t A 3.25 BS01 dna X 0 S7 A9 T44 T47 H65 G66 S3 A5 T40 T43 H61 G62 ? 0000062,0003677,0003700,0005737,0005829,0006355,0006631,0019217,0042803,0045723,0045892,0045893 remove_due_to_license_issue P0A8V6 11296236 1 ~ 19 AQSPAGFAEEYIIESIWNNRFPPGTILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNNFWETSGLNILETLARLDHESVPQLIDNLLSVRTNISTIFIRTAFRQHPDKAQEVLATANEVADHADAFAELDYNIFRGLAFASGNPIYGLILNGMKGLYTRIGRHYFANPEARSLALGFYHKLSALCSEGAHDQVYETVRRYGHESGEIWHRMQKNLLAIQGR 1h9t A 3.25 BS02 dna Y 0 A33 E34 R35 R45 R49 I63 Q64 H65 G66 K67 A29 E30 R31 R41 R45 I59 Q60 H61 G62 K63 ? 0000062,0003677,0003700,0005737,0005829,0006355,0006631,0019217,0042803,0045723,0045892,0045893 remove_due_to_license_issue P0A8V6 11296236 1 ~ 19 AQSPAGFAEEYIIESIWNNRFPPGTILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNNFWETSGLNILETLARLDHESVPQLIDNLLSVRTNISTIFIRTAFRQHPDKAQEVLATANEVADHADAFAELDYNIFRGLAFASGNPIYGLILNGMKGLYTRIGRHYFANPEARSLALGFYHKLSALCSEGAHDQVYETVRRYGHESGEIWHRMQKNLLAIQGR 1h9t B 3.25 BS01 dna X 0 A33 E34 R35 R45 R49 H65 G66 A29 E30 R31 R41 R45 H61 G62 ? 0000062,0003677,0003700,0005737,0005829,0006355,0006631,0019217,0042803,0045723,0045892,0045893 remove_due_to_license_issue P0A8V6 11296236 1 ~ 19 AQSPAGFAEEYIIESIWNNRFPPGTILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNNFWETSGLNILETLARLDHESVPQLIDNLLSVRTNISTIFIRTAFRQHPDKAQEVLATANEVADHADAFAELDYNIFRGLAFASGNPIYGLILNGMKGLYTRIGRHYFANPEARSLALGFYHKLSALCSEGAHDQVYETVRRYGHESGEIWHRMQKNL 1h9t B 3.25 BS02 dna Y 0 S7 P8 A9 V43 T44 T46 T47 H65 G66 S3 P4 A5 V39 T40 T42 T43 H61 G62 ? 0000062,0003677,0003700,0005737,0005829,0006355,0006631,0019217,0042803,0045723,0045892,0045893 remove_due_to_license_issue P0A8V6 11296236 1 ~ 19 AQSPAGFAEEYIIESIWNNRFPPGTILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNNFWETSGLNILETLARLDHESVPQLIDNLLSVRTNISTIFIRTAFRQHPDKAQEVLATANEVADHADAFAELDYNIFRGLAFASGNPIYGLILNGMKGLYTRIGRHYFANPEARSLALGFYHKLSALCSEGAHDQVYETVRRYGHESGEIWHRMQKNL 1h9z A 2.5 BS01 RWF A 1 W214 A215 R222 L238 H242 A291 W212 A213 R220 L236 H240 A289 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=3.8uM remove_due_to_license_issue Kd=1.2E4nM P02768 11285262 3001 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1ha2 A 2.5 BS01 SWF A 1 W214 A215 L219 L238 H242 L260 S287 A291 W212 A213 L217 L236 H240 L258 S285 A289 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=2.9uM remove_due_to_license_issue P02768 11285262 3001 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1hbj A 2.5 BS01 FBQ A 1 W84 G117 G118 G119 Y121 S200 A201 W233 F288 F290 F330 F331 W432 H440 W81 G114 G115 G116 Y118 S197 A198 W230 F285 F287 F327 F328 W429 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue IC50=11000nM P04058 11563919 1539 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1hbv A 2.3 BS01 GAN A 1 D25 G27 A28 D29 I47 G48 P81 V82 D25 G27 A28 D29 I47 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=430nM remove_due_to_license_issue P03366 7650677 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hbv B 2.3 BS01 GAN A 1 D25 G27 D29 G48 G49 I50 V82 I84 D25 G27 D29 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 7650677 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hdq A 2.3 BS01 INF A 1 R145 H196 I247 Y248 E270 R145 H196 I247 Y248 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=1.5uM remove_due_to_license_issue P00730 11937361 1308 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVEALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTLNN 1hdt H 2.6 BS02 0E7 H 1 H57 Y60A W60D D189 A190 C191 E192 S195 S214 W215 G216 E217 G219 C220 H43 Y47 W50 D199 A200 C201 E202 S205 S226 W227 G228 E229 G230 C231 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 7853394 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1hee A 1.75 BS02 LHY A 1 H69 E72 R127 N144 R145 S197 I243 T268 E270 H69 E72 R127 N144 R145 S197 I243 T268 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=4.6uM remove_due_to_license_issue P00730 11937361 1309 ARSTNTFNYATYHTLDEIYDFMDLLVAQHPELVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 1heg E 2.2 BS01 PSI E 1 D25 G27 A28 D29 G48 D25 G27 A28 D29 G48 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=18nM remove_due_to_license_issue P03366 1429626 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEENSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hfs A 1.7 BS06 L04 A 1 Y155 N162 V163 L164 A165 H166 Y168 H201 E202 H205 H211 L218 Y220 L222 Y223 H224 L226 Y68 N75 V76 L77 A78 H79 Y81 H114 E115 H118 H124 L131 Y133 L135 Y136 H137 L139 H201 E202 H205 H211 H114 E115 H118 H124 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=2nM remove_due_to_license_issue Ki=2nM P08254 9083493 256 GIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYG 1hge A 2.6 BS01 MNA A 1 Y98 R135 S136 N137 W153 H183 E190 L194 S228 Y98 R135 S136 N137 W153 H183 E190 L194 S228 ? 0019031,0019064,0046789 remove_due_to_license_issue P03438 1327122 349 QDLPGNDNSTATLCLGHHAVPNGTLVKTITDDQIEVTNATELVQSSSTGKICNNPHRILDGIDCTLIDALLGDPHCDVFQNETWDLFVERSKAFSNCYPYDVPDYASLRSLVASSGTLEFITEGFTWTGVTQNGRSNACKRGPGSGFFSRLNWLTKSGSTYPVLNVTMPNNDNFDKLYIWGIHHPSTNQEQTSLYVQASGRVTVSTRRSQQTIIPNIGSRPWVRGLSSRISIYWTIVKPGDVLVINSNGNLIAPRGYFKMRTGKSSIMRSDAPIDTCISECITPNGSIPNDKPFQNVNKITYGACPKYVKQNTLKLATGMRNVPEKQT 1hgi A 2.7 BS01 ANA A 1 Y98 G135 S136 N137 S145 W153 H183 E190 L194 L226 S228 Y98 G135 S136 N137 S145 W153 H183 E190 L194 L226 S228 ? 0019031,0019064,0046789 remove_due_to_license_issue P03438 1327122 349 QDLPGNDNSTATLCLGHHAVPNGTLVKTITDDQIEVTNATELVQSSSTGKICNNPHRILDGIDCTLIDALLGDPHCDVFQNETWDLFVERSKAFSNCYPYDVPDYASLRSLVASSGTLEFITEGFTWTGVTQNGGSNACKRGPGSGFFSRLNWLTKSGSTYPVLNVTMPNNDNFDKLYIWGIHHPSTNQEQTSLYVQASGRVTVSTRRSQQTIIPNIGSRPWVRGLSSRISIYWTIVKPGDVLVINSNGNLIAPRGYFKMRTGKSSIMRSDAPIDTCISECITPNGSIPNDKPFQNVNKITYGACPKYVKQNTLKLATGMRNVPEKQT 1hgj A 2.7 BS01 AMN A 1 Y98 G135 S136 N137 E190 L194 L226 Y98 G135 S136 N137 E190 L194 L226 ? 0019031,0019064,0046789 remove_due_to_license_issue P03438 1327122 349 QDLPGNDNSTATLCLGHHAVPNGTLVKTITDDQIEVTNATELVQSSSTGKICNNPHRILDGIDCTLIDALLGDPHCDVFQNETWDLFVERSKAFSNCYPYDVPDYASLRSLVASSGTLEFITEGFTWTGVTQNGGSNACKRGPGSGFFSRLNWLTKSGSTYPVLNVTMPNNDNFDKLYIWGIHHPSTNQEQTSLYVQASGRVTVSTRRSQQTIIPNIGSRPWVRGLSSRISIYWTIVKPGDVLVINSNGNLIAPRGYFKMRTGKSSIMRSDAPIDTCISECITPNGSIPNDKPFQNVNKITYGACPKYVKQNTLKLATGMRNVPEKQT 1hi3 A 1.8 BS01 A2P A 1 Q14 H15 H129 L130 Q15 H16 H130 L131 H15 K38 H129 H16 K39 H130 4.6.1.18 0001530,0002227,0003676,0004519,0004522,0004540,0005515,0005576,0005615,0005764,0006401,0006935,0016829,0035578,0043152,0050829,0050830,0051607,0070062 Ki=64uM remove_due_to_license_issue P10153 11154698 999 MKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII 1hi4 A 1.8 BS01 A3P A 1 M0 W7 Q14 H15 R68 N70 A110 V128 H129 M1 W8 Q15 H16 R69 N71 A111 V129 H130 H15 K38 H129 H16 K39 H130 4.6.1.18 0001530,0002227,0003676,0004519,0004522,0004540,0005515,0005576,0005615,0005764,0006401,0006935,0016829,0035578,0043152,0050829,0050830,0051607,0070062 Ki=32uM remove_due_to_license_issue P10153 11154698 301 MKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII 1hi5 A 1.8 BS01 ADP A 1 H15 K38 Q40 H82 H129 L130 H16 K39 Q41 H83 H130 L131 H15 K38 H129 H16 K39 H130 4.6.1.18 0001530,0002227,0003676,0004519,0004522,0004540,0005515,0005576,0005615,0005764,0006401,0006935,0016829,0035578,0043152,0050829,0050830,0051607,0070062 Ki=92uM remove_due_to_license_issue P10153 11154698 999 MKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII 1hih A 2.2 BS01 C20 B 1 D25 G27 A28 D29 G48 P81 V82 D25 G27 A28 D29 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 7613867 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hih B 2.2 BS01 C20 B 1 D25 G27 A28 G48 G49 I50 V82 I84 D25 G27 A28 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=9nM remove_due_to_license_issue P03366 7613867 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hii A 2.3 BS01 C20 B 1 D25 G27 A28 G48 G49 I82 D25 G27 A28 G48 G49 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 7613867 101 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hii B 2.3 BS01 C20 B 1 D25 G27 A28 D29 G48 G49 I50 P81 I82 D25 G27 A28 D29 G48 G49 I50 P81 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=53nM remove_due_to_license_issue P04584 7613867 101 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hiv A 2.0 BS01 1ZK A 1 R8 D25 G27 A28 D29 I47 G48 G49 I50 V82 R8 D25 G27 A28 D29 I47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki<1nM remove_due_to_license_issue P04585 1304383 100 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hiv B 2.0 BS01 1ZK A 1 D25 G27 A28 D29 G48 D25 G27 A28 D29 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 1304383 100 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hiy A 2.6 BS01 3AN A 1 F64 L68 R92 T98 R109 V116 N119 F59 L63 R87 T93 R104 V111 N114 K16 Y56 N119 H122 E133 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 11294625 1156 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIHGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1hiy B 2.6 BS01 3AN B 1 H259 F264 L268 R292 T298 N319 H54 F59 L63 R87 T93 N114 K216 Y256 N319 H322 E333 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 11294625 1356 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIHGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1hk1 A 2.65 BS01 T44 A 1 Y150 K199 W214 R218 L219 R222 L238 H242 R257 I290 A291 Y134 K183 W198 R202 L203 R206 L222 H226 R241 I274 A275 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3001 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFA 1hk1 A 2.65 BS02 T44 A 2 Q390 N391 A406 L407 R410 Y411 L453 S489 Q374 N375 A390 L391 R394 Y395 L437 S473 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3002 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFA 1hk1 A 2.65 BS03 T44 A 3 F507 T508 I513 K524 K525 A528 F551 A552 F568 F491 T492 I497 K508 K509 A512 F535 A536 F552 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3003 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFA 1hk1 A 2.65 BS04 T44 A 4 F502 F507 A528 E531 L532 F551 F486 F491 A512 E515 L516 F535 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3004 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFA 1hk2 A 2.8 BS01 T44 A 1 Y150 K199 H218 R222 L238 R257 A291 Y134 K183 H202 R206 L222 R241 A275 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3001 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAHLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLV 1hk2 A 2.8 BS02 T44 A 2 L387 Q390 N391 L394 A406 L407 Y411 L453 S489 L371 Q374 N375 L378 A390 L391 Y395 L437 S473 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3002 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAHLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLV 1hk2 A 2.8 BS03 T44 A 3 F507 T508 I513 K524 A528 M548 F551 F491 T492 I497 K508 A512 M532 F535 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3003 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAHLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLV 1hk2 A 2.8 BS04 T44 A 4 F502 F507 A528 E531 L532 F551 V576 F486 F491 A512 E515 L516 F535 V560 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3004 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAHLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLV 1hk3 A 2.8 BS01 T44 A 1 Y150 K199 W214 P218 L219 L238 H242 R257 A291 Y134 K183 W198 P202 L203 L222 H226 R241 A275 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3001 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAPLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKL 1hk3 A 2.8 BS02 T44 A 2 L387 Q390 N391 A406 L407 R410 Y411 L453 S489 L371 Q374 N375 A390 L391 R394 Y395 L437 S473 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3002 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAPLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKL 1hk3 A 2.8 BS03 T44 A 3 F507 T508 K524 F551 F491 T492 K508 F535 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3003 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAPLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKL 1hk3 A 2.8 BS04 T44 A 4 F502 F507 A528 E531 L532 V547 F551 L575 F486 F491 A512 E515 L516 V531 F535 L559 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 3004 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTDCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAPLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKL 1hk4 A 2.4 BS01 T44 A 1 D187 E188 K190 A191 K195 N429 K432 D451 Y452 D185 E186 K188 A189 K193 N427 K430 D449 Y450 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=4.9uM remove_due_to_license_issue P02768 12743361 1008 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1hk5 A 2.7 BS01 T44 A 1 D187 E188 K190 A191 K195 N429 K432 D451 Y452 D185 E186 K188 A189 K193 N427 K430 D449 Y450 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 12743361 1008 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVAHLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 1hkj A 2.6 BS01 NA1 B 1 W31 N100 E297 W10 N79 E276 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q13231 12639956 2 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEQSGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQELS 1hkj A 2.6 BS02 AMI A 1 Y27 W99 D138 E140 M210 Y212 Y267 M356 W358 Y6 W78 D117 E119 M189 Y191 Y246 M335 W337 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q13231 12639956 1389 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEQSGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQELS 1hkk A 1.85 BS01 AMI A 1 Y27 W99 D138 E140 M210 Y212 D213 Y267 W358 Y6 W78 D117 E119 M189 Y191 D192 Y246 W337 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q13231 12639956 1388 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEQSGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQEL 1hkk A 1.85 BS02 AMI A 2 Y141 Q145 A186 G187 Y190 D213 Y120 Q124 A165 G166 Y169 D192 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q13231 12639956 1391 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEQSGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQEL 1hkm A 2.55 BS01 ALI A 1 Y27 W99 D138 E140 M210 Y212 D213 Y267 W358 Y6 W78 D117 E119 M189 Y191 D192 Y246 W337 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q13231 12639956 1389 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEQSGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQELS 1hlf A 2.26 BS02 GL4 A 1 G135 L136 N284 H377 N484 E672 G675 G123 L124 N272 H365 N472 E660 G663 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=2.3uM remove_due_to_license_issue Ki=5100nM P00489 11741774 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1hlk A 2.5 BS03 113 A 1 W49 H162 C181 N193 H223 W29 H142 C161 N173 H203 H99 H101 D103 H162 C181 K184 N193 H223 H79 H81 D83 H142 C161 K164 N173 H203 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=10uM remove_due_to_license_issue P25910 12019104 2002 SVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQATSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGDYGGTELIEHTKQIVNQYIESTS 1hmr A 1.4 BS01 ELA A 1 K58 D76 L115 R126 Y128 K58 D76 L115 R126 Y128 ? 0005515,0005615,0005634,0005737,0005829,0008092,0008285,0008289,0015909,0032365,0036041,0042632,0046320,0050873,0055091,0070062,0070538,0071073,0140214,2001245 Kd=0.28uM remove_due_to_license_issue P05413 7922029 133 VDAFLGTWKLVDSKNFDDYMKSLGVGFATRQVASMTKPTTIIEKNGDILTLKTHSTFKNTEISFKLGVEFDETTADDRKVKSIVTLDGGKLVHLQKWDGQETTLVRELIDGKLILTLTHGTAVCTRTYEKE 1hn2 A 1.8 BS01 ANC A 1 T1038 F1056 F1089 N1103 T1116 T38 F56 F89 N103 T116 ? 0005549,0005576,0005615,0007608,0036094 Kd=1uM remove_due_to_license_issue P07435 11114310 3001 AQEEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPHPE 1hn2 B 1.8 BS01 ANC B 1 F2056 F2089 N2103 T2116 E2117 F2119 F54 F87 N101 T114 E115 F117 ? 0005549,0005576,0005615,0007608,0036094 Kd=1uM remove_due_to_license_issue P07435 11114310 3002 EEEAEQNLSELSGPWRTVYIGSTNPEKIQENGPFRTYFRELVFDDEKGTVDFYFSVKRDGKWKNVHVKATKQDDGTYVADYEGQNVFKIVSLSRTHLVAHNINVDKHGQTTELTELFVKLNVEDEDLEKFWKLTEDKGIDKKNVVNFLENENHPH 1hn4 A 1.5 BS04 MJI A 1 S-2 L2 C29 G30 C45 H48 D49 Y52 F106 S4 L7 C34 G35 C50 H53 D54 Y57 F111 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y33 G35 G37 H53 D54 Y57 Y78 D104 3.1.1.4 0002446,0004623,0005102,0005509,0005543,0005576,0006629,0006633,0006644,0008284,0009986,0010524,0016042,0016787,0019370,0030593,0032052,0032652,0032757,0032869,0035556,0043406,0045944,0046324,0046470,0046471,0046872,0047498,0047499,0048146,0050482,0050778,0051092,1904635 Kd=0.15mM remove_due_to_license_issue P00592 11560489 397 GISSRALWQFRSMIKCAIPGSHPLMDFNNYGCYCGLGGSGTPVDELDRCCETHDNCYRDAKNLDSCKFLVDNPYTESYSYSCSNTEITCNSKNNACEAFICNCDRNAAICFSKAPYNKEHKNLDTKKYC 1hnn A 2.4 BS02 SKF A 1 Y35 N39 Y40 R44 V53 K57 F182 E219 M258 Y14 N18 Y19 R23 V32 K36 F161 E198 M237 E185 E219 E164 E198 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=0.58uM remove_due_to_license_issue Ki=280nM P11086 11591352 3001 AVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKVGL 1hos A 2.3 BS01 PHP A 1 D25 G27 A28 G48 G49 P81 V82 I84 D25 G27 A28 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2.8nM remove_due_to_license_issue P03366 8347601 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hos B 2.3 BS01 PHP A 1 D25 G27 I47 G48 G49 I50 V82 D25 G27 I47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8347601 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hp0 A 2.1 BS02 AD3 A 1 N12 D14 D40 W83 M164 N173 E184 N186 Y257 W260 D261 N12 D14 D40 W83 M164 N173 E184 N186 Y249 W252 D253 D10 D15 D40 W83 T137 W185 N186 W260 D261 D10 D15 D40 W83 T137 W185 N186 W252 D253 3.2.2.1 0005829,0006139,0006152,0008477,0016798,0016799,0046872 Ki=0.2uM remove_due_to_license_issue Q9GPQ4 11292348 1315 SAKNVVLDHDGNLDDFVAMVLLASNTEKVRLIGALCTDADCFVENGFNVTGKIMCLMHNNMNLPLFPIGKSAATAVNPFPKEWRCLAKNMDDMPILNIPENVELWDKIKAENEKYEGQQLLADLVMNSEEKVTICVTGPLSNVAWCIDKYGEKFTSKVEECVIMGGAVDVRGNVFLPSTDGTAEWNIYWDPASAKTVFGCPGLRRIMFSLDSTNTVPVRSPYVQRFGEQTNFLLSILVGTMWAMCTHGYYAWDALTAAYVVDQKVANVDPVPIDVVVDKQPNEGATVRTDAENYPLTFVARNPEAEFFLDMLLRSARAC 1hp5 A 2.1 BS01 NGT A 1 R162 H250 D313 E314 W344 W361 Y393 D395 W408 W442 E444 R155 H243 D306 E307 W337 W354 Y386 D388 W401 W435 E437 D313 E314 D306 E307 3.2.1.52 0004553,0004563,0005975,0016020,0016231,0016798,0030203 remove_due_to_license_issue Ki=20000nM O85361 11124970 511 DRKAPVRPTPLDRVIPAPASVDPGGAPYRITRGTHIRVDDSREARRVGDYLADLLRPATGYRLPVTAHGHGGIRLRLAGGPYGDEGYRLDSGPAGVTITARKAAGLFHGVQTLRQLLPPAVEKDSAQPGPWLVAGGTIEDTPRYAWRSAMLDVSRHFFGVDEVKRYIDRVARYKYNKLHLHLSDDQGWRIAIDSWPRLATYGGSTEVGGGPGGYYTKAEYKEIVRYAASRHLEVVPEIDMPGHTNAALASYAELNCDGVAPPLYTGTKVGFSSLCVDKDVTYDFVDDVIGELAALTPGRYLHIGGDEAHSTPKADFVAFMKRVQPIVAKYGKTVVGWHQLAGAEPVEGALVQYWGLDRTGDAEKAEVAEAARNGTGLILSPADRTYLDMKYTKDTPLGLSWAGYVEVQRSYDWDPAGYLPGAPADAVRGVEAPLWTETLSDPDQLDYMAFPRLPGVAELGWSPASTHDWDTYKVRLAAQAPYWEAAGIDFYRSPQVPWT 1hpo A 2.5 BS01 UNI B 1 R8 D25 G27 G49 R8 D25 G27 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 9089336 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hpo B 2.5 BS01 UNI B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P03367 9089336 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hps A 2.3 BS01 RUN B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 7932533 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hps A 2.3 BS02 RUN B 2 R8 D25 G27 A28 I47 G48 G49 I50 V82 R8 D25 G27 A28 I47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 7932533 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hps B 2.3 BS01 RUN B 1 R8 D25 G27 A28 G48 G49 P81 R8 D25 G27 A28 G48 G49 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P03366 7932533 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hps B 2.3 BS02 RUN B 2 R8 L23 D25 G27 A28 D29 D30 G48 G49 I50 V82 R8 L23 D25 G27 A28 D29 D30 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P03366 7932533 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hpv A 1.9 BS01 478 B 1 D25 G27 D30 V32 D25 G27 D30 V32 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hpv B 1.9 BS01 478 B 1 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P04587 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hpx A 2.0 BS01 KNI B 1 R8 D25 G27 P81 V82 I84 R8 D25 G27 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 8590019 900 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hpx B 2.0 BS01 KNI B 1 D25 G27 A28 D29 D30 V32 G48 G49 I50 D25 G27 A28 D29 D30 V32 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=5.5pM remove_due_to_license_issue P03367 8590019 900 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hq1 A 1.52 BS01 rna B 0 R27 A30 N33 S34 M35 K38 S49 R50 R53 G57 S58 G59 M60 R20 A23 N26 S27 M28 K31 S42 R43 R46 G50 S51 G52 M53 3.6.5.4 0003924,0005525,0006614,0008312,0048500 remove_due_to_license_issue P0AGD7 11243816 130 ~ 178 GFDLNDFLEQLRQDDKVLVRMEAIINSMTMKERAKPEIIKGSRKRRIAAGSGMQVQDVNRLLKQFDDMQRMMKKMK 1hq5 A 2.3 BS03 S2C A 1 D124 H126 D128 S137 H141 D183 D232 D234 E277 D119 H121 D123 S132 H136 D178 D227 D229 E272 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 Kd=2.22uM remove_due_to_license_issue P07824 11258879 551 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTTSSGNLHGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHK 1hqf A 2.9 BS03 HAR A 1 D124 H126 D128 H141 E186 D232 D234 E277 D119 H121 D123 H136 E181 D227 D229 E272 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 remove_due_to_license_issue P07824 11258880 906 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTTSSGNLHGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHKPETDYL 1hqg A 2.0 BS03 ORN A 1 H126 N130 C141 D183 H121 N125 C136 D178 H101 D124 H126 D128 C141 D232 D234 E277 H96 D119 H121 D123 C136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 remove_due_to_license_issue P07824 11258880 801 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTTSSGNLCGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHKPETDYL 1hqh A 2.8 BS03 NNH A 1 H126 D128 H141 G142 D183 T246 H121 D123 H136 G137 D178 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 remove_due_to_license_issue IC50=2000nM P07824 11258880 901 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTTSSGNLHGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHKPETDYL 1hrn A 1.8 BS01 03D A 1 D32 G34 Y75 S76 P111 A115 F117 V120 L213 D215 G217 A218 S219 D35 G37 Y80 S81 P115 A119 F121 V124 L218 D220 G222 A223 S224 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D220 A223 3.4.23.15 0004190,0006508 ic50=9nM remove_due_to_license_issue P00797 7608971 391 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSESLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 1hs6 A 1.95 BS02 BES A 1 Q136 Y267 G268 G269 M270 E271 H295 E296 H299 F314 E318 Y378 Y383 Q136 Y267 G268 G269 M270 E271 H295 E296 H299 F314 E318 Y378 Y383 E271 H295 E296 H299 E318 D375 Y383 E271 H295 E296 H299 E318 D375 Y383 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=4000nM, Kd=2050nM, Ki=320nM P09960 11175901 901 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 1hsg A 2.0 BS01 MK1 B 1 R8 D25 G27 G48 G49 V82 R8 D25 G27 G48 G49 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 7929352 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hsg B 2.0 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.38nM remove_due_to_license_issue P03367 7929352 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hsh A 1.9 BS01 MK1 A 1 D25 G27 A28 D29 D30 I32 V47 G48 P81 D25 G27 A28 D29 D30 I32 V47 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=2.45nM remove_due_to_license_issue P04584 7929352 401 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hsh B 1.9 BS01 MK1 A 1 D25 G27 V47 G48 G49 I82 D25 G27 V47 G48 G49 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 7929352 401 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hsl A 1.89 BS01 HIS A 1 Y14 L52 S69 S70 L71 S72 R77 T120 T121 D161 Y14 L52 S69 S70 L71 S72 R77 T120 T121 D161 ? 0006865,0016020,0016597,0030288,0042597,0055052,0071705,1903810 Kd=0.064uM remove_due_to_license_issue P0AEU0 8161536 239 AIPQKIRIGTDPTYAPFESKNAQGELVGFDIDLAKELCKRINTQCTFVENPLDALIPSLKAKKIDAIMSSLSITEKRQQEIAFTDKLYAADSRLVVAKNSDIQPTVASLKGKRVGVLQGTTQETFGNEHWAPKGIEIVSYQGQDNIYSDLTAGRIDAAFQDEVAASEGFLKQPVGKDYKFGGPAVKDEKLFGVGTGMGLRKEDNELREALNKAFAEMRADGTYEKLAKKYFDFDVYGG 1hte A 2.8 BS01 G23 A 1 A28 D29 D30 V32 A28 D29 D30 V32 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8031777 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hte B 2.8 BS02 G23 A 1 R8 L10 I50 P81 V82 I84 R8 L10 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8031777 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htf A 2.2 BS01 G26 A 1 D25 G27 A28 D29 D30 V32 G48 D25 G27 A28 D29 D30 V32 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=148nM remove_due_to_license_issue P03366 8031777 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htf A 2.2 BS02 G26 B 1 R8 D25 G27 I50 R8 D25 G27 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=148nM remove_due_to_license_issue P03366 8031777 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htf B 2.2 BS01 G26 A 1 R8 D25 G27 P81 V82 R8 D25 G27 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=148nM remove_due_to_license_issue P03366 8031777 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htf B 2.2 BS02 G26 B 1 D25 A28 D29 D30 V32 G48 V82 I84 D25 A28 D29 D30 V32 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=148nM remove_due_to_license_issue P03366 8031777 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htg A 2.0 BS01 G37 A 1 D25 G27 A28 D29 D30 V32 I47 G48 V82 I84 D25 G27 A28 D29 D30 V32 I47 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=3.8nM remove_due_to_license_issue P03366 8031777 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htg A 2.0 BS02 G37 A 2 R8 D25 G27 D30 I47 G48 I50 R8 D25 G27 D30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=3.8nM remove_due_to_license_issue P03366 8031777 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htg B 2.0 BS01 G37 A 1 R8 D25 G27 D29 D30 I47 I50 R8 D25 G27 D29 D30 I47 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8031777 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1htg B 2.0 BS02 G37 A 2 D25 G27 A28 D29 V32 I47 G48 F53 I84 D25 G27 A28 D29 V32 I47 G48 F53 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 8031777 600 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hti B 2.8 BS01 PGA B 1 N11 K13 H95 E165 I170 G210 L230 G232 N11 K13 H95 E165 I170 G210 L230 G232 N11 K13 H95 E97 E165 G171 S211 N11 K13 H95 E97 E165 G171 S211 4.2.3.3,5.3.1.1 0004807,0005515,0005615,0005634,0005737,0005829,0006006,0006094,0006096,0008929,0016829,0016853,0019242,0019563,0019682,0031625,0042803,0046166,0061621,0070062 remove_due_to_license_issue P60174 8061610 549 APSRKFFVGGNWKMNGRKQSLGELIGTLNAAKVPADTEVVCAPPTAYIDFARQKLDPKIAVAAQNCYKVTNGAFTGEISPGMIKDCGATWVVLGHSERRHVFGESDELIGQKVAHALAEGLGVIACIGEKLDEREAGITEKVVFEQTKVIADNVKDWSKVVLAYEPVWAIGTGKTATPQQAQEVHEKLRGWLKSNVSDAVAQSTRIIYGGSVTGATCKELASQPDVDGFLVGGASLKPEFVDIINAKQ 1hv5 A 2.6 BS04 RXP A 1 L172 G179 I180 L181 A182 A184 Q215 H219 E220 F240 Y241 L72 G79 I80 L81 A82 A84 Q115 H119 E120 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=5nM Q02853 11254383 6001 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYG 1hvh A 1.8 BS01 Q82 B 1 R8 D25 A28 D30 I50 R8 D25 A28 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9554878 265 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1hvh B 1.8 BS01 Q82 B 1 D25 G27 G49 I50 P81 V82 D25 G27 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=11nM remove_due_to_license_issue P04585 9554878 265 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1hvi A 1.8 BS01 A77 A 1 R8 D25 G27 D29 G48 G49 I50 V82 R8 D25 G27 D29 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=84pM remove_due_to_license_issue O92139 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvi B 1.8 BS01 A77 A 1 R8 D25 G27 A28 D29 G48 G49 R8 D25 G27 A28 D29 G48 G49 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O92139 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvj A 2.0 BS01 A78 A 1 R8 D25 D29 G48 G49 I50 P81 V82 R8 D25 D29 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4pM remove_due_to_license_issue P04587 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvj B 2.0 BS01 A78 A 1 R8 D25 G27 A28 D29 G48 G49 I50 R8 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvk A 1.8 BS01 A79 A 1 R8 D25 G27 A28 D29 G48 G49 I50 P81 V82 R8 D25 G27 A28 D29 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=77pM remove_due_to_license_issue P03366 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvk B 1.8 BS01 A79 A 1 R8 D25 G27 A28 D29 G48 G49 I50 V82 I84 R8 D25 G27 A28 D29 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvl A 1.8 BS01 A76 B 1 R8 D25 G27 D29 G48 G49 I50 P81 R8 D25 G27 D29 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvl B 1.8 BS01 A76 B 1 R8 D25 G27 A28 D29 G48 G49 I50 V82 R8 D25 G27 A28 D29 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1000pM remove_due_to_license_issue P03367 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hvr A 1.8 BS01 XK2 A 1 D25 G27 A28 D30 I47 G49 I50 D25 G27 A28 D30 I47 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.31nM remove_due_to_license_issue P04585 8278812 263 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1hvr B 1.8 BS01 XK2 A 1 D25 G27 A28 D30 V32 G49 I50 D25 G27 A28 D30 V32 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 8278812 263 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1hvs A 2.25 BS01 A77 A 1 R8 D25 G27 D29 G48 G49 I50 A82 I84 R8 D25 G27 D29 G48 G49 I50 A82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=50pM remove_due_to_license_issue P04587 7773792 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 1hvs B 2.25 BS01 A77 A 1 R8 D25 A28 D29 G48 G49 I50 P81 I84 R8 D25 A28 D29 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 7773792 800 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 1hvy A 1.9 BS01 D16 A 1 F80 I108 W109 D218 L221 G222 F225 Y258 M311 F55 I83 W84 D193 L196 G197 F200 Y233 M286 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue IC50=29000nM P04818 11329255 414 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 1hvy B 1.9 BS02 D16 B 1 I108 W109 N112 D218 L221 G222 F225 Y258 M311 I83 W84 N87 D193 L196 G197 F200 Y233 M286 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue IC50=29000nM P04818 11329255 415 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 1hwr A 1.8 BS01 216 B 1 D25 G27 A28 I50 P81 V82 D25 G27 A28 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9575185 216 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1hwr B 1.8 BS01 216 B 1 D25 G27 A28 G49 I50 V82 D25 G27 A28 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.7nM remove_due_to_license_issue P04585 9575185 216 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1hww A 1.87 BS02 SWA A 1 H90 D92 W95 D204 F206 R228 D341 W415 H471 D472 Y727 H60 D62 W65 D174 F176 R198 D311 W385 H441 D442 Y697 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=20nM remove_due_to_license_issue IC50=37nM, Ki=3.0nM Q24451 11406577 1103 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 1hxb A 2.3 BS01 ROC A 1 D25 G27 D29 D30 I47 G48 I50 P81 I84 D25 G27 D29 D30 I47 G48 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.12nM remove_due_to_license_issue P04585 1956054 100 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hxb B 2.3 BS01 ROC A 1 R8 D25 G27 G49 I50 V82 R8 D25 G27 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 1956054 100 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hxk A 1.5 BS02 DMJ A 1 H90 D92 W95 D204 F206 H471 D472 Y727 R876 H60 D62 W65 D174 F176 H441 D442 Y697 R846 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=400uM remove_due_to_license_issue Q24451 11406577 1103 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 1hxw A 1.8 BS01 RIT B 1 D25 G27 G48 G49 V82 I84 D25 G27 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 7708670 301 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hxw B 1.8 BS01 RIT B 1 R8 D25 G27 D30 G49 I50 P81 V82 R8 D25 G27 D30 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=15pM remove_due_to_license_issue P12499 7708670 301 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hy7 B 1.5 BS06 MBS B 1 V663 L664 A665 H666 H701 E702 H711 L718 Y720 P721 L722 Y723 V81 L82 A83 H84 H119 E120 H129 L136 Y138 P139 L140 Y141 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=4090nM remove_due_to_license_issue IC50=4090nM P08254 11297453 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYLTDLTRFRLSQDDINGIQSLYGPPPDSPET 1hyv A 1.7 BS01 TTA A 1 D167 Q168 A169 T174 D104 Q105 A106 T111 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50>5mM remove_due_to_license_issue P12497 11264582 304 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGYSAGERIVDIIATDIQT 1i00 A 2.5 BS02 D16 A 1 F80 I108 D218 L221 G222 F225 Y258 F52 I80 D190 L193 G194 F197 Y230 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 Ki=0.46uM remove_due_to_license_issue IC50=29000nM P04818 11316879 315 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 1i00 B 2.5 BS03 D16 B 1 F80 W109 D218 L221 G222 F225 Y258 F52 W81 D190 L193 G194 F197 Y230 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 Ki=0.46uM remove_due_to_license_issue IC50=29000nM P04818 11316879 409 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 1i1e A 2.5 BS01 DM2 A 1 E1188 E1189 G1238 I1239 H1240 R1241 C1257 S1259 W1261 Y1262 E1185 E1186 G1235 I1236 H1237 R1238 C1254 S1256 W1258 Y1259 H229 E230 H233 E267 R369 H229 E230 H233 E267 R369 3.4.24.69 0004222,0005515,0005576,0006508,0008237,0008270,0008289,0008320,0016020,0020002,0030430,0035821,0044161,0044164,0044221,0044231,0046872,0071806,0090729 Kd=9.4uM remove_due_to_license_issue P10844 11679763 3001 PVTINNFNYNDPIDNNNIIMMEPPFARGTGRYYKAFKITDRIWIIPERYTFGYKPEDFNKSSGIFNRDVCEYYDPDYLNTNDKKNIFLQTMIKLFNRIKSKPLGEKLLEMIINGIPYLGDRRVPLEEFNTNIASVTVNKLISNPGEVERKKGIFANLIIFGPGPVLNENETIDIGIQNHFASREGFGGIMQMKFCPEYVSVFNNVQENKGASIFNRRGYFSDPALILMHELIHVLHGLYGIKVDDLPIVPNEKKFFMQSTDAIQAEELYTFGGQDPSIITPSTDKSIYDKVLQNFRGIVDRLNKVLVCISDPNININIYKNKFKDKYKFVEDSEGKYSIDVESFDKLYKSLMFGFTETNIAENYKIKTRASYFSDSLPPVKIKNLLDNEIYTIEEGFNISDKDMEKEYRGQNKAINKQAYEEISKEHLAVYKIQMCKSVGICIDVDNEDLFFIADKNSFSDDLSKNERIEYNTQSNYIENDFPINELILDTDLISKIELPSENTESLTDFNVDVPVYEKQPAIKKIFTDENTIFQYLYSQTFPLDIRDISLTSSFDDALLFSNKVYSFFSMDYIKTANKVVEAGLFAGWVKQIVNDFVIEANKSNTMDKIADISLIVPYIGLALNVGNETAKGNFENAFEIAGASILLEFIPELLIPVVGAFLLESYIDNKNKIIKTIDNALTKRNEKWSDMYGLIVAQWLSTVNTQFYTIKEGMYKALNYQAQALEEIIKYRYNIYSEKEKSNINIDFNDINSKLNEGINQAIDNINNFINGCSVSYLMKKMIPLAVEKLLDFDNTLKKNLLNYIDENKLYLIGSAEYEKSKVNKYLKTIMPFDLSIYTNDTILIEMFNKYNSEILNNIILNLRYKDNNLIDLSGYGAKVEVYDGVELNDKNQFKLTSSANSKIRVTQNQNIIFNSVFLDFSVSFWIRIPKYKNDGIQNYIHNEYTIINCMKNNSGWKISIRGNRIIWTLIDINGKTKSVFFEYNIREDISEYINRWFFVTITNNLNNAKIYINGKLESNTDIKDIREVIANGEIIFKLDGDIDRTQFIWMKYFSIFNTELSQSNIEERYKIQSYSEYLKDFWGNPLMYNKEYYMFNAGNKNSYIKLKKDSPVGEILTRSKYNQNSKYINYRDLYIGEKFIIRRKSNSQSINDDIVRKEDYIYLDFFNLNQEWRVYTYKYFKKEEEKLFLAPISDSDEFYNTIQIKEYDEQPTYSCQLLFKKDEESTDEIGLIGIHRFYESGIVFEEYKDYFCISKWYLKEVKRKPYNLKLGCNWQFIPKDEGWTE 1i32 A 2.6 BS01 NMD A 1 G9 D38 M39 S40 A90 Q91 R92 T111 G9 D38 M39 S40 A90 Q91 R92 T111 C166 H194 C166 H194 1.2.1.12 0004365,0005829,0006006,0006096,0016491,0016620,0020015,0050661,0051287 remove_due_to_license_issue Q27890 11371162 361 APIKVGINGFGRIGRMVFQAICDQGLIGTEIDVVAVVDMSTNAEYFAYQMKHDTVHGRPKYTVEAVKSSPSVETADVLVVNGHRIKCVKAQRNPADLPWGKLGVDYVIESTGLFTDKLKAEGHIKGGAKKVVISAPASGGAKTIVMGVNQHEYSPASHHVVSNASCTTNCLAPIVHVLTKENFGIETGLMTTIHSYTATQKTVDGVSLKDWRGGRAAAVNIIPSTTGAAKAVGMVIPSTKGKLTGMSFRVPTPDVSVVDLTFRATRDTSIQEIDKAIKKAAQTYMKGILGFTDEELVSADFINDNRSSVYDSKATLQNNLPGEKRFFKVVSWYDNEWAYSHRVVDLVRYMAAKDAASS 1i32 B 2.6 BS01 NMD B 1 G9 G11 D38 M39 S40 A90 Q91 R92 T111 L113 G9 G11 D38 M39 S40 A90 Q91 R92 T111 L113 C166 H194 C166 H194 1.2.1.12 0004365,0005829,0006006,0006096,0016491,0016620,0020015,0050661,0051287 remove_due_to_license_issue Q27890 11371162 362 APIKVGINGFGRIGRMVFQAICDQGLIGTEIDVVAVVDMSTNAEYFAYQMKHDTVHGRPKYTVEAVKSSPSVETADVLVVNGHRIKCVKAQRNPADLPWGKLGVDYVIESTGLFTDKLKAEGHIKGGAKKVVISAPASGGAKTIVMGVNQHEYSPASHHVVSNASCTTNCLAPIVHVLTKENFGIETGLMTTIHSYTATQKTVDGVSLKDWRGGRAAAVNIIPSTTGAAKAVGMVIPSTKGKLTGMSFRVPTPDVSVVDLTFRATRDTSIQEIDKAIKKAAQTYMKGILGFTDEELVSADFINDNRSSVYDSKATLQNNLPGEKRFFKVVSWYDNEWAYSHRVVDLVRYMAAKDAASS 1i33 A 3.0 BS01 TND A 1 G9 G11 D38 M39 S40 A90 Q91 R92 G9 G11 D38 M39 S40 A90 Q91 R92 C166 H194 C166 H194 1.2.1.12 0004365,0005829,0006006,0006096,0016491,0016620,0020015,0050661,0051287 remove_due_to_license_issue Q27890 11371162 361 APIKVGINGFGRIGRMVFQAICDQGLIGTEIDVVAVVDMSTNAEYFAYQMKHDTVHGRPKYTVEAVKSSPSVETADVLVVNGHRIKCVKAQRNPADLPWGKLGVDYVIESTGLFTDKLKAEGHIKGGAKKVVISAPASGGAKTIVMGVNQHEYSPASHHVVSNASCTTNCLAPIVHVLTKENFGIETGLMTTIHSYTATQKTVDGVSLKDWRGGRAAAVNIIPSTTGAAKAVGMVIPSTKGKLTGMSFRVPTPDVSVVDLTFRATRDTSIQEIDKAIKKAAQTYMKGILGFTDEELVSADFINDNRSSVYDSKATLQNNLPGEKRFFKVVSWYDNEWAYSHRVVDLVRYMAAKDAASS 1i33 B 3.0 BS01 TND A 1 V206 L208 V206 L208 C166 H194 C166 H194 1.2.1.12 0004365,0005829,0006006,0006096,0016491,0016620,0020015,0050661,0051287 remove_due_to_license_issue Q27890 11371162 361 APIKVGINGFGRIGRMVFQAICDQGLIGTEIDVVAVVDMSTNAEYFAYQMKHDTVHGRPKYTVEAVKSSPSVETADVLVVNGHRIKCVKAQRNPADLPWGKLGVDYVIESTGLFTDKLKAEGHIKGGAKKVVISAPASGGAKTIVMGVNQHEYSPASHHVVSNASCTTNCLAPIVHVLTKENFGIETGLMTTIHSYTATQKTVDGVSLKDWRGGRAAAVNIIPSTTGAAKAVGMVIPSTKGKLTGMSFRVPTPDVSVVDLTFRATRDTSIQEIDKAIKKAAQTYMKGILGFTDEELVSADFINDNRSSVYDSKATLQNNLPGEKRFFKVVSWYDNEWAYSHRVVDLVRYMAAKDAASS 1i33 B 3.0 BS02 TND B 1 G9 G11 D38 M39 S40 A90 Q91 R92 T111 L113 G9 G11 D38 M39 S40 A90 Q91 R92 T111 L113 C166 H194 C166 H194 1.2.1.12 0004365,0005829,0006006,0006096,0016491,0016620,0020015,0050661,0051287 remove_due_to_license_issue Q27890 11371162 362 APIKVGINGFGRIGRMVFQAICDQGLIGTEIDVVAVVDMSTNAEYFAYQMKHDTVHGRPKYTVEAVKSSPSVETADVLVVNGHRIKCVKAQRNPADLPWGKLGVDYVIESTGLFTDKLKAEGHIKGGAKKVVISAPASGGAKTIVMGVNQHEYSPASHHVVSNASCTTNCLAPIVHVLTKENFGIETGLMTTIHSYTATQKTVDGVSLKDWRGGRAAAVNIIPSTTGAAKAVGMVIPSTKGKLTGMSFRVPTPDVSVVDLTFRATRDTSIQEIDKAIKKAAQTYMKGILGFTDEELVSADFINDNRSSVYDSKATLQNNLPGEKRFFKVVSWYDNEWAYSHRVVDLVRYMAAKDAASS 1i37 A 2.0 BS01 DHT A 1 L704 N705 L707 Q711 M745 M749 F764 M780 T877 M895 L33 N34 L36 Q40 M74 M78 F93 M109 T206 M224 ? remove_due_to_license_issue IC50=3.1nM, EC50=0.97nM, Ki=0.43nM P15207 11320241 201 IFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 1i41 A 3.2 BS01 HEN A 1 G138 M139 Y163 E207 D236 T238 S258 T260 K261 P387 S388 R423 G89 M90 Y114 E158 D187 T189 S209 T211 K212 P338 S339 R374 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 500 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i41 A 3.2 BS02 HEN C 1 E107 Y108 R110 Y111 E58 Y59 R61 Y62 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 502 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i41 C 3.2 BS01 HEN A 1 E107 Y108 R110 Y111 E58 Y59 R61 Y62 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 500 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i41 C 3.2 BS02 HEN C 1 S137 G138 M139 Y163 E207 D236 S258 T260 K261 S388 F389 S403 R423 S88 G89 M90 Y114 E158 D187 S209 T211 K212 S339 F340 S354 R374 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 502 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i43 A 3.1 BS02 PMC A 1 Y163 K261 P387 S403 R423 Y114 K212 P338 S354 R374 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 600 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i43 A 3.1 BS04 PMC C 1 E107 Y111 E58 Y62 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 602 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i43 C 3.1 BS02 PMC A 1 E107 Y108 Y111 E58 Y59 Y62 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 600 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i43 C 3.1 BS04 PMC C 1 Y163 K261 P387 S403 R423 Y114 K212 P338 S354 R374 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 602 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i48 A 3.25 BS02 CCO A 1 Y163 R164 A386 P387 S388 D397 S403 R423 S425 Y114 R115 A337 P338 S339 D348 S354 R374 S376 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 600 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i48 C 3.25 BS03 CCO C 1 Y163 R164 A386 P387 S388 F389 D397 S403 R423 S425 Y114 R115 A337 P338 S339 F340 D348 S354 R374 S376 R110 Y163 D236 K261 R61 Y114 D187 K212 4.2.99.9 0003962,0009086,0019346,0030170 remove_due_to_license_issue Q9ZPL5 11518531 602 YASFLNSDGSVAIHAGERLGRGIVTDAITTPVVNTSAYFFNKTSELIDFKEKRRASFEYGRYGNPTTVVLEEKISALEGAESTLLMASGMCASTVMLLALVPAGGHIVTTTDCYRKTRIFIETILPKMGITATVIDPADVGALELALNQKKVNLFFTESPTNPFLRCVDIELVSKLCHEKGALVCIDGTFATPLNQKALALGADLVLHSATKFLGGHNDVLAGCISGPLKLVSEIRNLHHILGGALNPNAAYLIIRGMKTLHLRVQQQNSTALRMAEILEAHPKVRHVYYPGLQSHPEHHIAKKQMTGFGGAVSFEVDGDLLTTAKFVDALKIPYIAPSFGGCESIVDQPAIMSYWDLSQSDRAKYGIMDNLVRFSFGVEDFDDLKADILQALDSI 1i5d A 2.9 BS01 128 A 1 H413 G414 I454 K458 I459 K462 K494 H64 G65 I105 K109 I110 K113 K145 N409 N60 2.7.13.3 0016310,0016772 remove_due_to_license_issue Q56310 11276258 999 VMKIRMVPISFVFNRFPRMVRDLAKKMNKEVNFIMRGEDTELDRTFVEEIGEPLLHLLRNAIDHGIEPKEERIAKGKPPIGTLILSARHEGNNVVIEVEDDGRGIDKEKIIRKAIEKGLIDESKAATLSDQEILNFLFVPGFSTKEKVSEVSGRGVGMDVVKNVVESLNGSISIESEKDKGTKVTIRLPL 1i5r A 1.6 BS01 HYC A 1 G9 S11 S12 R37 L64 D65 V66 R67 A91 G92 L93 G94 S142 G144 M147 L149 Y155 G186 F192 M193 Y218 H221 V225 F259 G9 S11 S12 R37 L64 D65 V66 R67 A91 G92 L93 G94 S142 G144 M147 L149 Y155 G186 F192 M193 Y218 H221 V225 F259 1.1.1.51,1.1.1.62 0003824,0004303,0005496,0005515,0005737,0005829,0006629,0006694,0006703,0007040,0007519,0008210,0010467,0016491,0030283,0036094,0042803,0047035,0047045,0050661,0060348,0060612,0061370,0070401,0071248,0072582,1903924 Ki=3nM remove_due_to_license_issue IC50=52nM, Ki=3nM P14061 12223444 328 ARTVVLITGCSSGIGLHLAVRLASDPSQSFKVYATLRDLKTQGRLWEAARALACPPGSLETLQLDVRDSKSVAAARERVTEGRVDVLVCNAGLGLLGPLEALGEDAVASVLDVNVVGTVRMLQAFLPDMKRRGSGRVLVTGSVGGLMGLPFNDVYCASKFALEGLCESLAVLLLPFGVHLSLIECGPVHTAFMEKVLGSPEEVLDRTDIHTFHRFYQYLAHSKQVFREAAQNPEEVAEVFLTALRAPKPTLRYFTTERFLPLLRMRLDDPSGSNYVTAMHREVFG 1i6v C 3.3 BS01 RFP C 1 Q390 S392 Q393 F394 D396 R409 S411 E445 I452 Q389 S391 Q392 F393 D395 R408 S410 E444 I451 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue Q9KWU7 11290327 1640 KIKRFGRIREVIPLPPLTEIQVESYKKALQADVPPEKRENVGIQAAFKETFPIEEGDKGKGGLVLDFLEYRIGDPPFSQDECREKDLTYQAPLYARLQLIHKDTGLIKEDEVFLGHLPLMTEDGSFIINGADRVIVSQIHRSPGVYFTPDPARPGRYIASIIPLPKRGPWIDLEVEASGVVTMKVNKRKFPLVLLLRVLGYDQETLVRELSAYGDLVQGLLDEAVLAMRPEEAMVRLFTLLRPGDPPKKDKALAYLFGLLADPKRYDLGEAGRYKAEEKLGVGLSGRTLVRFEDGEFKDEVFLPTLRYLFALTAGVPGHEVDDIDHLGNRRIRTVGELMADQFRVGLARLARGVRERMVMGSPDTLTPAKLVNSRPLEAALREFFSRSQLSQFKDETNPLSSLRHKRRISALGPGGLTRERAGFDVRDVHRTHYGRICPVETPEGANIGLITSLAAYARVDALGFIRTPYRRVKNGVVTEEVVYMTASEEDRYTIAQANTPLEGDRIATDRVVARRRGEPVIVAPEEVEFMDVSPKQVFSLNTNLIPFLEHDDANRALMGSNMQTQAVPLIRAQAPVVMTGLEERVVRDSLAALYAEEDGEVVKVDGTRIAVRYEDGRLVHPLRRYARSNQGTAFDQRPRVRVGQRVKKGDLLADGPASEEGFLALGQNVLVAIMPFDGYNFEDAIVISEELLKRDFYTSIHIERYEIEARDTKLGPERITRDIPHLSEAALRDLDEEGIVRIGAEVKPGDILVGRTSFKGEQEPSPEERLLRSIFGEKARDVKDTSLRVPPGEGGIVVGRLRLRRGDPGVELKPGVREVVRVFVAQKRKLQVGDKLANRHGNKGVVAKILPVEDMPHLPDGTPVDVILNPLGVPSRMNLGQILETHLGLAGYFLGQRYISPVFDGATEPEIKELLAEAFNLYFGKRQGEGFGVDKREKEVLARAEKLGLVSPGKSPEEQLKELFDLGKVVLYDGRTGEPFEGPIVVGQMFIMKLYHMVEDKMHARSTGPYSLITQQPLGGKAQFGGQRFGEMEVWALEAYGAAHTLQEMLTIKSDDIEGRNAAYQAIIKGEDVPEPSVPESFRVLVKELQALALDVQTLDEKDNPVDVFEGL 1i72 A 2.0 BS01 MAO A 1 X68 F223 C226 G227 Y228 S229 H243 I244 T245 E247 X1 F152 C155 G156 Y157 S158 H172 I173 T174 E176 S229 H243 S157 H171 4.1.1.50 0004014,0006597,0008295 remove_due_to_license_issue IC50=55nM P17707 11583147 368 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAGYCMGRMNSDCWYLYTLDFPESQPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQSSKCRPQKIEGFKRLDCQSAMFNDYNFVFTSFAKK 1i72 B 2.0 BS01 MAO A 1 F7 L65 S66 E67 F4 L59 S60 E61 E67 E61 4.1.1.50 0004014,0008295 remove_due_to_license_issue IC50=55nM P17707 11583147 368 AHFFEGTEKLLEVWFSRQQPQGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 1i7c A 2.4 BS02 MGB A 1 X68 F223 C226 S229 E247 X1 F156 C159 S162 E180 S229 H243 S161 H175 4.1.1.50 0004014,0006597,0008295 ic50=0.4uM remove_due_to_license_issue P17707 11583147 375 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAGYCMGRMNSDCWYLYTLDFPESRVISQPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQSTVLASPQKIEGFKRLDCQSAMFNDYNFVFTSFAKKQ 1i7c B 2.4 BS01 MGB A 1 F7 L65 S66 F4 L59 S60 E67 E61 4.1.1.50 0004014,0008295 remove_due_to_license_issue P17707 11583147 375 AHFFEGTEKLLEVWFSRQQPQGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 1i7g A 2.2 BS01 AZ2 A 1 F273 C275 C276 S280 Y314 M330 V332 H440 Y464 F64 C66 C67 S71 Y105 M121 V123 H231 Y255 ? 0003677,0004879,0005634,0006355 ic50=1uM remove_due_to_license_issue EC50=820nM, Ki=1000nM Q07869 11587644 469 ETADLKSLAKRIYEAYLKNFNMNKVKARVILSGSNNPPFVIHDMETLCMAEKTLQNKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANLDLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFDFAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDIFLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDMY 1i7i A 2.35 BS01 AZ2 A 1 F282 G284 C285 S289 H323 I341 M364 H449 L469 Y473 F64 G66 C67 S71 H105 I123 M146 H231 L251 Y255 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=704nM, Ki=18nM P37231 11587644 101 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 1i7m A 2.24 BS02 CG A 1 X68 F223 S229 H243 I244 E247 X1 F149 S155 H169 I170 E173 S229 H243 S154 H168 4.1.1.50 0004014,0006597,0008295 ic50=0.23nM remove_due_to_license_issue P17707 11583147 375 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAGYCMGRMNSDCWYLYTLDFQPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQSSKCPQKIEGFKRLDCQSAMFNDYNFVFTSFAKKQ 1i7m B 2.24 BS01 CG A 1 F7 L65 S66 E67 F4 L55 S56 E57 E67 E57 4.1.1.50 0004014,0008295 remove_due_to_license_issue P17707 11583147 375 AHFFEGTEKLLEVWFSRGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 1i7z A 2.3 BS01 COC A 1 Y32 H34 S91 R92 E93 Y36 H38 S95 R96 E97 ? 0002250,0003823,0005576,0005615,0005886,0006955,0016064,0019814,0050853,0070062,0071735,0071738,0071742,0071745,0071753,0072562 Kd=0.4uM remove_due_to_license_issue P01834 11469854 301 DLVLTQSPASLAVSLGQRATISCRASKSVSTSGYNYMHWYQQKPGQPPKLLIYLASNLASGVPARFSGSGSGTDFTLNIHPVEEEDAATYYCLYSREFPPWTFGGGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 1i7z B 2.3 BS01 COC A 1 Y95 S97 P98 D101 Y99 S101 P102 D105 ? remove_due_to_license_issue P01857 11469854 301 QVQLQQSGPELKKPGETVKISCKTSGYSFTNYGMNWVKQAPGKGLKWMGWINTYTGEPTYADDFRGRFAFSLATSASTAYLQIINLKNEDTATYFCETYDSPLGDYWGQGTTVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 1i80 B 2.0 BS01 9HX B 1 A120 A121 G122 Y188 E189 V205 G206 T230 N231 A115 A116 G117 Y183 E184 V200 G201 T225 N226 S36 H68 H90 Y92 E93 A120 M207 S208 N231 A233 H243 S31 H63 H85 Y87 E88 A115 M202 S203 N226 A228 H238 2.4.2.1 0003824,0004731,0005737,0006139,0006154,0006161,0009116,0016757,0016763 Kd=0.39uM remove_due_to_license_issue P9WP01 11444966 302 PDPDELARRAAQVIADRTGIGEHDVAVVLGSGWLPAVAALGSPTTVLPQAELPGFVPPTAAGHAGELLSVPIGAHRVLVLAGRIHAYEGHDLRYVVHPVRAARAAGAQIMVLTNAAGGLRADLQVGQPVLISDHLNLTARSPLVGGEFVDLTDAYSPRLRELARQSDPQLAEGVYAGLPGPHYETPAEIRMLQTLGADLVGMSTVHETIAARAAGAEVLGVSLVTNLAAGITGEPLSHAEVLAAGAASATRMGALLADVIARF 1i80 C 2.0 BS01 9HX C 1 A120 A121 G122 Y188 E189 V205 G206 M207 T230 N231 A114 A115 G116 Y182 E183 V199 G200 M201 T224 N225 S36 H68 H90 Y92 E93 A120 M207 S208 N231 A233 H243 S30 H62 H84 Y86 E87 A114 M201 S202 N225 A227 H237 2.4.2.1 0003824,0004731,0005737,0006139,0006154,0006161,0009116,0016757,0016763 Kd=0.39uM remove_due_to_license_issue P9WP01 11444966 303 DPDELARRAAQVIADRTGIGEHDVAVVLGSGWLPAVAALGSPTTVLPQAELPGFVPPTAAGHAGELLSVPIGAHRVLVLAGRIHAYEGHDLRYVVHPVRAARAAGAQIMVLTNAAGGLRADLQVGQPVLISDHLNLTARSPLVGGEFVDLTDAYSPRLRELARQSDPQLAEGVYAGLPGPHYETPAEIRMLQTLGADLVGMSTVHETIAARAAGAEVLGVSLVTNLAAGITGEPLSHAEVLAAGAASATRMGALLADVIARF 1i8j A 1.9 BS02 DSB A 1 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue P0ACB2 11444968 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 1i8m A 2.1 BS01 dna D 0 Y92 T94 Y92 T94 ? remove_due_to_license_issue Q7TS98 11733999 2 ~ 3 ELQMTQSPASLSASVGETVTITCRASENIYSYLAWYQQKQGKSPQLLVYNAKTLAEGVPSRFSGSGSGTQFSLKINSLQPEDFGSYYCQHHYGTPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1i8m B 2.1 BS01 dna T 0 Y97 Y102 Y101 Y109 ? remove_due_to_license_issue Q924Q6 11733999 1 ~ 5 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 1i8m B 2.1 BS02 dna D 0 V33 H35 Y100A V33 H35 Y105 ? remove_due_to_license_issue Q924Q6 11733999 2 ~ 3 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 1i8m H 2.1 BS01 dna T 0 Y97 Y100 Y100A A100B Y101 Y104 Y105 A106 ? remove_due_to_license_issue Q924Q6 11733999 1 ~ 5 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 1i8m L 2.1 BS01 dna T 0 Y32 Y49 N50 H91 Y92 Y32 Y49 N50 H91 Y92 ? remove_due_to_license_issue Q7TS98 11733999 1 ~ 5 ELQMTQSPASLSASVGETVTITCRASENIYSYLAWYQQKQGKSPQLLVYNAKTLAEGVPSRFSGSGSGTQFSLKINSLQPEDFGSYYCQHHYGTPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1i8z A 1.93 BS02 INL A 1 Q92 H94 H119 F131 L198 T199 T200 Q90 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=1.27nM remove_due_to_license_issue Ki=0.15nM, IC50=1.3nM P00918 11831900 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i90 A 2.0 BS02 INM A 1 Q92 H94 H119 F131 V143 L198 T199 T200 Q90 H92 H117 F128 V140 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=1.28nM remove_due_to_license_issue P00918 11831900 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i91 A 2.0 BS02 INQ A 1 Q92 H94 H96 H119 L198 T199 T200 Q90 H92 H94 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=1.15nM remove_due_to_license_issue Ki=0.15nM, IC50=1.2nM P00918 11831900 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9l A 1.93 BS02 INV A 1 H94 H96 H119 L198 T199 T200 P202 L204 H92 H94 H117 L195 T196 T197 P199 L201 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.3nM remove_due_to_license_issue P00918 11572683 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9l A 1.93 BS03 INV A 2 F70 D72 I91 V131 V135 F68 D70 I89 V128 V132 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.3nM remove_due_to_license_issue P00918 11572683 666 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9m A 1.84 BS02 INW A 1 Q92 H94 H96 H119 V121 L198 T199 T200 P202 W209 Q90 H92 H94 H117 V119 L195 T196 T197 P199 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.3nM remove_due_to_license_issue P00918 11572683 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9m A 1.84 BS03 INW A 2 E69 F70 D72 I91 E67 F68 D70 I89 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.3nM remove_due_to_license_issue P00918 11572683 666 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9n A 1.86 BS02 IOA A 1 H94 H96 H119 L198 T199 T200 P202 H92 H94 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=2.2nM remove_due_to_license_issue P00918 11572683 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9o A 1.86 BS02 IOC A 1 H94 H96 H119 V135 L198 T199 T200 P202 L204 H92 H94 H117 V132 L195 T196 T197 P199 L201 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.8nM remove_due_to_license_issue Kd=2.3nM P00918 11572683 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9o A 1.86 BS03 IOC A 2 E69 F70 I91 E67 F68 I89 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.8nM remove_due_to_license_issue Kd=2.3nM P00918 11572683 666 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1i9p A 1.92 BS02 IOE A 1 H94 H96 H119 V135 L198 T199 T200 P202 H92 H94 H117 V132 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.9nM remove_due_to_license_issue P00918 11572683 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1ibg H 2.7 BS01 OBN H 1 H35 F95 Y100 Y100C H34 F97 Y102 Y105 remove_due_to_license_issue 7739045 1 VHLVQSGPGLVAPSQSLSITCTVSGFSLTTYGVHWFRQPPGKGLEWLGLIWAGGNTDYNSALMSRLSINKDNSKSQVFLKMNSLQADDTAMYYCARFRFASYYDYAVDYWGQGTSVTVSSAKTTPPSVYPLAPGCGDTTGSSVTSGCLVKGYFPEPVTVTWNSGSLSSSVHTFPALLQSGLYTMSSSVTVPSSTWPSQTVTCSVAHPASSTTVDKKL 1ibg L 2.7 BS01 OBN H 1 T27D H32 S91 Y94 L96 T30 H35 S94 Y97 L99 remove_due_to_license_issue 7739045 1 IVLTQSPASLAVSLGQRATISCRASKSVSTSGYSHIHWYQQKPGQPPKLLIYLASILESGVPARFSGSGSGTDFTLNIHPVEEEDAATYYCQHSREYPLTFGAGTELELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 1ida A 1.7 BS01 0PO B 1 R8 D25 D30 G48 G49 P81 R8 D25 D30 G48 G49 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 7743130 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1ida B 1.7 BS01 0PO B 1 D25 G27 A28 D29 G48 G49 I50 P81 I82 I84 D25 G27 A28 D29 G48 G49 I50 P81 I82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 ic50<2nM remove_due_to_license_issue P04584 7743130 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1idb A 2.2 BS01 0DO B 1 D25 G27 G48 G49 I50 I84 D25 G27 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 7743130 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1idb B 2.2 BS01 0DO B 1 D25 G27 A28 D29 D30 V47 G49 I50 P81 I82 D25 G27 A28 D29 D30 V47 G49 I50 P81 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 ic50=11nM remove_due_to_license_issue P04584 7743130 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1ie9 A 1.4 BS01 VDX A 1 Y143 L233 S237 R274 S275 S278 W286 H305 H397 Y26 L65 S69 R106 S107 S110 W118 H137 H229 ? 0003677,0004879,0006355 remove_due_to_license_issue EC50=10nM, IC50=1.1nM, Kd=0.065nM P11473 11344298 500 DSLRPKLSEEQQRIIAILLDAHHKTYDPTYSDFCQFRPPVRVNDGGGSVTLELSQLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSEDQIVLLKSSAIEVIMLRSNESFTMDDMSWTCGNQDYKYRVSDVTKAGHSLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAALIEAIQDRLSNTLQTYIRCRHPPPGSHLLYAKMIQKLADLRSLNEEHSKQYRCLSFQPECSMKLTPLVLEVFG 1iem A 2.3 BS01 CB4 A 1 S64 Y150 N152 Y221 A318 G320 S61 Y147 N149 Y218 A315 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 11478888 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1iep A 2.1 BS01 STI A 1 L248 Y253 A269 K271 E286 M290 V299 I313 T315 F317 M318 I360 H361 R362 A380 D381 F382 L24 Y29 A45 K47 E62 M66 V75 I89 T91 F93 M94 I136 H137 R138 A156 D157 F158 D363 A365 R367 N368 D381 P402 D139 A141 R143 N144 D157 P178 2.7.10.2 0004672,0004713,0005524,0006468 ic50=100nM remove_due_to_license_issue IC50=10.8nM P00520 12154025 201 MDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ 1iew A 2.55 BS01 G2F A 1 D95 R158 K206 H207 Y253 D285 W286 M316 D95 R158 K206 H207 Y253 D285 W286 M316 D285 E491 D285 E491 3.2.1.21 0004553,0005975,0016798 remove_due_to_license_issue Q9XEI3 11709165 620 DYVLYKDATKPVEDRVADLLGRMTLAEKIGQMTQIERLVATPDVLRDNFIGSLLSGGGSVPRKGATAKEWQDMVDGFQKACMSTRLGIPMIYGIDAVHGQNNVYGATIFPHNVGLGATRDPYLVKRIGEATALEVRATGIQYAFAPCIAVCRDPRWGRCYESYSEDRRIVQSMTELIPGLQGDVPKDFTSGMPFVAGKNKVAACAKHFVGDGGTVDGINENNTIINREGLMNIHMPAYKNAMDKGVSTVMISYSSWNGVKMHANQDLVTGYLKDTLKFKGFVISDWEGIDRITTPAGSDYSYSVKASILAGLDMIMVPNKYQQFISILTGHVNGGVIPMSRIDDAVTRILRVKFTMGLFENPYADPAMAEQLGKQEHRDLAREAARKSLVLLKNGKTSTDAPLLPLPKKAPKILVAGSHADNLGYQCGGWTIEWQGDTGRTTVGTTILEAVKAAVDPSTVVVFAENPDAEFVKSGGFSYAIVAVGEHPYTETKGDNLNLTIPEPGLSTVQAVCGGVRCATVLISGRPVVVQPLLAASDALVAAWLPGSEGQGVTDALFGDFGFTGRLPRTWFKSVDQLPMNVGDAHYDPLFRLGYGLTTNAT 1if7 A 1.98 BS02 SBR A 1 H94 H96 H119 L198 T199 T200 H92 H94 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=30pM remove_due_to_license_issue P00918 11818565 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1if8 A 1.94 BS02 SBS A 1 H94 H96 H119 L198 T199 T200 P202 H92 H94 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=230pM remove_due_to_license_issue P00918 11818565 555 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1igb A 2.3 BS03 IPO A 1 D117 E151 E152 D179 C223 C227 F244 F248 Y251 H256 D117 E151 E152 D179 C223 C227 F244 F248 Y251 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=0.4uM remove_due_to_license_issue Q01693 8647077 520 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 1igj D 2.5 BS01 DGX D 1 Y33 N35 Y47 Y50 S95 W100 A100A M100B Y32 N34 Y46 Y49 S98 W103 A104 M105 Kd=0.1nM remove_due_to_license_issue 8234291 228 VQLQQSGPELVKPGASVRMSCKSSGYIFTDFYMNWVRQSHGKSLDYIGYISPYSGVTGYNQKFKGKATLTVDKSSSTAYMELRSLTSEDSAVYYCAGSSGNKWAMDYWGHGASVTVSSAKTTAPSVYPLAPVCGDTTGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEP 1ign A 2.25 BS01 dna C 0 K360 A361 S362 F363 H398 T399 N401 S402 H405 R406 Y410 K446 R447 F449 H536 T537 N539 D543 R544 F548 K575 N576 T578 T588 P589 G590 N591 N593 S594 K1 A2 S3 F4 H39 T40 N42 S43 H46 R47 Y51 K87 R88 F90 H146 T147 N149 D153 R154 F158 K178 N179 T181 T183 P184 G185 N186 N188 S189 ? 0000723,0003677 remove_due_to_license_issue P11938 8620531 1 ~ 19 KASFTDEEDEFILDVVRKNPTRRTTHTLYDEISHYVPNHTGNSIRHRFRVYLSKRLEYVYEVDKFGKLVRDDDGNLIKTKVLPPSIKRKFSADEDYTLAIAVKKQFYRDLFQIDPDTGRSLIRTQSRRGPIAREFFKHFAEEHAAHTENAWRDRFRKFLLAYGIDDYISYYEAEEPMKNLTPTPGNYNS 1ign A 2.25 BS02 dna D 0 K360 T383 T384 H385 T386 R404 R408 S444 I445 K446 R518 P520 I521 R523 E524 E538 R542 R546 P589 G590 K1 T24 T25 H26 T27 R45 R49 S85 I86 K87 R128 P130 I131 R133 E134 E148 R152 R156 P184 G185 ? 0000723,0003677 remove_due_to_license_issue P11938 8620531 20 ~ 38 KASFTDEEDEFILDVVRKNPTRRTTHTLYDEISHYVPNHTGNSIRHRFRVYLSKRLEYVYEVDKFGKLVRDDDGNLIKTKVLPPSIKRKFSADEDYTLAIAVKKQFYRDLFQIDPDTGRSLIRTQSRRGPIAREFFKHFAEEHAAHTENAWRDRFRKFLLAYGIDDYISYYEAEEPMKNLTPTPGNYNS 1ign B 2.25 BS01 dna E 0 K360 A361 S362 F363 H398 T399 N401 S402 H405 R406 Y410 K446 R447 F449 H536 T537 N539 A540 D543 R544 F548 K575 N576 T578 T588 P589 G590 N591 N593 S594 K1 A2 S3 F4 H39 T40 N42 S43 H46 R47 Y51 K87 R88 F90 H146 T147 N149 A150 D153 R154 F158 K178 N179 T181 T183 P184 G185 N186 N188 S189 ? 0000723,0003677 remove_due_to_license_issue P11938 8620531 2 ~ 19 KASFTDEEDEFILDVVRKNPTRRTTHTLYDEISHYVPNHTGNSIRHRFRVYLSKRLEYVYEVDKFGKLVRDDDGNLIKTKVLPPSIKRKFSADEDYTLAIAVKKQFYRDLFQIDPDTGRSLIRTQSRRGPIAREFFKHFAEEHAAHTENAWRDRFRKFLLAYGIDDYISYYEAEEPMKNLTPTPGNYNS 1ign B 2.25 BS02 dna F 0 T383 T384 H385 T386 R404 R408 S444 I445 R518 P520 I521 R523 E524 E538 R542 R546 T24 T25 H26 T27 R45 R49 S85 I86 R128 P130 I131 R133 E134 E148 R152 R156 ? 0000723,0003677 remove_due_to_license_issue P11938 8620531 20 ~ 38 KASFTDEEDEFILDVVRKNPTRRTTHTLYDEISHYVPNHTGNSIRHRFRVYLSKRLEYVYEVDKFGKLVRDDDGNLIKTKVLPPSIKRKFSADEDYTLAIAVKKQFYRDLFQIDPDTGRSLIRTQSRRGPIAREFFKHFAEEHAAHTENAWRDRFRKFLLAYGIDDYISYYEAEEPMKNLTPTPGNYNS 1ih0 A -1.00 BS03 EMD A 1 F104 L121 T124 L136 G140 I148 F153 F156 M157 V160 E161 F14 L31 T34 L46 G50 I58 F63 F66 M67 V70 E71 ? 0005509 remove_due_to_license_issue P63316 11320096 1 GKSEEELSDLFRMFDKNADGYIDLEELKIMLQATGETITEDDIEELMKDGDKNNDGRIDYDEFLEFMKGVE 1ihy A 3.0 BS01 APR A 1 G9 R10 I11 D32 P33 F34 M77 T96 T179 A180 G9 R10 I11 D31 P32 F33 M76 T95 T178 A179 1.2.1.12 0004365,0005737,0005829,0006006,0006096,0016491,0016620,0050661,0051287 remove_due_to_license_issue P56649 12136140 335 SKIGINGFGRIGRLVLRTALEMGAQVVAVNDPFIALEYMVYMFKYDSTHGMFKGEVKVEDGALVVDGKKITVFNEMKPENIPWSKAGAEYIVESTGVFTTIEKASAHFKGGAKKVIISAPSADAPMFVCGVNLEKYSKDMKVVSNASCTTNCLAPVAKVLHENFEIVEGLMTTVHAVTATQKTVDGPSAKDWRGGRGAAQNIIPSSTGAAKAVGKVIPELDGKLTGMAFRVPTPNVSVVDLTVRLGKECSYDDIKAAMKTASEGPLQGVLGYTEDDVVSCDFTGDNRSSIFDAKAGIQLSKTFVKVVSWYDNEFGYSQRVIDLIKHMQKVDSA 1ihy C 3.0 BS01 APR C 1 G9 R10 I11 D32 P33 F34 M77 T96 F99 T179 A180 G9 R10 I11 D31 P32 F33 M76 T95 F98 T178 A179 1.2.1.12 0004365,0005737,0005829,0006006,0006096,0016491,0016620,0050661,0051287 remove_due_to_license_issue P56649 12136140 338 SKIGINGFGRIGRLVLRTALEMGAQVVAVNDPFIALEYMVYMFKYDSTHGMFKGEVKVEDGALVVDGKKITVFNEMKPENIPWSKAGAEYIVESTGVFTTIEKASAHFKGGAKKVIISAPSADAPMFVCGVNLEKYSKDMKVVSNASCTTNCLAPVAKVLHENFEIVEGLMTTVHAVTATQKTVDGPSAKDWRGGRGAAQNIIPSSTGAAKAVGKVIPELDGKLTGMAFRVPTPNVSVVDLTVRLGKECSYDDIKAAMKTASEGPLQGVLGYTEDDVVSCDFTGDNRSSIFDAKAGIQLSKTFVKVVSWYDNEFGYSQRVIDLIKHMQKVDSA 1ii5 A 1.6 BS01 GLU A 1 N13 I54 P72 S74 R79 T125 T126 F161 D162 N13 I49 P67 S69 R74 T120 T121 F156 D157 ? 0015276,0016020 Kd=240nM remove_due_to_license_issue P73797 11518533 999 GSAMALKVGVVGNPPFVFYGAFTGISLDVWRAVAESQKWNSEYVRQNSISAGITAVAEGELDILIGPISVTPERAAIEGITFTQPYFSSGIGLLIPGTATPLFRSVGDLKNKEVAVVRDTTAVDWANFYQADVRETNNLTAAITLLQKKQVEAVMFDRPALIYYTRQNPNLNLEVTEIRVSLEPYGFVLKENSPLQKTINVEMLNLLYSRVIAEFTERWLG 1iig B 2.6 BS01 3PP B 1 K313 H395 E467 I472 G473 S513 G534 K12 H94 E166 I171 G172 S212 G233 N311 K313 H395 E397 E467 G473 S513 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 remove_due_to_license_issue P04789 2062828 600 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 1iiq A 1.83 BS01 0ZR A 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 F53 P81 D25 G27 A28 D29 D30 I47 G48 G49 I50 F53 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=33nM remove_due_to_license_issue P03367 11906284 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1iiq B 1.83 BS01 0ZR A 1 D25 G27 G49 P81 V82 I84 D25 G27 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 11906284 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ijr A 2.2 BS01 CC0 A 1 R12 R32 S34 E35 S36 C42 H58 Y59 K60 I71 G93 R12 R32 S34 E35 S36 C42 H58 Y59 K60 I71 G93 2.7.10.2 remove_due_to_license_issue P06239 11527723 150 APEPWFFKNLSRKDAERQLLAPGNTHGSFLIRESESTAGSFCLSVRDFDQNQGEVVKHYKIRNLDNGGFYISPRITFPGLHELVRHYTNASDGLCTRLSRPCQT 1ijw C 2.4 BS01 dna A 0 G139 R140 R142 A143 I171 G172 S174 T175 R178 Y179 G1 R2 R4 A5 I33 G34 S36 T37 R40 Y41 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 2 ~ 15 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASSI 1ijw C 2.4 BS02 dna B 0 G139 R140 P141 Y177 P181 A182 S183 G1 R2 P3 Y39 P43 A44 S45 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 16 ~ 29 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASSI 1ik4 A 2.0 BS01 PGH A 1 V17 H19 K23 T45 T47 T48 S65 G66 D71 H98 V17 H19 K23 T45 T47 T48 S65 G66 D71 H98 H19 G66 D71 D91 H98 D101 R107 H19 G66 D71 D91 H98 D101 R107 4.2.3.3 0005737,0005829,0008929,0016829,0019242,0034214,0042802 Ki=39nM remove_due_to_license_issue P0A731 11389594 153 MELTTRTLPARKHIALVAHDHCKQMLMSWVERHQPLLEQHVLYATGTTGNLISRATGMNVNAMLSGPMGGDQQVGALISEGKIDVLIFFWDPLNAVPHDPDVKALLRLATVWNIPVATNVATADFIIQSPHFNDAVDILIPDYQRYLADRLK 1ik4 F 2.0 BS01 PGH F 1 V17 H19 K23 T45 T47 T48 S65 G66 D71 H98 V17 H19 K23 T45 T47 T48 S65 G66 D71 H98 H19 G66 D71 D91 H98 D101 R107 H19 G66 D71 D91 H98 D101 R107 4.2.3.3 0005737,0005829,0008929,0016829,0019242,0034214,0042802 Ki=39nM remove_due_to_license_issue P0A731 11389594 153 MELTTRTLPARKHIALVAHDHCKQMLMSWVERHQPLLEQHVLYATGTTGNLISRATGMNVNAMLSGPMGGDQQVGALISEGKIDVLIFFWDPLNAVPHDPDVKALLRLATVWNIPVATNVATADFIIQSPHFNDAVDILIPDYQRYLADRL 1ikt A 1.75 BS01 OXN A 1 W36 F79 Q90 F93 S107 Q108 Q111 W31 F74 Q85 F88 S102 Q103 Q106 1.1.1.n12,4.2.1.107,4.2.1.119 remove_due_to_license_issue P51659 11700068 123 LQSTFVFEEIGRRLKDIGPEVVKKVNAVFEWHITKGGNIGAKWTIDLKSGSGKVYQGPAKGAADTTIILSDEDFMEVVLGKLDPQKAFFSGRLKARGNIMLSQKLQMILKDYAKL 1ikv A 3.0 BS01 EFZ A 1 L100 K101 V106 V179 Y181 Y188 G190 W229 L234 H235 Y318 L100 K101 V105 V178 Y180 Y187 G189 W228 L233 H234 Y317 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 11895437 2000 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTQLQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 1ikw A 3.0 BS01 EFZ A 1 L100 K101 V106 V179 Y181 Y188 F227 W229 L234 H235 Y318 L100 K101 V106 V179 Y181 Y188 F227 W229 L234 H235 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 11895437 2000 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTQLQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 1ikx A 2.8 BS01 PNU A 1 P95 K101 N103 Y181 Y188 F227 W229 L234 Y318 P95 K101 N103 Y181 Y188 F227 W229 L234 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 11895437 2000 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTQLQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 1iky A 3.0 BS01 MSD A 1 L100 K101 N103 V179 Y181 Y188 F227 W229 L234 H235 P236 Y318 L100 K101 N103 V179 Y181 Y188 F227 W229 L234 H235 P236 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 11895437 2000 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTQLQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 1il2 A 2.6 BS01 rna C 0 R26 R28 D29 L30 G31 S32 L33 F35 Q46 F48 R64 R76 N82 N84 E93 P109 D111 N113 H114 V115 N116 T117 E118 E119 E171 G172 A173 R217 E219 D220 R222 A223 R225 I343 F433 M447 E482 R549 T557 T558 R26 R28 D29 L30 G31 S32 L33 F35 Q46 F48 R64 R76 N82 N84 E93 P109 D111 N113 H114 V115 N116 T117 E118 E119 E171 G172 A173 R217 E219 D220 R222 A223 R225 I343 F433 M447 E482 R549 T557 T558 E482 G485 R537 E482 G485 R537 6.1.1.12 0000166,0003676,0004812,0004815,0005524,0005737,0005829,0006412,0006418,0006422,0016874,0140640 remove_due_to_license_issue P21889 11566892 901 ~ 976 MRTEYCGQLRLSHVGQQVTLCGWVNRRRDLGSLIFIDMRDREGIVQVFFDPDRADALKLASELRNEFCIQVTGTVRARDEKNINRDMATGEIEVLASSLTIINRADVLPLDSNHVNTEEARLKYRYLDLRRPEMAQRLKTRAKITSLVRRFMDDHGFLDIETPMLTKATPEGARDYLVPSRVHKGKFYALPQSPQLFKQLLMMSGFDRYYQIVKCFRDEDLRADRQPEFTQIDVETSFMTAPQVREVMEALVRHLWLEVKGVDLGDFPVMTFAEAERRYGSDKPDLRNPMELTDVADLLKSVEFAVFAGPANDPKGRVAALRVPGGASLTRKQIDEYGNFVKIYGAKGLAYIKVNERAKGLEGINSPVAKFLNAEIIEDILDRTAAQDGDMIFFGADNKKIVADAMGALRLKVGKDLGLTDESKWAPLWVIDFPMFEDDGEGGLTAMHHPFTSPKDMTAAELKAAPENAVANAYDMVINGYEVGGGSVRIHNGDMQQTVFGILGINEEEQREKFGFLLDALKYGTPPHAGLAFGLDRLTMLLTGTDNIRDVIAFPKTTAAACLMTEAPSFANPTALAELSIQVVK 1il2 B 2.6 BS01 rna D 0 R1026 R1028 D1029 L1030 G1031 S1032 L1033 F1035 Q1046 F1048 R1064 R1078 N1082 N1084 E1093 P1109 D1111 N1113 H1114 V1115 N1116 T1117 R26 R28 D29 L30 G31 S32 L33 F35 Q46 F48 R64 R78 N82 N84 E93 P109 D111 N113 H114 V115 N116 T117 E1482 G1485 R1537 E482 G485 R537 6.1.1.12 0000166,0003676,0004812,0004815,0005524,0005737,0005829,0006412,0006418,0006422,0016874,0140640 remove_due_to_license_issue P21889 11566892 1902 ~ 1972 MRTEYCGQLRLSHVGQQVTLCGWVNRRRDLGSLIFIDMRDREGIVQVFFDPDRADALKLASELRNEFCIQVTGTVRARDEKNINRDMATGEIEVLASSLTIINRADVLPLDSNHVNTEEARLKYRYLDLRRPEMAQRLKTRAKITSLVRRFMDDHGFLDIETPMLTKATPEGARDYLVPSRVHKGKFYALPQSPQLFKQLLMMSGFDRYYQIVKCFRDEDLRADRQPEFTQIDVETSFMTAPQVREVMEALVRHLWLEVKGVDLGDFPVMTFAEAERRYGSDKPDLRNPMELTDVADLLKSVEFAVFAGPANDPKGRVAALRVPGGASLTRKQIDEYGNFVKIYGAKGLAYIKVNERAKGLEGINSPVAKFLNAEIIEDILDRTAAQDGDMIFFGADNKKIVADAMGALRLKVGKDLGLTDESKWAPLWVIDFPMFEDDGEGGLTAMHHPFTSPKDMTAAELKAAPENAVANAYDMVINGYEVGGGSVRIHNGDMQQTVFGILGINEEEQREKFGFLLDALKYGTPPHAGLAFGLDRLTMLLTGTDNIRDVIAFPKTTAAACLMTEAPSFANPTALAELSIQVVK 1il3 A 2.8 BS01 7DG A 1 Y80 V81 G121 Y123 I172 E177 R180 Y80 V81 G121 Y123 I172 E177 R180 V81 E177 R180 V81 E177 R180 3.2.2.22 0017148,0030598 remove_due_to_license_issue P02879 11754581 301 IFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 1il4 A 2.6 BS01 9DG A 1 Y80 V81 G121 Y123 I172 E177 R180 Y80 V81 G121 Y123 I172 E177 R180 V81 E177 R180 V81 E177 R180 3.2.2.22 0017148,0030598 remove_due_to_license_issue IC50=1400000nM P02879 11754581 301 IFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 1il5 A 2.8 BS01 DDP A 1 Y80 N122 Y123 R180 Y79 N121 Y122 R179 V81 E177 R180 V80 E176 R179 3.2.2.22 0017148,0030598 remove_due_to_license_issue P02879 11754581 301 IFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPQF 1il9 A 3.1 BS01 MOG A 1 A79 Y80 V81 F93 G121 N122 Y123 I172 R180 A79 Y80 V81 F93 G121 N122 Y123 I172 R180 V81 E177 R180 V81 E177 R180 3.2.2.22 0017148,0030598 remove_due_to_license_issue IC50=400000nM P02879 11754581 301 IFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 1ilh A 2.76 BS01 SRL A 1 M243 M246 S247 F251 F281 C284 Q285 F288 W299 M82 M85 S86 F90 F120 C123 Q124 F127 W138 ? 0003677,0004879,0006355 remove_due_to_license_issue EC50=440nM O75469 11408620 1 GLTEEQRMMIRELMDAQMKTFDTTFSHFKNFRLPGVKWSQVRKDLCSLKVSLQLRGEDGSVWNYKPPADSGGKEIFSLLPHMADMSTYMFKGIISFAKVISYFRDLPIEDQISLLKGAAFELCQLRFNTVFNAETGTWECGRLSYCLEDTAGGFQQLLLEPMLKFHYMLKKLQLHEEEYVLMQAISLFSPDRPGVLQHRVVDQLQEQFAITLKSYIECNRPQPAHRFLFLKIMAMLTELRSINAQHTQRLLRIQDIHPFATPLMQELFGI 1imh C 2.86 BS01 dna A 0 R217 G224 S225 R226 G227 Q364 K392 R30 G37 S38 R39 G40 Q177 K205 ? 0000978,0003677,0003700,0006355 remove_due_to_license_issue O94916 11780147 4001 ~ 4015 KKSPMLCGQYPVKSEGKELKIVVQPETQHRARYLTEGSRGSVKDRTQQGFPTVKLEGHNEPVVLQVFVGNDSGRVKPHGFYQACRVTGRNTTPCKEVDIEGTTVIEVGLDPSNNMTLAVDCVGILKLRNADVEARIGIAGSKKKSTRARLVFRVNIMRKDGSTLTLQTPSSPILCTQPAGVPEILKKSLHSCSVKGEEEVFLIGKNFLKGTKVIFQENVSDENSWKSEAEIDMELFHQNHLIVKVPPYHDQHITLPVSVGIYVVTNAGRSHDVQPFTYTPD 1imh C 2.86 BS02 dna B 0 Y220 T222 E223 R315 N316 T333 Y33 T35 E36 R128 N129 T146 ? 0000978,0003677,0003700,0006355 remove_due_to_license_issue O94916 11780147 5001 ~ 5015 KKSPMLCGQYPVKSEGKELKIVVQPETQHRARYLTEGSRGSVKDRTQQGFPTVKLEGHNEPVVLQVFVGNDSGRVKPHGFYQACRVTGRNTTPCKEVDIEGTTVIEVGLDPSNNMTLAVDCVGILKLRNADVEARIGIAGSKKKSTRARLVFRVNIMRKDGSTLTLQTPSSPILCTQPAGVPEILKKSLHSCSVKGEEEVFLIGKNFLKGTKVIFQENVSDENSWKSEAEIDMELFHQNHLIVKVPPYHDQHITLPVSVGIYVVTNAGRSHDVQPFTYTPD 1imh D 2.86 BS01 dna A 0 Y220 T222 R315 N316 Y33 T35 R128 N129 ? 0000978,0003677,0003700,0006355 remove_due_to_license_issue O94916 11780147 4001 ~ 4015 KKSPMLCGQYPVKSEGKELKIVVQPETQHRARYLTEGSRGSVKDRTQQGFPTVKLEGHNEPVVLQVFVGNDSGRVKPHGFYQACRVTGRNTTPCKEVDIEGTTVIEVGLDPSNNMTLAVDCVGILKLRNADVEARIGIAGSKKKSTRARLVFRVNIMRKDGSTLTLQTPSSPILCTQPAGVPEILKKSLHSCSVKGEEEVFLIGKNFLKGTKVIFQENVSDENSWKSEAEIDMELFHQNHLIVKVPPYHDQHITLPVSVGIYVVTNAGRSHDVQPFTYTPD 1imx A 1.82 BS01 CPQ A 1 L5 F16 L3 F14 ? 0005179,0005576,0005615,0008083 remove_due_to_license_issue P05019 11551198 101 ETLCGAELVDALQFVCGDRGFYFNKPTGYGSSTGIVDECCFRSCDLRRLEMYCAPL 1inc A 1.94 BS02 ICL A 1 T41 H57 L151 Q192 S195 V216 T29 H45 L141 Q185 S188 V209 H57 D102 Q192 G193 D194 S195 G196 H45 D93 Q185 G186 D187 S188 G189 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 3430613 260 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 1ind H 2.2 BS01 EOT H 1 T33 L52 H99 R100 T33 L52 H99 R100 Ka=11000000000M^-1 remove_due_to_license_issue 8218161 801 EVTLVESGGDSVKPGGSLKLSCAASGFTLSGETMSWVRQTPEKRLEWVATTLSGGGFTFYSASVKGRFTISRDNAQNNLYLQLNSLRSEDTALYFCASHRFVHWGHGTLVTVSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLESDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPR 1ind L 2.2 BS01 EOT H 1 Y34 W93 W98 Y33 W92 W97 remove_due_to_license_issue 8218161 801 AVVTQESALTTSPGETVTLTCRSSTGAVTTSNYANWVQEKPDHLFTGLIGGTNNRAPGVPARFSGSLIGDKAALTITGAQTEDEARYFCALWYSNLWVFGGGTKLTVLGQPKSSPSVTLFPPSSEELETNKATLVCTIIDFYPGVVTVDWKVDGTPVTQGMETTQPSKQSNNKYMASSYLTLTAREWERHSSYSCQVTHEGHTVEKSLSRA 1inf A 2.4 BS02 ST4 A 1 R116 E117 D149 W177 R223 E275 E276 R292 R374 Y409 R40 E41 D73 W101 R147 E199 E200 R216 R298 Y333 D149 E276 R292 R374 Y409 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=10uM remove_due_to_license_issue P03474 7650674 471 EPEWTYPRLSCQGSTFQKALLISPHRFGEIKGNSAPLIIREPFVACGPKECRHFALTHYAAQPGGYYNGTRKDRNKLRHLVSVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDNDALVKIKYGEAYTDTYHSYAHNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEILPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTKTYLDTPRPDDGSIAGPCESNGDKWLGGIKGGFVHQRMASKIGRWYSRTMSKTNRMGMELYVKYDGDPWTDSDALTLSGVMVSIEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKDTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1ing A 2.4 BS02 ST5 A 1 D151 R152 A246 E276 R371 Y406 D70 R71 A165 E195 R290 Y325 D151 E277 R292 R371 Y406 D70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue P06820 7650674 471 VEYRNWSKPQCQITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPVKCYQFALGQGTTLDNKHSNDTVHDRIPHRTLLMNELGVPFHLGTRQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYDGRLVDSIGSWSQNILRTQESECVCINGTCTVVMTDGSASGRADTRILFIEEGKIVHISPLAGSAQHVEECSCYPRYPGVRCICRDNWKGSNRPVVDINMEDYSIDSSYVCSGLVGDTPRNDDRSSNSNCRDPNNERGTQGVKGWAFDNGNDLWMGRTISKDLRSGYETFKVIGGWSTPNSKSQINRQVIVDSDNRSGYSGIFSVEGKSCINRCFYVELIRGRKQETRVWWTSNSIVVFCGTSGTYGTGSWPDGANINFMPI 1inh A 2.4 BS03 ST6 A 1 R118 E119 D151 W178 E276 E277 Y406 R37 E38 D70 W97 E195 E196 Y325 D151 E277 R292 R371 Y406 D70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue P06820 7650674 471 VEYRNWSKPQCQITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPVKCYQFALGQGTTLDNKHSNDTVHDRIPHRTLLMNELGVPFHLGTRQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYDGRLVDSIGSWSQNILRTQESECVCINGTCTVVMTDGSASGRADTRILFIEEGKIVHISPLAGSAQHVEECSCYPRYPGVRCICRDNWKGSNRPVVDINMEDYSIDSSYVCSGLVGDTPRNDDRSSNSNCRDPNNERGTQGVKGWAFDNGNDLWMGRTISKDLRSGYETFKVIGGWSTPNSKSQINRQVIVDSDNRSGYSGIFSVEGKSCINRCFYVELIRGRKQETRVWWTSNSIVVFCGTSGTYGTGSWPDGANINFMPI 1io4 A 3.0 BS01 dna E 0 R280 V285 K287 S288 R12 V17 K19 S20 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11257229 1 ~ 26 KHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLF 1io4 A 3.0 BS02 dna F 0 R278 N282 R286 R289 R10 N14 R18 R21 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11257229 1 ~ 26 KHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLF 1io4 B 3.0 BS01 dna E 0 K269 Y274 R278 N281 N282 R289 K5 Y10 R14 N17 N18 R25 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11257229 1 ~ 26 KTVDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQL 1io4 B 3.0 BS02 dna F 0 R280 K287 S288 R16 K23 S24 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 11257229 1 ~ 26 KTVDKHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQL 1io4 C 3.0 BS01 dna E 0 R80 R135 R174 R177 R21 R76 R115 R118 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q03347 11257229 1 ~ 26 GELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPRRH 1io4 C 3.0 BS02 dna F 0 R139 R142 G143 K167 T169 V170 D171 R80 R83 G84 K108 T110 V111 D112 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q03347 11257229 1 ~ 26 GELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPRRH 1it6 A 2.0 BS03 CYU A 1 S129 Y134 V195 P196 D197 W206 D208 R221 V223 Q249 Y272 S123 Y128 V189 P190 D191 W200 D202 R215 V217 Q243 Y266 D64 H66 D92 D95 R96 N124 H125 H173 R221 H248 D58 H60 D86 D89 R90 N118 H119 H167 R215 H242 3.1.3.16 0000070,0000165,0000775,0000776,0000781,0001824,0003723,0004721,0004722,0005515,0005521,0005634,0005654,0005694,0005730,0005737,0005739,0005741,0005815,0005829,0005856,0005925,0005977,0006338,0006357,0006470,0007283,0008157,0016607,0016787,0016791,0017018,0019901,0019903,0019904,0030182,0030496,0032154,0032922,0032991,0033192,0042752,0043153,0043197,0044877,0046822,0046872,0048511,0051301,0060252,0072357,0098793,0098794,0098978,0140791,0180004,0180005,0180006,0180007,0180008,1990439 Ki=4.1nM remove_due_to_license_issue P36873 12015153 501 LNIDSIIQRLLEVRGSKPGKNVQLQENEIRGLCLKSREIFLSQPILLELEAPLKICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFLLRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDLQSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVLGWGENDRGVSFTFGAEVVAKFLHKHDLDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYCGEFDNAGAMMSVDETLMCSFQILKPA 1iup A 1.6 BS01 ALQ A 1 Y76 W81 M190 W198 Y74 W79 M188 W196 S34 G35 G37 N102 A103 F104 G127 V142 R174 F187 D224 H252 W253 S32 G33 G35 N100 A101 F102 G125 V140 R172 F185 D222 H250 W251 3.7.1.9 0003824,0016020,0016787 Ki=2.9mM remove_due_to_license_issue P96965 12192074 1302 NLEIGKSILAAGVLTNYHDVGEGQPVILIHGSGPGVSAYANWRLTIPALSKFYRVIAPDMVGFGFTDRPENYNYSKDSWVDHIIGIMDALEIEKAHIVGNAFGGGLAIATALRYSERVDRMVLMGAAGTRFDVTEGLNAVWGYTPSIENMRNLLDIFAYDRSLVTDELARLRYEASIQPGFQESFSSMFPEPRQRWIDALASSDEDIKTLPNETLIIHGREDQVVPLSSSLRLGELIDRAQLHVFGRCGHWTQIEQTDRFNRLVVEFFNEA 1iup A 1.6 BS02 ALQ A 2 S34 A103 F104 L139 W143 V226 H252 S32 A101 F102 L137 W141 V224 H250 S34 G35 G37 N102 A103 F104 G127 V142 R174 F187 D224 H252 W253 S32 G33 G35 N100 A101 F102 G125 V140 R172 F185 D222 H250 W251 3.7.1.9 0003824,0016020,0016787 Ki=2.9mM remove_due_to_license_issue P96965 12192074 1300 NLEIGKSILAAGVLTNYHDVGEGQPVILIHGSGPGVSAYANWRLTIPALSKFYRVIAPDMVGFGFTDRPENYNYSKDSWVDHIIGIMDALEIEKAHIVGNAFGGGLAIATALRYSERVDRMVLMGAAGTRFDVTEGLNAVWGYTPSIENMRNLLDIFAYDRSLVTDELARLRYEASIQPGFQESFSSMFPEPRQRWIDALASSDEDIKTLPNETLIIHGREDQVVPLSSSLRLGELIDRAQLHVFGRCGHWTQIEQTDRFNRLVVEFFNEA 1iup A 1.6 BS03 ALQ A 3 A42 N43 R174 W253 A40 N41 R172 W251 S34 G35 G37 N102 A103 F104 G127 V142 R174 F187 D224 H252 W253 S32 G33 G35 N100 A101 F102 G125 V140 R172 F185 D222 H250 W251 3.7.1.9 0003824,0016020,0016787 Ki=2.9mM remove_due_to_license_issue P96965 12192074 1301 NLEIGKSILAAGVLTNYHDVGEGQPVILIHGSGPGVSAYANWRLTIPALSKFYRVIAPDMVGFGFTDRPENYNYSKDSWVDHIIGIMDALEIEKAHIVGNAFGGGLAIATALRYSERVDRMVLMGAAGTRFDVTEGLNAVWGYTPSIENMRNLLDIFAYDRSLVTDELARLRYEASIQPGFQESFSSMFPEPRQRWIDALASSDEDIKTLPNETLIIHGREDQVVPLSSSLRLGELIDRAQLHVFGRCGHWTQIEQTDRFNRLVVEFFNEA 1ivp A 2.5 BS01 1ZK B 1 R8 L23 D25 G27 A28 D29 G48 P81 I82 I84 R8 L23 D25 G27 A28 D29 G48 P81 I82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 8514751 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTLEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1ivp B 2.5 BS01 1ZK B 1 D25 A28 D29 D30 V47 G48 G49 D25 A28 D29 D30 V47 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=30nM remove_due_to_license_issue P04584 8514751 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTLEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1iy7 A 2.0 BS02 CXA A 1 H69 E72 R127 N144 R145 I243 Y248 A250 T268 E270 H69 E72 R127 N144 R145 I243 Y248 A250 T268 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=0.64uM remove_due_to_license_issue P00730 12431056 500 ARSTNTFNYATYHTLDEIYDFMDLLVAQHPELVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 1iyl A 3.2 BS01 R64 A 1 Y107 D110 Y119 F176 Y225 H227 F240 F339 N392 C393 L451 Y40 D43 Y52 F109 Y158 H160 F173 F272 N325 C326 L384 N175 F176 L177 T211 L451 N108 F109 L110 T144 L384 2.3.1.97 0004379,0006499 remove_due_to_license_issue IC50=1nM P30418 12401496 452 TPEDVPNDPLPLISDFEWSTLDIDDNLQLDELYKLLYDNYVEDIDATFRFKYSHEFFQWALKPPGWRKDWHVGVRVKSTGKLVAFIAATPVTFKLNKSNKVIDSVEINFLCIHKKLRNKRLAPVLIKEITRRVNKQNIWQALYTGGSILPTPLTTCRYQHRPINWSKLHDVGFSHLPPNQTKSSMVASYTLPNNPKLKGLRPMTGKDVSTVLSLLYKYQERFDIVQLFTEEEFKHWMLGHDENSDSNVVKSYVVEDENGIITDYFSYYLLPFTVLDNAQHDELGIAYLFYYASDSFEKPNYKKRLNELITDALITSKKFGVDVFNCLTCQDNTYFLKDCKFGSGDGFLNYYLFNYRTFPMDGGIDKKTKEVVEDQTSGIGVVLL 1izh A 1.9 BS01 Q50 B 1 R8 D25 G27 A28 P81 V82 I84 R8 D25 G27 A28 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q90EB9 12460574 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1izh B 1.9 BS01 Q50 B 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 F53 D25 G27 A28 D29 D30 I47 G48 G49 I50 F53 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=0.02uM remove_due_to_license_issue Q90EB9 12460574 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1izi A 2.15 BS01 Q50 B 1 R8 D25 G27 A28 T82 R8 D25 G27 A28 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 12460574 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKVIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1izi B 2.15 BS01 Q50 B 1 D25 G27 A28 D29 D30 I47 G48 G49 T82 D25 G27 A28 D29 D30 I47 G48 G49 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.26nM remove_due_to_license_issue P03367 12460574 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKVIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1j01 A 2.0 BS01 XIL A 1 E43 N44 K47 H80 W84 Q87 Q203 E233 W273 W281 E43 N44 K47 H80 W84 Q87 Q203 E233 W273 W281 E127 N169 H205 E233 D235 E127 N169 H205 E233 D235 3.2.1.8,3.2.1.91 0004553,0005975 Ki=0.34uM remove_due_to_license_issue P07986 601 ATTLKEAADGAGRDFGFALDPNRLSEAQYKAIADSEFNLVVAENAMKWDATEPSQNSFSFGAGDRVASYAADTGKELYGHTLVWHSQLPDWAKNLNGSAFESAMVNHVTKVADHFEGKVASWDVVNEAFADGGGRRQDSAFQQKLGNGYIETAFRAARAADPTAKLCINDYNVEGINAKSNSLYDLVKDFKARGVPLDCVGFQSHLIVGQVPGDFRQNLQRFADLGVDVRITELDIRMRTPSDATKLATQAADYKKVVQACMQVTRCQGVTVWGITDKYSWVPDVFPGEGAALVWDASYAKKPAYAAVMEAF 1j07 A 2.35 BS02 DCU A 1 Y72 W286 H287 L289 Q291 S293 Y72 W280 H281 L283 Q285 S287 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Ki=0.021uM remove_due_to_license_issue P21836 12505979 951 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 1j14 A 2.4 BS02 BEN A 1 D189 S190 C191 Q192 S195 V213 W215 G216 D171 S172 C173 Q174 S177 V191 W193 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=32.2uM remove_due_to_license_issue P00763 12527302 1 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRETYNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASYPGKITDNMVCVGFLEGGKDSCQGDSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN 1j15 A 2.0 BS02 BEN A 1 D189 A190 C191 Q192 V213 W215 G216 G219 D171 A172 C173 Q174 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=143uM remove_due_to_license_issue P00763 12527302 1 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRETYNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASSSFIITDNMVCVGFLEGGKDACQGDSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN 1j16 A 1.6 BS02 BEN A 1 D189 A190 C191 Q192 V213 W215 G216 G219 D171 A172 C173 Q174 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=143uM remove_due_to_license_issue P00763 12527302 1 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRETYNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASSSFIITDNMVCVGFLEGGKDACQGDSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN 1j16 A 1.6 BS03 BEN A 2 R62 I63 Q64 N84 R45 I46 Q47 N66 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=143uM remove_due_to_license_issue P00763 12527302 4 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRETYNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASSSFIITDNMVCVGFLEGGKDACQGDSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN 1j17 T 2.0 BS02 ZEN T 1 E97 T98 Y99 F174 A190 C191 Q192 V213 W215 G216 G219 C220 G226 V227 Y228 E79 T80 Y81 F154 A172 C173 Q174 V191 W193 G194 G196 C197 G204 V205 Y206 G193 S195 G196 G175 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=6.05uM remove_due_to_license_issue P00763 12527302 1 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRETYNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASSSFIITDNMVCVGFLEGGKDACQGDSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN 1j1a A 2.2 BS03 BHP A 1 L2 F5 H6 A17 G29 G31 C44 H47 D48 Y51 L2 F5 H6 A17 G29 G31 C44 H47 D48 Y51 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 ic50=0.029uM remove_due_to_license_issue P14555 12616631 1301 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 1j1a B 2.2 BS03 BHP B 1 F5 G29 G31 C44 H47 D48 Y51 K62 F5 G29 G31 C44 H47 D48 Y51 K62 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 ic50=0.029uM remove_due_to_license_issue P14555 12616631 2301 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 1j36 A 2.4 BS02 LPR A 1 Q265 H337 A338 E368 E395 K495 H497 Y504 Y507 Q243 H315 A316 E346 E373 K473 H475 Y482 Y485 H337 A338 H367 E368 H371 E395 H497 Y507 H315 A316 H345 E346 H349 E373 H475 Y485 3.4.15.1 0006508,0008237,0008241,0016020 Ki=18nM remove_due_to_license_issue Q10714 12633854 801 IQAKEYLENLNKELAKRTNVETEAAWAYRSAITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQAYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLIDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSARAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWITSNKCVSSHHHHH 1j37 A 2.4 BS02 X8Z A 1 Q265 H337 H367 E368 H371 E395 H497 Y504 Y507 Q243 H315 H345 E346 H349 E373 H475 Y482 Y485 H337 A338 H367 E368 H371 E395 H497 Y507 H315 A316 H345 E346 H349 E373 H475 Y485 3.4.15.1 0006508,0008237,0008241,0016020 Ki=1.1nM remove_due_to_license_issue Q10714 12633854 801 IQAKEYLENLNKELAKRTNVETEAAWAYRSAITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQAYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLIDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSARAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWITSNKCVSSHHHHH 1j4r A 1.8 BS01 001 A 1 Y26 F36 D37 R42 F46 Q53 V55 I56 W59 Y82 H87 I90 Y26 F36 D37 R42 F46 Q53 V55 I56 W59 Y82 H87 I90 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 Ki=0.019uM remove_due_to_license_issue P62942 11735566 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1j5a K 3.5 BS01 rna A 0 T54 G63 N66 H69 F77 P86 P96 R159 L170 G174 T53 G62 N65 H68 F76 P85 P95 R158 L169 G173 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q9RXK1 11677599 1 ~ 2877 AQINVIGQNGGRTIELPLPEVNSGVLHEVVTWQLASRRRGTASTRTRAQVSKTGRKMYGQKGTGNARHGDRSVPTFVGGGVAFGPKPRSYDYTLPRQVRQLGLAMAIASRQEGGKLVAVDGFDIADAKTKNFISWAKQNGLDGTEKVLLVTDDENTRRAARNVSWVSVLPVAGVNVYDILRHDRLVIDAAALEIVEE 1j5a L 3.5 BS01 rna A 0 K15 R62 S74 P108 G112 A114 K11 R58 S70 P104 G108 A110 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue Q9RXJ7 11677599 1 ~ 2877 EQTFRNKKQRKQQVKLRKPGFAVAKYVRMSPRKVRLVVDVIRGKSVQDAEDLLRFIPRSASEPVAKVLNSAKANALHNDEMLEDRLFVKEAYVDAGPTLKRLIPRARGSANIIKKRTSHITIIVAEKGNK 1j5a M 3.5 BS01 rna A 0 H4 P7 K10 H43 H3 P6 K9 H42 ? 0003735,0005840,0006412,0015934,0019843,0046872,1990904 remove_due_to_license_issue P49228 11677599 1 ~ 2877 AKHPVPKKKTSKSKRDMRRSHHALTAPNLTECPQCHGKKLSHHICPNCGYYDGRQVLA 1j5i A -1.00 BS01 NCZ A 1 C37 L45 C47 D51 G96 S98 G102 N103 E106 C37 L45 C47 D51 G96 S98 G102 N103 E106 ? 0003677,0006952,0042742 remove_due_to_license_issue P0A3R9 12269815 130 AAPTATVTPSSGLSDGTVVKVAGAGLQAGTAYDVGQCAWVDTGVLACNPADFSSVTADANGSASTSLTVRRSFEGFLFDGTRWGTVDCTTAACQVGLSDAAGNGPEGVAISFN 1j5k A -1.00 BS01 dna B 0 A25 G26 S27 I29 G30 K31 G32 G33 R40 I47 K48 I49 R59 A16 G17 S18 I20 G21 K22 G23 G24 R31 I38 K39 I40 R50 ? 0003676,0003723 remove_due_to_license_issue P61978 12093748 105 ~ 109 GGPIITTQVTIPKDLAGSIIGKGGQRIKQIRHESGASIKIDEPLEGSEDRIITITGTQDQIQNAQYLLQNSVKQYS 1j5n A -1.00 BS01 dna B 0 R13 K14 K16 K22 R23 L25 Y28 M29 R36 R40 T47 F48 R13 K14 K16 K22 R23 L25 Y28 M29 R36 R40 T47 F48 ? 0001195,0003676,0003677,0005515,0005634,0005694,0006281,0006325,0006338,0008301,0031491,0032407,0032993,0051123,0065004,0070898 remove_due_to_license_issue P11632 12381320 101 ~ 115 MVTPREPKKRTTRKKKDPNAPKRALSAYMFFANENRDIVRSENPDITFGQVGKKLGEKWKALTPEEKQPYEAKAQADKKRYESEKELYNATLA 1j5n A -1.00 BS02 dna C 0 T11 T12 R23 S26 Y28 F48 K53 W59 K60 K78 Y81 K85 T11 T12 R23 S26 Y28 F48 K53 W59 K60 K78 Y81 K85 ? 0001195,0003676,0003677,0005515,0005634,0005694,0006281,0006325,0006338,0008301,0031491,0032407,0032993,0051123,0065004,0070898 remove_due_to_license_issue P11632 12381320 116 ~ 130 MVTPREPKKRTTRKKKDPNAPKRALSAYMFFANENRDIVRSENPDITFGQVGKKLGEKWKALTPEEKQPYEAKAQADKKRYESEKELYNATLA 1j75 A 1.85 BS01 dna B 0 K143 N146 Q147 Y150 P163 K31 N34 Q35 Y38 P51 ? 0003677,0003723,0003726,0060340 remove_due_to_license_issue Q9QY24 11524677 200 ~ 206 NLEQKILQVLSDDGGPVKIGQLVKKCQVPKKTLNQVLYRLKKEDRVSSPEPATWSIG 1jak A 1.75 BS02 IFG A 1 R162 D313 E314 W344 W361 Y393 D395 W408 W442 E444 R155 D306 E307 W337 W354 Y386 D388 W401 W435 E437 D313 E314 D306 E307 3.2.1.52 0004553,0004563,0005975,0016020,0016231,0016798,0030203 Ki=2.7uM remove_due_to_license_issue O85361 11522797 601 DRKAPVRPTPLDRVIPAPASVDPGGAPYRITRGTHIRVDDSREARRVGDYLADLLRPATGYRLPVTAHGHGGIRLRLAGGPYGDEGYRLDSGPAGVTITARKAAGLFHGVQTLRQLLPPAVEKDSAQPGPWLVAGGTIEDTPRYAWRSAMLDVSRHFFGVDEVKRYIDRVARYKYNKLHLHLSDDQGWRIAIDSWPRLATYGGSTEVGGGPGGYYTKAEYKEIVRYAASRHLEVVPEIDMPGHTNAALASYAELNCDGVAPPLYTGTKVGFSSLCVDKDVTYDFVDDVIGELAALTPGRYLHIGGDEAHSTPKADFVAFMKRVQPIVAKYGKTVVGWHQLAGAEPVEGALVQYWGLDRTGDAEKAEVAEAARNGTGLILSPADRTYLDMKYTKDTPLGLSWAGYVEVQRSYDWDPAGYLPGAPADAVRGVEAPLWTETLSDPDQLDYMAFPRLPGVAELGWSPASTHDWDTYKVRLAAQAPYWEAAGIDFYRSPQVPWT 1jao A 2.4 BS01 0D3 A 1 I159 L160 Y189 V194 H197 E198 H201 P217 N218 Y219 I75 L76 Y105 V110 H113 E114 H117 P133 N134 Y135 H197 E198 H201 H207 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 Ki=1.2uM remove_due_to_license_issue P22894 7737183 1 NPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1jaq A 2.4 BS02 01S A 1 I159 L160 A161 H197 E198 H201 H207 P217 N218 Y219 I75 L76 A77 H113 E114 H117 H123 P133 N134 Y135 H197 E198 H201 H207 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 Ki=33uM remove_due_to_license_issue Ki=121000nM P22894 7737183 1 NPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1jbr A 2.15 BS01 rna C 0 Y47 H49 W50 F51 T52 N53 R65 K110 K111 K113 D143 Y47 H49 W50 F51 T52 N53 R65 K110 K111 K113 D143 3.1.27.- 0003723,0004518,0004521,0004540,0005576,0017148 remove_due_to_license_issue P67876 11685244 0 ~ 17 ATWTCINQQLNPKTNKWEDKRLLYSQAKAESNSHHAPLSDGKTGSSYPHWFTNGYDGNGKLIKGRTPIKFGKADCDRPPKHSQNGMGKDDHYLLEFPTFPDGHDYKFDSKKPKEDPGPARVIYTYPNKVFCGIVAHQRGNQGDLRLCSH 1jbr B 2.15 BS01 rna D 0 G44 S46 H49 W50 F51 T52 I62 R65 E95 K110 K113 G44 S46 H49 W50 F51 T52 I62 R65 E95 K110 K113 3.1.27.- 0003723,0004518,0004521,0004540,0005576,0017148 remove_due_to_license_issue P67876 11685244 0 ~ 30 ATWTCINQQLNPKTNKWEDKRLLYSQAKAESNSHHAPLSDGKTGSSYPHWFTNGYDGNGKLIKGRTPIKFGKADCDRPPKHSQNGMGKDDHYLLEFPTFPDGHDYKFDSKKPKEDPGPARVIYTYPNKVFCGIVAHQRGNQGDLRLCSH 1jcx A 1.8 BS01 PAI A 1 K1041 K1046 N1048 R1049 S1050 Q1099 P1101 A1102 K1124 R1154 H1185 Q1188 F1220 E1222 K40 K45 N47 R48 S49 Q98 P100 A101 K123 R153 H184 Q187 F211 E213 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0046364 Ki=7uM remove_due_to_license_issue O66496 11747443 1300 EKFLVIAGPCAIESEELLLKVGEEIKRLSEKFKEVEFVFKSSFDKANRSSIHSFRGHGLEYGVKALRKVKEEFGLKITTDIHESWQAEPVAEVADIIQIPAFLCRQTDLLLAAAKTGRAVNVKKGQFLAPWDTKNVVEKLKFGGAKEIYLTERGTTFGYNNLVVDFRSLPIMKQWAKVIYDATHSVQLPGMREFIFPLIRAAVAVGCDGVFMETHPEPEKALSDASTQLPLSQLEGIIEAILEIREVASKYYETI 1jcx B 1.8 BS01 PAI B 1 K2041 K2046 N2048 R2049 S2050 Q2099 P2101 A2102 K2124 R2154 H2185 F2220 K39 K44 N46 R47 S48 Q97 P99 A100 K122 R152 H183 F210 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0046364 Ki=7uM remove_due_to_license_issue O66496 11747443 2300 KFLVIAGPCAIESEELLLKVGEEIKRLSEKFKEVEFVFKSSFDKANRSSIHSFRGHGLEYGVKALRKVKEEFGLKITTDIHESWQAEPVAEVADIIQIPAFLCRQTDLLLAAAKTGRAVNVKKGQFLAPWDTKNVVEKLKFGGAKEIYLTERGTTFGYNNLVVDFRSLPIMKQWAKVIYDATHSVQLPGMREFIFPLIRAAVAVGCDGVFMETHPEPEKALSDASTQLPLSQLEGIIEAILEIREVASKYYETI 1jd0 A 1.5 BS02 AZM A 1 Q92 H94 H119 V121 L198 T199 T200 Q87 H89 H115 V117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 remove_due_to_license_issue Ki=5.7nM, Kd=130nM, IC50=60nM O43570 11493685 1400 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFS 1jdj A 2.2 BS01 CFP A 1 W44 M46 F97 W36 M38 F89 K210 T267 K202 T259 1.1.1.8 0005829,0005975,0006072,0006116,0016491,0016616,0020015,0046168,0051287,0141152 remove_due_to_license_issue P90551 12445769 367 KDELLYLNKAVVFGSGAFGTALAMVLSKKCREVCVWHMNEEEVRLVNEKRENVLFLKGVQLASNITFTSDVEKAYNGAEIILFVIPTQFLRGFFEKSGGNLIAYAKEKQVPVLVCTKGIERSTLKFPAEIIGEFLPSPLLSVLAGPSFAIEVATGVFTCVSIASADINVARRLQRIMSTGDRSFVCWATTDTVGCEVASAVKNVLAIGSGVANGLGMGLNARAALIMRGLLEIRDLTAALGGDGSAVFGLAGLGDLQLTCSSELSRNFTVGKKLGKGLPIEEIQRAVAEGVATADPLMRLAKQLKVKMPLCHQIYEIVYKKKNPRDALADLLSCGLQDEGLPPLFK 1je8 A 2.12 BS01 dna C 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 A 2.12 BS02 dna D 0 T157 P158 R159 I182 T183 S185 T186 V189 H190 T7 P8 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 B 2.12 BS01 dna C 0 T157 P158 R159 I182 T183 S185 T186 V189 H190 T7 P8 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 B 2.12 BS02 dna D 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 E 2.12 BS01 dna G 0 P172 N173 K188 K192 S202 R203 P23 N24 K39 K43 S53 R54 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 1 ~ 20 ERDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 E 2.12 BS02 dna H 0 T157 P158 R159 I182 T183 S185 T186 V189 H190 T8 P9 R10 I33 T34 S36 T37 V40 H41 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 21 ~ 40 ERDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 F 2.12 BS01 dna G 0 T157 P158 R159 I182 T183 S185 T186 V189 H190 T7 P8 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1je8 F 2.12 BS02 dna H 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 12352954 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1jey A 2.5 BS01 dna C 0 R80 L256 K338 R47 L215 K297 3.6.4.-,4.2.99.- 0000723,0000725,0000781,0000783,0000976,0002218,0003677,0003678,0003684,0003690,0003691,0003723,0004386,0005515,0005524,0005576,0005634,0005654,0005667,0005694,0005730,0005829,0005958,0006266,0006281,0006303,0006310,0008094,0010558,0016020,0016787,0016829,0016887,0030332,0032508,0032991,0032993,0034774,0042162,0043564,0044877,0045027,0045087,0045621,0045860,0045892,0045893,0045944,0048660,0051575,0070418,0070419,0071475,0071480,0071481,0097110,0097680,1904813 remove_due_to_license_issue P12956 11493912 1 ~ 18 GRDSLIFLVDASKAMFESQSEDELTPFDMSIQCIQSVYISKIISSDRDLLAVVFYGTEKDKNSVNFKNIYVLQELDNPGAKRILELDQFKGQQGQKRFQDMMGHGSDYSLSEVLWVCANLFSDVQFKMSHKRIMLFTNEDNPHGNDSAKASRARTKAGDLRDTGIFLDLMHLKKPGGFDISLFYRDIISVHFEESSKLEDLLRKVRAKETRKRALSRLKLKLNKDIVISVGIYNLVQKALKPPPIKLYRETNEPVKTKTRTFNTSTGGLLLPSDTKRSQIYGSRQIILEKEETEELKRFDDPGLMLMGFKPLVLLKKHHYLRPSLFVYPEESLVIGSSTLFSALLIKCLEKEVAALCRYTPRRNIPPYFVALVPQEEELDDQKIQVTPPGFQLVFLPFADDKRKMPFTEKIMATPEQVGKMKAIVEKLRFTYRSDSFENPVLQQHFRNLEALALDLMEPEQAVDLTLPKVEAMNKRLGSLVDEFKELVYPPDY 1jey A 2.5 BS02 dna D 0 A255 R403 R404 A214 R362 R363 3.6.4.-,4.2.99.- 0000723,0000725,0000781,0000783,0000976,0002218,0003677,0003678,0003684,0003690,0003691,0003723,0004386,0005515,0005524,0005576,0005634,0005654,0005667,0005694,0005730,0005829,0005958,0006266,0006281,0006303,0006310,0008094,0010558,0016020,0016787,0016829,0016887,0030332,0032508,0032991,0032993,0034774,0042162,0043564,0044877,0045027,0045087,0045621,0045860,0045892,0045893,0045944,0048660,0051575,0070418,0070419,0071475,0071480,0071481,0097110,0097680,1904813 remove_due_to_license_issue P12956 11493912 4 ~ 34 GRDSLIFLVDASKAMFESQSEDELTPFDMSIQCIQSVYISKIISSDRDLLAVVFYGTEKDKNSVNFKNIYVLQELDNPGAKRILELDQFKGQQGQKRFQDMMGHGSDYSLSEVLWVCANLFSDVQFKMSHKRIMLFTNEDNPHGNDSAKASRARTKAGDLRDTGIFLDLMHLKKPGGFDISLFYRDIISVHFEESSKLEDLLRKVRAKETRKRALSRLKLKLNKDIVISVGIYNLVQKALKPPPIKLYRETNEPVKTKTRTFNTSTGGLLLPSDTKRSQIYGSRQIILEKEETEELKRFDDPGLMLMGFKPLVLLKKHHYLRPSLFVYPEESLVIGSSTLFSALLIKCLEKEVAALCRYTPRRNIPPYFVALVPQEEELDDQKIQVTPPGFQLVFLPFADDKRKMPFTEKIMATPEQVGKMKAIVEKLRFTYRSDSFENPVLQQHFRNLEALALDLMEPEQAVDLTLPKVEAMNKRLGSLVDEFKELVYPPDY 1jey B 2.5 BS01 dna C 0 T275 K338 D398 K399 R400 T260 K323 D383 K384 R385 3.6.4.- 0000723,0003677,0003678,0003684,0005634,0006303,0006310,0042162,0043564 remove_due_to_license_issue P13010 11493912 1 ~ 18 NKAAVVLCMDVGFTMSNSIPGIESPFEQAKKVITMFVQRQVFAENKDEIALVLFGTDGTDNPLSGGDQYQNITVHRHLMLPDFDLLEDIESKIQPGSQQADFLDALIVSMDVIQHETIGKKFEKRHIEIFTDLSSRFSKSQLDIIIHSLKKCDISLQFFLPFSLGGPFRLGGHGPSFPLKGITEQQKEGLEIVKMVMISLEGEDGLDEIYSFSESLRKLCVFKKIERHSIHWPCRLTIGSNLSIRIAAYKSILQERVKKTWTVVDAKTLKKEDIQKETVYCLNDDDETEVLKEDIIQGFRYGSDIVPFSKVDEEQMKYKSEGKCFSVLGFCKSSQVQRRFFMGNQVLKVFAARDDEAAAVALSSLIHALDDLDMVAIVRYAYDKRANPQVGVAFPHIKHNYECLVYVQLPFMEDLRQYMFSSLKNSKKYAPTEAQLNAVDALIDSMSLAKKDEKTDTLEDLFPTTKIPNPRFQRLFQCLLHRALHPREPLPPIQQHIWNMLNPPAEVTTKSQIPLSKIKTLFPLIEAKKK 1jey B 2.5 BS02 dna D 0 E53 L85 K126 R242 K265 Y397 R400 A401 N402 E48 L80 K121 R227 K250 Y382 R385 A386 N387 3.6.4.- 0000723,0003677,0003678,0003684,0005634,0006303,0006310,0042162,0043564 remove_due_to_license_issue P13010 11493912 4 ~ 34 NKAAVVLCMDVGFTMSNSIPGIESPFEQAKKVITMFVQRQVFAENKDEIALVLFGTDGTDNPLSGGDQYQNITVHRHLMLPDFDLLEDIESKIQPGSQQADFLDALIVSMDVIQHETIGKKFEKRHIEIFTDLSSRFSKSQLDIIIHSLKKCDISLQFFLPFSLGGPFRLGGHGPSFPLKGITEQQKEGLEIVKMVMISLEGEDGLDEIYSFSESLRKLCVFKKIERHSIHWPCRLTIGSNLSIRIAAYKSILQERVKKTWTVVDAKTLKKEDIQKETVYCLNDDDETEVLKEDIIQGFRYGSDIVPFSKVDEEQMKYKSEGKCFSVLGFCKSSQVQRRFFMGNQVLKVFAARDDEAAAVALSSLIHALDDLDMVAIVRYAYDKRANPQVGVAFPHIKHNYECLVYVQLPFMEDLRQYMFSSLKNSKKYAPTEAQLNAVDALIDSMSLAKKDEKTDTLEDLFPTTKIPNPRFQRLFQCLLHRALHPREPLPPIQQHIWNMLNPPAEVTTKSQIPLSKIKTLFPLIEAKKK 1jfh A 2.03 BS01 MA3 B 1 W59 Q63 H305 W59 Q63 H305 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 9385631 1 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAIKSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKIAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGEPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCDVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAEDPFIAIHAESKL 1jfh A 2.03 BS02 MA2 B 1 W59 V163 W59 V163 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 9385631 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAIKSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKIAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGEPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCDVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAEDPFIAIHAESKL 1jfs A 2.9 BS01 dna B 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S13 T15 T16 R25 V27 A28 T31 L53 K54 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 11781089 699 ~ 715 ATIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDFGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1jft A 2.5 BS01 dna B 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S13 T15 T16 R25 V27 A28 T31 L53 K54 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 11781089 699 ~ 715 ATIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDAGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYRR 1jg0 A 2.0 BS02 DDT A 1 I55 I79 D169 L172 G173 F176 V262 A263 I55 I79 D169 L172 G173 F176 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 ic50=5uM remove_due_to_license_issue IC50=5.0e+3nM, Ki=1.8e+3nM P0A884 11590022 304 MKQYLELMQKVLDEGTQKNDATGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGAHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVA 1jg0 B 2.0 BS02 DDT B 1 I55 I79 W83 D169 L172 G173 F176 V262 I55 I79 W83 D169 L172 G173 F176 V262 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 ic50=5uM remove_due_to_license_issue IC50=5.0e+3nM, Ki=1.8e+3nM P0A884 11590022 306 MKQYLELMQKVLDEGTQKNDATGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGAHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVA 1jgl H 2.15 BS01 EST L 1 Q35 W95 G97 Q33 W94 G96 remove_due_to_license_issue 11451948 911 QIQLVQSGPELKKPGETVRISCKASDYMTSGMQWVQQMPGKGLKWIGWLNTQSGVPEYAEDFKGRFAFSLETTAYLQINNLKNEDTATYFCATWGGNSAYWGQGTTLTVSSAKTTPPSVYPLAPGNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 1jgl L 2.15 BS01 EST L 1 Y36 Y49 H89 F91 W96 Y36 Y49 H89 F91 W96 ? Kd=2nM remove_due_to_license_issue Q7TS98 11451948 911 DIQMTQSPASLSASVGETVTITCRASGNIHNYLAWYQQKQGKSPQLLVYNAKTLADGVPSRFSGSGSGTQYSLKINSLQPEDFGTYYCHHFWSTPWTFGGGTKLEVKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1jh1 A 2.7 BS05 JST A 1 H162 A163 H197 E198 H201 H78 A79 H113 E114 H117 H197 E198 H201 H207 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P22894 11563922 1000 NPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1jh9 A 2.55 BS01 dna B 0 V13 S14 T16 T17 R26 A29 T32 L54 K55 V12 S13 T15 T16 R25 A28 T31 L53 K54 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 11781089 699 ~ 715 ATIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDRGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1jif A 1.6 BS01 BLM B 1 F33 F38 H49 S51 F33 F38 H49 S51 ? 0046677 remove_due_to_license_issue Q53793 11706014 401 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif A 1.6 BS02 BLM B 2 D60 W65 Y86 P101 R109 G113 C115 D60 W65 Y86 P101 R109 G113 C115 ? 0046677 remove_due_to_license_issue Q53793 11706014 402 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif B 1.6 BS01 BLM B 1 D260 W265 Y286 A302 R309 G313 C315 D60 W65 Y86 A102 R109 G113 C115 ? 0046677 remove_due_to_license_issue Q53793 11706014 401 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif B 1.6 BS02 BLM B 2 F233 F238 S251 F33 F38 S51 ? 0046677 remove_due_to_license_issue Q53793 11706014 402 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jii A 3.2 BS01 383 A 1 Y36 G38 A39 D40 H50 L70 D80 Y170 Q174 D177 D195 Q196 Y35 G37 A38 D39 H49 L69 D79 Y169 Q173 D176 D194 Q195 T42 H47 H50 K84 R88 Q174 D195 K231 K234 S235 T41 H46 H49 K83 R87 Q173 D194 K230 K233 S234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0043039 remove_due_to_license_issue A6QHR2 11567092 421 TNVLIEDLKWRGLIYQQTDEQGIEDLLNKEQVTLYCGADPTADSLHIGHLLPFLTLRRFQEHGHRPIVLIGGGTGMIGDPSGKSEERVLQTEEQVDKNIEGISKQMHNIFEFGTDHGAVLVNNRDWLGQISLISFLRDYGKHVGVNYMLGKDSIQSRLEHGISYTEFTYTILQAIDFGHLNRELNCKIQVGGSDQWGNITSGIELMRRMYGQTDAYGLTIPLVTKSDGKKFGKSESGAVWLDAEKTSPYEFYQFWINQSDEDVIKFLKYFTFLGKEEIDRLEQSKNEAPHLREAQKTLAEEVTKFIHGEDALNDAIRIS 1jij A 3.2 BS01 629 A 1 G38 A39 H50 L70 D80 Y170 Q174 D177 G193 D195 Q196 G37 A38 H49 L69 D79 Y169 Q173 D176 G192 D194 Q195 T42 H47 H50 K84 R88 Q174 D195 K231 K234 S235 T41 H46 H49 K83 R87 Q173 D194 K230 K233 S234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0043039 remove_due_to_license_issue A6QHR2 11567092 421 TNVLIEDLKWRGLIYQQTDEQGIEDLLNKEQVTLYCGADPTADSLHIGHLLPFLTLRRFQEHGHRPIVLIGGGTGMIGDPSGKSEERVLQTEEQVDKNIEGISKQMHNIFEFGTDHGAVLVNNRDWLGQISLISFLRDYGKHVGVNYMLGKDSIQSRLEHGISYTEFTYTILQAIDFGHLNRELNCKIQVGGSDQWGNITSGIELMRRMYGQTDAYGLTIPLVTKSDGKKFGKSESGAVWLDAEKTSPYEFYQFWINQSDEDVIKFLKYFTFLGKEEIDRLEQSKNEAPHLREAQKTLAEEVTKFIHGEDALNDAIRIS 1jik A 2.8 BS01 545 A 1 G38 A39 D40 H50 P53 L70 D80 I103 Y170 Q174 D177 G193 D195 Q196 G37 A38 D39 H49 P52 L69 D79 I102 Y169 Q173 D176 G192 D194 Q195 T42 H47 H50 K84 R88 Q174 D195 K231 K234 S235 T41 H46 H49 K83 R87 Q173 D194 K230 K233 S234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0043039 remove_due_to_license_issue A6QHR2 11567092 421 TNVLIEDLKWRGLIYQQTDEQGIEDLLNKEQVTLYCGADPTADSLHIGHLLPFLTLRRFQEHGHRPIVLIGGGTGMIGDPSGKSEERVLQTEEQVDKNIEGISKQMHNIFEFGTDHGAVLVNNRDWLGQISLISFLRDYGKHVGVNYMLGKDSIQSRLEHGISYTEFTYTILQAIDFGHLNRELNCKIQVGGSDQWGNITSGIELMRRMYGQTDAYGLTIPLVTKSDGKKFGKSESGAVWLDAEKTSPYEFYQFWINQSDEDVIKFLKYFTFLGKEEIDRLEQSKNEAPHLREAQKTLAEEVTKFIHGEDALNDAIRIS 1jil A 2.2 BS01 485 A 1 Y36 G38 A39 D40 H50 L70 D80 Y170 Q174 D177 G192 G193 D195 Q196 Y35 G37 A38 D39 H49 L69 D79 Y169 Q173 D176 G191 G192 D194 Q195 T42 H47 H50 K84 R88 Q174 D195 K231 K234 S235 T41 H46 H49 K83 R87 Q173 D194 K230 K233 S234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0043039 ic50=4nM remove_due_to_license_issue A6QHR2 11567092 421 TNVLIEDLKWRGLIYQQTDEQGIEDLLNKEQVTLYCGADPTADSLHIGHLLPFLTLRRFQEHGHRPIVLIGGGTGMIGDPSGKSEERVLQTEEQVDKNIEGISKQMHNIFEFGTDHGAVLVNNRDWLGQISLISFLRDYGKHVGVNYMLGKDSIQSRLEHGISYTEFTYTILQAIDFGHLNRELNCKIQVGGSDQWGNITSGIELMRRMYGQTDAYGLTIPLVTKSDGKKFGKSESGAVWLDAEKTSPYEFYQFWINQSDEDVIKFLKYFTFLGKEEIDRLEQSKNEAPHLREAQKTLAEEVTKFIHGEDALNDAIRISQALF 1jiz A 2.6 BS06 CGS A 1 I81 L82 A83 T116 H119 E120 H123 H129 P139 Y141 I82 L83 A84 T117 H120 E121 H124 H130 P140 Y142 H119 E120 H123 H129 H120 E121 H124 H130 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 11575929 998 GFREMPGGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1jj4 A 2.4 BS01 dna C 0 R296 K300 R303 Y304 R307 S318 T319 R11 K15 R18 Y19 R22 S33 T34 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue P06790 10906136 602 ~ 617 MTPIIHLKGDRNSLKCLRYRLRKHSDHYRDISSTWHWTKTGILTVTYHSETQRTKFLNTVAIPDSVQILVGYMT 1jj4 A 2.4 BS02 dna D 0 N297 S298 C301 R305 S355 N12 S13 C16 R20 S65 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue P06790 10906136 902 ~ 917 MTPIIHLKGDRNSLKCLRYRLRKHSDHYRDISSTWHWTKTGILTVTYHSETQRTKFLNTVAIPDSVQILVGYMT 1jj4 B 2.4 BS01 dna C 0 N297 S298 C301 R305 S355 N13 S14 C17 R21 S67 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue P06790 10906136 602 ~ 617 HMTPIIHLKGDRNSLKCLRYRLRKHSDHYRDISSTWHWTEKTGILTVTYHSETQRTKFLNTVAIPDSVQILVGYMT 1jj4 B 2.4 BS02 dna D 0 R296 K300 R303 Y304 S318 T319 R12 K16 R19 Y20 S34 T35 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue P06790 10906136 902 ~ 917 HMTPIIHLKGDRNSLKCLRYRLRKHSDHYRDISSTWHWTEKTGILTVTYHSETQRTKFLNTVAIPDSVQILVGYMT 1jj9 A 2.0 BS05 BBT A 1 L160 A161 H197 E198 H201 H207 P217 N218 L76 A77 H113 E114 H117 H123 P133 N134 H197 E198 H201 H207 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=1700nM remove_due_to_license_issue IC50=1700nM P22894 11278347 1000 NPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1jje A 1.8 BS04 BYS A 1 V25 W28 H79 D81 H139 C158 K161 G166 N167 H197 V23 W26 H77 D79 H137 C156 K159 G164 N165 H195 H77 H79 D81 H139 C158 K161 N167 H197 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.0037uM remove_due_to_license_issue Q79MP6 11390410 250 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESKK 1jjk A 3.0 BS01 BMP A 1 A20 D22 K44 K73 L130 T131 P189 R192 Q201 G221 R222 A9 D11 K33 K62 L119 T120 P178 R181 Q190 G210 R211 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 remove_due_to_license_issue P08244 11526316 301 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1jjk A 3.0 BS02 BMP B 1 D76 I77 T80 D65 I66 T69 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 remove_due_to_license_issue P08244 11526316 302 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1jjk B 3.0 BS01 BMP A 1 D76 I77 T80 D65 I66 T69 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 remove_due_to_license_issue P08244 11526316 301 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1jjk B 3.0 BS02 BMP B 1 A20 D22 K44 K73 L130 T131 P189 R192 Q201 G221 R222 A9 D11 K33 K62 L119 T120 P178 R181 Q190 G210 R211 K44 D71 K73 D76 T131 R222 K33 D60 K62 D65 T120 R211 4.1.1.23 0004590,0005515,0005737,0005829,0006207,0006221,0015949,0016831,0044205 remove_due_to_license_issue P08244 11526316 302 VTNSPVVVALDYHNRDDALAFVDKIDPRDCRLKVGKEMFTLFGPQFVRELQQRGFDIFLDLKFHDIPNTAAHAVAAAADLGVWMVNVHASGGARMMTAAREALVPFGKDAPLLIAVTVLTSMEASDLVDLGMTLSPADYAERLAALTQKCGLDGVVCSAQEAVRFKQVFGQEFKLVTPGIRPQGSEAGDQRRIMTPEQALSAGVDYMVIGRPVTQSVDPAQTLKAINASLQ 1jjt A 1.8 BS04 BDS A 1 V25 W28 F51 H79 S80 D81 H139 C158 K161 G166 N167 H197 V23 W26 F49 H77 S78 D79 H137 C156 K159 G164 N165 H195 H77 H79 D81 H139 C158 K161 N167 H197 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.009uM remove_due_to_license_issue Q79MP6 11390410 250 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESKK 1jk1 A 1.9 BS01 dna B 0 R114 F116 R118 E121 R124 H125 I128 R142 S145 R146 H149 H153 T156 R174 E177 R180 R12 F14 R16 E19 R22 H23 I26 R40 S43 R44 H47 H51 T54 R72 E75 R78 ? remove_due_to_license_issue P08046 11800559 1 ~ 11 RPYACPVESCDRRFSRSAELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLR 1jk1 A 1.9 BS02 dna C 0 D148 S175 D176 K179 D46 S73 D74 K77 ? remove_due_to_license_issue P08046 11800559 51 ~ 61 RPYACPVESCDRRFSRSAELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLR 1jk2 A 1.65 BS01 dna B 0 R103 F116 R118 E121 R124 H125 I128 R142 S145 R146 H149 H153 T156 R170 R174 E177 R180 R1 F14 R16 E19 R22 H23 I26 R40 S43 R44 H47 H51 T54 R68 R72 E75 R78 ? remove_due_to_license_issue P08046 11800559 1 ~ 11 RPYACPVESCDRRFSRSAELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLR 1jk2 A 1.65 BS02 dna C 0 D148 S175 K179 D46 S73 K77 ? remove_due_to_license_issue P08046 11800559 51 ~ 61 RPYACPVESCDRRFSRSAELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLR 1jk7 A 1.9 BS03 OKA A 1 R96 H125 I130 Y134 D220 R221 Y272 C273 F276 R91 H120 I125 Y129 D215 R216 Y267 C268 F271 D64 H66 D92 D95 R96 N124 H125 H173 R221 H248 D59 H61 D87 D90 R91 N119 H120 H168 R216 H243 3.1.3.16 0000070,0000165,0000775,0000776,0000781,0001824,0003723,0004721,0004722,0005515,0005521,0005634,0005654,0005694,0005730,0005737,0005739,0005741,0005815,0005829,0005856,0005925,0005977,0006338,0006357,0006470,0007283,0008157,0016607,0016787,0016791,0017018,0019901,0019903,0019904,0030182,0030496,0032154,0032922,0032991,0033192,0042752,0043153,0043197,0044877,0046822,0046872,0048511,0051301,0060252,0072357,0098793,0098794,0098978,0140791,0180004,0180005,0180006,0180007,0180008,1990439 remove_due_to_license_issue IC50=>5000nM P36873 11535607 501 KLNIDSIIQRLLEVRGSKPGKNVQLQENEIRGLCLKSREIFLSQPILLELEAPLKICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFLLRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDLQSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVLGWGENDRGVSFTFGAEVVAKFLHKHDLDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYCGEFDNAGAMMSVDETLMCSFQILKPA 1jko C 2.24 BS01 dna A 0 G139 R140 R142 S174 T175 R178 Y179 G1 R2 R4 S36 T37 R40 Y41 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 2 ~ 15 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASS 1jko C 2.24 BS02 dna B 0 G139 R140 P141 Y177 A182 G1 R2 P3 Y39 A44 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 16 ~ 29 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASS 1jkp C 2.8 BS01 dna A 0 G139 R140 R142 A143 S174 T175 R178 Y179 G1 R2 R4 A5 S36 T37 R40 Y41 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 2 ~ 15 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASSI 1jkp C 2.8 BS02 dna B 0 R140 P141 Y177 P181 A182 S183 R2 P3 Y39 P43 A44 S45 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 16 ~ 29 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASSI 1jkq C 2.86 BS01 dna A 0 R140 R142 A143 G172 S174 T175 R178 Y179 R1 R3 A4 G33 S35 T36 R39 Y40 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 2 ~ 15 RPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASSI 1jkq C 2.86 BS02 dna B 0 R140 Y177 P181 A182 S183 R1 Y38 P42 A43 S44 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 16 ~ 29 RPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASSI 1jkr C 2.28 BS01 dna A 0 G139 R140 R142 A143 S174 T175 R178 Y179 G1 R2 R4 A5 S36 T37 R40 Y41 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 2 ~ 15 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASS 1jkr C 2.28 BS02 dna B 0 G139 R140 P141 Y177 A182 G1 R2 P3 Y39 A44 ? 0000150,0003677,0006310 remove_due_to_license_issue P03013 11847127 16 ~ 29 GRPRAINKHEQEQISRLLEKGHPRQQLAIIFGIGVSTLYRYFPASS 1jld A 2.5 BS01 0PP A 1 D25 G27 D29 D30 G48 I82 D25 G27 D29 D30 G48 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 ic50=185nM remove_due_to_license_issue P04584 9216835 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1jld B 2.5 BS01 0PP A 1 D25 G27 D29 G48 F53 I84 D25 G27 D29 G48 F53 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 9216835 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1jlq A 3.0 BS01 SBN A 1 L100 K101 K103 V106 Y181 Y188 G190 W229 H235 Y318 L94 K95 K97 V100 Y175 Y182 G184 W223 H229 Y312 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 11384233 999 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHK 1jlx A 2.2 BS01 GAL C 1 N74 H75 N74 H75 ? remove_due_to_license_issue Q71QF2 9334739 2 AGLPVIMCLKSNNHQKYLRYQSDNIQQYGLLQFSADKILDPLAQFEVEPSKTYDGLVHIKSRYTNKYLVRWSPNHYWITASANEPDENKSNWACTLFKPLYVEEGNMKKVRLLHVQLGHYTQNYTVGGSFVSYLFAESSQIDTGSKDVFHVIDWKSIFQFPKGYVTFKGNNGKYLGVITINQLPCLQFGYDNLNDPKVAHQMFVTSNGTICIKSNYMNKFWRLSTDDWILVDGNDPRETNEAAALFRSDVHDFNVISLLNMQKTWFIKRFTSGKPGFINCMNAATQNVDETAILEIIEL 1jlx B 2.2 BS01 GAL D 1 N74 H75 N74 H75 ? remove_due_to_license_issue Q71QF2 9334739 2 AGLPVIMCLKSNNHQKYLRYQSDNIQQYGLLQFSADKILDPLAQFEVEPSKTYDGLVHIKSRYTNKYLVRWSPNHYWITASANEPDENKSNWACTLFKPLYVEEGNMKKVRLLHVQLGHYTQNYTVGGSFVSYLFAESSQIDTGSKDVFHVIDWKSIFQFPKGYVTFKGNNGKYLGVITINQLPCLQFGYDNLNDPKVAHQMFVTSNGTICIKSNYMNKFWRLSTDDWILVDGNDPRETNEAAALFRSDVHDFNVISLLNMQKTWFIKRFTSGKPGFINCMNAATQNVDETAILEIIEL 1jmf A 2.5 BS01 UMP A 1 R23 L195 C198 H199 Q217 R218 S219 A220 D221 G225 H259 R23 L195 C198 H199 Q217 R218 S219 A220 D221 G225 H259 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=1.7uM remove_due_to_license_issue P00469 9514716 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFAIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1jmg A 2.2 BS01 UMP A 1 R23 C198 H199 Q217 R218 S219 A220 D221 G225 H259 R23 C198 H199 Q217 R218 S219 A220 D221 G225 H259 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=0.85uM remove_due_to_license_issue P00469 9514716 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFGIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1jmi A 2.5 BS01 UMP A 1 R23 L195 C198 R218 S219 A220 D221 G225 H259 Y261 R23 L195 C198 R218 S219 A220 D221 G225 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=0.87uM remove_due_to_license_issue P00469 9514716 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFSIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1jn2 P 1.9 BS03 SFP P 1 D16 G227 R228 D16 G227 R228 ? 0030246 Ka=12200M^-1 remove_due_to_license_issue P02866 11504727 1001 ADTIVAVELDTYPNTDIGDPSYPHIGIDIKSVRSKKTAKWNMQNGKVGTAHIIYNSVDKRLSAVVSYPNADSATVSYDVDLDNVLPEWVRVGLSASTGLYKETNTILSWSFTSKLKSNSTHETNALHFMFNQFSKDQKDLILQGDATTGTDGNLELTRVSSNGSPQGSSVGRALFYAPVHIWESSAVVASFEATFTFLIKSPDSHPADGIAFFISNIDSSIPSGSTGRLLGLFPDAN 1jn4 A 1.8 BS01 139 A 1 Q11 H12 K41 V43 N44 T45 C65 N67 Q69 N71 A109 E111 V118 H119 F120 Q11 H12 K41 V43 N44 T45 C65 N67 Q69 N71 A109 E111 V118 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=11.3uM remove_due_to_license_issue P61823 11513604 901 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1joc A 2.2 BS03 ITP A 1 D1352 R1370 R1371 H1372 H1373 R1375 D64 R82 R83 H84 H85 R87 ? 0046872 Kd=24uM remove_due_to_license_issue Q15075 11741531 101 QDERRALLERCLKGEGEIEKLQTKVLELQRKLDNTTAAVQELGRENQSLQIKHTQALNRKWAEDNEVQNCMACGKGFSVTVRRHHCRQCGNIFCAECSAKNALTPSSKKPVRVCDACFNDLQG 1joc B 2.2 BS03 ITP B 1 D1352 R1370 R1371 H1372 H1373 R1375 D64 R82 R83 H84 H85 R87 ? 0046872 Kd=24uM remove_due_to_license_issue Q15075 11741531 102 QDERRALLERCLKGEGEIEKLQTKVLELQRKLDNTTAAVQELGRENQSLQIKHTQALNRKWAEDNEVQNCMACGKGFSVTVRRHHCRQCGNIFCAECSAKNALTPSSKKPVRVCDACFNDLQG 1jq3 A 1.8 BS01 AAT A 1 L62 M67 Y76 H77 G98 D101 E121 V122 N152 G153 D170 S171 T172 Q178 L182 Y239 L61 M66 Y75 H76 G97 D100 E120 V121 N151 G152 D169 S170 T171 Q177 L181 Y238 2.5.1.16 0003824,0004766,0005737,0005829,0006596,0008295,0010487,0016740,0043918,0043919,0050314 ic50=0.2uM remove_due_to_license_issue Q9WZC2 11731804 800 RTLKELERELQPRQHLWYFEYYTGNNVGLFMKMNRVIYSGQSDIQRIDIFENPDLGVVFALDGITMTTEKDEFMYHEMLAHVPMFLHPNPKKVLIIGGGDGGTLREVLKHDSVEKAILCEVDGLVIEAARKYLKQTSCGFDDPRAEIVIANGAEYVRKFKNEFDVIIIDSTDPTAGQGGHLFTEEFYQACYDALKEDGVFSAETEDPFYDIGWFKLAYRRISKVFPITRVYLGFMTTYPSGMWSYTFASKGIDPIKDFDPEKVRKFNKELKYYNEEVHVASFALPNFVKKELGLM 1jqd A 2.28 BS01 SAH A 1 G60 E89 P90 Q94 T119 S120 I142 Q143 M144 Y147 G54 E83 P84 Q88 T113 S114 I136 Q137 M138 Y141 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 Ki=6.9uM remove_due_to_license_issue Ki=18100nM P50135 11566133 400 MRSLFHGKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKTSNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 1jqe A 1.91 BS02 QUN A 1 Y15 V16 Y146 Y147 W179 W183 D193 L195 C196 F243 Y3 V4 Y134 Y135 W167 W171 D181 L183 C184 F231 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 remove_due_to_license_issue P50135 11566133 500 GKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKISNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 1jqy D 2.14 BS01 A32 D 1 Y12 E51 Q56 H57 Q61 W88 N90 K91 Y12 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 Ki=12uM remove_due_to_license_issue P32890 11880036 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1jqy D 2.14 BS02 A32 H 1 G33 K34 G33 K34 ? 0005576,0031640,0035821,0090729 Ki=12uM remove_due_to_license_issue P32890 11880036 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1jqy E 2.14 BS01 A32 D 1 G33 K34 G33 K34 ? 0005576,0031640,0035821,0090729 Ki=12uM remove_due_to_license_issue P32890 11880036 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1jqy E 2.14 BS02 A32 E 1 E11 Y12 R13 E51 Q56 H57 Q61 W88 N90 K91 E11 Y12 R13 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 Ki=12uM remove_due_to_license_issue P32890 11880036 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1jr1 A 2.6 BS02 MOA A 1 D274 S275 S276 N303 G326 C331 T333 M414 G415 Q441 D212 S213 S214 N241 G264 C269 T271 M352 G353 Q363 1.1.1.205 0000166,0003824,0003938,0005634,0005737,0005829,0006164,0006177,0006183,0007623,0016491,0046651,0046872,0071353,0097294 remove_due_to_license_issue P12269 8681386 1332 GLTAQQLFNCGDGLTYNDFLILPGYIDFTADQVDLTSALTKKITLKTPLVSSPMDTVTEAGMAIAMALTGGIGFIHHNCTPEFQANEVRKVKKYEQGFITDPVVDRVRFEAKMGSRLVIMTKREDLVVAPAGITLKEANEILQRSKLPIVNENDELVAIIARTDLKKNRDYPLASKDAKKQLLCGAAIGTHEDDKYRLDLLALAGVDVVVLDSSQGNSIFQINMIKYMKEKYPNLQVIGGNVVTAAQAKNLIDAGVDALRVGMGCGSICITQEVLACGRPQATAVYKVSEYARRFGVPVIADGGIQNVGHIAKALALGASTVMMGSLLAATTEAPGEYFFSDGIRLKKYRGMGSLDAMIKVAQGVSGAVQDKGSIHKFVPYLIAGIQHSCQDIGAKSLTQVRAMMYSGELKFEKRTSSAQVEGGVHSLHSYEKRLF 1jsv A 1.96 BS01 U55 A 1 A31 K33 F82 L83 H84 Q85 D86 K89 L134 A31 K33 F71 L72 H73 Q74 D75 K78 L123 D127 K129 Q131 N132 D145 T158 T165 D116 K118 Q120 N121 D134 T147 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=1900nM P24941 11604388 400 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1jt0 A 2.9 BS01 dna E 0 L3 S34 S35 G37 N38 Y41 H42 L2 S33 S34 G36 N37 Y40 H41 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLSKH 1jt0 A 2.9 BS02 dna F 0 T24 T25 K36 Y40 T45 K46 T23 T24 K35 Y39 T44 K45 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLSKH 1jt0 B 2.9 BS01 dna E 0 T24 T25 K36 Y40 T45 K46 T23 T24 K35 Y39 T44 K45 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLSKH 1jt0 B 2.9 BS02 dna F 0 L3 S34 S35 G37 N38 Y41 H42 L2 S33 S34 G36 N37 Y40 H41 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLSKH 1jt0 C 2.9 BS01 dna E 0 T24 T25 K36 Y40 T45 K46 T23 T24 K35 Y39 T44 K45 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLSKH 1jt0 C 2.9 BS02 dna F 0 S34 S35 K36 G37 N38 Y41 H42 S33 S34 K35 G36 N37 Y40 H41 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLSKH 1jt0 D 2.9 BS01 dna E 0 N2 L3 S34 S35 G37 N38 Y41 H42 N1 L2 S33 S34 G36 N37 Y40 H41 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGL 1jt0 D 2.9 BS02 dna F 0 T24 T25 K36 Y40 T45 K46 T23 T24 K35 Y39 T44 K45 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 11867549 7 ~ 34 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGL 1jt1 A 1.78 BS03 MCO A 1 S221 G223 M266 Y293 K297 D300 S173 G175 M217 Y244 K248 D251 H116 H118 D120 H121 H196 Y228 H263 H70 H72 D74 H75 H148 Y180 H214 3.5.2.6 Ki=400uM remove_due_to_license_issue Q9K578 12507470 700 YPMPNPFPPFRIAGNLYYVGTDDLASYLIVTPRGNILINSDLEANVPMIKASIKKLGFKFSDTKILLISHAHFDHAAGSELIKQQTKAKYMVMDEDVSVILSGGKSDFHYANDSSTYFTQSTVDKVLHDGERVELGGTVLTAHLTPGHTRGCTTWTMKLKDHGKQYQAVIIGSIGVNPGYKLVDNITYPKIAEDYKHSIKVLESMRCDIFLGSHAGMFDLKNKYVLLSKGQNNPFVDPTGCKNYIEQKANDFYTELKKQETG 1jtq A 2.5 BS02 LY3 A 1 H51 I79 W83 D169 G173 A263 H51 I79 W83 D169 G173 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 11697906 501 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1jtq B 2.5 BS03 LY3 B 1 H51 I79 W80 W83 D169 G173 V262 A263 H51 I79 W80 W83 D169 G173 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 11697906 502 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1juj A 3.0 BS02 LYA A 1 K77 F80 I108 W109 G222 F225 A312 K50 F53 I81 W82 G195 F198 A285 E87 W109 Y135 C195 R215 D218 E60 W82 Y108 C168 R188 D191 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue IC50=9500nM, Ki=1.3nM P04818 11697906 315 HGELQYLGQIQHILRCGVEKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 1juj B 3.0 BS03 LYA B 1 K77 F80 I108 W109 G222 F225 A312 K50 F53 I81 W82 G195 F198 A285 E87 W109 Y135 C195 R215 D218 E60 W82 Y108 C168 R188 D191 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue IC50=9500nM, Ki=1.3nM P04818 11697906 315 HGELQYLGQIQHILRCGVEKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 1jut A 2.7 BS02 LYD A 1 W80 W83 D169 L172 G173 F176 W80 W83 D169 L172 G173 F176 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 11697906 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1jut B 2.7 BS03 LYD B 1 W80 G173 F176 V262 W80 G173 F176 V262 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 11697906 305 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1juy A 2.5 BS03 H5P A 1 N38 G127 T128 T129 Q224 L228 V238 T239 V273 N38 G127 T128 T129 Q224 L228 V238 T239 V273 D13 K16 G40 H41 Q224 D13 K16 G40 H41 Q224 6.3.4.4 0000166,0000287,0004019,0005515,0005525,0005737,0005829,0006164,0006974,0015949,0016020,0016874,0044208,0046040,0046086,0046872,0097216 remove_due_to_license_issue P0A7D4 8961938 433 GNNVVVLGTQWGDEGKGKIVDLLTERAKYVVRYQGGHNAGHTLVINGEKTVLHLIPSGILRENVTSIIGNGVVLSPAALMKEMKELEDRGIPVRERLLLSEACPLILDYHVALDNAREKARGAKAIGTTGRGIGPAYEDKVARRGLRVGDLFDKETFAEKLKEVMEYHNFQLVNYYKAEAVDYQKVLDDTMAVADILTSMVVDVSDLLDQARQRGDFVMFEGAQGTLLDIDHGTYPYVTSSNTTAGGVATGSGLGPRYVDYVLGILKAYSTRVGAGPFPTELFDETGEFLCKQGNEFGATTGRRRRTGWLDTVAVRRAVQLNSLSGFCLTKLDVLDGLKEVKLCVAYRMPDGREVTTTPLAADDWKGVEPIYETMPGWSESTFGVKDRSGLPQAALNYIKRIEELTGVPIDIISTGPDRTETMILRDPFDA 1jvu A 1.78 BS01 C2P A 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue Ki=7000nM P61823 11746706 130 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1jwt A 2.5 BS01 BLI A 1 H79 N131 I209 D229 C231 W257 G258 G260 G268 H79 N131 I209 D229 C231 W257 G258 G260 G268 H79 D135 E232 G233 D234 S235 G236 H79 D135 E232 G233 D234 S235 G236 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=14nM remove_due_to_license_issue P00734 11720865 300 TFGSGEADCGLRPLFEKKSLEDKTERELLESYIDGRIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGEDFEEIPEEYL 1jys A 1.9 BS01 ADE A 1 F151 I152 E172 M173 F151 I152 E172 M173 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=300uM remove_due_to_license_issue P0AF12 11591349 233 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQSFDEFLAVAAKQSSLMVESLVQKLA 1jys B 1.9 BS01 ADE B 1 F151 I152 E172 F151 I152 E172 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=300uM remove_due_to_license_issue P0AF12 11591349 234 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQSFDEFLAVAAKQSSLMVESLVQKLA 1jzs A 2.5 BS03 MRC A 1 P46 G56 E550 G551 D553 Q554 P46 G56 E550 G551 D553 Q554 P46 H54 H57 D85 W518 Q554 W558 K591 K594 P46 H54 H57 D85 W518 Q554 W558 K591 K594 6.1.1.5 0000049,0000166,0002161,0004812,0004822,0005524,0006418,0006428 Ki=0.25uM remove_due_to_license_issue P56690 11584022 1301 MFKEVGEPNFPKLEEEVLAFWKREKIFQKSVENRKGGPRYTVYEGPPTANGLPHVGHAQARSYKDLFPRYKTMRGYYAPRRAGWDTHGLPVELEVEKKLGLKSKREIEAYGIERFNQACRESVFTYEKEWEAFTERIAYWVDLEDAYATLEPTYIESIWWSLKNLFDRGLLYRDHKVVPYCPRCGTPLSSHEVALGYKEIQDPSVYVRFPLKEPKKLGLEKASLLIWTTTPWTLPGNVAAAVHPEYTYAAFQVGDEALILEEGLGRKLLGEGTQVLKTFPGKALEGLPYTPPYPQALEKGYFVVLADYVSQEDGTGIVHQAPAFGAEDLETARVYGLPLLKTVDEEGKLLVEPFKGLYFREANRAILRDLRGRGLLFKEESYLHSYPHCWRCSTPLMYYATESWFIKNTLFKDELIRNNQEIHWVPPHIKEGRYGEWLKNLVDWALSRNRYWGTPLPIWVCQACGKEEAIGSFQELKARATKPLPEPFDPHRPYVDQVELACACGGTMRRVPYVIDVWYDSGAMPFASLHYPFEHEEVFRESFPADFIAEGIDQTRGWFNSLHQLGVMLFGSIAFKNVICHGLILDEKGQKMSKSKGNVVDPWDIIRKFGADALRWYIYVSAPPEADRRFGPNLVRETVRDYFLTLWNVYSFFVTYANLDRPDLKNPPPPEKRPEMDRWLLARMQDLIQRVTEALEAYDPTTSARALRDFVVEDLSQWYVRRNRRRFWKNEDALDREAAYATLYEALVLVATLAAPFTPFLAEVLWQNLVRSVRLEAKESVHLADWPEADPALADEALVAQMRAVLKVVDLARAARAKSGV 1k03 A 2.7 BS02 HBA A 1 W116 H191 N194 Y196 F250 F296 Y375 W116 H191 N194 Y196 F250 F296 Y375 T37 H191 N194 Y196 R243 N251 T37 H191 N194 Y196 R243 N251 1.6.99.1 0003959,0010181,0016491 remove_due_to_license_issue Q02899 11668181 450 SFVKDFKPQALGDTNLFKPIKIGNNELLHRAVIPPLTRMRALHPGNIPNRDWAVEYYTQRAQRPGTMIITEGAFISPQAGGYDNAPGVWSEEQMVEWTKIFNAIHEKKSFVWVNLWVLGWAAFPDNLARDGLRYDSASDNVFMDAEQEAKAKKANNPQHSLTKDEIKQYIKEYVQAAKNSIAAGADGVEIHSANGYLLNQFLDPHSNTRTDEYGGSIENRARFTLEVVDALVEAIGHEKVGLRLSPYGVFNSMSGGAETGIVAQYAYVAGELEKRAKAGKRLAFVHLVEPRVTNPFLTEGEGEYEGGSNDFVYSIWKGPVIRAGNFALHPEVVREEVKDKRTLIGYGRFFISNPDLVDRLEKGLPLNKYDRDTFYQMSAHGYIDYPTYEEALKLGWDKK 1k06 A 1.8 BS01 BZD A 1 E88 G135 L136 N282 D283 H377 N484 E672 S674 G675 E76 G123 L124 N261 D262 H347 N454 E642 S644 G645 H377 K568 R569 K574 T676 K680 H347 K538 R539 K544 T646 K650 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.6uM remove_due_to_license_issue Ki=4600nM P00489 11895439 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1k06 A 1.8 BS02 BZD A 2 R60 W67 W189 E190 K191 P229 R48 W55 W177 E178 K179 P217 H377 K568 R569 K574 T676 K680 H347 K538 R539 K544 T646 K650 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.6uM remove_due_to_license_issue Ki=4600nM P00489 11895439 920 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1k08 A 2.26 BS01 BZD A 1 E88 G135 L136 N282 D283 H341 H377 N484 E672 S674 G675 E76 G123 L124 N270 D271 H321 H357 N464 E652 S654 G655 H377 K568 R569 K574 T676 K680 H357 K548 R549 K554 T656 K660 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.6uM remove_due_to_license_issue Ki=4600nM P00489 11895439 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1k08 A 2.26 BS02 BZD A 2 R60 W67 W189 E190 K191 P229 R48 W55 W177 E178 K179 P217 H377 K568 R569 K574 T676 K680 H357 K548 R549 K554 T656 K660 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.6uM remove_due_to_license_issue Ki=4600nM P00489 11895439 920 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1k1g A -1.00 BS01 rna B 0 N151 V153 G154 L155 I157 G158 R160 L164 M176 I177 R178 G179 S182 V183 K184 R190 M195 L196 K241 L244 L247 T253 L254 R255 N18 V20 G21 L22 I24 G25 R27 L31 M43 I44 R45 G46 S49 V50 K51 R57 M62 L63 K108 L111 L114 T120 L121 R122 ? 0003676,0003723 remove_due_to_license_issue Q15637 11691992 501 ~ 511 TRVSDKVMIPQDEYPEINFVGLLIGPRGNTLKNIEKECNAKIMIRGKGSVKEGKVGRKDGQMLPGEDEPLHALVTANTMENVKKAVEQIRNILKQGIETPEDQNDLRKMQLRELARLNGTLR 1k1i A 2.2 BS02 FD1 A 1 H57 D189 S190 S195 V213 W215 G216 G219 H40 D171 S172 S177 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=264nM remove_due_to_license_issue Ki=99999999999999nM P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k1j A 2.2 BS02 FD2 A 1 H57 L99 D189 S190 S195 W215 G216 S217 G219 H40 L81 D171 S172 S177 W193 G194 S195 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=28nM remove_due_to_license_issue Ki=36nM P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k1l A 2.5 BS02 FD3 A 1 L99 D189 S190 C191 Q192 W215 G216 S217 G219 L81 D171 S172 C173 Q174 W193 G194 S195 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=125nM remove_due_to_license_issue Ki=220nM P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k1m A 2.2 BS02 FD4 A 1 H57 L99 D189 S190 C191 Q192 W215 G216 G219 H40 L81 D171 S172 C173 Q174 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=40nM remove_due_to_license_issue Ki=99999999999999nM P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k1n A 2.0 BS02 CCR A 1 H57 D189 S190 C191 Q192 S214 W215 G216 G219 H40 D171 S172 C173 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=153nM remove_due_to_license_issue P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k1o A 2.0 BS02 IGN A 1 H57 N97 T98 D189 S190 C191 S195 S214 W215 G216 G219 H40 N79 T80 D171 S172 C173 S177 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue Ki=675nM P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k1p A 1.9 BS02 MEL A 1 L99 D189 S190 C191 S214 W215 G216 G219 L81 D171 S172 C173 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue IC50=11nM P00760 11676542 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1k21 H 1.86 BS05 IGN H 1 H57 Y60A W60D D189 A190 C191 S195 S214 W215 G216 E217 G219 H43 Y47 W50 D192 A193 C194 S198 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=4.2nM remove_due_to_license_issue Ki=15nM, IC50=1300nM P00734 11676542 999 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 1k22 H 1.93 BS05 MEL H 1 H57 Y60A W60D L99 I174 D189 A190 S195 W215 G216 E217 G219 C220 H43 Y47 W50 L96 I172 D192 A193 S198 W220 G221 E222 G223 C224 3.4.21.5 0004252,0005509,0006508,0007596 Ki=4nM remove_due_to_license_issue IC50=69nM, Ki=1.2nM P00734 11676542 999 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1k27 A 1.95 BS02 MTM A 1 A94 C95 G96 F177 N195 M196 D220 V236 A86 C87 G88 F169 N187 M188 D212 V225 T18 P41 H65 I67 M68 A94 M196 T197 D220 D222 V233 T10 P33 H57 I59 M60 A86 M188 T189 D212 D214 V222 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Ki=1nM remove_due_to_license_issue Q13126 14705926 401 AVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGRQHTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLP 1k2i 1 1.8 BS01 SN1 1 1 S190 C191 M192 S195 W215 G216 S217 S181 C182 M183 S186 W206 G207 S208 D102 D97 3.4.21.1 0004252,0005515,0005576,0006508,0007586,0008236,0097180,0097655 remove_due_to_license_issue P00766 11846564 400 CGVPAIQPVLIVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGVTTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKYNSLTINNDITLLKLSTAASFSQTVSAVCLPSASDDFAAGTTCVTTGWGLTRYTPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 1k2v N 1.97 BS01 DEF N 1 W43 W68 R84 Y106 L189 W217 W273 F274 Y275 W12 W37 R53 Y75 L158 W186 W242 F243 Y244 ? 0005515,0006826,0015687,0030288,0042597,0055052,0098711,1901678 Kd=36uM remove_due_to_license_issue P07822 11805094 1 AIDPNRIVALEWLPVELLLALGIVPYGVADTINYRLWVSEPPLPDSVIDVGLRTEPNLELLTEMKPSFMVWSAGYGPSPEMLARIAPGRGFNFSDGKQPLAMARKSLTEMADLLNLQSAAETHLAQYEDFIRSMKPRFVKRGARPLLLTTLIDPRHMLVFGPNSLFQEILDEYGIPNAWQGETNFWGSTAVSIDRLAAYKDVDVLCFDHDNSKDMDALMATPLWQAMPFVRAGRFQRVPAVWFYGATLSAMHFVRVLDNAIG 1k3t C 1.95 BS01 BRZ C 1 C166 H194 N335 C166 H194 N335 C166 H194 C166 H194 1.2.1.12 0004365,0005829,0006006,0006096,0016491,0016620,0020015,0050661,0051287 ic50=64uM remove_due_to_license_issue P22513 12044862 960 MPIKVGINGFGRIGRMVFQALCEDGLLGTEIDVVAVVDMNTDAEYFAYQMRYDTVHGKFKYEVTTTKSSPSVAKDDTLVVNGHRILCVKAQRNPADLPWGKLGVEYVIESTGLFTAKAAAEGHLRGGARKVVISAPASGGAKTLVMGVNHHEYNPSEHHVVSNASCTTNCLAPIVHVLVKEGFGVQTGLMTTIHSYTATQKTVDGVSVKDWRGGRAAAVNIIPSTTGAAKAVGMVIPSTQGKLTGMSFRVPTPDVSVVDLTFTAARDTSIQEIDAALKRASKTYMKGILGYTDEELVSADFINDNRSSIYDSKATLQNNLPKERRFFKIVSWYDNEWGYSHRVVDLVRHMASKDRSARL 1k4g A 1.7 BS02 AIQ A 1 Y106 C158 G229 M260 G261 D280 Y96 C148 G219 M250 G251 D270 D102 D280 C318 C320 C323 H349 D92 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=1.4uM remove_due_to_license_issue P28720 11921407 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1k4h A 1.8 BS02 APQ A 1 N70 D102 Y106 C158 G229 L231 M260 G261 D280 N60 D92 Y96 C148 G219 L221 M250 G251 D270 D102 D280 C318 C320 C323 H349 D92 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=7.7uM remove_due_to_license_issue P28720 11921407 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1k6c A 2.2 BS01 MK1 B 1 R8 D25 G27 G48 R8 D25 G27 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 11790852 902 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6c B 2.2 BS01 MK1 B 1 D25 G27 A28 D29 D30 G48 P81 D25 G27 A28 D29 D30 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=33nM remove_due_to_license_issue P35963 11790852 902 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6p A 2.2 BS01 XN3 B 1 R8 D25 G27 G48 P81 T82 R8 D25 G27 G48 P81 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 11790852 807 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6p B 2.2 BS01 XN3 B 1 D25 G27 A28 D29 D30 G48 P81 D25 G27 A28 D29 D30 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=44nM remove_due_to_license_issue P35963 11790852 807 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6t A 2.25 BS01 XN1 B 1 R8 D25 G48 G49 R8 D25 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 11790852 509 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6t B 2.25 BS01 XN1 B 1 D25 G27 A28 D29 D30 V32 I47 G48 P81 D25 G27 A28 D29 D30 V32 I47 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=24nM remove_due_to_license_issue P35963 11790852 509 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6v A 2.0 BS01 XN2 B 1 R8 D25 G27 G48 F53 R8 D25 G27 G48 F53 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 11790852 252 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6v B 2.0 BS01 XN2 B 1 D25 G27 A28 D29 D30 G48 P81 D25 G27 A28 D29 D30 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=120nM remove_due_to_license_issue P35963 11790852 252 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k9s A 2.0 BS02 FM2 A 1 M64 S90 C91 G92 F159 V178 E179 M180 E181 S203 M64 S90 C91 G92 F159 V178 E179 M180 E181 S203 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0006974,0009116,0009164,0016020,0016757,0016763,0019686,0042278,0042802,0047975 remove_due_to_license_issue P0ABP8 11786017 9901 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHIRTHEQTTAAERQTTFNDMIKIALESVLLGDK 1k9s D 2.0 BS01 FM2 A 1 H4 R43 H4 R43 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0006974,0009116,0009164,0016020,0016757,0016763,0019686,0042278,0042802,0047975 remove_due_to_license_issue P0ABP8 11786017 9901 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHIRTHEQTTAAERQTTFNDMIKIALESVLLGDK 1kak A 2.5 BS01 FNP A 1 Y46 V49 D181 F182 A217 Q262 Y45 V48 D180 F181 A216 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=26uM remove_due_to_license_issue P18031 11741477 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1kav A 2.35 BS01 FEP A 1 Y46 R47 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 R46 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=1.5uM remove_due_to_license_issue P18031 11741477 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1kc7 A 2.2 BS02 PPR A 1 R561 R617 E745 G766 T767 N768 D769 R560 R616 E744 G765 T766 N767 D768 K22 R92 G101 M103 R337 H455 E745 S764 D769 C831 Y851 K21 R91 G100 M102 R336 H454 E744 S763 D768 C830 Y850 2.7.9.1 0003824,0005524,0006090,0016301,0016310,0016772,0046872,0050242 Ki=3uM remove_due_to_license_issue P22983 11790099 1000 AKWVYKFEEGNASMRNLLGGKGCNLAEMTILGMPIPQGFTVTTEACTEYYNSGKQITQEIQDQIFEAITWLEELNGKKFGDTEDPLLVSVRSGARASMPGMMDTILNLGLNDVAVEGFAKKTGNPRFAYDSYRRFIQMYSDVVMEVPKSHFEKIIDAMKEEKGVHFDTDLTADDLKELAEKFKAVYKEAMNGEEFPQEPKDQLMGAVKAVFRSWDNPRAIVYRRMNDIPGDWGTAVNVQTMVFGNKGETSGTGVAFTRNPSTGEKGIYGEYLINAQGEDVVAGVRTPQPITQLENDMPDCYKQFMDLAMKLEKHFRDMQDMEFTIEEGKLYFLQTRNGKRTAPAALQIACDLVDEGMITEEEAVVRIEAKSLDQLLHPTFNPAALKAGEVIGSALPASPGAAAGKVYFTADEAKAAHEKGERVILVRLETSPEDIEGMHAAEGILTVRGGMTSHAAVVARGMGTCCVSGCGEIKINEEAKTFELGGHTFAEGDYISLDGSTGKIYKGDIETQEASVSGSFERIMVWADKFRTLKVRTNADTPEDTLNAVKLGAEGIGLCRTEHMFFEADRIMKIRKMILSDSVEAREEALNELIPFQKGDFKAMYKALEGRPMTVRYLDPPLHEFVPHTEEEQAELAKNMGLTLAEVKAKVDELHEFNPMMGHRGCRLAVTYPEIAKMQTRAVMEAAIEVKEETGIDIVPEIMIPLVGEKKELKFVKDVVVEVAEQVKKEKGSDMQYHIGTMIEIPRAALTADAIAEEAEFFSFGTNDLTQMTFGFSRDDAGKFLDSYYKAKIYESDPFARLDQTGVGQLVEMAVKKGRQTRPGLKCGICGEHGGDPSSVEFCHKVGLNYVSCSPFRVPIARLAAAQAALNN 1kdk A 1.7 BS01 DHT A 1 S41 S42 D65 F67 N82 L171 S30 S31 D54 F56 N71 L160 ? Kd=0.9nM remove_due_to_license_issue IC50=3.8nM, Kd=0.182000nM P04278 12054810 301 DPPAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGPLTSKRHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAEISASAPTSLRSC 1kds A 2.15 BS01 NPB A 1 S64 Y150 N152 Y221 G317 A318 S61 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=1700nM, IC50=5000nM P00811 12109906 364 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1kdw A 2.28 BS01 4CB A 1 S64 Q120 Y150 N152 Y221 A318 S61 Q117 Y147 N149 Y218 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=2900nM P00811 12109906 364 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1ke0 A 2.3 BS01 CVB A 1 S64 Q120 Y150 N152 Y221 G317 A318 S61 Q117 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=4200nM P00811 12109906 364 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1ke3 A 2.15 BS01 BDB A 1 S64 Q120 Y150 N152 Y221 G317 A318 S61 Q117 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=200nM P00811 12109906 364 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1ke5 A 2.2 BS01 LS1 A 1 I10 A31 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F73 E74 F75 L76 H77 Q78 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T148 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=560nM remove_due_to_license_issue IC50=560nM P24941 11728181 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1ke6 A 2.0 BS01 LS2 A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 I10 A31 F73 F75 L76 H77 Q78 D79 K82 L127 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T147 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=5.7nM remove_due_to_license_issue IC50=5.7nM P24941 11728181 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1ke7 A 2.0 BS01 LS3 A 1 I10 A31 K33 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 K33 F73 E74 F75 L76 H77 Q78 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T148 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=8.9nM remove_due_to_license_issue IC50=8.9nM P24941 11728181 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1ke8 A 2.0 BS01 LS4 A 1 E8 I10 A31 F80 E81 F82 L83 H84 D86 K89 L134 D145 E8 I10 A31 F73 E74 F75 L76 H77 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1000nM remove_due_to_license_issue IC50=1000nM P24941 11728181 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1ke9 A 2.0 BS01 LS5 A 1 I10 A31 F80 E81 F82 L83 H84 Q85 D86 K89 L134 I10 A31 F73 E74 F75 L76 H77 Q78 D79 K82 L127 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T148 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=660nM remove_due_to_license_issue Kd=210nM, koff=4.97E-02s-1, kon=175033.3M-1-s-1, IC50=660nM P24941 11728181 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1kel H 1.9 BS01 AAH H 1 Y33 N35 F50 R52 K56 W101 Y33 N35 F50 R52 K56 W101 ? Kd=52nM remove_due_to_license_issue P01868 8643580 219 EVKLVESGGGLGQPGGSLRLSCATSGFTFTDYYFNWARQPPGKALEWLGFIRNKAKGYTTEYSASVKGRFTISRDNSQGILYLQMNTLRAEDSATYYCARWGSYAMDYWGQGTSVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVP 1kel L 1.9 BS01 AAH H 1 Y37 F94 G96 Y37 F94 G96 remove_due_to_license_issue 8643580 219 DVLMTQTPLSLPVSLGDQASISCRFSQSIVHSNGNTYLEWYLQKSGQSPKLLIYKVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFQGSHVPRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRN 1kf0 A 2.5 BS01 ACP A 1 G213 A214 G237 G238 G340 V341 E343 G213 A214 G237 G238 G340 V341 E343 R38 K215 G373 G396 R38 K215 G373 G396 2.7.2.3 0004618,0005524,0005737,0005759,0005829,0006094,0006096,0016301,0043531 Kd=2.8mM remove_due_to_license_issue Q7SIB7 12102622 418 SLSNKLTLDKLNVKGKRVVMRVDFNVPMKNNQITNNQRIKAAVPSIKFCLDDGAKSVVLMSHLGRPDGSPMPDKYSLQPVAVELKSLLGKDVLFLKDCVGPEVEKACADPAAGSVILLENLRFHVEEEGKGKDASGNKVKAEPAKIKTFRASLSKLGDVYVNDAFGTAHRAHSSMVGVNLPKKAGGFLMKKELNYFAKALESPERPFLAILGGAKVADKIQLINNMLDKVNEMIIGGGMAFTFLKVLNNMEIGTSLFDEEGAKIVKNLMSKAEKNGVKITLPVDFVTADKFDEHAKTGQATVASGIPAGWMGLDCGPESSKKYSEAVARAKQIVWNGPVGVFEWEAFAQGTKALMDEVVKATSRGCITIIGGGDTATCCAKWNTEDKVSHVSTGGGASLELLEGKVLPGVDALSNV 1kf6 B 2.7 BS04 HQO C 1 T205 F206 Q225 K228 T205 F206 Q225 K228 1.3.5.1 0005515,0005829,0005886,0006099,0006113,0008177,0009055,0009061,0016020,0016491,0019645,0044780,0045283,0046872,0051536,0051537,0051538,0051539 remove_due_to_license_issue P0AC47 11850430 700 AEMKNLKIEVVRYNPEVDTAPHSAFYEVPYDATTSLLDALGYIKDNLAPDLSYRWSCRMAICGSCGMMVNNVPKLACKTFLRDYTDGMKVEALANFPIERDLVVDMTHFIESLEAIKPYIIGNSRTADQGTNIQTPAQMAKYHQFSGCINCGLCYAACPQFGLNPEFIGPAAITLAHRYNEDSRDHGKKERMAQLNSQNGVWSCTFVGYCSEVCPKHVDPAAAIQQGKVESSKDFLIATLKPR 1kf6 C 2.7 BS01 HQO C 1 R28 E29 R28 E29 ? 0000104,0005886,0006113,0009061,0016020,0019645,0044780,0045283 remove_due_to_license_issue P0A8Q0 11850430 700 TTKRKPYVRPMTSTWWKKLPFYRFYMLREGTAVPAVWFSIELIFGLFALKNGPEAWAGFVDFLQNPVIVIINLITLAAALLHTKTWFELAPKAANIIVKDEKMGPEPIIKSLWAVTVVATIVILFVALYW 1kf6 D 2.7 BS01 HQO C 1 W14 F17 W15 F18 ? 0000104,0005886,0006106,0006113,0009061,0016020,0019645,0044780,0045283 remove_due_to_license_issue P0A8Q3 11850430 700 MINPNPKRSDEPVFWGLFGAGGMWSAIIAPVMILLVGILLPLGLFPGDALSYERVLAFAQSFIGRVFLFLMIVLPLWCGLHRMHHAMHDLKIHVPAGKWVFYGLAAILTVVTLIGVVTI 1kfv A 2.55 BS01 dna D 0 E2 K57 H72 R74 M75 R109 K129 G170 N171 Y238 K254 K256 R260 E2 K57 H72 R74 M75 R109 K129 G170 N171 Y231 K247 K249 R253 G1 G1 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 12065399 1 ~ 13 GELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSISTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1kfv A 2.55 BS02 dna E 0 H91 V108 R109 F111 H91 V108 R109 F111 G1 G1 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 12065399 14 ~ 26 GELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSISTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1kfv B 2.55 BS01 dna G 0 G1 E2 K57 H72 R74 M75 R109 K129 G170 N171 Y238 K254 K256 R260 G1 E2 K57 H72 R74 M75 R109 K129 G170 N171 Y227 K243 K245 R249 G1 G1 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 12065399 1 ~ 13 GELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1kfv B 2.55 BS02 dna H 0 H91 V108 R109 K110 F111 H91 V108 R109 K110 F111 G1 G1 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 12065399 14 ~ 26 GELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1kfy B 3.6 BS04 BRS B 1 T205 F206 Q225 K228 T205 F206 Q225 K228 1.3.5.1 0005515,0005829,0005886,0006099,0006113,0008177,0009055,0009061,0016020,0016491,0019645,0044780,0045283,0046872,0051536,0051537,0051538,0051539 remove_due_to_license_issue P0AC47 11850430 700 AEMKNLKIEVVRYNPEVDTAPHSAFYEVPYDATTSLLDALGYIKDNLAPDLSYRWSCRMAICGSCGMMVNNVPKLACKTFLRDYTDGMKVEALANFPIERDLVVDMTHFIESLEAIKPYIIGNSRTADQGTNIQTPAQMAKYHQFSGCINCGLCYAACPQFGLNPEFIGPAAITLAHRYNEDSRDHGKKERMAQLNSQNGVWSCTFVGYCSEVCPKHVDPAAAIQQGKVESSKDFLIATLKPR 1kfy C 3.6 BS01 BRS B 1 R28 W86 L89 R28 W86 L89 ? 0000104,0005886,0006113,0009061,0016020,0019645,0044780,0045283 remove_due_to_license_issue P0A8Q0 11850430 700 TTKRKPYVRPMTSTWWKKLPFYRFYMLREGTAVPAVWFSIELIFGLFALKNGPEAWAGFVDFLQNPVIVIINLITLAAALLHTKTWFELAPKAANIIVKDEKMGPEPIIKSLWAVTVVATIVILFVALYW 1kfy D 3.6 BS01 BRS B 1 W14 G18 W15 G19 ? 0000104,0005886,0006106,0006113,0009061,0016020,0019645,0044780,0045283 remove_due_to_license_issue P0A8Q3 11850430 700 MINPNPKRSDEPVFWGLFGAGGMWSAIIAPVMILLVGILLPLGLFPGDALSYERVLAFAQSFIGRVFLFLMIVLPLWCGLHRMHHAMHDLKIHVPAGKWVFYGLAAILTVVTLIGVVTI 1kjr A 1.55 BS01 GAL B 1 H158 R162 W181 E184 H46 R50 W69 E72 ? 0030246 remove_due_to_license_issue P17931 15701008 2 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 1kjr A 1.55 BS02 BEK A 1 R144 H158 N160 R32 H46 N48 ? 0030246 remove_due_to_license_issue P17931 15701008 500 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 1kkq A 3.0 BS02 471 A 1 L254 I272 F273 C275 C276 Y314 V332 I354 H440 L55 I73 F74 C76 C77 Y115 V133 I155 H241 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Q07869 11845213 775 TADLKSLAKRIYEAYLKNFNMNKVKARVILSGKASNNPPFVIHDMETLCMAEKTLVAKLVANGIQNKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANLDLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFDFAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDIFLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDMY 1kll A 1.5 BS01 MC A 1 L7 H38 D52 Y60 L5 H36 D50 Y58 ? remove_due_to_license_issue O05205 12121648 9138 ARISLFAVVVEDMAKSMEFYRKMGVEIPAEADSAPHTEAVLDGGIRLAWDTVETVRSYDPEWQAPTGGHRFAIAFEFPDTASVDKKYAELVDAGYEGHLKPWNAVWGQRYAIVKDPDGNVVDLFAPLP 1km3 A 1.5 BS01 UP6 A 1 D20 K72 M126 S127 P180 Q185 G202 R203 D10 K62 M116 S117 P170 Q175 G192 R193 A42 D70 K72 D75 A32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=12400nM O26232 11900543 2001 VMNRLILAMDLMNRDDALRVTGEVREYIDTVAIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESI 1kmv A 1.05 BS01 LII A 1 I7 V8 E30 F31 F34 P61 V115 I7 V8 E30 F31 F34 P61 V115 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 remove_due_to_license_issue P00374 12096917 201 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFQRMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKN 1kmy A 2.0 BS02 BPY A 1 H146 F187 H195 H210 H241 N243 Y250 E260 H145 F186 H194 H209 H240 N242 Y249 E259 1.13.11.39 0003824,0005506,0008198,0009056,0018583,0042178,0046872,0051213 Kd=8uM remove_due_to_license_issue P47228 9857017 300 SIRSLGYMGFAVSDVAAWRSFLTQKLGLMEAGTTDNGDLFRIDSRAWRIAVQQGEVDDLAFAGYEVADAAGLAQMADKLKQAGIAVTTGDASLARRRGVTGLITFADPFGLPLEIYYGASEVFEKPFLPGAAVSGFLTGEQGLGHFVRCVPDSDKALAFYTDVLGFQLSDVIDMKMGPDVTVPAYFLHCNERHHTLAIAAFPLPKRIHHFMLEVASLDDVGFAFDRVDADGLITSTLGRHTNDHMVSFYASTPSGVEVEYGWSARTVDRSWVVVRHDSPSMWGHKSVR 1knz A 2.45 BS01 rna W 0 N62 G65 K66 T69 S80 R83 N84 W87 D100 G131 K132 S133 S134 S135 N56 G59 K60 T63 S74 R77 N78 W81 D94 G122 K123 S124 S125 S126 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 TQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNNKFGSAIRNRNWLADTSRPAKLDEDVNKLRMMLGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVEVDDSFVDEKM 1knz B 2.45 BS01 rna W 0 D98 R105 R118 V119 K146 R149 D83 R90 R103 V104 K131 R134 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 GSMESTQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNDTSRPAKLDEDVNKLRMMLSSKGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVE 1knz C 2.45 BS01 rna X 0 N62 G65 K66 T69 S80 R83 N84 W87 R93 D100 G131 K132 S133 S134 S135 N56 G59 K60 T63 S74 R77 N78 W81 R87 D94 G122 K123 S124 S125 S126 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 TQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNNKFGSAIRNRNWLADTSRPAKLDEDVNKLRMMLGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVEVDDSFVDEKM 1knz D 2.45 BS01 rna X 0 D98 R105 R118 V119 K146 R149 D83 R90 R103 V104 K131 R134 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 GSMESTQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNDTSRPAKLDEDVNKLRMMLSSKGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVE 1knz I 2.45 BS01 rna Y 0 N62 G65 K66 T69 S80 R83 N84 W87 D100 G131 K132 S133 S134 S135 N56 G59 K60 T63 S74 R77 N78 W81 D94 G122 K123 S124 S125 S126 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 TQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNNKFGSAIRNRNWLADTSRPAKLDEDVNKLRMMLGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVEVDDSFVDEKM 1knz J 2.45 BS01 rna Y 0 D98 R105 R118 V119 K146 R149 D83 R90 R103 V104 K131 R134 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 GSMESTQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNDTSRPAKLDEDVNKLRMMLSSKGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVE 1knz M 2.45 BS01 rna Z 0 N62 G65 K66 T69 R83 N84 W87 R93 D100 G131 K132 S133 S134 S135 N56 G59 K60 T63 R77 N78 W81 R87 D94 G122 K123 S124 S125 S126 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 TQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNNKFGSAIRNRNWLADTSRPAKLDEDVNKLRMMLGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVEVDDSFVDEKM 1knz N 2.45 BS01 rna Z 0 D98 R105 R118 V119 K146 R149 D83 R90 R103 V104 K131 R134 ? 0003723 remove_due_to_license_issue P03536 11792322 2 ~ 6 GSMESTQQMAVSIINSSFEAAVVAATSALENMGIEYDYQDIYSRVKNKFDFVMDDSGVKNNPIGKAITIDQALNDTSRPAKLDEDVNKLRMMLSSKGIDQKMRVLNACFSVKRIPGKSSSIIKCTKLMRDKLERGEVE 1kog A 3.5 BS01 rna I 0 K249 I547 D549 N575 K577 F580 I582 R583 R609 K8 I306 D308 N334 K336 F339 I341 R342 R368 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog A 3.5 BS02 rna J 0 G344 L345 S347 Y348 R349 V498 E500 N502 G103 L104 S106 Y107 R108 V257 E259 N261 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog B 3.5 BS01 rna I 0 G344 L345 S347 Y348 R349 V498 E500 N502 G103 L104 S106 Y107 R108 V257 E259 N261 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog B 3.5 BS02 rna J 0 K249 I547 T548 D549 N575 K577 F580 I582 R583 R609 K8 I306 T307 D308 N334 K336 F339 I341 R342 R368 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog C 3.5 BS01 rna K 0 K249 I547 T548 D549 N575 E576 K577 F580 I582 R583 G597 K599 E600 K8 I306 T307 D308 N334 E335 K336 F339 I341 R342 G356 K358 E359 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog C 3.5 BS02 rna L 0 G344 L345 S347 Y348 R349 V498 G499 E500 N502 G103 L104 S106 Y107 R108 V257 G258 E259 N261 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog D 3.5 BS01 rna K 0 Q343 G344 L345 S347 Y348 R349 V498 E500 N502 Q102 G103 L104 S106 Y107 R108 V257 E259 N261 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog D 3.5 BS02 rna L 0 K246 K249 I547 T548 D549 N575 K577 F580 I582 R583 T586 K599 R609 K5 K8 I306 T307 D308 N334 K336 F339 I341 R342 T345 K358 R368 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog E 3.5 BS01 rna M 0 K246 K249 I547 T548 D549 N575 K577 F580 I582 R583 T586 V595 K599 E600 A607 R609 K5 K8 I306 T307 D308 N334 K336 F339 I341 R342 T345 V354 K358 E359 A366 R368 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog E 3.5 BS02 rna N 0 L345 S347 Y348 R349 V498 E500 N502 L104 S106 Y107 R108 V257 E259 N261 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog F 3.5 BS01 rna M 0 L345 S347 Y348 R349 V498 E500 N502 L104 S106 Y107 R108 V257 E259 N261 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog F 3.5 BS02 rna N 0 K246 K249 I547 T548 D549 N575 K577 G579 F580 I582 R583 T586 D598 K599 E600 K5 K8 I306 T307 D308 N334 K336 G338 F339 I341 R342 T345 D357 K358 E359 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog G 3.5 BS01 rna O 0 K246 K249 I547 T548 D549 N575 K577 F580 I582 R583 T586 G597 K599 E600 A607 R609 K5 K8 I306 T307 D308 N334 K336 F339 I341 R342 T345 G356 K358 E359 A366 R368 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kog H 3.5 BS01 rna P 0 I547 T548 D549 N575 K577 I578 F580 I582 R583 V595 G597 K599 E600 R609 I306 T307 D308 N334 K336 I337 F339 I341 R342 V354 G356 K358 E359 R368 Q381 D383 K465 Q140 D142 K224 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P0A8M3 11953757 69 ~ 105 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEE 1kpm A 1.8 BS01 VIT A 1 L2 L3 G6 K7 A18 I19 Y22 S23 C45 H48 D49 L2 L3 G6 K7 A17 I18 Y21 S22 C44 H47 D48 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 Ki=1.59uM remove_due_to_license_issue P59071 12079380 401 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 1kq2 A 2.71 BS01 rna R 0 Q8 K41 Y42 K57 H58 Q3 K36 Y37 K52 H53 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue A0A0H3JV59 12093755 26 ~ 32 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTV 1kq2 B 2.71 BS01 rna R 0 Q8 K41 Y42 K57 H58 Q3 K36 Y37 K52 H53 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue A0A0H3JV59 12093755 26 ~ 32 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTVE 1kq2 H 2.71 BS01 rna R 0 Q8 K41 Y42 K57 H58 Q4 K37 Y38 K53 H54 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue A0A0H3JV59 12093755 26 ~ 32 ENIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTVE 1kq2 I 2.71 BS01 rna R 0 Q8 K41 Y42 K57 H58 Q3 K36 Y37 K52 H53 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue A0A0H3JV59 12093755 26 ~ 32 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTV 1kq2 K 2.71 BS01 rna R 0 Q8 K41 Y42 K57 H58 Q3 K36 Y37 K52 H53 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue A0A0H3JV59 12093755 26 ~ 32 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTVE 1kq2 M 2.71 BS01 rna R 0 Q8 K41 Y42 K57 H58 Q3 K36 Y37 K52 H53 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue A0A0H3JV59 12093755 26 ~ 32 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTVE 1kqq A -1.00 BS01 dna B 0 I48 M49 S90 T92 I46 M47 S88 T90 ? 0003677,0006357 remove_due_to_license_issue Q24573 11867548 401 ~ 415 GWSFEEQFKQVRQLYEINDDPKRKEFLDDLFSFMQKRGTPINRLPIMAKSVLDLYELYNLVIARGGLVDVINKKLWQEIIKGLHLPSSITSAALTLRTQYMKYLYPYECEKKNLSTPAELQAAIDGNRREG 1kqq A -1.00 BS02 dna C 0 K76 W78 Q79 T92 S93 A95 L96 R99 N129 K74 W76 Q77 T90 S91 A93 L94 R97 N127 ? 0003677,0006357 remove_due_to_license_issue Q24573 11867548 416 ~ 430 GWSFEEQFKQVRQLYEINDDPKRKEFLDDLFSFMQKRGTPINRLPIMAKSVLDLYELYNLVIARGGLVDVINKKLWQEIIKGLHLPSSITSAALTLRTQYMKYLYPYECEKKNLSTPAELQAAIDGNRREG 1ksn A 2.1 BS02 FXV A 1 E97 T98 Y99 E147 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G219 C220 E83 T84 Y85 E135 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.4nM remove_due_to_license_issue P00742 12039587 401 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1kti A 1.97 BS01 AZC A 1 G135 L136 N284 H377 T378 N484 E672 S674 G675 G123 L124 N263 H346 T347 N453 E641 S643 G644 H377 K568 R569 K574 T676 K680 H346 K537 R538 K543 T645 K649 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=370uM remove_due_to_license_issue Ki=305000nM P00489 11895439 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 1ktt B 2.1 BS03 C02 B 1 H57 Y60A W60D E97A N98 L99 I174 D189 A190 V213 S214 W215 G216 G219 C220 H43 Y47 W50 E94 N95 L96 I172 D192 A193 V218 S219 W220 G221 G223 C224 H57 D102 E192 G193 D194 S195 G196 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 ic50=1.5uM remove_due_to_license_issue IC50=1500nM P00734 11960487 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1kv1 A 2.5 BS01 BMU A 1 E71 L75 M78 I84 D168 E67 L71 M74 I80 D160 D150 K152 N155 D168 T185 D142 K144 N147 D160 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=1.16uM remove_due_to_license_issue Kd=1160nM, kon=118000M-1-s-1, koff=0.140000s-1, IC50=21000nM Q16539 11896401 391 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1kv2 A 2.8 BS01 B96 A 1 V38 R67 E71 L75 T106 L108 M109 G110 H148 L167 D168 F169 V34 R63 E67 L71 T102 L104 M105 G106 H136 L155 D156 F157 D150 K152 N155 D168 T185 D138 K140 N143 D156 T158 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Kd=0.1nM, IC50=12nM, Ki=22nM, koff=0.000008s-1, kon=84900M-1-s-1 Q16539 11896401 391 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1kv5 A 1.65 BS01 PGA A 1 K13 H95 E167 I172 G212 S213 G234 K12 H94 E166 I171 G211 S212 G233 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=60uM remove_due_to_license_issue P04789 11997014 1350 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALISSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 1kv5 B 1.65 BS01 PGA B 1 K13 H95 E167 I172 G212 S213 G234 G235 K12 H94 E166 I171 G211 S212 G233 G234 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=60uM remove_due_to_license_issue P04789 11997014 2350 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALISSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 1kvo A 2.0 BS03 OAP A 1 F5 A17 A18 G22 G29 V30 C44 H47 D48 Y51 F5 A17 A18 G22 G29 V30 C44 H47 D48 Y51 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 ic50=0.013uM remove_due_to_license_issue IC50=21nM P14555 8831753 190 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 1kwq A 2.6 BS02 SG1 A 1 H94 V121 F131 L198 T199 T200 H92 V119 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue IC50=0.62nM P00918 12166932 900 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1kwr A 2.25 BS02 SG2 A 1 Q92 H94 H96 V121 L198 T199 T200 Q90 H92 H94 V119 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=0.25uM remove_due_to_license_issue IC50=245.5nM P00918 12166932 900 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1kyn A 3.5 BS01 KTP A 1 H57 A190 F191 K192 S195 G216 K217 H44 A176 F177 K178 S181 G198 K199 H57 D102 K192 G193 D194 S195 G196 H44 D88 K178 G179 D180 S181 G182 3.4.21.20 0002003,0002548,0004252,0005515,0005576,0005615,0005634,0005737,0005764,0005829,0005886,0006468,0006508,0006935,0006955,0008201,0008233,0008236,0010494,0016020,0016485,0016787,0019221,0019731,0022617,0030141,0030168,0032496,0035578,0035590,0042119,0042742,0048018,0050778,0050829,0050830,0050832,0050868,0051604,0062023,0070062,0070946,0071222,0089720,0098786,1901731 remove_due_to_license_issue IC50=4100nM P08311 11942800 601 IIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMR 1kz8 A 2.0 BS04 PFE A 1 K50 I53 H55 L56 K71 L73 K42 I45 H47 L48 K55 L57 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=0.83uM remove_due_to_license_issue P00636 12190310 738 NIVTLTRFVMEQGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGVKKLDVLSNDLVINVLKSSFATCVLVTEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRNVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1kz8 F 2.0 BS04 PFE F 1 K50 I53 H55 L56 K71 L73 K42 I45 H47 L48 K55 L57 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=0.83uM remove_due_to_license_issue P00636 12190310 838 NIVTLTRFVMEQGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGVKKLDVLSNDLVINVLKSSFATCVLVTEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRNVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1kzk A 1.09 BS01 JE2 A 1 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=41pM remove_due_to_license_issue P03369 11926820 701 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1kzk B 1.09 BS01 JE2 A 1 D25 G27 A28 D30 I47 G48 G49 P81 I84 D25 G27 A28 D30 I47 G48 G49 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 11926820 701 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1kzn A 2.3 BS01 CBN A 1 N46 E50 V71 D73 R76 G77 I78 P79 I90 R136 T165 N32 E36 V57 D59 R62 G63 I64 P65 I76 R103 T132 5.6.2.2 0003677,0003918,0005524,0006265 Kd=1.2nM remove_due_to_license_issue IC50=73nM P0AES6 12044152 1 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIGVSAAEVIMTVLHAHGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 1l1c A -1.00 BS01 rna C 0 V6 N9 N10 M25 G26 R27 F31 Q32 V6 N9 N10 M25 G26 R27 F31 Q32 ? 0003723 remove_due_to_license_issue P39805 11953318 1 ~ 29 MKIAKVINNNVISVVNEQGKELVVMGRGLAFQKKSGDDVDEARIEKVFTLDNKDV 1l1c B -1.00 BS01 rna C 0 K5 V6 I7 N8 N9 N10 R27 F31 Q32 K5 V6 I7 N8 N9 N10 R27 F31 Q32 ? 0003723 remove_due_to_license_issue P39805 11953318 1 ~ 29 MKIAKVINNNVISVVNEQGKELVVMGRGLAFQKKSGDDVDEARIEKVFTLDNKDV 1l2s A 1.94 BS01 STC A 1 S64 N152 Y221 G317 A318 T319 G320 S61 N149 Y218 G311 A312 T313 G314 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K309 A312 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=26uM remove_due_to_license_issue Ki=26000nM P00811 12121656 1115 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNLAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1l2s A 1.94 BS02 STC B 2 A79 Q250 L254 S257 P306 A76 Q247 L251 S254 P300 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K309 A312 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=26uM remove_due_to_license_issue Ki=26000nM P00811 12121656 3115 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNLAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1l5q A 2.25 BS04 CFF A 1 F285 A610 G612 Y613 F254 A571 G573 Y574 H377 K568 R569 K574 T676 K680 H338 K529 R530 K535 T637 K641 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=108uM remove_due_to_license_issue P06737 12204691 863 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1l5q A 2.25 BS05 CFF A 2 W174 H614 W153 H575 H377 K568 R569 K574 T676 K680 H338 K529 R530 K535 T637 K641 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=108uM remove_due_to_license_issue P06737 12204691 864 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1l5r A 2.1 BS04 RBF A 1 F285 E382 H571 A610 G612 Y613 R770 F771 F254 E343 H532 A571 G573 Y574 R731 F732 H377 K568 R569 K574 T676 K680 H338 K529 R530 K535 T637 K641 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=17uM remove_due_to_license_issue P06737 12204691 859 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEP 1l5s A 2.1 BS04 URC A 1 N282 F285 A610 G612 Y613 N252 F255 A572 G574 Y575 H377 K568 R569 K574 T676 K680 H339 K530 R531 K536 T638 K642 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=550uM remove_due_to_license_issue P06737 12204691 863 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPSD 1l5s B 2.1 BS05 URC B 1 N282 F285 A610 G612 Y613 N251 F254 A571 G573 Y574 H377 K568 R569 K574 T676 K680 H338 K529 R530 K535 T637 K641 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=550uM remove_due_to_license_issue P06737 12204691 1863 NVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1l6m A 2.4 BS01 DBH A 1 S68 W79 K134 S65 W76 K131 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 remove_due_to_license_issue P80188 12453412 201 TSDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCID 1l6m A 2.4 BS02 DBH A 2 W79 L94 Y100 Y106 K125 W76 L91 Y97 Y103 K122 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 remove_due_to_license_issue P80188 12453412 202 TSDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCID 1l6s A 1.7 BS02 DSB A 1 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue P0ACB2 11909869 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 1l6y A 1.9 BS02 4OX A 1 K194 Y200 F203 R204 R215 Q219 K246 V271 S272 Y311 K194 Y200 F203 R204 R215 Q219 K246 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue P0ACB2 11909869 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 1l7x A 2.3 BS04 CFF A 1 F285 H571 A610 G612 Y613 F256 H535 A574 G576 Y577 H377 K568 R569 K574 T676 K680 H341 K532 R533 K538 T640 K644 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=92uM remove_due_to_license_issue P06737 12204691 863 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFTVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEP 1l7x A 2.3 BS05 CFF A 2 W174 H614 W153 H578 H377 K568 R569 K574 T676 K680 H341 K532 R533 K538 T640 K644 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=92uM remove_due_to_license_issue P06737 12204691 864 ENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFTVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEP 1l7x B 2.3 BS05 CFF B 1 F285 H571 A610 G612 Y613 F258 H536 A575 G577 Y578 H377 K568 R569 K574 T676 K680 H342 K533 R534 K539 T641 K645 2.4.1.1 0000166,0002060,0004645,0005515,0005524,0005536,0005576,0005737,0005829,0005975,0005977,0005980,0006015,0008184,0009617,0016208,0016757,0019842,0030170,0030246,0031220,0032052,0034774,0042593,0042802,0070062,0070266,1904813 Kd=92uM remove_due_to_license_issue P06737 12204691 1863 GVENVAELKKSFNRHLHFTLVKDRNVATTRDYYFALAHTVRDHLVGRWIRTQQHYYDKCPKRVYYLSLEFYMGRTLQNTMINLGLQNACDEAIYQLGLDIEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEYGIFNQKIRDGWQVEEADDWLRYGNPWEKSRPEFMLPVHFYGKVEHTNTGTKWIDTQVVLALPYDTPVPGYMNNTVNTMRLWSARAPNDGDYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKASKFVFDAFPDQVAIQLNDTHPALAIPELMRIFVDIEKLPWSKAWELTQKTFAYTNHTVLPEALERWPVDLVEKLLPRHLEIIYEINQKHLDRIVALFPKDVDRLRRMSLIEEEGSKRINMAHLCIVGSHAVNGVAKIHSDIVKTKVFKDFSELEPDKFQNKTNGITPRRWLLLCNPGLAELIAEKIGEDYVKDLSQLTKLHSFLGDDVFLRELAKVKQENKLKFSQFLETEYKVKINPSSMFDVQVKRIHEYKRQLLNCLHVITMYNRIKKDPKKLFVPRTVIIGGKAAPGYHMAKMIIKLITSVADVVNNDPMVGSKLKVIFLENYRVSLAEKVIPATDLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENLFIFGMRIDDVAALDKKGYEAKEYYEALPELKLVIDQIDNGFFSPKQPDLFKDIINMLFYHDRFKVFADYEAYVKCQDKVSQLYMNPKAWNTMVLKNIAASGKFSSDRTIKEYAQNIWNVEPS 1l83 A 1.7 BS01 BNZ A 1 V87 A99 V111 L118 V87 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=0.4mM remove_due_to_license_issue P00720 1731252 400 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 1l8g A 2.5 BS01 DBD A 1 Y46 D48 V49 K120 D181 F182 C215 S216 A217 I219 G220 R221 M258 Q262 Y45 D47 V48 K119 D180 F181 C214 S215 A216 I218 G219 R220 M257 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=1100nM P18031 11732900 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKTYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1laf E 2.06 BS01 ARG E 1 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=14nM remove_due_to_license_issue P02911 7929349 240 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 1lag E 2.06 BS01 HIS E 1 Y14 F52 S69 S70 L71 S72 R77 L117 S120 Q122 D161 Y14 F52 S69 S70 L71 S72 R77 L117 S120 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=500nM remove_due_to_license_issue P02911 7929349 240 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 1lah E 2.06 BS01 ORN E 1 Y14 F52 S70 S72 R77 S120 Q122 D161 Y14 F52 S70 S72 R77 S120 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=30nM remove_due_to_license_issue P02911 7929349 240 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 1lan A 1.9 BS03 LEU A 1 D255 D273 D332 E334 T359 L360 D255 D273 D332 E334 T359 L360 K262 R336 K262 R336 3.4.11.1,3.4.11.5,3.4.13.23 0004177,0004180,0005737,0005739,0006508,0008233,0016805,0019538,0030145,0046872,0070006,0097718 Ki=60nM remove_due_to_license_issue P00727 7578088 500 TKGLVLGIYSKEKEEDEPQFTSAGENFNKLVSGKLREILNISGPPLKAGKTRTFYGLHEDFPSVVVVGLGKKTAGIDEQENWHEGKENIRAAVAAGCRQIQDLEIPSVEVDPCGDAQAAAEGAVLGLYEYDDLKQKRKVVVSAKLHGSEDQEAWQRGVLFASGQNLARRLMETPANEMTPTKFAEIVEENLKSASIKTDVFIRPKSWIEEQEMGSFLSVAKGSEEPPVFLEIHYKGSPNASEPPLVFVGKGITFDSGGISIKAAANMDLMRADMGGAATICSAIVSAAKLDLPINIVGLAPLCENMPSGKANKPGDVVRARNGKTIQVDNTDAEGRLILADALCYAHTFNPKVIINAATLTGAMDIALGSGATGVFTNSSWLWNKLFEASIETGDRVWRMPLFEHYTRQVIDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHLDIAGVMTNKDEVPYLRKGMAGRPTRTLIEFLFRFSQ 1lbf A 2.05 BS01 137 A 1 W8 E51 K53 S56 P57 S58 F89 K110 R182 L184 L187 S211 G212 L231 G233 S234 W7 E50 K52 S55 P56 S57 F88 K109 R181 L183 L186 S210 G211 L230 G232 S233 E51 K53 K110 E159 N180 E210 S211 E50 K52 K109 E158 N179 E209 S210 4.1.1.48 0000162,0004425,0004640,0006568,0006586,0009072,0016830,0016831,1901605 Kd=0.014uM remove_due_to_license_issue Q06121 12054868 300 PRYLKGWLKDVVQLSLRRPSFRASRQRPIISLNERILEFNKRNITAIIAEYKRKSPSGLDVERDPIEYSKFMERYAVGLSILTEEKYFNGSYETLRKIASSVSIPILMKDFIVKESQIDDAYNLGADTVLLIVKILTERELESLLEYARSYGMEPLIEINDENDLDIALRIGARFIGINSRDLETLEINKENQRKLISMIPSNVVKVAESGISERNEIEELRKLGVNAFLIGSSLMRNPEKIKEFIL 1lcp A 1.65 BS03 PLU A 1 K250 D255 K262 M270 D273 D332 E334 T359 K250 D255 K262 M270 D273 D332 E334 T359 K262 R336 K262 R336 3.4.11.1,3.4.11.5,3.4.13.23 0004177,0004180,0005737,0005739,0006508,0008233,0016805,0019538,0030145,0046872,0070006,0097718 Ki=0.23uM remove_due_to_license_issue P00727 7619821 500 TKGLVLGIYSKEKEEDEPQFTSAGENFNKLVSGKLREILNISGPPLKAGKTRTFYGLHEDFPSVVVVGLGKKTAGIDEQENWHEGKENIRAAVAAGCRQIQDLEIPSVEVDPCGDAQAAAEGAVLGLYEYDDLKQKRKVVVSAKLHGSEDQEAWQRGVLFASGQNLARRLMETPANEMTPTKFAEIVEENLKSASIKTDVFIRPKSWIEEQEMGSFLSVAKGSEEPPVFLEIHYKGSPNASEPPLVFVGKGITFDSGGISIKAAANMDLMRADMGGAATICSAIVSAAKLDLPINIVGLAPLCENMPSGKANKPGDVVRARNGKTIQVDNTDAEGRLILADALCYAHTFNPKVIINAATLTGAMDIALGSGATGVFTNSSWLWNKLFEASIETGDRVWRMPLFEHYTRQVIDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHLDIAGVMTNKDEVPYLRKGMAGRPTRTLIEFLFRFSQ 1ld7 B 2.0 BS05 U66 B 1 S599 W602 W606 R702 D797 C799 Y861 H862 S83 W86 W90 R186 D281 C283 Y345 H346 H748 R791 K794 D797 C799 Y800 D852 D859 H862 H232 R275 K278 D281 C283 Y284 D336 D343 H346 2.5.1.58 0003824,0004659,0004660,0005515,0005829,0005875,0005965,0006629,0008270,0008318,0018343,0046872 ic50=1.1nM remove_due_to_license_issue P49356 12036349 1003 PVWSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPEGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYDIINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKRERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVLGVPENALQPTHPVYNIGPDKVIQATTYFLQKPVPGF 1ld8 B 1.8 BS05 U49 B 1 S599 W602 W606 R702 D797 C799 Y861 H862 S83 W86 W90 R186 D281 C283 Y345 H346 H748 R791 K794 D797 C799 Y800 D852 D859 H862 H232 R275 K278 D281 C283 Y284 D336 D343 H346 2.5.1.58 0003824,0004659,0004660,0005515,0005829,0005875,0005965,0006629,0008270,0008318,0018343,0046872 ic50=3.5nM remove_due_to_license_issue P49356 12036349 1003 PVWSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPEGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYDIINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKRERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVLGVPENALQPTHPVYNIGPDKVIQATTYFLQKPVPGF 1le8 A 2.3 BS01 dna C 0 K100 R115 I119 R122 M123 K27 R42 I46 R49 M50 ? 0000981,0003677,0006355 remove_due_to_license_issue P0CY10 12121651 2 ~ 21 KSSISPQARAFLEQVFRRKQSLNSKEKEEVAKKCGITPLQVRVWFINKRMRSK 1le8 A 2.3 BS02 dna D 0 R82 Q113 V116 N120 R124 R9 Q40 V43 N47 R51 ? 0000981,0003677,0006355 remove_due_to_license_issue P0CY10 12121651 23 ~ 42 KSSISPQARAFLEQVFRRKQSLNSKEKEEVAKKCGITPLQVRVWFINKRMRSK 1le8 B 2.3 BS01 dna C 0 R135 Y156 R184 K188 R4 Y25 R53 K57 ? 0003677 remove_due_to_license_issue P0CY08 12121651 2 ~ 21 RGHRFTKENVRILESWFAKNIENPYLDTKGLENLMKNTSLSRIQIKNWVAARRAKEKTITIAPELADLLSGEPL 1le8 B 2.3 BS02 dna D 0 H134 R135 F136 Q175 N178 W179 H3 R4 F5 Q44 N47 W48 ? 0003677 remove_due_to_license_issue P0CY08 12121651 23 ~ 42 RGHRFTKENVRILESWFAKNIENPYLDTKGLENLMKNTSLSRIQIKNWVAARRAKEKTITIAPELADLLSGEPL 1lee A 1.9 BS01 R36 A 1 D34 G36 N76 Y77 V78 S79 F111 I123 L131 Y192 D214 G216 T217 I290 I300 D36 G38 N78 Y79 V80 S81 F113 I125 L133 Y194 D216 G218 T219 I292 I302 D34 S37 N39 W41 Y77 D214 T217 D36 S39 N41 W43 Y79 D216 T219 3.4.23.39 0004190,0006508 remove_due_to_license_issue P46925 12454457 500 LGSSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 1lei A 2.7 BS01 dna C 0 Y36 C38 E39 K122 K123 Q220 R246 Q247 Y18 C20 E21 K104 K105 Q202 R228 Q229 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04207 11970949 1 ~ 17 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 1lei A 2.7 BS02 dna D 0 R33 R35 S42 S45 R15 R17 S24 S27 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04207 11970949 1 ~ 17 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 1lei B 2.7 BS01 dna C 0 R54 S63 H64 G65 R16 S25 H26 G27 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P25799 11970949 1 ~ 17 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 1lei B 2.7 BS02 dna D 0 Y57 C59 E60 K144 K241 P243 Q274 K275 Q306 Y19 C21 E22 K106 K203 P205 Q236 K237 Q268 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P25799 11970949 1 ~ 17 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 1lev A 2.15 BS04 CLI A 1 V17 E20 G21 G26 G28 M30 T31 L34 V9 E12 G13 G18 G20 M22 T23 L26 D74 E97 E98 D118 L120 D121 E280 D50 E73 E74 D94 L96 D97 E256 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=2.5uM remove_due_to_license_issue P00636 12781194 342 NIVTLTRFVMEEGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHKLDVLSNDLVINVLKSSFATCVLVTEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRDVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1lf2 A 1.8 BS01 R37 A 1 D34 G36 N76 Y77 V78 S79 F111 I123 Y192 D214 G216 T217 S218 F294 D34 G36 N76 Y77 V78 S79 F111 I123 Y192 D214 G216 T217 S218 F294 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue P46925 12454457 330 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 1lf3 A 2.7 BS01 EH5 A 1 D34 G36 Y77 V78 S79 Y192 D214 G216 S218 F294 D36 G38 Y79 V80 S81 Y194 D216 G218 S220 F296 D34 S37 N39 W41 Y77 D214 T217 D36 S39 N41 W43 Y79 D216 T219 3.4.23.39 0004190,0006508 remove_due_to_license_issue P46925 12614616 332 LGSSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 1lfo A 2.3 BS01 OLA A 1 K31 G55 S56 K57 K31 G55 S56 K57 ? 0003682,0005324,0005504,0005515,0005543,0005634,0005654,0005737,0005782,0005829,0008289,0015908,0015909,0016209,0032000,0032052,0032991,0033552,0043066,0045179,0050892,0051977,0051978,0070301,0070538,0071456,0098869,1901363 Kd~2uM remove_due_to_license_issue Ki=2900nM P02692 9054409 128 MNFSGKYQVQSQENFEPFMKAMGLPEDLIQKGKDIKGVSEIVHEGKKVKLTITYGSKVIHNEFTLGEECELETMTGEKVKAVVKMEGDNKMVTTFKGIKSVTEFNGDTITNTMTLGDIVYKRVSKRI 1lfo A 2.3 BS02 OLA A 2 S39 M74 T102 S39 M74 T102 ? 0003682,0005324,0005504,0005515,0005543,0005634,0005654,0005737,0005782,0005829,0008289,0015908,0015909,0016209,0032000,0032052,0032991,0033552,0043066,0045179,0050892,0051977,0051978,0070301,0070538,0071456,0098869,1901363 Kd~2uM remove_due_to_license_issue Ki=2900nM P02692 9054409 129 MNFSGKYQVQSQENFEPFMKAMGLPEDLIQKGKDIKGVSEIVHEGKKVKLTITYGSKVIHNEFTLGEECELETMTGEKVKAVVKMEGDNKMVTTFKGIKSVTEFNGDTITNTMTLGDIVYKRVSKRI 1lgt A 1.7 BS03 BP3 A 1 H146 V148 M175 F187 H195 F202 H210 H241 N243 Y250 E260 H145 V147 M174 F186 H194 F201 H209 H240 N242 Y249 E259 1.13.11.39 0003824,0005506,0008198,0009056,0018583,0042178,0046872,0051213 Kd=0.8uM remove_due_to_license_issue P47228 12415290 300 SIRSLGYMGFAVSDVAAWRSFLTQKLGLMEAGTTDNGDLFRIDSRAWRIAVQQGEVDDLAFAGYEVADAAGLAQMADKLKQAGIAVTTGDASLARRRGVTGLITFADPFGLPLEIYYGASEVFEKPFLPGAAVSGFLTGEQGLGHFVRCVPDSDKALAFYTDVLGFQLSDVIDMKMGPDVTVPAYFLHCNERHHTLAIAAFPLPKRIHHFMLEVASLDDVGFAFDRVDADGLITSTLGRHTNDHMVSFYASTPSGVEVEYGWSARTVDRSWVVVRHDSPSMWGHKSV 1lgt A 1.7 BS04 BP3 A 2 L204 P205 K206 G256 E258 L203 P204 K205 G255 E257 1.13.11.39 0003824,0005506,0008198,0009056,0018583,0042178,0046872,0051213 Kd=0.8uM remove_due_to_license_issue P47228 12415290 301 SIRSLGYMGFAVSDVAAWRSFLTQKLGLMEAGTTDNGDLFRIDSRAWRIAVQQGEVDDLAFAGYEVADAAGLAQMADKLKQAGIAVTTGDASLARRRGVTGLITFADPFGLPLEIYYGASEVFEKPFLPGAAVSGFLTGEQGLGHFVRCVPDSDKALAFYTDVLGFQLSDVIDMKMGPDVTVPAYFLHCNERHHTLAIAAFPLPKRIHHFMLEVASLDDVGFAFDRVDADGLITSTLGRHTNDHMVSFYASTPSGVEVEYGWSARTVDRSWVVVRHDSPSMWGHKSV 1lgw A 1.85 BS01 1AN A 1 A99 L118 A99 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=100uM remove_due_to_license_issue P00720 12217695 401 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINQVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 1lhc H 1.95 BS03 DP7 H 1 H57 Y60A I174 D189 A190 E192 S195 W215 G216 G219 H43 Y47 I171 D191 A192 E194 S197 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=0.040000nM P00734 7893672 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1lhd H 2.35 BS03 DI2 H 1 H57 Y60A N98 L99 I174 A190 C191 E192 S195 S214 W215 G216 G219 H43 Y47 N95 L96 I171 A192 C193 E194 S197 S218 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=0.240000nM P00734 7893672 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1lhe H 2.25 BS03 DI3 H 1 H57 Y60A N98 L99 I174 D189 A190 C191 S195 W215 G216 G219 H43 Y47 N95 L96 I171 D191 A192 C193 S197 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 7893672 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1lhf H 2.4 BS03 DI4 H 1 H57 W60D L99 I174 D189 A190 C191 S195 S214 W215 G216 H43 W50 L96 I171 D191 A192 C193 S197 S218 W219 G220 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 7893672 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1lhg H 2.25 BS03 DI5 H 1 H57 Y60A W60D I174 A190 C191 S195 W215 G216 E217 G219 H43 Y47 W50 I171 A192 C193 S197 W219 G220 E221 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 7893672 400 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1lhu A 1.8 BS02 EST A 1 S42 G58 D65 F67 V105 M107 K134 I141 S29 G45 D52 F54 V92 M94 K121 I128 ? remove_due_to_license_issue IC50=50nM, Kd=1.5nM P04278 12065592 301 PAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGPLTSKRHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAEISASAPTSLRSC 1lhv A 2.0 BS03 NOG A 1 S41 S42 D65 F67 N82 V105 M107 M139 L171 S29 S30 D53 F55 N70 V93 M95 M123 L155 ? remove_due_to_license_issue Kd=1.2nM P04278 12065592 301 PPAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGPLHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAEISASAPTSLRSCD 1lhw A 1.75 BS02 ESM A 1 S42 G58 D65 F67 L80 N82 V127 K134 I141 S30 G46 D53 F55 L68 N70 V115 K119 I126 ? Kd=6.9nM remove_due_to_license_issue Kd=0.832000nM P04278 12228253 301 PPAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGPKRHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAEISASAPTSLRSCD 1li3 A 1.85 BS01 3CH A 1 A99 Q102 L118 A99 Q102 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=56uM remove_due_to_license_issue P00720 12217695 401 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINQVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 1li6 A 2.0 BS01 5MP A 1 Y88 A99 Q102 V111 Y88 A99 Q102 V111 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Ka=6300M^-1 remove_due_to_license_issue P00720 12217695 400 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINQVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 1ljt A 2.0 BS01 HDI A 1 P1 M2 K32 Y36 H62 I64 V106 P1 M2 K32 Y36 H62 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM, Ki=21000nM P14174 11997397 115 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 1ljt A 2.0 BS02 HDI C 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM, Ki=21000nM P14174 11997397 115 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 1ljt B 2.0 BS01 HDI A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM, Ki=21000nM P14174 11997397 115 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 1ljt B 2.0 BS02 HDI B 1 P1 M2 K32 Y36 H62 I64 F113 P1 M2 K32 Y36 H62 I64 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM, Ki=21000nM P14174 11997397 115 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 1lke A 1.9 BS01 DOG A 1 Q28 Y39 Y47 R58 H86 F114 W129 L131 Q24 Y35 Y43 R54 H82 F110 W120 L122 ? 0000302,0005576,0005737,0006629,0006950,0031409 Kd=30.2nM remove_due_to_license_issue P09464 12823976 500 DGACPEVKPVDNFDWSQYHGKWWQVAAYPDHITKYGKCGWAEYTPEGKSVKVSRYSVIHGKEYFSEGTAYPVGDSKIGKIYHSYTIGGVTQEGVFNVLSTDNKNYIIGYFCSYGHMDLVWVLSRSMVLTGEAKTAVENYLIGSPVVDSQKLVYSDFS 1lkx A 3.0 BS02 ADP A 1 N49 K52 G104 G106 K107 T108 E109 N154 N156 N41 K44 G96 G98 K99 T100 E101 N146 N148 S103 G104 T108 N154 S157 S158 G389 E391 S95 G96 T100 N146 S149 S150 G367 E369 ? 0003774,0005524,0016459 remove_due_to_license_issue Q03479 12032065 791 GVPDFVLLNQITENAFIENLTMRHKSDNIYTYIGDVVISTNPFKNLNIYKESDIKAYNGRYKYEMPPHMYALANDAYRSMRQSQENQCVIISGESGAGKTEASKKIMQFLTFVSSNQSPNGERISKMLLDSNPLLEAFGNAKTLRNDNSSRFGKYMEMQFNAVGSPIGGKITNYLLEKSRVVGRTQGERSFHIFYQMLKGLSQSKLDELGLTPNAPAYEYLKKSGCFDVSTIDDSGEFKIIVKAMETLGLKESDQNSIWRILAAILHIGNITFAEAAEQTTVKVSDTKSLAAAASCLKTDQQSLSIALCYRSVISVPMDCNQAAYSRDALAKALYERLFNWLVSKINTIINCTTEKGPVIGILDIYGFEVFQNNSFEQLNINFCNEKLQQLFIELTLKSEQEEYVREGIEWKNIEYFNNKPICELIEKKPIGLISLLDEACLIAKSTDQTFLDSICKQFEKNPHLQSYVVSKDRSIGDTCFRLKHYAGDVTYDVRGFLDKNKDTLFGDLISSMQSSSDPLVQGLFPETAGSQFRNAMNALITTLLACSPHYVRCIKSNDNKQAGVIDEDRVRHQVRYLGLLENVRVRRAGFAGRIEYTRFYNRYKMLCKKKQATELILQQHNIDKEEIRMGKTKVFIRNPTTLFYFEEKR 1ll4 A 2.8 BS01 AMI A 1 Y43 F71 D169 E171 M237 Y239 D240 Y293 W378 Y8 F36 D134 E136 M202 Y204 D205 Y258 W343 D167 D169 E171 Y239 D132 D134 E136 Y204 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P0CB51 12079386 503 GGFRSVVYFVNWAIYGRGHNPQDLKADQFTHILYAFANIRPSGEVYLSDTWADTDKHYPGDKWDEPGNNVYGCIKQMYLLKKNNRNLKTLLSIGGWTYSPNFKTPASTEEGRKKFADTSLKLMKDLGFDGIDIDWEYPEDEKQANDFVLLLKACREALDAYSAKHPNGKKFLLTIASPAGPQNYNKLKLAEMDKYLDFWNLMAYDFSGSWDKVSGHMSNVFPSTTKPESTPFSSDKAVKDYIKAGVPANKIVLGMPLYGRAFASTDGIGTSFNGVGGGSWENGVWDYKDMPQQGAQVTELEDIAASYSYDKNKRYLISYDTVKIAGKKAEYITKNGMGGGMWWESSSDKTGNESLVGTVVNGLGGTGKLEQRENELSYPESVYDNLKNGMPS 1llb B 1.72 BS01 PCN B 1 S64 L119 Q120 N289 L293 G317 A318 G320 S61 L116 Q117 N286 L290 G314 A315 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 12323371 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1lnm A 1.9 BS01 DTX A 1 Y39 H86 F114 W129 Y35 H82 F110 W121 ? 0000302,0005576,0005737,0006629,0006950,0031409 Kd=2nM remove_due_to_license_issue P09464 12823976 700 DGACPEVKPVDNFDWSQYHGKWWQVAAYPDHITKYGKCGWAEYTPEGKSVKVSRYSVIHGKEYFSEGTAYPVGDSKIGKIYHSYTIGGVTQEGVFNVLSTDNKNYIIGYFCSYKGHMDLVWVLSRSMVLTGEAKTAVENYLIGSPVVDSQKLVYSDFSCK 1lo1 A -1.00 BS01 dna B 0 R101 Y113 H114 Y115 K124 K128 Q132 R174 R177 V178 R179 G180 R182 Q183 K184 R5 Y17 H18 Y19 K28 K32 Q36 R78 R81 V82 R83 G84 R86 Q87 K88 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue O95718 12654265 1 ~ 13 AIPKRLCLVCGDIASGYHYGVASCEACKAFFKRTIQGNIEYSCPATNECEITKRRRKSCQACRFMKALKVGMLKEGVRLDRVRGGRQKYK 1lo1 A -1.00 BS02 dna C 0 E121 R129 R152 K153 Q156 R159 R179 G180 G181 R182 E25 R33 R56 K57 Q60 R63 R83 G84 G85 R86 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue O95718 12654265 14 ~ 26 AIPKRLCLVCGDIASGYHYGVASCEACKAFFKRTIQGNIEYSCPATNECEITKRRRKSCQACRFMKALKVGMLKEGVRLDRVRGGRQKYK 1lol A 1.9 BS02 XMP A 1 A18 D20 K42 S127 S158 P180 G202 R203 A8 D10 K32 S117 S148 P170 G184 R185 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=0.41uM remove_due_to_license_issue O26232 12011084 2001 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGGETLRFADAIIVGRSIYLADNPAAAAAGIIESI 1lol B 1.9 BS02 XMP B 1 A1018 D1020 K1042 S1158 G1202 R1203 A8 D10 K32 S148 G187 R188 K1042 D1070 K1072 D1075 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=0.41uM remove_due_to_license_issue O26232 12011084 2002 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDLLIPE 1loq A 1.5 BS01 U A 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D7 K29 D57 K59 M113 S114 P167 Q172 G189 R190 K42 D70 K72 D75 K29 D57 K59 D62 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=0.2mM remove_due_to_license_issue O26232 12011084 2001 RLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESI 1lor A 1.6 BS01 BMP A 1 D20 K42 K72 M126 S127 P180 Q185 G202 R203 D7 K29 K59 M113 S114 P167 Q172 G189 R190 K42 D70 K72 D75 K29 D57 K59 D62 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=8.8pM remove_due_to_license_issue O26232 12011084 2001 RLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESI 1lox A 2.4 BS02 RS7 A 1 E357 H361 L362 H366 L408 F415 H545 Q548 I593 L597 E343 H347 L348 H352 L394 F401 H531 Q534 I579 L583 H361 H366 H541 H545 I663 H347 H352 H527 H531 I647 1.13.11.-,1.13.11.12,1.13.11.31,1.13.11.33 0001503,0002820,0004052,0005506,0005546,0005737,0005811,0005829,0005886,0006629,0006631,0006646,0008289,0009898,0010811,0016020,0016165,0016702,0019369,0019372,0019395,0030282,0030838,0034440,0034976,0035358,0035963,0042060,0043277,0043651,0046872,0050473,0050727,0051122,0051213,0070374,0071277,1901074,2001303 Ki=3uM remove_due_to_license_issue P12530 9406550 841 GVYRVCVSTGASIYAGSKNKVELWLVGQHGEVELGSCLRPTRNKEEEFKVNVSKYLGSLLFVRLRKKHFLKEDAWFCNWISVQALGAAEDKYWFPCYRWVVGDGVQSLPVGTGCTTVGDPQGLFQKHREQELEERRKLYQWGSWKEGLILNVAGSKLTDLPVDERFLEDKKIDFELKNSLNILAPWKTLDDFNRIFWRSKLARRVRDSWQEDSLFGYQFLNGANPMLLRRSVQLPARLVFPPGMEELQAQLEKELKAGTLFEADFALLDNIKANVILYCQQYLAAPLVMLKLQPDGKLMPMVIQLHLPKIGSSPPPLFLPTDPPMVWLLAKCWVRSSDFQVHELNSHLLRGHLMAEVFTVATMRCLPSIHPVFKLIVPHLRYTLEINVRARNGLVSDFGIFDQIMSTGGGGHVQLLQQAGAFLTYRSFCPPDDLADRGLLGVESSFYAQDALRLWEIISRYVQGIMGLYYKTDEAVRDDLELQSWCREITEIGLQGAQKQGFPTSLQSVAQACHFVTMCIFTCTGQHSSIHLGQLDWFTWVPNAPCTMRLPPPTTKDATLETVMATLPNLKQSSLQMSIVWQLGRDIMVPLGQHQEEYFSGPEPRAVLEKFREELAIMDKEIEVRNEKLDIPYEYLRPSIVENSVAI 1lpg B 2.0 BS02 IMA B 1 E97 T98 Y99 R143 E147 K148 F174 D189 A190 C191 Q192 S195 W215 G216 G219 C220 E83 T84 Y85 R132 E135 K136 F162 D179 A180 C181 Q182 S185 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=82nM remove_due_to_license_issue Ki=82nM P00742 12061878 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1lpk B 2.2 BS02 CBB B 1 R143 F174 D189 A190 C191 Q192 W215 G216 G219 C220 R132 F162 D179 A180 C181 Q182 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=28nM remove_due_to_license_issue P00742 12061878 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1lpz B 2.4 BS02 CMB B 1 T98 Y99 R143 D189 A190 C191 Q192 W215 G216 G219 C220 T84 Y85 R132 D179 A180 C181 Q182 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=25nM remove_due_to_license_issue Ki=25nM P00742 12061878 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1lq2 A 2.7 BS01 IDD A 1 D95 R158 K206 H207 M250 D285 W286 W434 E491 D95 R158 K206 H207 M250 D285 W286 W434 E491 D285 E491 D285 E491 3.2.1.21 0004553,0005975,0016798 remove_due_to_license_issue Q9XEI3 14597633 621 DYVLYKDATKPVEDRVADLLGRMTLAEKIGQMTQIERLVATPDVLRDNFIGSLLSGGGSVPRKGATAKEWQDMVDGFQKACMSTRLGIPMIYGIDAVHGQNNVYGATIFPHNVGLGATRDPYLVKRIGEATALEVRATGIQYAFAPCIAVCRDPRWGRCYESYSEDRRIVQSMTELIPGLQGDVPKDFTSGMPFVAGKNKVAACAKHFVGDGGTVDGINENNTIINREGLMNIHMPAYKNAMDKGVSTVMISYSSWNGVKMHANQDLVTGYLKDTLKFKGFVISDWEGIDRITTPAGSDYSYSVKASILAGLDMIMVPNKYQQFISILTGHVNGGVIPMSRIDDAVTRILRVKFTMGLFENPYADPAMAEQLGKQEHRDLAREAARKSLVLLKNGKTSTDAPLLPLPKKAPKILVAGSHADNLGYQCGGWTIEWQGDTGRTTVGTTILEAVKAAVDPSTVVVFAENPDAEFVKSGGFSYAIVAVGEHPYTETKGDNLNLTIPEPGLSTVQAVCGGVRCATVLISGRPVVVQPLLAASDALVAAWLPGSEGQGVTDALFGDFGFTGRLPRTWFKSVDQLPMNVGDAHYDPLFRLGYGLTTNAT 1lqd B 2.7 BS02 CMI B 1 D189 A190 C191 Q192 W215 G216 C220 G226 D179 A180 C181 Q182 W205 G206 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=9nM P00742 12061878 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1lqe A 2.2 BS02 IMA A 1 L99 D189 S190 C191 Q192 W215 G216 G219 C220 L81 D171 S172 C173 Q174 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Ki=1507nM remove_due_to_license_issue P00760 12061878 250 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1lrr A 2.65 BS01 dna B 0 G115 R116 T117 R118 Y120 N133 Q134 N150 R155 G52 R53 T54 R55 Y57 N70 Q71 N87 R92 ? 0003677 remove_due_to_license_issue P0AFY8 12379844 1 ~ 12 TIKDKVRAMRELLLSDEYAEQKRAVNRFMLLLSTLYSLDAQAFAEATESLHGRTRVYFAADEQTLLKNGNQTKPKHVPGTPYWVITNTNTGRKCSMIEHIMQSMQFPAELIEKVCGTI 1lrr A 2.65 BS02 dna C 0 R86 A87 V88 R116 K138 N152 T153 R23 A24 V25 R53 K75 N89 T90 ? 0003677 remove_due_to_license_issue P0AFY8 12379844 1 ~ 12 TIKDKVRAMRELLLSDEYAEQKRAVNRFMLLLSTLYSLDAQAFAEATESLHGRTRVYFAADEQTLLKNGNQTKPKHVPGTPYWVITNTNTGRKCSMIEHIMQSMQFPAELIEKVCGTI 1lrr D 2.65 BS01 dna E 0 G115 R116 T117 R118 Y120 N150 R155 G52 R53 T54 R55 Y57 N87 R92 ? 0003677 remove_due_to_license_issue P0AFY8 12379844 1 ~ 12 TIKDKVRAMRELLLSDEYAEQKRAVNRFMLLLSTLYSLDAQAFAEATESLHGRTRVYFAADEQTLLKNGNQTKPKHVPGTPYWVITNTNTGRKCSMIEHIMQSMQFPAELIEKVCGTI 1lrr D 2.65 BS02 dna F 0 R86 A87 V88 K138 T151 N152 T153 R23 A24 V25 K75 T88 N89 T90 ? 0003677 remove_due_to_license_issue P0AFY8 12379844 1 ~ 12 TIKDKVRAMRELLLSDEYAEQKRAVNRFMLLLSTLYSLDAQAFAEATESLHGRTRVYFAADEQTLLKNGNQTKPKHVPGTPYWVITNTNTGRKCSMIEHIMQSMQFPAELIEKVCGTI 1lrt A 2.2 BS02 TAD A 1 T240 R241 D261 S262 S263 W269 I313 E408 E431 T109 R110 D130 S131 S132 W138 I182 E274 E284 1.1.1.205 0003824,0003938,0006164,0016491 Ki=2.3uM remove_due_to_license_issue P50097 12403633 901 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFKRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIRDKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICEQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWEEGVDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVE 1lrt B 2.2 BS02 TAD B 1 T240 R241 D261 S262 S263 W269 I313 E408 T109 R110 D130 S131 S132 W138 I182 E274 1.1.1.205 0003824,0003938,0006164,0016491 Ki=2.3uM remove_due_to_license_issue P50097 12403633 902 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFKRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIRDKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICEQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVE 1lst A 1.8 BS01 LYS A 1 Y14 F52 S70 S72 R77 L117 S120 T121 Q122 D161 Y14 F52 S70 S72 R77 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 remove_due_to_license_issue P02911 8496186 240 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 1lt6 D 2.2 BS01 GAA D 1 Y12 E51 H57 Q61 W88 N90 K91 Y12 E51 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 remove_due_to_license_issue P32890 9384564 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1lt6 E 2.2 BS01 GAA E 1 E51 H57 Q61 W88 N90 K91 E51 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 remove_due_to_license_issue P32890 9384564 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1lv8 A 2.3 BS02 9PP A 1 G32 S33 H86 N115 A116 A117 G118 F200 E201 M219 S220 N243 G30 S31 H84 N113 A114 A115 G116 F198 E199 M217 S218 N241 S33 H64 Y88 A116 M219 S220 S31 H62 Y86 A114 M217 S218 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Kd=3.5uM remove_due_to_license_issue P55859 15342253 3001 NGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGQNPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDQAAQKLEQFVSLLMASIPV 1lv8 B 2.3 BS02 9PP B 1 G1032 S1033 H1086 N1115 A1116 A1117 G1118 F1200 E1201 M1219 S1220 N1243 G30 S31 H84 N113 A114 A115 G116 F198 E199 M217 S218 N241 S1033 H1064 Y1088 A1116 M1219 S1220 S31 H62 Y86 A114 M217 S218 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Kd=3.5uM remove_due_to_license_issue P55859 15342253 3002 NGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGQNPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDQAAQKLEQFVSLLMASIPV 1lvc A 3.6 BS01 DOT A 1 K346 H351 K353 S354 K382 E386 D493 H577 G578 T579 N583 F586 K55 H60 K62 S63 K91 E95 D202 H286 G287 T288 N292 F295 4.6.1.1 0005576,0008294 remove_due_to_license_issue P40136 12485993 999 RIDVLKGEKALKASGLVPEHADAFKKIARELNTYILFRPVNKLATNLIKSGVATKGLNVHGKSSDWGPVAGYIPFDQDLSKKHGQQLAVEKGNLENKKSITEHEGEIGKIPLKLDHLRIEELKENGIILKGKKEIDNGKKYYLLESNNQVYEFRISDENNEVQYKTKEGKITVLGEKFNWRNIEVMAKNVEGVLKPLTADYDLFALAPSLTEIKKQIPQKEWDKVVNTPNSLEKQKGVTNLLIKYGIERKPDSTKGTLSNWQKQMLDRLNEAVKYTGYTGGDVVNHGTEQDNEEFPEKDNEIFIINPEGEFILTKNWEMTGRFIEKNITGKDYLYYFNRSYNKIAPGNKAYIEWTDPITKAKINTIPTSAEFIKNLSSIRRSSSVKKIAGYLSDYYNSANHIFSQEKKRKISIFRGIQAYNEIENVLKSKQIAPEYKNYFQYLKERITNQVQLLLTHQKFKLLYKQLNFTENETDNFEVFQKIID 1lvk A 1.9 BS02 MNT A 1 N127 P128 S181 G182 G184 K185 T186 E187 N233 N234 N235 N126 P127 S180 G181 G183 K184 T185 E186 N229 N230 N231 S181 G182 T186 N233 S236 S237 G457 E459 S180 G181 T185 N229 S232 S233 G453 E455 ? 0003774,0005524,0016459,0051015 remove_due_to_license_issue P08799 9405148 999 NPIHDRTSDYHKYLKVKQGDSDLFKLTVSDKRYIWYNPDPKERDSYECGEIVSETSDSFTFKTSDGQDRQVKKDDANQRNPIKFDGVEDMSELSYLNEPAVFHNLRVRYNQDLIYTYSGLFLVAVNPFKRIPIYTQEMVDIFKGRRRNEVAPHIFAISDVAYRSMLDDRQNQSLLITGESGAGKTENTKKVIQYLASVAGRNQAGVLEQQILQANPILEAFGNAKTTRNNNSSRFGKFIEIQFNNAGFISGASIQSYLLEKSRVVFQSTSERNYHIFYQLLAGATAEEKKALHLAGPESFNYLNQSGCVDIKGVSDEDEFKITRQAMDIVGFSQEEQMSIFKIIAGILHLGNIKFEKGAGEGAVLKDKTALNAASTVFGVNPSVLEKALMEPRILAGRDLVAQHLNVEKSSSSRDALVKALYGRLFLWLVKKINNVLCSERKAYFIGVLDISGFEIFKVNSFEQLCINYTNEKLQQFFNHHMFKVEQEKYLKEKINLDSQATIDLIDGRQPPGILALLDEQSVFPNATDNTLITKLHSHFSKKNAKYEEPRFSKTEFGVTHYAGQVMYEIQDWLEKNKDPLQQDLELCFKDSSDNVVTKLFNDPNIASRAFLTVAAQYKEQLASLMATLETTNPHFVRCIIPNNKQLPAKLEDKVVLDQLRCNGVLEGIRITRKGFPNRIIYADFVKRYYDLAPNVPRDAEDSQKATDAVLKHLNIDPEQFRFGITKIFFRAGQLARIEEARE 1lvu A 2.05 BS02 9PP A 1 G32 S33 H86 N115 A116 G118 F200 E201 V217 M219 S220 N243 G31 S32 H85 N114 A115 G117 F199 E200 V216 M218 S219 N242 S33 H64 Y88 A116 M219 S220 S32 H63 Y87 A115 M218 S219 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Kd=4.8uM remove_due_to_license_issue P55859 15342253 6100 QNGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGQNPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYEEAGKQAAQKLEQFVSLLMASIPV 1lvu B 2.05 BS02 9PP B 1 G1032 S1033 R1084 H1086 N1115 A1116 A1117 G1118 F1200 E1201 V1217 M1219 S1220 N1243 G31 S32 R83 H85 N114 A115 A116 G117 F199 E200 V216 M218 S219 N242 S1033 H1064 Y1088 A1116 M1219 S1220 H1257 S32 H63 Y87 A115 M218 S219 H250 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Kd=4.8uM remove_due_to_license_issue P55859 15342253 6200 QNGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESTVPGHAGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGQNPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYEHEEVLEAGKQAAQKLEQFVSLLMASIPV 1lxf C -1.00 BS03 BEP C 1 L41 L48 M60 I61 V72 F77 M80 M81 L41 L48 M60 I61 V72 F77 M80 M81 ? 0005509 remove_due_to_license_issue P63316 12060657 92 MDDIYKAAVEQLTEEQKNEFKAAFDIFVLGAEDGCISTKELGKVMRMLGQNPTPEELQEMIDEVDEDGSGTVDFDEFLVMMVRCMKDDS 1lyx A 1.9 BS01 PGA A 1 K12 H95 E165 I170 G171 G210 S211 G232 N233 K10 H93 E163 I168 G169 G208 S209 G230 N231 N10 K12 H95 E97 E165 G171 S211 N8 K10 H93 E95 E163 G169 S209 5.3.1.1 0004807,0005829,0006094,0006096,0016853,0019563,0042802,0046166 Ki=0.029mM remove_due_to_license_issue Q07412 12403619 401 RKYFVAANWKCNGTLESIKSLTNSFNNLDFDPSKLDVVVFPVSVHYDHTRKLLQSKFSTGIQNVSKFGNGSYTGEVSAEIAKDLNIEYVIIGHFERRKYFHETDEDVREKLQASLKNNLKAVVCFGESLEQREQNKTIEVITKQVKAFVDLIDNFDNVILVYEPLWAIGTGKTATPEQAQLVHKEIRKIVKDTCGEKQANQIRILYGGSVNTENCSSLIQQEDIDGFLVGNASLKESFVDIIKSAM 1lzo B 2.8 BS01 PGA B 1 K12 S211 G232 N233 K10 S209 G230 N231 N10 K12 H95 E97 E165 G171 S211 N8 K10 H93 E95 E163 G169 S209 5.3.1.1 0004807,0005829,0006094,0006096,0016853,0019563,0042802,0046166 remove_due_to_license_issue Q07412 12403619 7251 RKYFVAANWKCNGTLESIKSLTNSFNNLDFDPSKLDVVVFPVSVHYDHTRKLLQSKFSTGIQNVSKFGNGSYTGEVSAEIAKDLNIEYVIIGHFERRKYFHETDEDVREKLQASLKNNLKAVVCFGESLEQREQNKTIEVITKQVKAFVDLIDNFDNVILVYEPLWAIGTGKTATPEQAQLVHKEIRKIVKDTCGEKQANQIRILYGGSVNTENCSSLIQQEDIDGFLVGNASLKESFVDIIKSAM 1lzq A 2.2 BS01 0ZQ A 1 R8 D25 G27 A28 D29 D30 I47 G48 G49 I50 R8 D25 G27 A28 D29 D30 I47 G48 G49 I50 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.1nM remove_due_to_license_issue P03367 12699382 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKVIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1lzq B 2.2 BS01 0ZQ A 1 D125 G127 V132 G148 G149 P181 T182 D25 G27 V32 G48 G49 P81 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 12699382 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKVIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1m0b A 2.45 BS01 0ZQ B 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 D25 G27 A28 D29 D30 I47 G48 G49 I50 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15560786 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1m0b B 2.45 BS01 0ZQ B 1 D125 G127 A128 D130 G148 G149 P181 V182 I184 D25 G27 A28 D30 G48 G49 P81 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.53nM remove_due_to_license_issue P03367 15560786 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1m0n A 2.2 BS01 HCP A 1 Q52 M53 A112 N115 W138 H139 E210 S215 D243 A245 Q246 K272 R406 Q50 M51 A110 N113 W136 H137 E208 S213 D241 A243 Q244 K270 R404 G21 W138 E210 D243 Q246 K272 T303 R406 G19 W136 E208 D241 Q244 K270 T301 R404 4.1.1.64 0008483,0016831,0030170,0047432 Ki=6mM remove_due_to_license_issue P16932 12369820 434 LNDDATFWRNARHHLVRYGGTFEPMIIERAKGSFVYDADGRAILDFTSGQMSAVLGHCHPEIVSVIGEYAGKLDHLFSEMLSRPVVDLATRLANITPPGLDRALLLSTGAESNEAAIRMAKLVTGKYEIVGFAQSWHGMTGAAASATYSAGRKGVGPAAVGSFAIPAPFTYRPRFERNGAYDYLAELDYAFDLIDRQSSGNLAAFIAEPILSSGGIIELPDGYMAALKRKCEARGMLLILDEAQTGVGRTGTMFACQRDGVTPDILTLSKTLGAGLPLAAIVTSAAIEERAHELGYLFYTTHVSDPLPAAVGLRVLDVVQRDGLVARANVMGDRLRRGLLDLMERFDCIGDVRGRGLLLGVEIVKDRRTKEPADGLGAKITRECMNLGLSMNIVQLPGMGGVFRIAPPLTVSEDEIDLGLSLLGQAIERAL 1m0o A 2.4 BS01 MPM A 1 Q52 G111 A112 W138 H139 E210 D243 Q246 K272 R406 Q50 G109 A110 W136 H137 E208 D241 Q244 K270 R404 G21 W138 E210 D243 Q246 K272 T303 R406 G19 W136 E208 D241 Q244 K270 T301 R404 4.1.1.64 0008483,0016831,0030170,0047432 Ki=4.9mM remove_due_to_license_issue P16932 12369820 434 LNDDATFWRNARHHLVRYGGTFEPMIIERAKGSFVYDADGRAILDFTSGQMSAVLGHCHPEIVSVIGEYAGKLDHLFSEMLSRPVVDLATRLANITPPGLDRALLLSTGAESNEAAIRMAKLVTGKYEIVGFAQSWHGMTGAAASATYSAGRKGVGPAAVGSFAIPAPFTYRPRFERNGAYDYLAELDYAFDLIDRQSSGNLAAFIAEPILSSGGIIELPDGYMAALKRKCEARGMLLILDEAQTGVGRTGTMFACQRDGVTPDILTLSKTLGAGLPLAAIVTSAAIEERAHELGYLFYTTHVSDPLPAAVGLRVLDVVQRDGLVARANVMGDRLRRGLLDLMERFDCIGDVRGRGLLLGVEIVKDRRTKEPADGLGAKITRECMNLGLSMNIVQLPGMGGVFRIAPPLTVSEDEIDLGLSLLGQAIERAL 1m0q A 2.0 BS01 EPC A 1 Q52 T110 A112 W138 H139 E210 S215 D243 A245 Q246 K272 R406 Q50 T108 A110 W136 H137 E208 S213 D241 A243 Q244 K270 R404 G21 W138 E210 D243 Q246 K272 T303 R406 G19 W136 E208 D241 Q244 K270 T301 R404 4.1.1.64 0008483,0016831,0030170,0047432 Ki=1.1mM remove_due_to_license_issue P16932 12369820 435 LNDDATFWRNARHHLVRYGGTFEPMIIERAKGSFVYDADGRAILDFTSGQMSAVLGHCHPEIVSVIGEYAGKLDHLFSEMLSRPVVDLATRLANITPPGLDRALLLSTGAESNEAAIRMAKLVTGKYEIVGFAQSWHGMTGAAASATYSAGRKGVGPAAVGSFAIPAPFTYRPRFERNGAYDYLAELDYAFDLIDRQSSGNLAAFIAEPILSSGGIIELPDGYMAALKRKCEARGMLLILDEAQTGVGRTGTMFACQRDGVTPDILTLSKTLGAGLPLAAIVTSAAIEERAHELGYLFYTTHVSDPLPAAVGLRVLDVVQRDGLVARANVMGDRLRRGLLDLMERFDCIGDVRGRGLLLGVEIVKDRRTKEPADGLGAKITRECMNLGLSMNIVQLPGMGGVFRIAPPLTVSEDEIDLGLSLLGQAIERAL 1m13 A 2.15 BS01 HYF A 1 L209 M243 S247 F281 C284 Q285 F288 W299 M323 H407 I414 L48 M82 S86 F120 C123 Q124 F127 W138 M162 H246 I253 ? 0003677,0004879,0006355 Kd=27nM remove_due_to_license_issue O75469 12578355 435 GLTEEQRMMIRELMDAQMKTFDTTFSHFKNFRLPGVKWSQVRKDLCSLKVSLQLRGEDGSVWNYKPPADSGGKEIFSLLPHMADMSTYMFKGIISFAKVISYFRDLPIEDQISLLKGAAFELCQLRFNTVFNAETGTWECGRLSYCLEDTAGGFQQLLLEPMLKFHYMLKKLQLHEEEYVLMQAISLFSPDRPGVLQHRVVDQLQEQFAITLKSYIECNRPQPAHRFLFLKIMAMLTELRSINAQHTQRLLRIQDIHPFATPLMQELFGITGS 1m18 A 2.45 BS01 dna I 0 R442 T445 R463 R472 R483 F484 Q485 R516 V517 T518 R5 T8 R26 R35 R46 F47 Q48 R79 V80 T81 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 1 ~ 146 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m18 A 2.45 BS02 dna J 0 R440 Y441 G444 V446 A447 R449 R463 K464 L465 P466 R469 R483 R3 Y4 G7 V9 A10 R12 R26 K27 L28 P29 R32 R46 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 147 ~ 292 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m18 B 2.45 BS01 dna I 0 P32 R36 R45 P9 R13 R22 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 1 ~ 146 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m18 B 2.45 BS02 dna J 0 R35 R45 I46 S47 R78 K79 T80 R12 R22 I23 S24 R55 K56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 147 ~ 292 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m18 C 2.45 BS01 dna I 0 R817 G828 R832 R877 R4 G15 R19 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 1 ~ 146 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKKT 1m18 C 2.45 BS02 dna J 0 R829 R835 R842 A845 K875 T876 R877 R16 R22 R29 A32 K62 T63 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 147 ~ 292 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKKT 1m18 D 2.45 BS01 dna I 0 T1229 R1230 S1252 S1253 S1284 T1285 T1 R2 S24 S25 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m18 D 2.45 BS02 dna J 0 R1230 K1231 E1232 S1233 I1236 Y1237 R2 K3 E4 S5 I8 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 147 ~ 292 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m18 E 2.45 BS01 dna I 0 H639 R640 Y641 P643 G644 V646 A647 R649 R663 K664 L665 P666 R669 R683 H3 R4 Y5 P7 G8 V10 A11 R13 R27 K28 L29 P30 R33 R47 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 1 ~ 146 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m18 E 2.45 BS02 dna J 0 R640 Y641 R642 P643 T645 R663 R672 R683 F684 Q685 R716 V717 T718 R4 Y5 R6 P7 T9 R27 R36 R47 F48 Q49 R80 V81 T82 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 147 ~ 292 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m18 F 2.45 BS01 dna I 0 R235 R245 I246 S247 G248 R278 K279 T280 R16 R26 I27 S28 G29 R59 K60 T61 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 1 ~ 146 KVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m18 F 2.45 BS02 dna J 0 T230 P232 R236 R245 T11 P13 R17 R26 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 147 ~ 292 KVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m18 G 2.45 BS01 dna I 0 R1029 R1035 R1042 G1044 A1045 K1075 T1076 R1077 R16 R22 R29 G31 A32 K62 T63 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 1 ~ 146 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKK 1m18 G 2.45 BS02 dna J 0 R1017 R1020 R1032 R1042 R1077 R4 R7 R19 R29 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 147 ~ 292 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKK 1m18 H 2.45 BS01 dna I 0 R1430 K1431 S1433 I1436 Y1437 R2 K3 S5 I8 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m18 H 2.45 BS02 dna J 0 T1429 R1430 S1452 S1453 R1483 S1484 T1485 T1 R2 S24 S25 R55 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 147 ~ 292 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m19 A 2.3 BS01 dna I 0 Y441 R442 T445 R463 R472 R483 F484 Q485 R516 V517 T518 Y6 R7 T10 R28 R37 R48 F49 Q50 R81 V82 T83 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 1 ~ 146 KKPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m19 A 2.3 BS02 dna J 0 K436 R440 Y441 P443 G444 V446 A447 R449 R463 K464 L465 R469 R483 K1 R5 Y6 P8 G9 V11 A12 R14 R28 K29 L30 R34 R48 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 147 ~ 292 KKPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m19 B 2.3 BS01 dna I 0 T30 P32 R36 R45 T7 P9 R13 R22 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 1 ~ 146 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m19 B 2.3 BS02 dna J 0 R45 I46 S47 G48 R78 K79 T80 R22 I23 S24 G25 R55 K56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 147 ~ 292 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m19 C 2.3 BS01 dna I 0 R817 G828 R832 R842 R877 R4 G15 R19 R29 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 1 ~ 146 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKKT 1m19 C 2.3 BS02 dna J 0 R829 R842 V843 G844 T876 R877 R16 R29 V30 G31 T63 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 147 ~ 292 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKKT 1m19 D 2.3 BS01 dna I 0 Y1239 S1252 S1253 R1283 S1284 T1285 K1322 Y11 S24 S25 R55 S56 T57 K94 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m19 D 2.3 BS02 dna J 0 R1230 K1231 E1232 S1233 I1236 Y1237 R2 K3 E4 S5 I8 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 147 ~ 292 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m19 E 2.3 BS01 dna I 0 R640 Y641 P643 G644 V646 A647 R649 R663 K664 L665 P666 R669 R683 R3 Y4 P6 G7 V9 A10 R12 R26 K27 L28 P29 R32 R46 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 1 ~ 146 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m19 E 2.3 BS02 dna J 0 Y641 R642 T645 R672 R683 F684 Q685 R716 V717 T718 Y4 R5 T8 R35 R46 F47 Q48 R79 V80 T81 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 147 ~ 292 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m19 F 2.3 BS01 dna I 0 R235 R245 I246 S247 G248 R278 K279 T280 R19 R29 I30 S31 G32 R62 K63 T64 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 1 ~ 146 RHRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m19 F 2.3 BS02 dna J 0 R219 P232 R236 R245 R3 P16 R20 R29 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 147 ~ 292 RHRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m19 G 2.3 BS01 dna I 0 R1029 R1042 V1043 G1044 A1045 K1075 T1076 R1077 R15 R28 V29 G30 A31 K61 T62 R63 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 1 ~ 146 KTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKK 1m19 G 2.3 BS02 dna J 0 R1017 R1032 R1042 R1077 R3 R18 R28 R63 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 147 ~ 292 KTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKK 1m19 H 2.3 BS01 dna I 0 R1430 K1431 S1433 Y1437 R2 K3 S5 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m19 H 2.3 BS02 dna J 0 R1430 G1450 I1451 S1452 S1453 R1483 S1484 T1485 R2 G22 I23 S24 S25 R55 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 147 ~ 292 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSAK 1m1a A 2.65 BS01 dna I 0 R440 Y441 R442 P443 T445 R463 R472 R483 F484 Q485 R516 V517 T518 R4 Y5 R6 P7 T9 R27 R36 R47 F48 Q49 R80 V81 T82 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 1 ~ 146 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m1a A 2.65 BS02 dna J 0 H439 R440 Y441 G444 T445 V446 A447 R449 R463 K464 L465 R469 R483 H3 R4 Y5 G8 T9 V10 A11 R13 R27 K28 L29 R33 R47 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 147 ~ 292 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m1a B 2.65 BS01 dna I 0 R23 T30 P32 R36 R45 R1 T8 P10 R14 R23 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 1 ~ 146 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m1a B 2.65 BS02 dna J 0 R45 I46 S47 G48 R78 K79 T80 R23 I24 S25 G26 R56 K57 T58 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 147 ~ 292 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m1a C 2.65 BS01 dna I 0 R817 R820 R829 R832 R842 R877 R4 R7 R16 R19 R29 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 1 ~ 146 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPK 1m1a C 2.65 BS02 dna J 0 R829 R835 R842 G844 T876 R877 R16 R22 R29 G31 T63 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 147 ~ 292 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPK 1m1a D 2.65 BS01 dna I 0 T1229 R1230 S1252 S1253 R1283 S1284 T1285 T1 R2 S24 S25 R55 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 1m1a D 2.65 BS02 dna J 0 R1230 K1231 E1232 S1233 I1236 Y1237 R2 K3 E4 S5 I8 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 147 ~ 292 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 1m1a E 2.65 BS01 dna I 0 R640 Y641 P643 G644 T645 V646 A647 R649 K656 R663 K664 L665 R669 R3 Y4 P6 G7 T8 V9 A10 R12 K19 R26 K27 L28 R32 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 1 ~ 146 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m1a E 2.65 BS02 dna J 0 H639 R640 R642 P643 R672 R683 F684 Q685 R716 V717 T718 H2 R3 R5 P6 R35 R46 F47 Q48 R79 V80 T81 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02302 12559907 147 ~ 292 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 1m1a F 2.65 BS01 dna I 0 R245 I246 S247 G248 R278 K279 T280 R36 I37 S38 G39 R69 K70 T71 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 1 ~ 146 LGKGGAKRHRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m1a F 2.65 BS02 dna J 0 R219 P232 R236 R245 R10 P23 R27 R36 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 12559907 147 ~ 292 LGKGGAKRHRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 1m1a G 2.65 BS01 dna I 0 R1029 R1035 R1042 G1044 A1045 K1075 T1076 R1077 R16 R22 R29 G31 A32 K62 T63 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 1 ~ 146 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKK 1m1a G 2.65 BS02 dna J 0 A1014 K1015 R1017 R1020 R1029 R1032 R1042 R1077 A1 K2 R4 R7 R16 R19 R29 R64 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 12559907 147 ~ 292 AKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPKK 1m1a H 2.65 BS01 dna I 0 R1430 K1431 S1433 I1436 Y1437 R2 K3 S5 I8 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 1m1a H 2.65 BS02 dna J 0 Y1439 S1453 R1483 S1484 T1485 Y11 S25 R55 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 12559907 147 ~ 292 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 1m1b A 2.25 BS02 SPV A 1 S46 G47 L48 D85 N122 S123 L124 R159 S42 G43 L44 D81 N118 S119 L120 R155 W44 S46 G47 L48 D58 D85 D87 C112 E114 K120 N122 S123 R159 H190 V215 W40 S42 G43 L44 D54 D81 D83 C108 E110 K116 N118 S119 R155 H186 V211 5.4.2.9 0003824,0016853,0032923,0046872,0050188 Ki=22uM remove_due_to_license_issue P56839 12162742 996 VKKTTQLKQMLNSKDLEFIMEAHNGLSARIVQEAGFKGIWGSGLSVSAQLGVRDSNEASWTQVVEVLEFMSDASDVPILLDADTGYGNFNNARRLVRKLEDRGVAGACLEDKLFPKTNSLHDGRAQPLADIEEFALKIKACKDSQTDPDFCIVARVEAFIAGWGLDEALKRAEAYRNAGADAILMHSKKADPSDIEAFMKAWNNQGPVVIVPTKYYKTPTDHFRDMGVSMVIWANHNLRASVSAIQQTTKQIYDDQSLVNVEDKIVSVKEIFRLQRDDELVQAEDKYLPKN 1m2p A 2.0 BS01 HNA A 1 V45 G46 R47 V53 K68 V95 F113 I174 D175 V39 G40 R41 V47 K62 V89 F107 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue Ki=780nM P28523 12419810 351 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 1m2q A 1.79 BS01 MNX A 1 R47 G48 V53 I66 K68 F113 V116 M163 I174 D175 R41 G42 V47 I60 K62 F107 V110 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue Ki=800nM P28523 12419810 351 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 1m2r A 1.7 BS01 MNY A 1 V45 V53 I66 F113 V116 N118 M163 I174 V39 V47 I60 F107 V110 N112 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue Ki=350nM P28523 12419810 351 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 1m2x A 1.5 BS04 MCO A 1 H118 D119 D120 K167 H196 Y233 H74 D75 D76 K106 H135 Y166 H116 H118 D120 H196 C221 K224 Y233 H263 H72 H74 D76 H135 C154 K157 Y166 H196 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki~85uM remove_due_to_license_issue O08498 12684522 811 DVKIEKLKDNLYVYTTYNTFNGTKYAANAVYLVTDKGVVVIDCPWGEDKFKSFTDEIYKKHGKKVIMNIATHSHDDRAGGLEYFGKIGAKTYSTKMTDSILAKENKPRAQYTFDNNKSFKVGKSEFQVYYPGKGHTADNVVVWFPKEKVLVGGCIIKSADSKDLGYIGEAYVNDWTQSVHNIQQKFSGAQYVVAGHDDWKDQRSIQHTLDLINEYQQKQ 1m48 A 1.95 BS01 FRG A 1 K35 R38 M39 T41 F42 K43 Y45 E62 P65 L72 A73 K32 R35 M36 T38 F39 K40 Y42 E59 P62 L69 A70 ? 0002250,0002366,0002639,0002903,0005125,0005134,0005515,0005576,0005615,0006366,0006955,0007155,0007186,0007204,0007267,0008083,0008284,0010467,0019209,0030101,0030217,0030246,0030307,0030890,0031851,0032729,0032740,0034105,0038110,0042098,0042102,0042104,0043066,0043208,0045471,0045582,0045591,0045944,0046013,0046651,0048304,0050672,0050728,0050729,0050798,0060999,0097192,0097696,1900100,1901327,2000320,2000561 Kd=8.2uM remove_due_to_license_issue P60568 12582206 301 SSSTKKTQLQLEHLLLDLQMILNGINNYKNPKLTRMLTFKFYMPKKATELKHLQCLEEELKPLEEVLNLAQRPRDLISNINVIVLELKGSETTFMCEYADETATIVEFLNRWITFCQSIISTL 1m51 A 2.25 BS02 TSX A 1 N292 L293 W516 F517 F525 P528 F530 N533 N281 L282 W497 F498 F506 P509 F511 N514 R87 Y235 K244 H264 S286 C288 D311 R405 R78 Y224 K233 H253 S275 C277 D300 R394 2.7.11.-,4.1.1.32 0000287,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0016301,0016831,0017076,0018105,0019543,0030145,0031406,0032868,0032869,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070062,0070365,0071333,0071549,0072350,0106264 ic50=18.8uM remove_due_to_license_issue P35558 14552798 1001 NLSAKVVQGSLDSLPQAVREFLENNAELCQPDHIHICDGSEEENGRLLGQMEEEGILRRLKKYDNCWLALTDPRDVARIESKTVIVTQEQRDTVPIPKTGLSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSSKIGIELTDSPYVVASMRIMTRMGTPVLEALGDGEFVKCLHSVGCPLPLQKPLVNNWPCNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRMASRLAKEEGWLAEHMLVLGITNPEGEKKYLAAAFPSACGKTNLAMMNPSLPGWKVECVGDDIAWMKFDAQGHLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLASGVTITSWKNKEWSSEDGEPCAHPNSRFCTPASQCPIIDAAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEAKIIMHDPFAMRPFFGYNFGKYLAHWLSMAQHPAAKLPKIFHVNWFRKDKEGKFLWPGFGENSRVLEWMFNRIDGKASTKLTPIGYIPKEDALNLKGLGHINMMELFSISKEFWDKEVEDIEKYLVDQVNADLPCEIEREILALKQRISQM 1m5c A 1.65 BS01 BRH A 1 E13 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 E10 Y58 L87 T88 R93 L135 G138 S139 T140 L189 E190 ? 0015276,0016020 ic50=0.5uM remove_due_to_license_issue P19491 12215417 611 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1m5d A 1.73 BS01 BRH A 1 E13 Y61 T91 R96 L138 G141 S142 T143 L192 E193 E10 Y58 T88 R93 L135 G138 S139 T140 L189 E190 ? 0015276,0016020 ic50=9.2uM remove_due_to_license_issue P19491 12215417 611 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1m5w A 1.96 BS01 DXP A 1 D11 H12 R47 E72 T102 T103 H193 D10 H11 R46 E71 T101 T102 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM remove_due_to_license_issue P0A794 12269807 1001 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w E 1.96 BS01 DXP E 1 D11 H52 K97 H193 G215 H216 D10 H51 K96 H192 G214 H215 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM remove_due_to_license_issue P0A794 12269807 1005 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m6p A 1.8 BS02 M6P A 1 Y45 Q66 D103 N104 H105 R111 E133 R135 Y143 Y37 Q58 D95 N96 H97 R103 E125 R127 Y135 ? 0005768,0005794,0006622,0019904 Kd=8uM remove_due_to_license_issue P11456 9604938 200 EKTCDLVGEKGKESEKELALLKRLTPLFQKSFESTMYSYVFRVCREAGQHSSGAGLVQIQKSNGKETVVGRFNETQIFQGSNWIMLIYKGGDEYDNHCGREQRRAVVMISCNRHTLADNFNPVSEERGKVQDCFYLFEMDSSLACS 1m74 A 3.0 BS01 ADP A 1 M79 F80 P81 F82 Q85 G103 G105 K106 T107 L108 D492 M79 F80 P81 F82 Q85 G103 G105 K106 T107 L108 D492 7.4.2.8 0005524,0005737,0005886,0006605,0006886,0008564,0015031,0016020,0017038,0031522,0043952,0045121,0046872,0065002 remove_due_to_license_issue P28366 12242434 901 MLGILNKMFDPTKRTLNRYEKIANDIDAIRGDYENLSDDALKHKTIEFKERLEKGATTDDLLVEAFAVVREASRRVTGMFPFKVQLMGGVALHDGNIAEMKTGEGKTLTSTLPVYLNALTGKGVHVVTVNEYLASRDAEQMGKIFEFLGLTVGLNLNSMSKDEKREAYAADITYSTNNELGFDYLRDNMVLYKEQMVQRPLHFAVIDEVDSILIDEARTPLIISGQAAKSTKLYVQANAFVRTLKAEKDYTYDIKTKAVQLTEEGMTKAEKAFGIDNLFDVKHVALNHHINQALKAHVAMQKDVDYVVEDGQVVIVDSFTGRLMKGRRYSEGLHQAIEAKEGLEIQNESMTLATITFQNYFRMYEKLAGMTGTAKTEEEEFRNIYNMQVVTIPTNRPVVRDDRPDLIYRTMEGKFKAVAEDVAQRYMTGQPVLVGTVAVETSELISKLLKNKGIPHQVLNAKNHEREAQIIEEAGQKGAVTIATNMAGRGTDIKLGEGVKELGGLAVVGTERHESRRIDNQLRGRSGRQGDPGITQFYLSMEDELMRRFGAERTMAMLDRFGMDDSTPIQSKMVSRAVESSQKRVEGNNFDSRKQLLQYDDVLRQQREVIYKQRFEVIDSENLREIVENMIKSSLERAIAAYTPREELPEEWKLDGLVDLINTTYLDEGALEKSDIFGKEPDEMLELIMDRIITKYNEKEEQFGKEQMREFEKVIVLRAVDSKWMDHIDAMDQLRQGIHLRAYAQTNPLREYQMEGFAMFEHMIESIEDEVAKFVMKAEIENNLEREEVVQGQTTAHQPQEG 1m7d A 2.3 BS01 MAG C 1 H27D Y32 T91 T92 H93 P95 H31 Y37 T96 T97 H98 P100 ? 0046872 remove_due_to_license_issue A2NHM3 12427018 1 DVVLTQTPLSLPVRLGDQASISCRSSQSLLHSDGNTYLHWYLQKPGQSPKLLIYKVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYFCSQTTHVPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 1m7d B 2.3 BS01 RAE C 1 G95 G99 G101 G105 ? 0002250,0003823,0005576,0016064,0019814 remove_due_to_license_issue P01801 12427018 2 EVKVEESGGGLVQPGGSMKLSCVASGFTFSNYWMEWVRQSPEKGLEWVAEIRLKSNNYATHYAESVKGRFTISRDDSKSSVYLQMNNLRAEDTGIYYCTRGGAVGAMDYWGQGTSVTVSSATTTAPSVYPLVPGCSDTSGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKVDLIKEPSGP 1m7i B 2.5 BS01 RAM C 1 W33 G95 W33 G101 ? 0002250,0003823,0005576,0016064,0019814 remove_due_to_license_issue P01801 12427018 5 EVKVEESGGGLVQPGGSMKLSCVASGFTFSNYWMEWVRQSPEKGLEWVAEIRLKSNNYATHYAESVKGRFTISRDDSKSSVYLQMNNLRAEDTGIYYCTRGGAVGAMDYWGQGTSVTVSSATTTAPSVYPLVPGCSDTSGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKVDLIKEPSGP 1m7q A 2.4 BS01 DQO A 1 Y35 A51 K53 T106 H107 L108 M109 G110 A111 A157 L167 D168 Y32 A48 K50 T103 H104 L105 M106 G107 A108 A154 L164 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=2.6nM remove_due_to_license_issue IC50=2.6nM Q16539 12482439 501 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 1m7y A 1.6 BS01 PPG A 1 Y19 W23 L45 A46 E47 G119 A120 T121 Y145 N202 D230 I232 Y233 S270 S272 K273 R281 R407 Y10 W14 L36 A37 E38 G110 A111 T112 Y136 N193 D221 I223 Y224 S261 S263 K264 R272 R398 Y145 D230 I232 K273 Y136 D221 I223 K264 1.4.-.-,4.4.1.14 0003824,0006520,0008483,0009058,0009693,0009835,0016491,0016829,0016847,0030170,0042218 remove_due_to_license_issue P37821 12228256 600 MLSRNATSSYFLGWQEYEKNPYHEVHNTNGIIQMGLAENQLCFDLLESWLAKNPEAAAFKKNGESIFAELALFQDYHGLPAFKKAMVDFMAEIRGNKVTFDPNHLVLTAGATSANETFIFCLADPGEAVLIPTPYYPGFDRDLKWRTGVEIVPIHCTSSNGFQITETALEEAYQEAEKRNLRVKGVLVTNPSNPLGTTMTRNELYLLLSFVEDKGIHLISDEIYSGTAFSSPSFISVMEVLKDRNCDENSEVWQRVHVVYSLSKDLGLPGFRVGAIYSNDDMVVAAATKMSSFGLVSSQTQHLLSAMLSDKKLTKNYIAENHKRLKQRQKKLVSGLQKSGISCLNGNAGLFCWVDMRHLLRSNTFEAEMELWKKIVYEVHLNISPGSSCHCTEPGWFRVCFANLPERTLDLAMQRLKAFVGEYY 1m83 A 2.2 BS01 ATP A 1 Q9 S11 G17 N18 G21 V143 G144 D146 A181 R182 I183 K192 M193 S194 K195 S196 Q9 S11 G17 N18 G21 V143 G144 D146 A181 R182 I183 K192 M193 S194 K195 S196 K111 K192 K195 K111 K192 K195 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0005829,0006412,0006418,0006436 Kd=0.4mM remove_due_to_license_issue P00953 12473451 400 MKTIFSGIQPSGVITIGNYIGALRQFVELQHEYNCYFCIVDQHAITVWQDPHELRQNIRRLAALYLAVGIDPTQATLFIQSEVPAHAQAAWMLQCIVYIGELERMTQFKEKSAGKEAVSAGLLTYPPLMAADILLYNTDIVPVGEDQKQHIELTRDLAERFNKRYGELFTIPEARIPKVGARIMSLVDPTKKMSKSDPNPKAYITLLDDAKTIEKKIKSAVTDSEGTIRYDKEAKPGISNLLNIYSTLSGQSIEELERQYEGKGYGVFKADLAQVVIETLRPIQERYHHWMESEELDRVLDEGAEKANRVASEMVRKMEQAMGLGRRR 1m8w A 2.2 BS01 rna C 0 N899 Y900 R936 Q939 H972 Q975 C1007 R1008 Q1011 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 Q1126 Y1156 H1159 N72 Y73 R109 Q112 H145 Q148 C180 R181 Q184 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 Q299 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 12 ~ 19 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 1m8w A 2.2 BS02 rna E 0 Y900 Q903 R936 Q939 H972 R1008 Y1041 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 Q1126 Y1156 H1159 Y73 Q76 R109 Q112 H145 R181 Y214 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 Q299 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 2 ~ 9 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 1m8w B 2.2 BS01 rna D 0 N899 Y900 Q903 Y933 R936 Q939 H972 C1007 R1008 Q1011 Y1041 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 Y1156 H1159 N72 Y73 Q76 Y106 R109 Q112 H145 C180 R181 Q184 Y214 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 13 ~ 19 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 1m8w B 2.2 BS02 rna F 0 Y900 R936 Q939 H972 R1008 Y1041 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 Y1156 H1159 Y73 R109 Q112 H145 R181 Y214 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 3 ~ 9 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 1m8x A 2.2 BS01 rna C 0 N899 Y900 R936 Q939 H972 C1007 R1008 Q1011 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 N1122 Y1123 Q1126 Y1156 H1159 N72 Y73 R109 Q112 H145 C180 R181 Q184 N216 Y217 Q220 F250 S252 N253 E256 N295 Y296 Q299 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 12 ~ 19 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 1m8x B 2.2 BS01 rna D 0 N899 Y900 Q903 Y933 R936 Q939 H972 Q975 C1007 R1008 Q1011 Y1041 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 Y1156 H1159 N72 Y73 Q76 Y106 R109 Q112 H145 Q148 C180 R181 Q184 Y214 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 13 ~ 19 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 1m8y A 2.6 BS01 rna C 0 Q860 R864 Q867 F897 N899 Y900 Y933 R936 Q939 H972 C1007 R1008 Q1011 N1043 Y1044 F1077 N1080 E1083 N1122 Y1123 Y1156 H1159 Q33 R37 Q40 F70 N72 Y73 Y106 R109 Q112 H145 C180 R181 Q184 N216 Y217 F250 N253 E256 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 11 ~ 20 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 1m8y B 2.6 BS01 rna D 0 Q860 R864 Q867 F897 N899 Y900 Y933 R936 Q939 H972 R1008 Q1011 N1043 Y1044 Q1047 K1076 F1077 N1080 E1083 Y1120 N1122 Y1123 H1159 Q33 R37 Q40 F70 N72 Y73 Y106 R109 Q112 H145 R181 Q184 N216 Y217 Q220 K249 F250 N253 E256 Y293 N295 Y296 H332 ? 0003723 remove_due_to_license_issue Q14671 12202039 11 ~ 20 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYYM 1m9n A 1.93 BS02 XMP A 1 S11 V12 S13 S35 G37 T38 G64 R65 K67 T68 C102 N103 L104 Y105 D126 G128 G129 S8 V9 S10 S32 G34 T35 G61 R62 K64 T65 C99 N100 L101 Y102 D123 G125 G126 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.12uM remove_due_to_license_issue P31335 12501179 1003 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1m9n B 1.93 BS03 XMP B 1 S11 V12 S13 S35 G37 T38 R65 K67 T68 N103 L104 Y105 D126 G128 G129 S8 V9 S10 S32 G34 T35 R62 K64 T65 N100 L101 Y102 D123 G125 G126 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.12uM remove_due_to_license_issue P31335 12501179 1004 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1ma7 A 2.3 BS01 dna C 0 F37 S38 H40 T41 R173 I174 A175 K244 E262 R282 Y283 S287 G288 H289 F19 S20 H22 T23 R155 I156 A157 K226 E244 R264 Y265 S269 G270 H271 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 12779336 1 ~ 34 TSDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 1ma7 A 2.3 BS02 dna D 0 M44 S47 R50 R81 L83 A84 K86 T87 Q90 A131 R159 T202 R241 V242 K244 S257 R259 A260 R282 W315 I320 Y324 M26 S29 R32 R63 L65 A66 K68 T69 Q72 A113 R141 T184 R223 V224 K226 S239 R241 A242 R264 W297 I302 Y306 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 12779336 1 ~ 34 TSDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 1ma7 B 2.3 BS01 dna C 0 K43 M44 S47 R50 R81 L83 A84 K86 T87 Q90 R118 A131 K132 Q156 R159 R173 K201 T202 R241 V242 K244 L256 S257 R259 R282 W315 T316 N317 I320 Y324 K24 M25 S28 R31 R62 L64 A65 K67 T68 Q71 R99 A112 K113 Q137 R140 R154 K182 T183 R222 V223 K225 L237 S238 R240 R263 W296 T297 N298 I301 Y305 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 12779336 1 ~ 34 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNGAMVRLLED 1ma7 B 2.3 BS02 dna D 0 F37 S38 H40 T41 M97 R100 R101 R106 R121 R173 I174 A175 K201 R243 K244 N245 R259 E262 R282 Y283 S287 G288 H289 F18 S19 H21 T22 M78 R81 R82 R87 R102 R154 I155 A156 K182 R224 K225 N226 R240 E243 R263 Y264 S268 G269 H270 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 12779336 1 ~ 34 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNGAMVRLLED 1mai A 1.9 BS01 I3P A 1 K30 K32 W36 R40 S55 R56 K57 K19 K21 W25 R29 S44 R45 K46 3.1.4.11 0035556 Kd=210nM remove_due_to_license_issue P10688 8521504 200 GLQDDPDLQALLKGSQLLKVKSSSWRRERFYKLQEDCKTIWQESRKVMRSPESQLFSIEDIQEVRMGHRTEGLEKFARDIPEDRCFSIVFKDQRNTLDLIAPSPADAQHWVQGLRKIIH 1mau A 2.15 BS01 ATP A 1 I8 Q9 S11 G17 N18 G21 V143 G144 D146 A181 R182 I183 K192 M193 S194 K195 S196 I8 Q9 S11 G17 N18 G21 V143 G144 D146 A181 R182 I183 K192 M193 S194 K195 S196 K111 K192 K195 K111 K192 K195 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0005829,0006412,0006418,0006436 remove_due_to_license_issue P00953 12473451 400 MKTIFSGIQPSGVITIGNYIGALRQFVELQHEYNCYFCIVDQHAITVWQDPHELRQNIRRLAALYLAVGIDPTQATLFIQSEVPAHAQAAWMLQCIVYIGELERMTQFKEKSAGKEAVSAGLLTYPPLMAADILLYNTDIVPVGEDQKQHIELTRDLAERFNKRYGELFTIPEARIPKVGARIMSLVDPTKKMSKSDPNPKAYITLLDDAKTIEKKIKSAVTDSEGTIRYDKEAKPGISNLLNIYSTLSGQSIEELERQYEGKGYGVFKADLAQVVIETLRPIQERYHHWMESEELDRVLDEGAEKANRVASEMVRKMEQAMGLGRRR 1maw A 3.0 BS01 ATP A 1 G17 N18 I183 K192 M193 S194 K195 S196 G17 N18 I183 K192 M193 S194 K195 S196 K111 K192 K195 K111 K192 K195 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0005829,0006412,0006418,0006436 remove_due_to_license_issue P00953 12473451 400 MKTIFSGIQPSGVITIGNYIGALRQFVELQHEYNCYFCIVDQHAITVWQDPHELRQNIRRLAALYLAVGIDPTQATLFIQSEVPAHAQAAWMLQCIVYIGELERMTQFKEKSAGKEAVSAGLLTYPPLMAADILLYNTDIVPVGEDQKQHIELTRDLAERFNKRYGELFTIPEARIPKVGARIMSLVDPTKKMSKSDPNPKAYITLLDDAKTIEKKIKSAVTDSEGTIRYDKEAKPGISNLLNIYSTLSGQSIEELERQYEGKGYGVFKADLAQVVIETLRPIQERYHHWMESEELDRVLDEGAEKANRVASEMVRKMEQAMGLGR 1mcz A 2.8 BS04 RMN A 1 H281 T377 F464 H280 T376 F463 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 S525 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 S524 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 12590569 534 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTVS 1mcz A 2.8 BS06 RMN B 1 S26 H70 L110 S25 H69 L109 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 S525 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 S524 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 12590569 534 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTVS 1mcz B 2.8 BS03 RMN A 1 G25 S26 H70 L110 G24 S25 H69 L109 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 S525 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 S524 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 12590569 534 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTVS 1mcz B 2.8 BS06 RMN B 1 H281 T377 H280 T376 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 S525 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 S524 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 12590569 534 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTVS 1mdl A 1.85 BS02 RMN A 1 V22 F52 R166 V20 F50 R164 V22 S139 K164 R166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 R164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 remove_due_to_license_issue Ki=810000nM P11444 7893690 398 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTRIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 1mdm A 2.8 BS01 dna C 0 N29 G30 C52 R56 H62 S66 G84 G85 S86 P88 K89 V90 A91 S131 S133 S134 R137 N11 G12 C34 R38 H44 S48 G66 G67 S68 P70 K71 V72 A73 S113 S115 S116 R119 ? 0003677,0006355 remove_due_to_license_issue Q02548 12221090 1 ~ 26 GVNQLGGVFVNGRPLPDVVRQRIVELAHQGVRPCDISRQLRVSHGCVSKILGRYYETGSIKPGVIGGSKPKVATPKVVEKIAEYKRQNPTMFAWEIRDRLLAERVCDNDTVPSVSSINRIIRTK 1mdm A 2.8 BS02 dna D 0 N21 Q22 F27 G30 P32 L33 S61 C64 K67 P80 G81 V82 I83 G84 G85 F110 A111 N3 Q4 F9 G12 P14 L15 S43 C46 K49 P62 G63 V64 I65 G66 G67 F92 A93 ? 0003677,0006355 remove_due_to_license_issue Q02548 12221090 1 ~ 26 GVNQLGGVFVNGRPLPDVVRQRIVELAHQGVRPCDISRQLRVSHGCVSKILGRYYETGSIKPGVIGGSKPKVATPKVVEKIAEYKRQNPTMFAWEIRDRLLAERVCDNDTVPSVSSINRIIRTK 1mdm B 2.8 BS01 dna C 0 R391 R394 Y397 K404 R409 R83 R86 Y89 K96 R101 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P27577 12221090 1 ~ 26 RDRADLNKDKPVIPAAALAGYTGSGPIQLWQFLLELLTDKSCQSFISWTGDGWEFKLSDPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTAGKRYVYRFVCDLQSLLGYTPEELHAMLDVKP 1mdm B 2.8 BS02 dna D 0 Q336 L337 W375 K379 M384 K388 R391 Y396 Q28 L29 W67 K71 M76 K80 R83 Y88 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P27577 12221090 1 ~ 26 RDRADLNKDKPVIPAAALAGYTGSGPIQLWQFLLELLTDKSCQSFISWTGDGWEFKLSDPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTAGKRYVYRFVCDLQSLLGYTPEELHAMLDVKP 1me3 A 1.2 BS01 P10 A 1 G23 C25 S61 S64 G65 G66 L67 A133 D158 H159 G23 C25 S61 S64 G65 G66 L67 A138 D161 H162 Q19 C25 H159 N175 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 12467703 300 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 1me4 A 1.2 BS01 T10 A 1 Q19 G23 C25 S61 G65 G66 A133 D158 H159 Q19 G23 C25 S61 G65 G66 A138 D161 H162 Q19 C25 H159 N175 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 12467703 300 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 1me7 A 2.15 BS01 RVP A 1 M59 G316 S317 I318 C319 D358 G381 R382 Y405 G407 E408 G409 M58 G203 S204 I205 C206 D245 G268 R269 Y292 G294 E295 G296 1.1.1.205 0000166,0003824,0003938,0005737,0006164,0006177,0006183,0016491,0032991,0042802,0046872 Ki=65nM remove_due_to_license_issue P50097 12235158 602 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFKAGFVVSDVCHNELVDSQKRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIREKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICITREQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWEGVDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVEGGAHDVI 1me8 A 1.9 BS01 RVP A 1 M59 G316 S317 I318 C319 D358 L380 G381 R382 Y405 G407 E408 G409 M58 G195 S196 I197 C198 D237 L259 G260 R261 Y284 G286 E287 G288 1.1.1.205 0000166,0003824,0003938,0005737,0006164,0006177,0006183,0016491,0032991,0042802,0046872 Ki=65nM remove_due_to_license_issue P50097 12235158 602 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFKAHNELVDSQKRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIREKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICITREQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWEGVDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVEGGAHDVI 1mem A 1.8 BS01 0D6 A 1 Q19 G23 C25 D61 G64 G65 G66 Y67 L157 N158 H159 W177 Q19 G23 C25 D61 G64 G65 G66 Y67 L160 N161 H162 W184 Q19 C25 H159 N175 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 9033587 280 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1mes A 1.9 BS01 DMP B 1 D25 G27 D30 G49 I50 P81 V82 D25 G27 D30 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9048541 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 1mes B 1.9 BS01 DMP B 1 D25 G27 A28 D30 I50 V82 D25 G27 A28 D30 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P03366 9048541 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 1met A 1.9 BS01 DMP A 1 D25 G27 D30 G49 I50 P81 F82 D25 G27 D30 G49 I50 P81 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.4nM remove_due_to_license_issue P03366 9048541 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNIIGRNLLTQIGCTLNF 1met B 1.9 BS01 DMP A 1 D25 G27 A28 D30 V32 G49 I50 P81 F82 D25 G27 A28 D30 V32 G49 I50 P81 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9048541 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNIIGRNLLTQIGCTLNF 1meu A 1.9 BS01 DMP A 1 L23 D25 G27 D30 V32 G49 I50 P81 F82 L23 D25 G27 D30 V32 G49 I50 P81 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.8uM remove_due_to_license_issue P03366 9048541 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1meu B 1.9 BS01 DMP A 1 D25 G27 A28 D30 G48 I50 D25 G27 A28 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9048541 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1mfa L 1.7 BS01 ABE A 1 W93 W98 W93 W98 remove_due_to_license_issue 7517550 3 QIVVTQESALTTSPGETVTLTCRSSTGTVTSGNHANWVQEKPDHLFTGLIGDTNNRAPGVPARFSGSLIGDKAALTITGAQPEDEAIYFCALWSNNHWIFGGGTKLTVLGQG 1mfd H 2.1 BS01 MMA A 1 W283 H351 W33 H101 remove_due_to_license_issue 8172893 1 EVQVQQSGTVLARPGASVKMSCKASGYTFTNYWMHWIKQRPGQGLEWIGAIYPGNSATFYNHKFRAKTKLTAVTSTITAYMELSSLTNEDSAVYYCTRGGHGYYGDYWGQGASLTVSSAKTTPPSVYPLAPGMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 1mfd H 2.1 BS02 ABE A 1 W283 H285 G350 G352 W33 H35 G100 G102 remove_due_to_license_issue 8172893 3 EVQVQQSGTVLARPGASVKMSCKASGYTFTNYWMHWIKQRPGQGLEWIGAIYPGNSATFYNHKFRAKTKLTAVTSTITAYMELSSLTNEDSAVYYCTRGGHGYYGDYWGQGASLTVSSAKTTPPSVYPLAPGMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 1mfd L 2.1 BS01 ABE A 1 W93 W98 W93 W98 remove_due_to_license_issue 8172893 3 QAVVTQESALTTSPGETVTLTCRSSTGTVTSGNHANWVQEKPDHLFTGLIGDTNNRAPGVPARFSGSLIGDKAALTITGAQPEDEAIYFCALWCNNHWIFGGGTKLTVLGQPKSSPSVTLFPPSSEELETNKATLVCTITDFYPGVVTVDWKVDGTPVTQGMETTQPSKQSNNKYMASSYLTLTARAWERHSSYSCQVTHEGHTVEKSLSRA 1mfi A 1.8 BS01 FHC A 1 P1 M2 K32 Y36 H62 I64 V106 P1 M2 K32 Y36 H62 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0001934,0002020,0002821,0002906,0004167,0005125,0005126,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0032760,0033033,0042056,0042127,0042327,0042802,0043066,0043209,0043406,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070207,0070374,0090238,0090398,0141163,1902166,2000343,2000773 Ki=2.6uM remove_due_to_license_issue P34884 10360941 115 PMFIVNTNVPRASVPEGFLSELTQQLAQATGKPAQYIAVHVVPDQLMTFSGTNDPCALCSLHSIGKIGGAQNRNYSKLLCGLLSDRLHISPDRVYINYYDMNAANVGWNGSTFA 1mfi A 1.8 BS02 FHC B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0001934,0002020,0002821,0002906,0004167,0005125,0005126,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0032760,0033033,0042056,0042127,0042327,0042802,0043066,0043209,0043406,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070207,0070374,0090238,0090398,0141163,1902166,2000343,2000773 Ki=2.6uM remove_due_to_license_issue P34884 10360941 116 PMFIVNTNVPRASVPEGFLSELTQQLAQATGKPAQYIAVHVVPDQLMTFSGTNDPCALCSLHSIGKIGGAQNRNYSKLLCGLLSDRLHISPDRVYINYYDMNAANVGWNGSTFA 1mfi B 1.8 BS01 FHC B 1 P1 M2 K32 Y36 H62 S63 I64 V106 P1 M2 K32 Y36 H62 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0001934,0002020,0002821,0002906,0004167,0005125,0005126,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0032760,0033033,0042056,0042127,0042327,0042802,0043066,0043209,0043406,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070207,0070374,0090238,0090398,0141163,1902166,2000343,2000773 Ki=2.6uM remove_due_to_license_issue P34884 10360941 116 PMFIVNTNVPRASVPEGFLSELTQQLAQATGKPAQYIAVHVVPDQLMTFSGTNDPCALCSLHSIGKIGGAQNRNYSKLLCGLLSDRLHISPDRVYINYYDMNAANVGWNGSTFA 1mfi B 1.8 BS02 FHC C 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0001934,0002020,0002821,0002906,0004167,0005125,0005126,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0032760,0033033,0042056,0042127,0042327,0042802,0043066,0043209,0043406,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070207,0070374,0090238,0090398,0141163,1902166,2000343,2000773 Ki=2.6uM remove_due_to_license_issue P34884 10360941 117 PMFIVNTNVPRASVPEGFLSELTQQLAQATGKPAQYIAVHVVPDQLMTFSGTNDPCALCSLHSIGKIGGAQNRNYSKLLCGLLSDRLHISPDRVYINYYDMNAANVGWNGSTFA 1mh5 A 2.1 BS01 HAL B 1 H27D Y32 L89 H91 L92 Y94 F96 H31 Y37 L94 H96 L97 Y99 F101 ? 0005576,0005886,0030183 remove_due_to_license_issue P01837 12948492 601 DIVMTQAAPSVSVTPGESVSISCRSSKSLLHSNGNTYLYWFLQRPGQSPQLLIYRMSNLASGVPDRFSGSGSGTAFTLRISRVEAEDVGVYYCLQHLEYPFTFGAGTKLELKRADAAPTVSIFPPASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKRHNSYTCEATSPIVKSFN 1mh5 B 2.1 BS01 HAL B 1 W33 N35 K95 W32 N34 K98 ? Kd=0.61nM remove_due_to_license_issue P01863 12948492 601 VQLQQPGAELVKPGASVKLSCKASGYTFTSNWINWVKQRPGQGLEWIGNIYPDSYRTNYNEKFKRKATLTVDTSSSTAYMQLSSLTSDDSAVYYCVRKHYSYDGVVYWGQGTLVTVSAAKTTAPSVYPLAPVVTLGCLVKGYFPEPVTLTWVHTFPAVLQSDLYTLSSSVTV 1mhd A 2.8 BS01 dna C 0 S70 L71 Q76 K81 S61 L62 Q67 K72 ? 0005667,0006355 remove_due_to_license_issue P84022 9741623 1001 ~ 1013 PIVKRLLGWKKGEQNGQEEKWCEKAVKSLVKKLKKTGQLDELEKAITTQNVNTKCITIPRSLDGRLQVSHRKGLPHVIYCRLWRWPDLHSHHELRAMELCEFAFNMKKDEVCVNPYHYQRVET 1mhd A 2.8 BS02 dna D 0 R74 H100 R65 H91 ? 0005667,0006355 remove_due_to_license_issue P84022 9741623 2001 ~ 2014 PIVKRLLGWKKGEQNGQEEKWCEKAVKSLVKKLKKTGQLDELEKAITTQNVNTKCITIPRSLDGRLQVSHRKGLPHVIYCRLWRWPDLHSHHELRAMELCEFAFNMKKDEVCVNPYHYQRVET 1mhd B 2.8 BS01 dna C 0 R74 K81 R65 K72 ? 0005667,0006355 remove_due_to_license_issue P84022 9741623 1001 ~ 1013 PIVKRLLGWKKGEQNGQEEKWCEKAVKSLVKKLKKTGQLDELEKAITTQNVNTKCITIPRSLDGRLQVSHRKGLPHVIYCRLWRWPDLHSHHELRAMELCEFAFNMKKDEVCVNPYHYQRVET 1mhd B 2.8 BS02 dna D 0 S70 L71 Q76 K81 S61 L62 Q67 K72 ? 0005667,0006355 remove_due_to_license_issue P84022 9741623 2001 ~ 2014 PIVKRLLGWKKGEQNGQEEKWCEKAVKSLVKKLKKTGQLDELEKAITTQNVNTKCITIPRSLDGRLQVSHRKGLPHVIYCRLWRWPDLHSHHELRAMELCEFAFNMKKDEVCVNPYHYQRVET 1mj7 H 2.25 BS01 HAL H 1 W33 N35 V93 K95 W103 W22 N24 V83 K85 W90 Kd=4.5nM remove_due_to_license_issue 12948492 301 LQQPGAELVKPGASVKLSCSSWINWVKQRPGQGLEWIGNVYPSTNYNEKFKNKATLTVDTSSSTAYMQLSSLTSDDSAFYYCVRKDFPYWGQGTLVTVSAAKTTAPSVYPLAPSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEPR 1mj7 L 2.25 BS01 HAL H 1 Y32 M89 H91 L92 Y94 F96 Y37 M94 H96 L97 Y99 F101 remove_due_to_license_issue 12948492 301 EIVMTQAAPSVPVTPGESVSISCRSSKSLLHSNGNTYLNWFLQRPGQSPQLLIYRMSNLASGVPDRFSGSGSETAFTLRTSRVEAEDVGVYYCMQHLEYPFTFGSGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1mjj A 2.1 BS01 HAL A 1 Y32 L89 H91 L92 Y94 F96 Y37 L94 H96 L97 Y99 F101 Kd=1.83nM remove_due_to_license_issue 12948492 1001 DIVMTQAAPSVPVTPGESVSISCRSSKSLLHSNGNTYLYWFLQRPGQSPQLLIYRMSNLASGVPDRFSGSGSGTAFTLRISRVEAEDVGVYYCLQHLEYPFTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1mjj B 2.1 BS01 HAL A 1 W33 N35 N50 K95 W33 N35 N50 K99 remove_due_to_license_issue 12948492 1001 QVQLQQPGAELVKPGASVKLSCKASGYTFTNYWINWVKQRPGQGLEWIGNIYPGSSYTHYNEKFKNKATLTVDTSSSTAYMQLSSLTSDDSAVYYCANKLGWFPYWGQGTLVTVSAAKTTAPSVYPLAPVCSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEPR 1mkd A 2.9 BS02 ZAR A 1 M370 Y426 W429 T430 M454 Q466 F469 M188 Y244 W247 T248 M272 Q284 F287 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=390nM Q08499 12387865 3001 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFPQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQS 1ml1 A 2.6 BS01 PGA A 1 N11 K13 H95 E167 I172 G173 S213 G234 G235 N10 K12 H86 E158 I163 G164 S204 G225 G226 N11 K13 H95 E97 E167 G173 S213 N10 K12 H86 E88 E158 G164 S204 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 remove_due_to_license_issue P04789 9089815 600 SKPQPIAAANWKSGSPDSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAGNADALASLKDFGVNWIVLGHSERRWYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 1mm6 A 2.15 BS01 QUS A 1 Y61 T91 R96 L138 G141 S142 T143 L192 E193 Y60 T90 R95 L137 G140 S141 T142 L191 E192 ? 0015276,0016020 ic50=20nM remove_due_to_license_issue P19491 12501192 500 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1mm7 A 1.65 BS02 QUS A 1 Y61 T91 R96 L138 G141 S142 T143 L192 E193 Y58 T88 R93 L135 G138 S139 T140 L189 E190 ? 0015276,0016020 ic50=20nM remove_due_to_license_issue P19491 12501192 801 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1mmp B 2.3 BS05 RSS B 1 N179 L181 H218 E219 H228 P238 T239 Y240 N80 L82 H120 E121 H130 P140 T141 Y142 H218 E219 H222 H228 H120 E121 H124 H130 3.4.24.23 0004222,0006508,0008237,0008270,0031012 Ki=0.85uM remove_due_to_license_issue Ki=850nM P09237 7756291 269 YSLFPNSPKWTSKVVTYRIVSYTRDLPHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAFAPGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYGNGDPQNFKLSQDDIKGIQKLYGK 1mmq A 1.9 BS05 RRS A 1 N179 L181 A182 H218 E219 H222 H228 P238 T239 Y240 N80 L82 A83 H120 E121 H124 H130 P140 T141 Y142 H218 E219 H222 H228 H120 E121 H124 H130 3.4.24.23 0004222,0006508,0008237,0008270,0031012 Ki=0.03uM remove_due_to_license_issue Ki=3nM P09237 7756291 269 YSLFPNSPKWTSKVVTYRIVSYTRDLPHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAFAPGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYGNGDPQNFKLSQDDIKGIQKLYGK 1mmr A 2.4 BS05 SRS A 1 N179 T180 L181 A182 H218 E219 H222 H228 P238 T239 Y240 N80 T81 L82 A83 H120 E121 H124 H130 P140 T141 Y142 H218 E219 H222 H228 H120 E121 H124 H130 3.4.24.23 0004222,0006508,0008237,0008270,0031012 Ki=4uM remove_due_to_license_issue P09237 7756291 269 YSLFPNSPKWTSKVVTYRIVSYTRDLPHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAFAPGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYGNGDPQNFKLSQDDIKGIQKLYGKR 1mn9 A 2.9 BS01 RTP A 1 K16 Y56 F64 L68 R92 R109 V116 N119 G122 G123 K11 Y51 F59 L63 R87 R104 V111 N114 G117 G118 K16 Y56 N119 G122 E133 K11 Y51 N114 G117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 12606760 160 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1mn9 B 2.9 BS01 RTP A 2 K16 Y56 H59 F64 L68 R92 T98 R109 V116 N119 G122 G123 K11 Y51 H54 F59 L63 R87 T93 R104 V111 N114 G117 G118 K16 Y56 N119 G122 E133 K11 Y51 N114 G117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 12606760 161 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1mnc A 2.1 BS04 PLH A 1 G179 I180 L181 A182 H218 E219 H222 H228 P238 N239 Y240 G74 I75 L76 A77 H113 E114 H117 H123 P133 N134 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.34 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P22894 7656015 280 GPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTGISQGEADINIAFYQRDHGDGSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1mns A 2.0 BS02 APG A 1 K164 K166 D195 E247 H297 E317 L319 K162 K164 D193 E245 H295 E315 L317 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 remove_due_to_license_issue P11444 8292591 361 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 1moq A 1.57 BS01 GLP A 1 T302 S303 S347 Q348 S349 T352 V399 A602 K603 T60 S61 S105 Q106 S107 T110 V157 A360 K361 E481 K485 E488 H504 K603 E239 K243 E246 H262 K361 2.6.1.16 0004360,0097367,1901135,1901137 Ki=0.35mM remove_due_to_license_issue P17169 9739095 609 GDKGIYRHYMQKEIYEQPNAIKNTLTGRISHGQVDLSELGPNADELLSKVEHIQILACGTSYNSGMVSRYWFESLAGIPCDVEIASEFRYRKSAVRRNSLMITLSQSGETADTLAGLRLSKELGYLGSLAICNVPGSSLVRESDLALMTNAGTEIGVASTKAFTTQLTVLLMLVAKLSRLKGLDASIEHDIVHGLQALPSRIEQMLSQDKRIEALAEDFSDKHHALFLGRGDQYPIALEGALKLKEISYIHAEAYAAGELKHGPLALIDADMPVIVVAPNNELLEKLKSNIEEVRARGGQLYVFADQDAGFVSSDNMHIIEMPHVEEVIAPIFYTVPLQLLAYHVALIKGTDVDQPRNLAKSVTVE 1mpl A 1.12 BS01 RE1 A 1 S62 F120 T123 Y159 N161 W233 G300 T301 Q303 S326 N327 S60 F118 T121 Y157 N159 W231 G298 T299 Q301 S324 N325 S62 K65 D114 T116 V130 Y159 N161 V165 T227 H298 G304 S60 K63 D112 T114 V128 Y157 N159 V163 T225 H296 G302 3.4.16.4 0004180,0005576,0006508,0008360,0009002,0009252,0071555 remove_due_to_license_issue P15555 12564922 400 LPAPDDTGLQAVLHTALSQGAPGAMVRVDDNGTIHQLSEGVADRATGRAITTTDRFRVGSVTKSFSAVVLLQLVDEGKLDLDASVNTYLPGLLPDDRITVRQVMSHRSGLYDYTNDMFAQTVPGFESVRNKVFSYQDLITLSLKHGVTNAPGAAYSYSNTNFVVAGMLIEKLTGHSVATEYQNRIFTPLNLTDTFYVHPDTVIPGTHANGYLTPDEAGGALVDSTEQTVSWAQSAGAVISSTQDLDTFFSALMSGQLMSAAQLAQMQQWTTVNSTQGYGLGLRRRDLSCGISVYGHTGTVQGYYTYAFASKDGKRSVTALANTSNNVNVLNTMARTLESAFCGKP 1mq5 A 2.1 BS02 XLC A 1 K96 E97 Y99 R143 E146 F174 D189 A190 V213 W215 G216 E217 G218 C220 G226 I227 Y228 K82 E83 Y85 R132 E135 F162 D179 A180 V203 W205 G206 E207 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=1nM remove_due_to_license_issue Ki=0.76nM P00742 12501180 500 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 1mq6 A 2.1 BS02 XLD A 1 E97 Y99 E146 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 Y228 E83 Y85 E135 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=7pM remove_due_to_license_issue Ki=0.007nM P00742 12501180 500 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 1mqd A 1.46 BS01 SHI A 1 Y58 T88 R93 G138 S139 T140 E190 M193 Y58 T88 R93 G138 S139 T140 E190 M193 ? 0015276,0016020 ic50=0.17uM remove_due_to_license_issue P19491 12417307 3001 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1mqg A 2.15 BS01 IWD A 1 Y61 L90 T91 R96 G141 S142 T143 E193 M196 Y58 L87 T88 R93 G138 S139 T140 E190 M193 ? 0015276,0016020 ic50=0.52uM remove_due_to_license_issue Ki=105nM P19491 12872125 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1mqh A 1.8 BS01 BWD A 1 Y61 L90 T91 R96 G141 S142 T143 L192 E193 M196 Y59 L88 T89 R94 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 ic50=0.3uM remove_due_to_license_issue Ki=61nM P19491 12872125 301 NKTVVVTTILESPYVMMKKNHEALEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1mqi A 1.35 BS01 FWD A 1 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y59 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 ic50=23.53nM remove_due_to_license_issue Ki=4nM, EC50=460nM P19491 12872125 401 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1mqj A 1.65 BS02 HWD A 1 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y59 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 ic50=4.76uM remove_due_to_license_issue Ki=1220nM P19491 12872125 301 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1mrn A 2.45 BS02 T5A A 1 D9 F36 P37 Y39 A49 E50 H53 F70 R74 R95 S99 N100 Y103 R160 Y165 D9 F36 P37 Y39 A49 E50 H53 F70 R74 R95 S99 N100 Y103 R160 Y165 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 Ki=30uM remove_due_to_license_issue P9WKE1 12454011 301 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAELAGERSRGRAQRDPGRARDNYERDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLA 1mrs A 2.0 BS02 5HU A 1 D9 P37 Y39 F70 R74 R95 N100 Y103 Y165 D9 P37 Y39 F70 R74 R95 N100 Y103 Y165 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 Ki=110uM remove_due_to_license_issue P9WKE1 12454011 217 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAELAGERSRGRAQRDPGRARDNYERDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLA 1mrw A 2.0 BS01 K57 A 1 R8 D25 G27 A28 G48 G49 I50 V82 R8 D25 G27 A28 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.2nM remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1mrw B 2.0 BS01 K57 A 1 D25 G27 A28 D29 D30 G48 G49 D25 G27 A28 D29 D30 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1mrx A 2.0 BS01 K57 B 1 D25 G27 A28 G48 G49 I50 F82 D25 G27 A28 G48 G49 I50 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1mrx B 2.0 BS01 K57 B 1 D25 G27 A28 D29 D30 G48 G49 I50 P81 D25 G27 A28 D29 D30 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=55nM remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1ms0 A 2.5 BS03 DAN A 1 R53 D59 D96 W120 Q195 E230 R245 R314 Y342 R53 D59 D96 W120 Q195 E230 R245 R314 Y342 3.2.1.18 0004308,0005737,0006689,0009313,0016020,0043231 remove_due_to_license_issue Ki=12300000nM Q26966 12419220 700 LAPGSSRVELFKRQSSKVPFEKDGKVTERVVHSFRLPALVNVDGVMVAIADARYETSFDNSLIDTVAKYSVDDGETWETQIAIKNSRASSVSRVVDPTVIVKGNKLYVLVGSYNSSRSYWTSHGDARDWDILLAVGEVTKSTAGGKITASIKWGSPVSLKEFFPAEMEGMHTNQFLGGAGVAIVASNGNLVYPVQVTNKKKQVFSKIFYSEDEGKTWKFGKGRSAFGCSEPVALEWEGKLIINTRVDYRRRLVYESSDMGNTWLEAVGTLSRVWGPSPKSNQPGSQSSFTAVTIEGMRVMLFTHPLNFKGRWLRDRLNLWLTDNQRIYNVGQVSIGDENSAYSSVLYKDDKLYCLHEINSNEVYSLVFARLVGELRIIKSVLQSWKNWDSHLSSICTPAGCGPAVTTVGLVGFLSHSATKTEWEDAYRCVNASTANAERVPNGLKFAGVGGGALWPVSQQGQNQRYHFANHAFTLVASVTIHEVPKGASPLLGASLDSSGGKKLLGLSYDKRHQWQPIYGSTPVTPTGSWEMGKRYHVVLTMANKIGSVYIDGEPLEGSGQTVVPDERTPDISHFYVGGYKRSGMPTDSRVTVNNVLLYNRQLNAEEIRTLFLSQDLIGTEAH 1ms6 A 1.9 BS01 BLN A 1 G23 C25 G68 G69 F70 M71 A140 F146 N163 G23 C25 G68 G69 F70 M71 A140 F146 N163 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue P25774 12459015 281 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 1ms7 A 1.97 BS02 SHI A 1 Y58 T88 R93 G138 S139 T140 L189 E190 M193 Y58 T88 R93 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 ic50=0.17uM remove_due_to_license_issue P19491 12417307 2001 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1msm A 2.0 BS01 JE2 B 1 D25 G27 A28 D30 I47 G48 I50 V82 I84 D25 G27 A28 D30 I47 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1msm B 2.0 BS01 JE2 B 1 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=33pM remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1msn A 2.0 BS01 JE2 B 1 D25 G27 A28 D30 V32 I47 G48 G49 P81 F82 D25 G27 A28 D30 V32 I47 G48 G49 P81 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1msn B 2.0 BS01 JE2 B 1 D25 G27 A28 D29 D30 I50 F82 D25 G27 A28 D29 D30 I50 F82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd<1nM remove_due_to_license_issue P03367 15103623 1001 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPFNVIGRNLLTQIGCTLNF 1mto A 3.2 BS01 F6P A 1 D127 M169 R171 E222 H249 R252 D127 M169 R171 E222 H249 R252 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 2.7.1.11 0003872,0005524,0005737,0005945,0006002,0006096,0008443,0016208,0016301,0030388,0042802,0046872,0048029,0061621,0070095 remove_due_to_license_issue P00512 12390023 1002 MKRIGVLTSGGDSPGMNAAIRSVVRKAIYHGVEVYGVYHGYAGLIAGNIKKLEVGDVGDIIHRGGTILYTARCPEFKTEEGQKKGIEQLKKHGIEGLVVIGGDGSYQGAKKLTEHGFPCVGVPGTIDNDIPGTDFTIGFDTALNTVIDAIDKIRDTATSHERTWVIEVMGRHAGDIALYSGLAGGAETILIPEADYDMNDVIARLKRGHERGKKHSIIIVAEGVGSGVDFGRQIQEATGFETRVTVLGHVQRGGSPTAFDRVLASRLGARAVELLLEGKGGRCVGIQNNQLVDHDIAEALANKHTIDQRMYALSKELSI 1mto A 3.2 BS02 F6P B 1 R162 R243 R162 R243 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 2.7.1.11 0003872,0005524,0005737,0005945,0006002,0006096,0008443,0016208,0016301,0030388,0042802,0046872,0048029,0061621,0070095 remove_due_to_license_issue P00512 12390023 1001 MKRIGVLTSGGDSPGMNAAIRSVVRKAIYHGVEVYGVYHGYAGLIAGNIKKLEVGDVGDIIHRGGTILYTARCPEFKTEEGQKKGIEQLKKHGIEGLVVIGGDGSYQGAKKLTEHGFPCVGVPGTIDNDIPGTDFTIGFDTALNTVIDAIDKIRDTATSHERTWVIEVMGRHAGDIALYSGLAGGAETILIPEADYDMNDVIARLKRGHERGKKHSIIIVAEGVGSGVDFGRQIQEATGFETRVTVLGHVQRGGSPTAFDRVLASRLGARAVELLLEGKGGRCVGIQNNQLVDHDIAEALANKHTIDQRMYALSKELSI 1mto B 3.2 BS01 F6P A 1 R162 R243 R162 R243 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 2.7.1.11 0003872,0005524,0005737,0005945,0006002,0006096,0008443,0016208,0016301,0030388,0042802,0046872,0048029,0061621,0070095 remove_due_to_license_issue P00512 12390023 1002 MKRIGVLTSGGDSPGMNAAIRSVVRKAIYHGVEVYGVYHGYAGLIAGNIKKLEVGDVGDIIHRGGTILYTARCPEFKTEEGQKKGIEQLKKHGIEGLVVIGGDGSYQGAKKLTEHGFPCVGVPGTIDNDIPGTDFTIGFDTALNTVIDAIDKIRDTATSHERTWVIEVMGRHAGDIALYSGLAGGAETILIPEADYDMNDVIARLKRGHERGKKHSIIIVAEGVGSGVDFGRQIQEATGFETRVTVLGHVQRGGSPTAFDRVLASRLGARAVELLLEGKGGRCVGIQNNQLVDHDIAEALANKHTIDQRMYALSKELSI 1mto B 3.2 BS02 F6P B 1 D127 M169 R171 E222 H249 R252 D127 M169 R171 E222 H249 R252 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 G11 R72 C73 D103 G104 G124 T125 D127 D129 R171 2.7.1.11 0003872,0005524,0005737,0005945,0006002,0006096,0008443,0016208,0016301,0030388,0042802,0046872,0048029,0061621,0070095 remove_due_to_license_issue P00512 12390023 1001 MKRIGVLTSGGDSPGMNAAIRSVVRKAIYHGVEVYGVYHGYAGLIAGNIKKLEVGDVGDIIHRGGTILYTARCPEFKTEEGQKKGIEQLKKHGIEGLVVIGGDGSYQGAKKLTEHGFPCVGVPGTIDNDIPGTDFTIGFDTALNTVIDAIDKIRDTATSHERTWVIEVMGRHAGDIALYSGLAGGAETILIPEADYDMNDVIARLKRGHERGKKHSIIIVAEGVGSGVDFGRQIQEATGFETRVTVLGHVQRGGSPTAFDRVLASRLGARAVELLLEGKGGRCVGIQNNQLVDHDIAEALANKHTIDQRMYALSKELSI 1mtr A 1.75 BS01 PI6 B 1 R8 D25 G48 G49 I50 P81 V82 R8 D25 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1mtr B 1.75 BS01 PI6 B 1 D25 G27 A28 D29 G48 I50 P81 D25 G27 A28 D29 G48 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4nM remove_due_to_license_issue P03369 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1mu6 B 1.99 BS03 CDA B 1 H57 Y60A N98 L99 A190 C191 S195 S214 W215 G216 H43 Y47 N95 L96 A192 C193 S197 S218 W219 G220 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 Ki=4.2nM remove_due_to_license_issue Ki=4.2nM P00734 12570369 248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1mu8 B 2.0 BS03 CDB B 1 H57 Y60A N98 A190 S195 V213 S214 W215 G216 H43 Y47 N95 A192 S197 V217 S218 W219 G220 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 Ki=1nM remove_due_to_license_issue P00734 12570369 248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1mue B 2.0 BS03 CDD B 1 H57 Y60A L99 A190 S195 S214 W215 G216 H43 Y47 L96 A192 S197 S218 W219 G220 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 Ki=2.3nM remove_due_to_license_issue Ki=2.3nM P00734 12657281 248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1mui A 2.8 BS01 AB1 B 1 D25 G27 D29 D30 G49 I50 P81 D25 G27 D29 D30 G49 I50 P81 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q903J0 12057670 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1mui B 2.8 BS01 AB1 B 1 D25 G27 A28 D29 G48 G49 P81 V82 I84 D25 G27 A28 D29 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q903J0 12057670 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1mwt A 2.45 BS01 PNM A 1 S403 Y446 S462 N464 Q521 S598 T600 Q613 S377 Y420 S436 N438 Q495 S572 T574 Q580 2.4.1.129 0005886,0008658,0016020,0016757,0046677,0071555,0071972 remove_due_to_license_issue Q93IC2 12389036 1007 DKEINNTIDAIEDKNFKQVYKDSSYISKSDNGEVEMTERPIKIYNSLGVKDINIQDRKIKKVSKNKKRVDAQYKIKTNYGNIDRNVQFNFVKEDGMWKLDWDHSVIIPGMQKDQSIHIENLKSERGKILDRNNVELANTGTAYEIGIVPKNVSKKDYKAIAKELSISEDYIKQQMDQNWVQDDTFVPLKTVKKMDEYLSDFAKKFHLTTNETESRNYPLEKATSHLLGYVGPINSEELKQKEYKGYKDDAVIGKKGLEKLYDKKLQHEDGYRVTIVDDNSNTIAHTLIEKKKKDGKDIQLTIDAKVQKSIYNNMKNDYGSGTAIHPQTGELLALVSTPSYDVYPFMYGMSNEEYNKLTEDKKEPLLNKFQITTSPGSTQKILTAMIGLNNKTLDDKTSYKIDGKGWQKDKSWGGYNVTRYEVVNGNIDLKQAIESSDNIFFARVALELGSKKFEKGMKKLGVGEDIPSDYPFYNAQISNKNLDNEILLADSGYGQGEILINPVQILSIYSALENNGNINAPHLLKDTKNKVWKKNIISKENINLLTDGMQQVVNKTHKEDIYRSYANLIGKSGTAELGRQIGWFISYDKDNPNMMMAINVKDVQDKGMASYNAKISGKVYDELYENGNKKYDIDE 1mx1 A 2.4 BS02 THA A 1 L1097 F1101 S1221 H1468 L77 F81 S201 H447 G1142 G1143 S1221 A1222 E1354 H1468 G122 G123 S201 A202 E334 H447 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 remove_due_to_license_issue IC50=>100000nM, Ki=>100000nM P23141 12725862 1 SSPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1mxo A 1.83 BS01 SM2 A 1 S64 L119 Y150 Y221 N289 G317 A318 T319 S61 L116 Y147 Y218 N286 G314 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 12526668 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1mxu A 1.8 BS02 BWD A 1 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y58 L87 T88 R93 L135 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 ic50=4uM remove_due_to_license_issue Ki=61nM P19491 12731861 300 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1my3 A 1.75 BS02 BWD A 1 Y61 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y58 T88 R93 L135 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 remove_due_to_license_issue Ki=61nM P19491 12731861 800 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1my4 A 1.9 BS02 IWD A 1 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y58 L87 T88 R93 L135 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 remove_due_to_license_issue Ki=105nM P19491 12731861 601 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1my8 A 1.72 BS01 SM3 A 1 S64 L119 Y150 Y221 G317 A318 T319 S61 L116 Y147 Y218 G314 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.035uM remove_due_to_license_issue P00811 12526668 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1mzc B 2.0 BS05 BNE B 1 W602 W606 R702 D797 C799 Y800 Y861 H862 W86 W90 R186 D281 C283 Y284 Y345 H346 H748 R791 K794 D797 C799 Y800 D852 D859 H862 H232 R275 K278 D281 C283 Y284 D336 D343 H346 2.5.1.58 0003824,0004659,0004660,0005515,0005829,0005875,0005965,0006629,0008270,0008318,0018343,0046872 ic50=0.06nM remove_due_to_license_issue IC50=0.06nM P49356 12825937 1003 PVWSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPEGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYDIINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKRERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVLGVPENALQPTHPVYNIGPDKVIQATTYFLQKPVPGF 1mzs A 2.1 BS01 669 A 1 W32 R36 R151 G152 I156 M207 G209 F213 A246 N247 F304 W32 R36 R151 G152 I156 M207 G209 F213 A246 N247 F304 2.3.1.180 0004315,0005737,0005829,0006631,0006633,0016746,0033818,0044281 ic50=7uM remove_due_to_license_issue P0A6R0 12502353 350 MYTKIIGTGSYLPEQVRTNADLEKMVDTSDEWIVTRTGIRERHIAAPNETVSTMGFEAATRAIEMAGIEKDQIGLIVVATTSATHAFPSAACQIQSMLGIKGCPAFDVAAACAGFTYALSVADQYVKSGAVKYALVVGSDVLARTCDPTDRGTIIIFGDGAGAAVLAASEEPGIISTHLHADGSYGELLTLPNADRVNPENSIHLTMAGNEVFKVAVTELAHIVDETLAANNLDRSQLDWLVPHQANLRIISATAKKLGMSMDNVVVTLDRHGNTSAASVPCALDEAVRDGRIKPGQLVLLEAFGGGFTWGSALVRF 1n0s A 2.0 BS01 FLU A 1 Y22 E28 Y47 R58 M69 H86 F99 H127 W129 Y22 E28 Y47 R58 M69 H86 F99 H127 W129 ? 0000302,0005576,0005737,0006629,0006950,0031409 Kd=35.2nM remove_due_to_license_issue P09464 12945055 500 DVYHDGACPEVKPVDNFDWSQYHGKWWEVAKYPSPNGKYGKCGWAEYTPEGKSVKVSRYDVIHGKEYFMEGTAYPVGDSKIGKIYHSRTVGGYTRKTVFNVLSTDNKNYIIGYSCRYDEDKKGHWDHVWVLSRSMVLTGEAKTAVENYLIGSPVVDSQKLVYSDFSEAACKVN 1n0t A 2.1 BS01 AT1 A 1 E13 Y61 P89 L90 T91 R96 G141 S142 T143 E193 Y220 E9 Y57 P85 L86 T87 R92 G137 S138 T139 E189 Y216 ? 0015276,0016020 ic50=12.2uM remove_due_to_license_issue P19491 12519060 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1n1g A 2.5 BS01 BCP A 1 M225 R336 L339 M217 R325 L328 K210 T267 K202 T259 1.1.1.8 0005829,0005975,0006072,0006116,0016491,0016616,0020015,0046168,0051287,0141152 ic50=5mM remove_due_to_license_issue P90551 12445769 402 KDELLYLNKAVVFGSGAFGTALAMVLSKKCREVCVWHMNEEEVRLVNEKRENVLFLKGVQLASNITFTSDVEKAYNGAEIILFVIPTQFLRGFFEKSGGNLIAYAKEKQVPVLVCTKGIERSTLKFPAEIIGEFLPSPLLSVLAGPSFAIEVATGVFTCVSIASADINVARRLQRIMSTGDRSFVCWATTDTVGCEVASAVKNVLAIGSGVANGLGMGLNARAALIMRGLLEIRDLTAALGGDGSAVFGLAGLGDLQLTCSSELSRNFTVGKKLGKGLPIEEIQRAVAEGVATADPLMRLAKQLKVKMPLCHQIYEIVYKKKNPRDALADLLSCGLQDEGLPPLFK 1n1g A 2.5 BS02 BCP A 2 W44 M46 F97 W36 M38 F89 K210 T267 K202 T259 1.1.1.8 0005829,0005975,0006072,0006116,0016491,0016616,0020015,0046168,0051287,0141152 ic50=5mM remove_due_to_license_issue P90551 12445769 403 KDELLYLNKAVVFGSGAFGTALAMVLSKKCREVCVWHMNEEEVRLVNEKRENVLFLKGVQLASNITFTSDVEKAYNGAEIILFVIPTQFLRGFFEKSGGNLIAYAKEKQVPVLVCTKGIERSTLKFPAEIIGEFLPSPLLSVLAGPSFAIEVATGVFTCVSIASADINVARRLQRIMSTGDRSFVCWATTDTVGCEVASAVKNVLAIGSGVANGLGMGLNARAALIMRGLLEIRDLTAALGGDGSAVFGLAGLGDLQLTCSSELSRNFTVGKKLGKGLPIEEIQRAVAEGVATADPLMRLAKQLKVKMPLCHQIYEIVYKKKNPRDALADLLSCGLQDEGLPPLFK 1n1m A 2.5 BS01 A3M A 1 E205 E206 S630 V656 Y662 Y666 N710 V711 E167 E168 S592 V618 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=2uM remove_due_to_license_issue IC50=4000nM, Ki=470nM P27487 12483204 954 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 1n1t A 1.6 BS01 DAN A 1 R39 D63 M99 D100 W124 R249 R318 Y346 R39 D63 M99 D100 W124 R249 R318 Y346 3.2.1.18 0004308,0005737,0006689,0009313,0016020,0016798,0043231 remove_due_to_license_issue O44049 12507479 700 AASLAPGSSRVELFKRKNSTVPFEESNGTIRERVVHSFRIPTIVNVDGVMVAIADARYETSFDNSFIETAVKYSVDDGATWNTQIAIKNSRASSVSRVMDATVIVKGNKLYILVGSFNKTRNSWTQHRDGSDWEPLLVVGEVTKSAANGKTTATISWGKPVSLKPLFPAEFDGILTKEFVGGVGAAIVASNGNLVYPVQIADMGGRVFTKIMYSEDDGNTWKFAEGRSKFGCSEPAVLEWEGKLIINNRVDGNRRLVYESSDMGKTWVEALGTLSHVWTNSPTSNQQDCQSSFVAVTIEGKRVMLFTHPLNLKGRWMRDRLHLWMTDNQRIFDVGQISIGDENSGYSSVLYKDDKLYSLHEINTNDVYSLVFVRLIGELQLMKSVVRTWKEEDNHLASICTPVVPAGCGAAVPTAGLVGFLSHSANGSVWEDVYRCVDANVANAERVPNGLKFNGVGGGAVWPVARQGQTRRYQFANYRFTLVATVTIDELPKGTSPLLGAGLEGPGDAKLLGLSYDKNRQWRPLYGAAPASPTGSWELHKKYHVVLTMADRQGSVYVDGQPLAGSGNTVVRGATLPDISHFYIGGPRSKGAPTDSRVTVTNVVLYNRRLNSSEIRTLFLSQDMIGTD 1n1v A 2.1 BS01 DAN A 1 R39 D63 D100 W124 R249 R318 Y346 R39 D63 D100 W124 R249 R318 Y346 3.2.1.18 0004308,0005737,0006689,0009313,0016020,0016798,0043231 Ki=140uM remove_due_to_license_issue O44049 12507479 670 AASLAPGSSRVELFKRKNSTVPFEESNGTIRERVVHSFRIPTIVNVDGVMVAIADARYETSFDNSFIETAVKYSVDDGATWNTQIAIKNSRASSVSRVMDATVIVKGNKLYILVGSFNKTRNSWTQHRDGSDWEPLLVVGEVTKSAANGKTTATISWGKPVSLKPLFPAEFDGILTKEFVGGVGAAIVASNGNLVYPVQIADMGGRVFTKIMYSEDDGNTWKFAEGRSKFGCSEPAVLEWEGKLIINNRVDGNRRLVYESSDMGKTWVEALGTLSHVWTNSPTSNQQDCQSSFVAVTIEGKRVMLFTHPLNLKGRWMRDRLHLWMTDNQRIFDVGQISIGDENSGYSSVLYKDDKLYSLHEINTNDVYSLVFVRLIGELQLMKSVVRTWKEEDNHLASICTPVVPAGCGAAVPTAGLVGFLSHSANGSVWEDVYRCVDANVANAERVPNGLKFNGVGGGAVWPVARQGQTRRYQFANYRFTLVATVTIDELPKGTSPLLGAGLEGPGDAKLLGLSYDKNRQWRPLYGAAPASPTGSWELHKKYHVVLTMADRQGSVYVDGQPLAGSGNTVVRGATLPDISHFYIGGPRSKGAPTDSRVTVTNVVLYNRRLNSSEIRTLFLSQDMIGTD 1n2v A 2.1 BS02 BDI A 1 Y106 D156 G229 M260 G261 Y96 D146 G219 M250 G251 D102 D280 C318 C320 C323 H349 D92 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=83uM remove_due_to_license_issue P28720 12646024 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1n32 B 3.0 BS01 rna A 0 W24 P26 G99 T103 N104 R111 R144 I172 E176 K179 W18 P20 G93 T97 N98 R105 R138 I166 E170 K173 ? 0003735,0005840,0006412,0015935,0019843,0022627,1990904 remove_due_to_license_issue P80371 12464183 5 ~ 1544 VKELLEAGVHFGHERKRWNPKFARYIYAERNGIHIIDLQKTMEELERTFRFIEDLAMRGGTILFVGTKKQAQDIVRMEAERAGMPYVNQRWLGGMLTNFKTISQRVHRLEELEALFASPEIEERPKKEQVRLKHELERLQKYLSGFRLLKRLPDAIFVVDPTKEAIAVREARKLFIPVIALADTDSDPDLVDYIIPGNDDAIRSIQLILSRAVDLIIQARGGVVEPSPSYALVQ 1n32 C 3.0 BS01 rna A 0 G2 N3 K4 I5 K27 S154 R156 E161 Q162 A163 W167 R172 V173 P174 H176 T177 L178 R179 F186 T192 Y193 G194 V195 K199 G1 N2 K3 I4 K26 S153 R155 E160 Q161 A162 W166 R171 V172 P173 H175 T176 L177 R178 F185 T191 Y192 G193 V194 K198 ? 0003676,0003723,0003729,0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P80372 12464183 5 ~ 1544 GNKIHPIGFRLGITRDWESRWYAGKKQYRHLLLEDQRIRGLLEKELYSAGLARVDIERAADNVAVTVHVAKPGVVIGRGGERIRVLREELAKLTGKNVALNVQEVQNPNLSAPLVAQRVAEQIERRFAVRRAIKQAVQRVMESGAKGAKVIVSGRIGGAEQARTEWAAQGRVPLHTLRANIDYGFALARTTYGVLGVKAYIFLGEV 1n32 D 3.0 BS01 rna A 0 G2 I5 P7 V8 C9 R10 R13 R14 K22 E24 R25 K30 R35 R36 Y38 P40 G41 Q42 H43 K46 S52 Y54 A55 R59 Q62 R66 E72 R73 Q74 S113 R115 Q116 R118 Q119 R122 H123 H125 R132 V133 D134 L135 S137 Y138 L155 S208 R209 G1 I4 P6 V7 C8 R9 R12 R13 K21 E23 R24 K29 R34 R35 Y37 P39 G40 Q41 H42 K45 S51 Y53 A54 R58 Q61 R65 E71 R72 Q73 S112 R114 Q115 R117 Q118 R121 H122 H124 R131 V132 D133 L134 S136 Y137 L154 S207 R208 ? 0003723,0003735,0005840,0006412,0015935,0019843,0042274,0046872,1990904 remove_due_to_license_issue P80373 12464183 5 ~ 1544 GRYIGPVCRLCRREGVKLYLKGERCYSPKCAMERRPYPPGQHGQKRARRPSDYAVRLREKQKLRRIYGISERQFRNLFEEASKKKGVTGSVFLGLLESRLDNVVYRLGFAVSRRQARQLVRHGHITVNGRRVDLPSYRVRPGDEIAVAEKSRNLELIRQNLEAMKGRKVGPWLSLDVEGMKGKFLRLPDREDLALPVNEQLVIEFYSR 1n32 E 3.0 BS01 rna A 0 R14 T16 A17 R18 M19 Q20 A21 G22 R24 R25 K47 P49 K57 A86 K92 A94 A95 T98 I101 A102 G103 L119 T120 K121 E122 L123 S125 R126 N127 N130 R10 T12 A13 R14 M15 Q16 A17 G18 R20 R21 K43 P45 K53 A82 K88 A90 A91 T94 I97 A98 G99 L115 T116 K117 E118 L119 S121 R122 N123 N126 ? 0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHQ5 12464183 5 ~ 1544 DFEEKMILIRRTARMQAGGRRFRFGALVVVGDRQGRVGLGFGKAPEVPLAVQKAGYYARRNMVEVPLQNGTIPHEIEVEFGASKIVLKPAAPGTGVIAGAVPRAILELAGVTDILTKELGSRNPINIAYATMEALRQLRTKADVERLRKG 1n32 F 3.0 BS01 rna A 0 R2 Y4 Y50 K54 E69 N73 R87 V90 K92 R2 Y4 Y50 K54 E69 N73 R87 V90 K92 ? 0003735,0005737,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLP8 12464183 5 ~ 1544 MRRYEVNIVLNPNLDQSQLALEKEIIQRALENYGARVEKVEELGLRRLAYPIAKDPQGYFLWYQVEMPEDRVNDLARELRIRDNVRRVMVVKSQEPFLANA 1n32 G 3.0 BS01 rna A 0 A2 R3 R4 R6 A7 R10 L12 N28 K29 I30 R32 D33 G34 K35 K36 L38 R41 I42 R76 G81 R94 R95 S98 R102 N109 R114 A116 R119 A1 R2 R3 R5 A6 R9 L11 N27 K28 I29 R31 D32 G33 K34 K35 L37 R40 I41 R75 G80 R93 R94 S97 R101 N108 R113 A115 R118 ? 0000049,0003723,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P17291 12464183 5 ~ 1544 ARRRRAEVRQLQPDLVYGDVLVTAFINKIMRDGKKNLAARIFYDACKIIQEKTGQEPLKVFKQAVENVKPRMEVRSRRVGGANYQVPMEVSPRRQQSLALRWLVQAANQRPERRAAVRIAHELMDAAEGKGGAVKKKEDVERMAEANRAYAHYRW 1n32 H 3.0 BS01 rna A 0 M1 L2 T3 P5 D8 T11 R12 R14 N15 S29 R30 F31 K56 R75 K88 P89 G90 R92 Y94 V95 G96 V97 S113 T114 S115 G128 G130 E132 M1 L2 T3 P5 D8 T11 R12 R14 N15 S29 R30 F31 K56 R75 K88 P89 G90 R92 Y94 V95 G96 V97 S113 T114 S115 G128 G130 E132 ? 0003735,0005737,0005840,0006412,0019843,1990904 remove_due_to_license_issue P0DOY9 12464183 5 ~ 1544 MLTDPIADMLTRIRNATRVYKESTDVPASRFKEEILRILAREGFIKGYERVDVDGKPYLRVYLKYGPRRQGPDPRPEQVIHHIRRISKPGRRVYVGVKEIPRVRRGLGIAILSTSKGVLTDREARKLGVGGELICEVW 1n32 I 3.0 BS01 rna A 0 Q3 Y5 T7 R9 K11 E12 V14 R16 R20 Y36 Q38 Y62 R66 G67 G68 G69 K70 S71 Q73 R83 K97 T103 R104 A106 R107 V108 E110 R111 K112 K113 Y114 G115 H117 K118 R120 R121 A122 Q124 Y125 S126 K127 R128 Q2 Y4 T6 R8 K10 E11 V13 R15 R19 Y35 Q37 Y61 R65 G66 G67 G68 K69 S70 Q72 R82 K96 T102 R103 A105 R106 V107 E109 R110 K111 K112 Y113 G114 H116 K117 R119 R120 A121 Q123 Y124 S125 K126 R127 ? 0000049,0003723,0003735,0005737,0005840,0006412,0019843,0022627,0043232,1990904 remove_due_to_license_issue P80374 12464183 5 ~ 1544 EQYYGTGRRKEAVARVFLRPGNGKVTVNGQDFNEYFQGLVRAVAALEPLRAVDALGRFDAYITVRGGGKSGQIDAIKLGIARALVQYNPDYRAKLKPLGFLTRDARVVERKKYGKHKARRAPQYSKR 1n32 J 3.0 BS01 rna A 0 R5 R9 H13 D17 S35 P37 I38 P39 L40 P41 R43 R45 T48 R51 G52 F54 K55 H56 K57 R60 H62 H68 D73 R3 R7 H11 D15 S33 P35 I36 P37 L38 P39 R41 R43 T46 R49 G50 F52 K53 H54 K55 R58 H60 H66 D71 ? 0000049,0003723,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q5SHN7 12464183 5 ~ 1544 KIRIKLRGFDHKTLDASAQKIVEAARRSGAQVSGPIPLPTRVRRFTVIRGPFKHKDSREHFELRTHNRLVDIINPNRKTIEQLMTLDLPTGVEIEIKT 1n32 K 3.0 BS01 rna A 0 R12 Y20 N26 N27 I29 T31 G37 N38 P39 W42 S44 G46 G52 S53 K55 R85 V114 H116 N117 G118 C119 R120 K122 K123 K124 R2 Y10 N16 N17 I19 T21 G27 N28 P29 W32 S34 G36 G42 S43 K45 R75 V104 H106 N107 G108 C109 R110 K112 K113 K114 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P80376 12464183 5 ~ 1544 KRQVASGRAYIHASYNNTIVTITDPDGNPITWSSGGVIGYKGSRKGTPYAAQLAALDAAKKAMAYGMQSVDVIVRGTGAGREQAIRALQASGLQVKSIVDDTPVPHNGCRPKKKFRKAS 1n32 L 3.0 BS01 rna A 0 P5 T6 N8 Q9 L10 R12 R15 E16 K17 K20 K21 K23 K28 G29 A30 P31 F32 R33 R34 K46 N49 S50 A51 L52 R53 K54 K57 T61 Y69 G72 E73 R86 G87 K91 D92 P94 R97 R113 K114 K115 S116 R117 S118 K119 T122 K123 K124 P1 T2 N4 Q5 L6 R8 R11 E12 K13 K16 K17 K19 K24 G25 A26 P27 F28 R29 R30 K42 N45 S46 A47 L48 R49 K50 K53 T57 Y65 G68 E69 R82 G83 K87 D88 P90 R93 R109 K110 K111 S112 R113 S114 K115 T118 K119 K120 ? 0000049,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHN3 12464183 5 ~ 1544 PTINQLVRKGREKVRKKSKVPALKGAPFRRGVCTVVRTVTPKKPNSALRKVAKVRLTSGYEVTAYIPGEGHNLQEHSVVLIRGGRVKDLPGVRYHIVRGVYDAAGVKDRKKSRSKYGTKKPKEA 1n32 M 3.0 BS01 rna A 0 K13 R14 V17 Y23 G24 I25 G26 A28 R29 R44 N77 Y87 R88 R91 H92 L96 P97 V98 R99 Q101 R102 T103 R104 T105 N106 A107 R108 T109 R110 K111 R114 K115 T116 V117 K12 R13 V16 Y22 G23 I24 G25 A27 R28 R43 N76 Y86 R87 R90 H91 L95 P96 V97 R98 Q100 R101 T102 R103 T104 N105 A106 R107 T108 R109 K110 R113 K114 T115 V116 ? 0000049,0003676,0003723,0003735,0005829,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P80377 12464183 5 ~ 1544 ARIAGVEIPRNKRVDVALTYIYGIGKARAKEALEKTGINPATRVKDLTEAEVVRLREYVENTWKLEGELRAEVAANIKRLMDIGCYRGLRHRRGLPVRGQRTRTNARTRKGPRKTVAG 1n32 N 3.0 BS01 rna A 0 R3 K4 A5 L6 K15 F16 V18 R19 Y21 T22 C27 R29 R31 S32 R35 R41 I42 R45 E46 K58 S60 W61 R2 K3 A4 L5 K14 F15 V17 R18 Y20 T21 C26 R28 R30 S31 R34 R40 I41 R44 E45 K57 S59 W60 ? 0003735,0005737,0005840,0006412,0008270,0015935,0019843,0046872,1990904 remove_due_to_license_issue P0DOY6 12464183 5 ~ 1544 ARKALIEKAKRTPKFKVRAYTRCVRCGRARSVYRFFGLCRICLRELAHKGQLPGVRKASW 1n32 O 3.0 BS01 rna A 0 P2 K5 K8 F18 D21 T22 G23 S24 Q28 L31 R35 L39 H42 H46 K48 D49 H51 S52 R54 G55 M58 Q62 R64 R65 Y69 R72 P1 K4 K7 F17 D20 T21 G22 S23 Q27 L30 R34 L38 H41 H45 K47 D48 H50 S51 R53 G54 M57 Q61 R63 R64 Y68 R71 ? 0003735,0005737,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue Q5SJ76 12464183 5 ~ 1544 PITKEEKQKVIQEFARFPGDTGSTEVQVALLTLRINRLSEHLKVHKKDHHSHRGLLMMVGQRRRLLRYLQREDPERYRALIEKLGIRG 1n32 P 3.0 BS01 rna A 0 M1 K3 R5 L6 R8 F9 G10 S11 K12 H13 N14 H16 Y17 R18 D23 R25 K27 R28 G30 K31 I33 Y38 P41 R42 K43 T44 T45 W59 V62 G63 Q65 T67 D68 T69 R72 R75 F80 R81 Q82 E83 M1 K3 R5 L6 R8 F9 G10 S11 K12 H13 N14 H16 Y17 R18 D23 R25 K27 R28 G30 K31 I33 Y38 P41 R42 K43 T44 T45 W59 V62 G63 Q65 T67 D68 T69 R72 R75 F80 R81 Q82 E83 ? 0003735,0005737,0005840,0006412,0015935,1990904 remove_due_to_license_issue Q5SJH3 12464183 5 ~ 1544 MVKIRLARFGSKHNPHYRIVVTDARRKRDGKYIEKIGYYDPRKTTPDWLKVDVERARYWLSVGAQPTDTARRLLRQAGVFRQE 1n32 Q 3.0 BS01 rna A 0 P2 K3 S12 K14 M15 Q16 K17 T18 R25 L31 Y32 K34 R38 S39 K40 K41 Y42 E61 S62 R63 P64 I65 S66 K67 R68 K69 R70 R72 R91 N94 Y95 L98 S99 K100 R101 G102 A105 P1 K2 S11 K13 M14 Q15 K16 T17 R24 L30 Y31 K33 R37 S38 K39 K40 Y41 E60 S61 R62 P63 I64 S65 K66 R67 K68 R69 R71 R90 N93 Y94 L97 S98 K99 R100 G101 A104 ? 0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P0DOY7 12464183 5 ~ 1544 PKKVLTGVVVSDKMQKTVTVLVERQFPHPLYGKVIKRSKKYLAHDPEEKYKLGDVVEIIESRPISKRKRFRVLRLVESGRMDLVEKYLIRRQNYQSLSKRGGKA 1n32 R 3.0 BS01 rna A 0 K49 I50 K61 Q63 R64 K68 K71 R72 R74 I75 F81 K34 I35 K46 Q48 R49 K53 K56 R57 R59 I60 F66 ? 0003735,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLQ0 12464183 5 ~ 1544 PSRKAKVKATLGEFDLRDYRNVEVLKRFLSETGKILPRRRTGLSGKEQRILAKTIKRARILGLLPFTEKLVRK 1n32 S 3.0 BS01 rna A 0 P2 R3 S4 L5 K6 F10 H14 K18 W34 R36 R37 Y52 N53 G54 K55 K70 G72 E73 T77 R78 T79 Y80 P1 R2 S3 L4 K5 F9 H13 K17 W33 R35 R36 Y51 N52 G53 K54 K69 G71 E72 T76 R77 T78 Y79 ? 0000028,0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHP2 12464183 5 ~ 1544 PRSLKKGVFVDDHLLEKVLELNAKGEKRLIKTWSRRSTIVPEMVGHTIAVYNGKQHVPVYITENMVGHKLGEFAPTRTYR 1n32 T 3.0 BS01 rna A 0 L10 K14 R15 H16 R17 S19 R22 R23 R25 N26 K27 A28 K29 S31 T35 L36 K38 K39 E60 S61 D64 K65 K68 S70 K74 N75 A78 R79 K81 S82 R83 M85 R86 K87 R89 G101 G102 G103 S105 L3 K7 R8 H9 R10 S12 R15 R16 R18 N19 K20 A21 K22 S24 T28 L29 K31 K32 E53 S54 D57 K58 K61 S63 K67 N68 A71 R72 K74 S75 R76 M78 R79 K80 R82 G94 G95 G96 S98 ? 0003723,0003735,0005840,0006412,0015935,0019843,0070181,1990904 remove_due_to_license_issue P80380 12464183 5 ~ 1544 RNLSALKRHRQSLKRRLRNKAKKSAIKTLSKKAIQLAQEGKAEEALKIMRKAESLIDKAAKGSTLHKNAAARRKSRLMRKVRQLLEAAGAPLIGGGLSA 1n33 B 3.35 BS01 rna A 0 W24 G99 T103 N104 T107 R111 I172 E176 W18 G93 T97 N98 T101 R105 I166 E170 ? 0003735,0005840,0006412,0015935,0019843,0022627,1990904 remove_due_to_license_issue P80371 12464183 5 ~ 1544 VKELLEAGVHFGHERKRWNPKFARYIYAERNGIHIIDLQKTMEELERTFRFIEDLAMRGGTILFVGTKKQAQDIVRMEAERAGMPYVNQRWLGGMLTNFKTISQRVHRLEELEALFASPEIEERPKKEQVRLKHELERLQKYLSGFRLLKRLPDAIFVVDPTKEAIAVREARKLFIPVIALADTDSDPDLVDYIIPGNDDAIRSIQLILSRAVDLIIQARGGVVEPSPSYALVQ 1n33 C 3.35 BS01 rna A 0 G2 N3 K4 I5 K27 S154 E161 Q162 A163 R172 V173 P174 H176 T177 L178 R179 T192 Y193 G194 V195 K199 G1 N2 K3 I4 K26 S153 E160 Q161 A162 R171 V172 P173 H175 T176 L177 R178 T191 Y192 G193 V194 K198 ? 0003676,0003723,0003729,0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P80372 12464183 5 ~ 1544 GNKIHPIGFRLGITRDWESRWYAGKKQYRHLLLEDQRIRGLLEKELYSAGLARVDIERAADNVAVTVHVAKPGVVIGRGGERIRVLREELAKLTGKNVALNVQEVQNPNLSAPLVAQRVAEQIERRFAVRRAIKQAVQRVMESGAKGAKVIVSGRIGGAEQARTEWAAQGRVPLHTLRANIDYGFALARTTYGVLGVKAYIFLGEV 1n33 D 3.35 BS01 rna A 0 G2 P7 V8 C9 R10 R13 R14 K22 E24 R25 K30 R35 R36 Y38 P40 G41 Q42 H43 Q45 S52 Y54 A55 R59 Q62 R66 E72 R73 Q74 R76 R115 Q116 R118 Q119 R122 H123 H125 R132 D134 L135 S137 R141 L155 E205 S208 R209 G1 P6 V7 C8 R9 R12 R13 K21 E23 R24 K29 R34 R35 Y37 P39 G40 Q41 H42 Q44 S51 Y53 A54 R58 Q61 R65 E71 R72 Q73 R75 R114 Q115 R117 Q118 R121 H122 H124 R131 D133 L134 S136 R140 L154 E204 S207 R208 ? 0003723,0003735,0005840,0006412,0015935,0019843,0042274,0046872,1990904 remove_due_to_license_issue P80373 12464183 5 ~ 1544 GRYIGPVCRLCRREGVKLYLKGERCYSPKCAMERRPYPPGQHGQKRARRPSDYAVRLREKQKLRRIYGISERQFRNLFEEASKKKGVTGSVFLGLLESRLDNVVYRLGFAVSRRQARQLVRHGHITVNGRRVDLPSYRVRPGDEIAVAEKSRNLELIRQNLEAMKGRKVGPWLSLDVEGMKGKFLRLPDREDLALPVNEQLVIEFYSR 1n33 E 3.35 BS01 rna A 0 R14 T16 A17 R18 M19 Q20 G22 R24 R25 K47 P49 K57 Y61 A86 K92 A94 T98 I101 A102 T120 K121 E122 L123 S125 R126 N127 N130 Y133 R10 T12 A13 R14 M15 Q16 G18 R20 R21 K43 P45 K53 Y57 A82 K88 A90 T94 I97 A98 T116 K117 E118 L119 S121 R122 N123 N126 Y129 ? 0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHQ5 12464183 5 ~ 1544 DFEEKMILIRRTARMQAGGRRFRFGALVVVGDRQGRVGLGFGKAPEVPLAVQKAGYYARRNMVEVPLQNGTIPHEIEVEFGASKIVLKPAAPGTGVIAGAVPRAILELAGVTDILTKELGSRNPINIAYATMEALRQLRTKADVERLRKG 1n33 F 3.35 BS01 rna A 0 R2 Y50 K54 E69 N73 R87 V90 K92 R2 Y50 K54 E69 N73 R87 V90 K92 ? 0003735,0005737,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLP8 12464183 5 ~ 1544 MRRYEVNIVLNPNLDQSQLALEKEIIQRALENYGARVEKVEELGLRRLAYPIAKDPQGYFLWYQVEMPEDRVNDLARELRIRDNVRRVMVVKSQEPFLANA 1n33 G 3.35 BS01 rna A 0 A2 R3 R4 R6 R10 L12 K29 I30 R32 D33 G34 K35 K36 N37 R41 I42 G81 R94 R95 R102 N109 R114 A116 R119 A1 R2 R3 R5 R9 L11 K28 I29 R31 D32 G33 K34 K35 N36 R40 I41 G80 R93 R94 R101 N108 R113 A115 R118 ? 0000049,0003723,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P17291 12464183 5 ~ 1544 ARRRRAEVRQLQPDLVYGDVLVTAFINKIMRDGKKNLAARIFYDACKIIQEKTGQEPLKVFKQAVENVKPRMEVRSRRVGGANYQVPMEVSPRRQQSLALRWLVQAANQRPERRAAVRIAHELMDAAEGKGGAVKKKEDVERMAEANRAYAHYRW 1n33 H 3.35 BS01 rna A 0 M1 T3 T11 R12 R14 N15 S29 R30 K56 R75 K88 P89 R92 Y94 G96 V97 K98 S113 T114 S115 G128 V129 G130 E132 M1 T3 T11 R12 R14 N15 S29 R30 K56 R75 K88 P89 R92 Y94 G96 V97 K98 S113 T114 S115 G128 V129 G130 E132 ? 0003735,0005737,0005840,0006412,0019843,1990904 remove_due_to_license_issue P0DOY9 12464183 5 ~ 1544 MLTDPIADMLTRIRNATRVYKESTDVPASRFKEEILRILAREGFIKGYERVDVDGKPYLRVYLKYGPRRQGPDPRPEQVIHHIRRISKPGRRVYVGVKEIPRVRRGLGIAILSTSKGVLTDREARKLGVGGELICEVW 1n33 I 3.35 BS01 rna A 0 Q3 Y5 R9 R10 K11 E12 V14 R16 F18 R20 Y36 Q38 G39 G67 G68 G69 K70 S71 Q73 R83 K97 T103 R104 R107 E110 R111 K112 K113 Y114 G115 H117 K118 R120 R121 A122 Q124 Y125 S126 R128 Q2 Y4 R8 R9 K10 E11 V13 R15 F17 R19 Y35 Q37 G38 G66 G67 G68 K69 S70 Q72 R82 K96 T102 R103 R106 E109 R110 K111 K112 Y113 G114 H116 K117 R119 R120 A121 Q123 Y124 S125 R127 ? 0000049,0003723,0003735,0005737,0005840,0006412,0019843,0022627,0043232,1990904 remove_due_to_license_issue P80374 12464183 5 ~ 1544 EQYYGTGRRKEAVARVFLRPGNGKVTVNGQDFNEYFQGLVRAVAALEPLRAVDALGRFDAYITVRGGGKSGQIDAIKLGIARALVQYNPDYRAKLKPLGFLTRDARVVERKKYGKHKARRAPQYSKR 1n33 J 3.35 BS01 rna A 0 R5 R9 H13 S35 G36 P37 I38 P39 L40 P41 T42 R43 V44 R45 R51 G52 F54 K55 H56 K57 R60 H62 H68 D73 R3 R7 H11 S33 G34 P35 I36 P37 L38 P39 T40 R41 V42 R43 R49 G50 F52 K53 H54 K55 R58 H60 H66 D71 ? 0000049,0003723,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q5SHN7 12464183 5 ~ 1544 KIRIKLRGFDHKTLDASAQKIVEAARRSGAQVSGPIPLPTRVRRFTVIRGPFKHKDSREHFELRTHNRLVDIINPNRKTIEQLMTLDLPTGVEIEIKT 1n33 K 3.35 BS01 rna A 0 Y20 N26 N27 I29 T31 G37 N38 P39 I40 W42 G46 G52 S53 K55 R85 P115 H116 N117 C119 R120 K122 K123 K124 Y10 N16 N17 I19 T21 G27 N28 P29 I30 W32 G36 G42 S43 K45 R75 P105 H106 N107 C109 R110 K112 K113 K114 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P80376 12464183 5 ~ 1544 KRQVASGRAYIHASYNNTIVTITDPDGNPITWSSGGVIGYKGSRKGTPYAAQLAALDAAKKAMAYGMQSVDVIVRGTGAGREQAIRALQASGLQVKSIVDDTPVPHNGCRPKKKFRKAS 1n33 L 3.35 BS01 rna A 0 P5 T6 N8 Q9 L10 R12 R15 E16 R19 K20 K21 A30 P31 F32 R33 R34 R41 K46 K47 N49 S50 A51 L52 R53 K54 K57 T61 Y69 P71 E73 R86 K91 D92 P94 R97 V104 R113 K114 K115 S116 R117 S118 K119 T122 K123 K124 P1 T2 N4 Q5 L6 R8 R11 E12 R15 K16 K17 A26 P27 F28 R29 R30 R37 K42 K43 N45 S46 A47 L48 R49 K50 K53 T57 Y65 P67 E69 R82 K87 D88 P90 R93 V100 R109 K110 K111 S112 R113 S114 K115 T118 K119 K120 ? 0000049,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHN3 12464183 5 ~ 1544 PTINQLVRKGREKVRKKSKVPALKGAPFRRGVCTVVRTVTPKKPNSALRKVAKVRLTSGYEVTAYIPGEGHNLQEHSVVLIRGGRVKDLPGVRYHIVRGVYDAAGVKDRKKSRSKYGTKKPKEA 1n33 M 3.35 BS01 rna A 0 K13 R14 V17 Y23 I25 G26 A28 R29 V74 N77 Y87 R88 R91 H92 L96 P97 V98 R99 Q101 R102 T103 R104 T105 N106 A107 R108 T109 R110 K111 R114 K115 T116 K12 R13 V16 Y22 I24 G25 A27 R28 V73 N76 Y86 R87 R90 H91 L95 P96 V97 R98 Q100 R101 T102 R103 T104 N105 A106 R107 T108 R109 K110 R113 K114 T115 ? 0000049,0003676,0003723,0003735,0005829,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P80377 12464183 5 ~ 1544 ARIAGVEIPRNKRVDVALTYIYGIGKARAKEALEKTGINPATRVKDLTEAEVVRLREYVENTWKLEGELRAEVAANIKRLMDIGCYRGLRHRRGLPVRGQRTRTNARTRKGPRKTVAG 1n33 N 3.35 BS01 rna A 0 A2 R3 K4 A5 L6 F16 V18 R19 Y21 R29 R31 S32 V33 R35 R41 I42 R45 K58 S60 W61 A1 R2 K3 A4 L5 F15 V17 R18 Y20 R28 R30 S31 V32 R34 R40 I41 R44 K57 S59 W60 ? 0003735,0005737,0005840,0006412,0008270,0015935,0019843,0046872,1990904 remove_due_to_license_issue P0DOY6 12464183 5 ~ 1544 ARKALIEKAKRTPKFKVRAYTRCVRCGRARSVYRFFGLCRICLRELAHKGQLPGVRKASW 1n33 O 3.35 BS01 rna A 0 P2 K5 K8 T22 G23 S24 Q28 L31 R35 H42 H46 K48 D49 H50 H51 S52 R54 L57 R65 Y69 R72 P1 K4 K7 T21 G22 S23 Q27 L30 R34 H41 H45 K47 D48 H49 H50 S51 R53 L56 R64 Y68 R71 ? 0003735,0005737,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue Q5SJ76 12464183 5 ~ 1544 PITKEEKQKVIQEFARFPGDTGSTEVQVALLTLRINRLSEHLKVHKKDHHSHRGLLMMVGQRRRLLRYLQREDPERYRALIEKLGIRG 1n33 P 3.35 BS01 rna A 0 M1 K3 R5 L6 R8 F9 S11 K12 H13 H16 D23 R25 K27 R28 K31 K35 P41 K43 T44 W59 V62 G63 Q65 T67 T69 R72 R75 R81 Q82 E83 M1 K3 R5 L6 R8 F9 S11 K12 H13 H16 D23 R25 K27 R28 K31 K35 P41 K43 T44 W59 V62 G63 Q65 T67 T69 R72 R75 R81 Q82 E83 ? 0003735,0005737,0005840,0006412,0015935,1990904 remove_due_to_license_issue Q5SJH3 12464183 5 ~ 1544 MVKIRLARFGSKHNPHYRIVVTDARRKRDGKYIEKIGYYDPRKTTPDWLKVDVERARYWLSVGAQPTDTARRLLRQAGVFRQE 1n33 Q 3.35 BS01 rna A 0 P2 K3 S12 K14 M15 Q16 K17 T18 R25 L31 Y32 K34 R38 S39 K40 K41 Y42 E61 S62 R63 P64 I65 S66 K67 R68 K69 R70 R72 R91 N94 Y95 L98 S99 K100 R101 G102 G103 K104 A105 P1 K2 S11 K13 M14 Q15 K16 T17 R24 L30 Y31 K33 R37 S38 K39 K40 Y41 E60 S61 R62 P63 I64 S65 K66 R67 K68 R69 R71 R90 N93 Y94 L97 S98 K99 R100 G101 G102 K103 A104 ? 0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P0DOY7 12464183 5 ~ 1544 PKKVLTGVVVSDKMQKTVTVLVERQFPHPLYGKVIKRSKKYLAHDPEEKYKLGDVVEIIESRPISKRKRFRVLRLVESGRMDLVEKYLIRRQNYQSLSKRGGKA 1n33 R 3.35 BS01 rna A 0 K49 I50 L51 K61 Q63 R64 K68 K71 R72 R74 F81 K34 I35 L36 K46 Q48 R49 K53 K56 R57 R59 F66 ? 0003735,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLQ0 12464183 5 ~ 1544 PSRKAKVKATLGEFDLRDYRNVEVLKRFLSETGKILPRRRTGLSGKEQRILAKTIKRARILGLLPFTEKLVRK 1n33 S 3.35 BS01 rna A 0 P2 S4 K6 F10 H14 W34 R36 R37 Y52 N53 G54 K55 K70 G72 E73 T77 R78 Y80 P1 S3 K5 F9 H13 W33 R35 R36 Y51 N52 G53 K54 K69 G71 E72 T76 R77 Y79 ? 0000028,0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHP2 12464183 5 ~ 1544 PRSLKKGVFVDDHLLEKVLELNAKGEKRLIKTWSRRSTIVPEMVGHTIAVYNGKQHVPVYITENMVGHKLGEFAPTRTYR 1n33 T 3.35 BS01 rna A 0 L10 K14 R15 H16 R17 Q18 S19 R22 R23 R25 N26 K27 K29 S31 K34 T35 K38 K39 R57 E60 S61 D64 K65 K68 S70 K74 N75 R79 K81 S82 R83 M85 R86 R89 G102 G103 L104 S105 L3 K7 R8 H9 R10 Q11 S12 R15 R16 R18 N19 K20 K22 S24 K27 T28 K31 K32 R50 E53 S54 D57 K58 K61 S63 K67 N68 R72 K74 S75 R76 M78 R79 R82 G95 G96 L97 S98 ? 0003723,0003735,0005840,0006412,0015935,0019843,0070181,1990904 remove_due_to_license_issue P80380 12464183 5 ~ 1544 RNLSALKRHRQSLKRRLRNKAKKSAIKTLSKKAIQLAQEGKAEEALKIMRKAESLIDKAAKGSTLHKNAAARRKSRLMRKVRQLLEAAGAPLIGGGLSA 1n34 B 3.8 BS01 rna A 0 K22 W24 P26 N37 L98 G99 T103 N104 R111 K133 R144 I172 E176 K179 K16 W18 P20 N31 L92 G93 T97 N98 R105 K127 R138 I166 E170 K173 ? 0003735,0005840,0006412,0015935,0019843,0022627,1990904 remove_due_to_license_issue P80371 12464183 5 ~ 1544 VKELLEAGVHFGHERKRWNPKFARYIYAERNGIHIIDLQKTMEELERTFRFIEDLAMRGGTILFVGTKKQAQDIVRMEAERAGMPYVNQRWLGGMLTNFKTISQRVHRLEELEALFASPEIEERPKKEQVRLKHELERLQKYLSGFRLLKRLPDAIFVVDPTKEAIAVREARKLFIPVIALADTDSDPDLVDYIIPGNDDAIRSIQLILSRAVDLIIQARGGVVEPSPSYALVQ 1n34 C 3.8 BS01 rna A 0 G2 N3 K4 I5 F10 R127 S154 G155 R156 G159 A160 E161 A163 R172 V173 P174 H176 T177 L178 R179 R190 T191 Y193 G194 V195 L196 K199 G1 N2 K3 I4 F9 R126 S153 G154 R155 G158 A159 E160 A162 R171 V172 P173 H175 T176 L177 R178 R189 T190 Y192 G193 V194 L195 K198 ? 0003676,0003723,0003729,0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P80372 12464183 5 ~ 1544 GNKIHPIGFRLGITRDWESRWYAGKKQYRHLLLEDQRIRGLLEKELYSAGLARVDIERAADNVAVTVHVAKPGVVIGRGGERIRVLREELAKLTGKNVALNVQEVQNPNLSAPLVAQRVAEQIERRFAVRRAIKQAVQRVMESGAKGAKVIVSGRIGGAEQARTEWAAQGRVPLHTLRANIDYGFALARTTYGVLGVKAYIFLGEV 1n34 D 3.8 BS01 rna A 0 G2 R3 I5 P7 V8 C9 R10 R13 R14 E24 R25 K30 R35 R36 Y38 P40 G41 Q42 H43 K46 S52 L58 R59 Q62 R65 S71 E72 R73 S113 R115 Q116 R118 Q119 R122 H123 H125 V133 D134 L135 S137 Y138 L155 E156 S208 R209 G1 R2 I4 P6 V7 C8 R9 R12 R13 E23 R24 K29 R34 R35 Y37 P39 G40 Q41 H42 K45 S51 L57 R58 Q61 R64 S70 E71 R72 S112 R114 Q115 R117 Q118 R121 H122 H124 V132 D133 L134 S136 Y137 L154 E155 S207 R208 ? 0003723,0003735,0005840,0006412,0015935,0019843,0042274,0046872,1990904 remove_due_to_license_issue P80373 12464183 5 ~ 1544 GRYIGPVCRLCRREGVKLYLKGERCYSPKCAMERRPYPPGQHGQKRARRPSDYAVRLREKQKLRRIYGISERQFRNLFEEASKKKGVTGSVFLGLLESRLDNVVYRLGFAVSRRQARQLVRHGHITVNGRRVDLPSYRVRPGDEIAVAEKSRNLELIRQNLEAMKGRKVGPWLSLDVEGMKGKFLRLPDREDLALPVNEQLVIEFYSR 1n34 E 3.8 BS01 rna A 0 T16 A17 R18 M19 Q20 A21 G22 R24 R25 K47 P49 K57 Y60 A86 K92 A94 A95 T98 I101 A102 G103 R107 L119 T120 K121 E122 L123 S125 R126 N127 N130 T12 A13 R14 M15 Q16 A17 G18 R20 R21 K43 P45 K53 Y56 A82 K88 A90 A91 T94 I97 A98 G99 R103 L115 T116 K117 E118 L119 S121 R122 N123 N126 ? 0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHQ5 12464183 5 ~ 1544 DFEEKMILIRRTARMQAGGRRFRFGALVVVGDRQGRVGLGFGKAPEVPLAVQKAGYYARRNMVEVPLQNGTIPHEIEVEFGASKIVLKPAAPGTGVIAGAVPRAILELAGVTDILTKELGSRNPINIAYATMEALRQLRTKADVERLRKG 1n34 F 3.8 BS01 rna A 0 Y4 Y50 K54 N73 R87 V91 K92 Y4 Y50 K54 N73 R87 V91 K92 ? 0003735,0005737,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLP8 12464183 5 ~ 1544 MRRYEVNIVLNPNLDQSQLALEKEIIQRALENYGARVEKVEELGLRRLAYPIAKDPQGYFLWYQVEMPEDRVNDLARELRIRDNVRRVMVVKSQEPFLANA 1n34 G 3.8 BS01 rna A 0 A2 R3 R4 R6 R10 N28 I30 R32 D33 G34 N37 L38 R41 I42 R94 R95 S98 R102 R114 A116 R119 A1 R2 R3 R5 R9 N27 I29 R31 D32 G33 N36 L37 R40 I41 R93 R94 S97 R101 R113 A115 R118 ? 0000049,0003723,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P17291 12464183 5 ~ 1544 ARRRRAEVRQLQPDLVYGDVLVTAFINKIMRDGKKNLAARIFYDACKIIQEKTGQEPLKVFKQAVENVKPRMEVRSRRVGGANYQVPMEVSPRRQQSLALRWLVQAANQRPERRAAVRIAHELMDAAEGKGGAVKKKEDVERMAEANRAYAHYRW 1n34 H 3.8 BS01 rna A 0 M1 T3 P5 T11 R12 R14 N15 S29 R30 F31 K56 K88 P89 G90 R92 Y94 G96 V97 S113 T114 S115 G130 E132 M1 T3 P5 T11 R12 R14 N15 S29 R30 F31 K56 K88 P89 G90 R92 Y94 G96 V97 S113 T114 S115 G130 E132 ? 0003735,0005737,0005840,0006412,0019843,1990904 remove_due_to_license_issue P0DOY9 12464183 5 ~ 1544 MLTDPIADMLTRIRNATRVYKESTDVPASRFKEEILRILAREGFIKGYERVDVDGKPYLRVYLKYGPRRQGPDPRPEQVIHHIRRISKPGRRVYVGVKEIPRVRRGLGIAILSTSKGVLTDREARKLGVGGELICEVW 1n34 I 3.8 BS01 rna A 0 Q3 Y5 T7 R9 K11 E12 V14 R16 F18 R20 Y36 Y62 R66 G68 G69 K70 S71 G72 Q73 R83 K97 T103 R104 R107 V108 V109 E110 R111 K112 K113 Y114 H117 K118 R120 R121 A122 Q124 Y125 S126 R128 Q2 Y4 T6 R8 K10 E11 V13 R15 F17 R19 Y35 Y61 R65 G67 G68 K69 S70 G71 Q72 R82 K96 T102 R103 R106 V107 V108 E109 R110 K111 K112 Y113 H116 K117 R119 R120 A121 Q123 Y124 S125 R127 ? 0000049,0003723,0003735,0005737,0005840,0006412,0019843,0022627,0043232,1990904 remove_due_to_license_issue P80374 12464183 5 ~ 1544 EQYYGTGRRKEAVARVFLRPGNGKVTVNGQDFNEYFQGLVRAVAALEPLRAVDALGRFDAYITVRGGGKSGQIDAIKLGIARALVQYNPDYRAKLKPLGFLTRDARVVERKKYGKHKARRAPQYSKR 1n34 J 3.8 BS01 rna A 0 R5 R9 H13 S35 G36 P37 I38 L40 P41 T42 R43 V44 R45 T48 I50 R51 G52 P53 F54 K55 H56 K57 H62 H68 D73 R3 R7 H11 S33 G34 P35 I36 L38 P39 T40 R41 V42 R43 T46 I48 R49 G50 P51 F52 K53 H54 K55 H60 H66 D71 ? 0000049,0003723,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q5SHN7 12464183 5 ~ 1544 KIRIKLRGFDHKTLDASAQKIVEAARRSGAQVSGPIPLPTRVRRFTVIRGPFKHKDSREHFELRTHNRLVDIINPNRKTIEQLMTLDLPTGVEIEIKT 1n34 K 3.8 BS01 rna A 0 Y20 N26 N27 I29 T31 P39 I40 W42 S44 G45 G46 G52 S53 K55 R85 V114 P115 H116 N117 C119 R120 K122 K123 Y10 N16 N17 I19 T21 P29 I30 W32 S34 G35 G36 G42 S43 K45 R75 V104 P105 H106 N107 C109 R110 K112 K113 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P80376 12464183 5 ~ 1544 KRQVASGRAYIHASYNNTIVTITDPDGNPITWSSGGVIGYKGSRKGTPYAAQLAALDAAKKAMAYGMQSVDVIVRGTGAGREQAIRALQASGLQVKSIVDDTPVPHNGCRPKKKFRKAS 1n34 L 3.8 BS01 rna A 0 P5 T6 N8 Q9 R12 K13 R15 E16 K17 R19 K20 K28 G29 A30 P31 F32 R33 R34 K47 N49 S50 L52 R53 K54 T61 Y69 P71 E73 R86 R89 D92 R97 R113 K114 K115 S116 R117 S118 K119 G121 T122 K123 K124 P1 T2 N4 Q5 R8 K9 R11 E12 K13 R15 K16 K24 G25 A26 P27 F28 R29 R30 K43 N45 S46 L48 R49 K50 T57 Y65 P67 E69 R82 R85 D88 R93 R109 K110 K111 S112 R113 S114 K115 G117 T118 K119 K120 ? 0000049,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHN3 12464183 5 ~ 1544 PTINQLVRKGREKVRKKSKVPALKGAPFRRGVCTVVRTVTPKKPNSALRKVAKVRLTSGYEVTAYIPGEGHNLQEHSVVLIRGGRVKDLPGVRYHIVRGVYDAAGVKDRKKSRSKYGTKKPKEA 1n34 M 3.8 BS01 rna A 0 R14 Y23 I25 G26 K27 A28 R29 R44 N77 I78 Y87 R91 H92 V98 R99 Q101 R102 T103 R104 N106 R108 T109 R110 K111 R114 K115 T116 G119 R13 Y22 I24 G25 K26 A27 R28 R43 N76 I77 Y86 R90 H91 V97 R98 Q100 R101 T102 R103 N105 R107 T108 R109 K110 R113 K114 T115 G118 ? 0000049,0003676,0003723,0003735,0005829,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P80377 12464183 5 ~ 1544 ARIAGVEIPRNKRVDVALTYIYGIGKARAKEALEKTGINPATRVKDLTEAEVVRLREYVENTWKLEGELRAEVAANIKRLMDIGCYRGLRHRRGLPVRGQRTRTNARTRKGPRKTVAG 1n34 N 3.8 BS01 rna A 0 R3 K4 A5 L6 E8 K15 F16 K17 V18 R19 Y21 T22 C27 R29 A30 R31 S32 Y34 R35 R41 I42 R45 K58 S60 W61 R2 K3 A4 L5 E7 K14 F15 K16 V17 R18 Y20 T21 C26 R28 A29 R30 S31 Y33 R34 R40 I41 R44 K57 S59 W60 ? 0003735,0005737,0005840,0006412,0008270,0015935,0019843,0046872,1990904 remove_due_to_license_issue P0DOY6 12464183 5 ~ 1544 ARKALIEKAKRTPKFKVRAYTRCVRCGRARSVYRFFGLCRICLRELAHKGQLPGVRKASW 1n34 O 3.8 BS01 rna A 0 P2 K5 K8 F18 D21 T22 G23 S24 T25 Q28 R35 L39 H42 H46 K48 D49 H50 H51 S52 R54 L57 Y69 R72 P1 K4 K7 F17 D20 T21 G22 S23 T24 Q27 R34 L38 H41 H45 K47 D48 H49 H50 S51 R53 L56 Y68 R71 ? 0003735,0005737,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue Q5SJ76 12464183 5 ~ 1544 PITKEEKQKVIQEFARFPGDTGSTEVQVALLTLRINRLSEHLKVHKKDHHSHRGLLMMVGQRRRLLRYLQREDPERYRALIEKLGIRG 1n34 P 3.8 BS01 rna A 0 M1 V2 K3 R5 L6 R8 F9 G10 S11 K12 H13 H16 Y17 R18 D23 R25 K27 R28 K31 I33 K35 K43 W59 V62 G63 T67 T69 R72 R75 F80 R81 Q82 M1 V2 K3 R5 L6 R8 F9 G10 S11 K12 H13 H16 Y17 R18 D23 R25 K27 R28 K31 I33 K35 K43 W59 V62 G63 T67 T69 R72 R75 F80 R81 Q82 ? 0003735,0005737,0005840,0006412,0015935,1990904 remove_due_to_license_issue Q5SJH3 12464183 5 ~ 1544 MVKIRLARFGSKHNPHYRIVVTDARRKRDGKYIEKIGYYDPRKTTPDWLKVDVERARYWLSVGAQPTDTARRLLRQAGVFRQE 1n34 Q 3.8 BS01 rna A 0 P2 K3 S12 M15 Q16 K17 R25 L31 Y32 K34 S39 K40 K41 Y42 E61 S62 R63 P64 I65 S66 K67 R68 K69 R70 R72 K87 N94 Y95 L98 S99 K100 R101 G102 G103 K104 A105 P1 K2 S11 M14 Q15 K16 R24 L30 Y31 K33 S38 K39 K40 Y41 E60 S61 R62 P63 I64 S65 K66 R67 K68 R69 R71 K86 N93 Y94 L97 S98 K99 R100 G101 G102 K103 A104 ? 0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P0DOY7 12464183 5 ~ 1544 PKKVLTGVVVSDKMQKTVTVLVERQFPHPLYGKVIKRSKKYLAHDPEEKYKLGDVVEIIESRPISKRKRFRVLRLVESGRMDLVEKYLIRRQNYQSLSKRGGKA 1n34 R 3.8 BS01 rna A 0 K49 I50 K61 Q63 R64 K68 K71 R72 R74 I75 F81 K34 I35 K46 Q48 R49 K53 K56 R57 R59 I60 F66 ? 0003735,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLQ0 12464183 5 ~ 1544 PSRKAKVKATLGEFDLRDYRNVEVLKRFLSETGKILPRRRTGLSGKEQRILAKTIKRARILGLLPFTEKLVRK 1n34 S 3.8 BS01 rna A 0 P2 R3 S4 K6 F10 W34 R36 R37 Y52 N53 G54 K55 G72 E73 T77 R78 Y80 P1 R2 S3 K5 F9 W33 R35 R36 Y51 N52 G53 K54 G71 E72 T76 R77 Y79 ? 0000028,0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHP2 12464183 5 ~ 1544 PRSLKKGVFVDDHLLEKVLELNAKGEKRLIKTWSRRSTIVPEMVGHTIAVYNGKQHVPVYITENMVGHKLGEFAPTRTYR 1n34 T 3.8 BS01 rna A 0 L10 K14 R15 H16 R17 Q18 R22 R23 N26 K27 A28 S31 T35 K38 K39 E60 S61 K65 K68 S70 K74 A78 R79 K81 S82 R83 M85 R89 G102 G103 L104 S105 L3 K7 R8 H9 R10 Q11 R15 R16 N19 K20 A21 S24 T28 K31 K32 E53 S54 K58 K61 S63 K67 A71 R72 K74 S75 R76 M78 R82 G95 G96 L97 S98 ? 0003723,0003735,0005840,0006412,0015935,0019843,0070181,1990904 remove_due_to_license_issue P80380 12464183 5 ~ 1544 RNLSALKRHRQSLKRRLRNKAKKSAIKTLSKKAIQLAQEGKAEEALKIMRKAESLIDKAAKGSTLHKNAAARRKSRLMRKVRQLLEAAGAPLIGGGLSA 1n36 B 3.65 BS01 rna A 0 W24 N37 G99 T103 N104 R111 K133 I172 E176 K179 W18 N31 G93 T97 N98 R105 K127 I166 E170 K173 ? 0003735,0005840,0006412,0015935,0019843,0022627,1990904 remove_due_to_license_issue P80371 12464183 5 ~ 1544 VKELLEAGVHFGHERKRWNPKFARYIYAERNGIHIIDLQKTMEELERTFRFIEDLAMRGGTILFVGTKKQAQDIVRMEAERAGMPYVNQRWLGGMLTNFKTISQRVHRLEELEALFASPEIEERPKKEQVRLKHELERLQKYLSGFRLLKRLPDAIFVVDPTKEAIAVREARKLFIPVIALADTDSDPDLVDYIIPGNDDAIRSIQLILSRAVDLIIQARGGVVEPSPSYALVQ 1n36 C 3.65 BS01 rna A 0 G2 N3 K4 I5 R127 S154 G155 R156 G158 G159 E161 A163 R172 V173 P174 H176 T177 L178 R179 F186 T191 Y193 G194 V195 G1 N2 K3 I4 R126 S153 G154 R155 G157 G158 E160 A162 R171 V172 P173 H175 T176 L177 R178 F185 T190 Y192 G193 V194 ? 0003676,0003723,0003729,0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P80372 12464183 5 ~ 1544 GNKIHPIGFRLGITRDWESRWYAGKKQYRHLLLEDQRIRGLLEKELYSAGLARVDIERAADNVAVTVHVAKPGVVIGRGGERIRVLREELAKLTGKNVALNVQEVQNPNLSAPLVAQRVAEQIERRFAVRRAIKQAVQRVMESGAKGAKVIVSGRIGGAEQARTEWAAQGRVPLHTLRANIDYGFALARTTYGVLGVKAYIFLGEV 1n36 D 3.65 BS01 rna A 0 G2 R3 I5 P7 V8 C9 R10 R13 R14 E24 R25 K30 R36 Y38 G41 H43 Q45 K46 S52 Y54 R59 Q62 E72 R73 Q74 K84 R115 Q116 R118 Q119 R122 H123 H125 V133 L135 S137 Y138 R209 G1 R2 I4 P6 V7 C8 R9 R12 R13 E23 R24 K29 R35 Y37 G40 H42 Q44 K45 S51 Y53 R58 Q61 E71 R72 Q73 K83 R114 Q115 R117 Q118 R121 H122 H124 V132 L134 S136 Y137 R208 ? 0003723,0003735,0005840,0006412,0015935,0019843,0042274,0046872,1990904 remove_due_to_license_issue P80373 12464183 5 ~ 1544 GRYIGPVCRLCRREGVKLYLKGERCYSPKCAMERRPYPPGQHGQKRARRPSDYAVRLREKQKLRRIYGISERQFRNLFEEASKKKGVTGSVFLGLLESRLDNVVYRLGFAVSRRQARQLVRHGHITVNGRRVDLPSYRVRPGDEIAVAEKSRNLELIRQNLEAMKGRKVGPWLSLDVEGMKGKFLRLPDREDLALPVNEQLVIEFYSR 1n36 E 3.65 BS01 rna A 0 R14 T16 A17 R18 M19 Q20 A21 G22 R24 R25 R27 P49 K57 A86 A95 T98 I101 A102 G103 T120 K121 E122 L123 S125 R126 N127 N130 R10 T12 A13 R14 M15 Q16 A17 G18 R20 R21 R23 P45 K53 A82 A91 T94 I97 A98 G99 T116 K117 E118 L119 S121 R122 N123 N126 ? 0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHQ5 12464183 5 ~ 1544 DFEEKMILIRRTARMQAGGRRFRFGALVVVGDRQGRVGLGFGKAPEVPLAVQKAGYYARRNMVEVPLQNGTIPHEIEVEFGASKIVLKPAAPGTGVIAGAVPRAILELAGVTDILTKELGSRNPINIAYATMEALRQLRTKADVERLRKG 1n36 F 3.65 BS01 rna A 0 Y4 Y50 K54 E69 N73 R80 R87 V90 V91 K92 Y4 Y50 K54 E69 N73 R80 R87 V90 V91 K92 ? 0003735,0005737,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLP8 12464183 5 ~ 1544 MRRYEVNIVLNPNLDQSQLALEKEIIQRALENYGARVEKVEELGLRRLAYPIAKDPQGYFLWYQVEMPEDRVNDLARELRIRDNVRRVMVVKSQEPFLANA 1n36 G 3.65 BS01 rna A 0 A2 R3 R4 R6 R10 I30 R32 D33 G34 K35 K36 N37 L38 R41 R94 R95 S98 R102 N109 R114 R115 A116 R119 A1 R2 R3 R5 R9 I29 R31 D32 G33 K34 K35 N36 L37 R40 R93 R94 S97 R101 N108 R113 R114 A115 R118 ? 0000049,0003723,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P17291 12464183 5 ~ 1544 ARRRRAEVRQLQPDLVYGDVLVTAFINKIMRDGKKNLAARIFYDACKIIQEKTGQEPLKVFKQAVENVKPRMEVRSRRVGGANYQVPMEVSPRRQQSLALRWLVQAANQRPERRAAVRIAHELMDAAEGKGGAVKKKEDVERMAEANRAYAHYRW 1n36 H 3.65 BS01 rna A 0 M1 T3 D8 T11 R12 R14 N15 K21 S29 R30 F31 K56 R75 K88 P89 G90 R92 Y94 G96 V97 S113 T114 S115 G130 E132 M1 T3 D8 T11 R12 R14 N15 K21 S29 R30 F31 K56 R75 K88 P89 G90 R92 Y94 G96 V97 S113 T114 S115 G130 E132 ? 0003735,0005737,0005840,0006412,0019843,1990904 remove_due_to_license_issue P0DOY9 12464183 5 ~ 1544 MLTDPIADMLTRIRNATRVYKESTDVPASRFKEEILRILAREGFIKGYERVDVDGKPYLRVYLKYGPRRQGPDPRPEQVIHHIRRISKPGRRVYVGVKEIPRVRRGLGIAILSTSKGVLTDREARKLGVGGELICEVW 1n36 I 3.65 BS01 rna A 0 E2 Q3 Y5 T7 R9 R10 K11 E12 V14 F18 R20 Q38 Y62 R66 G67 G68 G69 K70 S71 Q73 T103 R104 R107 V108 V109 E110 R111 K112 K113 Y114 H117 K118 R120 R121 A122 P123 Q124 Y125 R128 E1 Q2 Y4 T6 R8 R9 K10 E11 V13 F17 R19 Q37 Y61 R65 G66 G67 G68 K69 S70 Q72 T102 R103 R106 V107 V108 E109 R110 K111 K112 Y113 H116 K117 R119 R120 A121 P122 Q123 Y124 R127 ? 0000049,0003723,0003735,0005737,0005840,0006412,0019843,0022627,0043232,1990904 remove_due_to_license_issue P80374 12464183 5 ~ 1544 EQYYGTGRRKEAVARVFLRPGNGKVTVNGQDFNEYFQGLVRAVAALEPLRAVDALGRFDAYITVRGGGKSGQIDAIKLGIARALVQYNPDYRAKLKPLGFLTRDARVVERKKYGKHKARRAPQYSKR 1n36 J 3.65 BS01 rna A 0 R5 K7 H13 S35 G36 P37 P39 L40 P41 T42 R43 V44 I50 R51 F54 K55 H56 K57 S59 R60 H62 H68 R3 K5 H11 S33 G34 P35 P37 L38 P39 T40 R41 V42 I48 R49 F52 K53 H54 K55 S57 R58 H60 H66 ? 0000049,0003723,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q5SHN7 12464183 5 ~ 1544 KIRIKLRGFDHKTLDASAQKIVEAARRSGAQVSGPIPLPTRVRRFTVIRGPFKHKDSREHFELRTHNRLVDIINPNRKTIEQLMTLDLPTGVEIEIKT 1n36 K 3.65 BS01 rna A 0 Y20 N26 N27 I29 T31 N38 P39 W42 S44 G46 V47 K51 G52 S53 K55 V114 P115 H116 N117 G118 C119 R120 K123 Y10 N16 N17 I19 T21 N28 P29 W32 S34 G36 V37 K41 G42 S43 K45 V104 P105 H106 N107 G108 C109 R110 K113 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P80376 12464183 5 ~ 1544 KRQVASGRAYIHASYNNTIVTITDPDGNPITWSSGGVIGYKGSRKGTPYAAQLAALDAAKKAMAYGMQSVDVIVRGTGAGREQAIRALQASGLQVKSIVDDTPVPHNGCRPKKKFRKAS 1n36 L 3.65 BS01 rna A 0 P5 T6 N8 Q9 L10 R12 K13 R15 E16 K20 G29 P31 F32 R33 R34 K46 K47 N49 S50 L52 R53 K54 T61 Y69 P71 E73 R86 V90 K91 D92 R97 V104 R113 K114 K115 S116 R117 S118 K119 Y120 K123 K124 P1 T2 N4 Q5 L6 R8 K9 R11 E12 K16 G25 P27 F28 R29 R30 K42 K43 N45 S46 L48 R49 K50 T57 Y65 P67 E69 R82 V86 K87 D88 R93 V100 R109 K110 K111 S112 R113 S114 K115 Y116 K119 K120 ? 0000049,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHN3 12464183 5 ~ 1544 PTINQLVRKGREKVRKKSKVPALKGAPFRRGVCTVVRTVTPKKPNSALRKVAKVRLTSGYEVTAYIPGEGHNLQEHSVVLIRGGRVKDLPGVRYHIVRGVYDAAGVKDRKKSRSKYGTKKPKEA 1n36 M 3.65 BS01 rna A 0 R14 Y23 G24 I25 G26 A28 R29 R44 N77 R88 R91 H92 P97 R99 R102 T103 R104 T105 N106 A107 R108 T109 K111 K115 T116 R13 Y22 G23 I24 G25 A27 R28 R43 N76 R87 R90 H91 P96 R98 R101 T102 R103 T104 N105 A106 R107 T108 K110 K114 T115 ? 0000049,0003676,0003723,0003735,0005829,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P80377 12464183 5 ~ 1544 ARIAGVEIPRNKRVDVALTYIYGIGKARAKEALEKTGINPATRVKDLTEAEVVRLREYVENTWKLEGELRAEVAANIKRLMDIGCYRGLRHRRGLPVRGQRTRTNARTRKGPRKTVAG 1n36 N 3.65 BS01 rna A 0 A2 R3 K4 K17 V18 R19 Y21 T22 R23 R29 A30 R31 R35 R41 I42 R45 K58 S60 W61 A1 R2 K3 K16 V17 R18 Y20 T21 R22 R28 A29 R30 R34 R40 I41 R44 K57 S59 W60 ? 0003735,0005737,0005840,0006412,0008270,0015935,0019843,0046872,1990904 remove_due_to_license_issue P0DOY6 12464183 5 ~ 1544 ARKALIEKAKRTPKFKVRAYTRCVRCGRARSVYRFFGLCRICLRELAHKGQLPGVRKASW 1n36 O 3.65 BS01 rna A 0 P2 K5 K8 F18 D21 T22 G23 S24 Q28 L31 R35 L39 H42 H46 D49 H51 S52 R54 G55 L57 M58 R65 Y69 R72 P1 K4 K7 F17 D20 T21 G22 S23 Q27 L30 R34 L38 H41 H45 D48 H50 S51 R53 G54 L56 M57 R64 Y68 R71 ? 0003735,0005737,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue Q5SJ76 12464183 5 ~ 1544 PITKEEKQKVIQEFARFPGDTGSTEVQVALLTLRINRLSEHLKVHKKDHHSHRGLLMMVGQRRRLLRYLQREDPERYRALIEKLGIRG 1n36 P 3.65 BS01 rna A 0 M1 V2 K3 R5 L6 F9 S11 K12 H13 H16 Y17 R18 D23 A24 R25 R26 K27 R28 G30 K31 I33 K35 Y38 P41 K43 T44 V62 G63 Q65 T67 T69 R72 R75 R81 Q82 M1 V2 K3 R5 L6 F9 S11 K12 H13 H16 Y17 R18 D23 A24 R25 R26 K27 R28 G30 K31 I33 K35 Y38 P41 K43 T44 V62 G63 Q65 T67 T69 R72 R75 R81 Q82 ? 0003735,0005737,0005840,0006412,0015935,1990904 remove_due_to_license_issue Q5SJH3 12464183 5 ~ 1544 MVKIRLARFGSKHNPHYRIVVTDARRKRDGKYIEKIGYYDPRKTTPDWLKVDVERARYWLSVGAQPTDTARRLLRQAGVFRQE 1n36 Q 3.65 BS01 rna A 0 P2 K3 K14 M15 Q16 K17 R25 L31 Y32 R38 S39 K40 K41 Y42 E61 S62 R63 P64 S66 K67 R68 K69 R70 R72 K87 N94 Y95 L98 S99 K100 R101 G102 G103 K104 A105 P1 K2 K13 M14 Q15 K16 R24 L30 Y31 R37 S38 K39 K40 Y41 E60 S61 R62 P63 S65 K66 R67 K68 R69 R71 K86 N93 Y94 L97 S98 K99 R100 G101 G102 K103 A104 ? 0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P0DOY7 12464183 5 ~ 1544 PKKVLTGVVVSDKMQKTVTVLVERQFPHPLYGKVIKRSKKYLAHDPEEKYKLGDVVEIIESRPISKRKRFRVLRLVESGRMDLVEKYLIRRQNYQSLSKRGGKA 1n36 R 3.65 BS01 rna A 0 K49 I50 K61 Q63 R64 K68 K71 R72 R74 I75 F81 K34 I35 K46 Q48 R49 K53 K56 R57 R59 I60 F66 ? 0003735,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLQ0 12464183 5 ~ 1544 PSRKAKVKATLGEFDLRDYRNVEVLKRFLSETGKILPRRRTGLSGKEQRILAKTIKRARILGLLPFTEKLVRK 1n36 S 3.65 BS01 rna A 0 P2 R3 S4 K6 F10 H14 K32 T33 W34 R36 R37 Y52 N53 G54 K55 G72 E73 T77 R78 T79 Y80 P1 R2 S3 K5 F9 H13 K31 T32 W33 R35 R36 Y51 N52 G53 K54 G71 E72 T76 R77 T78 Y79 ? 0000028,0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHP2 12464183 5 ~ 1544 PRSLKKGVFVDDHLLEKVLELNAKGEKRLIKTWSRRSTIVPEMVGHTIAVYNGKQHVPVYITENMVGHKLGEFAPTRTYR 1n36 T 3.65 BS01 rna A 0 L10 K14 H16 R17 S19 K21 R22 R23 N26 S31 K34 T35 K38 K39 R57 E60 S61 K65 K68 S70 K74 N75 A78 R79 K81 S82 R83 M85 R89 G102 G103 L104 S105 L3 K7 H9 R10 S12 K14 R15 R16 N19 S24 K27 T28 K31 K32 R50 E53 S54 K58 K61 S63 K67 N68 A71 R72 K74 S75 R76 M78 R82 G95 G96 L97 S98 ? 0003723,0003735,0005840,0006412,0015935,0019843,0070181,1990904 remove_due_to_license_issue P80380 12464183 5 ~ 1544 RNLSALKRHRQSLKRRLRNKAKKSAIKTLSKKAIQLAQEGKAEEALKIMRKAESLIDKAAKGSTLHKNAAARRKSRLMRKVRQLLEAAGAPLIGGGLSA 1n3c A 2.7 BS01 dna B 0 N149 R154 G202 Y203 R204 Q287 A288 N138 R143 G191 Y192 R193 Q276 A277 3.2.2.-,4.2.99.18 0000978,0003677,0003684,0003824,0004519,0005515,0005634,0005654,0005739,0005759,0005829,0006281,0006284,0006285,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045007,0045008,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O15527 12578369 1 ~ 15 GSEGHRTLASTPALWASIPCPRSELRLDLVLPSGQSFRWREQSPAHWSGVLADQVWTLTQTEEQLHCTVYRSQASRPTPDELEAVRKYFQLDVTLAQLYHHWGSVDSHFQEVAQKFQGVRLLRQDPIECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPSLQALAGPEVEAHLRKLGLGYRARYVSASARAILEEQGGLAWLQQLRESSYEEAHKALCILPGVGTKVADCICLMALDKPQAVPVNVHMWHIAQRDYSWHPTTSQAKGPSPQTNKELGNFFRSLWGPYAGWAQAVLFSADLRQ 1n3c A 2.7 BS02 dna C 0 G42 S147 S148 N149 N150 N151 I152 Y207 P244 G245 G247 K249 V250 N268 H270 Q315 F319 G34 S136 S137 N138 N139 N140 I141 Y196 P233 G234 G236 K238 V239 N257 H259 Q304 F308 3.2.2.-,4.2.99.18 0000978,0003677,0003684,0003824,0004519,0005515,0005634,0005654,0005739,0005759,0005829,0006281,0006284,0006285,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045007,0045008,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O15527 12578369 16 ~ 30 GSEGHRTLASTPALWASIPCPRSELRLDLVLPSGQSFRWREQSPAHWSGVLADQVWTLTQTEEQLHCTVYRSQASRPTPDELEAVRKYFQLDVTLAQLYHHWGSVDSHFQEVAQKFQGVRLLRQDPIECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPSLQALAGPEVEAHLRKLGLGYRARYVSASARAILEEQGGLAWLQQLRESSYEEAHKALCILPGVGTKVADCICLMALDKPQAVPVNVHMWHIAQRDYSWHPTTSQAKGPSPQTNKELGNFFRSLWGPYAGWAQAVLFSADLRQ 1n3i A 1.9 BS02 DIH A 1 Y92 A120 A121 G122 Y188 E189 V205 M207 N231 H243 Y86 A114 A115 G116 Y182 E183 V199 M201 N225 H237 H68 H90 Y92 E93 A120 M207 S208 N231 A233 H243 H62 H84 Y86 E87 A114 M201 S202 N225 A227 H237 6.3.2.1 0003824,0004731,0006139,0009116,0016763 Kd=1.3nM remove_due_to_license_issue P9WIL5 12755607 401 DPDELARRAAQVIADRTGIGEHDVAVVLGSGWLPAVAALGSPTTVLPQAELPGFVPPTAAGHAGELLSVPIGAHRVLVLAGRIHAYEGHDLRYVVHPVRAARAAGAQIMVLTNAAGGLRADLQVGQPVLISDHLNLTARSPLVGGEFVDLTDAYSPRLRELARQSDPQLAEGVYAGLPGPHYETPAEIRMLQTLGADLVGMSTVHETIAARAAGAEVLGVSLVTNLAAGITGEPLSHAEVLAAGAASATRMGALLADVIARF 1n3i B 1.9 BS02 DIH B 1 Y92 A120 A121 G122 Y188 E189 V205 M207 N231 H243 Y86 A114 A115 G116 Y182 E183 V199 M201 N225 H237 H68 H90 Y92 E93 A120 M207 S208 N231 A233 H243 H62 H84 Y86 E87 A114 M201 S202 N225 A227 H237 6.3.2.1 0003824,0004731,0006139,0009116,0016763 Kd=1.3nM remove_due_to_license_issue P9WIL5 12755607 402 DPDELARRAAQVIADRTGIGEHDVAVVLGSGWLPAVAALGSPTTVLPQAELPGFVPPTAAGHAGELLSVPIGAHRVLVLAGRIHAYEGHDLRYVVHPVRAARAAGAQIMVLTNAAGGLRADLQVGQPVLISDHLNLTARSPLVGGEFVDLTDAYSPRLRELARQSDPQLAEGVYAGLPGPHYETPAEIRMLQTLGADLVGMSTVHETIAARAAGAEVLGVSLVTNLAAGITGEPLSHAEVLAAGAASATRMGALLADVIARF 1n3z A 1.65 BS01 U3P A 1 K41 N44 T45 F120 K36 N39 T40 F115 H12 K41 H119 F120 D121 H12 K36 H114 F115 D116 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 remove_due_to_license_issue Ki=63200nM P00669 12833549 125 KESAAAKFERQHMDSGSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 1n43 A 1.89 BS01 BTN A 1 S27 Y43 S45 V47 N49 W79 T90 W108 D128 S12 Y28 S30 V32 N34 W64 T75 W93 D113 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 12925786 5100 GITGTWYAQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTK 1n43 D 1.89 BS01 BTN D 1 L25 S27 Y43 S45 V47 G48 N49 W79 S88 T90 W108 D128 L10 S12 Y28 S30 V32 G33 N34 W64 S73 T75 W93 D113 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 12925786 5400 GITGTWYAQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1n46 A 2.2 BS01 PFA A 1 I276 A279 R282 M310 M313 R316 A317 R320 L330 N331 L346 H435 M442 F455 I63 A66 R69 M97 M100 R103 A104 R107 L117 N118 L133 H222 M229 F242 ? 0003677,0004879,0006355 Ki=0.03nM remove_due_to_license_issue P10828 12565933 462 KPEPTDEEWELIKTVTEAHVATNAQWKQKRKFLPEDIGQAPIVNAPEGGKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 1n4h A 2.1 BS02 REA A 1 Q21 C55 V96 M100 A135 Q21 C55 V96 M100 A135 ? 0003677,0004879,0005634,0006355 Kd=280nM remove_due_to_license_issue P45446 12958591 500 TMSEIDRIAQNIIKSHLETCQYTMEELHQLAWQTHTYEEIKAYQSKSREALWQQCAIQITHAIQYVVEFAKRITGFMELCQNDQILLLKSGCLEVVLVRMCRAFNPLNNTVLFEGKYGGMQMFKALGSDDLVNEAFDFAKNLCSLQLTEEEIALFSSAVLISPDRAWLLEPRKVQKLQEKIYFALQHVIQKNHLDDETLAKLIAKIPTITAVCNLHGEKLQVFKQSHPDIVNTLFPPLYKELFN 1n4k A 2.2 BS01 I3P A 1 R265 T267 G268 R269 K508 Y567 R568 K569 R30 T32 G33 R34 K215 Y257 R258 K259 ? 0005220,0005262,0005783,0006816,0016020,0070588,0070679 Kd=0.09nM remove_due_to_license_issue P11881 12442173 1000 GGDVVRLFHAEQEKFLTCDEHRKKQHVFLRTTGRQSATSATSSKALWEVEVVQLFRFKHLATGHYLAAEVDMVYSLVSVPEGNDISSIFELDPYVRLRHLCTNTWVHSTNIPIDKEEEKPVMLKIGTSPLKEDKEAFAIVPVSPAEVRDLDFANDASKVLGSIAGKLEKGTITQNERRSVTKLLEDLVYFVTGGTNSGQDVLEVVFSKPNRERQKLMREQNILKQIFKLLQAPFTHAPFRHICRLCYRVLRHSQQDYRKNQEYIAKQFGFMQKQIGYDVLAEDTITALLHNN 1n5r A 2.25 BS01 PRM A 1 Y72 W286 H287 S293 Y72 W280 H281 S287 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Ki=2.2uM remove_due_to_license_issue P21836 12505979 951 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 1n77 A 2.4 BS01 rna C 0 E41 D44 R47 L112 R116 V145 R163 E172 V177 K180 S181 Y187 E207 E208 W209 L210 V211 R237 K241 K243 G274 E282 R297 S299 P303 V304 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 E41 D44 R47 L112 R116 V145 R163 E172 V177 K180 S181 Y187 E207 E208 W209 L210 V211 R237 K241 K243 G274 E282 R297 S299 P303 V304 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 K246 K246 6.1.1.17 0000049,0000166,0004812,0004818,0005524,0005737,0005829,0006412,0006418,0006424,0008270,0043039 remove_due_to_license_issue P27000 12554668 501 ~ 576 MVVTRIAPSPTGDPHVGTAYIALFNYAWARRNGGRFIVRIEDTDRARYVPGAEERILAALKWLGLSYDEGPDVGGPHGPYRQSERLPLYQKYAEELLKRGWAYRAFETPEELEQIRKEKGGYDGRARNIPPEEAEERARRGEPHVIRLKVPRPGTTEVKDELRGVVVYDNQEIPDVVLLKSDGYPTYHLANVVDDHLMGVTDVIRAEEWLVSTPIHVLLYRAFGWEAPRFYHMPLLRNPDKTKISKRKSHTSLDWYKAEGFLPEALRNYLCLMGFSMPDGREIFTLEEFIQAFTWERVSLGGPVFDLEKLRWMNGKYIREVLSLEEVAERVKPFLREAGLSWESEAYLRRAVELMRPRFDTLKEFPEKARYLFTEDYPVSEKAQRKLEEGLPLLKELYPRLRAQEEWTEAALEALLRGFAAEKGVKLGQVAQPLRAALTGSLETPGLFEILALLGKERALRRLERALA 1n77 B 2.4 BS01 rna D 0 E41 L112 R116 V145 R163 V166 Y168 E172 V177 K180 S181 Y187 E207 E208 W209 L210 V211 R237 K241 T242 K243 G274 E282 R297 S299 L300 G301 P303 V304 E308 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 E41 L112 R116 V145 R163 V166 Y168 E172 V177 K180 S181 Y187 E207 E208 W209 L210 V211 R237 K241 T242 K243 G274 E282 R297 S299 L300 G301 P303 V304 E308 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 K246 K246 6.1.1.17 0000049,0000166,0004812,0004818,0005524,0005737,0005829,0006412,0006418,0006424,0008270,0043039 remove_due_to_license_issue P27000 12554668 501 ~ 576 MVVTRIAPSPTGDPHVGTAYIALFNYAWARRNGGRFIVRIEDTDRARYVPGAEERILAALKWLGLSYDEGPDVGGPHGPYRQSERLPLYQKYAEELLKRGWAYRAFETPEELEQIRKEKGGYDGRARNIPPEEAEERARRGEPHVIRLKVPRPGTTEVKDELRGVVVYDNQEIPDVVLLKSDGYPTYHLANVVDDHLMGVTDVIRAEEWLVSTPIHVLLYRAFGWEAPRFYHMPLLRNPDKTKISKRKSHTSLDWYKAEGFLPEALRNYLCLMGFSMPDGREIFTLEEFIQAFTWERVSLGGPVFDLEKLRWMNGKYIREVLSLEEVAERVKPFLREAGLSWESEAYLRRAVELMRPRFDTLKEFPEKARYLFTEDYPVSEKAQRKLEEGLPLLKELYPRLRAQEEWTEAALEALLRGFAAEKGVKLGQVAQPLRAALTGSLETPGLFEILALLGKERALRRLERALA 1n78 A 2.1 BS01 rna C 0 S9 T43 D44 R47 V145 R163 V166 Y168 E172 V177 K180 S181 Y187 E207 E208 W209 L210 V211 R237 K241 M273 G274 E282 R297 P303 V304 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 S9 T43 D44 R47 V145 R163 V166 Y168 E172 V177 K180 S181 Y187 E207 E208 W209 L210 V211 R237 K241 M273 G274 E282 R297 P303 V304 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 K246 K246 6.1.1.17 0000049,0000166,0004812,0004818,0005524,0005737,0005829,0006412,0006418,0006424,0008270,0043039 remove_due_to_license_issue P27000 12554668 501 ~ 576 MVVTRIAPSPTGDPHVGTAYIALFNYAWARRNGGRFIVRIEDTDRARYVPGAEERILAALKWLGLSYDEGPDVGGPHGPYRQSERLPLYQKYAEELLKRGWAYRAFETPEELEQIRKEKGGYDGRARNIPPEEAEERARRGEPHVIRLKVPRPGTTEVKDELRGVVVYDNQEIPDVVLLKSDGYPTYHLANVVDDHLMGVTDVIRAEEWLVSTPIHVLLYRAFGWEAPRFYHMPLLRNPDKTKISKRKSHTSLDWYKAEGFLPEALRNYLCLMGFSMPDGREIFTLEEFIQAFTWERVSLGGPVFDLEKLRWMNGKYIREVLSLEEVAERVKPFLREAGLSWESEAYLRRAVELMRPRFDTLKEFPEKARYLFTEDYPVSEKAQRKLEEGLPLLKELYPRLRAQEEWTEAALEALLRGFAAEKGVKLGQVAQPLRAALTGSLETPGLFEILALLGKERALRRLERALA 1n78 B 2.1 BS01 rna D 0 S9 T43 R47 V145 R163 V166 Y168 E172 V177 K180 S181 Y187 E207 E208 W209 L210 R237 K241 T242 K243 G274 E282 L300 P303 V304 E308 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 S9 T43 R47 V145 R163 V166 Y168 E172 V177 K180 S181 Y187 E207 E208 W209 L210 R237 K241 T242 K243 G274 E282 L300 P303 V304 E308 K309 W312 R319 P357 R358 R417 L427 Q432 R435 L442 E443 T444 G446 L447 F448 K246 K246 6.1.1.17 0000049,0000166,0004812,0004818,0005524,0005737,0005829,0006412,0006418,0006424,0008270,0043039 remove_due_to_license_issue P27000 12554668 501 ~ 576 MVVTRIAPSPTGDPHVGTAYIALFNYAWARRNGGRFIVRIEDTDRARYVPGAEERILAALKWLGLSYDEGPDVGGPHGPYRQSERLPLYQKYAEELLKRGWAYRAFETPEELEQIRKEKGGYDGRARNIPPEEAEERARRGEPHVIRLKVPRPGTTEVKDELRGVVVYDNQEIPDVVLLKSDGYPTYHLANVVDDHLMGVTDVIRAEEWLVSTPIHVLLYRAFGWEAPRFYHMPLLRNPDKTKISKRKSHTSLDWYKAEGFLPEALRNYLCLMGFSMPDGREIFTLEEFIQAFTWERVSLGGPVFDLEKLRWMNGKYIREVLSLEEVAERVKPFLREAGLSWESEAYLRRAVELMRPRFDTLKEFPEKARYLFTEDYPVSEKAQRKLEEGLPLLKELYPRLRAQEEWTEAALEALLRGFAAEKGVKLGQVAQPLRAALTGSLETPGLFEILALLGKERALRRLERALA 1n7i A 2.8 BS02 LY1 A 1 Y35 N39 Y40 R44 V53 K57 F182 Y222 D267 V269 Y14 N18 Y19 R23 V32 K36 F161 Y201 D246 V248 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 remove_due_to_license_issue Ki=4400nM P11086 14695818 3002 AVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKVGL 1n7j A 2.7 BS02 IDI A 1 Y35 V53 F182 E219 Y222 Y14 V32 F161 E198 Y201 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 remove_due_to_license_issue Ki=93nM P11086 14695818 3003 AVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKVGL 1n8u A 1.8 BS01 BDD A 1 Y8 D9 Y26 V27 Y6 D7 Y24 V25 ? Kd=0.93uM remove_due_to_license_issue Q9NG96 12697900 411 KYTDKYDNINLDEILANKRLLVAYVNCVMERGKCSPEGKELKEHLQDAIENGCKKCTENQEKGAYRVIEHLIKNEIEIWRELTAKYDPTGNWRKKYEDRA 1n8u A 1.8 BS02 BDD A 2 E42 L43 A50 W94 Y98 E40 L41 A48 W92 Y96 ? Kd=0.93uM remove_due_to_license_issue Q9NG96 12697900 412 KYTDKYDNINLDEILANKRLLVAYVNCVMERGKCSPEGKELKEHLQDAIENGCKKCTENQEKGAYRVIEHLIKNEIEIWRELTAKYDPTGNWRKKYEDRA 1n8u A 1.8 BS03 BDD A 3 I51 D89 I49 D87 ? Kd=0.93uM remove_due_to_license_issue Q9NG96 12697900 413 KYTDKYDNINLDEILANKRLLVAYVNCVMERGKCSPEGKELKEHLQDAIENGCKKCTENQEKGAYRVIEHLIKNEIEIWRELTAKYDPTGNWRKKYEDRA 1n8v A 1.39 BS01 BDD A 1 L13 Y26 V30 L11 Y24 V28 ? Kd=0.93uM remove_due_to_license_issue Q9NG96 12697900 501 KYTDKYDNINLDEILANKRLLVAYVNCVMERGKCSPEGKELKEHLQDAIENGCKKCTENQEKGAYRVIEHLIKNEIEIWRELTAKYDPTGNWRKKYEDRAK 1n8v A 1.39 BS02 BDD A 2 E42 L43 A50 Y98 E40 L41 A48 Y96 ? Kd=0.93uM remove_due_to_license_issue Q9NG96 12697900 502 KYTDKYDNINLDEILANKRLLVAYVNCVMERGKCSPEGKELKEHLQDAIENGCKKCTENQEKGAYRVIEHLIKNEIEIWRELTAKYDPTGNWRKKYEDRAK 1n8v A 1.39 BS03 BDD A 3 G65 A66 I70 W81 T85 D89 G63 A64 I68 W79 T83 D87 ? Kd=0.93uM remove_due_to_license_issue Q9NG96 12697900 503 KYTDKYDNINLDEILANKRLLVAYVNCVMERGKCSPEGKELKEHLQDAIENGCKKCTENQEKGAYRVIEHLIKNEIEIWRELTAKYDPTGNWRKKYEDRAK 1n94 A 3.5 BS02 TIN A 1 K164 Y166 Q167 K110 Y112 Q113 K164 K110 2.5.1.58,2.5.1.59 0008318,0018342 remove_due_to_license_issue Q04631 12657282 1 FLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSEKFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVWHFRRVLLRSLQKDLQEEMNYIIAIIEEQPKNYQVWHHRRVLVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFRLWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRAVLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPNLLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDILNKALELCEILAKEKDTIRKEYWRYIGRSLQSKHSR 1n94 B 3.5 BS02 TIN A 1 S99 W106 S78 W85 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H227 R270 K273 D276 C278 Y279 D331 D338 H341 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 12657282 1 PLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQK 1n95 B 2.3 BS03 FTH B 1 Y93 L96 W102 W106 D359 H362 Y71 L74 W80 W84 D337 H340 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 12657282 1001 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1n9a B 3.2 BS03 FTI B 1 L96 W106 D359 Y361 L74 W84 D337 Y339 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 12657283 1 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1n9m A 1.6 BS01 BTN A 1 L25 Y43 S45 N49 W79 T90 W108 L12 Y30 S32 N36 W66 T77 W95 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 12925786 5100 EAGITGTWYNQLGATFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVK 1n9m D 1.6 BS01 BTN D 1 L25 Y43 S45 N49 W79 T90 W108 L13 Y31 S33 N37 W67 T78 W96 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 12925786 5400 AEAGITGTWYNQLGATFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKP 1nax A 2.7 BS01 IH5 A 1 F272 I275 I276 R282 M310 M313 L330 N331 H435 F455 F62 I65 I66 R72 M100 M103 L120 N121 H225 F245 ? 0003677,0004879,0006355 remove_due_to_license_issue IC50=1.1nM, Ki=0.37nM, EC50=1.12nM P10828 12699376 501 KPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGQAPIVNAPEGGKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 1nc1 A 2.0 BS01 MTH A 1 M9 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 M11 I52 S78 A79 G80 F153 I154 E174 M175 E176 D199 F209 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=0.75uM remove_due_to_license_issue P0AF12 12496243 233 FSMKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1nc1 B 2.0 BS01 MTH B 1 M9 I50 S76 A77 G78 F151 I152 E172 M173 E174 S196 D197 F207 M9 I50 S76 A77 G78 F151 I152 E172 M173 E174 S196 D197 F207 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=0.75uM remove_due_to_license_issue P0AF12 12496243 234 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1nc3 A 2.2 BS01 FMC A 1 S76 A77 G78 F151 I152 E172 M173 E174 D197 A199 F207 S79 A80 G81 F154 I155 E175 M176 E177 D200 A202 F210 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=10uM remove_due_to_license_issue P0AF12 12496243 233 EFSMKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1nc3 B 2.2 BS01 FMC B 1 S76 A77 F151 I152 E172 M173 E174 D197 A199 S76 A77 F151 I152 E172 M173 E174 D197 A199 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=10uM remove_due_to_license_issue P0AF12 12496243 234 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLA 1nc6 A 1.9 BS03 ABB A 1 H57 D189 S190 C191 Q192 G193 D194 S195 W215 G216 G219 H40 D171 S172 C173 Q174 G175 D176 S177 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 12930148 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1nd5 A 2.9 BS01 2BF A 1 R11 H12 R15 I18 R79 Y123 S175 H257 D258 T259 R11 H12 R15 I18 R79 Y123 S175 H257 D258 T259 3.1.3.2,3.1.3.48,3.1.3.5 0003993,0004725,0004726,0005515,0005576,0005615,0005634,0005737,0005764,0005765,0005771,0005829,0005886,0006144,0006338,0006629,0006772,0008253,0009117,0012506,0016020,0016311,0016787,0016791,0030141,0030175,0030946,0031985,0033265,0035577,0042131,0042802,0042803,0045177,0046085,0051930,0052642,0060090,0060168,0070062,0106411,0140793 remove_due_to_license_issue IC50=4nM P15309 12525165 6000 KELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRFQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMT 1nde A 3.0 BS01 MON A 1 M295 L298 A302 D303 E305 L339 R346 I373 I376 H475 L476 M33 L36 A40 D41 E43 L77 R84 I111 I114 H209 L210 ? 0003677,0004879,0006355 remove_due_to_license_issue Q92731 12459017 101 DALSPEQLVLTLLEAEPPHVLISRPSFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYATQDADSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKPVYDLLLEMLNAHVL 1ndj A 1.81 BS01 BTN A 1 S27 F43 S45 V47 G48 N49 W79 A86 T90 W108 S12 F28 S30 V32 G33 N34 W64 A71 T75 W93 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 12925786 5100 GITGTWYNQLGSTFIVTAGADGALTGTFESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTK 1ndj D 1.81 BS01 BTN D 1 N23 L25 S27 F43 S45 V47 G48 N49 W79 S88 T90 W108 D128 N8 L10 S12 F28 S30 V32 G33 N34 W64 S73 T75 W93 D113 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 12925786 5400 GITGTWYNQLGSTFIVTAGADGALTGTFESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTK 1ndv A 2.3 BS02 FR0 A 1 H17 D19 L56 F61 L62 G184 E217 T269 D296 H14 D16 L53 F58 L59 G181 E214 T266 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=1.2uM remove_due_to_license_issue P56658 14709046 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1ndw A 2.0 BS02 FR2 A 1 H17 D19 L62 F65 L106 W117 D296 H14 D16 L59 F62 L103 W114 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=5.9uM remove_due_to_license_issue P56658 14709046 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1ndy A 2.0 BS02 FR3 A 1 H17 D19 L62 F65 L106 M155 H157 G184 D185 D296 H14 D16 L59 F62 L103 M152 H154 G181 D182 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=0.68uM remove_due_to_license_issue P56658 14709046 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1ndz A 2.0 BS02 FR5 A 1 H17 D19 F61 L62 F65 M155 G184 D185 T269 D296 H14 D16 F58 L59 F62 M152 G181 D182 T266 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=7.7nM remove_due_to_license_issue P56658 14709046 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1nf8 A 1.6 BS01 ISC A 1 F43 Q78 R87 W94 K122 V150 Y151 G155 F43 Q78 R87 W94 K122 V150 Y151 G155 H37 A38 K122 H37 A38 K122 3.3.2.15 0002047,0008908,0016787,0017000 Kd=0.015uM remove_due_to_license_issue P0DPB9 12741825 220 MSGIPEITAYPLPTAQQLPANLARWSLEPRRAVLLVHAMQRYFLRPLPESLRAGLVANAARLRRWCVEQGVQIAYTAQPGSMTEEQRGLLKDFWGPGMRASPADREVVEELAPGPDDWLLTKWRYSAFFHSDLLQRMRAAGRDQLVLCGVYAHVGVLISTVDAYSNDIQPFLVADAIADFSEAHHRMALEYAASRCAMVVTTDEVLE 1nfs A 1.96 BS03 DED A 1 K21 R51 C67 G68 H69 R83 Y104 E114 E116 W161 K18 R48 C64 G65 H66 R80 Y101 E111 E113 W158 H25 H32 C67 H69 E87 Y104 E114 E116 W161 H22 H29 C64 H66 E84 Y101 E111 E113 W158 5.3.3.2 0000287,0003824,0004452,0005737,0006974,0008270,0008299,0016853,0046872,0050992 Kd<0.12nM remove_due_to_license_issue Q46822 12540835 301 EHVILLNAQGVPTGTLEKYAAHTADTRLHLAFSSWLFNAKGQLLVTRRALSKKAWPGVWTNSVCGHPQLGESNEDAVIRRCRYELGVEITPPESIYPDFRYRATDPSGIVENEVCPVFAARTTSALQINDDEVMDYQWCDLADVLHGIDATPWAFSPWMVMQATNREARKRLSAFT 1nfu A 2.05 BS02 RRP A 1 F174 D189 A190 C191 Q192 V213 W215 G216 E217 G219 C220 G226 I227 Y228 F162 D179 A180 C181 Q182 V203 W205 G206 E207 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=18nM remove_due_to_license_issue Ki=4nM P00742 12593649 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1nfw A 2.1 BS02 RRR A 1 Y99 F174 D189 A190 Q192 V213 W215 G216 E217 G218 C220 G226 I227 Y228 Y85 F162 D179 A180 Q182 V203 W205 G206 E207 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=1.1nM remove_due_to_license_issue Ki=1.1nM P00742 12593649 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1nfx A 2.15 BS02 RDR A 1 Y99 F174 D189 A190 C191 Q192 V213 W215 G216 E217 G218 C220 G226 I227 Y228 Y85 F162 D179 A180 C181 Q182 V203 W205 G206 E207 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=3nM remove_due_to_license_issue Ki=3.0nM P00742 12593649 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1nfy A 2.1 BS02 RTR A 1 Y99 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=1.3nM remove_due_to_license_issue Ki=1.3nM P00742 12593649 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1ng9 A 2.6 BS01 dna E 0 P12 M13 M33 G34 D35 F36 S61 Q95 P99 P105 V106 R108 P12 M13 M33 G34 D35 F36 S61 Q95 P99 P105 V106 R108 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 12554674 1 ~ 18 MSAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGAGRSTFMVEMTETANILHNATEYSLVLMDEIGAGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1ng9 A 2.6 BS02 dna F 0 F36 E38 I53 S54 T56 M68 G70 P72 H74 Y79 L495 K496 R500 F36 E38 I53 S54 T56 M68 G70 P72 H74 Y79 L495 K496 R500 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 12554674 14 ~ 30 MSAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGAGRSTFMVEMTETANILHNATEYSLVLMDEIGAGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1ng9 B 2.6 BS01 dna E 0 Q95 L495 K496 R500 Q79 L469 K470 R474 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 12554674 1 ~ 18 AHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTPIPMAGIPYHAVENYLAKLVNQGESVAICEQVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGASTFMVEMTETANILHNATEYSLVLMDEIGAGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1nhg A 2.43 BS02 TCL A 1 A217 N218 A219 Y267 Y277 A319 A320 I323 A121 N122 A123 Y171 Y181 A223 A224 I227 Y277 K285 Y181 K189 1.3.1.9 0004318,0006633 Ki=0.05uM remove_due_to_license_issue IC50=49nM Q9BH77 11792710 500 EDICFIAGIGDTNGYGWGIAKELSKRNVKIIFGIWPPVYNIFMKNYKNGKFDNDMIIDKDKKMNILDMLPFDASFDTANDIDEETKNNKRYNMLQNYTIEDVANLIHQKYGKINMLVHSLANAKEVQKDLLNTSRKGYLDALSKSSYSLISLCKYFVNIMKPQSSIISLTYHASQKVVPGYGGGMSSAKAALESDTRVLAYHLGRNYNIRINTISAGPLKSRAATAINK 1nhu A 2.0 BS01 153 A 1 L419 R422 M423 S476 Y477 L497 R501 W528 L414 R417 M418 S471 Y472 L492 R496 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Ki=2.2uM remove_due_to_license_issue P26663 12509436 5001 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 1nhv A 2.9 BS01 154 A 1 R422 M423 S476 Y477 L497 R501 R417 M418 S471 Y472 L492 R496 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 12509436 5001 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 1nhw A 2.35 BS02 TCC A 1 A217 N218 A219 V222 Y277 A319 A320 I323 A121 N122 A123 V126 Y181 A223 A224 I227 Y277 K285 Y181 K189 1.3.1.9 0004318,0006633 Ki=14.3uM remove_due_to_license_issue Q9BH77 11792710 600 EDICFIAGIGDTNGYGWGIAKELSKRNVKIIFGIWPPVYNIFMKNYKNGKFDNDMIIDKDKKMNILDMLPFDASFDTANDIDEETKNNKRYNMLQNYTIEDVANLIHQKYGKINMLVHSLANAKEVQKDLLNTSRKGYLDALSKSSYSLISLCKYFVNIMKPQSSIISLTYHASQKVVPGYGGGMSSAKAALESDTRVLAYHLGRNYNIRINTISAGPLKSRAATAINK 1nhx A 2.1 BS03 FTB A 1 A287 N292 L293 M296 W516 F517 F525 F530 N533 A278 N283 L284 M287 W499 F500 F508 F513 N516 R87 Y235 K244 H264 S286 C288 D311 R405 R78 Y226 K235 H255 S277 C279 D302 R396 2.7.11.-,4.1.1.32 0000287,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0016301,0016831,0017076,0018105,0019543,0030145,0031406,0032868,0032869,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070062,0070365,0071333,0071549,0072350,0106264 ic50=2.11uM remove_due_to_license_issue IC50=2110nM P35558 14552798 704 NLSAKVVQGSLDSLPQAVREFLENNAELCQPDHIHICDGSEEENGRLLGQMEEEGILRRLKKYDNCWLALTDPRDVARIESKTVIVTQEQRDTVPIPKTGLSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLSKIGIELTDSPYVVASMRIMTRMGTPVLEALGDGEFVKCLHSVGCPLPLQKPLVNNWPCNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRMASRLAKEEGWLAEHMLVLGITNPEGEKKYLAAAFPSACGKTNLAMMNPSLPGWKVECVGDDIAWMKFDAQGHLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLASGVTITSWKNKEWSSEDGEPCAHPNSRFCTPASQCPIIDAAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEAKIIMHDPFAMRPFFGYNFGKYLAHWLSMAQHPAAKLPKIFHVNWFRKDKEGKFLWPGFGENSRVLEWMFNRIDGKASTKLTPIGYIPKEDALNLKGLGHINMMELFSISKEFWDKEVEDIEKYLVDQVNADLPCEIEREILALKQRISQM 1nhz A 2.3 BS01 486 A 1 M560 L563 N564 G567 Q570 M601 M604 F623 Q642 M646 L732 M31 L34 N35 G38 Q41 M72 M75 F94 Q113 M117 L203 ? remove_due_to_license_issue IC50=1.1nM, Ki=1.2nM, EC50=872nM, Kd=15nM P04150 12686538 800 PTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNNIKKLLFHQ 1ni1 B 2.3 BS03 2C5 B 1 Y93 L96 W106 R202 D297 D359 Y361 Y71 L74 W84 R180 D275 D337 Y339 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=0.9nM remove_due_to_license_issue Q02293 12699757 10 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1nj1 A 2.55 BS03 5CA A 1 T117 E119 R148 I158 V160 I163 F166 E168 F212 Q232 G234 T235 H237 C265 Y266 G267 S269 R271 T99 E101 R130 I140 V142 I145 F148 E150 F194 Q214 G216 T217 H219 C247 Y248 G249 S251 R253 E119 R148 H170 E101 R130 H152 6.1.1.15 0000166,0004812,0004827,0005515,0005524,0005737,0006412,0006418,0006433,0017101,0046872 remove_due_to_license_issue O26708 12578991 512 EFSEWFHNILEEAEIIDQRYPVKGMHVWMPHGFMIRKNTLKILRRILDRDHEEVLFPLLVPEDELAKEAIHVKGFEDEVYWVTHGGLSKLQRKLALRPTSETVMYPMFALWVRSHTDLPMRFYQVVNTFRYETKHTRPLIRVREITTFKEAHTIHATASEAEEQVERAVEIYKEFFNSLGIPYLITRRPPWDKFPGSEYTVAFDTLMPDGKTLQIGTVHNLGQTFARTFEIKFETPEGDHEYVHQTCYGLSDRVIASVIAIHGDESGLCLPPDVAAHQVVIVPIIFKKAAEEVMEACRELRSRLEAAGFRVHLDDRDIRAGRKYYEWEMRGVPLRVEIGPRDLEKGAAVISRRDTGEKVTADLQGIEETLRELMKDILENLRTRAWERMESEIREAETLEEASRIVDEKRGIISFMWCGEEECGMDVEEKVRVDILGIQEEGSGTCINCGREAPYRAYLARTY 1nj5 A 2.8 BS03 P5A A 1 T117 E119 R148 I158 V160 I163 F166 E168 F212 Q232 T235 H237 C265 Y266 G267 S269 R271 T99 E101 R130 I140 V142 I145 F148 E150 F194 Q214 T217 H219 C247 Y248 G249 S251 R253 E119 R148 H170 E101 R130 H152 6.1.1.15 0000166,0004812,0004827,0005515,0005524,0005737,0006412,0006418,0006433,0017101,0046872 remove_due_to_license_issue O26708 12578991 510 EFSEWFHNILEEAEIIDQRYPVKGMHVWMPHGFMIRKNTLKILRRILDRDHEEVLFPLLVPEDELAKEAIHVKGFEDEVYWVTHGGLSKLQRKLALRPTSETVMYPMFALWVRSHTDLPMRFYQVVNTFRYETKHTRPLIRVREITTFKEAHTIHATASEAEEQVERAVEIYKEFFNSLGIPYLITRRPPWDKFPGSEYTVAFDTLMPDGKTLQIGTVHNLGQTFARTFEIKFETPEGDHEYVHQTCYGLSDRVIASVIAIHGDESGLCLPPDVAAHQVVIVPIIFKKAAEEVMEACRELRSRLEAAGFRVHLDDRDIRAGRKYYEWEMRGVPLRVEIGPRDLEKGAAVISRRDTGEKVTADLQGIEETLRELMKDILENLRTRAWERMESEIREAETLEEASRIVDEKRGIISFMWCGEEECGMDVEEKVRVDILGIQEEGSGTCINCGREAPYRAYLARTY 1nja A 2.5 BS01 DCM A 1 R23 L195 C198 H199 R218 S219 A220 D221 H259 Y261 R23 L195 C198 H199 R218 S219 A220 D221 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=0.49uM remove_due_to_license_issue P00469 8611496 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFCIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1njb A 2.74 BS01 UMP A 1 R23 C198 H199 R218 S219 A220 D221 H259 Y261 R23 C198 H199 R218 S219 A220 D221 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue P00469 8611496 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFCIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1njc A 2.5 BS01 DCM A 1 R23 Q217 R218 S219 A220 D221 D229 H259 R23 Q217 R218 S219 A220 D221 D229 H259 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=2.8uM remove_due_to_license_issue P00469 8611496 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFDIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1njd A 2.2 BS01 UMP A 1 R23 C198 R218 S219 A220 D221 D229 H259 Y261 R23 C198 R218 S219 A220 D221 D229 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=2.7uM remove_due_to_license_issue P00469 8611496 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFDIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1nje A 2.3 BS01 DCM A 1 R23 R218 S219 A220 D221 N229 H259 Y261 R23 R218 S219 A220 D221 N229 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=160uM remove_due_to_license_issue P00469 8611496 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1njf A 2.3 BS02 AGS A 1 A7 W10 R11 P12 V18 V19 R47 G48 V49 G50 K51 T52 S53 L214 R215 A3 W6 R7 P8 V14 V15 R43 G44 V45 G46 K47 T48 S49 L210 R211 2.7.7.7 0003887,0005524,0006260,0009360,0016887 Kd=0.62uM remove_due_to_license_issue P06710 12623013 402 VLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGT 1njj A 2.45 BS01 GET A 1 R22 D243 L339 L382 E384 D385 R3 D206 L287 L327 E329 D330 K69 H197 E274 K42 H160 E237 4.1.1.17 0003824,0004586,0005737,0006596,0016829,0033387 Ki=8mM remove_due_to_license_issue Q9TZZ6 12672797 601 NTRDALCKKGDPFFVADLGDIVRKHETWKKCLPRVTPFYAVKCNDDWRVLGTLAALGTGFDCASNTEIQRVRGIGVPPEKIIYANPCKQISHIRYARDSGVDVMTFDCVDELEKVAKTHPKAKMVLRISTVKFGAKVEDCRFILEQAKKLNIDVTGVSFHVGSGSTDASTFAQAISDSRFVFDMGTELGFNMHILDIGGGFPGTRDAPLKFEEIAGVINNALEKHFPPDLKLTIVAEPGRYYVASAFTLAVNVIAKKVTQSFMYYVNDGVYGSFNCILYDHAVVRPLPQREPEKLYPSSVWGPTCDGLDQIVERYYLPEMQVGEWLLFEDMGAYTVSPTIYYVVSGLPD 1njs A 1.98 BS01 KEU A 1 R64 L85 M89 R90 I91 L92 N106 H108 G117 S118 V139 A140 V143 D144 R64 L85 M89 R90 I91 L92 N106 H108 G117 S118 V139 A140 V143 D144 N106 H108 T135 D144 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=15nM remove_due_to_license_issue P22102 12755606 510 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 1nju A 2.7 BS01 0FP A 1 E31 N62 H63 S132 L133 S134 S135 R136 R137 C161 V163 G164 R165 I231 E28 N53 H54 S123 L124 S125 S126 R127 R128 C144 V146 G147 R148 I205 3.4.21.97 0004252,0006508 remove_due_to_license_issue P16753 12549906 260 DEQQSQAVAPVYVGGFLARYDQSPDEAELLLPRDVVEHWLHAQLSVALPLNINHDDTAVVGHVAAMQSVRDGLFCLGCVTSPRFLEIVRRASEKSELVSRGPVSPLQPDKVVEFLSGSYAGLSLSSRRCDDVEQTTPFKHVALCSVGRRRGTLAVYGRDPEWVTQRFPDLTAADRDGLRAQWQSGDPFRSDSYGLLGNSVDALYIRERLPKLRYDKQLVGVTERESYVKA 1nju B 2.7 BS01 0FP B 1 N362 H363 S432 L433 S434 S435 R436 R437 K456 C461 V463 G464 R465 N52 H53 S122 L123 S124 S125 R126 R127 K138 C143 V145 G146 R147 3.4.21.97 0004252,0006508 remove_due_to_license_issue P16753 12549906 560 DEQQSQAVAPVYVGGFLARYDQSPDEAELLLPRDVVEHWLHAQSVALPLNINHDDTAVVGHVAAMQSVRDGLFCLGCVTSPRFLEIVRRASEKSELVSRGPVSPLQPDKVVEFLSGSYAGLSLSSRRCDDVEQTTPFKHVALCSVGRRRGTLAVYGRDPEWVTQRFPDLTAADRDGLRAQWQASGDPFRSDSYGLLGNSVDALYIRERLPKLRYDKQLVGVTERESYVKA 1nk2 P -1.00 BS01 dna A 0 K109 K111 R113 V114 Q152 I155 N159 K163 K9 K11 R13 V14 Q52 I55 N59 K63 ? 0000981,0003677,0006355 remove_due_to_license_issue P22808 9154919 1 ~ 16 ASDGLPNKKRKRRVLFTKAQTYELERRFRQQRYLSAPEREHLASLIRLTPTQVKIWFQNHRYKTKRAQNEKGYEGHP 1nk2 P -1.00 BS02 dna B 0 R110 K111 R112 R113 Y162 R10 K11 R12 R13 Y62 ? 0000981,0003677,0006355 remove_due_to_license_issue P22808 9154919 17 ~ 32 ASDGLPNKKRKRRVLFTKAQTYELERRFRQQRYLSAPEREHLASLIRLTPTQVKIWFQNHRYKTKRAQNEKGYEGHP 1nki A 0.95 BS02 PPF A 1 Y62 H64 S94 Y100 R119 Y62 H64 S94 Y100 R119 2.5.1.18 0004364,0005737,0016740,0046677,0046872 Kd=0.2uM remove_due_to_license_issue Q9I4K6 15504029 5001 MLTGLNHLTLAVADLPASIAFYRDLLGFRLEARWDQGAYLELGSLWLCLSREPQYGGPAADYTHYAFGIAAADFARFAAQLRAHGVREWKQNRSEGDSFYFLDPDGHRLEAHVGDLRSRLAACRQAPYAGMRFA 1nki B 0.95 BS02 PPF B 1 Y62 H64 S94 Y100 E110 R119 Y62 H64 S94 Y100 E110 R119 2.5.1.18 0004364,0005737,0016740,0046677,0046872 Kd=0.2uM remove_due_to_license_issue Q9I4K6 15504029 5002 MLTGLNHLTLAVADLPASIAFYRDLLGFRLEARWDQGAYLELGSLWLCLSREPQYGGPAADYTHYAFGIAAADFARFAAQLRAHGVREWKQNRSEGDSFYFLDPDGHRLEAHVGDLRSRLAACRQAPYAGMRFA 1nkm A 2.7 BS01 0FP A 1 N62 H63 S132 S134 S135 R136 K156 C161 G164 R165 I231 N50 H51 S120 S122 S123 R124 K130 C135 G138 R139 I195 3.4.21.97 0004252,0006508 remove_due_to_license_issue P16753 12549906 260 DEQQSQAVAPVYVGGFLARYDQSPDEAELLLPRDVVEHWLHAQALPLNINHDDTAVVGHVAAMQSVRDGLFCLGCVTSPRFLEIVRRASEKSELVSRGPVSPLQPDKVVEFLSGSYAGLSLSSRRTTPFKHVALCSVGRRRGTLAVYGRDPEWVTQRFPDLTAADRDGLRAQWQGDPFRSDSYGLLGNSVDALYIRERLPKLRYDKQLVGVTERESYVKA 1nkp A 1.8 BS01 dna F 0 H898 K902 E910 R913 H2 K6 E14 R17 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 12553908 101 ~ 119 GHMNVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAEEQKLISEEDLLRKRREQLKHKLEQLGGC 1nkp A 1.8 BS02 dna G 0 R903 H906 N907 E910 R914 P938 K939 R7 H10 N11 E14 R18 P42 K43 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 12553908 301 ~ 319 GHMNVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAEEQKLISEEDLLRKRREQLKHKLEQLGGC 1nkp B 1.8 BS01 dna F 0 R204 H207 N208 E211 R212 R215 K219 S238 R239 R3 H6 N7 E10 R11 R14 K18 S37 R38 ? 0046983 remove_due_to_license_issue P61244 12553908 101 ~ 119 DKRAHHNALERKRRDHIKDSFHSLRDSVPSLQGEKASRAQILDKATEYIQYMRRKNHTHQQDIDDLKRQNALLEQQVRALGGC 1nkp B 1.8 BS02 dna G 0 H206 E211 R214 H5 E10 R13 ? 0046983 remove_due_to_license_issue P61244 12553908 301 ~ 319 DKRAHHNALERKRRDHIKDSFHSLRDSVPSLQGEKASRAQILDKATEYIQYMRRKNHTHQQDIDDLKRQNALLEQQVRALGGC 1nkp D 1.8 BS01 dna H 0 R503 H506 N507 E510 R511 R514 K518 P538 K539 R5 H8 N9 E12 R13 R16 K20 P40 K41 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 12553908 601 ~ 619 MNVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAEEQKLISEEDLLRKRREQLKHKLEQL 1nkp D 1.8 BS02 dna J 0 K502 E510 R513 K4 E12 R15 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 12553908 801 ~ 819 MNVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAEEQKLISEEDLLRKRREQLKHKLEQL 1nkp E 1.8 BS01 dna H 0 E711 R714 E8 R11 ? 0046983 remove_due_to_license_issue P61244 12553908 601 ~ 619 RAHHNALERKRRDHIKDSFHSLRDSVPSLQGEKASRAQILDKATEYIQYMRRKNHTHQQDIDDLKRQNALLEQQVRALGGC 1nkp E 1.8 BS02 dna J 0 R704 H707 N708 E711 R712 R715 K719 S738 R739 R1 H4 N5 E8 R9 R12 K16 S35 R36 ? 0046983 remove_due_to_license_issue P61244 12553908 801 ~ 819 RAHHNALERKRRDHIKDSFHSLRDSVPSLQGEKASRAQILDKATEYIQYMRRKNHTHQQDIDDLKRQNALLEQQVRALGGC 1nl4 B 2.7 BS03 FTL B 1 W102 W106 D297 D359 Y361 H362 W80 W84 D275 D337 Y339 H340 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 12657284 1 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1nl6 A 2.8 BS01 750 A 1 Q19 G23 C25 S58 E59 G65 G66 Y67 L160 N161 H162 W184 Q19 G23 C25 S58 E59 G65 G66 Y67 L160 N161 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=30nM, Ki=0.0048nM P43235 11311061 501 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1nl9 A 2.4 BS01 989 A 1 Y46 D48 C215 S216 A217 I219 G220 R221 Q262 T263 G283 Y45 D47 C214 S215 A216 I218 G219 R220 Q261 T262 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=631nM P18031 12670229 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1nli A 1.93 BS01 ADE A 1 Y70 I71 G109 Y111 I155 S159 R163 Y71 I72 G110 Y112 I156 S160 R164 I71 A160 R163 I72 A161 R164 3.2.2.22 0006952,0016787,0017148,0030598,0035821,0050688,0090729 Kd=260uM remove_due_to_license_issue P09989 12676436 248 MDVSFRLSGATSSSYGVFISNLRKALPNERKLYDIPLLRSSLPGSQRYALIHLTNYADETISVAIDVTNVYIMGYRAGDTSYFFNEASATEAAKYVFKDAMRKVTLPYSGNYERLQTAAGKIRENIPLGLPALDSAITTLFYYNANSAASALMVLIQSTSAAARYKFIEQQIGKRVDKTFLPSLAIISLANSWSALSKQIQIASTNNGQFESPVVLINAQNQRVTITNVDAGVVTSNIALLLNRNNMA 1nlj A 2.4 BS01 2CA A 1 Q19 G23 C25 D61 G65 G66 A137 L160 N161 H162 W184 Q19 G23 C25 D61 G65 G66 A137 L160 N161 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue Ki=0.16nM, IC50=70nM P43235 11311061 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1nm6 A 1.8 BS02 L86 A 1 H57 Y60A W60D E97A N98 L99 A190 S195 V213 S214 W215 G216 H69 Y73 W76 E120 N121 L122 A218 S223 V243 S244 W245 G246 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=0.09nM remove_due_to_license_issue Ki=0.090000nM P00734 12873514 247 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1nmk A 2.1 BS01 SFM A 1 R55 F60 Q63 T73 A101 N102 Q111 F113 H126 R55 F60 Q63 T73 A101 N102 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 ic50=5.7nM remove_due_to_license_issue P62937 12656618 166 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 1nnb A 2.8 BS02 DAN A 1 R119 D152 R153 A248 E278 E279 R294 R372 Y406 R36 D69 R70 A165 E195 E196 R211 R289 Y323 D152 E279 R294 R372 Y406 D69 E196 R211 R289 Y323 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue IC50=13000nM P03472 8371267 500 DFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1nnj A 1.9 BS01 dna D 0 E2 K57 H72 R74 M75 K129 G170 N171 Y238 K254 K256 R260 E2 K57 H72 R74 M75 K129 G170 N171 Y234 K250 K252 R256 G1 G1 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 16243784 1 ~ 14 GELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSIALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1nnj A 1.9 BS02 dna E 0 K90 H91 V108 R109 F111 K90 H91 V108 R109 F111 G1 G1 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 16243784 15 ~ 28 GELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSIALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1nnk A 1.85 BS02 CE2 A 1 E10 Y58 P86 L87 T88 R93 G138 S139 T140 E190 M193 Y217 E10 Y58 P86 L87 T88 R93 G138 S139 T140 E190 M193 Y217 ? 0015276,0016020 ic50=3.5uM remove_due_to_license_issue P19491 12593667 454 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1nnu A 2.5 BS02 TCT A 1 A217 A219 V222 Y267 Y277 A319 I323 A121 A123 V126 Y171 Y181 A223 I227 Y277 K285 Y181 K189 1.3.1.9 0004318,0006633 Ki=0.15uM remove_due_to_license_issue Q9BH77 11792710 500 EDICFIAGIGDTNGYGWGIAKELSKRNVKIIFGIWPPVYNIFMKNYKNGKFDNDMIIDKDKKMNILDMLPFDASFDTANDIDEETKNNKRYNMLQNYTIEDVANLIHQKYGKINMLVHSLANAKEVQKDLLNTSRKGYLDALSKSSYSLISLCKYFVNIMKPQSSIISLTYHASQKVVPGYGGGMSSAKAALESDTRVLAYHLGRNYNIRINTISAGPLKSRAATAINK 1nny A 2.4 BS01 515 A 1 R24 Y46 D48 K120 C215 S216 A217 I219 G220 R221 R254 Q262 T263 G283 R23 Y45 D47 K119 C214 S215 A216 I218 G219 R220 R253 Q261 T262 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=20nM P18031 12670229 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1no6 A 2.4 BS01 794 A 1 Y46 V49 C215 S216 A217 I219 G220 R221 Q262 T263 G283 Y45 V48 C214 S215 A216 I218 G219 R220 Q261 T262 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=39000nM, Kd=26000nM P18031 12670229 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1no9 H 1.9 BS02 4ND H 1 H57 A190 C191 S195 V213 S214 W215 H43 A194 C195 S199 V219 S220 W221 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 12885234 250 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1noi A 2.5 BS03 NTZ A 1 L136 H377 T378 N484 E672 G675 L127 H363 T364 N470 E658 G661 H377 K568 R569 K574 T676 K680 H363 K554 R555 K560 T662 K666 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=700uM remove_due_to_license_issue P00489 8652510 998 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKPAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 1noj A 2.4 BS04 NTZ A 1 L136 N284 H377 N484 E672 S674 G675 L125 N273 H366 N473 E661 S663 G664 H377 K568 R569 K574 T676 K680 H366 K557 R558 K563 T665 K669 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=700uM remove_due_to_license_issue P00489 8652510 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKPAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1nok A 2.4 BS02 NTZ A 1 G135 L136 L139 H377 N484 E672 S674 G675 G124 L125 L128 H366 N473 E661 S663 G664 H377 K568 R569 K574 T676 K680 H366 K557 R558 K563 T665 K669 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=700uM remove_due_to_license_issue P00489 8652510 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKPAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 1nox A 1.59 BS01 FMN A 1 R18 S19 R21 Q73 P156 M157 L158 G159 S193 R195 R13 S14 R16 Q68 P151 M152 L153 G154 S188 R190 7.1.1.2 0008137,0016491,1902600 Kd=90nM remove_due_to_license_issue Q60049 8846223 300 PVLDAKTAALKRRSIRRYRKDPVPEGLLREILEAALRAPSAWNLQPWRIVVVRDPATKRALREAAFGQAHVEEAPVVLVLYADLEDALAHLDEVIHPGVQGERREAQKQAIQRAFAAMGQEARKAWASGQSYILLGYLLLLLEAYGLGSVPMLGFDPERVRAILGLPSRAAIPALVALGYPAEEGYPSHRLPLERVVLWR 1npa A 2.0 BS01 3NH A 1 D25 G27 A28 D29 V32 G48 G49 I50 V82 D25 G27 A28 D29 V32 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=2nM remove_due_to_license_issue P03366 9258349 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1npa B 2.0 BS01 3NH A 1 D25 G27 D30 G49 P81 V82 D25 G27 D30 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 9258349 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1npv A 2.0 BS01 L27 A 1 D25 G27 A28 D30 V32 G48 G49 D25 G27 A28 D30 V32 G48 G49 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=5.7nM remove_due_to_license_issue P03366 12723947 479 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1npv B 2.0 BS01 L27 A 1 D225 G227 A228 D230 G248 G249 I250 P281 D25 G27 A28 D30 G48 G49 I50 P81 D225 T226 G227 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12723947 479 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1npw A 2.0 BS01 LGZ A 1 D25 G27 A28 D29 V32 G48 G49 I50 V82 D25 G27 A28 D29 V32 G48 G49 I50 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=2nM remove_due_to_license_issue P03366 12723947 479 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1npw B 2.0 BS01 LGZ A 1 D225 G227 D230 G249 P281 V282 D25 G27 D30 G49 P81 V82 D225 T226 G227 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 12723947 479 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1npz A 2.0 BS01 C1P A 1 Q19 C25 N67 G68 G69 F70 A140 N163 H164 W186 Q19 C25 N67 G68 G69 F70 A140 N163 H164 W186 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue P25774 12641451 468 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVTLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 1nq0 A 2.4 BS01 4HY A 1 F269 F272 I276 M310 M313 A317 R320 L330 N331 L346 H435 M442 F61 F64 I68 M102 M105 A109 R112 L122 N123 L138 H227 M234 ? 0003677,0004879,0006355 remove_due_to_license_issue IC50=0.0407nM P10828 12511610 500 AAMEELQKSIGHKPEPTDEEWELIKTVTEAHVATNTQGSHWKQKRKFLPEDIGQKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 1nq7 A 1.5 BS02 ARL A 1 C227 Q228 Y229 L300 V303 R306 M307 F330 C20 Q21 Y22 L93 V96 R99 M100 F123 ? 0003677,0004879,0005634,0006355 Ki=0.16uM remove_due_to_license_issue P45446 12958591 800 TMSEIDRIAQNIIKSHLETCQYTMEELHQLAWQTHTYEEIKAYQSKSREALWQQCAIQITHAIQYVVEFAKRITGFMELCQNDQILLLKSGCLEVVLVRMCRAFNPLNNTVLFEGKYGGMQMFKALGSDDLVNEAFDFAKNLCSLQLTEEEIALFSSAVLISPDRAWLLEPRKVQKLQEKIYFALQHVIQKNHLDDETLAKLIAKIPTITAVCNLHGEKLQVFKQSHPDIVNTLFPPLYKELFN 1nqc A 1.8 BS01 C4P A 1 G23 C25 K64 C66 G68 G69 F70 M71 V162 N163 G23 C25 K64 C66 G68 G69 F70 M71 V162 N163 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue P25774 12641451 218 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVTLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 1nt1 A 2.0 BS02 T76 A 1 H57 Y60A S195 V213 S214 W215 G216 G219 F227 H69 Y73 S223 V243 S244 W245 G246 G248 F257 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=1.3nM remove_due_to_license_issue Ki=1.3nM P00734 12873514 247 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1ntk C 2.6 BS03 AY1 C 1 I27 S35 M190 L197 F220 Y224 D228 I26 S34 M189 L196 F219 Y223 D227 H201 S205 K227 D228 E271 H200 S204 K226 D227 E270 ? 0005739,0005743,0006122,0008121,0009055,0016020,0016491,0020037,0022904,0031966,0045275,0046872,0048039,1902600 remove_due_to_license_issue P00157 12885240 383 TNIRKSHPLMKIVNNAFIDLPAPSNISSWWNFGSLLGICLILQILTGLFLAMHYTSDTTTAFSSVTHICRDVNYGWIIRYMHANGASMFFICLYMHVGRGLYYGSYTFLETWNIGVILLLTVMATAFMGYVLPWGQMSFWGATVITNLLSAIPYIGTNLVEWIWGGFSVDKATLTRFFAFHFILPFIIMAIAMVHLLFLHETGSNNPTGISSDVDKIPFHPYYTIKDILGALLLILALMLLVLFAPDLLGDPDNYTPANPLNTPPHIKPEWYFLFAYAILRSIPNKLGGVLALAFSILILALIPLLHTSKQRSMMFRPLSQCLFWALVADLLTLTWIGGQPVEHPYITIGQLASVLYFLLILVLMPTAGTIENKLLKW 1nu1 C 3.2 BS03 QNO C 1 F18 I27 S35 F220 Y224 D228 F17 I26 S34 F219 Y223 D227 H201 S205 K227 D228 E271 H200 S204 K226 D227 E270 ? 0005739,0005743,0006122,0008121,0009055,0016020,0016491,0020037,0022904,0031966,0045275,0046872,0048039,1902600 remove_due_to_license_issue P00157 12885240 383 TNIRKSHPLMKIVNNAFIDLPAPSNISSWWNFGSLLGICLILQILTGLFLAMHYTSDTTTAFSSVTHICRDVNYGWIIRYMHANGASMFFICLYMHVGRGLYYGSYTFLETWNIGVILLLTVMATAFMGYVLPWGQMSFWGATVITNLLSAIPYIGTNLVEWIWGGFSVDKATLTRFFAFHFILPFIIMAIAMVHLLFLHETGSNNPTGISSDVDKIPFHPYYTIKDILGALLLILALMLLVLFAPDLLGDPDNYTPANPLNTPPHIKPEWYFLFAYAILRSIPNKLGGVLALAFSILILALIPLLHTSKQRSMMFRPLSQCLFWALVADLLTLTWIGGQPVEHPYITIGQLASVLYFLLILVLMPTAGTIENKLLKW 1nu3 A 1.75 BS01 VPR A 1 I80 D101 L103 F134 F139 I76 D97 L99 F130 F135 Y53 N55 R99 D101 D132 Y49 N51 R95 D97 D128 3.3.2.8 0016787,0018744 remove_due_to_license_issue Q9ZAG3 12773375 4001 IEQPRWASKDSAAGAASTPDEKIVLEFMDALTSNDAAKLIEYFAEDTMYQNMPLPPAYGRDAVEQTLAGLFTVMSIDAVETFHIGSSNGLVYTERVDVLRALPTGKSYNLSILGVFQLTEGKITGWRDYFDLREFEEAVDLPLRG 1nvq A 2.0 BS02 UCN A 1 L15 G16 V23 A36 K38 V68 E85 Y86 C87 G90 E91 E134 L137 S147 D148 L13 G14 V21 A34 K36 V59 E76 Y77 C78 G81 E82 E125 L128 S138 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=5.6nM remove_due_to_license_issue IC50=9.9nM, Ki=5.6nM O14757 12244092 400 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 1nvr A 1.8 BS02 STU A 1 L15 Y20 V23 A36 K38 E85 Y86 C87 G90 E91 E134 L137 D148 L13 Y18 V21 A34 K36 E76 Y77 C78 G81 E82 E125 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=7.8nM remove_due_to_license_issue O14757 12244092 400 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 1nvs A 1.8 BS02 UCM A 1 L15 G16 V23 A36 K38 L84 E85 E91 L137 D148 L13 G14 V21 A34 K36 L75 E76 E82 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=15nM remove_due_to_license_issue IC50=15nM O14757 12244092 400 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 1nw4 A 2.2 BS01 IMH A 1 S91 C92 G93 Y160 E182 M183 E184 D206 W212 S89 C90 G91 Y158 E180 M181 E182 D204 W210 H7 G23 R27 R45 E77 R88 S91 D206 G207 P209 V222 H5 G21 R25 R43 E75 R86 S89 D204 G205 P207 V220 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006148,0006166,0006195,0006218,0009116,0016757,0017061,0047975 Kd=0.86nM remove_due_to_license_issue Q8I3X4 14982926 301 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKWDEGDFDNNLVPHQLENMIKIALGACAKLATKYA 1nw4 B 2.2 BS01 IMH B 1 S91 C92 G93 Y160 E182 M183 E184 D206 S89 C90 G91 Y158 E180 M181 E182 D204 H7 G23 R27 R45 E77 R88 S91 D206 G207 P209 V222 H5 G21 R25 R43 E75 R86 S89 D204 G205 P207 V220 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006148,0006166,0006195,0006218,0009116,0016757,0017061,0047975 Kd=0.86nM remove_due_to_license_issue Q8I3X4 14982926 302 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKWDEGDFDNNLVPHQLENMIKIALGACAKLATKYA 1nw5 A 2.05 BS01 SAM A 1 D46 C47 D65 H223 T225 Q226 K227 F250 G252 S253 D271 A272 D11 C12 D30 H188 T190 Q191 K192 F215 G217 S218 D236 A237 D65 P66 D30 P31 2.1.1.72 0003676,0003677,0008168,0008170,0009007,0009307,0032259 Kd=6.1uM remove_due_to_license_issue P14751 12732637 401 GTTRHVYDVCDCLDTLAKLPDDSVQLIICDPPYNIMLADWDDHMDYIGWAKRWLAEAERVLSPTGSIAIFGGLQYQGEAGSGDLISIISHMRQNSKMLLANLIIWNYPNGMSAQRFFANRHEEIAWFAKTKKYFFDLDAVREPYDEETKAAYMKDKRLNPESVEKGRNPTNVWRMSRLNGNSLERVGHPTQKPAAVIERLVRALSHPGSTVLDFFAGSGVTARVAIQEGRNSICTDAAPVFKEYYQKQLTFLRSYEIVEGAANFGAALQR 1nw7 A 2.1 BS02 SAH A 1 D46 C47 D65 H223 T225 F249 F250 D271 A272 D11 C12 D30 H188 T190 F214 F215 D236 A237 D65 P66 D30 P31 2.1.1.72 0003676,0003677,0008168,0008170,0009007,0009307,0032259 Kd=8.1uM remove_due_to_license_issue P14751 12732637 401 GTTRHVYDVCDCLDTLAKLPDDSVQLIICDPPYNIMLADWDDHMDYIGWAKRWLAEAERVLSPTGSIAIFGGLQYQGEAGSGDLISIISHMRQNSKMLLANLIIWNYPNGMSAQRFFANRHEEIAWFAKTKKYFFDLDAVREPYDEETKAAYMKDKRLNPESVEKGRNPTNVWRMSRLNGNSLERVGHPTQKPAAVIERLVRALSHPGSTVLDFFAGSGVTARVAIQEGRNSICTDAAPVFKEYYQKQLTFLQRSYEIVEGAANFGAALQR 1nwl A 2.4 BS01 964 A 1 Y46 C47 A217 I219 G220 R221 Q262 Q266 Y46 C47 A217 I219 G220 R221 Q262 Q266 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P18031 12733877 501 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPSRVAKLPKNKNRNRYCDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTVGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1nxy A 1.6 BS01 SM2 A 1 M69 S70 Y105 S130 N132 E166 N170 S235 G236 A237 G238 R244 M44 S45 Y80 S105 N107 E141 N145 S210 G211 A212 G213 R218 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 12859188 500 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1nxy A 1.6 BS02 SM2 A 2 R241 G267 S268 Q269 R215 G240 S241 Q242 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 12859188 501 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1ny0 A 1.75 BS01 NBF A 1 S70 K73 Y105 S130 N132 N170 G236 A237 G238 E240 S45 K48 Y80 S105 N107 N145 G211 A212 G213 E214 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 12859188 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1nym A 1.2 BS01 CXB A 1 S70 K73 Y105 S130 N132 G236 A237 G238 E240 S45 K48 Y80 S105 N107 G211 A212 G213 E214 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 12859188 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1nyx A 2.65 BS01 DRF A 1 I281 F282 C285 Q286 R288 S289 H323 I326 L330 I341 S342 M348 H449 L469 Y473 I65 F66 C69 Q70 R72 S73 H107 I110 L114 I125 S126 M132 H233 L253 Y257 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=575nM, Ki=90nM P37231 12672231 101 DQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 1nyy A 1.9 BS01 105 A 1 S70 Y105 S130 N132 G236 A237 S45 Y80 S105 N107 G211 A212 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P62593 12859188 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1nz7 A 2.4 BS01 901 A 1 R24 D29 Y46 D48 K120 C215 S216 A217 I219 G220 R221 M258 Q262 T263 Q266 G283 R23 D28 Y45 D47 K119 C214 S215 A216 I218 G219 R220 M257 Q261 T262 Q265 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=76nM P18031 12749891 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1nzq H 2.18 BS03 162 H 1 H57 Y60A W60D D189 A190 E192 S195 S214 W215 G216 E217 G219 H43 Y47 W50 D192 A193 E195 S198 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=11nM remove_due_to_license_issue P00734 12781189 248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1o0d H 2.44 BS02 163 H 1 H57 Y60A W60D D189 A190 C191 S195 S214 W215 G216 G219 H43 Y47 W50 D192 A193 C194 S198 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=6.2nM remove_due_to_license_issue P00734 12781189 248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1o0f A 1.5 BS01 A3P A 1 Q11 H12 Q69 N71 A109 H119 Q11 H12 Q69 N71 A109 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=5uM remove_due_to_license_issue P61823 14573867 1301 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1o0h A 1.2 BS01 ADP A 1 K7 Q11 H12 K41 C65 N67 Q69 N71 A109 E111 V118 H119 K7 Q11 H12 K41 C65 N67 Q69 N71 A109 E111 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=1.2uM remove_due_to_license_issue P61823 14573867 1125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1o0m A 1.5 BS01 U2P A 1 Q11 H12 K41 V43 N44 T45 H119 F120 Q11 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=7.1uM remove_due_to_license_issue Ki=11600nM P61823 14573867 1101 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1o0n A 1.5 BS01 U3P A 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=82uM remove_due_to_license_issue Ki=78500nM P61823 14573867 1101 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1o0o A 1.2 BS01 A2P A 1 Q11 H12 H119 F120 Q11 H12 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=8uM remove_due_to_license_issue P61823 14573867 998 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1o1s B 2.3 BS02 1NH B 1 W102 H149 A151 M193 R202 H248 G250 Y251 R291 K294 Y300 W303 W80 H127 A129 M171 R180 H226 G228 Y229 R269 K272 Y278 W281 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 Ki=49nM remove_due_to_license_issue Q02293 12667062 2001 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1o2g H 1.58 BS02 696 H 1 C42 H57 C58 W60D D189 A190 C191 E192 S195 V213 C28 H43 C44 W50 D191 A192 C193 E194 S197 V217 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.76uM remove_due_to_license_issue Ki=760nM P00734 12742021 410 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1o2h A 1.77 BS02 CR3 A 1 F41 H57 D189 S190 Q192 S195 W215 G216 G219 F24 H40 D171 S172 Q174 S177 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.068uM remove_due_to_license_issue Ki=68nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2j A 1.65 BS02 656 A 1 H57 D189 S190 C191 Q192 S195 V213 H40 D171 S172 C173 Q174 S177 V191 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.12uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2k A 1.63 BS02 656 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.12uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2n A 1.5 BS02 762 A 1 H57 D189 S190 C191 Q192 S195 V213 S214 W215 G216 G219 G226 H40 D171 S172 C173 Q174 S177 V191 S192 W193 G194 G196 G204 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.81uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2o A 1.63 BS02 950 A 1 H57 D189 S190 Q192 S195 V213 S214 W215 G216 G219 H40 D171 S172 Q174 S177 V191 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.44uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2p A 1.47 BS02 972 A 1 H57 D189 S190 Q192 S195 V213 S214 W215 G219 G226 V227 Y228 H40 D171 S172 Q174 S177 V191 S192 W193 G196 G204 V205 Y206 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2q A 1.5 BS02 991 A 1 H57 D189 S190 Q192 S195 V213 S214 W215 G219 G226 V227 H40 D171 S172 Q174 S177 V191 S192 W193 G196 G204 V205 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.021uM remove_due_to_license_issue Ki=21nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2r A 1.45 BS02 CR9 A 1 F41 H57 D189 S190 Q192 S195 S214 W215 G219 F24 H40 D171 S172 Q174 S177 S192 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2s A 1.65 BS02 CR4 A 1 H57 D189 S190 Q192 S195 V213 G216 H40 D171 S172 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=3.4uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2t A 1.62 BS02 783 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 G219 C220 H40 D171 S172 C173 Q174 S177 V191 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue Ki=14nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2u A 1.41 BS02 847 A 1 D189 S190 C191 Q192 S195 V213 G219 D171 S172 C173 Q174 S177 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.4uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2v A 1.5 BS02 847 A 1 H57 D189 S190 Q192 S195 V213 W215 G219 C220 H40 D171 S172 Q174 S177 V191 W193 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.4uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2w A 1.38 BS02 847 A 1 H57 D189 S190 Q192 S195 V213 S214 G219 C220 H40 D171 S172 Q174 S177 V191 S192 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.4uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2x A 1.46 BS02 847 A 1 H57 D189 S190 C191 Q192 S195 V213 S214 G219 C220 H40 D171 S172 C173 Q174 S177 V191 S192 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.4uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2y A 1.45 BS02 847 A 1 H57 D189 S190 C191 Q192 S195 V213 W215 G216 H40 D171 S172 C173 Q174 S177 V191 W193 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.4uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o2z A 1.65 BS02 312 A 1 H57 D189 S190 C191 Q192 S195 S214 W215 G216 G219 H40 D171 S172 C173 Q174 S177 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.78uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o30 A 1.55 BS02 693 A 1 H57 D189 S190 Q192 S195 S214 W215 G216 G219 C220 H40 D171 S172 Q174 S177 S192 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.17uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o32 A 1.78 BS02 801 A 1 D189 S190 C191 Q192 W215 G219 D171 S172 C173 Q174 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.8uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o33 A 1.46 BS02 801 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.8uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o34 A 1.5 BS02 801 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.8uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o35 A 1.41 BS02 802 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o36 A 1.7 BS02 607 A 1 C42 H57 D189 S190 C191 Q192 S195 V213 G219 C220 C25 H40 D171 S172 C173 Q174 S177 V191 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.1uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o37 A 1.45 BS02 653 A 1 H57 D189 S190 C191 Q192 S195 V213 W215 G216 G219 C220 H40 D171 S172 C173 Q174 S177 V191 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.15uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o38 A 1.38 BS02 653 A 1 H57 D189 S190 Q192 S195 V213 W215 G219 H40 D171 S172 Q174 S177 V191 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.15uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o39 A 1.59 BS02 780 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 G219 H40 D171 S172 C173 Q174 S177 V191 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.074uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3b A 1.75 BS02 780 A 1 H57 D189 S190 C191 Q192 S195 V213 G216 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.074uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3c A 1.64 BS02 780 A 1 H57 D189 S190 C191 Q192 S195 V213 H40 D171 S172 C173 Q174 S177 V191 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3d A 1.33 BS02 780 A 1 H57 D189 S190 Q192 S195 V213 S214 W215 G216 G219 H40 D171 S172 Q174 S177 V191 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.074uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3e A 1.64 BS02 696 A 1 C42 H57 D189 S190 C191 Q192 S195 V213 G216 C25 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.011uM remove_due_to_license_issue Ki=11nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3f A 1.55 BS02 696 A 1 C42 H57 D189 S190 C191 Q192 S195 V213 G216 C25 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.011uM remove_due_to_license_issue Ki=11nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3g A 1.55 BS02 696 A 1 C42 H57 D189 S190 C191 Q192 S195 V213 G216 C25 H40 D171 S172 C173 Q174 S177 V191 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.011uM remove_due_to_license_issue Ki=11nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3h A 1.53 BS02 907 A 1 H57 D189 S190 Q192 S195 W215 G216 G219 H40 D171 S172 Q174 S177 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.05uM remove_due_to_license_issue Ki=50nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3i A 1.51 BS02 907 A 1 H57 D189 S190 Q192 S195 V213 W215 G216 G219 H40 D171 S172 Q174 S177 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.05uM remove_due_to_license_issue Ki=50nM P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3j A 1.4 BS02 334 A 1 H57 D189 S190 Q192 S195 V213 W215 G216 H40 D171 S172 Q174 S177 V191 W193 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.17uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3k A 1.43 BS02 334 A 1 H57 D189 S190 Q192 S195 W215 G216 G219 C220 H40 D171 S172 Q174 S177 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.17uM remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3l A 1.4 BS02 678 A 1 H57 D189 S190 Q192 S195 V213 S214 W215 G216 G219 H40 D171 S172 Q174 S177 V191 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 12742021 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1o3p B 1.81 BS02 655 B 1 H57 C58 S190 C191 Q192 S195 V213 W215 H46 C47 S193 C194 Q195 S198 V216 W218 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.22uM remove_due_to_license_issue P00749 12742021 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 1o3s A 3.0 BS01 dna B 0 T168 R169 Q170 R180 R185 K188 T161 R162 Q163 R173 R178 K181 ? 0003677,0003680,0003700,0005515,0005829,0006351,0006355,0008301,0030552,0032993,0042802,0043565,0045013,0045892,0045893 remove_due_to_license_issue P0ACJ8 11724533 -2 ~ 9 DPTLEWFLSHCHIHKYPSKSTLIHQGEKAETLYYIVKGSVAVLIKDEEGKEMILSYLNQGDFIGELGLFEEGQERSAWVRAKTACEVAEISYKKFRQLIQVNPDILMRLSAQMARRLQVTSEKVGNLAFLDVTGRIAQTLLNLAKQPDAMTHPDGMQIKITRQEIGQIVGCSRDTVGRILKMLEDQNLISAHGKTIVVYG 1o3s A 3.0 BS02 dna C 0 D138 V139 S179 D181 T182 K201 D131 V132 S172 D174 T175 K194 ? 0003677,0003680,0003700,0005515,0005829,0006351,0006355,0008301,0030552,0032993,0042802,0043565,0045013,0045892,0045893 remove_due_to_license_issue P0ACJ8 11724533 13 ~ -2 DPTLEWFLSHCHIHKYPSKSTLIHQGEKAETLYYIVKGSVAVLIKDEEGKEMILSYLNQGDFIGELGLFEEGQERSAWVRAKTACEVAEISYKKFRQLIQVNPDILMRLSAQMARRLQVTSEKVGNLAFLDVTGRIAQTLLNLAKQPDAMTHPDGMQIKITRQEIGQIVGCSRDTVGRILKMLEDQNLISAHGKTIVVYG 1o41 A 1.7 BS01 300 A 1 R14 R34 E37 C44 H60 K62 R14 R34 E37 C44 H60 K62 2.7.10.2 remove_due_to_license_issue IC50=900000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o42 A 1.7 BS01 843 A 1 R14 R34 S36 E37 T38 C44 H60 Y61 K62 I73 G95 R14 R34 S36 E37 T38 C44 H60 Y61 K62 I73 G95 2.7.10.2 ic50=9nM remove_due_to_license_issue IC50=9nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o43 A 1.5 BS01 821 A 1 R14 R34 S36 E37 Y43 C44 H60 Y61 K62 Y89 G95 L96 R14 R34 S36 E37 Y43 C44 H60 Y61 K62 Y89 G95 L96 2.7.10.2 remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o44 A 1.7 BS01 852 A 1 R14 R34 S36 E37 T38 C44 H60 Y61 K62 I73 G95 R14 R34 S36 E37 T38 C44 H60 Y61 K62 I73 G95 2.7.10.2 ic50=3nM remove_due_to_license_issue IC50=3nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o45 A 1.8 BS01 687 A 1 R14 R34 S36 E37 Y43 C44 H60 Y61 K62 I73 G95 L96 R14 R34 S36 E37 Y43 C44 H60 Y61 K62 I73 G95 L96 2.7.10.2 remove_due_to_license_issue IC50=0.25nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o46 A 2.0 BS01 903 A 1 R14 R34 S36 E37 T38 C44 H60 Y61 K62 G95 L96 R14 R34 S36 E37 T38 C44 H60 Y61 K62 G95 L96 2.7.10.2 ic50=10nM remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o47 A 1.8 BS01 822 A 1 R14 R34 S36 E37 C44 H60 Y61 I73 G95 L96 R14 R34 S36 E37 C44 H60 Y61 I73 G95 L96 2.7.10.2 ic50=4nM remove_due_to_license_issue IC50=5nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o48 A 1.55 BS01 853 A 1 R14 R34 E37 T38 C44 H60 Y61 K62 I73 Y89 G95 L96 R14 R34 E37 T38 C44 H60 Y61 K62 I73 Y89 G95 L96 2.7.10.2 ic50=450nM remove_due_to_license_issue IC50=450nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o49 A 1.7 BS01 493 A 1 R14 R34 E37 C44 H60 Y61 K62 I73 Y89 G95 R14 R34 E37 C44 H60 Y61 K62 I73 Y89 G95 2.7.10.2 ic50=437nM remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4a A 1.5 BS01 197 A 1 R14 R34 S36 E37 T38 C44 H60 Y61 K62 Y89 G95 L96 R14 R34 S36 E37 T38 C44 H60 Y61 K62 Y89 G95 L96 2.7.10.2 remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4b A 1.85 BS01 876 A 1 R14 R34 S36 E37 T38 H60 Y61 K62 G95 R14 R34 S36 E37 T38 H60 Y61 K62 G95 2.7.10.2 ic50=2000nM remove_due_to_license_issue IC50=2000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4d A 1.85 BS01 262 A 1 R14 R34 S36 E37 C44 H60 Y61 K62 R14 R34 S36 E37 C44 H60 Y61 K62 2.7.10.2 remove_due_to_license_issue IC50=200000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCP 1o4e A 2.0 BS01 299 A 1 R14 R34 S36 E37 C44 H60 Y61 K62 R14 R34 S36 E37 C44 H60 Y61 K62 2.7.10.2 remove_due_to_license_issue IC50=39000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4f A 2.0 BS01 790 A 1 R14 R34 E37 T38 K62 R14 R34 E37 T38 K62 2.7.10.2 ic50=0.3mM remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCP 1o4g A 1.55 BS01 I59 A 1 R14 R34 S36 E37 T38 T39 C44 R14 R34 S36 E37 T38 T39 C44 2.7.10.2 ic50>5mM remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4h A 2.25 BS01 772 A 1 R14 R34 E37 C44 R14 R34 E37 C44 2.7.10.2 ic50=3.6mM remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4i A 1.75 BS01 219 A 1 R14 R34 S36 E37 T38 C44 H60 Y61 K62 R14 R34 S36 E37 T38 C44 H60 Y61 K62 2.7.10.2 remove_due_to_license_issue IC50=2300000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4j A 1.7 BS01 IS2 A 1 R14 R34 S36 E37 T38 C44 R14 R34 S36 E37 T38 C44 2.7.10.2 ic50=4.4mM remove_due_to_license_issue IC50=4400000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4k A 1.57 BS01 PSN A 1 R14 R34 S36 E37 C44 H60 Y61 K62 R14 R34 S36 E37 C44 H60 Y61 K62 2.7.10.2 remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4n A 1.6 BS01 OXD A 1 R14 R34 S36 E37 T38 C44 R14 R34 S36 E37 T38 C44 2.7.10.2 ic50>40mM remove_due_to_license_issue P12931 14613321 109 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4o A 1.7 BS01 HPS A 1 K54 K59 G95 L96 C97 K54 K59 G95 L96 C97 2.7.10.2 ic50=3.5mM remove_due_to_license_issue IC50=5000000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4o A 1.7 BS02 HPS A 2 R14 R34 S36 E37 H60 K62 R14 R34 S36 E37 H60 K62 2.7.10.2 ic50=3.5mM remove_due_to_license_issue IC50=5000000nM P12931 14613321 400 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4p A 1.9 BS01 791 A 1 R14 R34 S36 E37 T38 C44 H60 K62 R14 R34 S36 E37 T38 C44 H60 K62 2.7.10.2 ic50=2.5mM remove_due_to_license_issue IC50=200000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCP 1o4q A 1.7 BS01 256 A 1 R14 R34 S36 E37 T38 H60 K62 R14 R34 S36 E37 T38 H60 K62 2.7.10.2 ic50=3.2mM remove_due_to_license_issue IC50=3230000000nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT 1o4r A 1.5 BS01 787 A 1 R14 R34 S36 E37 T38 C44 H60 K62 R14 R34 S36 E37 T38 C44 H60 K62 2.7.10.2 ic50=3.9mM remove_due_to_license_issue P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCP 1o5a B 1.68 BS02 696 B 1 C42 H57 C58 A190 Q192 S195 V213 W215 G216 G219 C31 H46 C47 A193 Q195 S198 V216 W218 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.38uM remove_due_to_license_issue Ki=72nM P00749 15522303 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDACQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 1o5b B 1.85 BS02 ESI B 1 D189 A190 Q192 S195 W215 G216 G219 D192 A193 Q195 S198 W218 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=1.7uM remove_due_to_license_issue Ki=210nM P00749 15522303 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDACQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1o5c B 1.63 BS02 CR9 B 1 V41 H57 A190 Q192 S195 V213 G219 V30 H46 A193 Q195 S198 V216 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=6uM remove_due_to_license_issue Ki=30nM P00749 15522303 251 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEASTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDACQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 1o5e H 1.75 BS01 132 H 1 H57 D189 A190 C191 Q192 S195 V213 S214 W215 G219 C220 H41 D178 A179 C180 Q181 S184 V206 S207 W208 G211 C212 3.4.21.106 0004252,0006508 Ki=1.8uM remove_due_to_license_issue Ki=1800nM P05981 15522303 256 IVGGRDTSLGRWPWQVSLRYDGAHLCGGSLLSGDWVLTAAHCFPERNRVLSRWRVFAGAVAQASPHGLQLGVQAVVYHGGYLPFNSNDIALVHLSSPLPLTEYIQPVCLPAAGQALVDGKICTVTGWGNTQYYGQQAGVLQEARVPIISNDVCNGADFYGNQIKPKMFCAGYPEGGIDACQGDSGGPFVCEDSISRTPRWRLCGIVSWGTGCALAQKPGVYTKVSDFREWIFQAIKTHSEASGMVTQL 1o5f H 1.78 BS01 CR9 H 1 L41 H57 P60 D189 A190 C191 S195 V213 L25 H41 P44 D178 A179 C180 S184 V206 3.4.21.106 0004252,0006508 remove_due_to_license_issue Ki=850nM P05981 15522303 256 IVGGRDTSLGRWPWQVSLRYDGAHLCGGSLLSGDWVLTAAHCFPERNRVLSRWRVFAGAVAQASPHGLQLGVQAVVYHGGYLPFNSNDIALVHLSSPLPLTEYIQPVCLPAAGQALVDGKICTVTGWGNTQYYGQQAGVLQEARVPIISNDVCNGADFYGNQIKPKMFCAGYPEGGIDACQGDSGGPFVCEDSISRTPRWRLCGIVSWGTGCALAQKPGVYTKVSDFREWIFQAIKTHSEASGMVTQL 1o5g H 1.75 BS02 CR9 H 1 H57 C58 K60F D189 A190 C191 E192 S195 V213 H43 C44 K52 D192 A193 C194 E195 S198 V218 3.4.21.5 0004252,0005509,0006508,0007596 Ki=11uM remove_due_to_license_issue Ki=11000nM P00734 15522303 393 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1o5m A 2.3 BS01 336 B 1 K164 N165 Y166 H201 K111 N112 Y113 H148 K164 K111 2.5.1.58,2.5.1.59 0004659,0004660,0004661,0004662,0004663,0005515,0005737,0005875,0005953,0005965,0007167,0007323,0008017,0008270,0008284,0008318,0014070,0018342,0018343,0018344,0030971,0034097,0035022,0036094,0042277,0043014,0043066,0045787,0051770,0051771,0060090,0090044,1901363,1904395 remove_due_to_license_issue IC50=1.9nM Q04631 10377218 3001 GFLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSEKFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVWHFRRVLLRSLQKDLQEEMNYITAIIEEQPKNYQVWHHRRVLVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFRLWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRAVLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPNLLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDILNKALELCEILAKEKDTIRKEYWRYIGRSLQSKHS 1o5m B 2.3 BS03 336 B 1 A92 C95 L96 S99 W102 W106 D359 Y361 A70 C73 L74 S77 W80 W84 D337 Y339 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=1.9nM remove_due_to_license_issue Q02293 10377218 3001 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1o5p A -1.00 BS01 CHR A 1 G35 C37 W39 L45 F52 F76 F78 G96 S98 G102 N103 G35 C37 W39 L45 F52 F76 F78 G96 S98 G102 N103 ? 0003677,0006952,0042742 remove_due_to_license_issue P0A3R9 15640161 114 AAPTATVTPSSGLSDGTVVKVAGAGLQAGTAYDVGQCAWVDTGVLACNPADFSSVTADANGSASTSLTVRRSFEGFLFDGTRWGTVDCTTAACQVGLSDAAGNGPEGVAISFN 1o5r A 2.35 BS02 FR9 A 1 H17 D19 F61 L62 F65 M155 D185 T269 D296 H14 D16 F58 L59 F62 M152 D182 T266 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=7.5nM remove_due_to_license_issue P56658 15239652 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1o6h A 2.8 BS02 W37 A 1 F129 W169 A170 T173 P263 W312 F365 D374 D376 W489 F601 F605 F120 W160 A161 T164 P254 W303 F356 D365 D367 W480 F592 F596 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1o6i A 1.7 BS01 0HZ A 1 Y10 G96 W97 D142 E144 M212 Y214 W403 Y8 G94 W95 D140 E142 M210 Y212 W401 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0004553,0005576,0005975,0008061,0030246 Ki=0.65mM remove_due_to_license_issue P11797 12323074 1516 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1o6q A 2.8 BS02 R17 A 1 P263 W312 F365 D376 F437 W489 F601 F605 Y609 P254 W303 F356 D367 F428 W480 F592 F596 Y600 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1o6r A 2.7 BS02 R19 A 1 F129 P263 W312 D374 W489 F601 F605 Y609 F120 P254 W303 D365 W480 F592 F596 Y600 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1o79 A 2.8 BS01 R23 A 1 F129 P263 W312 F365 D374 D377 F437 W489 F601 F605 F120 P254 W303 F356 D365 D368 F428 W480 F592 F596 E45 E93 R127 W169 Q262 W312 F365 D374 D376 D377 Y420 H451 W489 Y495 F601 F605 Y609 E36 E84 R118 W160 Q253 W303 F356 D365 D367 D368 Y411 H442 W480 Y486 F592 F596 Y600 4.2.1.129,5.4.99.17 0005811,0005886,0008610,0016104,0016829,0016853,0016866,0051007 remove_due_to_license_issue P33247 12747780 800 AYARTLDRAVEYLLSCQKDEGYWWGPLLSNVTMEAEYVLLCHILDRVDRDRMEKIRRYLLHEQREDGTWALYPGGPPDLDTTIEAYVALKYIGMSRDEEPMQKALRFIQSQGGIESSRVFTRMWLALVGEYPWEKVPMVPPEIMFLGKRMPLNIYEFGSWARATVVALSIVMSRQPVFPLPERARVPELYETDVPPRRRGAKGGGGWIFDALDRALHGYQKLSVHPFRRAAEIRALDWLLERQAGDGSWGGIQPPWFYALIALKILDMTQHPAFIKGWEGLELYGVELDYGGWMFQASISPVWDTGLAVLALRAAGLPADHDRLVKAGEWLLDRQITVPGDWAVKRPNLKPGGFAFQFDNVYYPDVDDTAVVVWALNTLRLPDERRRRDAMTKGFRWIVGMQSSNGGWGAYDVDNTSDLPNHIPFCDFGEVTDPPSEDVTAHVLECFGSFGYDDAWKVIRRAVEYLKREQKPDGSWFGRWGVNYLYGTGAVVSALKAVGIDTREPYIQKALDWVEQHQNPDGGWGEDCRSYEDPAYAGKGASTPSQTAWALMALIAGGRAESEAARRGVQYLVETQRPDGGWDEPYYTGTGFPGDFYLGYTMYRHVFPTLALGRYKQAI 1o7o A 1.97 BS04 UDP A 1 F134 A135 V136 Y139 I198 R202 D225 V226 D227 K359 Y361 R365 F53 A54 V55 Y58 I117 R121 D144 V145 D146 K278 Y280 R284 Q247 H280 W314 Q317 W356 R365 Q166 H199 W233 Q236 W275 R284 2.4.1.87 0005975,0016020,0016758 Kd=0.032mM remove_due_to_license_issue P14769 14621997 1371 KLKLSDWFNPFKRPEVVTMTKWKAPVVWEGTYNRAVLDNYYAKQKITVGLTVFAVGRYIEHYLEEFLTSANKHFMVGHPVIFYIMVDDVSRMPLIELGPLRSFKVFKIKPEKRWQDISMMRMKTIGEHIVAHIQHEVDFLFCMDVDQVFQDKFGVETLGESVAQLQAWWYKADPNDFTYERRKESAAYIPFGEGDFYYHAAIFGGTPTQVLNITQECFKGILKDKKNDIEAQWHDQSHLNKYFLLNKPTKILSPEYCWDYHIGLPADIKLVKMSWQTKEYNVVRNNV 1o86 A 2.0 BS03 LPR A 1 Q281 H353 A354 H383 E384 H387 E411 K511 F512 H513 V518 Y520 Y523 Q242 H314 A315 H344 E345 H348 E372 K468 F469 H470 V475 Y477 Y480 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H470 Y480 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue IC50=1.2nM P12821 12540854 702 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWP 1o9e A 2.6 BS01 FSC A 1 N49 V53 F126 K129 P174 I175 K221 D222 N45 V49 F122 K125 P170 I171 K213 D214 ? 0005737,0007165,0008104 remove_due_to_license_issue P93343 12606564 1241 PTAREENVYMAKLAEQAERYEEMVEFMEKVSNSLGSEELTVEERNLLSVAYKNVIGARRASWRIISSIEQKEESRGNEEHVNSIREYRSKIENELSKICDGILKLLDAKLIPSAASGDSKVFYLKMKGDYHRYLAEFKTGAERKEAAESTLTAYKAAQDIATTELAPTHPIRLGLALNFSVFYYEILNSPDRACNLAKQAFDEAIAELDTLYKDSTLIMQLLRDNLTLWTS 1oar H 2.23 BS01 AZN H 1 W33 R50 K59 M99 Y105 W33 R50 K59 M99 Y105 Kd=40nM remove_due_to_license_issue 12610298 500 EVQLQQSGAELVKPGASVKLSCKASGYTFTSYWMHWVKQRPGRGLEWIGRIDPNGGGTKYNEKFKSKATLTVDKPSSTAYMQLSSLTSEDSAVYYCARMWYYGTYYFDYWGQGTTLTVSSAA 1oar L 2.23 BS01 AZN H 1 Y34 N36 W93 Y33 N35 W92 ? 0002250,0006955,0019814 remove_due_to_license_issue P01724 12610298 500 AVVTQESALTTSPGETVTLTCRSSTGAVTTSNYANWVQEKPDHLFTGLIGGTNNRAPGVPARFSGSLIGNKAALTITGAQTEDEAIYFCALWYSNHLVFGGGTKLTVL 1oau H 1.8 BS01 DNF H 1 W33 R50 M99 Y105 W33 R50 M99 Y105 remove_due_to_license_issue 12610298 501 EVQLQQSGAELVKPGASVKLSCKASGYTFTSYWMHWVKQRPGRGLEWIGRIDPNGGGTKYNEKFKSKATLTVDKPSSTAYMQLSSLTSEDSAVYYCARMWYYGTYYFDYWGQGTTLTVSSAA 1oau L 1.8 BS01 DNF H 1 Y34 W93 Y33 W92 ? 0002250,0006955,0019814 remove_due_to_license_issue P01724 12610298 501 AVVTQESALTTSPGETVTLTCRSSTGAVTTSNYANWVQEKPDHLFTGLIGGTNNRAPGVPARFSGSLIGNKAALTITGAQTEDEAIYFCALWYSNHLVFGGGTKLTVL 1oay H 2.66 BS01 FUR H 1 W33 H35 K59 M99 W32 H34 K58 M98 remove_due_to_license_issue 12610298 500 VQLQQSGAELVKPGASVKLSCKASGYTFTSYWMHWVKQRPGRGLEWIGRIDPNGGGTKYNLKFKSKATLTVDKPSSTAYMQLSSLTSEDSAVYYCARMWYYGTYYFDYWGQGTTLTVSSAA 1oay L 2.66 BS01 FUR H 1 W93 L98 W92 L97 ? 0002250,0006955,0019814 remove_due_to_license_issue P01724 12610298 500 AVVTQESALTTSPGETVTLTCRSSTGAVTTSNYANWVQEKPRHLFTGLIGGTNNRAPGVPARFSGSLIGNKAALTITGAQTEDEAIYFCALWYSNHLVFGGGTKLTVL 1oba A 2.45 BS01 CHT A 1 W223 W230 Y252 S277 W222 W229 Y251 S276 D10 D92 E94 D182 D9 D91 E93 D181 3.2.1.17 0003796,0005515,0009253,0016798,0016998,0031640,0042742,0044659 Kd=3.6mM remove_due_to_license_issue P15057 14527392 1340 VKKNDLFVDVSSHNGYDITGILEQMGTTNTIIKISESTTYLNRCLSAQVEQSNPIGFYHFARFGGDVAEAEREAQFFLDNVPMQVKYLVLDYEDDPSGDAQANTNACLRFMQMIADAGYKPIYYSYKPFTHDNVDYQQILAQFPNSLWIAGYGLNDGTANFEYFPSMDGIRWWQYSSNPFDKNIVLLDDEEDDKPKTAGTWKQDSKGWWFRRNNGSFPYNKWEKIGGVWYYFDSKGYCLTSEWLKDNEKWYYLKDNGAMATGWVLVGSEWYYMDDSGAMVTGWVKYKNNWYYMTNERGNMVSNEFIKSGKGWYFMNTNGELADNPSFTKEPDGLITVA 1oba A 2.45 BS02 CHT A 2 W202 W209 Y231 W201 W208 Y230 D10 D92 E94 D182 D9 D91 E93 D181 3.2.1.17 0003796,0005515,0009253,0016798,0016998,0031640,0042742,0044659 Kd=3.6mM remove_due_to_license_issue P15057 14527392 1341 VKKNDLFVDVSSHNGYDITGILEQMGTTNTIIKISESTTYLNRCLSAQVEQSNPIGFYHFARFGGDVAEAEREAQFFLDNVPMQVKYLVLDYEDDPSGDAQANTNACLRFMQMIADAGYKPIYYSYKPFTHDNVDYQQILAQFPNSLWIAGYGLNDGTANFEYFPSMDGIRWWQYSSNPFDKNIVLLDDEEDDKPKTAGTWKQDSKGWWFRRNNGSFPYNKWEKIGGVWYYFDSKGYCLTSEWLKDNEKWYYLKDNGAMATGWVLVGSEWYYMDDSGAMVTGWVKYKNNWYYMTNERGNMVSNEFIKSGKGWYFMNTNGELADNPSFTKEPDGLITVA 1ocn A 1.31 BS01 IFM A 1 W137 Y174 S186 A309 K399 D405 W47 Y84 S96 A219 K309 D315 Y174 R179 D180 S186 D226 D405 Y84 R89 D90 S96 D136 D315 3.2.1.91 0004553,0005975,0030245 remove_due_to_license_issue Q9C1S9 12744312 452 GNPFEGVQLWANNYYRSEVHTLAIPQITDPALRAAASAVAEVPSFQWLDRNVTVDTLLVQTLSEIREANQAGANPQYAAQIVVYDLPDRDCAAAASNGEWAIANNGVNNYKAYINRIREILISFSDVRTILVIEPDSLANMVTNMNVPKCSGAASTYRELTIYALKQLDLPHVAMYMDAGHAGWLGWPANIQPAAELFAKIYEDAGKPRAVRGLATNVANYNAWSVSSPPPYTSPNPNYDEKHYIEAFRPLLEARGFPAQFIVDQGRSGKQPTGQKEWGHWCNAIGTGFGMRPTANTGHQYVDAFVWVKPGGECDGTSDTTAARYAYHCGLEDALKPAPEAGQWFNEYFIQLLRNANPPF 1ocn A 1.31 BS02 BGC A 1 W137 D139 S186 K399 P400 E403 W47 D49 S96 K309 P310 E313 Y174 R179 D180 S186 D226 D405 Y84 R89 D90 S96 D136 D315 3.2.1.91 0004553,0005975,0030245 remove_due_to_license_issue Q9C1S9 12744312 453 GNPFEGVQLWANNYYRSEVHTLAIPQITDPALRAAASAVAEVPSFQWLDRNVTVDTLLVQTLSEIREANQAGANPQYAAQIVVYDLPDRDCAAAASNGEWAIANNGVNNYKAYINRIREILISFSDVRTILVIEPDSLANMVTNMNVPKCSGAASTYRELTIYALKQLDLPHVAMYMDAGHAGWLGWPANIQPAAELFAKIYEDAGKPRAVRGLATNVANYNAWSVSSPPPYTSPNPNYDEKHYIEAFRPLLEARGFPAQFIVDQGRSGKQPTGQKEWGHWCNAIGTGFGMRPTANTGHQYVDAFVWVKPGGECDGTSDTTAARYAYHCGLEDALKPAPEAGQWFNEYFIQLLRNANPPF 1ocn A 1.31 BS03 IFM A 2 N234 H271 W274 N144 H181 W184 Y174 R179 D180 S186 D226 D405 Y84 R89 D90 S96 D136 D315 3.2.1.91 0004553,0005975,0030245 remove_due_to_license_issue Q9C1S9 12744312 454 GNPFEGVQLWANNYYRSEVHTLAIPQITDPALRAAASAVAEVPSFQWLDRNVTVDTLLVQTLSEIREANQAGANPQYAAQIVVYDLPDRDCAAAASNGEWAIANNGVNNYKAYINRIREILISFSDVRTILVIEPDSLANMVTNMNVPKCSGAASTYRELTIYALKQLDLPHVAMYMDAGHAGWLGWPANIQPAAELFAKIYEDAGKPRAVRGLATNVANYNAWSVSSPPPYTSPNPNYDEKHYIEAFRPLLEARGFPAQFIVDQGRSGKQPTGQKEWGHWCNAIGTGFGMRPTANTGHQYVDAFVWVKPGGECDGTSDTTAARYAYHCGLEDALKPAPEAGQWFNEYFIQLLRNANPPF 1ocn A 1.31 BS04 BGC A 2 D226 H271 N310 W371 D136 H181 N220 W281 Y174 R179 D180 S186 D226 D405 Y84 R89 D90 S96 D136 D315 3.2.1.91 0004553,0005975,0030245 remove_due_to_license_issue Q9C1S9 12744312 455 GNPFEGVQLWANNYYRSEVHTLAIPQITDPALRAAASAVAEVPSFQWLDRNVTVDTLLVQTLSEIREANQAGANPQYAAQIVVYDLPDRDCAAAASNGEWAIANNGVNNYKAYINRIREILISFSDVRTILVIEPDSLANMVTNMNVPKCSGAASTYRELTIYALKQLDLPHVAMYMDAGHAGWLGWPANIQPAAELFAKIYEDAGKPRAVRGLATNVANYNAWSVSSPPPYTSPNPNYDEKHYIEAFRPLLEARGFPAQFIVDQGRSGKQPTGQKEWGHWCNAIGTGFGMRPTANTGHQYVDAFVWVKPGGECDGTSDTTAARYAYHCGLEDALKPAPEAGQWFNEYFIQLLRNANPPF 1ocq A 1.08 BS01 IFM A 1 Y66 H101 E139 Y202 E228 A234 T235 G236 W262 Y63 H98 E136 Y199 E225 A231 T232 G233 W259 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 12812472 500 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1ocq A 1.08 BS02 BGC A 1 H35 Y66 W262 K267 E269 H32 Y63 W259 K264 E266 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 12812472 501 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1odi A 2.4 BS02 ADN A 1 M65 T90 A91 G92 E156 F159 F178 E179 M180 E181 N204 M64 T89 A90 G91 E155 F158 F177 E178 M179 E180 N203 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=62uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odi A 2.4 BS03 ADN B 1 H5 R44 H4 R43 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=62uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odi B 2.4 BS01 ADN A 1 H5 R44 H4 R43 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=62uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odi B 2.4 BS03 ADN B 1 T90 A91 G92 E156 F159 E179 M180 E181 N204 T89 A90 G91 E155 F158 E178 M179 E180 N203 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=62uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odj A 2.4 BS02 GMP A 1 T90 A91 G92 E156 F159 F178 E179 M180 E181 T89 A90 G91 E155 F158 F177 E178 M179 E180 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=80uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odj A 2.4 BS03 GMP B 1 H5 R44 H4 R43 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=80uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odj B 2.4 BS01 GMP A 1 H5 R44 H4 R43 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=80uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1odj B 2.4 BS03 GMP B 1 T90 A91 G92 E156 F159 E179 M180 E181 T89 A90 G91 E155 F158 E178 M179 E180 H5 G21 R25 R44 E76 R87 T90 S203 N204 I206 L217 H4 G20 R24 R43 E75 R86 T89 S202 N203 I205 L216 2.4.2.3 0003824,0005829,0009116,0009164,0016757,0016763 Kd=80uM remove_due_to_license_issue Q5SID9 15046984 1237 SPIHVRAHPGDVAERVLLPGDPGRAEWIAKTFLQNPRRYNDHRGLWGYTGLYKGVPVSVQTTGMGTPSAAIVVEELVRLGARVLVRVGTAGAASSDLAPGELIVAQGAVPLDGTTRQYLEGRPYAPVPDPEVFRALWRRAEALGYPHRVGLVASEDAFYATTPEEARAWARYGVLAFEMEASALFLLGRMRGVRTGAILAVSNRIGDPELAPPEVLQEGVRRMVEVALEAVLEV 1ody A 2.0 BS01 LP1 A 1 D25 G27 A28 D29 I47 G48 G49 P81 V82 I84 D25 G27 A28 D29 I47 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8nM remove_due_to_license_issue P04585 9827997 201 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ody B 2.0 BS01 LP1 A 1 D25 G27 A28 D29 I47 G48 G49 P81 D25 G27 A28 D29 I47 G48 G49 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9827997 201 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1oe0 A 2.4 BS01 TTP A 1 I29 G30 S31 G32 K33 T34 W57 Y70 F80 Q81 E104 R105 A110 F114 R167 R169 E172 I18 G19 S20 G21 K22 T23 W46 Y59 F69 Q70 E93 R94 A99 F103 R156 R158 E161 E52 R105 E41 R94 2.7.1.145 0004136,0004137,0004138,0004797,0004849,0005524,0005737,0005739,0006139,0006170,0006222,0009157,0009224,0016301,0019136,0043174,0043771,0071897,1901293 Ki=5.3nM remove_due_to_license_issue Q9XZT6 12741827 300 TKYAEGTQPFTVLIEGNIGSGKTTYLNHFEKYKNDICLLTEPVEKWRNVNGVNLLELMYKDPKKWAMPFQSYVTLTMLQSHTAPTNKKLKIMERSIFSARYCFVENMRRNGSLEQGMYNTLEEWYKFIEESIHVQADLIIYLRTSPEVAYERIRQRARSEESCVPLKYLQELHELHEDWLIHQRRPQSCKVLVLDADL 1oe7 A 1.8 BS01 GSH A 1 Y10 F11 R16 W41 K45 R52 L53 E70 S71 Y7 F8 R13 W38 K42 R49 L50 E67 S68 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=9uM remove_due_to_license_issue P30114 12939136 301 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRA 1oe7 B 1.8 BS01 GSH B 1 F11 R16 W41 K45 R52 L53 E70 S71 F7 R12 W37 K41 R48 L49 E66 S67 Y10 R16 R21 Y6 R12 R17 2.5.1.18 0004364,0006749,0016740 Kd=9uM remove_due_to_license_issue P30114 12939136 301 HIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRA 1oe8 A 1.65 BS01 GSH A 1 R16 W41 K45 R52 L53 E70 S71 R13 W38 K42 R49 L50 E67 S68 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=9uM remove_due_to_license_issue P30114 12939136 301 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRA 1oe8 B 1.65 BS01 GSH B 1 R16 W41 K45 R52 L53 E70 S71 R14 W39 K43 R50 L51 E68 S69 Y10 R16 R21 Y8 R14 R19 2.5.1.18 0004364,0006749,0016740 Kd=9uM remove_due_to_license_issue P30114 12939136 301 GDHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRA 1ogg A 1.97 BS01 AMI A 1 Y10 F51 W97 N142 E144 M212 Y214 D215 Y292 M401 W403 Y8 F49 W95 N140 E142 M210 Y212 D213 Y290 M399 W401 D140 N142 E144 Y214 D138 N140 E142 Y212 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 14726210 1501 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDINWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1ogu A 2.6 BS01 ST8 A 1 I10 E12 G13 A31 F80 E81 L83 L134 I13 E15 G16 A34 F80 E81 L83 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue Ki=2400nM, IC50=34nM P24941 12941338 1298 PGSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 1ogz A 2.3 BS01 EQU A 1 Y14 S58 L63 F86 D99 F116 Y14 S58 L63 F86 D99 F116 Y14 D38 A96 D99 Y14 D38 A96 D99 5.3.3.1 0004769,0008202,0016853 Kd=1.4uM remove_due_to_license_issue P00947 12852789 1126 MNTPEHMTAVVQRYVAALNAGDLDGIVALFADDATVEDAVGSEPRSGTAAIREFYANSLKLPLAVELTQEVRAVANEAAFAFIVSFEYQGRKTVVAPIDHFRFNGAGKVVSMRALFGEKNIHAGA 1ohr A 2.1 BS01 1UN A 1 D25 G27 A28 D29 D30 P81 I84 D25 G27 A28 D29 D30 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=2nM remove_due_to_license_issue Q9Q288 9397180 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ohr B 2.1 BS01 1UN A 1 D25 G27 V32 G49 I50 I84 D25 G27 V32 G49 I50 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q9Q288 9397180 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1oi9 A 2.1 BS01 N20 A 1 I10 E12 A31 V64 F80 L83 H84 Q85 L134 I11 E13 A32 V64 F80 L83 H84 Q85 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=69nM remove_due_to_license_issue IC50=69nM P24941 15239650 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1oif A 2.12 BS01 IFM A 1 Q20 E166 Y295 E351 W398 E405 W406 F414 Q18 E164 Y293 E349 W396 E403 W404 F412 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E349 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Ka=51450000M^-1 remove_due_to_license_issue Q08638 14624580 1447 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLED 1oim A 2.15 BS01 NOJ A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 Q18 H119 N163 E164 Y292 E348 W395 E402 W403 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N290 Y292 E348 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Ka=210000M^-1 remove_due_to_license_issue Q08638 14624580 1447 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLED 1oiq A 2.31 BS01 HDU A 1 A31 K33 F80 E81 L83 L134 A27 K29 F62 E63 L65 L116 D127 K129 Q131 N132 D145 T165 D109 K111 Q113 N114 D127 T131 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=2.9uM remove_due_to_license_issue IC50=2884nM P24941 12941325 1299 MENFQKVEKIGGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1oir A 1.91 BS01 HDY A 1 V18 A31 F80 L83 H84 K89 L134 V18 A31 F71 L74 H75 K80 L125 D127 K129 Q131 N132 D145 T158 T165 D118 K120 Q122 N123 D136 T149 T156 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.032uM remove_due_to_license_issue IC50=32nM P24941 12941325 1298 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1oit A 1.6 BS01 HDT A 1 I10 V18 A31 L83 H84 Q85 D86 K89 L134 I8 V16 A28 L69 H70 Q71 D72 K75 L120 D127 K129 Q131 N132 D145 T165 D113 K115 Q117 N118 D131 T140 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50<0.003uM remove_due_to_license_issue IC50=1nM P24941 12941325 1299 NFQKVEKIGEGTYGVVYKARNKLGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLSFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1oiu A 2.0 BS01 N76 A 1 I10 E12 G13 A31 V64 F80 E81 F82 L83 H84 L134 I13 E15 G16 A34 V64 F80 E81 F82 L83 H84 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.21uM remove_due_to_license_issue IC50=210nM P24941 15239650 1298 PGSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 1oiy A 2.4 BS01 N41 A 1 I10 E12 A31 V64 F80 E81 L83 H84 Q85 D86 Q131 L134 I11 E13 A32 V62 F78 E79 L81 H82 Q83 D84 Q129 L132 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=64nM remove_due_to_license_issue IC50=64nM P24941 15239650 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1okl A 2.1 BS02 MNS A 1 H94 H119 V121 F130 L140 L197 T198 T199 H90 H115 V117 F126 L136 L193 T194 T195 H64 H94 H96 E106 H119 T198 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.93uM remove_due_to_license_issue P00918 8557623 862 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1oky A 2.3 BS01 STU A 1 L88 G89 V96 A109 K111 Y161 A162 G165 E166 E209 L212 T222 L17 G18 V25 A38 K40 Y90 A91 G94 E95 E138 L141 T151 D205 K207 E209 N210 D223 T245 D134 K136 E138 N139 D152 T168 2.7.11.1 0004672,0004674,0005524,0006468 ic50=6.5nM remove_due_to_license_issue O15530 12892559 1368 PQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 1okz A 2.51 BS01 UCN A 1 L88 G89 V96 A109 K111 L159 Y161 A162 G165 E166 E209 N210 L212 T222 D223 L16 G17 V24 A37 K39 L87 Y89 A90 G93 E94 E137 N138 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 12892559 1370 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLNSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 1om1 A 1.68 BS01 IQA A 1 V45 V53 I66 K68 F113 V116 M163 I174 D175 V39 V47 I60 K62 F107 V110 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.17uM remove_due_to_license_issue P28523 12816539 338 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 1omh A 1.95 BS01 dna B 0 M1 L2 S3 H4 M5 V6 S72 A73 R75 Q76 K79 R81 S89 A90 P91 K92 R128 Q129 K130 I131 Q132 R154 Q159 R172 R178 A179 N182 D183 N218 R226 S233 R235 T236 K258 K262 R266 M1 L2 S3 H4 M5 V6 S61 A62 R64 Q65 K68 R70 S78 A79 P80 K81 R117 Q118 K119 I120 Q121 R143 Q148 R161 R167 A168 N171 D172 N207 R215 S222 R224 T225 K247 K251 R255 ? remove_due_to_license_issue Q47673 14625590 1 ~ 25 MLSHMVLTRQDIGRAASYYGDASEWQGKGAEELGLSGEVDSKRFRELLAGNIGEGHRIMRSATRQDSKERIGLDLTFSAPKSVSLQALVAGDAEIIKAHDRAVARTLEQAEARAQARQKIQGKTRIETTGNLVIGKFRHETSRERDPQLHTHAVILNMTKRSDGQWRALKNDEIVKATRYLGAVYNAELAHELQKLGYQLRYGKDGNFDLAHIDRQQIEGFSKRTEQIAEWYAARGLDPNSVSLEQKQAAKVLSRAKKTSVDREALRAEWQATAKELGIDFS 1ong A 1.1 BS03 WY4 A 1 S70 Y105 S130 N132 N170 G236 A237 S45 Y80 S105 N107 N145 G211 A212 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 14609325 400 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 1onh A 1.38 BS01 WY4 A 1 S64 L119 Q120 N152 G320 S321 T322 G323 S63 L118 Q119 N151 G319 S320 T321 G322 S64 K67 Y112 V121 Y150 G156 E275 K318 S321 S63 K66 Y111 V120 Y149 G155 E274 K317 S320 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q59401 14609325 400 PVSEKQLAEVVANTVTPLMKAQSVPGMAVAVIYQGKPHYYTFGKADIAANKPVTPQTLFELGSISKTFTGVLGGDAIARGEISLDDPVTRYWPQLTGKQWQGIRMLDLATYTAGGLPLQVPDEVTDNASLLRFYQNWQPQWKPGTTRLYANASIGLFGALAVKPSGMPYEQAMTTRVLKPLKLDHTWINVPKAEEAHYAWGYRDGKAVRAVRVSPGMLDAQAYGVKTNVQDMANWVMANMAPENVADASLKQGIALAQSRYWRIGSMYQGLGWEMLNWPVEANTVVEGSDSKVALAPLPVAEVNPPAPPVKASWVHKTGSTGGFGSYVAFIPEKQIGIVMLANTSYPNPARVEAAYHILEALQ 1onp A 2.5 BS02 FOM A 1 E152 S186 W212 N227 K228 E152 S186 W212 N227 K228 1.1.1.267 0008299,0016491,0019288,0030145,0030604,0042802,0046872,0051484,0070402,1990065 remove_due_to_license_issue IC50=30nM P45568 12621040 1001 MKQLTILGSTGSIGCSTLDVVRHNPEHFRVVALVAGKNVTRMVEQCLEFSPRYAVMDDEASAKLLKTMLQQQGSRTEVLSGQQAACDMAALEDVDQVMAAIVGAAGLLPTLAAIRAGKTILLANKESLVTCGRLFMDAVKQSKAQLLPVDSEHNAIFQSLPQPIQHNLGYADLEQNGVVSILLTGSGGPFRETPLRDLATMTPDQACRHPNWSMGRKISVDSATMMNKGLEYIEARWLFNASASQMEVLIHPQSVIHSMVRYQDGSVLAQLGEPDMRTPIAHTMAWPNRVNSGVKPLDFCKLSALTFAAPDYDRYPCLKLAMEAFEQGQAATTALNAANEITVAAFLAQQIRFTDIAALNLSVLEKMDMREPQCVDDVLSVDANAREVARKEVMRLA 1ony A 2.15 BS01 588 A 1 Y46 D48 K120 C215 S216 A217 I219 G220 R221 Q262 T263 Q266 G283 Y45 D47 K119 C214 S215 A216 I218 G219 R220 Q261 T262 Q265 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=170nM P18031 12747781 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1onz A 2.4 BS01 968 A 1 Y46 K120 C215 S216 A217 I219 G220 R221 Q262 T263 Q266 G283 Y45 K119 C214 S215 A216 I218 G219 R220 Q261 T262 Q265 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=25119nM P18031 12747781 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1oq5 A 1.5 BS02 CEL A 1 N67 Q92 H94 H96 H119 F131 L198 T199 T200 P202 N64 Q89 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=21nM remove_due_to_license_issue Ki=21nM, IC50=21nM P00918 14736236 701 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1ork A 2.4 BS01 ATC A 1 H64 N82 F86 H100 R104 Q116 I134 S138 H63 N81 F85 H99 R103 Q115 I133 S137 ? 0000976,0003677,0003700,0006355,0045892,0046677,0046872 Kd=1.56nM remove_due_to_license_issue P0ACT4 9878420 222 SRLNRESVIDAALELLNETGIDGLTTRKLAQKLGIEQPTLYWHVKNKRALLDALAVEILARHHDYSLPAAGESWQSFLRNNAMSFRRALLRYRDGAKVHLGTRPDEKQYDTVETQLRFMTENGFSLRDGLYAISAVSHFTLGAVLEQQEHTAANLPPLLREALQIMDSDDGEQAFLHGLESLIRGFEVQLTALLQIV 1orw A 2.84 BS01 PHI A 1 R125 E205 E206 F357 R358 Y662 N710 R87 E167 E168 F319 R320 Y624 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P22411 12690074 801 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 1orw A 2.84 BS02 P2Y A 1 Y547 S630 Y631 Y662 Y666 Y509 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P22411 12690074 802 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 1os0 A 2.1 BS06 0PQ A 1 N112 A113 F114 V139 H142 E143 H146 E166 I188 L202 R203 H231 N112 A113 F114 V139 H142 E143 H146 E166 I188 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=0.93uM remove_due_to_license_issue P00800 12832763 605 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1os5 A 2.2 BS01 NH1 A 1 R422 M423 H475 S476 Y477 L497 W528 R422 M423 H475 S476 Y477 L497 W528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.14uM remove_due_to_license_issue P26663 12805457 901 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 1osb A 2.65 BS01 dna B 0 M1 S3 H4 S72 A73 T74 R75 Q76 D77 K79 R81 S89 A90 P91 K92 R128 K130 Q132 T152 R154 Q159 H161 H163 R172 R178 A179 N182 D183 K215 N218 R226 S233 R235 T236 I239 L255 K258 K262 R266 M1 S3 H4 S66 A67 T68 R69 Q70 D71 K73 R75 S83 A84 P85 K86 R122 K124 Q126 T146 R148 Q153 H155 H157 R166 R172 A173 N176 D177 K209 N212 R220 S227 R229 T230 I233 L249 K252 K256 R260 ? remove_due_to_license_issue Q47673 14625590 1 ~ 25 MLSHMVLTRQDIGRAASYYEDGADGDASEWQGKGAEELGLSGEVDSKRFRELLAGNIGEGHRIMRSATRQDSKERIGLDLTFSAPKSVSLQALVAGDAEIIKAHDRAVARTLEQAEARAQARQKIQGKTRIETTGNLVIGKFRHETSRERDPQLHTHAVILNMTKRSDGQWRALKNDEIVKATRYLGAVYNAELAHELQKLGYQLRYGKDGNFDLAHIDRQQIEGFSKRTEQIAEWYAARGLDPNSVSLEQKQAAKVLSRAKKTSVDREALRAEWQATAKELGIDFS 1osb C 2.65 BS01 dna D 0 M1 S3 H4 S72 A73 R75 Q76 K79 R81 S89 A90 P91 K92 R128 Q129 K130 Q132 R154 Q159 H161 H163 R172 R178 A179 N182 D183 K187 N218 R226 S233 R235 T236 I239 L255 K258 K262 R266 M1 S3 H4 S62 A63 R65 Q66 K69 R71 S79 A80 P81 K82 R118 Q119 K120 Q122 R144 Q149 H151 H153 R162 R168 A169 N172 D173 K177 N208 R216 S223 R225 T226 I229 L245 K248 K252 R256 ? remove_due_to_license_issue Q47673 14625590 1 ~ 25 MLSHMVLTRQDIGRAASYYEGDASEWQGKGAEELGLSGEVDSKRFRELLAGNIGEGHRIMRSATRQDSKERIGLDLTFSAPKSVSLQALVAGDAEIIKAHDRAVARTLEQAEARAQARQKIQGKTRIETTGNLVIGKFRHETSRERDPQLHTHAVILNMTKRSDGQWRALKNDEIVKATRYLGAVYNAELAHELQKLGYQLRYGKDGNFDLAHIDRQQIEGFSKRTEQIAEWYAARGLDPNSVSLEQKQAAKVLSRAKKTSVDREALRAEWQATAKELGIDF 1oss A 1.93 BS02 BEN A 1 D189 P190 C191 S195 V213 W215 G219 D166 P167 C168 S172 V191 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H37 D82 Q169 G170 D171 S172 G173 3.4.21.4 0004252,0006508,0008236 Ki=16.4uM remove_due_to_license_issue P00775 12885239 246 VVGGTRAAQGEFPFMVRLSMGCGGALYAQDIVLTAAHCVSGSGNNTSITATGGVVDLQSSSAVKVRSTKVLQAPGYNGTGKDWALIKLAQPINQPTLKIATTTAYNQGTFTVAGWGANREGGSQQRYLLKANVPFVSDAACRSAYGNELVANEEICAGYPDTGGVDPCQGDSGGPMFRKDNADEWIQVGIVSWGYGCARPGYPGVYTEVSTFASAIASAARTL 1oth A 1.85 BS01 PAO A 1 S90 T91 R92 T93 R141 L163 H168 N199 D263 S267 M268 C303 L304 R330 S57 T58 R59 T60 R108 L130 H135 N166 D230 S234 M235 C270 L271 R297 R92 T93 V120 R141 H168 Q171 D263 C303 R330 R59 T60 V87 R108 H135 Q138 D230 C270 R297 2.1.3.3 0000050,0001889,0004585,0005543,0005739,0005743,0005759,0006520,0006526,0006591,0006593,0007494,0009410,0010043,0016597,0016740,0016743,0019240,0031667,0032868,0042301,0042450,0042802,0055081,0070781,0097272 remove_due_to_license_issue Ki=100nM P00480 9852088 355 KVQLKGRDLLTLKNFTGEEIKYMLWLSADLKFRIKQKGEYLPLLQGKSLGMIFEKRSTRTRLSTETGFALLGGHPCFLTTQDIHLGVNESLTDTARVLSSMADAVLARVYKQSDLDTLAKEASIPIINGLSDLYHPIQILADYLTLQEHYSSLKGLTLSWIGDGNNILHSIMMSAAKFGMHLQAATPKGYEPDASVTKLAEQYAKENGTKLLLTNDPLEAAHGGNVLITDTWISMGREEEKKKRLQAFQGYQVTMKTAKVAASDWTFLHCLPRKPEEVDDEVFYSPRSLVFPEAENRKWTIMAVMVSLLTDYSPQLQKPKF 1ouk A 2.5 BS01 084 A 1 Y35 V38 A51 K53 L75 L104 T106 L108 M109 A111 D168 Y32 V35 A48 K50 L72 L101 T103 L105 M106 A108 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.13nM remove_due_to_license_issue IC50=110nM Q16539 12897767 501 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 1ouy A 2.5 BS01 094 A 1 Y35 V38 A51 K53 I84 L104 V105 T106 H107 L108 M109 G110 A111 A157 Y32 V35 A48 K50 I81 L101 V102 T103 H104 L105 M106 G107 A108 A154 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=4.3nM remove_due_to_license_issue Q16539 12897767 501 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 1ouz A 2.41 BS01 dna C 0 K45 R55 K57 P61 R63 P65 R82 K88 K44 R54 K56 P60 R62 P64 R81 K87 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 50 ~ 16 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1ouz A 2.41 BS02 dna D 0 G48 N51 K86 G47 N50 K85 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 15 ~ 29 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1ouz A 2.41 BS03 dna E 0 T4 K5 K57 R60 R63 N64 P65 K66 I73 R76 V78 T3 K4 K56 R59 R62 N63 P64 K65 I72 R75 V77 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 30 ~ 49 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1ouz B 2.41 BS01 dna C 0 K3 S4 K27 R46 G47 S50 R59 R62 N63 P64 L72 K75 K81 G83 K84 K3 S4 K27 R46 G47 S50 R59 R62 N63 P64 L72 K75 K81 G83 K84 ? 0003677,0005694,0005737,0005829,0006310,0006351,0006355,0006417,0030527,0043565,1990177 remove_due_to_license_issue P0A6Y1 12842466 50 ~ 16 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIAIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIYG 1ouz B 2.41 BS02 dna E 0 A44 R46 H54 R56 H79 A44 R46 H54 R56 H79 ? 0003677,0005694,0005737,0005829,0006310,0006351,0006355,0006417,0030527,0043565,1990177 remove_due_to_license_issue P0A6Y1 12842466 30 ~ 49 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIAIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIYG 1ove A 2.1 BS01 358 A 1 Y35 A51 T106 H107 M109 G110 A111 D168 Y32 A48 T103 H104 M106 G107 A108 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.74nM remove_due_to_license_issue IC50=0.740000nM Q16539 12897767 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1owd A 2.32 BS01 497 A 1 H45 D49 D191 S192 Q194 W217 G220 H46 D50 D192 S193 Q195 W218 G221 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=6.3nM remove_due_to_license_issue Ki=6.3nM P00749 14711304 1001 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1owe A 1.6 BS01 675 A 1 H54 H106 D205 S206 Q208 W231 G234 H46 H94 D192 S193 Q195 W218 G221 H54 D109 Q208 G209 D210 S211 G212 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.631uM remove_due_to_license_issue Ki=631nM, IC50=13000nM P00749 14711304 1001 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1owf A 1.95 BS01 dna C 0 K45 R55 K57 P61 R63 P65 R82 K88 K44 R54 K56 P60 R62 P64 R81 K87 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 50 ~ 16 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1owf A 1.95 BS02 dna D 0 G48 N51 K86 G47 N50 K85 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 15 ~ 29 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1owf A 1.95 BS03 dna E 0 T4 K5 K57 R60 R63 N64 P65 K66 I71 I73 R76 T3 K4 K56 R59 R62 N63 P64 K65 I70 I72 R75 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 30 ~ 49 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1owf B 1.95 BS01 dna C 0 S4 R42 R46 S50 R59 R62 N63 P64 L72 K75 K81 G83 K84 S4 R42 R46 S50 R59 R62 N63 P64 L72 K75 K81 G83 K84 ? 0003677,0005694,0005737,0005829,0006310,0006351,0006355,0006417,0030527,0043565,1990177 remove_due_to_license_issue P0A6Y1 12842466 50 ~ 16 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIAIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIYG 1owf B 1.95 BS02 dna E 0 A44 I45 R46 H54 R56 H79 A44 I45 R46 H54 R56 H79 ? 0003677,0005694,0005737,0005829,0006310,0006351,0006355,0006417,0030527,0043565,1990177 remove_due_to_license_issue P0A6Y1 12842466 30 ~ 49 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIAIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIYG 1owg A 2.1 BS01 dna C 0 K45 R55 K57 P61 R63 P65 K66 R82 K88 K44 R54 K56 P60 R62 P64 K65 R81 K87 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 50 ~ 16 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1owg A 2.1 BS02 dna D 0 G48 N51 K86 G47 N50 K85 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 15 ~ 29 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1owg A 2.1 BS03 dna E 0 T4 K5 K57 R60 R63 N64 P65 K66 I73 R76 T3 K4 K56 R59 R62 N63 P64 K65 I72 R75 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 12842466 30 ~ 49 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 1owg B 2.1 BS01 dna C 0 S4 K27 E44 R46 G47 S50 R59 R62 N63 P64 K75 G83 K84 S4 K27 E44 R46 G47 S50 R59 R62 N63 P64 K75 G83 K84 ? 0003677,0005694,0005737,0005829,0006310,0006351,0006355,0006417,0030527,0043565,1990177 remove_due_to_license_issue P0A6Y1 12842466 50 ~ 16 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIEIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIYG 1owg B 2.1 BS02 dna E 0 E44 R46 H54 R56 H79 E44 R46 H54 R56 H79 ? 0003677,0005694,0005737,0005829,0006310,0006351,0006355,0006417,0030527,0043565,1990177 remove_due_to_license_issue P0A6Y1 12842466 30 ~ 49 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIEIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIYG 1owh A 1.61 BS01 239 A 1 H54 H106 D205 S206 Q208 W231 G234 H46 H94 D192 S193 Q195 W218 G221 H54 D109 Q208 G209 D210 S211 G212 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=40nM remove_due_to_license_issue Ki=40nM, IC50=1200nM P00749 14711304 1001 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1owi A 2.93 BS01 426 A 1 H45 Y86 A88 H93 D191 S192 Q194 G220 H46 Y87 A89 H94 D192 S193 Q195 G221 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue Ki=25nM P00749 14711304 245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1owj A 3.1 BS01 155 A 1 H45 H93 D191 S192 Q194 V215 G218 G220 H46 H94 D192 S193 Q195 V216 G219 G221 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue Ki=48nM P00749 14711304 245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1owk A 2.8 BS01 303 A 1 H45 D49 D191 S192 Q194 S216 W217 G220 H46 D50 D192 S193 Q195 S217 W218 G221 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue Ki=23.5nM P00749 14711304 245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1owr M 3.0 BS01 dna A 0 R421 G428 S429 R430 I479 R537 Q571 R665 R27 G34 S35 R36 I85 R143 Q177 R271 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 4001 ~ 4015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr M 3.0 BS02 dna B 0 Y424 T426 E427 K520 R522 N523 R537 K538 T616 H672 Y30 T32 E33 K126 R128 N129 R143 K144 T222 H278 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 5001 ~ 5015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr N 3.0 BS01 dna C 0 R421 G428 S429 R430 R537 H575 R665 R27 G34 S35 R36 R143 H181 R271 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 4001 ~ 4015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr N 3.0 BS02 dna D 0 Y424 T426 K520 R522 N523 R537 K538 Y30 T32 K126 R128 N129 R143 K144 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 5001 ~ 5015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr P 3.0 BS01 dna E 0 R421 S429 R430 R537 R27 S35 R36 R143 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 4001 ~ 4015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr P 3.0 BS02 dna F 0 Y424 T426 K520 R522 N523 R537 R572 R665 Y30 T32 K126 R128 N129 R143 R178 R271 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 5001 ~ 5015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr Q 3.0 BS01 dna G 0 R421 G428 S429 R430 G431 I479 R537 Q571 R27 G34 S35 R36 G37 I85 R143 Q177 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 4001 ~ 4015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1owr Q 3.0 BS02 dna H 0 Y424 T426 K520 R522 N523 R537 K538 R572 Y30 T32 K126 R128 N129 R143 K144 R178 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 14643663 5001 ~ 5015 VPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1oxr A 1.93 BS01 AIN A 1 L2 G30 Y64 L2 G29 Y63 Y28 G30 G32 H48 D49 Y52 Y68 D94 Y27 G29 G31 H47 D48 Y51 Y67 D93 3.1.1.4 0004623,0005102,0005509,0005543,0005576,0006633,0006644,0016042,0016787,0046872,0047498,0047499,0048146,0050482 Kd=0.000000064M remove_due_to_license_issue P60045 15823962 141 NLYQFKNMIQCTVPSRSWQDFADYGCYCGKGGSGTPVDDLDRCCQVHDNCYNEAENISGCRPYFKTYSYECTQGTLTCKGDNNACAASVCDCDRLAAICFAGAPYNDANYNIDLKARCN 1oyn A 2.0 BS02 ROL A 1 Y159 N321 I336 F340 M357 Q369 F372 Y81 N243 I258 F262 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=0.55uM remove_due_to_license_issue Q08499 12842049 503 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 1oyq A 1.9 BS02 T87 A 1 H57 Q175 D189 S190 W215 G216 G219 H40 Q155 D171 S172 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=110nM remove_due_to_license_issue Ki=110nM P00760 11342132 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1oyt H 1.67 BS04 FSN H 1 H57 N98 D189 A190 S214 W215 G216 G219 H43 N95 D192 A193 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.057uM remove_due_to_license_issue P00734 12800172 501 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1oz0 A 2.5 BS02 MS1 A 1 Q450 R452 I453 A541 F542 F545 D547 S566 A567 R589 F591 Q447 R449 I450 A538 F539 F542 D544 S563 A564 R586 F588 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Kd=20nM remove_due_to_license_issue P31335 12974624 1002 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1oz0 A 2.5 BS03 MS1 B 1 R208 Y209 I239 K267 M313 F316 G317 D340 R205 Y206 I236 K264 M310 F313 G314 D337 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Kd=20nM remove_due_to_license_issue P31335 12974624 1001 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1oz0 B 2.5 BS01 MS1 A 1 Y209 I239 K267 M313 F316 G317 D340 Y206 I236 K264 M310 F313 G314 D337 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Kd=20nM remove_due_to_license_issue P31335 12974624 1002 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1oz0 B 2.5 BS03 MS1 B 1 Q450 S451 R452 I453 A541 F542 P544 F545 S566 A567 R589 F591 Q447 S448 R449 I450 A538 F539 P541 F542 S563 A564 R586 F588 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Kd=20nM remove_due_to_license_issue P31335 12974624 1001 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1ozv A 2.65 BS01 LYS A 1 R222 F224 R226 Y254 Y287 R173 F175 R177 Y205 Y229 Y287 Y229 2.1.1.127,2.1.1.259 0009507,0016279,0018022,0030785 remove_due_to_license_issue Q43088 12819771 700 LSPAVQTFWKWLQEEGVITAKTPVKASVVTEGLGLVALKDISRNDVILQVPKRLWINPDAVAASEIGRVCSELKPWLSVILFLIRERSREDSVWKHYFGILPQETDSTIYWSEEELQELQGSQLLKTTVSVKEYVKNECLKLEQEIILPNKRLFPDPVTLDDFFWAFGILRSRAFSRLRNENLVVVPMADLINHSAGVTTEDHAYEVKYLFSLKSPLSVKAGEQVYIQYDLNKSNAELALDYGFIEPNENRHAYTLTLEISESDPFFDDKLDVAESNGFAQTAYFDIFYNRTLPPGLLPYLRLVALGGTDAFLLESLFRDTIWGHLELSVSRDNEELLCKAVREACKSALAGYHTTIEQDRELKEGNLDSRLAIAVGIREGEKMVLQQIDGIFEQKELELDQLEYYQERRLKDLGLCGENGDILENLYF 1p01 A 2.0 BS01 0EG A 1 H57 Y171 G192A R192B G193 S195 S214 G215 G216 H36 Y123 G139 R140 G141 S143 S159 G160 G161 H57 D102 G193 S195 S214 H36 D63 G141 S143 S159 3.4.21.12 0004252,0006508 remove_due_to_license_issue P00778 3122831 4 ANIVGGIEYSINNASLCSVGFSVTRGATKGFVTAGHCGTVNATARIGGAVVGTFAARVFPGNDRAWVSLTSAQTLLPRVANGSSFVTVRGSTEAAVGAAVCRSGRTTGYQCGTITAKNVTANYAEGAVRGLTQGNACMGRGDSGGSWITSAGQAQGVMSGGNVQSNGNNCGIPASQRSSLFERLQPILSQYGLSLVTG 1p17 A 2.7 BS01 IMP A 1 E111 D112 I113 V114 D115 T116 A117 T119 F164 E107 D108 I109 V110 D111 T112 A113 T115 F160 E111 D112 D115 F164 R177 E107 D108 D111 F160 R173 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0046100,0046872,0052657 remove_due_to_license_issue Q4DRC4 14698288 3000 PREYEFAEKILFTEEEIRTRIKEVAKRIADDYKGKGLRPYVNPLVLISVLRGSFMFTADLCRALCDFNVPVRMEFICVSSYGTSSGQVRMLLDTRHSIEGHHVLIVEDIVDTALTLNYLYHMYFTRRPASLKTVVLLDKREGRRVPFSADYVVANIPNAFVIGYGLDYDDTYRELRDIVVLRPEVYAEREAARQ 1p19 A 2.3 BS01 IMP A 1 D112 I113 D115 T116 A117 K143 F164 V165 D109 I110 D112 T113 A114 K140 F161 V162 E111 D112 D115 F164 R177 E108 D109 D112 F161 R174 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0046100,0046872,0052657 Kd=76.8uM remove_due_to_license_issue Q4DRC4 14698288 1300 PREYEFAEKILFTEEEIRTRIKEVAKRIADDYKGKGLRPYVNPLVLISVLKGSFMFTADLCRALCDFNVPVRMEFICVSSYGLTSSGQVRMLLDTRHSIEGHHVLIVEDIVDTALTLNYLYHMYFTRRPASLKTVVLLDKREGRRVPFSADYVVANIPNAFVIGYGLDYDDTYRELRDIVVLRPEVY 1p1n A 1.6 BS01 KAI A 1 Y61 P89 T91 R96 G141 S142 T143 E193 Y58 P86 T88 R93 G138 S139 T140 E190 ? 0015276,0016020 Kd=0.16uM remove_due_to_license_issue EC50=380000nM, Ki=3690nM P19491 12730367 999 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTTDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1p1o A 1.6 BS01 QUS A 1 Y61 L90 T91 R96 G141 S142 T143 L192 E193 Y59 L88 T89 R94 G139 S140 T141 L190 E191 ? 0015276,0016020 Kd=1.74uM remove_due_to_license_issue P19491 12730367 301 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTTDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1p2a A 2.5 BS01 5BN A 1 I10 A31 F80 F82 L83 H84 N132 L134 D145 I10 A28 F67 F69 L70 H71 N119 L121 D132 D127 K129 Q131 N132 D145 T165 D114 K116 Q118 N119 D132 T138 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=12nM remove_due_to_license_issue IC50=12nM P24941 12852944 301 MENFQKVEKIGEGVVYKARNKLTGEVVALKKIRLAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1p47 A 2.2 BS01 dna C 0 R103 R114 F116 R118 E121 R124 H125 R142 F144 S145 R146 H149 H153 T156 R170 F172 R174 E177 R180 H181 I184 R2 R13 F15 R17 E20 R23 H24 R41 F43 S44 R45 H48 H52 T55 R69 F71 R73 E76 R79 H80 I83 ? remove_due_to_license_issue P08046 12818197 1 ~ 22 ERPYACPVESCDRRFSRSDELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLRQ 1p47 A 2.2 BS02 dna D 0 D120 D148 S175 D176 K179 D19 D47 S74 D75 K78 ? remove_due_to_license_issue P08046 12818197 42 ~ 63 ERPYACPVESCDRRFSRSDELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLRQ 1p47 B 2.2 BS01 dna C 0 F116 R118 R124 H125 R142 R146 H149 H153 T156 R170 R174 E177 R180 H181 I184 F14 R16 R22 H23 R40 R44 H47 H51 T54 R68 R72 E75 R78 H79 I82 ? remove_due_to_license_issue P08046 12818197 1 ~ 22 RPYACPVESCDRRFSRSDELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHL 1p47 B 2.2 BS02 dna D 0 D148 S175 K179 D46 S73 K77 ? remove_due_to_license_issue P08046 12818197 42 ~ 63 RPYACPVESCDRRFSRSDELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHL 1p4r A 2.55 BS02 354 A 1 Q449 S450 R451 I452 P543 F544 D546 N547 S565 A566 Q446 S447 R448 I449 P540 F541 D543 N544 S562 A563 K266 H267 N431 H592 K263 H264 N428 H589 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue P31939 14966129 1801 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1p4r A 2.55 BS05 354 B 1 K266 M312 F315 N489 K263 M309 F312 N486 K266 H267 N431 H592 K263 H264 N428 H589 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue P31939 14966129 1802 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1p4r B 2.55 BS02 354 A 1 K266 M312 F315 G316 N489 K262 M308 F311 G312 N485 K266 H267 N431 H592 K262 H263 N427 H588 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue P31939 14966129 1801 QLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1p4r B 2.55 BS04 354 B 1 Q449 S450 R451 I452 P543 F544 D546 N547 S565 A566 Q445 S446 R447 I448 P539 F540 D542 N543 S561 A562 K266 H267 N431 H592 K262 H263 N427 H588 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue P31939 14966129 1802 QLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1p51 A 2.5 BS01 dna E 0 R55 R58 R61 P63 R55 R58 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 A 2.5 BS02 dna F 0 R58 G60 R61 N62 M69 I71 R58 G60 R61 N62 M69 I71 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 B 2.5 BS01 dna E 0 R58 R61 N62 P63 K64 M69 I71 R58 R61 N62 P63 K64 M69 I71 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 B 2.5 BS02 dna F 0 R53 R55 K56 R58 R61 P63 R53 R55 K56 R58 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 B 2.5 BS03 dna H 0 K41 T43 S49 K83 K41 T43 S49 K83 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 C 2.5 BS01 dna I 0 R53 R55 K56 R58 R61 P63 R53 R55 K56 R58 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 C 2.5 BS02 dna H 0 R58 R61 N62 P63 K64 M69 I71 R58 R61 N62 P63 K64 M69 I71 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 D 2.5 BS01 dna F 0 K41 T43 K83 K41 T43 K83 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 D 2.5 BS02 dna I 0 R58 N62 P63 M69 I71 R58 N62 P63 M69 I71 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p51 D 2.5 BS03 dna H 0 R53 R55 K56 R58 R61 P63 R53 R55 K56 R58 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 2 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p57 B 1.75 BS01 CR4 B 1 H57 D189 A190 C191 Q192 S195 V213 H41 D178 A179 C180 Q181 S184 V206 H57 D102 Q192 G193 D194 S195 G196 H41 D88 Q181 G182 D183 S184 G185 3.4.21.106 0004252,0006508 Ki=40uM remove_due_to_license_issue P05981 12962630 346 IVGGRDTSLGRWPWQVSLRYDGAHLCGGSLLSGDWVLTAAHCFPERNRVLSRWRVFAGAVAQASPHGLQLGVQAVVYHGGYLPFNSNDIALVHLSSPLPLTEYIQPVCLPAAGQALVDGKICTVTGWGNTQYYGQQAGVLQEARVPIISNDVCNGADFYGNQIKPKMFCAGYPEGGIDACQGDSGGPFVCEDSISRTPRWRLCGIVSWGTGCALAQKPGVYTKVSDFREWIFQAIKTHSEASGMVTQ 1p5e A 2.22 BS01 TBS A 1 I10 A31 V64 F80 L83 L134 I11 A32 V65 F81 L84 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 12869192 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 1p6d A 2.0 BS04 3PC A 1 W1 E4 N55 F66 H118 D122 H128 T133 N134 E146 W1 E4 N55 F66 H118 D122 H128 T133 N134 E146 H14 N55 H69 H118 D122 H128 H142 E146 H14 N55 H69 H118 D122 H128 H142 E146 3.1.4.3 0004629,0008270,0016787,0016788,0031640,0034480,0046872 Ki=1.15mM remove_due_to_license_issue P09598 12921783 601 WSAEDKHKEGVNSHLWIVNRAIDIMSRNTTLVKQDRVAQLNEWRTELENGIYAANYENPYYDNSTFASHFYDPDNGKTYIPFAKQAKETGAKYFKLAGESYKNKDMKQAFFYLGLSLHYLGDVNQPMHAANFTNLSYPQGFHSKYENFVDTIKDNYKVTDGNGYWNWKGTNPEEWIHGAAVVAKQDYSGIVNDNTKDWFVKAAVSQEYADKWRAEVTPMTGKRLMDAQRVTAGYIQLWFDTYGDR 1p6e A 2.3 BS04 PC5 A 1 W1 E4 N55 F66 H118 D122 H128 T133 N134 S143 E146 W1 E4 N55 F66 H118 D122 H128 T133 N134 S143 E146 H14 N55 H69 H118 D122 H128 H142 E146 H14 N55 H69 H118 D122 H128 H142 E146 3.1.4.3 0004629,0008270,0016787,0016788,0031640,0034480,0046872 Ki=1.21mM remove_due_to_license_issue P09598 12921783 601 WSAEDKHKEGVNSHLWIVNRAIDIMSRNTTLVKQDRVAQLNEWRTELENGIYAANYENPYYDNSTFASHFYDPDNGKTYIPFAKQAKETGAKYFKLAGESYKNKDMKQAFFYLGLSLHYLGDVNQPMHAANFTNLSYPQGFHSKYENFVDTIKDNYKVTDGNGYWNWKGTNPEEWIHGAAVVAKQDYSGIVNDNTKDWFVKAAVSQEYADKWRAEVTPMTGKRLMDAQRVTAGYIQLWFDTYGDR 1p71 A 1.9 BS01 dna C 0 R55 K56 R58 R61 P63 R55 K56 R58 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPPKA 1p71 A 1.9 BS02 dna D 0 R58 G60 R61 N62 P63 K64 M69 R58 G60 R61 N62 P63 K64 M69 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPPKA 1p71 B 1.9 BS01 dna C 0 R58 G60 R61 N62 P63 K64 M69 I71 R58 G60 R61 N62 P63 K64 M69 I71 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPPK 1p71 B 1.9 BS02 dna D 0 R55 K56 R58 E59 R61 P63 R55 K56 R58 E59 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPPK 1p78 A 2.25 BS01 dna C 0 R55 K56 R58 E59 R61 P63 K68 R55 K56 R58 E59 R61 P63 K68 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p78 A 2.25 BS02 dna D 0 R58 G60 R61 N62 P63 K64 M69 R58 G60 R61 N62 P63 K64 M69 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 21 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p78 B 2.25 BS01 dna C 0 R58 G60 R61 N62 P63 K64 M69 I71 R58 G60 R61 N62 P63 K64 M69 I71 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 20 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p78 B 2.25 BS02 dna D 0 R53 R55 E59 R61 P63 R53 R55 E59 R61 P63 ? 0003677,0005829,0030261,0030527,0043158 remove_due_to_license_issue P05514 12853489 1 ~ 21 MNKGELVDAVAEKASVTKKQADAVLTAALETIIEAVSSGDKVTLVGFGSFESRERKAREGRNPKTNEKMEIPATRVPAFSAGKLFREKVAPP 1p7h L 2.6 BS01 dna A 0 Y424 T426 E427 K520 R522 N523 R537 K538 Y32 T34 E35 K128 R130 N131 R145 K146 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h L 2.6 BS02 dna B 0 R421 R430 R537 Q571 H575 G663 K664 R665 K666 R29 R38 R145 Q179 H183 G271 K272 R273 K274 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h M 2.6 BS01 dna A 0 R421 R430 R537 Q571 R29 R38 R145 Q179 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h M 2.6 BS02 dna B 0 Y424 T426 K520 R522 N523 R537 K538 Y32 T34 K128 R130 N131 R145 K146 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h N 2.6 BS01 dna C 0 R421 R430 R537 Q571 H575 G663 K664 R665 K666 R29 R38 R145 Q179 H183 G271 K272 R273 K274 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h N 2.6 BS02 dna D 0 Y424 T426 K520 R522 N523 R537 K538 K664 R665 Y32 T34 K128 R130 N131 R145 K146 K272 R273 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h O 2.6 BS01 dna C 0 Y424 T426 E427 K520 R522 N523 R537 K538 Y32 T34 E35 K128 R130 N131 R145 K146 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7h O 2.6 BS02 dna D 0 R421 R430 R537 Q571 R29 R38 R145 Q179 ? 0003677,0003700,0006355 remove_due_to_license_issue Q13469 12949493 1 ~ 15 SSVPLEWPLSSQSGSYELRIEVQPKPHHRAHYETEGSRGAVKAPTGGHPVVQLHGYMENKPLGLQIFIGTADERILKPHAFYQVHRITGKTVTTTSYEKIVGNTKVLEIPLEPKNNMRATIDCAGILKLRNADIELRKGETDIGRKNTRVRLVFRVHIPESSGRIVSLQTASNPIECSQRSAHELPMVERQDTDSCLVYGGQQMILTGQNFTSESKVVFTEKTTDGQQIWEMEATVDKDKSQPNMLFVEIPEYRNKHIRTPVKVNFYVINGKRKRSQPQHFTYHPV 1p7m A -1.00 BS02 ADK A 1 W6 Y13 Y16 W21 E38 W46 W6 Y13 Y16 W21 E38 W46 Y16 E38 W46 Y16 E38 W46 3.2.2.20 0003824,0005515,0006281,0006284,0006307,0008725,0016787,0046872 remove_due_to_license_issue IC50=1500000nM P05100 13129925 189 MERCGWVSQDPLYIAYHDNEWGVPETDSKKLFEMICLEGQQAGLSWITVLKKRENYRACFHQFDPVKVAAMQEEDVERLVQDAGIIRHRGKIQAIIGNARAYLQMEQNGEPFADFVWSFVNHQPQMTQATTLSEIPTSTPASDALSKALKKRGFKFVGTTICYSFMQACGLVNDHVVGCCCYPGNKP 1p8k Z 2.6 BS01 dna A 0 K24 Y27 I55 R59 R61 R70 R72 K74 E148 Q171 R172 K24 Y27 I55 R59 R61 R70 R72 K74 E148 Q171 R172 3.1.-.- 0004519 remove_due_to_license_issue P03880 14633971 399 ~ 416 GSDLTYAYLVGLFEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSFILPIFEKYPMFSNKQYDYLRFRNALLSGIISLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYLLWLKQLRKISRYSEKIKIPSNY 1p8k Z 2.6 BS02 dna B 0 D16 A147 E148 C150 S152 Y154 D168 K200 K202 K227 Q230 D16 A147 E148 C150 S152 Y154 D168 K200 K202 K227 Q230 3.1.-.- 0004519 remove_due_to_license_issue P03880 14633971 417 ~ 429 GSDLTYAYLVGLFEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSFILPIFEKYPMFSNKQYDYLRFRNALLSGIISLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYLLWLKQLRKISRYSEKIKIPSNY 1p8k Z 2.6 BS03 dna C 0 D16 E35 L36 S37 M66 Y162 K190 Y192 K200 T204 S205 V206 R243 D16 E35 L36 S37 M66 Y162 K190 Y192 K200 T204 S205 V206 R243 3.1.-.- 0004519 remove_due_to_license_issue P03880 14633971 501 ~ 516 GSDLTYAYLVGLFEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSFILPIFEKYPMFSNKQYDYLRFRNALLSGIISLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYLLWLKQLRKISRYSEKIKIPSNY 1p8k Z 2.6 BS04 dna D 0 D16 G17 Y18 S20 T22 K23 E35 K94 D16 G17 Y18 S20 T22 K23 E35 K94 3.1.-.- 0004519 remove_due_to_license_issue P03880 14633971 517 ~ 531 GSDLTYAYLVGLFEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSFILPIFEKYPMFSNKQYDYLRFRNALLSGIISLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYLLWLKQLRKISRYSEKIKIPSNY 1p93 A 2.7 BS03 DEX A 1 M560 L563 N564 G567 Q570 M601 M604 R611 Q642 Y735 T739 I747 M34 L37 N38 G41 Q44 M75 M78 R85 Q116 Y206 T210 I218 ? remove_due_to_license_issue EC50=2.5nM, Ki=1.2nM, IC50=5nM, Kd=19nM P04150 12686538 1999 QLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKRSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 1pa9 A 2.0 BS01 CSN A 1 F67 I70 D194 Q195 C241 R242 A243 V245 G246 R247 Q284 F44 I47 D171 Q172 C214 R215 A216 V218 G219 R220 Q257 E128 W192 D194 H240 C241 R247 T248 E105 W169 D171 H213 C214 R220 T221 3.1.3.48 0004725,0006470,0016311 Ki=25uM remove_due_to_license_issue P15273 12810712 737 VSPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCRRQTAVRADLNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGLGDGIMADMYTLTIREAGQKTISVPVVHVGNWPDQTAVSSEVTKALASLVDQTAETKRNMYESKGSDDSKLRPVIHCRAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS 1pb8 A 1.45 BS01 DSN A 1 F92 T126 R131 S179 S180 W223 D224 F82 T116 R121 S169 S170 W213 D214 ? 0015276,0016020 Ki=7.02uM remove_due_to_license_issue IC50=670.0nM P35439 12805203 901 TRLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPNRHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINTERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQECDS 1pb9 A 1.6 BS01 4AX A 1 F92 T126 R131 S179 S180 W223 D224 F81 T115 R120 S168 S169 W212 D213 ? 0015276,0016020 Ki=241uM remove_due_to_license_issue P35439 12805203 901 TRLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPNHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINTERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQECDS 1pbk A 2.5 BS01 RAP A 1 Y135 D146 L162 G169 K170 V171 W175 Y198 I208 Y27 D38 L54 G61 K62 V63 W67 Y90 I100 Y135 F145 D146 I172 Y198 F216 Y27 F37 D38 I64 Y90 F108 5.2.1.8 0003755 Ki=0.9nM remove_due_to_license_issue Q00688 225 PKYTKSVLKKGDKTNFPKKGDVVHCWYTGTLQDGTVFDTNIQTSAKKKKNAKPLSFKVGVGKVIRGWDEALLTMSKGEKARLEIEPEWAYGKKGQPDAKIPPNAKLTFEVELVDID 1pbq A 1.9 BS01 DK1 A 1 Q13 F16 F92 P124 L125 T126 R131 W223 D224 F250 Q9 F12 F76 P108 L109 T110 R115 W207 D208 F234 ? 0015276,0016020 Ki=0.54uM remove_due_to_license_issue Ki=40nM, EC50=330nM, IC50=860nM P35439 12805203 1001 RLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQEC 1pdz A 2.2 BS01 PGA A 1 S36 K344 R373 S374 S36 K344 R373 S374 S39 H157 E166 E209 D244 E294 D319 K344 H372 K395 S39 H157 E166 E209 D244 E294 D319 K344 H372 K395 4.2.1.11 0000015,0000287,0004634,0005737,0006096,0016829,0046872 Ki=0.2mM remove_due_to_license_issue P56252 7547999 439 SITKVFARTIFDSRGNPTVEVDLYTSKGLFRAAVPSGASTGVHEALEMRDGDKSKYHGKSVFNAVKNVNDVIVPEIIKSGLKVTQQKECDEFMCKLDGTENKSSLGANAILGVSLAICKAGAAELGIPLYRHIANLANYDEVILPVPAFNVINGGSHAGNKLAMQEFMILPTGATSFTEAMRMGTEVYHHLKAVIKARFGLDATAVGDEGGFAPNILNNKDALDLIQEAIKKAGYTGKIEIGMDVAASEFYKQNNIYDLDFKTANNDGSQKISGDQLRDMYMEFCKDFPIVSIEDPFDQDDWETWSKMTSGTTIQIVGDDLTVTNPKRITTAVEKKACKCLLLKVNQIGSVTESIDAHLLAKKNGWGTMVSHRSGETEDCFIADLVVGLCTGQIKTGAPCRSERLAKYNQILRIEEELGSGAKFAGKNFRAPS 1pf7 E 2.6 BS01 IMH E 1 Y88 A116 E201 M219 T242 N243 H257 Y87 A115 E200 M218 T241 N242 H256 S33 H64 H86 Y88 E89 A116 M219 S220 N243 H257 S32 H63 H85 Y87 E88 A115 M218 S219 N242 H256 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 13679061 290 ENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS 1pf8 A 2.51 BS01 SU9 A 1 I10 A31 F80 F82 L83 H84 Q85 L134 D145 I10 A31 F80 F82 L83 H84 Q85 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=22nM P24941 14550307 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pfu A 1.91 BS02 MPJ A 1 A12 L13 D52 W253 P257 Y260 A9 L10 D49 W250 P254 Y257 L13 H21 H24 D52 D129 K132 S175 S178 K332 K335 L10 H18 H21 D49 D126 K129 S172 S175 K329 K332 6.1.1.10 0000166,0004812,0004825,0005524,0006418,0006431 Kd=1900uM remove_due_to_license_issue P00959 12946347 553 AKKILVTCALPYANGSIHLGHMLEHIQADVWVRYQRMRGHEVNFICADDAHGTPIMLKAQQLGITPEQMIGEMSQEHQTDFAGFNISYDNYHSTHSEENRQLSELIYSRLKENGFIKNRTISQLYDPEKGMFLPDRFVKGTCPKCKSPDQYGDNCEVCGATYSPTELIEPKSVVSGATPVMRDSEHFFFDLPSFSEMLQAWTRSGALQEQVANKMQEWFESGLQQWDISRDAPYFGFEIPNAPGKYFYVWLDAPIGYMGSFKNLCDKRGDSVSFDEYWKKDSTAELYHFIGKDIVYFHSLFWPAMLEGSNFRKPSNLFVHGYVTVNGAKMSKSRGTFIKASTWLNHFDADSLRYYYTAKLSSRIDDIDLNLEDFVQRVNADIVNKVVNLASRNAGFINKRFDGVLASELADPQLYKTFTDAAEVIGEAWESREFGKAVREIMALADLANRYVDEQAPWVVAKQEGRDADLQAICSMGINLFRVLMTYLKPVLPKLTERAEAFLNTELTWDGIQQPLLGHKVNPFKALYNRIDMRQVEALVEASKEEV 1pfy A 1.93 BS02 MSP A 1 A12 L13 Y15 G23 H24 E27 D52 W253 A256 P257 Y260 G294 D296 I297 H301 Y325 V326 A9 L10 Y12 G20 H21 E24 D49 W250 A253 P254 Y257 G291 D293 I294 H298 Y322 V323 L13 H21 H24 D52 D129 K132 S175 S178 K332 K335 L10 H18 H21 D49 D126 K129 S172 S175 K329 K332 6.1.1.10 0000166,0004812,0004825,0005524,0006418,0006431 ic50~7nM remove_due_to_license_issue P00959 12946347 553 AKKILVTCALPYANGSIHLGHMLEHIQADVWVRYQRMRGHEVNFICADDAHGTPIMLKAQQLGITPEQMIGEMSQEHQTDFAGFNISYDNYHSTHSEENRQLSELIYSRLKENGFIKNRTISQLYDPEKGMFLPDRFVKGTCPKCKSPDQYGDNCEVCGATYSPTELIEPKSVVSGATPVMRDSEHFFFDLPSFSEMLQAWTRSGALQEQVANKMQEWFESGLQQWDISRDAPYFGFEIPNAPGKYFYVWLDAPIGYMGSFKNLCDKRGDSVSFDEYWKKDSTAELYHFIGKDIVYFHSLFWPAMLEGSNFRKPSNLFVHGYVTVNGAKMSKSRGTFIKASTWLNHFDADSLRYYYTAKLSSRIDDIDLNLEDFVQRVNADIVNKVVNLASRNAGFINKRFDGVLASELADPQLYKTFTDAAEVIGEAWESREFGKAVREIMALADLANRYVDEQAPWVVAKQEGRDADLQAICSMGINLFRVLMTYLKPVLPKLTERAEAFLNTELTWDGIQQPLLGHKVNPFKALYNRIDMRQVEALVEASKEEV 1pg2 A 1.75 BS02 MET A 1 A12 L13 Y15 D52 W253 A256 P257 Y260 A9 L10 Y12 D49 W191 A194 P195 Y198 L13 H21 H24 D52 K332 K335 L10 H18 H21 D49 K270 K273 6.1.1.10 0000166,0004812,0004825,0005524,0006418,0006431 remove_due_to_license_issue P00959 12946347 553 AKKILVTCALPYANGSIHLGHMLEHIQADVWVRYQRMRGHEVNFICADDAHGTPIMLKAQQLGITPEQMIGEMSQEHQTDFAGFNISYDNYHSTHSEENRQLSELIYSRLKENGFIKNRTISRDSEHFFFDLPSFSEMLQAWTRSGALQEQVANKMQEWFESGLQQWDISRDAPYFGFEIPNAPGKYFYVWLDAPIGYMGSFKNLCDKRGDSVSFDEYWKKDSTAELYHFIGKDIVYFHSLFWPAMLEGSNFRKPSNLFVHGYVTVNGAKMSKSRGTFIKASTWLNHFDADSLRYYYTAKLSSRIDDIDLNLEDFVQRVNADIVNKVVNLASRNAGFINKRFDGVLASELADPQLYKTFTDAAEVIGEAWESREFGKAVREIMALADLANRYVDEQAPWVVAKQEGRDADLQAICSMGINLFRVLMTYLKPVLPKLTERAEAFLNTELTWDGIQQPLLGHKVNPFKALYNRIDMRQVEALVEASKEEV 1pgp A 2.5 BS01 6PG A 1 S128 K183 N187 Y191 K260 T262 S128 K183 N187 Y191 K260 T262 S128 K183 H186 N187 E190 S128 K183 H186 N187 E190 1.1.1.44 0004616,0005737,0006098,0016491,0019521,0050661 Kd=2uM remove_due_to_license_issue P00349 7922042 502 AQADIALIGLAVMGQNLILNMNDHGFVVCAFNRTVSKVDDFLANEAKGTKVLGAHSLEEMVSKLKKPRRIILLVKAGQAVDNFIEKLVPLLDIGDIIIDGGNSEYRDTMRRCRDLKDKGILFVGSGVSGGEDGARYGPSLMPGGNKEAWPHIKAIFQGIAAKVGTGEPCCDWVGDDGAGHFVKMVHNGIEYGDMQLICEAYHLMKDVLGLGHKEMAKAFEEWNKTELDSFLIEITASILKFQDADGKHLLPKIRDSAGQKGTGKWTAISALEYGVPVTLIGEAVFARCLSSLKDERIQASKKLKGPQNIPFEGDKKSFLEDIRKALYASKIISYAQGFMLLRQAATEFGWTLNYGGIALMWRGGCIIRSVFLGKIKDAFDRNPGLQNLLLDDFFKSAVENCQDSWRRAISTGVQAGIPMPCFTTALSFYDGYRHAMLPANLIQAQRDYFGAHTYELLAKPGQFIHTNWTGHGG 1ph0 A 2.2 BS01 418 A 1 Y20 R24 Y46 D48 C215 S216 A217 I219 G220 R221 R254 G259 Q262 T263 Q266 M282 G283 Y19 R23 Y45 D47 C214 S215 A216 I218 G219 R220 R253 G258 Q261 T262 Q265 M281 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=120nM P18031 12877578 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1phw A 2.36 BS01 N A 1 P1115 A1116 F1117 K1138 R1168 H1202 P115 A116 F117 K138 R168 H202 N1026 K1060 D1250 N26 K60 D238 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0032991,0042802 Ki=0.5mM remove_due_to_license_issue P0A715 16023668 70 MKQKVVSIGDINVANDLPFVLFGGMNVLESRDLAMRICEHYVTVTQKLGIPYVFKASFDKANRSSIHSYRGPGLEEGMKIFQELKQTFGVKIITDVHEPSQAQPVADVVDVIQLPAFLARQTDLVEAMAKTGAVINVKKPQFVSPGQMGNIVDKFKEGGNEKVILCDRGANFGYDNLVVDMLGFSIMKKVSGNSPVIFDVTHALQRAQVAELARAGMAVGLAGLFIEAHPDPEHAKCDGPSALPLAKLEPFLKQMKAIDDLVKGFEELDTSK 1pi4 A 1.39 BS01 SM3 A 1 S64 L119 Y150 Y221 G317 A318 T319 G320 S61 L116 Y147 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=37nM remove_due_to_license_issue P00811 14661960 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDAKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1pi5 A 1.49 BS01 SM2 A 1 S64 L119 Y150 Y221 G317 A318 T319 G320 S61 L116 Y147 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=17nM remove_due_to_license_issue P00811 14661960 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDAKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1pig A 2.2 BS01 GLC B 1 W58 W59 Q63 H305 W58 W59 Q63 H305 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 1 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS02 AGL B 1 W59 V163 W59 V163 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS03 GLC C 1 Y151 K200 E240 Y151 K200 E240 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS04 AGL C 1 A198 H201 E233 D300 A198 H201 E233 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 3 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS05 GLC D 1 K322 W388 E390 K322 W388 E390 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 1 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS06 GLC D 2 R387 W388 R389 E390 R387 W388 R389 E390 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS07 GLC E 1 E272 W284 E272 W284 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 1 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS08 BGC E 1 K261 G283 W284 K261 G283 W284 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS09 HMC A 1 W58 H101 D197 E233 H299 D300 W58 H101 D197 E233 H299 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 703 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pig A 2.2 BS10 BGC A 1 T439 Y468 S470 T474 A475 T439 Y468 S470 T474 A475 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8757803 1002 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAISSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGQPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCNVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAQDPFIAIHAESKL 1pk0 A 3.3 BS01 EMA A 1 R329 K346 L348 K353 S354 K372 A490 D493 T548 H577 G578 T579 N583 R38 K55 L57 K62 S63 K81 A199 D202 T257 H286 G287 T288 N292 4.6.1.1 0005576,0008294 remove_due_to_license_issue P40136 14978283 1999 RIDVLKGEKALKASGLVPEHADAFKKIARELNTYILFRPVNKLATNLIKSGVATKGLNVHGKSSDWGPVAGYIPFDQDLSKKHGQQLAVEKGNLENKKSITEHEGEIGKIPLKLDHLRIEELKENGIILKGKKEIDNGKKYYLLESNNQVYEFRISDENNEVQYKTKEGKITVLGEKFNWRNIEVMAKNVEGVLKPLTADYDLFALAPSLTEIKKQIPQKEWDKVVNTPNSLEKQKGVTNLLIKYGIERKPDSTKGTLSNWQKQMLDRLNEAVKYTGYTGGDVVNHGTEQDNEEFPEKDNEIFIINPEGEFILTKNWEMTGRFIEKNITGKDYLYYFNRSYNKIAPGNKAYIEWTDPITKAKINTIPTSAEFIKNLSSIRRSSVKKIAGYLSDYYNSANHIFSQEKKRKISIFRGIQAYNEIENVLKSKQIAPEYKNYFQYLKERITNQVQLLLTHQKFKLLYKQLNFTENETDNFEVFQKIID 1pkx A 1.9 BS01 XMP A 1 S10 V11 S12 S34 G36 T37 R64 K66 T67 N102 L103 Y104 D125 I126 G127 G128 S8 V9 S10 S32 G34 T35 R62 K64 T65 N100 L101 Y102 D123 I124 G125 G126 K266 H267 N431 H592 K264 H265 N429 H588 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 Ki=0.12uM remove_due_to_license_issue P31939 14756553 1901 PGQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1pl0 A 2.6 BS03 BW2 B 1 K266 M312 F315 K263 M309 F312 K266 H267 N431 H592 K263 H264 N428 H589 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue Ki=6.0nM, IC50=1000nM P31939 14966129 802 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1pl0 B 2.6 BS02 BW2 B 1 S450 R451 I452 F541 P543 F544 N547 S447 R448 I449 F536 P538 F539 N542 K266 H267 N431 H592 K263 H264 N428 H587 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue Ki=6.0nM, IC50=1000nM P31939 14966129 802 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 1pme A 2.0 BS01 SB2 A 1 A52 L103 V104 T105 H106 L107 M108 K151 S153 N154 L156 A34 L85 V86 T87 H88 L89 M90 K133 S135 N136 L138 D149 K151 S153 N154 D167 T190 D131 K133 S135 N136 D149 T172 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Ki=0.76nM remove_due_to_license_issue P28482 9827991 1001 GQVFDVGPRYTNLSYIGYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYLVTHLMGADLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFLPKEKLKELIFEETARFQPGYRS 1pmn A 2.2 BS01 984 A 1 V78 A91 I92 K93 I124 L144 M146 M149 D150 A151 S193 N194 V34 A47 I48 K49 I80 L100 M102 M105 D106 A107 S149 N150 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 ic50=7.1nM remove_due_to_license_issue IC50=1.6nM P53779 12954329 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPQLDEREHTIEEWKELIYKEVMN 1pmu A 2.7 BS01 9HP A 1 I70 Q75 V78 A91 M146 L148 M149 Q155 L206 I26 Q31 V34 A47 M102 L104 M105 Q111 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T174 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=590nM P53779 12954329 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQDEREHTIEEWKELIYKEVMN 1pmv A 2.5 BS01 537 A 1 I70 A91 M146 L148 M149 D150 A151 V196 L206 I26 A47 M102 L104 M105 D106 A107 V152 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 ic50=150nM remove_due_to_license_issue IC50=190nM, Kd=22nM P53779 12954329 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQQLDEREHTIEEWKELIYKEVMN 1po6 A 2.1 BS01 dna B 0 K15 F17 G19 G20 D42 M46 R55 F57 F59 E85 A89 V90 R92 S95 H101 K8 F10 G12 G13 D35 M39 R48 F50 F52 E78 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 12904298 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1pot A 1.8 BS01 SPD A 1 W34 E36 Y37 S83 D168 E171 W255 D257 Y293 Q327 W9 E11 Y12 S58 D143 E146 W230 D232 Y268 Q302 ? 0015846,0015847,0015848,0016020,0019808,0019809,0019810,0030288,0042597,1903711 Kd=3.2uM remove_due_to_license_issue P0AFK9 8897598 350 NNTLYFYNWTEYVPPGLLEQFTKETGIKVIYSTYESNETMYAKLKTYKDGAYDLVVPSTYYVDKMRKEGMIQKIDKSKLTNFSNLDPDMLNKPFDPNNDYSIPYIWGATAIGVNGDAVDPKSVTSWADLWKPEYKGSLLLTDDAREVFQMALRKLGYSGNTTDPKEIEAAYNELKKLMPNVAAFNSDNPANPYMEGEVNLGMIWNGSAFVARQAGTPIDVVWPKEGGIFWMDSLAIPANAKNKEGALKLINFLLRPDVAKQVAETIGYPTPNLAARKLLSPEVANDKTLYPDAETIKNGEWQNDVGAASSIYEEYYQKLKAG 1pp8 F 3.05 BS01 dna K 0 S26 R28 R33 F34 I78 K79 T82 S25 R27 R32 F33 I77 K78 T81 ? remove_due_to_license_issue Q95VR4 14622596 26 ~ 37 DSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTRNS 1pp8 F 3.05 BS02 dna J 0 R24 K25 K69 R88 Q94 D98 R23 K24 K68 R87 Q93 D97 ? remove_due_to_license_issue Q95VR4 14622596 3 ~ 14 DSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTRNS 1pp8 M 3.05 BS01 dna Y 0 S26 R33 F34 I78 K79 N81 T82 N86 S26 R33 F34 I78 K79 N81 T82 N86 ? remove_due_to_license_issue Q95VR4 14622596 26 ~ 37 MDSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTRNSVFED 1pp8 M 3.05 BS02 dna R 0 K25 K69 K25 K69 ? remove_due_to_license_issue Q95VR4 14622596 3 ~ 14 MDSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTRNSVFED 1pp8 P 3.05 BS01 dna I 0 S26 R33 I78 K79 N81 T82 N86 S26 R33 I78 K79 N81 T82 N86 ? remove_due_to_license_issue Q95VR4 14622596 26 ~ 37 MDSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTRNSVFED 1pp8 P 3.05 BS02 dna T 0 K25 R28 K69 R88 Q94 D98 K25 R28 K69 R88 Q94 D98 ? remove_due_to_license_issue Q95VR4 14622596 3 ~ 14 MDSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTRNSVFED 1pp8 U 3.05 BS01 dna E 0 R33 I78 K79 N81 T82 N86 R32 I77 K78 N80 T81 N85 ? remove_due_to_license_issue Q95VR4 14622596 26 ~ 37 DSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTR 1pp8 U 3.05 BS02 dna G 0 R24 K25 S27 K69 R88 Q94 H97 D98 R23 K24 S26 K68 R87 Q93 H96 D97 ? remove_due_to_license_issue Q95VR4 14622596 3 ~ 14 DSNDLEASFTSRLPPEIVAALKRKSSRDPNSRFPRKLHMLLTYLASNPQLEEEIGLSWISDTEFKMKKKNVALVMGIKLNTLNVNLRDLAFEQLQHDKGGWTQWKRSGFTR 1ppc E 1.8 BS01 MID E 1 H57 N97 L99 D189 S190 S195 W215 G216 G219 H40 N79 L81 D171 S172 S177 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.69uM remove_due_to_license_issue Ki=325nM P00760 2226434 5 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1pph E 1.9 BS02 0ZG E 1 D189 S190 C191 V213 W215 G216 G219 D171 S172 C173 V191 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.2uM remove_due_to_license_issue Ki=99999999999999nM P00760 1879520 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1ppi A 2.2 BS01 GLC B 1 W58 W59 Q63 H305 W58 W59 Q63 H305 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8193143 1 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAIKSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGEPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCDVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAEDPFIAIHAESKL 1ppi A 2.2 BS02 GLC B 2 W59 Q63 V163 L165 W59 Q63 V163 L165 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8193143 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAIKSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGEPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCDVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAEDPFIAIHAESKL 1ppi A 2.2 BS03 BGC C 1 K200 I235 E240 G306 K200 I235 E240 G306 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8193143 1 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAIKSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGEPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCDVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAEDPFIAIHAESKL 1ppi A 2.2 BS04 DAF C 1 W58 Y62 H101 D197 A198 H201 E233 H299 D300 G306 W58 Y62 H101 D197 A198 H201 E233 H299 D300 G306 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0046872 remove_due_to_license_issue P00690 8193143 2 QYAPQTQSGRTSIVHLFEWRWVDIALECERYLGPKGFGGVQVSPPNENVVVTNPSRPWWERYQPVSYKLCTRSGNENEFRDMVTRCNNVGVRIYVDAVINHMCGSGAAAGTGTTCGSYCNPGSREFPAVPYSAWDFNDGKCKTASGGIESYNDPYQVRDCQLVGLLDLALEKDYVRSMIADYLNKLIDIGVAGFRIDASKHMWPGDIKAVLDKLHNLNTNWFPAGSRPFIFQEVIDLGGEAIKSSEYFGNGRVTEFKYGAKLGTVVRKWSGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGSSILTFWDARLYKVAVGFMLAHPYGFTRVMSSYRWARNFVNGEDVNDWIGPPNNNGVIKEVTINADTTCGNDWVCEHRWREIRNMVWFRNVVDGEPFANWWDNGSNQVAFGRGNRGFIVFNNDDWQLSSTLQTGLPGGTYCDVISGDKVGNSCTGIKVYVSSDGTAQFSISNSAEDPFIAIHAESKL 1ppk E 1.8 BS01 IVV E 1 E15 D33 G35 Y75 G76 D77 D213 G215 T216 T217 Y274 E15 D33 G35 Y75 G76 D77 D213 G215 T216 T217 Y274 3.4.23.20 0004190,0005576,0006508 Ki=22nM remove_due_to_license_issue P00798 1606144 700 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 1ppl E 1.7 BS01 1Z7 E 1 D33 Y75 G76 D77 D213 G215 T216 T217 Y274 I297 D33 Y75 G76 D77 D213 G215 T216 T217 Y274 I297 3.4.23.20 0004190,0005576,0006508 Ki=2.8nM remove_due_to_license_issue P00798 1606144 324 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 1ppm E 1.7 BS01 0P1 E 1 D33 Y75 G76 D77 D213 G215 T216 T217 A242 D33 Y75 G76 D77 D213 G215 T216 T217 A242 3.4.23.20 0004190,0005576,0006508 Ki=1600nM remove_due_to_license_issue P00798 1606144 324 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 1ppw A 2.21 BS03 EIP A 1 K21 R51 K55 C67 G68 H69 Y104 E114 E116 W161 K18 R48 K52 C64 G65 H66 Y101 E111 E113 W158 H25 H32 C67 H69 E87 Y104 E114 E116 W161 H22 H29 C64 H66 E84 Y101 E111 E113 W158 5.3.3.2 0000287,0003824,0004452,0005737,0006974,0008270,0008299,0016853,0046872,0050992 ic50~50uM remove_due_to_license_issue Q46822 15643873 301 EHVILLNAQGVPTGTLEKYAAHTADTRLHLAFSSWLFNAKGQLLVTRRALSKKAWPGVWTNSVCGHPQLGESNEDAVIRRCRYELGVEITPPESIYPDFRYRATDPSGIVENEVCPVFAARTTSALQINDDEVMDYQWCDLADVLHGIDATPWAFSPWMVMQATNREARKRLSAFT 1pq3 A 2.7 BS03 S2C A 1 H145 D147 S156 H160 D202 D251 E296 H122 D124 S133 H137 D179 D228 E273 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 remove_due_to_license_issue P78540 12859189 551 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 1pq6 A 2.4 BS01 965 A 1 F271 L274 A275 S278 M312 L313 T316 R319 F329 L330 F340 L345 F349 I350 I353 F354 H435 W457 F43 L46 A47 S50 M84 L85 T88 R91 F101 L102 F112 L117 F121 I122 I125 F126 H207 W229 ? 0003677,0004879,0006629 remove_due_to_license_issue EC50=40.0nM, IC50=23nM, Ki=2.2nM P55055 12819202 1500 LTAAQELMIQQLVAAQLQCNKRSPKVTPWPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVH 1pqc A 2.8 BS01 444 A 1 F271 A275 M312 T316 F329 L345 F349 H435 F45 A49 M86 T90 F103 L119 F123 H209 ? 0003677,0004879,0006629 remove_due_to_license_issue IC50=9nM, EC50=170nM, Ki=41nM, Kd=103nM P55055 12819202 1500 LTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWD 1pr1 A 2.3 BS02 FMB A 1 M64 R87 S90 C91 G92 F159 V178 M180 E181 D204 M64 R87 S90 C91 G92 F159 V178 M180 E181 D204 H4 G20 R24 R43 E75 R87 S90 S203 D204 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 R206 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0009116,0009164,0016757,0016763,0042278 Ki=5uM remove_due_to_license_issue P0ABP9 12937174 245 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHRQTTFNDMIKIALESVLLGDK 1pr5 A 2.5 BS02 TBN A 1 M64 R87 S90 C91 G92 F159 V178 M180 E181 D204 M64 R87 S90 C91 G92 F159 V178 M180 E181 D204 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R211 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0009116,0009164,0016757,0016763,0042278 Ki=120uM remove_due_to_license_issue P0ABP9 12937174 1245 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHITAAERQTTFNDMIKIALESVLLGDK 1pro A 1.8 BS01 A88 A 1 D25 G27 A28 D29 D30 I50 P81 V82 D25 G27 A28 D29 D30 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=5pM remove_due_to_license_issue P12499 8558507 301 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1pro B 1.8 BS01 A88 A 1 D25 A28 D29 D30 G49 I50 P81 D25 A28 D29 D30 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 8558507 301 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ps3 A 1.8 BS02 KIF A 1 H90 D92 W95 D204 Y269 D341 W415 H471 D472 Y727 R876 H60 D62 W65 D174 Y239 D311 W385 H441 D442 Y697 R846 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=5.2mM remove_due_to_license_issue Q24451 14636047 1501 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 1pu7 A 1.93 BS01 39A A 1 W24 W25 F45 K211 W23 W24 F44 K210 ? 0003824,0004519,0006281,0006284,0046872,0051539 Ki=0.8mM remove_due_to_license_issue O25323 14517230 219 LDSFEILKALKSLDLLKNAPAWWWPNALKFEALLGAVLTQNTKFEAVLKSLENLKNAFILENDDEINLKKIAYIEFSKLAECVRPSGFYNQKAKRLIDLSGNILKDFQSFENFKQEVTREWLLDQKGIGKESADAILCYACAKEVMVVDKYSYLFLKKLGIEIEDYDELQHFFEKGVQENLNSALALYENTISLAQLYARFHGKIVEFSKQKLEL 1pu8 A 2.13 BS01 EA1 A 1 W24 W25 F45 K211 W23 W24 F44 K210 ? 0003824,0004519,0006281,0006284,0046872,0051539 Ki=0.8mM remove_due_to_license_issue O25323 14517230 219 LDSFEILKALKSLDLLKNAPAWWWPNALKFEALLGAVLTQNTKFEAVLKSLENLKNAFILENDDEINLKKIAYIEFSKLAECVRPSGFYNQKAKRLIDLSGNILKDFQSFENFKQEVTREWLLDQKGIGKESADAILCYACAKEVMVVDKYSYLFLKKLGIEIEDYDELQHFFEKGVQENLNSALALYENTISLAQLYARFHGKIVEFSKQKLEL 1puf A 1.9 BS01 dna D 0 R203 K207 R209 C210 P211 Y212 R247 Q248 I251 N255 K259 R11 K15 R17 C18 P19 Y20 R55 Q56 I59 N63 K67 ? 0000981,0003677,0006355 remove_due_to_license_issue P09631 12923056 1 ~ 20 NNPAANWLHARSTRKKRCPYTKHQTLELEKEFLFNMYLTRDRRYEVARLLNLTERQVKIWFQNRRMKMKKINKDRAK 1puf A 1.9 BS02 dna E 0 L200 A202 R209 P211 Y229 R232 R235 Q254 R257 M258 K261 L8 A10 R17 P19 Y37 R40 R43 Q62 R65 M66 K69 ? 0000981,0003677,0006355 remove_due_to_license_issue P09631 12923056 21 ~ 40 NNPAANWLHARSTRKKRCPYTKHQTLELEKEFLFNMYLTRDRRYEVARLLNLTERQVKIWFQNRRMKMKKINKDRAK 1puf B 1.9 BS01 dna D 0 R237 R238 N239 F240 Q279 N282 N286 R290 R5 R6 N7 F8 Q47 N50 N54 R58 ? 0000981,0003677,0006355 remove_due_to_license_issue P40424 12923056 1 ~ 20 ARRKRRNFNKQATEILNEYFYSHLSNPYPSEEAKEELAKKCGITVSQVSNWFGNKRIRYKKNIGKFQEEANIY 1puf B 1.9 BS02 dna E 0 R237 R238 Y260 R288 K292 K293 R5 R6 Y28 R56 K60 K61 ? 0000981,0003677,0006355 remove_due_to_license_issue P40424 12923056 21 ~ 40 ARRKRRNFNKQATEILNEYFYSHLSNPYPSEEAKEELAKKCGITVSQVSNWFGNKRIRYKKNIGKFQEEANIY 1pun A -1.00 BS02 8OG A 1 I6 E41 I6 E41 3.6.1.55 0000287,0005515,0006203,0006260,0006281,0006289,0008413,0016787,0030145,0035539,0044715,0044716,0046067,0046872,0047693 remove_due_to_license_issue P08337 12939141 131 MKKLQIAVGIIRNENNEIFITRRAADAHMANKLEFPGGKIEMGETPEQAVVRELQEEVGITPQHFSLFEKLEYEFPDRHITLWFWLVERWEGEPWGKEGQPGEWMSLVGLNADDFPPANEPVIAKLKRL 1puq A -1.00 BS02 8OG A 1 L4 I6 E34 F75 R78 I80 A118 N119 L4 I6 E34 F75 R78 I80 A118 N119 3.6.1.55 0000287,0005515,0006203,0006260,0006281,0006289,0008413,0016787,0030145,0035539,0044715,0044716,0046067,0046872,0047693 remove_due_to_license_issue P08337 12939141 131 MKKLQIAVGIIRNENNEIFITRRAADAHMANKLEFPGGKIEMGETPEQAVVRELQEEVGITPQHFSLFEKLEYEFPDRHITLWFWLVERWEGEPWGKEGQPGEWMSLVGLNADDFPPANEPVIAKLKRL 1pus A -1.00 BS02 8OG A 1 L4 I6 E34 I80 L82 P116 N119 L4 I6 E34 I80 L82 P116 N119 3.6.1.55 0000287,0005515,0006203,0006260,0006281,0006289,0008413,0016787,0030145,0035539,0044715,0044716,0046067,0046872,0047693 remove_due_to_license_issue P08337 12939141 131 MKKLQIAVGIIRNENNEIFITRRAADAHMANKLEFPGGKIEMGETPEQAVVRELQEEVGITPQHFSLFEKLEYEFPDRHITLWFWLVERWEGEPWGKEGQPGEWMSLVGLNADDFPPANEPVIAKLKRL 1pvn A 2.0 BS01 MZP A 1 A57 M59 G316 S317 I318 C319 D358 L380 G381 R382 Y405 G407 E408 G409 R418 Y419 E431 G432 A56 M58 G184 S185 I186 C187 D226 L248 G249 R250 Y273 G275 E276 G277 R286 Y287 E299 G300 1.1.1.205 0003824,0003938,0006164,0016491 Ki=0.15nM remove_due_to_license_issue P50097 12549902 971 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIREKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICITREQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWQRYDLGGKQKLSFEEGVDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVEGGAHDVIVK 1pvn B 2.0 BS01 MZP B 1 A57 M59 G316 S317 I318 C319 D358 L380 G381 R382 Y405 G407 E408 G409 R418 Y419 E431 G432 A56 M58 G184 S185 I186 C187 D226 L248 G249 R250 Y273 G275 E276 G277 R286 Y287 E299 G300 1.1.1.205 0003824,0003938,0006164,0016491 Ki=0.15nM remove_due_to_license_issue P50097 12549902 972 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIREKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICITREQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWQRYDLGGKQKLSFEEGVDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVEGGAHDVIVK 1pwp A 2.9 BS02 NSC A 1 D328 F329 S655 Y659 H690 Y728 E735 D299 F300 S611 Y615 H646 Y684 E691 H686 E687 H690 Y728 E735 H642 E643 H646 Y684 E691 3.4.24.83 0003824,0004222,0005515,0005576,0006508,0008237,0008270,0030430,0035821,0044164,0046872,0090729 remove_due_to_license_issue Ki=500nM, IC50=3200nM P15917 14718925 9002 KTQEEHLKEIMKHIVKIEVKGEEAVKKEAAEKLLEKVPSDVLEMYKAIGGKIYIVDGDITKHISLEALSEDKKKIKDIYGKDALLHEHYVYAKEGYEPVLVIQSSEDYVENTEKALNVYYEIGKILSRDILSKINQPYQKFLDVLNTIKNASDSDGQDLLFTNQLKEHPTDFSVEFLEQNSNEVQEVFAKAFAYYIEPQHRDVLQLYAPEAFNYMDKFNEQEINLSLEELKDQRMLSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 1pwq A 3.52 BS02 SD2 A 1 H654 S655 L658 K673 G674 L677 H686 E687 H690 Y728 E735 E739 H610 S611 L614 K629 G630 L633 H642 E643 H646 Y684 E691 E695 H686 E687 H690 Y728 E735 H642 E643 H646 Y684 E691 3.4.24.83 0003824,0004222,0005515,0005576,0006508,0008237,0008270,0030430,0035821,0044164,0046872,0090729 remove_due_to_license_issue P15917 14718924 9002 ERNKTQEEHLKEIMKHIVKIEVKGEEAVKKEAAEKLLEKVPSDVLEMYKAIGGKIYIVDGDITKHISLEALSEDKKKIKDIYGKDALLHEHYVYAKEGYEPVLVIQSSEDYVENTEKALNVYYEIGKILSRDILSKINQPYQKFLDVLNTIKNASDSDGQDLLFTNQLKEHPTDFSVEFLEQNSNEVQEVFAKAFAYYIEPQHRDVLQLYAPEAFNYMDKFNEQEINLSLEELKDQRMLSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 1pwu A 2.7 BS02 GM6 A 1 D328 H654 S655 K656 G657 G674 V675 L677 H686 H690 Y728 D299 H625 S626 K627 G628 G645 V646 L648 H657 H661 Y699 H686 C687 H690 Y728 E735 H657 C658 H661 Y699 E706 3.4.24.83 0003824,0004222,0005515,0005576,0006508,0008237,0008270,0030430,0035821,0044164,0046872,0090729 remove_due_to_license_issue P15917 14718924 1001 KTQEEHLKEIMKHIVKIEVKGEEAVKKEAAEKLLEKVPSDVLEMYKAIGGKIYIVDGDITKHISLEALSEDKKKIKDIYGKDALLHEHYVYAKEGYEPVLVIQSSEDYVENTEKALNVYYEIGKILSRDILSKINQPYQKFLDVLNTIKNASDSDGQDLLFTNQLKEHPTDFSVEFLEQNSNEVQEVFAKAFAYYIEPQHRDVLQLYAPEAFNYMDKFNEQEINLSLEELKDQRMLSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEEEKELLNRIQVDSSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHCFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 1pwy E 2.8 BS01 AC2 E 1 A116 A117 G118 F200 E201 V217 M219 T242 N243 H257 A115 A116 G117 F199 E200 V216 M218 T241 N242 H256 S33 H64 Y88 A116 M219 S220 H257 S32 H63 Y87 A115 M218 S219 H256 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=180000nM P00491 12914786 290 ENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS 1px4 A 1.6 BS03 IPT A 1 N102 D201 E461 E537 H540 N604 W999 N90 D189 E449 E525 H528 N592 W987 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.59mM remove_due_to_license_issue Ki=7.6e+4nM P00722 14621996 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIAVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 1px4 D 1.6 BS03 IPT D 1 N102 D201 E461 E537 H540 N604 W999 N90 D189 E449 E525 H528 N592 W987 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.59mM remove_due_to_license_issue Ki=7.6e+4nM P00722 14621996 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIAVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 1pxh A 2.15 BS01 SNA A 1 Y46 R47 D48 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 R46 D47 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P18031 12547827 401 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1pxi A 1.95 BS01 CK1 A 1 G11 E12 A31 K33 N132 L134 G11 E12 A31 K33 N128 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 12679018 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxj A 2.3 BS01 CK2 A 1 I10 V18 A31 K33 F82 L83 L134 I10 V18 A31 K33 F78 L79 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue Ki=6500nM, Kd=30300nM, IC50=6.50e+3nM, kon=8.22E+04M-1-s-1, koff=1.42E+00s-1 P24941 12679018 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxk A 2.8 BS01 CK3 A 1 I10 A31 F82 L83 H84 L134 D145 I10 A31 F74 L75 H76 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 12679018 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxl A 2.5 BS01 CK4 A 1 I10 A31 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F72 E73 F74 L75 H76 Q77 D78 K81 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=2.9e+2nM, Ki=290nM P24941 12679018 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxm A 2.53 BS01 CK5 A 1 I10 A31 F80 F82 L83 H84 D86 L134 I10 A31 F72 F74 L75 H76 D78 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue Ki=60nM P24941 15027857 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxn A 2.5 BS01 CK6 A 1 I10 V18 A31 F82 L83 H84 Q85 K89 L134 D145 I10 V18 A31 F78 L79 H80 Q81 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.07uM remove_due_to_license_issue Ki=70nM P24941 15027857 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxo A 1.96 BS01 CK7 A 1 I10 A31 F80 E81 L83 D86 K89 Q131 L134 A144 D145 I10 A31 F76 E77 L79 D82 K85 Q127 L130 A140 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=2nM remove_due_to_license_issue IC50=10.0nM, Ki=2nM P24941 15027857 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pxp A 2.3 BS01 CK8 A 1 I10 A31 F82 L83 H84 K89 L134 D145 I10 A31 F78 L79 H80 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.22uM remove_due_to_license_issue IC50=2.2e+2nM, Ki=220nM P24941 15027857 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1py2 A 2.8 BS01 FRH A 1 P34 R38 M39 F42 K43 Y45 E62 P65 L72 A73 P27 R31 M32 F35 K36 Y38 E55 P58 L65 A66 ? 0002250,0002366,0002639,0002903,0005125,0005134,0005515,0005576,0005615,0006366,0006955,0007155,0007186,0007204,0007267,0008083,0008284,0010467,0019209,0030101,0030217,0030246,0030307,0030890,0031851,0032729,0032740,0034105,0038110,0042098,0042102,0042104,0043066,0043208,0045471,0045582,0045591,0045944,0046013,0046651,0048304,0050672,0050728,0050729,0050798,0060999,0097192,0097696,1900100,1901327,2000320,2000561 remove_due_to_license_issue P60568 14664558 201 STKKTQLQLEHLLLDLQMILNGINNYPKLTRMLTFKFYMPKKATELKHLQCLEEELKPLEEVLNLAFRPRDLISNINVIVLELKETTFMCEYADETATIVEFLNRWITFCQSIISTL 1py5 A 2.3 BS01 PY1 A 1 I211 A230 V231 K232 L260 L278 S280 D281 Y282 H283 L340 D351 I12 A31 V32 K33 L61 L79 S81 D82 Y83 H84 L141 D152 D333 K335 N338 D351 T375 D134 K136 N139 D152 T176 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=51nM remove_due_to_license_issue IC50=51nM, Kd=5nM P36897 15177479 700 TIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG 1pye A 2.0 BS01 PM1 A 1 I10 V18 A31 K33 F80 F82 L83 L134 A144 D145 I10 V15 A28 K30 F64 F66 L67 L118 A128 D129 D127 K129 Q131 N132 D145 T165 D111 K113 Q115 N116 D129 T133 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=386nM remove_due_to_license_issue IC50=324nM P24941 14749470 700 MENFQKVEKIGEGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTELYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1pyg A 2.87 BS01 AMP A 1 W67 Q71 Y75 R309 R310 F316 G317 W58 Q62 Y66 R274 R275 F281 G282 H377 K568 R569 K574 T676 K680 H342 K533 R534 K539 T641 K645 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1962195 843 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPQAVLDRNLAENISKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 1pyg A 2.87 BS03 AMP B 1 D42 N44 V45 D33 N35 V36 H377 K568 R569 K574 T676 K680 H342 K533 R534 K539 T641 K645 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1962195 843 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPQAVLDRNLAENISKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 1pyg B 2.87 BS01 AMP A 1 D42 N44 V45 D23 N25 V26 H377 K568 R569 K574 T676 K680 H332 K523 R524 K529 T631 K635 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1962195 843 GVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPQAVLDRNLAENISKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 1pyg B 2.87 BS02 AMP B 1 W67 Q71 Y75 R309 R310 F316 G317 W48 Q52 Y56 R264 R265 F271 G272 H377 K568 R569 K574 T676 K680 H332 K523 R524 K529 T631 K635 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1962195 843 GVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPQAVLDRNLAENISKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 1pyn A 2.2 BS01 941 A 1 Y20 R24 Y46 D48 C215 S216 A217 G220 R221 R254 G259 Q262 G283 Y19 R23 Y45 D47 C214 S215 A216 G219 R220 R253 G258 Q261 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=3.2uM remove_due_to_license_issue Ki=3200nM P18031 12951078 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1pzi D 1.99 BS01 1DM D 1 Y12 E51 Q61 W88 N90 K91 Y12 E51 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 Kd=60uM remove_due_to_license_issue P32890 14980603 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1pzi E 1.99 BS01 1DM E 1 Y12 E51 Q56 H57 Q61 W88 N90 K91 Y12 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 Kd=60uM remove_due_to_license_issue P32890 14980603 105 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1pzj D 1.46 BS01 15B D 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0046872 ic50=0.32mM remove_due_to_license_issue Q57193 14980603 104 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 1pzj D 1.46 BS02 15B H 1 G33 K34 R35 G33 K34 R35 ? 0005576,0046872 ic50=0.32mM remove_due_to_license_issue Q57193 14980603 108 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 1pzo A 1.9 BS01 CBT A 1 L220 S235 G236 R244 G245 I246 N276 I279 L195 S210 G211 R218 G219 I220 N249 I252 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 Ki=460uM remove_due_to_license_issue P62593 15037085 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1pzo A 1.9 BS02 CBT A 2 L220 L221 A224 N276 I279 A280 G283 L195 L196 A199 N249 I252 A253 G256 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 Ki=460uM remove_due_to_license_issue P62593 15037085 301 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQNDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTTPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1pzp A 1.45 BS01 FTA A 1 A224 I263 A280 G283 A284 A199 I236 A253 G256 A257 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 Ki=480uM remove_due_to_license_issue P62593 15037085 300 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQRDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTMPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1pzp A 1.45 BS02 FTA A 2 P27 L30 K34 F60 R61 P2 L5 K9 F35 R36 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0005515,0008800,0016787,0017001,0030655,0046677 Ki=480uM remove_due_to_license_issue P62593 15037085 301 HPETLVKVKDAEDQLGARVGYIELDLNSGKILESFRPEERFPMMSTFKVLLCGAVLSRVDAGQEQLGRRIHYSQRDLVEYSPVTEKHLTDGMTVRELCSAAITMSDNTAANLLLTTIGGPKELTAFLHNMGDHVTRLDRWEPELNEAIPNDERDTTMPAAMATTLRKLLTGELLTLASRQQLIDWMEADKVAGPLLRSALPAGWFIADKSGAGERGSRGIIAALGPDGKPSRIVVIYTTGSQATMDERNRQIAEIGASLIKHW 1q0b A 1.9 BS02 NAT A 1 E116 E118 R119 W127 D130 A133 I136 P137 Y211 E101 E103 R104 W112 D115 A118 I121 P122 Y196 ? 0003777,0005524,0007018,0008017 ic50=6.7uM remove_due_to_license_issue IC50=10000nM P52732 14672662 604 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 1q1g A 2.02 BS01 MTI A 1 V66 S91 C92 G93 Y160 E182 M183 E184 D206 V64 S89 C90 G91 Y158 E180 M181 E182 D204 H7 G23 R27 R45 E77 R88 S91 D206 G207 P209 V222 H5 G21 R25 R43 E75 R86 S89 D204 G205 P207 V220 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006148,0006166,0006195,0006218,0009116,0016757,0017061,0047975 Kd=2.7nM remove_due_to_license_issue Q8I3X4 14982926 301 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKWDEGDFDNNLVPHQLENMIKIALGACAKLATKYA 1q1g B 2.02 BS01 MTI A 1 H7 V73 H5 V71 H7 G23 R27 R45 E77 R88 S91 D206 G207 P209 V222 H5 G21 R25 R43 E75 R86 S89 D204 G205 P207 V220 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006148,0006166,0006195,0006218,0009116,0016757,0017061,0047975 Kd=2.7nM remove_due_to_license_issue Q8I3X4 14982926 301 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKWDEGDFDNNLVPHQLENMIKIALGACAKLATKYA 1q1g B 2.02 BS02 MTI B 1 V66 S91 C92 G93 Y160 E182 M183 E184 D206 W212 V64 S89 C90 G91 Y158 E180 M181 E182 D204 W210 H7 G23 R27 R45 E77 R88 S91 D206 G207 P209 V222 H5 G21 R25 R43 E75 R86 S89 D204 G205 P207 V220 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006148,0006166,0006195,0006218,0009116,0016757,0017061,0047975 Kd=2.7nM remove_due_to_license_issue Q8I3X4 14982926 302 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKWDEGDFDNNLVPHQLENMIKIALGACAKLATKYA 1q1m A 2.6 BS01 234 A 1 R24 Y46 V49 F182 C215 S216 A217 I219 G220 R221 R254 G259 Q262 L299 R23 Y45 V48 F181 C214 S215 A216 I218 G219 R220 R253 G258 Q261 L298 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Ki=6900nM, IC50=110000nM P18031 13678400 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 1q1y A 1.9 BS02 BB2 A 1 R56 S57 G58 V59 G60 Q65 E109 A111 L112 V151 H154 E155 H158 R56 S57 G58 V59 G60 Q65 E109 A111 L112 V151 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 3.5.1.88 0006412,0016787,0042586,0043686,0046872 remove_due_to_license_issue IC50=<5nM P68826 15382235 301 MLTMKDIIRDGHPTLRQKAAELELPLTKEEKETLIAMREFLVNSQDEEIAKRYGLRSGVGLAAPQINISKRMIAVLIPDDGSGKSYDYMLVNPKIVSHSVQEAYLPTGEGCLSVDDNVAGLVHRHNRITIKAKDIEGNDIQLRLKGYPAIVFQHEIDHLNGVMFYDHIDKDHPLQPHTDAVEVLEH 1q3d A 2.2 BS01 STU A 1 I62 G63 V70 D133 Y134 V135 Q185 L188 D200 I28 G29 V36 D93 Y94 V95 Q145 L148 D160 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=15nM remove_due_to_license_issue P49841 14529625 451 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQ 1q3d B 2.2 BS01 STU B 1 I62 G63 G65 A83 K85 D133 Y134 V135 L188 D200 I28 G29 G31 A49 K51 D95 Y96 V97 L150 D162 D181 K183 N186 D200 S219 D143 K145 N148 D162 S181 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=15nM remove_due_to_license_issue P49841 14529625 452 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 1q3w B 2.3 BS01 ATU B 1 K85 Y134 V135 P136 T138 R141 L188 C199 D200 K51 Y97 V98 P99 T101 R104 L151 C162 D163 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=4nM remove_due_to_license_issue IC50=4nM P49841 14529625 501 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 1q41 A 2.1 BS01 IXM A 1 I62 A83 Y134 V135 P136 T138 R141 L188 C199 I28 A49 Y94 V95 P96 T98 R101 L148 C159 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=22nM remove_due_to_license_issue IC50=200nM P49841 14529625 451 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQA 1q4l A 2.77 BS01 679 A 1 I62 G63 N64 G65 K85 Y134 V135 R141 Q185 L188 C199 D200 I28 G29 N30 G31 K51 Y97 V98 R104 Q148 L151 C162 D163 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue IC50=76nM P49841 14529625 451 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQA 1q4w A 1.93 BS02 DQU A 1 D102 Y106 D156 G229 G230 M260 D92 Y96 D144 G217 G218 M248 D102 D280 C318 C320 C323 H349 D92 D268 C299 C301 C304 H330 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=0.35uM remove_due_to_license_issue P28720 15050823 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 1q4x A 2.8 BS01 G24 A 1 F269 F272 T273 L330 N331 L346 H435 F451 F455 F47 F50 T51 L108 N109 L124 H213 F229 F233 ? 0003677,0004879,0006355 remove_due_to_license_issue P10828 14673100 462 GHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPGKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 1q54 A 1.93 BS03 BHI A 1 R51 K55 A67 G68 R83 E87 E114 E116 W161 R48 K52 A64 G65 R80 E84 E111 E113 W158 H25 H32 A67 H69 E87 Y104 E114 E116 W161 H22 H29 A64 H66 E84 Y101 E111 E113 W158 5.3.3.2 0000287,0003824,0004452,0005737,0006974,0008270,0008299,0016853,0046872,0050992 Ki=1.4uM remove_due_to_license_issue Q46822 12630859 301 EHVILLNAQGVPTGTLEKYAAHTADTRLHLAFSSWLFNAKGQLLVTRRALSKKAWPGVWTNSVAGHPQLGESNEDAVIRRCRYELGVEITPPESIYPDFRYRATDPSGIVENEVCPVFAARTTSALQINDDEVMDYQWCDLADVLHGIDATPWAFSPWMVMQATNREARKRLSAFT 1q5k A 1.94 BS01 TMU A 1 I62 A83 Y134 V135 P136 R141 L188 I28 A49 Y98 V99 P100 R105 L152 D181 K183 N186 D200 S219 D145 K147 N150 D164 S183 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 Ki=38nM remove_due_to_license_issue IC50=104nM, Ki=38nM P49841 12928438 901 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 1q63 A 1.85 BS02 AIQ A 1 D102 D156 C158 G229 M260 D280 D92 D140 C142 G213 M244 D264 D102 D280 C318 C320 C323 H349 D92 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=1.4uM remove_due_to_license_issue P28720 15050823 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSTKQSEEGVTFKSHRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1q65 A 2.1 BS02 BHB A 1 D102 Y106 Q107 D156 G229 M260 D92 Y96 Q97 D143 G216 M247 D102 D280 C318 C320 C323 H349 D92 D267 C305 C307 C310 H336 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=3.5uM remove_due_to_license_issue P28720 15050823 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1q66 A 1.75 BS02 KMB A 1 L68 N70 D102 Y106 D156 G229 G230 L231 A232 M260 L58 N60 D92 Y96 D141 G214 G215 L216 A217 M245 D102 D280 C318 C320 C323 H349 D92 D265 C300 C302 C305 H331 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=1.7uM remove_due_to_license_issue P28720 15050823 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLTKQSEEGVTFKSHLSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1q6j A 2.2 BS01 335 A 1 Y46 R47 D48 V49 S118 L119 F182 C215 S216 A217 I219 G220 R221 Q262 Y50 R51 D52 V53 S122 L123 F186 C219 S220 A221 I223 G224 R225 Q266 D181 C215 R221 S222 Q262 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=0.016uM remove_due_to_license_issue IC50=16nM P18031 14516196 301 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6k A 2.1 BS01 TCO A 1 G23 C25 G64 G65 G66 L160 N161 G23 C25 G64 G65 G66 L160 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 ic50=26nM remove_due_to_license_issue IC50=26nM P43235 14684342 0 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1q6m A 2.2 BS01 P27 A 1 Y46 R47 D48 V49 S118 L119 F182 C215 S216 A217 I219 G220 R221 Q262 Y50 R51 D52 V53 S122 L123 F186 C219 S220 A221 I223 G224 R225 Q266 D181 C215 R221 S222 Q262 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=0.013uM remove_due_to_license_issue IC50=120nM P18031 14516196 301 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6n A 2.1 BS01 P90 A 1 Y546 R547 D548 V549 L619 F682 C715 S716 A717 I719 G720 R721 M758 Q762 Y50 R51 D52 V53 L123 F186 C219 S220 A221 I223 G224 R225 M262 Q266 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=0.023uM remove_due_to_license_issue P18031 14516196 801 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6n A 2.1 BS02 P90 B 1 A518 Q521 A22 Q25 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=0.023uM remove_due_to_license_issue P18031 14516196 1301 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6p A 2.3 BS01 213 A 1 Y546 R547 D548 F682 C715 S716 A717 I719 G720 R721 M758 G759 Q762 Y50 R51 D52 F186 C219 S220 A221 I223 G224 R225 M262 G263 Q266 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=3nM remove_due_to_license_issue IC50=3nM P18031 14516196 801 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1q6p A 2.3 BS02 213 B 1 D522 H525 E526 D26 H29 E30 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=3nM remove_due_to_license_issue IC50=3nM P18031 14516196 1301 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1q6s A 2.2 BS01 214 A 1 R524 D529 Y546 R547 D548 F682 C715 S716 A717 I719 G720 R721 R754 M758 Q762 R28 D33 Y50 R51 D52 F186 C219 S220 A221 I223 G224 R225 R258 M262 Q266 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=12nM remove_due_to_license_issue IC50=220nM P18031 14516196 801 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6s A 2.2 BS02 214 B 1 A518 D522 H525 E526 A22 D26 H29 E30 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=12nM remove_due_to_license_issue IC50=220nM P18031 14516196 1301 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6t A 2.3 BS01 600 A 1 R524 S528 D529 Y546 R547 D548 F552 F682 C715 S716 A717 I719 G720 R721 M758 Q762 R28 S32 D33 Y50 R51 D52 F56 F186 C219 S220 A221 I223 G224 R225 M262 Q266 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=5nM remove_due_to_license_issue IC50=5340nM P18031 14516196 801 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q6t A 2.3 BS02 600 B 1 D522 H525 E526 D26 H29 E30 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=5nM remove_due_to_license_issue IC50=5340nM P18031 14516196 1301 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 1q72 H 1.7 BS01 COC H 1 D31 W33 V95 Q97 D31 W33 V101 Q103 Kd=0.0000123M remove_due_to_license_issue 15885702 401 EVTLQESGGGLVQPGGSMKLSCAASGFTFSDAWVDWVRQSPGKGLEWVAEIRNKANNHATKYTESVKGRFTISRDDSKSSVYLQMNSLRAEDTGIYYCTSVPQLGRGFAYWGQGTLVTVSAASTTPPSVYPLAPGSGGAGSMVTLGCLVKGYFPEPVTVTWNSGALSSGVHTFPAVLNGDLYTLSSSVTVPSSTWPSQTVTCNVAHPASSTQVDKKIVPK 1q72 L 1.7 BS01 COC H 1 Y32 H91 F96 Y37 H96 F101 remove_due_to_license_issue 15885702 401 DIVMTQAAPSVPVTPGESVSISCRSSKSLLHSNGYTYLHWFLQRPGQSPQLLIYRVSNLASGVPDRFSGSGSGTAFTLRFSRVEAEDVGVYYCMQHLEYPFTFGSGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPQDITVSWKIDGAERSSGVLNSWTDQDSSDSTYSMSSTLTLTKDEYERHSSYTCEATHKTSTSPITKSFNRGE 1q7a A 1.6 BS02 OPB A 1 L2 F5 G29 W30 H47 Y51 K60 L2 F5 G29 W30 H47 Y51 K60 Y27 G29 G31 H47 D48 Y51 Y64 D89 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 Kd=0.000000064M remove_due_to_license_issue P59071 15544328 124 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 1q83 A 2.65 BS01 TZ5 A 1 Y72 W86 G121 Y124 E202 W286 Y337 Y341 W439 H447 Y72 W86 G121 Y124 E202 W281 Y332 Y336 W434 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0004104 remove_due_to_license_issue Ki=0.410nM, Kd=0.00041nM P21836 14757816 1951 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 1q84 A 2.45 BS01 TZ4 A 1 Y72 W86 G121 Y124 E202 W286 L289 S293 Y337 Y341 W439 H447 Y72 W86 G121 Y124 E202 W281 L284 S288 Y332 Y336 W434 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0004104 Ki=8900fM remove_due_to_license_issue P21836 14757816 951 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 1q8t A 2.0 BS02 Y27 A 1 A70 Y122 V123 N171 F327 A61 Y113 V114 N162 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=17.5uM remove_due_to_license_issue IC50=42000nM P00517 14656443 930 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1q8u A 1.9 BS02 H52 A 1 T51 V57 A70 M120 E121 Y122 V123 E170 L173 F327 T45 V51 A64 M114 E115 Y116 V117 E164 L167 F321 D166 K168 E170 N171 D184 T201 D160 K162 E164 N165 D178 T195 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=1.1uM remove_due_to_license_issue IC50=394nM P00517 14656443 961 KKGSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1q8u A 1.9 BS03 H52 A 2 E86 K189 T197 E80 K183 T191 D166 K168 E170 N171 D184 T201 D160 K162 E164 N165 D178 T195 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=1.1uM remove_due_to_license_issue IC50=394nM P00517 14656443 962 KKGSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1q8w A 2.2 BS02 M77 A 1 V57 A70 M120 Y122 V123 E170 T183 F327 V44 A57 M107 Y109 V110 E157 T170 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=5.7uM remove_due_to_license_issue IC50=1494nM P00517 14656443 960 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1q91 A 1.6 BS03 DPB A 1 F49 F75 W76 V77 W96 S131 I133 K134 R163 F16 F42 W43 V44 W63 S98 I100 K101 R130 D41 D43 D176 D8 D10 D143 3.1.3.- 0008253,0009264 Ki=70uM remove_due_to_license_issue Q9NPB1 15044615 1 RALRVLVDMDGVLADFEGGFLRKFRARFPDQPFIALEDRRGFWVSEQYGRLRPGLSEKAISIWESKNFFFELEPLPGAVEAVKEMASLQNTDVFICTSPIKMFKYCPYEKYAWVEKYFGPDFLEQIVLTRDKTVVSADLLIDDRPDITGAEPTPSWEHVLFTACHNQHLQLQPPRRRLHSWADDWKAILDSKRP 1q95 A 2.46 BS01 PAL A 1 T53 R54 T55 R105 H134 R167 R229 Q231 P268 T53 R54 T55 R105 H134 R167 R229 Q231 P268 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=27nM remove_due_to_license_issue P0A786 15157075 1001 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 1q95 B 2.46 BS01 PAL A 1 S80 K84 S80 K84 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=27nM remove_due_to_license_issue P0A786 15157075 1001 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 1q95 B 2.46 BS02 PAL B 1 T53 R54 T55 R105 H134 R167 T168 R229 Q231 P266 P268 T53 R54 T55 R105 H134 R167 T168 R229 Q231 P266 P268 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=27nM remove_due_to_license_issue P0A786 15157075 1002 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 1q9d A 2.35 BS06 OI1 A 1 D187 A189 I190 D180 A182 I183 D68 D74 E97 E98 D118 L120 D121 E280 D61 D67 E90 E91 D111 L113 D114 E273 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=1.87uM remove_due_to_license_issue P00636 14530289 416 TNIVTLTRFVMEEGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGSTNVTGDQVKKLDVLSNDLVINVLKSSFATCVLVSEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRDVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1q9d A 2.35 BS07 OI1 B 1 G52 H55 G45 H48 D68 D74 E97 E98 D118 L120 D121 E280 D61 D67 E90 E91 D111 L113 D114 E273 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=1.87uM remove_due_to_license_issue P00636 14530289 406 TNIVTLTRFVMEEGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGSTNVTGDQVKKLDVLSNDLVINVLKSSFATCVLVSEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRDVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1q9d B 2.35 BS01 OI1 A 1 G52 H55 G45 H48 D68 D74 E97 E98 D118 L120 D121 E280 D61 D67 E90 E91 D111 L113 D114 E273 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=1.87uM remove_due_to_license_issue P00636 14530289 416 TNIVTLTRFVMEEGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGSTNVTGDQVKKLDVLSNDLVINVLKSSFATCVLVSEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRDVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1q9d B 2.35 BS07 OI1 B 1 D187 A189 I190 D180 A182 I183 D68 D74 E97 E98 D118 L120 D121 E280 D61 D67 E90 E91 D111 L113 D114 E273 3.1.3.11 0000122,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0071286,0071466 ic50=1.87uM remove_due_to_license_issue P00636 14530289 406 TNIVTLTRFVMEEGRKARGTGEMTQLLNSLCTAVKAISTAVRKAGIAHLYGIAGSTNVTGDQVKKLDVLSNDLVINVLKSSFATCVLVSEEDKNAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSIGTIFGIYRKNSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMVNGVNCFMLDPAIGEFILVDRDVKIKKKGSIYSINEGYAKEFDPAITEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFMYPANKKSPKGKLRLLYECNPMAYVMEKAGGLATTGKEAVLDIVPTDIHQRAPIILGSPEDVTELLEIYQKHA 1q9m A 2.3 BS02 ROL A 1 Y159 H160 I336 M357 Q369 F372 Y81 H82 I258 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=0.33uM remove_due_to_license_issue Q08499 12842049 503 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 1q9x A 2.69 BS01 dna E 0 S360 Y391 P392 G393 A394 V396 G571 W574 K705 K706 R707 K800 K844 K878 S360 Y391 P392 G393 A394 V396 G571 W574 K705 K706 R707 K800 K844 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 910 ~ 928 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x A 2.69 BS02 dna I 0 N284 K706 M728 K734 S735 S783 S784 N786 Y791 K800 H804 N284 K706 M728 K734 S735 S783 S784 N786 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 940 ~ 952 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x A 2.69 BS03 dna H 0 S36 F38 Y49 G84 D95 F370 K374 K378 I380 S36 F38 Y49 G84 D95 F370 K374 K378 I380 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 910 ~ 928 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x B 2.69 BS01 dna F 0 Y391 P392 G393 F395 V396 Y567 G571 N572 W574 K705 K706 R707 K800 C801 K844 K874 K878 Y391 P392 G393 F395 V396 Y567 G571 N572 W574 K705 K706 R707 K800 C801 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 910 ~ 928 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x B 2.69 BS02 dna J 0 N284 K706 M728 G729 Q733 K734 S735 S784 N786 K790 Y791 K800 H804 N284 K706 M728 G729 Q733 K734 S735 S784 N786 K790 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 940 ~ 952 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x C 2.69 BS01 dna G 0 Y391 G393 A394 F395 V396 Y567 G571 N572 W574 K705 K706 R707 K800 K844 K874 Y391 G393 A394 F395 V396 Y567 G571 N572 W574 K705 K706 R707 K800 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 910 ~ 928 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x C 2.69 BS02 dna K 0 N284 K706 M728 G729 K734 S735 S783 S784 N786 K790 Y791 K800 H804 N284 K706 M728 G729 K734 S735 S783 S784 N786 K790 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 940 ~ 952 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x D 2.69 BS01 dna H 0 S360 Y391 G393 A394 F395 V396 Y567 G571 N572 W574 K705 R707 K800 C801 F803 K874 S360 Y391 G393 A394 F395 V396 Y567 G571 N572 W574 K705 R707 K800 C801 F803 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 910 ~ 928 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9x D 2.69 BS02 dna L 0 N284 K706 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 K706 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 940 ~ 952 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 1q9y A 2.8 BS01 dna T 0 S363 P364 I365 Y394 P395 G396 N567 S568 Y570 G571 N575 W577 K708 K709 R710 K803 F806 K847 K877 S363 P364 I365 Y394 P395 G396 N567 S568 Y570 G571 N575 W577 K708 K709 R710 K803 F806 K847 K877 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 907 ~ 924 HGSMKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFD 1q9y A 2.8 BS02 dna P 0 N287 D624 T625 K709 M731 G732 K737 S738 S739 S786 S787 N789 Y794 K803 H807 N287 D624 T625 K709 M731 G732 K737 S738 S739 S786 S787 N789 Y794 K803 H807 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 15057282 925 ~ 938 HGSMKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFD 1qan A 2.4 BS01 SAH A 1 N11 F12 G38 S39 G40 E59 I60 L64 D84 I85 N101 N3 F4 G30 S31 G32 E51 I52 L56 D76 I77 N93 G38 E59 N101 Y104 F163 G30 E51 N93 Y96 F155 2.1.1.184 0000154,0000179,0003723,0005829,0008168,0031167,0032259,0046677,0052910 Ki=33uM remove_due_to_license_issue P13956 10366505 501 SQNFITSKHNIDKIMTNIRLNEHDNIFEIGSGKGHFTLELVQRCNFVTAIEIDHKLCKTTENKLVDHDNFQVLNKDILQFKFPKNQSYKIFGNIPYNISTDIIRKIVFDSIADEIYLIVEYGFAKRLLNTKRSLALFLMAEVDISILSMVPREYFHPKPKVNSSLIRLNRKKSRISHKDKQKYNYFVMKWVNKEYKKIFTKNQFNNSLKHAGIDDLNNISFEQFLSLFNSYKLFNK 1qaq A 2.8 BS01 SFG A 1 Q10 N11 F12 I13 G38 S39 G40 E59 I60 L64 D84 I85 N101 P103 I106 Q2 N3 F4 I5 G30 S31 G32 E51 I52 L56 D76 I77 N93 P95 I98 G38 E59 N101 Y104 F163 G30 E51 N93 Y96 F155 2.1.1.184 0000154,0000179,0003723,0005829,0008168,0031167,0032259,0046677,0052910 remove_due_to_license_issue P13956 10366505 245 SQNFITSKHNIDKIMTNIRLNEHDNIFEIGSGKGHFTLELVQRCNFVTAIEIDHKLCKTTENKLVDHDNFQVLNKDILQFKFPKNQSYKIFGNIPYNISTDIIRKIVFDSIADEIYLIVEYGFAKRLLNTKRSLALFLMAEVDISILSMVPREYFHPKPKVNSSLIRLNRKKSRISHKDKQKYNYFVMKWVNKEYKKIFTKNQFNNSLKHAGIDDLNNISFEQFLSLFNSYKLFNK 1qaw A 2.5 BS01 TRP A 1 T25 G27 D29 T30 S53 T19 G21 D23 T24 S47 ? 0003723,0005515,0006353,0006355,0042802 Kd=7.5uM remove_due_to_license_issue Q9X6J6 10369778 81 SDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESE 1qaw A 2.5 BS02 TRP K 1 G23 A46 T49 T52 G17 A40 T43 T46 ? 0003723,0005515,0006353,0006355,0042802 Kd=7.5uM remove_due_to_license_issue Q9X6J6 10369778 81 SDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESE 1qaw B 2.5 BS01 TRP A 1 G23 T49 G17 T43 ? 0003723,0005515,0006353,0006355,0042802 Kd=7.5uM remove_due_to_license_issue Q9X6J6 10369778 81 SDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEGKK 1qaw B 2.5 BS02 TRP B 1 R26 G27 T30 S53 R20 G21 T24 S47 ? 0003723,0005515,0006353,0006355,0042802 Kd=7.5uM remove_due_to_license_issue Q9X6J6 10369778 81 SDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEGKK 1qaw K 2.5 BS01 TRP J 1 G23 H34 T49 G17 H28 T43 ? 0003723,0005515,0006353,0006355,0042802 Kd=7.5uM remove_due_to_license_issue Q9X6J6 10369778 81 SDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1qaw K 2.5 BS02 TRP K 1 T25 G27 T30 S53 T19 G21 T24 S47 ? 0003723,0005515,0006353,0006355,0042802 Kd=7.5uM remove_due_to_license_issue Q9X6J6 10369778 81 SDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1qb1 A 1.8 BS02 974 A 1 N85 T86 D177 S178 Q180 S183 V197 W199 G200 G202 N79 T80 D171 S172 Q174 S177 V191 W193 G194 G196 H46 D90 Q180 G181 D182 S183 G184 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=170nM remove_due_to_license_issue P00760 10417407 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1qb6 A 1.8 BS02 623 A 1 L87 D177 S178 Q180 W199 G200 G202 L81 D171 S172 Q174 W193 G194 G196 H46 D90 Q180 G181 D182 S183 G184 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=870nM remove_due_to_license_issue P00760 10417407 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1qb9 A 1.8 BS03 806 A 1 N85 T86 L87 Q161 D177 S178 W199 G200 G202 N79 T80 L81 Q155 D171 S172 W193 G194 G196 H46 D90 Q180 G181 D182 S183 G184 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=36nM remove_due_to_license_issue Ki=36nM P00760 10417407 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1qbn A 1.8 BS03 688 A 1 N85 D177 S178 Q180 W199 G200 G202 C203 N79 D171 S172 Q174 W193 G194 G196 C197 H46 D90 Q180 G181 D182 S183 G184 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1400nM remove_due_to_license_issue P00760 10417407 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1qbo A 1.8 BS03 711 A 1 N85 T86 Q161 D177 S178 W199 G200 G202 C203 N79 T80 Q155 D171 S172 W193 G194 G196 C197 H46 D90 Q180 G181 D182 S183 G184 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=18nM remove_due_to_license_issue P00760 10417407 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1qbq B 2.4 BS03 HFP B 1 Y205 H248 G250 Y251 C254 R291 W303 Y183 H226 G228 Y229 C232 R269 W281 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 Ki=5nM remove_due_to_license_issue Q02293 9843427 2001 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 1qbr A 1.8 BS01 XV6 A 1 R8 D25 G27 A28 D30 I47 G48 G49 I50 P81 I84 R8 D25 G27 A28 D30 I47 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.027nM remove_due_to_license_issue P04585 9003516 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbr B 1.8 BS01 XV6 A 1 D25 G27 A28 D29 D30 V32 I47 G48 G49 I50 P81 V82 I84 D25 G27 A28 D29 D30 V32 I47 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9003516 638 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbs A 1.8 BS01 DMP A 1 D25 G27 D30 V32 I47 G49 I50 P81 V82 I84 D25 G27 D30 V32 I47 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.34nM remove_due_to_license_issue P04585 8784449 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbs B 1.8 BS01 DMP A 1 D25 G27 D30 G49 I50 D25 G27 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 8784449 323 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbt A 2.1 BS01 146 B 1 D25 G27 A28 D30 I47 G48 G49 I50 I84 D25 G27 A28 D30 I47 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9003516 300 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbt B 2.1 BS01 146 B 1 R8 D25 G27 A28 D30 V32 K45 G48 G49 I50 P81 V82 I84 R8 D25 G27 A28 D30 V32 K45 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.024nM remove_due_to_license_issue P04585 9003516 300 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbu A 1.8 BS01 846 B 1 D25 G27 A28 D29 D30 G48 V82 D25 G27 A28 D29 D30 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 9003516 300 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbu B 1.8 BS01 846 B 1 D25 G27 G49 I50 V82 D25 G27 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.058nM remove_due_to_license_issue P04585 9003516 300 PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1qbv H 1.8 BS03 PPX H 1 Y60A E97A D189 A190 S195 W215 G216 G219 G226 Y47 E94 D191 A192 S197 W219 G220 G222 G230 3.4.21.5 0004252,0005509,0006508,0007596 Ki=4100nM remove_due_to_license_issue Ki=4100nM P00734 9622548 907 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1qca A 2.2 BS02 FUA A 1 C92 F103 F135 F146 F168 C86 F97 F129 F138 F160 R18 T174 H195 D199 R13 T166 H187 D191 2.3.1.28 0008811,0016746,0046677 Ki=5.4uM remove_due_to_license_issue P00484 7500366 221 MNYTKFDVKNWVRREHFEFYRHRLPCGFSLTSKIDITTLKKSLDDSAYKFYPVMIYLIAQAVNQFDELRMAIKDDELIVWDSVDPCFTVFHQETETFSALSCPYSSDIDQFMVNYLSVMERYKSDTKLFPQGPENHLFISALPWVNFDSFNLNVANFTDFFAPVITMAKYQQEGDRLLLPLSVQVHHAVCDGFHVARFINRLQELCNSKLK 1qcp A 1.8 BS02 RWJ A 1 C42 H57 L99 D189 S190 C191 Q192 G193 D194 S195 S214 G216 G219 C25 H40 L81 D171 S172 C173 Q174 G175 D176 S177 S192 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 10531473 300 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1qf0 A 2.2 BS06 TI2 A 1 N112 A113 F114 F130 V139 E143 H146 E166 I188 G189 L202 R203 H231 N112 A113 F114 F130 V139 E143 H146 E166 I188 G189 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=42nM remove_due_to_license_issue P00800 10504225 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1qf1 A 2.0 BS06 TI1 A 1 N112 A113 V139 H142 E143 H146 E166 I188 G189 L202 R203 H231 N112 A113 V139 H142 E143 H146 E166 I188 G189 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=48nM remove_due_to_license_issue P00800 10504225 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1qf2 A 2.06 BS06 TI3 A 1 N112 F130 L133 V139 H142 E143 L202 R203 H231 N112 F130 L133 V139 H142 E143 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=1200nM remove_due_to_license_issue P00800 10504225 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1qf4 A 2.2 BS04 RPD A 1 D13 N38 G40 G127 T128 T129 Q224 L228 V238 V273 G298 A299 T300 T301 R303 D13 N38 G40 G127 T128 T129 Q224 L228 V238 V273 G298 A299 T300 T301 R303 D13 K16 G40 H41 Q224 D13 K16 G40 H41 Q224 6.3.4.4 0000166,0000287,0004019,0005515,0005525,0005737,0005829,0006164,0006974,0015949,0016020,0016874,0044208,0046040,0046086,0046872,0097216 ic50=0.665uM remove_due_to_license_issue P0A7D4 10556888 435 GNNVVVLGTQWGDEGKGKIVDLLTERAKYVVRYQGGHNAGHTLVINGEKTVLHLIPSGILRENVTSIIGNGVVLSPAALMKEMKELEDRGIPVRERLLLSEACPLILDYHVALDNAREKARGAKAIGTTGRGIGPAYEDKVARRGLRVGDLFDKETFAEKLKEVMEYHNFQLVNYYKAEAVDYQKVLDDTMAVADILTSMVVDVSDLLDQARQRGDFVMFEGAQGTLLDIDHGTYPYVTSSNTTAGGVATGSGLGPRYVDYVLGILKAYSTRVGAGPFPTELFDETGEFLCKQGNEFGATTGRRRRTGWLDTVAVRRAVQLNSLSGFCLTKLDVLDGLKEVKLCVAYRMPDGREVTTTPLAADDWKGVEPIYETMPGWSESTFGVKDRSGLPQAALNYIKRIEELTGVPIDIISTGPDRTETMILRDPFDA 1qf5 A 2.0 BS04 RPL A 1 D13 N38 G40 G127 T128 T129 Q224 L228 V238 V273 G298 A299 T300 T301 R303 D13 N38 G40 G127 T128 T129 Q224 L228 V238 V273 G298 A299 T300 T301 R303 D13 K16 G40 H41 Q224 D13 K16 G40 H41 Q224 6.3.4.4 0000166,0000287,0004019,0005515,0005525,0005737,0005829,0006164,0006974,0015949,0016020,0016874,0044208,0046040,0046086,0046872,0097216 ic50=0.043uM remove_due_to_license_issue P0A7D4 10556888 435 GNNVVVLGTQWGDEGKGKIVDLLTERAKYVVRYQGGHNAGHTLVINGEKTVLHLIPSGILRENVTSIIGNGVVLSPAALMKEMKELEDRGIPVRERLLLSEACPLILDYHVALDNAREKARGAKAIGTTGRGIGPAYEDKVARRGLRVGDLFDKETFAEKLKEVMEYHNFQLVNYYKAEAVDYQKVLDDTMAVADILTSMVVDVSDLLDQARQRGDFVMFEGAQGTLLDIDHGTYPYVTSSNTTAGGVATGSGLGPRYVDYVLGILKAYSTRVGAGPFPTELFDETGEFLCKQGNEFGATTGRRRRTGWLDTVAVRRAVQLNSLSGFCLTKLDVLDGLKEVKLCVAYRMPDGREVTTTPLAADDWKGVEPIYETMPGWSESTFGVKDRSGLPQAALNYIKRIEELTGVPIDIISTGPDRTETMILRDPFDA 1qfq B -1.00 BS01 rna A 0 D2 A3 Q4 R6 R7 R8 R11 K14 Q15 W18 K19 D1 A2 Q3 R5 R6 R7 R10 K13 Q14 W17 K18 ? remove_due_to_license_issue P03045 10759866 1 ~ 15 DAQTRRRERRAEKQAQWKAANPLLVGVSAKPVNRP 1qfs A 2.0 BS01 ZPR A 1 M235 Y473 F476 S554 N555 A594 W595 R643 V644 M235 Y473 F476 S554 N555 A594 W595 R643 V644 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue IC50=0.33nM P23687 9695945 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 1qft A 1.25 BS01 HSM A 1 S20 D24 Y29 F98 Y100 D120 W137 S20 D24 Y29 F98 Y100 D120 W137 ? 0005576,0030682,0043176 Kd=1.7nM remove_due_to_license_issue O77421 10360182 176 NQPDWADEAANGAHQDAWKSLKADVENVYYMVKATYKNDPVWGNDFTCVGVMANDVNEDEKSIQAEFLFMNNADTNMQFATEKVTAVKMYGYNRENAFRYETEDGQVFTDVIAYSDDNCDVIYVPGTDGNEEGYELWTTDYDNIPANCLNKFNEYAVGRETRDVFTSACLEIAAA 1qft A 1.25 BS02 HSM A 2 D39 W42 E82 Y100 F108 D110 E135 D39 W42 E82 Y100 F108 D110 E135 ? 0005576,0030682,0043176 Kd=1.7nM remove_due_to_license_issue O77421 10360182 177 NQPDWADEAANGAHQDAWKSLKADVENVYYMVKATYKNDPVWGNDFTCVGVMANDVNEDEKSIQAEFLFMNNADTNMQFATEKVTAVKMYGYNRENAFRYETEDGQVFTDVIAYSDDNCDVIYVPGTDGNEEGYELWTTDYDNIPANCLNKFNEYAVGRETRDVFTSACLEIAAA 1qhc A 1.7 BS01 PUA A 1 K7 H12 K41 V43 N44 T45 C65 N67 Q69 N71 A109 E111 V118 H119 F120 K7 H12 K41 V43 N44 T45 C65 N67 Q69 N71 A109 E111 V118 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=27nM remove_due_to_license_issue P61823 10441122 901 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1qhr B 2.2 BS02 157 B 1 H57 W60D W148 D189 A190 C191 E192 G193 S195 V213 G216 H43 W50 W148 D199 A200 C201 E202 G203 S205 V225 G228 H57 D102 E192 G193 D194 S195 G196 H43 D99 E202 G203 D204 S205 G206 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=130nM P00734 10387040 500 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1qin A 2.0 BS02 GIP A 1 R122 H126 K150 G155 K156 M157 E172 M179 R115 H119 K143 G148 K149 M150 E165 M172 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Ki=10nM remove_due_to_license_issue Q04760 10521255 300 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 1qin A 2.0 BS03 GIP B 1 Q33 R37 F67 L69 F71 E99 T101 N103 Q26 R30 F60 L62 F64 E92 T94 N96 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Ki=10nM remove_due_to_license_issue Q04760 10521255 400 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 1qin B 2.0 BS01 GIP A 1 Q33 R37 F67 L69 F71 E99 T101 N103 Q26 R30 F60 L62 F64 E92 T94 N96 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Ki=10nM remove_due_to_license_issue Q04760 10521255 300 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 1qin B 2.0 BS03 GIP B 1 R122 H126 K150 G155 K156 M157 E172 M179 R115 H119 K143 G148 K149 M150 E165 M172 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Ki=10nM remove_due_to_license_issue Q04760 10521255 400 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 1qj7 B 2.2 BS02 GR1 B 1 H57 E97A N98 W148 I174 D189 A190 E192 G193 S195 W215 G216 G219 H43 E94 N95 W148 I179 D199 A200 E202 G203 S205 W227 G228 G230 H57 D102 E192 G193 D194 S195 G196 H43 D99 E202 G203 D204 S205 G206 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 10387040 1248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1qji A 2.14 BS02 PKF A 1 C64 W65 S66 Y67 H92 E93 H96 H102 Y149 D175 C64 W65 S66 Y67 H92 E93 H96 H102 Y149 D175 H92 E93 H96 H102 Y149 H92 E93 H96 H102 Y149 3.4.24.21 0004222,0006508,0008237,0008270 Ki=14uM remove_due_to_license_issue P07584 8756323 1202 AAILGDEYLWSGGVIPYTFAGVSGADQSAILSGMQELEEKTCIRFVPRTTESDYVEIFTSGSGCWSYVGRISGAQQVSLQANGCVYHGTIIHELMHAIGFYHEHTRMDRDNYVTINYQNVDPSMTSNFDIDTYSRYVGEDYQYYSIMHYGKYSFSIQWGVLETIVPLQNGIDLTDPYDKAHMLQTDANQINNLYTNECSL 1qk3 A 1.65 BS01 5GP A 1 I148 D150 T151 G152 T154 K178 W199 I200 I148 D150 T151 G152 T154 K178 W199 I200 E146 D147 D150 W199 R212 E146 D147 D150 W199 R212 2.4.2.22,2.4.2.8 0000166,0000287,0000310,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032265,0046100,0046872,0052657 Kd=7.1uM remove_due_to_license_issue Q26997 10545170 300 MASKPIEDYGKGKGRIEPMYIPDNTFYNADDFLVPPHCKPYIDKILLPGGLVKDRVEKLAYDIHRTYFGEELHIICILKGSRGFFNLLIDYLATIQKYSGRESSVPPFFEHYVRLKSYQNDNSTGQLTVLSDDLSIFRDKHVLIVEDIVDTGFTLTEFGERLKAVGPKSMRIATLVEKRTDRSNSLKGDFVGFSIEDVWIVGCCYDFNEMFRDFDHVAVLSDAARKKF 1qk3 B 1.65 BS01 5GP B 1 K79 E146 I148 D150 G152 T154 K178 W199 I200 K82 E149 I151 D153 G155 T157 K181 W202 I203 E146 D147 D150 W199 R212 E149 D150 D153 W202 R215 2.4.2.22,2.4.2.8 0000166,0000287,0000310,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032265,0046100,0046872,0052657 Kd=7.1uM remove_due_to_license_issue Q26997 10545170 300 GSHMASKPIEDYGKGKGRIEPMYIPDNTFYNADDFLVPPHCKPYIDKILLPGGLVKDRVEKLAYDIHRTYFGEELHIICILKGSRGFFNLLIDYLATIQKYSGRESSVPPFFEHYVRLKSYQNDNSTGQLTVLSDDLSIFRDKHVLIVEDIVDTGFTLTEFGERLKAVGPKSMRIATLVEKRTDRSNSLKGDFVGFSIEDVWIVGCCYDFNEMFRDFDHVAVLSDAARKKF 1qk4 A 1.9 BS01 IMP A 1 E146 D147 I148 D150 T151 G152 T154 K178 W199 I200 E141 D142 I143 D145 T146 G147 T149 K173 W194 I195 E146 D147 D150 W199 R212 E141 D142 D145 W194 R207 2.4.2.22,2.4.2.8 0000166,0000287,0000310,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032265,0046100,0046872,0052657 Kd=61uM remove_due_to_license_issue Q26997 10545170 300 MASKPIEDYGKGKGRIEPMYIPDNTFYNADDFLVPPHCKPYIDKILLPGGLVKDRVEKLAYDIHRTYFGEELHIICILKGSRGFFNLLIDYLATIQKYSGRESSVPPFFEHYVRLKSYQGQLTVLSDDLSIFRDKHVLIVEDIVDTGFTLTEFGERLKAVGPKSMRIATLVEKRTDRSNSLKGDFVGFSIEDVWIVGCCYDFNEMFRDFDHVAVLSDAARKKFE 1qkn A 2.25 BS01 RAL A 1 T254 A257 E260 L261 M291 L298 F311 I328 I331 G427 H430 L431 T38 A41 E44 L45 M75 L82 F95 I112 I115 G211 H214 L215 ? remove_due_to_license_issue Q62986 10469641 600 TLSPEQLVLTLLEAEPPNVLVSRPSMPFTEASMMMSLTKLADKELVHMIGWAKKIPGFVELSLLDQVRLLESCWMEVLMVGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLASANQEAESSRKLTHLLNAVTDALVWVIAKSGISSQQQSVRLANLLMLLSHVRHISNKGMEHLLSMKDLLLEMLNA 1qkt A 2.2 BS01 EST A 1 L346 E353 L387 F404 M421 L43 E50 L84 F101 M118 ? Kd=0.92nM remove_due_to_license_issue IC50=1.3nM, Kd=0.2nM, EC50=0.75nM, Ki=0.21nM P03372 11278577 600 NSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKSKNVVPLYDLLLEMLDAHRLHA 1qku A 3.2 BS01 EST A 1 E353 L387 F404 H524 L525 E53 L87 F104 H224 L225 ? remove_due_to_license_issue IC50=1.3nM, Kd=0.2nM, EC50=0.75nM, Ki=0.21nM P03372 11278577 600 SKKNSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLH 1ql7 A 2.1 BS02 ZEN A 1 T98 S190 Q192 V213 W215 G216 S217 G219 C220 G226 V227 Y228 T80 S172 Q174 V191 W193 G194 S195 G196 C197 G204 V205 Y206 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=15uM remove_due_to_license_issue P00760 11921406 999 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1ql9 A 2.3 BS02 ZEN A 1 T98 Y99 S190 Q192 V213 W215 G216 Y217 C220 G226 V227 Y228 T80 Y81 S172 Q174 V191 W193 G194 Y195 C197 G204 V205 Y206 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0005509,0005515,0005576,0005615,0006508,0007584,0007586,0008236,0030574,0046872 Ki=4.45uM remove_due_to_license_issue P00763 12527302 999 IVGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIKHPNFDRETYNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASYPGKITDNMVCVGFLEGGKDSCQGDSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN 1qm5 A 2.0 BS01 GLC C 1 E350 H536 E350 H536 H345 K533 R534 K539 T641 K645 H345 K533 R534 K539 T641 K645 2.4.1.1 0004645,0005737,0005829,0005975,0005980,0008184,0016757,0030170,0030980,0031220,0042803 remove_due_to_license_issue P00490 10469642 1 SQPIFNDKQFQEALSRQWQRYGLNSAAEMTPRQWWLAVSEALAEMLRAQPFAKPVANQRHVNYISMEFLIGRLTGNNLLNLGWYQDVQDSLKAYDINLTDLLEEEIDPALGNGGLGRLAACFLDSMATVGQSATGYGLNYQYGLFRQSFVDGKQVEAPDDWHRSNYPWFRHNEALDVQVGIGGKVTKDGRWEPEFTITGQAWDLPVVGYRNGVAQPLRLWQATHAHPFDLTKFNDGDFLRAEQQGINAEKLTKVLYPNDNHTAGKKLRLMQQYFQCACSVADILRRHHLAGRKLHELADYEVIQLNDTHPTIAIPELLRVLIDEHQMSWDDAWAITSKTFAYTNHTLMPEALERWDVKLVKGLLPRHMQIINEINTRFKTLVEKTWPGDEKVWAKLAVVHDKQVHMANLCVVGGFAVNGVAALHSDLVVKDLFPEYHQLWPNKFHNVTNGITPRRWIKQCNPALAALLDKSLQKEWANDLDQLINLEKFADDAKFRDQYREIKQANKVRLAEFVKVRTGIEINPQAIFDIQIKRLHEYKRQHLNLLHILALYKEIRENPQADRVPRVFLFGAKAAPGYYLAKNIIFAINKVADVINNDPLVGDKLKVVFLPDYCVSAAEKLIPAADISEQISTAGKEASGTGNMKLALNGALTVGTLDGANVEIAEKVGEENIFIFGHTVEQVKAILAKGYDPVKWRKKDKVLDAVLKELESGKYSDGDKHAFDQMLHSIGKQGGDPYLVMADFAAYVEAQKQVDVLYRDQEAWTRAAILNTARCGMFSSDRSIRDYQARIWQAKR 1qm5 A 2.0 BS02 GLC C 2 E350 R534 Y578 E350 R534 Y578 H345 K533 R534 K539 T641 K645 H345 K533 R534 K539 T641 K645 2.4.1.1 0004645,0005737,0005829,0005975,0005980,0008184,0016757,0030170,0030980,0031220,0042803 remove_due_to_license_issue P00490 10469642 2 SQPIFNDKQFQEALSRQWQRYGLNSAAEMTPRQWWLAVSEALAEMLRAQPFAKPVANQRHVNYISMEFLIGRLTGNNLLNLGWYQDVQDSLKAYDINLTDLLEEEIDPALGNGGLGRLAACFLDSMATVGQSATGYGLNYQYGLFRQSFVDGKQVEAPDDWHRSNYPWFRHNEALDVQVGIGGKVTKDGRWEPEFTITGQAWDLPVVGYRNGVAQPLRLWQATHAHPFDLTKFNDGDFLRAEQQGINAEKLTKVLYPNDNHTAGKKLRLMQQYFQCACSVADILRRHHLAGRKLHELADYEVIQLNDTHPTIAIPELLRVLIDEHQMSWDDAWAITSKTFAYTNHTLMPEALERWDVKLVKGLLPRHMQIINEINTRFKTLVEKTWPGDEKVWAKLAVVHDKQVHMANLCVVGGFAVNGVAALHSDLVVKDLFPEYHQLWPNKFHNVTNGITPRRWIKQCNPALAALLDKSLQKEWANDLDQLINLEKFADDAKFRDQYREIKQANKVRLAEFVKVRTGIEINPQAIFDIQIKRLHEYKRQHLNLLHILALYKEIRENPQADRVPRVFLFGAKAAPGYYLAKNIIFAINKVADVINNDPLVGDKLKVVFLPDYCVSAAEKLIPAADISEQISTAGKEASGTGNMKLALNGALTVGTLDGANVEIAEKVGEENIFIFGHTVEQVKAILAKGYDPVKWRKKDKVLDAVLKELESGKYSDGDKHAFDQMLHSIGKQGGDPYLVMADFAAYVEAQKQVDVLYRDQEAWTRAAILNTARCGMFSSDRSIRDYQARIWQAKR 1qm5 A 2.0 BS03 GLC C 3 N112 Y256 R268 H309 R534 N112 Y256 R268 H309 R534 H345 K533 R534 K539 T641 K645 H345 K533 R534 K539 T641 K645 2.4.1.1 0004645,0005737,0005829,0005975,0005980,0008184,0016757,0030170,0030980,0031220,0042803 remove_due_to_license_issue P00490 10469642 3 SQPIFNDKQFQEALSRQWQRYGLNSAAEMTPRQWWLAVSEALAEMLRAQPFAKPVANQRHVNYISMEFLIGRLTGNNLLNLGWYQDVQDSLKAYDINLTDLLEEEIDPALGNGGLGRLAACFLDSMATVGQSATGYGLNYQYGLFRQSFVDGKQVEAPDDWHRSNYPWFRHNEALDVQVGIGGKVTKDGRWEPEFTITGQAWDLPVVGYRNGVAQPLRLWQATHAHPFDLTKFNDGDFLRAEQQGINAEKLTKVLYPNDNHTAGKKLRLMQQYFQCACSVADILRRHHLAGRKLHELADYEVIQLNDTHPTIAIPELLRVLIDEHQMSWDDAWAITSKTFAYTNHTLMPEALERWDVKLVKGLLPRHMQIINEINTRFKTLVEKTWPGDEKVWAKLAVVHDKQVHMANLCVVGGFAVNGVAALHSDLVVKDLFPEYHQLWPNKFHNVTNGITPRRWIKQCNPALAALLDKSLQKEWANDLDQLINLEKFADDAKFRDQYREIKQANKVRLAEFVKVRTGIEINPQAIFDIQIKRLHEYKRQHLNLLHILALYKEIRENPQADRVPRVFLFGAKAAPGYYLAKNIIFAINKVADVINNDPLVGDKLKVVFLPDYCVSAAEKLIPAADISEQISTAGKEASGTGNMKLALNGALTVGTLDGANVEIAEKVGEENIFIFGHTVEQVKAILAKGYDPVKWRKKDKVLDAVLKELESGKYSDGDKHAFDQMLHSIGKQGGDPYLVMADFAAYVEAQKQVDVLYRDQEAWTRAAILNTARCGMFSSDRSIRDYQARIWQAKR 1qm5 A 2.0 BS04 SGC C 1 E67 G113 G114 L115 Y256 D307 T346 R534 E67 G113 G114 L115 Y256 D307 T346 R534 H345 K533 R534 K539 T641 K645 H345 K533 R534 K539 T641 K645 2.4.1.1 0004645,0005737,0005829,0005975,0005980,0008184,0016757,0030170,0030980,0031220,0042803 remove_due_to_license_issue P00490 10469642 4 SQPIFNDKQFQEALSRQWQRYGLNSAAEMTPRQWWLAVSEALAEMLRAQPFAKPVANQRHVNYISMEFLIGRLTGNNLLNLGWYQDVQDSLKAYDINLTDLLEEEIDPALGNGGLGRLAACFLDSMATVGQSATGYGLNYQYGLFRQSFVDGKQVEAPDDWHRSNYPWFRHNEALDVQVGIGGKVTKDGRWEPEFTITGQAWDLPVVGYRNGVAQPLRLWQATHAHPFDLTKFNDGDFLRAEQQGINAEKLTKVLYPNDNHTAGKKLRLMQQYFQCACSVADILRRHHLAGRKLHELADYEVIQLNDTHPTIAIPELLRVLIDEHQMSWDDAWAITSKTFAYTNHTLMPEALERWDVKLVKGLLPRHMQIINEINTRFKTLVEKTWPGDEKVWAKLAVVHDKQVHMANLCVVGGFAVNGVAALHSDLVVKDLFPEYHQLWPNKFHNVTNGITPRRWIKQCNPALAALLDKSLQKEWANDLDQLINLEKFADDAKFRDQYREIKQANKVRLAEFVKVRTGIEINPQAIFDIQIKRLHEYKRQHLNLLHILALYKEIRENPQADRVPRVFLFGAKAAPGYYLAKNIIFAINKVADVINNDPLVGDKLKVVFLPDYCVSAAEKLIPAADISEQISTAGKEASGTGNMKLALNGALTVGTLDGANVEIAEKVGEENIFIFGHTVEQVKAILAKGYDPVKWRKKDKVLDAVLKELESGKYSDGDKHAFDQMLHSIGKQGGDPYLVMADFAAYVEAQKQVDVLYRDQEAWTRAAILNTARCGMFSSDRSIRDYQARIWQAKR 1qm5 A 2.0 BS06 GLC A 1 G114 L115 H345 N449 E637 G640 G114 L115 H345 N449 E637 G640 H345 K533 R534 K539 T641 K645 H345 K533 R534 K539 T641 K645 2.4.1.1 0004645,0005737,0005829,0005975,0005980,0008184,0016757,0030170,0030980,0031220,0042803 remove_due_to_license_issue P00490 10469642 998 SQPIFNDKQFQEALSRQWQRYGLNSAAEMTPRQWWLAVSEALAEMLRAQPFAKPVANQRHVNYISMEFLIGRLTGNNLLNLGWYQDVQDSLKAYDINLTDLLEEEIDPALGNGGLGRLAACFLDSMATVGQSATGYGLNYQYGLFRQSFVDGKQVEAPDDWHRSNYPWFRHNEALDVQVGIGGKVTKDGRWEPEFTITGQAWDLPVVGYRNGVAQPLRLWQATHAHPFDLTKFNDGDFLRAEQQGINAEKLTKVLYPNDNHTAGKKLRLMQQYFQCACSVADILRRHHLAGRKLHELADYEVIQLNDTHPTIAIPELLRVLIDEHQMSWDDAWAITSKTFAYTNHTLMPEALERWDVKLVKGLLPRHMQIINEINTRFKTLVEKTWPGDEKVWAKLAVVHDKQVHMANLCVVGGFAVNGVAALHSDLVVKDLFPEYHQLWPNKFHNVTNGITPRRWIKQCNPALAALLDKSLQKEWANDLDQLINLEKFADDAKFRDQYREIKQANKVRLAEFVKVRTGIEINPQAIFDIQIKRLHEYKRQHLNLLHILALYKEIRENPQADRVPRVFLFGAKAAPGYYLAKNIIFAINKVADVINNDPLVGDKLKVVFLPDYCVSAAEKLIPAADISEQISTAGKEASGTGNMKLALNGALTVGTLDGANVEIAEKVGEENIFIFGHTVEQVKAILAKGYDPVKWRKKDKVLDAVLKELESGKYSDGDKHAFDQMLHSIGKQGGDPYLVMADFAAYVEAQKQVDVLYRDQEAWTRAAILNTARCGMFSSDRSIRDYQARIWQAKR 1qp0 A 2.9 BS01 dna M 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S12 T14 T15 R24 V26 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 10438625 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1qp4 A 3.0 BS01 dna M 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S12 T14 T15 R24 V26 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 10438625 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1qp7 A 2.9 BS01 dna M 0 S14 T16 T17 R26 V28 A29 T32 L54 S12 T14 T15 R24 V26 A27 T30 L52 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 10438625 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLAVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1qp9 A 2.8 BS01 dna E 0 R55 K56 N58 R70 K71 R1 K2 N4 R16 K17 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 1 ~ 20 RKRNRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTLSK 1qp9 A 2.8 BS02 dna F 0 R55 R57 K71 K73 R1 R3 K17 K19 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 1 ~ 20 RKRNRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTLSK 1qp9 B 2.8 BS01 dna E 0 R57 N58 R59 K71 W100 R2 N3 R4 K16 W45 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 1 ~ 20 KRNRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTLS 1qp9 B 2.8 BS02 dna F 0 K56 R57 R59 R68 K71 K73 K1 R2 R4 R13 K16 K18 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 1 ~ 20 KRNRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTLS 1qp9 C 2.8 BS01 dna G 0 R59 K71 R2 K14 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 1 ~ 20 NRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTL 1qp9 C 2.8 BS02 dna H 0 R68 K71 K73 R11 K14 K16 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 3 ~ 19 NRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTL 1qp9 D 2.8 BS01 dna G 0 R57 N58 R59 K71 R3 N4 R5 K17 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 1 ~ 20 RKRNRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTLS 1qp9 D 2.8 BS02 dna H 0 K56 R57 R59 P61 K71 V72 K73 K2 R3 R5 P7 K17 V18 K19 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P0CS82 11024163 3 ~ 19 RKRNRIPLGCTICRKRKVKCDKLRPHCQQCTKTGVAHLCHYMEQTWAEEAEKELLKDNELKKLRERVKSLEKTLS 1qpb A 2.4 BS03 PYM A 1 Y157 H225 D226 Y156 H224 D225 L25 G27 D28 F29 N30 E51 T73 H114 H115 L117 G118 A169 T266 N293 T388 G413 I415 D444 N471 G473 Y474 I476 E477 I480 V542 L24 G26 D27 F28 N29 E50 T72 H113 H114 L116 G117 A168 T265 N292 T387 G412 I414 D443 N470 G472 Y473 I475 E476 I479 V541 4.1.1.-,4.1.1.43,4.1.1.72,4.1.1.74 0000287,0000949,0000955,0003824,0004737,0005515,0005634,0005737,0005829,0006090,0006559,0006569,0009083,0016831,0019655,0030976,0046872,0047433,0047434,0050177 Kd=44mM remove_due_to_license_issue P06169 10651824 602 SEITLGKYLFERLKQVNVNTVFGLPGDFNLSLLDKIYEVEGMRWAGNANELNAAYAADGYARIKGMSCIITTFGVGELSALNGIAGSYAEHVGVLHVVGVPSISAQAKQLLLHHTLGNGDFTVFHRMSANISETTAMITDIATAPAEIDRCIRTTYVTQRPVYLGLPANLVDLNVPAKLLQTPIDMSLKPNDAESEKEVIDTILVLIKDAKNPVILADACCSRHDVKAETKKLIDLTQFPAFVTPMGKGSIDEQHPRYGGVYVGTLSKPEVKEAVESADLILSVGALLSDFNTGSFSYSYKTKNIVEFHSDHMKIRNATFPGVQMKFVLQKLLTAIADAAKGYKPVAVPARTPANAAVPASTPLKQEWMWNQLGNFLQEGDVVIAETGTSAFGINQTTFPNNTYGISQVLWGSIGFTTGATLGAAFAAEEIDPKKRVILFIGDGSLQLTVQEISTMIRWGLKPYLFVLNNDGYTIEKLIHGPKAQYNEIQGWDHLSLLPTFGAKDYETHRVATTGEWDKLTQDKSFNDNSKIRMIEVMLPVFDAPQNLVEQAKLT 1qpb B 2.4 BS04 PYM B 1 D28 H115 D27 H114 L25 G27 D28 F29 N30 E51 T73 H114 H115 L117 G118 A169 T266 N293 T388 G413 I415 D444 N471 G473 Y474 I476 E477 I480 V542 L24 G26 D27 F28 N29 E50 T72 H113 H114 L116 G117 A168 T265 N292 T387 G412 I414 D443 N470 G472 Y473 I475 E476 I479 V541 4.1.1.-,4.1.1.43,4.1.1.72,4.1.1.74 0000287,0000949,0000955,0003824,0004737,0005515,0005634,0005737,0005829,0006090,0006559,0006569,0009083,0016831,0019655,0030976,0046872,0047433,0047434,0050177 Kd=44mM remove_due_to_license_issue P06169 10651824 602 SEITLGKYLFERLKQVNVNTVFGLPGDFNLSLLDKIYEVEGMRWAGNANELNAAYAADGYARIKGMSCIITTFGVGELSALNGIAGSYAEHVGVLHVVGVPSISAQAKQLLLHHTLGNGDFTVFHRMSANISETTAMITDIATAPAEIDRCIRTTYVTQRPVYLGLPANLVDLNVPAKLLQTPIDMSLKPNDAESEKEVIDTILVLIKDAKNPVILADACCSRHDVKAETKKLIDLTQFPAFVTPMGKGSIDEQHPRYGGVYVGTLSKPEVKEAVESADLILSVGALLSDFNTGSFSYSYKTKNIVEFHSDHMKIRNATFPGVQMKFVLQKLLTAIADAAKGYKPVAVPARTPANAAVPASTPLKQEWMWNQLGNFLQEGDVVIAETGTSAFGINQTTFPNNTYGISQVLWGSIGFTTGATLGAAFAAEEIDPKKRVILFIGDGSLQLTVQEISTMIRWGLKPYLFVLNNDGYTIEKLIHGPKAQYNEIQGWDHLSLLPTFGAKDYETHRVATTGEWDKLTQDKSFNDNSKIRMIEVMLPVFDAPQNLVEQAKLT 1qpe A 2.0 BS01 PP2 A 1 A271 K273 E288 T316 M319 L371 A41 K43 E58 T86 M89 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=20nM remove_due_to_license_issue P06239 10404594 1904 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 1qpf D 2.5 BS01 858 D 1 Y226 F236 D237 F246 V255 W259 Y282 F299 Y26 F36 D37 F46 V55 W59 Y82 F99 Y226 F236 D237 I256 Y282 F299 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 ic50=27nM remove_due_to_license_issue P62942 10425089 308 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1qpl A 2.9 BS01 587 A 1 Y26 F36 D37 F46 V55 I56 W59 Y82 F99 Y26 F36 D37 F46 V55 I56 W59 Y82 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 remove_due_to_license_issue P62942 10425089 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1qpl C 2.9 BS01 587 C 1 Y226 D237 F246 E254 V255 I256 W259 Y282 Y26 D37 F46 E54 V55 I56 W59 Y82 Y226 F236 D237 I256 Y282 F299 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006357,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,0140839,0140840,1902991,1990000,1990425 remove_due_to_license_issue P62942 10425089 308 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1qpz A 2.5 BS01 dna M 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S13 T15 T16 R25 V27 A28 T31 L53 K54 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 10438625 699 ~ 715 ATIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1qq9 A 1.53 BS04 MET A 1 H85 D97 E131 E132 D160 R202 F219 Y246 H247 H85 D97 E131 E132 D160 R202 F219 Y246 H247 N77 D97 E131 E132 D160 N77 D97 E131 E132 D160 3.4.11.24 0004177,0006508,0008235 Ki=8.7mM remove_due_to_license_issue P80561 10771423 903 APDIPLANVKAHLTQLSTIAANNGGNRAHGRPGYKASVDYVKAKLDAAGYTTTLQQFTSGGATGYNLIANWPGGDPNKVLMAGAHLDSVSSGAGINDNGSGSAAVLETALAVSRAGYQPDKHLRFAWWGAEELGLIGSKFYVNNLPSADRSKLAGYLNFDMIGSPNPGYFVYDDDPVIEKTFKNYFAGLNVPTEIETEGDGRSDHAPFKNVGVPVGGLFTGAGYTKSAAQAQKWGGTAGQAFDRCYHSSCDSLSNINDTALDRNSDAAAHAIWTLSS 1qqa A 3.0 BS01 dna M 0 S14 T16 T17 R26 V28 A29 T32 L54 A55 S12 T14 T15 R24 V26 A27 T30 L52 A53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 10438625 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLAVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1qqb A 2.7 BS01 dna M 0 S14 T16 T17 R26 V28 A29 T32 L54 A55 S12 T14 T15 R24 V26 A27 T30 L52 A53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 10438625 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLAVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1qs4 A 2.1 BS02 100 A 1 T66 I151 E152 N155 K156 K159 T11 I92 E93 N96 K97 K100 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=2.3uM remove_due_to_license_issue P12497 10557269 1004 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACEWGGIKQEFGPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGIGGYSAGERIVDIIATDIQ 1qti A 2.5 BS01 GNT A 1 W84 G117 G118 Y121 E199 S200 F288 F290 F331 H440 W81 G114 G115 Y118 E196 S197 F285 F287 F328 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue IC50=1069nM, Ki=1.9e+2nM P04058 11119642 600 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1qtq A 2.25 BS01 rna B 0 Q13 E34 T68 N69 I129 R130 R133 T135 L136 T137 G168 P181 F182 I183 V189 R192 K194 M210 Y211 F233 Q234 D235 R238 I313 T316 K317 Q318 N320 T321 E323 S326 R341 P369 Q399 K401 R402 R410 R412 N413 V455 Q517 E519 R520 R545 Q6 E27 T61 N62 I122 R123 R126 T128 L129 T130 G161 P174 F175 I176 V182 R185 K187 M203 Y204 F226 Q227 D228 R231 I306 T309 K310 Q311 N313 T314 E316 S319 R334 P362 Q392 K394 R395 R403 R405 N406 V437 Q499 E501 R502 R527 6.1.1.18 0000166,0004812,0004819,0005524,0005737,0005829,0006412,0006418,0006424,0006425,0043039 remove_due_to_license_issue P00962 9562563 902 ~ 976 TNFIRQIIDEDLASGKHTTVHTRFPPEPNGYLHIGHAKSICLNFGIAQDYKGQCNLRFDDTNPVKEDIEYVESIKNDVEWLGFHWSGNVRYSSDYFDQLHAYAIELINKGLAYVDELTPEQIREYRGTLTQPGKNSPYRDRSVEENLALFEKMRAGGFEEGKACLRAKIDMASPFIVMRDPVLYRIKFAEHHQTGNKWCIYPMYDFTHCISDALEGITHSLCTLEFQDNRRLYDWVLDNITIPVHPRQYEFSRLNLEYTVMSKRKLNLLVTDKHVEGWDDPRMPTISGLRRRGYTAASIREFCKRIGVTKQDNTIEMASLESCIREDLNENAPRAMAVIDPVKLVIENYQGEGEMVTMPNHPNKPEMGSRQVPFSGEIWIDRADFREEANKQYKRLVLGKEVRLRNAYVIKAERVEKDAEGNITTIFCTYDADTLGVIHWVSAAHALPVEIRLYDRLFSVPNPGAADDFLSVINPESLVIKQGFAEPSLKDAVAGKAFQFEREGYFCLDSRHSTAEKPVFNRTVGLRDT 1qvt A 2.89 BS01 PRL A 1 W61 T89 Y93 W60 T88 Y92 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 15257299 311 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKCKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 1qvu A 2.96 BS02 PRL A 1 E58 T89 E90 Y93 Y103 E57 T88 E89 Y92 Y102 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N4 15257299 196 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKKEQIKCKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 1qwu A 2.03 BS02 GUL A 1 H90 D92 W95 D204 F206 R228 H471 D472 Y727 R876 H60 D62 W65 D174 F176 R198 H441 D442 Y697 R846 H90 D92 D204 N341 H471 H60 D62 D174 N311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 remove_due_to_license_issue Q24451 12960159 2003 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDNFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 1qx1 A 1.3 BS02 FMF A 1 H90 D92 W95 D204 F206 R228 W415 H471 D472 Y727 R876 H60 D62 W65 D174 F176 R198 W385 H441 D442 Y697 R846 H90 D92 D204 N341 H471 H60 D62 D174 N311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 remove_due_to_license_issue Q24451 12960159 2003 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDNFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 1qxk A 2.3 BS01 429 A 1 Y20 R24 Y46 D48 F182 A217 G220 R221 R254 G259 Q262 Q266 G283 Y19 R23 Y45 D47 F181 A216 G219 R220 R253 G258 Q261 Q265 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=9uM remove_due_to_license_issue Ki=9000nM, IC50=9000nM P18031 14592481 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 1qxl A 2.25 BS02 FR8 A 1 H17 D19 L56 L62 M155 G184 D185 T269 D296 H14 D16 L53 L59 M152 G181 D182 T266 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=11nM remove_due_to_license_issue P56658 15239652 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELLNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1qxw A 1.67 BS03 M1C A 1 C67 H76 D93 D104 H168 E202 F204 E233 C67 H76 D93 D104 H168 E202 F204 E233 D93 D104 H168 H175 E202 E233 D93 D104 H168 H175 E202 E233 3.4.11.18 0004177,0004239,0006508,0008235,0046872,0070006 ic50=7uM remove_due_to_license_issue P0A078 14998322 3001 MIVKTEEELQALKEIGYICAKVRNTMQAATKPGITTKELDNIAKELFEEYGAISAPIHDENFPGQTCISVNEEVAHGIPSKRVIREGDLVNIDVSALKNGYYADTGISFVVGESDDPMKQKVCDVATMAFENAIAKVKPGTKLSNIGKAVHNTARQNDLKVIKNLTGHGVGLSLHEAPAHVLNYFDPKDKTLLTEGMVLAIEPFISSNASFVTEGKNEWAFETSDKSFVAQIEHTVIVTKDGPILTTKI 1qxy A 1.04 BS04 M2C A 1 P56 E60 H76 D93 D104 H168 L174 H175 E202 E233 P56 E60 H76 D93 D104 H168 L174 H175 E202 E233 D93 D104 H168 H175 E202 E233 D93 D104 H168 H175 E202 E233 3.4.11.18 0004177,0004239,0006508,0008235,0046872,0070006 ic50=16uM remove_due_to_license_issue P0A078 14998322 3001 MIVKTEEELQALKEIGYICAKVRNTMQAATKPGITTKELDNIAKELFEEYGAISAPIHDENFPGQTCISVNEEVAHGIPSKRVIREGDLVNIDVSALKNGYYADTGISFVVGESDDPMKQKVCDVATMAFENAIAKVKPGTKLSNIGKAVHNTARQNDLKVIKNLTGHGVGLSLHEAPAHVLNYFDPKDKTLLTEGMVLAIEPFISSNASFVTEGKNEWAFETSDKSFVAQIEHTVIVTKDGPILTTKI 1qxz A 1.68 BS04 M3C A 1 H79 D97 D108 H178 E204 F206 E235 H76 D93 D104 H175 E202 F204 E233 D97 D108 H171 H178 E204 E235 D93 D104 H168 H175 E202 E233 3.4.11.18 0004177,0004239,0006508,0008235,0046872,0070006 ic50=19uM remove_due_to_license_issue P0A078 14998322 2001 MIVKTEEELQALKEIGYICAKVRNTMQAATKPGITTKELDNIAKELFEEYGAISAPIHDENFPGQTCISVNEEVAHGIPSKRVIREGDLVNIDVSALKNGYYADTGISFVVGESDDPMKQKVCDVATMAFENAIAKVKPGTKLSNIGKAVHNTARQNDLKVIKNLTGHGVGLSLHEAPAHVLNYFDPKDKTLLTEGMVLAIEPFISSNASFVTEGKNEWAFETSDKSFVAQIEHTVIVTKDGPILTTKI 1qy1 A 1.7 BS01 PRZ A 1 L40 F56 F90 A103 L116 Y120 L40 F56 F90 A103 L116 Y120 ? 0036094 Kd=0.3uM remove_due_to_license_issue P11588 14871097 300 EEASSTGRNFNVEKINGEWHTIILASDKREKIEDNGNFRLFLEQIHVLEKSLVLKFHTVRDEECSELSMVADKTEKAGEYSVTYDGFNTFTIPKTDYDNFLMAHLINEKDGETFQLMGLYGREPDLSSDIKERFAQLCEEHGILRENIIDLSNANRC 1qy2 A 1.75 BS01 IPZ A 1 L40 F56 Y120 L40 F56 Y120 ? 0036094 Kd=1.8uM remove_due_to_license_issue P11589 14871097 300 EEASSTGRNFNVEKINGEWHTIILASDKREKIEDNGNFRLFLEQIHVLEKSLVLKFHTVRDEECSELSMVADKTEKAGEYSVTYDGFNTFTIPKTDYDNFLMAHLINEKDGETFQLMGLYGREPDLSSDIKERFAQLCEEHGILRENIIDLSNANRC 1qyg H 1.81 BS01 BCG H 1 D31 W33 V95 Q97 L98 G99 D31 W33 V101 Q103 L104 G105 remove_due_to_license_issue 15885702 401 EVTLQESGGGLVQPGGSMKLSCAASGFTFSDAWVDWVRQSPGKGLEWVAEIRNKANNHATKYTESVKGRFTISRDDSKSSVYLQMNSLRAEDTGIYYCTSVPQLGRGFAYWGQGTLVTVSAASTTPPSVYPLAPGSGGAGSMVTLGCLVKGYFPEPVTVTWNSGALSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSQTVTCNVAHPASSTQVDKKIVPK 1qyg L 1.81 BS01 BCG H 1 Y32 H91 F96 Y37 H96 F101 remove_due_to_license_issue 15885702 401 DIVMTQAAPSVPVTPGESVSISCRSSKSLLHSNGYTYLHWFLQRPGQSPQLLIYRVSNLASGVPDRFSGSGSGTAFTLRFSRVEAEDVGVYYCMQHLEYPFTFGSGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPQDITVSWKIDGAERSSGVLNSWTDQDSSDSTYSMSSTLTLTKDEYERHSSYTCEATHKTSTSPITKSFNRGE 1qzg A 1.9 BS01 dna C 0 S58 L59 G61 T62 D64 F88 K90 T111 L122 S123 K124 D125 S54 L55 G57 T58 D60 F84 K86 T107 L118 S119 K120 D121 ? 0000723,0000781,0003677,0043047 remove_due_to_license_issue O13988 14614509 1 ~ 5 VIDSLQLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTN 1qzg B 1.9 BS01 dna D 0 R56 S58 L59 H60 G61 T62 D64 F88 K90 T111 L122 S123 K124 D125 R52 S54 L55 H56 G57 T58 D60 F84 K86 T107 L118 S119 K120 D121 ? 0000723,0000781,0003677,0043047 remove_due_to_license_issue O13988 14614509 1 ~ 5 VIDSLQLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTN 1r0p A 1.8 BS01 KSA A 1 I1084 V1092 A1108 K1110 P1158 Y1159 M1160 M1211 R1227 M1229 Y1230 I35 V43 A55 K57 P105 Y106 M107 M158 R174 M176 Y177 D1204 A1206 R1208 N1209 D1222 A1243 D151 A153 R155 N156 D169 A190 2.7.10.1 0004672,0004713,0005524,0006468 Kd=10nM remove_due_to_license_issue P08581 14559966 0 TVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEFDSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 1r0x A 2.2 BS02 ATP A 1 W401 L409 T460 G461 S462 G463 K464 T465 S466 W12 L20 T54 G55 S56 G57 K58 T59 S60 5.6.1.6 0005524,0016887 Kd=149uM remove_due_to_license_issue P26361 14685259 1 TGIIMENVTAFWEEGFGELLEKSFSHLCLVGNPVLKNINLNIEKGEMLAITGSTGSGKTSLLMLILGELEASEGIIKHSGRVSFCSQFSWIMPGTIKENIIFGVSYDEYRYKSVVKACQLQQDITKFAEQDNTVLGEGGVTLSGGQRARISLARAVYKDADLYLLDSPFGYLDVFTEEQVFESCVCKLMANKTRILVTSKMEHLRKADKILILHQGSSYFYGTFSELQSLRPDFSSKLMGYDTFDQFTEERRSSILTETLRRFS 1r10 A 3.0 BS02 ATP A 1 W401 L409 F430 G461 S462 G463 K464 T465 S466 W11 L19 F24 G55 S56 G57 K58 T59 S60 5.6.1.6 0005524,0016887 remove_due_to_license_issue P26361 14685259 1 GIIMENVTAFWEEGFGELLEKVSFSHLCLVGNPVLKNINLNIEKGEMLAITGSTGSGKTSLLMLILGELEASEGIIKHSGRVSFCSQFSWIMPGTIKENIIFGVSYDEYRYKSVVKACQLQQDITKFAEQDNTVLGEGGVTLSGGQRARISLARAVYKDADLYLLDSPFGYLDVFTEEQVFESCVCKLMANKTRILVTSKMEHLRKADKILILHQGSSYFYGTFSELQSLRPDFSSKLMGYDTFDQFTEERRSSILTETLRRFS 1r1h A 1.95 BS02 BIR A 1 F106 N542 A543 M579 V580 H583 E584 H587 E646 F689 V692 W693 H711 R717 F53 N489 A490 M526 V527 H530 E531 H534 E593 F636 V639 W640 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 Ki=1.2nM remove_due_to_license_issue P08473 14747736 2001 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 1r1i A 2.6 BS02 TI1 A 1 F106 N542 A543 M579 V580 H583 E584 H587 E646 W693 H711 R717 F53 N489 A490 M526 V527 H530 E531 H534 E593 W640 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 remove_due_to_license_issue P08473 14747736 2001 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 1r1j A 2.35 BS02 OIR A 1 F106 N542 A543 F544 M579 V580 H583 E584 H587 E646 W693 H711 R717 F53 N489 A490 F491 M526 V527 H530 E531 H534 E593 W640 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 Ki=2.3nM remove_due_to_license_issue P08473 14747736 2001 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 1r4w A 2.5 BS01 GSH A 1 S16 Y18 F181 G182 L183 F198 G199 S200 D201 S15 Y17 F180 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005737,0005739,0005759,0005777,0006749,0016491,0016740,0030855,0043231,0098869 Kd=90uM remove_due_to_license_issue P24473 14717589 301 GPAPRVLELFYDVLSPYSWLGFEVLCRYQHLWNIKLKLRPALLAGIMKDSGNQPPAMVPHKGQYILKEIPLLKQLFQVPMSVPKDFFGEHVKKGTVNAMRFLTAVSMEQPEMLEKVSRELWMRIWSRDEDITESQNILSAAEKAGMATAQAQHLLNKISTELVKSKLRETTGAACKYGAFGLPTTVAHVDGKTYMLFGSDRMELLAYLLGEKWMGPVPPTL 1r4w B 2.5 BS01 GSH B 1 S16 Y18 N53 G182 L183 F198 G199 S200 D201 S15 Y17 N52 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005737,0005739,0005759,0005777,0006749,0016491,0016740,0030855,0043231,0098869 Kd=90uM remove_due_to_license_issue P24473 14717589 401 GPAPRVLELFYDVLSPYSWLGFEVLCRYQHLWNIKLKLRPALLAGIMKDSGNQPPAMVPHKGQYILKEIPLLKQLFQVPMSVPKDFFGEHVKKGTVNAMRFLTAVSMEQPEMLEKVSRELWMRIWSRDEDITESQNILSAAEKAGMATAQAQHLLNKISTELVKSKLRETTGAACKYGAFGLPTTVAHVDGKTYMLFGSDRMELLAYLLGEKWMGPVPPTL 1r58 A 1.9 BS03 AO5 A 1 F219 H231 D251 D262 H331 H339 E364 M384 A414 Y444 E459 F110 H122 D142 D153 H222 H230 E255 M275 A305 Y335 E350 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 remove_due_to_license_issue IC50=110nM P50579 15012983 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 1r5g A 2.0 BS03 AO1 A 1 F219 H231 D262 N329 H331 H339 E364 Y444 E459 F110 H122 D153 N220 H222 H230 E255 Y335 E350 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 remove_due_to_license_issue IC50=22nM P50579 15012983 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 1r5h A 2.4 BS03 AO2 A 1 F219 H231 D251 D262 L328 N329 H331 H339 E364 M384 Y444 E459 F110 H122 D142 D153 L219 N220 H222 H230 E255 M275 Y335 E350 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 ic50=0.17uM remove_due_to_license_issue IC50=170nM P50579 15012983 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 1r5n A 2.9 BS01 GDP A 1 V247 D248 G250 K251 S252 T253 K278 N384 K385 D387 E388 S427 Y429 V33 D34 G36 K37 S38 T39 K64 N130 K131 D133 E134 S173 Y175 D248 K251 S252 D34 K37 S38 3.6.5.- 0000288,0003747,0003924,0005525,0006415 remove_due_to_license_issue O74718 15099522 663 TEDATDLQNEVDQELLKDMYGKEHVNIVFIGHVDAGKSTLGGNILFLTGMVDKRTMEKIEREAKRAYFETEHRRFSLLDAPGASQADIGVLVISARRGEFEAGFERGGQTREHAVLARTQGINHLVVVINKMDEPSVQWSEERYKECVDKLSMFLRRVAGYNSKTDVKYMPVSAYTGQNVKDRVDSSVCPWYQGPSLLEYLDSMTHLERKVNAPFIMPIASKYKDLGTILEGKIEAGSIKKNSNVLVMPINQTLEVTAIYDEADEEISSSICGDQVRLRVRGDDSDVQTGYVLTSTKNPVHATTRFIAQIAILELPSILTTGYSCVMHIHTAVEEVSFAKLLHKLDKTNRKSKKPPMFATKGMKIIAELETQTPVCMERFEDYQYMGRFTLRDQGTTVAVGKVVKILD 1r5y A 1.2 BS02 DQU A 1 D102 Y106 D156 C158 G229 M260 D92 Y96 D135 C137 G208 M239 D102 D280 C318 C320 C323 H349 D92 D259 C297 C299 C302 H328 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=0.35uM remove_due_to_license_issue P28720 15050823 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMLSLTKQSEEGVTFMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1r6g A 3.0 BS01 442 A 1 F272 I276 A279 R282 M313 R320 L330 N331 G345 L346 H435 R438 F439 M442 F455 F51 I55 A58 R61 M92 R99 L109 N110 G124 L125 H214 R217 F218 M221 F234 ? 0003677,0004879,0006355 remove_due_to_license_issue P10828 15177471 500 ELQKSIGKKPEPTDEEWELIKTVTEAHVATNARKFLPEDIGQVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 1r6n A 2.4 BS01 434 A 1 H32 W33 L94 Q95 S98 Y99 E100 H32 W33 L94 Q95 S98 Y99 E100 ? 0006275,0006355,0016032 Kd=40nM remove_due_to_license_issue P04015 14634007 1111 HEAIAKRLDACQDQLLELYEENSIDIHKHIMHWKCIRLESVLLHKAKQMGLSHIGLQVVPPLTVSETKGHNAIEMQMHLESLAKTQYGVEPWTLQDTSYEMWLTPPKRCFKKQGNTVEVKFDGCEDNVMEYVVWTHIYLQDNDSWVKVTSSVDAKGIYYTCGQFKTYYVNFNKEAQKYGSTNHWEVCYGSTVICSP 1r6n A 2.4 BS02 434 A 2 W33 T63 V64 T67 K68 N71 W33 T63 V64 T67 K68 N71 ? 0006275,0006355,0016032 Kd=40nM remove_due_to_license_issue P04015 14634007 1112 HEAIAKRLDACQDQLLELYEENSIDIHKHIMHWKCIRLESVLLHKAKQMGLSHIGLQVVPPLTVSETKGHNAIEMQMHLESLAKTQYGVEPWTLQDTSYEMWLTPPKRCFKKQGNTVEVKFDGCEDNVMEYVVWTHIYLQDNDSWVKVTSSVDAKGIYYTCGQFKTYYVNFNKEAQKYGSTNHWEVCYGSTVICSP 1r78 A 2.0 BS01 FMD A 1 I10 G11 E12 V18 A31 F80 F82 L83 Q131 L134 D145 I10 G11 E12 V18 A31 F71 F73 L74 Q122 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T140 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=3nM remove_due_to_license_issue IC50=3nM P24941 15012993 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1r8d A 2.7 BS01 dna C 0 V5 K6 R17 H20 Y38 R39 V5 K6 R17 H20 Y38 R39 ? 0003677,0003700,0006355 remove_due_to_license_issue P71039 14985361 -14 ~ 13 MKYQVKQVAEISGVSIRTLHHYDNIELLNPSALTDAGYRLYSDADLERLQQILFFKEIGFRLDEIKEMLDHPNFDRKAALQSQKEILMKKKQRMDEMIQTIDRTLLSVD 1r8d A 2.7 BS02 dna D 0 S15 R17 T18 H21 Y22 A36 Y38 R61 L62 S15 R17 T18 H21 Y22 A36 Y38 R61 L62 ? 0003677,0003700,0006355 remove_due_to_license_issue P71039 14985361 -14 ~ 13 MKYQVKQVAEISGVSIRTLHHYDNIELLNPSALTDAGYRLYSDADLERLQQILFFKEIGFRLDEIKEMLDHPNFDRKAALQSQKEILMKKKQRMDEMIQTIDRTLLSVD 1r8d B 2.7 BS01 dna C 0 S15 R17 T18 H21 Y22 A36 Y38 K56 R61 L62 S15 R17 T18 H21 Y22 A36 Y38 K56 R61 L62 ? 0003677,0003700,0006355 remove_due_to_license_issue P71039 14985361 -14 ~ 13 MKYQVKQVAEISGVSIRTLHHYDNIELLNPSALTDAGYRLYSDADLERLQQILFFKEIGFRLDEIKEMLDHPNFDRKAALQSQKEILMKKKQRMDEMIQTIDRTLLS 1r8d B 2.7 BS02 dna D 0 Q4 V5 K6 R17 H20 Y38 R39 Q4 V5 K6 R17 H20 Y38 R39 ? 0003677,0003700,0006355 remove_due_to_license_issue P71039 14985361 -14 ~ 13 MKYQVKQVAEISGVSIRTLHHYDNIELLNPSALTDAGYRLYSDADLERLQQILFFKEIGFRLDEIKEMLDHPNFDRKAALQSQKEILMKKKQRMDEMIQTIDRTLLS 1r8e A 2.4 BS01 dna B 0 S7 I8 G9 R23 Y42 R43 S5 I6 G7 R21 Y40 R41 ? 0003677,0003700,0006355 remove_due_to_license_issue P39075 14985361 -12 ~ 12 ESYYSIGEVSKLANVSIKALRYYDKIDLFKPAYVDPDTSYRYYTDSQLIHLDLIKSLKYIGTPLEEMKKAQDLEMEELFAFYTEQERQIREKLDFLSALEQTISLVKKRMKRQMEYPALGEVFVLDEEEIRIIQTEAEGIGPENVLNASYSKLKKFIESADGFTNNSYGATFSFQPYTSIDEMTYRHIFTPVLTNKQISSITPDMEITTIPKGRYACIAYNFSPEHYFLNLQKLIKYIADRQLTVVSDVYELIIPIHYSPKKQEEYRVEMKIRIA 1rbo L 2.3 BS01 CAP L 1 K175 D203 R295 H327 K334 L335 S379 G380 G403 K167 D195 R287 H319 K326 L327 S371 G372 G395 D203 E204 H294 H327 K334 D195 E196 H286 H319 K326 4.1.1.39 0000287,0004497,0009507,0009853,0015977,0015979,0016829,0016984,0019253,0046872 Kd=0.19pM remove_due_to_license_issue P00875 8955130 476 ASVGFKAGVKDYKLTYYTPEYETLDTDILAAFRVSPQPGVPPEEAGAAVAAESSTGTWTTVWTDGLTNLDRYKGRCYHIEPVAGEENQYICYVAYPLDLFEEGSVTNMFTSIVGNVFGFKALRALRLEDLRIPVAYVKTFQGPPHGIQVERDKLNKYGRPLLGCTIKPKLGLSAKNYGRAVYECLRGGLDFTKDDENVNSQPFMRWRDRFLFCAEALYKAQAETGEIKGHYLNATAGTCEDMMKRAVFARELGVPIVMHDYLTGGFTANTTLSHYCRDNGLLLHIHRAMHAVIDRQKNHGMHFRVLAKALRLSGGDHIHSGTVVGKLEGERDITLGFVDLLRDDYTEKDRSRGIYFTQSWVSTPGVLPVASGGIHVWHMPALTEIFGDDSVLQFGGGTLGHPWGNAPGAVANRVALEACVQARNEGRDLAREGNTIIREATKWSPELAAACEVWKEIKFEFPAMDTV 1rbp A 2.0 BS01 RTL A 1 L35 F36 A55 K58 V61 Q98 C174 L35 F36 A55 K58 V61 Q98 C174 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 Kd=0.19uM remove_due_to_license_issue P02753 2217163 183 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYC 1rd4 A 2.4 BS01 L08 A 1 F153 Y166 V233 I235 I255 Y257 I259 E284 F285 V286 K287 L298 E301 K305 F26 Y39 V106 I108 I128 Y130 I132 E157 F158 V159 K160 L171 E174 K178 ? Kd=18.3nM remove_due_to_license_issue Kd=18nM P20701 14992576 328 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKRKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVIEG 1rdi 1 1.8 BS01 MFU 1 1 E190 N192 E198 N210 E76 N78 E84 N96 ? Ki=8.8mM remove_due_to_license_issue P08661 8557671 1 KYFMSSVRRMPLNRAKALCSELQGTVATPRNAEENRAIQNVAKDVAFLGITDQRTENVFEDLTGNRVRYTNWNEGEPNNVGSGENCVVLLTNGKWNDVPCSDSFLVVCEFS 1rdj 1 1.8 BS01 MFB 1 1 E190 N192 E198 N210 E76 N78 E84 N96 ? Ki=21.7mM remove_due_to_license_issue P08661 8557671 1 KYFMSSVRRMPLNRAKALCSELQGTVATPRNAEENRAIQNVAKDVAFLGITDQRTENVFEDLTGNRVRYTNWNEGEPNNVGSGENCVVLLTNGKWNDVPCSDSFLVVCEFS 1rdl 1 1.7 BS01 MMA 1 1 E190 N192 E198 N210 E76 N78 E84 N96 ? Ki=5.7mM remove_due_to_license_issue P08661 8557671 1 KYFMSSVRRMPLNRAKALCSELQGTVATPRNAEENRAIQNVAKDVAFLGITDQRTENVFEDLTGNRVRYTNWNEGEPNNVGSGENCVVLLTNGKWNDVPCSDSFLVVCEFS 1rdt A 2.4 BS02 L79 A 1 I268 A272 Q275 W305 L309 F313 R316 L326 A327 V342 I345 I23 A27 Q30 W60 L64 F68 R71 L81 A82 V97 I100 ? 0003677,0003707,0005634,0006355,0008270 Ki=6nM remove_due_to_license_issue P19793 15056000 463 EDMPVERILEAELAVEPDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLE 1re1 A 2.5 BS01 NA3 A 1 R179 S236 H237 Q283 A284 C285 R31 S87 H88 Q128 A129 C130 T177 S178 H237 G238 C285 R286 T29 S30 H88 G89 C130 R131 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=6000nM P42574 15115390 501 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 1re1 B 2.5 BS01 NA3 A 1 Y338 S339 W340 R341 Y19 S20 W21 R22 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=6000nM P42574 15115390 501 KIPVEADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFY 1re8 A 2.1 BS01 BD2 A 1 G50 T51 G52 F54 V57 A70 K72 L74 E91 M120 E121 E127 E170 L173 T183 D184 G186 G39 T40 G41 F43 V46 A59 K61 L63 E80 M109 E110 E116 E159 L162 T172 D173 G175 D166 K168 E170 N171 D184 T201 D155 K157 E159 N160 D173 T190 2.7.11.11 0000122,0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,0141156,1904262,1904539,1990044,2000810 Ki=0.3nM remove_due_to_license_issue P05132 14705934 351 QESVKEFLAKAKEDFLKKWETPSQNTAQLDQFDRIKTLGTGSFGRVMLVKHKESGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 1rej A 2.2 BS01 B1L A 1 G50 T51 G52 S53 F54 G55 R56 V57 A70 K72 L74 E121 Y122 E127 E170 L173 T183 D184 F327 G35 T36 G37 S38 F39 G40 R41 V42 A55 K57 L59 E106 Y107 E112 E155 L158 T168 D169 F312 D166 K168 E170 N171 D184 T201 D151 K153 E155 N156 D169 T186 2.7.11.11 0000122,0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,0141156,1904262,1904539,1990044,2000810 Ki=5nM remove_due_to_license_issue P05132 14705934 351 KEFLAKAKEDFLKKWETPSQNTAQLDQFDRIKTLGTGSFGRVMLVKHKESGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 1rek A 2.3 BS01 B8L A 1 G50 T51 G52 F54 V57 A70 K72 L74 E91 E121 Y122 V123 E127 E170 L173 T183 D184 G186 G38 T39 G40 F42 V45 A58 K60 L62 E79 E109 Y110 V111 E115 E158 L161 T171 D172 G174 D166 K168 E170 N171 D184 T201 D154 K156 E158 N159 D172 T189 2.7.11.11 0000122,0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,0141156,1904262,1904539,1990044,2000810 Ki=200nM remove_due_to_license_issue P05132 14705934 351 ESVKEFLAKAKEDFLKKWETPSQNTAQLDQFDRIKTLGTGSFGRVMLVKHKESGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 1rev A 2.6 BS01 TB9 A 1 L100 K101 V106 Y181 Y188 W229 L234 H235 L97 K98 V103 Y178 Y185 W226 L231 H232 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 8535785 999 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAH 1rgk A 1.87 BS01 2AM A 1 N36 Y38 H40 E58 G74 R77 H92 N36 Y38 H40 E58 G74 R77 H92 Y38 H40 E58 D76 R77 T91 H92 F100 Y38 H40 E58 D76 R77 T91 H92 F100 4.6.1.24 0001411,0003723,0004519,0004521,0004540,0008150,0016829,0030428,0046589 Kd=49.1uM remove_due_to_license_issue P00651 1350642 105 ACDYTCGSNCYSSSDVSTAQAAGYKLHEDGETVGSNSYPHKYNNYQGFDFSVSSPYYEWPILSSGDVYSGGSPGADRVVFNENNQLAGVITHTGASGNNFVECT 1rgl A 2.0 BS01 2GP A 1 N36 Y38 H40 E58 R77 H92 G97 N36 Y38 H40 E58 R77 H92 G97 Y38 H40 E58 D76 R77 T91 H92 F100 Y38 H40 E58 D76 R77 T91 H92 F100 4.6.1.24 0001411,0003723,0004519,0004521,0004540,0008150,0016829,0030428,0046589 Kd=37uM remove_due_to_license_issue P00651 1350642 105 ACDYTCGSNCYSSSDVSTAQAAGYKLHEDGETVGSNSYPHKYNNYQGFDFSVSSPYYEWPILSSGDVYSGGSPGADRVVFNENNQLAGVITHTGASGNNFVECT 1rhm A 2.5 BS01 NA4 A 1 R179 S236 H237 C285 R31 S87 H88 C130 T177 S178 G238 C285 T29 S30 G89 C130 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=1735nM P42574 15115390 501 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 1rhm B 2.5 BS01 NA4 A 1 Y338 S339 W340 R341 Y19 S20 W21 R22 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=1735nM P42574 15115390 501 KIPVEADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFY 1rhq A 3.0 BS01 0ZZ A 1 R179 S236 H237 G238 E239 F244 A284 C285 R31 S87 H88 G89 E90 F95 A129 C130 T177 S178 H237 G238 C285 R286 T29 S30 H88 G89 C130 R131 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue P42574 15115390 551 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 1rhq B 3.0 BS01 0ZZ A 1 Y338 S339 W340 R341 S381A F381B Y19 S20 W21 R22 S64 F65 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue P42574 15115390 551 KIPVEADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFY 1rhr A 3.0 BS01 CNE A 1 M176 R179 H237 G238 E239 C285 G287 M28 R31 H88 G89 E90 C130 G132 T177 S178 H237 G238 C285 R286 T29 S30 H88 G89 C130 R131 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=8nM P42574 15115390 501 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 1rhr B 3.0 BS01 CNE A 1 S339 W340 R341 W348 F381B S381C F381H S20 W21 R22 W29 F65 S66 F71 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=8nM P42574 15115390 501 KIPVEADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFY 1rhu A 2.51 BS01 3CY A 1 R179 H237 E239 C285 T288 R31 H88 E90 C130 T133 T177 S178 H237 G238 C285 R286 T29 S30 H88 G89 C130 R131 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=3nM P42574 15115390 501 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 1rhu B 2.51 BS01 3CY A 1 Y338 S339 W340 R341 N342 S343 S381A F381B F381H Y19 S20 W21 R22 N23 S24 S64 F65 F71 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue IC50=3nM P42574 15115390 501 KIPVEADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFY 1rin A 2.6 BS01 MAN A 1 A80 D81 G99 F123 A80 D81 G99 F123 ? 0030246 remove_due_to_license_issue P02867 8486683 250 TETTSFLITKFSPDQQNLIFQGDGYTTKEKLTLTKAVKNTVGRALYSSPIHIWDRETGNVANFVTSFTFVINAPNSYNVADGFTFFIAPVDTKPQTGGGYLGVFNSAEYDKTTETVAVEFDTFYNAAWDPSNRDRHIGIDVNSIKSVNTKSWKLQNGEEANVVIAFNAATNVLTVSLTYP 1rin B 2.6 BS01 MAN A 1 G216 A217 E218 G29 A30 E31 ? 0030246 remove_due_to_license_issue P02867 8486683 250 VTSYTLSDVVSLKDVVPEWVRIGFSATTGAEYAAHEVLSWSFHSELS 1riw B 2.04 BS03 OSC C 1 H79 Y83 W86 L132 E182 H43 Y47 W50 L96 E146 H79 D135 H43 D99 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=28nM P00734 15137772 1001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKET 1riw C 2.04 BS02 OSC C 1 D229 A230 S235 S256 W257 G258 G260 R263 D45 A46 S51 S72 W73 G74 G76 R79 E232 G233 D234 S235 G236 E48 G49 D50 S51 G52 3.4.21.5 0004252,0006508 ic50=28nM remove_due_to_license_issue IC50=28nM P00734 15137772 1001 GQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 1rjk A 1.99 BS02 VDZ A 1 Y143 S233 R270 S271 S274 W282 C284 H301 H393 Y21 S52 R89 S90 S93 W101 C103 H120 H212 ? 0003677,0004879,0006355 remove_due_to_license_issue Ki=0.1nM P13053 15065852 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 1rkj A -1.00 BS01 rna B 0 F17 R49 T52 F56 Y58 K89 R91 D92 K94 K95 L103 K105 R127 V129 K136 I138 Y140 F17 R49 T52 F56 Y58 K89 R91 D92 K94 K95 L103 K105 R127 V129 K136 I138 Y140 ? 0003676,0003723 remove_due_to_license_issue P08199 15033352 1 ~ 21 GSHMVEGSESTTPFNLFIGNLNPNKSVAELKVAISELFAKNDLAVVDVRTGTNRKFGYVDFESAEDLEKALELTGLKVFGNEIKLEKPKGRDSKKVRAARTLLAKNLSFNITEDELKEVFEDALEIRLVSQDGKSKGIAYIEFKSEADAEKNLEEKQGAEIDGRSVSLYYTGEKG 1rm8 A 1.8 BS05 BAT A 1 G204 F205 L206 A207 V243 H246 E247 H250 H256 P266 F267 Y268 G81 F82 L83 A84 V120 H123 E124 H127 H133 P143 F144 Y145 H246 E247 H250 H256 H123 E124 H127 H133 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P51512 14741217 800 GQKWQHKHITYSIKNVTPKVGDPETRKAIRRAFDVWQNVTPLTFEEVPYSELENGKRDVDITIIFASGFHGDSSPFDGEGGFLAHAYFPGPGIGGDTHFDSDEPWTLGNPNHDGNDLFLVAVHELGHALGLEHSNDPTAIMAPFYQYMETDNFKLPNDDLQGIQKIYGP 1rmz A 1.34 BS06 NGH A 1 I180 L181 A182 T215 H218 E219 H222 H228 P238 T239 Y240 I76 L77 A78 T111 H114 E115 H118 H124 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=4.3nM P39900 15809432 269 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 1rne A 2.4 BS01 C60 A 1 Q13 D32 G34 Y75 S76 T77 F117 D215 G217 A218 S219 Y220 S222 A300 Q15 D34 G36 Y79 S80 T81 F120 D215 G217 A218 S219 Y220 S222 A303 D32 S35 N37 W39 Y75 D215 A218 D34 S37 N39 W41 Y79 D215 A218 3.4.23.15 0004190,0006508 ic50=2nM remove_due_to_license_issue IC50=0.830000nM, Ki=0.7nM P00797 1807356 350 NTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 1rnm E 2.0 BS01 C5P E 1 H12 V43 N44 T45 F120 H12 V43 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue P61823 200 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1rnt A 1.9 BS01 2GP A 1 Y38 H40 Y42 N43 N44 Y45 E46 E58 N98 F100 Y38 H40 Y42 N43 N44 Y45 E46 E58 N98 F100 Y38 H40 E58 D76 R77 T91 H92 F100 Y38 H40 E58 D76 R77 T91 H92 F100 4.6.1.24 0001411,0003723,0004519,0004521,0004540,0008150,0016829,0030428,0046589 Kd=6.5uM remove_due_to_license_issue P00651 105 ACDYTCGSNCYSSSDVSTAQAAGYKLHEDGETVGSNSYPHKYNNYEGFDFSVSSPYYEWPILSSGDVYSGGSPGADRVVFNENNQLAGVITHTGASGNNFVECT 1ro6 A 2.0 BS03 ROL A 1 Y233 H234 T407 I410 F414 Q443 F446 Y82 H83 T256 I259 F263 Q292 F295 3.1.4.53 0004114,0007165,0008081 Ki~375nM remove_due_to_license_issue Q07343 15003452 601 SISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPQAPAPPLDEQ 1ro7 A 1.8 BS01 CSF C 1 G8 G10 C30 N31 Q32 N51 L54 T131 S132 G133 I153 D154 F155 Y156 S161 Y162 F178 H188 G8 G10 C30 N31 Q32 N51 L54 T131 S132 G133 I153 D154 F155 Y156 S161 Y162 F178 H188 R129 Y156 Y162 H188 R129 Y156 Y162 H188 2.4.99.- remove_due_to_license_issue Q9LAK3 14730352 1001 MKKVIIAGNGPSLKEIDYSRLPNDFDVFRCNQFYFEDKYYLGKKCKAVFYNPSLFFEQYYTLKHLIQNQEYETELIMCSNYNQAHLENENFVKTFYDYFPDAHLGYDFFKQLKDFNAYFKFHEIYFNQRITSGVYMCAVAIALGYKEIYLSGIDFYQNGSSYAFDTKQKNLLKLAPNFKNDNSHYIGHSKNTDIKALEFLEKTYKIKLYCLCPNSLLANFIELAPNLNSNFIIQEKNNYTKDILIPSSEAYGKFSKNI 1ros A 2.0 BS06 DEO A 1 L181 A182 H183 A184 H218 E219 H222 H228 V235 P238 T239 Y240 K241 F248 L76 A77 H78 A79 H113 E114 H117 H123 V130 P133 T134 Y135 K136 F143 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.0017uM remove_due_to_license_issue P39900 15289103 1 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1rp7 A 2.09 BS02 TZD A 1 S109 Q140 H142 V192 S193 M194 G229 D230 G231 E232 N260 Q262 L264 K392 S54 Q85 H87 V137 S138 M139 G174 D175 G176 E177 N205 Q207 L209 K337 1.2.4.1 0000287,0003824,0004738,0004739,0005515,0005829,0016020,0016491,0030976,0036094,0042802,0042803,0042867,0045254,0046872,0060090 Ki>0.003uM remove_due_to_license_issue P0AFG8 14992577 889 ISNYINTIPVEEQPEYPGNLELERRIRSAIRWNAIMTVLRASKKDLELGGHMASFQSSATIYDVCFNHFFRARNEQDGGDLVYFQGHISPGVYARAFLEGRLTQEQLDNFRQEVHGNGLSSYPHPKLMPEFWQFPTVSMGLGPIGAIYQAKFLKYLEHRGLKDTSKQTVYAFLGDGEMDEPESKGAITIATREKLDNLVFVINCNLQRLDGPVTGNGKIINELEGIFEGAGWNVIKVMWGSRWDELLRKDTSGKLIQLMNETVDGDYQTFKSKDGAYVREHFFGKYPETAALVADWTDEQIWALNRGGHDPKKIYAAFKKAQETKGKATVILAHTIKGYGMGDAAMDGVRHIRDRFNVPVSDADIEKLPYITFPEGSEEHTYLHAQRQKLHGYLPSRQPNFTEKLELPSLQDFGALLEEQSKEISTTIAFVRALNVMLKNKSIKDRLVPIIADEARTFGMEGLFRQIGIYSPEDEKGQILQEGINELGAGCSWLAAATSYSTNNLPMIPFYIYYSMFGFQRIGDLCWAAGDQQARGFLIGGTSGRTTLNGEGLQHEDGHSHIQSLTIPNCISYDPAYAYEVAVIMHDGLERMYGEKQENVYYYITTLNENYHMPAMPEGAEEGIRKGIYKLETIEGSKGKVQLLGSGSILRHVREAAEILAKDYGVGSDVYSVTSFTELARDGQDCERWNMLHPLETPRVPYIAQVMNDAPAVASTDYMKLFAEQVRTYVPADDYRVLGTDGFGRSDSRENLRHHFEVDASYVVVAALGELAKRGEIDKKVVADAIAKFNIDADKVNPRLA 1rp7 A 2.09 BS03 TZD B 1 I569 E571 F602 I484 E486 F517 1.2.4.1 0000287,0003824,0004738,0004739,0005515,0005829,0016020,0016491,0030976,0036094,0042802,0042803,0042867,0045254,0046872,0060090 Ki>0.003uM remove_due_to_license_issue P0AFG8 14992577 887 ISNYINTIPVEEQPEYPGNLELERRIRSAIRWNAIMTVLRASKKDLELGGHMASFQSSATIYDVCFNHFFRARNEQDGGDLVYFQGHISPGVYARAFLEGRLTQEQLDNFRQEVHGNGLSSYPHPKLMPEFWQFPTVSMGLGPIGAIYQAKFLKYLEHRGLKDTSKQTVYAFLGDGEMDEPESKGAITIATREKLDNLVFVINCNLQRLDGPVTGNGKIINELEGIFEGAGWNVIKVMWGSRWDELLRKDTSGKLIQLMNETVDGDYQTFKSKDGAYVREHFFGKYPETAALVADWTDEQIWALNRGGHDPKKIYAAFKKAQETKGKATVILAHTIKGYGMGDAAMDGVRHIRDRFNVPVSDADIEKLPYITFPEGSEEHTYLHAQRQKLHGYLPSRQPNFTEKLELPSLQDFGALLEEQSKEISTTIAFVRALNVMLKNKSIKDRLVPIIADEARTFGMEGLFRQIGIYSPEDEKGQILQEGINELGAGCSWLAAATSYSTNNLPMIPFYIYYSMFGFQRIGDLCWAAGDQQARGFLIGGTSGRTTLNGEGLQHEDGHSHIQSLTIPNCISYDPAYAYEVAVIMHDGLERMYGEKQENVYYYITTLNENYHMPAMPEGAEEGIRKGIYKLETIEGSKGKVQLLGSGSILRHVREAAEILAKDYGVGSDVYSVTSFTELARDGQDCERWNMLHPLETPRVPYIAQVMNDAPAVASTDYMKLFAEQVRTYVPADDYRVLGTDGFGRSDSRENLRHHFEVDASYVVVAALGELAKRGEIDKKVVADAIAKFNIDADKVNPRLA 1rp7 B 2.09 BS01 TZD A 1 E522 I569 E571 F602 E454 I484 E486 F517 1.2.4.1 0000287,0003824,0004738,0004739,0005515,0005829,0016020,0016491,0030976,0036094,0042802,0042803,0042867,0045254,0046872,0060090 Ki>0.003uM remove_due_to_license_issue P0AFG8 14992577 889 ISNYINTIPVEEQPEYPGNLELERRIRSAIRWNAIMTVLRASKKDLELGGHMASFQSSATIYDVCFNHFFRARNEQDGGDLVYFQGHISPGVYARAFLEGRLTQEQLDNFRQEVHGNGLSSYPHPKLMPEFWQFPTVSMGLGPIGAIYQAKFLKYLEHRGLKDTSKQTVYAFLGDGEMDEPESKGAITIATREKLDNLVFVINCNLQRLDGPVTGNGKIINELEGIFEGAGWNVIKVMWGSRWDELLRKDTSGKLIQLMNETVDGDYQTFKSKDGAYVREHFFGKYPETAALVADWTDEQIWALNRGGHDPKKIYAAFKKAQETKGKATVILAHTIKGYGMGDAAMDGVRHIRDRFNVPVSDADIEKLPYITFPEGSEEHTYLHAQRQKLHGYLPSRQPNFTEKLELPSLQDFGALLEEQSKEISTTIAFVRALNVMLKNKSIKDRLVPIIADEARTFGMEGLFRQIGIYSPEDEKGQILQEGINELGAGCSWLAAATSYSTNNLPMIPFYIYYSMFGFQRIGDLCWAAGDQQARGFLIGGTSGRTTLNGEGLQHEDGHSHIQSLTIPNCISYDPAYAYEVAVIMHDGLERMYGEKQENVYYYITTLNENYHMPAMPEGAEEGIRKGIYKLETIEGSKGKVQLLGSGSILRHVREAAEILAKDYGVGSDVYSVTSFTELARDGQDCERWNMLHPLETPRVPYIAQVMNDAPAVASTDYMKLFAEQVRTYVPADDYRVLGTDGFGRSDSRENLRHHFEVDASYVVVAALGELAKRGEIDKKVVADAIAKFNIDADKVNPRLA 1rp7 B 2.09 BS03 TZD B 1 S109 Q140 H142 V192 S193 M194 G229 D230 G231 E232 N260 Q262 K392 S54 Q85 H87 V137 S138 M139 G174 D175 G176 E177 N205 Q207 K337 1.2.4.1 0000287,0003824,0004738,0004739,0005515,0005829,0016020,0016491,0030976,0036094,0042802,0042803,0042867,0045254,0046872,0060090 Ki>0.003uM remove_due_to_license_issue P0AFG8 14992577 887 ISNYINTIPVEEQPEYPGNLELERRIRSAIRWNAIMTVLRASKKDLELGGHMASFQSSATIYDVCFNHFFRARNEQDGGDLVYFQGHISPGVYARAFLEGRLTQEQLDNFRQEVHGNGLSSYPHPKLMPEFWQFPTVSMGLGPIGAIYQAKFLKYLEHRGLKDTSKQTVYAFLGDGEMDEPESKGAITIATREKLDNLVFVINCNLQRLDGPVTGNGKIINELEGIFEGAGWNVIKVMWGSRWDELLRKDTSGKLIQLMNETVDGDYQTFKSKDGAYVREHFFGKYPETAALVADWTDEQIWALNRGGHDPKKIYAAFKKAQETKGKATVILAHTIKGYGMGDAAMDGVRHIRDRFNVPVSDADIEKLPYITFPEGSEEHTYLHAQRQKLHGYLPSRQPNFTEKLELPSLQDFGALLEEQSKEISTTIAFVRALNVMLKNKSIKDRLVPIIADEARTFGMEGLFRQIGIYSPEDEKGQILQEGINELGAGCSWLAAATSYSTNNLPMIPFYIYYSMFGFQRIGDLCWAAGDQQARGFLIGGTSGRTTLNGEGLQHEDGHSHIQSLTIPNCISYDPAYAYEVAVIMHDGLERMYGEKQENVYYYITTLNENYHMPAMPEGAEEGIRKGIYKLETIEGSKGKVQLLGSGSILRHVREAAEILAKDYGVGSDVYSVTSFTELARDGQDCERWNMLHPLETPRVPYIAQVMNDAPAVASTDYMKLFAEQVRTYVPADDYRVLGTDGFGRSDSRENLRHHFEVDASYVVVAALGELAKRGEIDKKVVADAIAKFNIDADKVNPRLA 1rpf A 2.2 BS01 C3P A 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue Ki=103000nM P61823 7756988 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1rpj A 1.8 BS01 ALL A 1 K9 N13 F15 E42 D91 S147 R151 W175 N201 D227 Q247 K9 N13 F15 E42 D91 S147 R151 W175 N201 D227 Q247 ? 0015752,0015754,0016020,0030246,0030288,0042597,0048029,0055052,0055085 Kd=0.33uM remove_due_to_license_issue P39265 10064713 291 AAEYAVVLKTLSNPFWVDMKKGIEDEAKTLGVSVDIFASPSEGDFQSQLQLFEDLSNKNYKGIAFAPLSSVNLVMPVARAWKKGIYLVNLDEKIDMDNLKKAGGNVEAFVTTDNVAVGAKGASFIIDKLGAEGGEVAIIEGKAGNASGEARRNGATEAFKKASQIKLVASQPADWDRIKALDVATNVLQRNPNIKAIYCANDTMAMGVAQAVANAGKTGKVLVVGTDGIPEARKMVEAGQMTATVAQNPADIGATGLKLMVDAEKSGKVIPLDKAPEFKLVDSILVTQ 1rpu A 2.5 BS01 rna C 0 R11 W39 T40 R43 K67 S113 R115 S120 R3 W31 T32 R35 K53 S99 R101 S106 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 14697199 1 ~ 21 DTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDENPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLTPVEV 1rpu A 2.5 BS02 rna D 0 R18 P37 W39 W42 K60 Y73 Q107 V108 G109 G125 G126 R10 P29 W31 W34 K46 Y59 Q93 V94 G95 G111 G112 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 14697199 1 ~ 21 DTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDENPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLTPVEV 1rpu B 2.5 BS01 rna C 0 R18 W39 W42 K60 Y73 Q107 V108 G109 S124 G125 G126 R11 W32 W35 K47 Y60 Q94 V95 G96 S111 G112 G113 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 14697199 1 ~ 21 NDTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDENPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLTP 1rpu B 2.5 BS02 rna D 0 W39 T40 S62 K67 V69 T111 S113 R115 S120 T122 W32 T33 S49 K54 V56 T98 S100 R102 S107 T109 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 14697199 1 ~ 21 NDTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDENPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLTP 1rql B 2.4 BS02 VSO B 1 D12 A14 T126 Y128 D8 A10 T122 Y124 D12 A14 A45 M49 K53 H56 R160 D186 D8 A10 A41 M45 K49 H52 R156 D182 3.11.1.1 0000287,0003824,0005829,0006281,0008967,0016787,0019700,0046872,0050194 Ki=1.79mM remove_due_to_license_issue O31156 14670958 600 KIEAVIFDWAGTTVDYGCFAPLEVFMEIFHKRGVAITAEEARKPMGLLKIDHVRALTEMPRIASEWNRVFRQLPTEADIQEMYEEFEEILFAILPRYASPINAVKEVIASLRERGIKIGSTTGYTREMMDIVAKEAALQGYKPDFLVTPDDVPAGRPYPWMCYKNAMELGVYPMNHMIKVGDTVSDMKEGRNAGMWTVGVILGSSELGLTEEEVENMDSVELREKIEVVRNRFVENGAHFTIETMQELESVMEHIEK 1rr6 A 2.5 BS01 IMH A 1 A116 A117 G118 F200 E201 V217 M219 N243 H257 A114 A115 G116 F198 E199 V215 M217 N241 H255 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S31 H62 H84 Y86 E87 A114 M217 S218 N241 V243 H255 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 14982926 300 NGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPL 1rri A 2.0 BS01 A45 A 1 Y13 G14 Y15 H16 M65 E66 G67 A69 Y13 G14 Y15 H16 M65 E66 G67 A69 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 ic50=1.5uM remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rrw A 2.21 BS01 9MG A 1 L72 L73 E74 L72 L73 E74 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 ic50=28uM remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rry A 2.7 BS01 204 A 1 A18 E22 L72 L73 E74 A18 E22 L72 L73 E74 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rs2 A 2.31 BS01 209 A 1 N71 L72 E74 N71 L72 E74 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 ic50=50uM remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rs4 A 2.7 BS01 45P A 1 L19 L73 E74 P104 I105 L19 L73 E74 P104 I105 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rsd A 2.5 BS01 PSB A 1 L72 E74 P104 P106 L72 E74 P104 P106 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 ic50=0.3uM remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rsi A 2.2 BS01 977 A 1 A18 L72 L73 E74 A18 L72 L73 E74 E22 K100 E22 K100 4.1.2.25,5.1.99.8 0004150,0005737,0006760,0016829,0016853,0046654,0046656 ic50=38uM remove_due_to_license_issue P56740 15027862 1001 MQDTIFLKGMRFYGYHGALSAENEIGQIFKVDVTLKVDLSEAGRTDNVIDTVHYGEVFEEVKSIMEGKAVNLLEHLAERIANRINSQYNRVMETKVRITKENPPIPGHYDGVGIEIVRENK 1rt1 A 2.55 BS01 MKC A 1 L100 K101 K103 V106 Y181 Y188 G190 F227 W229 L234 Y318 L100 K101 K103 V106 Y181 Y188 G190 F227 W229 L234 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 8648598 999 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAH 1rt2 A 2.55 BS01 TNK A 1 L100 K101 K103 V106 Y181 Y188 F227 W229 H235 P236 Y318 L100 K101 K103 V106 Y181 Y188 F227 W229 H235 P236 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 8648598 999 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIG 1rt9 A 2.3 BS01 IMH A 1 Y88 A116 A117 G118 F200 E201 V217 M219 N243 H257 Y86 A114 A115 G116 F198 E199 V215 M217 N241 H255 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S31 H62 H84 Y86 E87 A114 M217 S218 N241 V243 H255 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 300 NGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPL 1rth A 2.2 BS01 U05 A 1 P95 L100 Y181 Y188 Y318 P95 L100 Y181 Y188 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=0.4uM remove_due_to_license_issue P04585 7540934 999 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIG 1rti A 3.0 BS01 HEF A 1 L100 K101 K103 V106 Y188 P225 F227 P236 L100 K101 K103 V106 Y188 P225 F227 P236 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 7540934 999 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIG 1rtl A 2.75 BS04 CPX A 1 Q41 H57 I132 S139 F154 A156 A157 Q41 H57 I132 S139 F154 A156 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P26664 14627400 201 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVTKAVDFIPVENLETTMR 1ru1 A 1.4 BS03 APC A 1 Q74 D95 D97 I98 R110 L111 T112 H115 Y116 R121 Q68 D80 D82 I83 R95 L96 T97 H100 Y101 R106 R92 D95 D97 R77 D80 D82 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 remove_due_to_license_issue P26281 14769023 171 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPPDYLNAAVALETSLAPEELLNHTQRIELQQGRRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 1ru2 A 1.48 BS03 APC A 1 L70 Q74 D95 D97 I98 R110 L111 T112 H115 Y116 R121 L64 Q68 D83 D85 I86 R98 L99 T100 H103 Y104 R109 R92 D95 D97 R80 D83 D85 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=0.32uM remove_due_to_license_issue P26281 14769023 171 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPPDYLNAAVALETSLAPEELLNHTQRIELQQGRGGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 1rv1 A 2.3 BS01 IMZ A 1 L54 G58 I61 M62 Q72 H73 V93 H96 Y100 L30 G34 I37 M38 Q48 H49 V69 H72 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.14uM remove_due_to_license_issue IC50=140nM Q00987 14704432 110 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 1rv1 A 2.3 BS02 IMZ A 2 M50 Y100 M26 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.14uM remove_due_to_license_issue IC50=140nM Q00987 14704432 111 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 1rv1 A 2.3 BS03 IMZ C 1 L54 H96 Y100 L30 H72 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.14uM remove_due_to_license_issue IC50=140nM Q00987 14704432 110 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 1rv1 C 2.3 BS01 IMZ C 1 L54 L57 G58 I61 M62 Q72 V93 H96 Y100 L30 L33 G34 I37 M38 Q48 V69 H72 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.14uM remove_due_to_license_issue IC50=140nM Q00987 14704432 110 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 1rw8 A 2.4 BS01 580 A 1 A230 K232 Y249 L260 L278 S280 N338 L340 A31 K33 Y50 L61 L79 S81 N139 L141 D333 K335 N338 D351 T375 D134 K136 N139 D152 T176 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.175uM remove_due_to_license_issue IC50=1320nM P36897 15177479 501 TIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG 1rwq A 2.2 BS01 5AP A 1 R125 E205 E206 Y547 S630 Y662 Y666 R87 E167 E168 Y509 S592 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.0001uM remove_due_to_license_issue IC50=0.1nM P27487 15006388 900 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 1rww A 2.8 BS01 OQB A 1 R179 H237 Q283 C285 R57 H115 Q161 C163 P177 R178 H237 G238 C285 R286 P55 R56 H115 G116 C163 R164 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue IC50=5nM, Ki=5nM P29466 16274992 501 MPTSSGSEGNVKLCSLEEAQRIWKQKSAEIYPIMDKSSRTRLALIICNEEFDSIPRRTGAEVDITGMTMLLQNLGYSVDVKKNLTASDMTTELEAFAHRPEHKTSDSTFLVFMSHGIREGICGKKHSEQVPDILQLNAIFNMLNTKNCPSLKDKPKVIIIQACRGDSPGVVWFKD 1rww B 2.8 BS01 OQB A 1 S339 W340 R341 H342 M345 S347 R383 S23 W24 R25 H26 M29 S31 R67 E390 E74 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue IC50=5nM, Ki=5nM P29466 16274992 501 AIKKAHIEKDFIAFCSSTPDNVSWRHPTMGSVFIGRLIEHMQEYACSCDVEEIFRKVRFSFEQPDGRAQMPTTERVTLTRCFYLFPGH 1rwx A 1.85 BS01 YBH A 1 R179 H237 Q283 C285 R60 H118 Q164 C166 P177 R178 H237 G238 C285 R286 P58 R59 H118 G119 C166 R167 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 16274992 501 NPAMPTSSGSEGNVKLCSLEEAQRIWKQKSAEIYPIMDKSSRTRLALIICNEEFDSIPRRTGAEVDITGMTMLLQNLGYSVDVKKNLTASDMTTELEAFAHRPEHKTSDSTFLVFMSHGIREGICGKKHSEQVPDILQLNAIFNMLNTKNCPSLKDKPKVIIIQACRGDSPGVVWFKD 1rwx B 1.85 BS01 YBH A 1 S339 R341 H342 R352 D381 R383 S23 R25 H26 R36 D65 R67 E390 E74 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 16274992 501 AIKKAHIEKDFIAFCSSTPDNVSWRHPTMGSVFIGRLIEHMQEYACSCDVEEIFRKVRFSFEQPDGRAQMPTTERVTLTRCFYLFPGH 1rxp A 1.7 BS02 169 A 1 F41 H57 K60 D189 S190 C191 Q192 S195 V213 F24 H40 K43 D171 S172 C173 Q174 S177 V191 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 15081015 991 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1ryf A 1.75 BS01 GDP A 1 A13 G15 K16 T17 C18 F28 K135 D137 L138 S177 A178 L179 A15 G17 K18 T19 C20 F30 K104 D106 L107 S146 A147 L148 3.6.5.2 0003924,0005525,0007264 remove_due_to_license_issue P63000 14625275 538 GSMQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAIADVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLRDDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPPPV 1ryh A 1.75 BS01 GNP A 1 A13 G15 K16 T17 C18 F28 K135 D137 L138 S177 A178 L179 A15 G17 K18 T19 C20 F30 K105 D107 L108 S147 A148 L149 3.6.5.2 0003924,0005525,0007264 remove_due_to_license_issue P63000 14625275 538 GSMQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAGIADVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLRDDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPPPV 1s03 G 2.7 BS01 rna B 0 P5 S29 K30 R83 Y85 R87 K88 S104 T105 S106 K107 G119 G121 P2 S26 K27 R80 Y82 R84 K85 S101 T102 S103 K104 G116 G118 ? 0000028,0002181,0003735,0005737,0005829,0005840,0006412,0006417,0019843,0022627,0043488,1990904 remove_due_to_license_issue P0A7W7 15146079 1 ~ 47 DPIADMLTRIRNGQAANKAAVTMPSSKLKVAIANVLKEEGFIEDFKVEGDTKPELELTLKYFQGKAVVESIQRVSRPGLRIYKRKDELPKVMAGLGIAVVSTSKGVMTDRAARQAGLGGEIICYVA 1s03 H 2.7 BS01 rna A 0 P27 S29 K30 R83 Y85 K86 R87 K88 S104 T105 S106 K107 G119 G121 P25 S27 K28 R81 Y83 K84 R85 K86 S102 T103 S104 K105 G117 G119 ? 0000028,0002181,0003735,0005737,0005829,0005840,0006412,0006417,0019843,0022627,0043488,1990904 remove_due_to_license_issue P0A7W7 15146079 1 ~ 47 QDPIADMLTRIRNGQAANKAAVTMPSSKLKVAIANVLKEEGFIEDFKVEGDTKPELELTLKYFQGKAVVESIQRVSRPGLRIYKRKDELPKVMAGLGIAVVSTSKGVMTDRAARQAGLGGEIICYVA 1s17 A 1.95 BS01 GNR A 1 G44 I45 G46 Q51 Y88 E90 G91 C92 L93 H134 E135 H138 G43 I44 G45 Q50 Y87 E89 G90 C91 L92 H133 E134 H137 G46 Q51 C92 L93 H134 E135 H138 G45 Q50 C91 L92 H133 E134 H137 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50<5nM remove_due_to_license_issue Q9I7A8 15006385 501 AILNILEFPDPRLRTIAKPVEVVDDAVRQLIDDMFETMYEAPGIGLAATQVNVHKRIVVMDLSEDKSEPRVFINPEFEPLTEEMDQYQEGCLSVPGFYENVDRPQKVRIKALDRDGNPFEEVAEGLLAVCIQHECDHLNGKLFVDYLSTLKRDRIRKKLEKQHRQQ 1s19 A 2.1 BS01 MC9 A 1 Y143 V234 S237 R274 S275 S278 W286 H305 H397 Y24 V64 S67 R104 S105 S108 W116 H135 H227 ? 0003677,0004879,0006355 remove_due_to_license_issue Kd=0.31nM P11473 15055995 500 LRPKLSEEQQRIIAILLDAHHKTYDPTYSDFCQFRPPVRVNDGGGSVTLELSQLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSEDQIVLLKSSAIEVIMLRSNESFTMDDMSWTCGNQDYKYRVSDVTKAGHSLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAALIEAIQDRLSNTLQTYIRCRHPPPGSHLLYAKMIQKLADLRSLNEEHSKQYRCLSFQPECSMKLTPLVLEVFG 1s26 A 3.0 BS01 APC A 1 K346 H351 S354 K372 K382 D493 N583 F586 K55 H60 S63 K81 K91 D202 N292 F295 4.6.1.1 0005576,0008294 remove_due_to_license_issue P40136 15063758 1139 RIDVLKGEKALKASGLVPEHADAFKKIARELNTYILFRPVNKLATNLIKSGVATKGLNVHGKSSDWGPVAGYIPFDQDLSKKHGQQLAVEKGNLENKKSITEHEGEIGKIPLKLDHLRIEELKENGIILKGKKEIDNGKKYYLLESNNQVYEFRISDENNEVQYKTKEGKITVLGEKFNWRNIEVMAKNVEGVLKPLTADYDLFALAPSLTEIKKQIPQKEWDKVVNTPNSLEKQKGVTNLLIKYGIERKPDSTKGTLSNWQKQMLDRLNEAVKYTGYTGGDVVNHGTEQDNEEFPEKDNEIFIINPEGEFILTKNWEMTGRFIEKNITGKDYLYYFNRSYNKIAPGNKAYIEWTDPITKAKINTIPTSAEFIKNLSSIRRSSSVKKIAGYLSDYYNSANHIFSQEKKRKISIFRGIQAYNEIENVLKSKQIAPEYKNYFQYLKERITNQVQLLLTHQKFKLLYKQLNFTENETDNFEVFQKIID 1s38 A 1.81 BS02 MAQ A 1 D102 Y106 D156 C158 G229 L231 M260 G261 D92 Y96 D138 C140 G211 L213 M242 G243 D102 D280 C318 C320 C323 H349 D92 D262 C300 C302 C305 H331 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=7uM remove_due_to_license_issue P28720 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1s39 A 1.95 BS02 AQO A 1 D102 Y106 D156 G229 G230 M260 G261 D92 Y96 D140 G213 G214 M244 G245 D102 D280 C318 C320 C323 H349 D92 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=20nM remove_due_to_license_issue P28720 900 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLTKQSEEGVTFKSHSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 1s40 A -1.00 BS01 dna B 0 T25 Y27 S38 K41 A43 F44 S46 Y61 L62 Y63 D64 Y66 Y70 K73 K81 I83 Y85 D112 N114 K127 K129 Y131 L135 N136 I138 T21 Y23 S34 K37 A39 F40 S42 Y57 L58 Y59 D60 Y62 Y66 K69 K77 I79 Y81 D108 N110 K123 K125 Y127 L131 N132 I134 ? 0000723,0000781,0003677 remove_due_to_license_issue P32797 15066429 1 ~ 11 KMARKDPTIEFCQLGLDTFETKYITMFGMLVSCSFDKPAFISFVFSDFTKNDIVQNYLYDRYLIDYENKLELNEGFKAIMYKNQFETFDSKLRKIFNNGLRDLQNGRDENLSQYGIVCKMNIKVKMYNGKLNAIVRECEPVPHSQISSIASPSQCEHLRLFYQRAFKRIGESAISRYFEEYRRFFPI 1s4d A 2.7 BS01 SAH A 1 G100 G101 D102 V105 T130 A131 Y183 M184 N212 A213 P240 A241 I242 G93 G94 D95 V98 T123 A124 Y169 M170 N198 A199 P226 A227 I228 D47 K69 M184 D42 K64 M170 2.1.1.107 0004851,0006779,0008168,0009236,0019354,0032259 remove_due_to_license_issue P21631 15522295 1501 FAGLPALEKGSVWLVGAGPGDPGLLTLHAANALRQADVIVHDALVNEDCLKLARPGAVLEFAGKRGPSPKQRDISLRLVELARAGNRVLRLKGGDPFVFGRGGEEALTLVEHQVPFRIVPGITAGIGGLAYAGIPVTHREVNHAVTFLTGHDRINWQGIASGSPVIVMYMAMKHIGAITANLIAGGRSPDEPVAFVCNAATPQQAVLETTLARAEADVAAAGLEPPAIVVVGEVVRLRAALDWIGALDGRKLAADP 1s4d B 2.7 BS01 SAH B 1 P24 L49 G100 G101 D102 V105 T130 A131 Y183 M184 N212 A213 P240 A241 I242 P21 L46 G97 G98 D99 V102 T127 A128 Y179 M180 N208 A209 P236 A237 I238 D47 K69 M184 D44 K66 M180 2.1.1.107 0004851,0006779,0008168,0009236,0019354,0032259 remove_due_to_license_issue P21631 15522295 1511 DLFAGLPALEKGSVWLVGAGPGDPGLLTLHAANALRQADVIVHDALVNEDCLKLARPGAVLEFAGKRGGKPSPKQRDISLRLVELARAGNRVLRLKGGDPFVFGRGGEEALTLVEHQVPFRIVPGITAGIGGLAYAGIPVTHREVNHAVTFLTGHDSSGVPDRINWQGIASGSPVIVMYMAMKHIGAITANLIAGGRSPDEPVAFVCNAATPQQAVLETTLARAEADVAAAGLEPPAIVVVGEVVRLRAALDWIGALDGRKLA 1s50 A 1.65 BS01 GLU A 1 Y61 P89 L90 A91 R96 G141 A142 T143 E191 Y60 P88 L89 A90 R95 G140 A141 T142 E190 ? 0015276,0016020 Ki=1.4uM remove_due_to_license_issue P42260 15721240 999 SNRSLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCPE 1s5z A 2.0 BS01 SON A 1 K16 H59 F64 T98 R109 V116 N119 K11 H54 F59 T93 R104 V111 N114 K16 Y56 N119 H122 E133 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 remove_due_to_license_issue P22887 16787337 1160 VNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIHGSDSVESANREIALWFKPEELLTEVKPNPNLYE 1s63 B 1.9 BS05 778 B 1 W102 W106 R202 D297 C299 Y361 H362 W88 W92 R188 D283 C285 Y347 H348 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H234 R277 K280 D283 C285 Y286 D338 D345 H348 2.5.1.58 0003824,0004659,0004660,0005515,0005829,0005875,0005965,0006629,0008270,0008318,0018343,0046872 Ki=0.9nM remove_due_to_license_issue IC50=2nM P49356 15248757 3012 SSPVWSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPEGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYDIINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKRERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVLGVPENALQPTHPVYNIGPDKVIQATTYFLQKPVPGFE 1s64 B 2.55 BS02 778 B 1 R173 Q212 H219 G221 D269 C271 Y272 W275 H321 R156 Q195 H202 G204 D252 C254 Y255 W258 H304 H219 R263 K266 D269 C271 Y272 K311 D318 H321 H202 R246 K249 D252 C254 Y255 K294 D301 H304 2.5.1.59 0003824,0004659,0004661,0004662,0005515,0005953,0008270,0008284,0008318,0018344,0034097,0036094,0042277,0045787,0046872,0051771,1901363 remove_due_to_license_issue P53610 15248757 380 LDFLRDRHVRFFQRCLQVLPERYSSLETSRLTIAFFALSGLDMLDSLDVVNKDDIIEWIYSLQVLPTEDRSNLDRCGFRGSSYLGIPFNPSKNPGTAHPYDSGHIAMTYTGLSCLIILGDDLSRVDKEACLAGLRALQLEDGSFCAVPEGSENDMRFVYCASCICYMLNNWSGMDMKKAISYIRRSMSYDNGLAQGAGLESHGGSTFCGIASLCLMGKLEEVFSEKELNRIKRWCIMRQQNGYHGRPNKPVDTCYSFWVGATLKLLKIFQYTNFEKNRNYILSTQDRLVGGFAKWPDSHPDALHAYFGICGLSLMEESGICKVHPALNVSTRTSERLRDLHQSWKT 1s89 A 2.22 BS01 PGA A 1 V17 H19 K23 T45 T47 T48 S65 G66 D71 V17 H19 K23 T45 T47 T48 S65 G66 D71 H19 G66 D71 D91 N98 D101 R107 H19 G66 D71 D91 N98 D101 R107 4.2.3.3 0005737,0005829,0008929,0016829,0019242,0034214,0042802 Ki=5.8uM remove_due_to_license_issue P0A731 15049687 201 MELTTRTLPARKHIALVAHDHCKQMLMSWVERHQPLLEQHVLYATGTTGNLISRATGMNVNAMLSGPMGGDQQVGALISEGKIDVLIFFWDPLNAVPNDPDVKALLRLATVWNIPVATNVATADFIIQSPHFNDAVDILIPDYQRYLADRLK 1s89 F 2.22 BS01 PGA F 1 K23 T45 T47 T48 S65 G66 D71 K23 T45 T47 T48 S65 G66 D71 H19 G66 D71 D91 N98 D101 R107 H19 G66 D71 D91 N98 D101 R107 4.2.3.3 0005737,0005829,0008929,0016829,0019242,0034214,0042802 Ki=5.8uM remove_due_to_license_issue P0A731 15049687 206 MELTTRTLPARKHIALVAHDHCKQMLMSWVERHQPLLEQHVLYATGTTGNLISRATGMNVNAMLSGPMGGDQQVGALISEGKIDVLIFFWDPLNAVPNDPDVKALLRLATVWNIPVATNVATADFIIQSPHFNDAVDILIPDYQRYLADRLK 1s9t A 1.8 BS01 QUS A 1 Y61 P89 R96 V138 G141 A142 T143 N174 M190 E191 Y59 P87 R94 V136 G139 A140 T141 N172 M188 E189 ? 0015276,0016020 Ki=253nM remove_due_to_license_issue Ki=134nM P42260 15721240 1001 NRSLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWWR 1sb1 H 1.9 BS03 165 H 1 H57 Y60A W60D N98 I174 D189 A190 S195 W215 G216 E217 G219 R221A H43 Y47 W50 N95 I171 D191 A192 S197 W219 G220 E221 G222 R225 3.4.21.5 0004252,0005509,0006508,0007596 Ki=128nM remove_due_to_license_issue P00734 15051174 1001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1sbg A 2.3 BS01 IM1 A 1 D25 G27 V82 I84 D25 G27 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=18nM remove_due_to_license_issue P03366 7918383 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1sbg B 2.3 BS01 IM1 A 1 D25 G27 A28 D29 D30 G49 V82 D25 G27 A28 D29 D30 G49 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 7918383 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1sbr A 2.3 BS02 VIB A 1 F15 S16 L17 D45 H46 I47 S48 T49 F7 S8 L9 D37 H38 I39 S40 T41 ? 0030975 Kd~10uM remove_due_to_license_issue O34911 15451668 501 RIAGFRFSLYPMTDDFISVIKSALAATDTSKVWTKTDHISTVLRGSIDHVFDAAKAIYLHAANSEQHIVMNGTFSIGCPGDTQGDTYLKRVNEDAVRGLKAEAPCQFALYPMNEPDYMGLIMEAVDIAKAQGTFVQGVHYASELDGDAHDVFSTLEAVFRMAEQQTNHITMTVNLSANSPSR 1sbr A 2.3 BS03 VIB A 2 F119 A120 L121 M130 I133 S154 F107 A108 L109 M118 I121 S142 ? 0030975 Kd~10uM remove_due_to_license_issue O34911 15451668 502 RIAGFRFSLYPMTDDFISVIKSALAATDTSKVWTKTDHISTVLRGSIDHVFDAAKAIYLHAANSEQHIVMNGTFSIGCPGDTQGDTYLKRVNEDAVRGLKAEAPCQFALYPMNEPDYMGLIMEAVDIAKAQGTFVQGVHYASELDGDAHDVFSTLEAVFRMAEQQTNHITMTVNLSANSPSR 1sbr B 2.3 BS01 VIB B 1 F15 S16 L17 I25 T44 D45 H46 I47 S48 T49 F7 S8 L9 I17 T36 D37 H38 I39 S40 T41 ? 0030975 Kd~10uM remove_due_to_license_issue O34911 15451668 503 RIAGFRFSLYPMTDDFISVIKSALAATDTSKVWTKTDHISTVLRGSIDHVFDAAKAIYLHAANSEQHIVMNGTFSIGCPGDTQGDTYLSDKRVNEDAVRGLKAEAPCQFALYPMNEPDYMGLIMEAVDIAKAQGTFVQGVHYASELDGDAHDVFSTLEAVFRMAEQQTNHITMTVNLSANSP 1sbr B 2.3 BS02 VIB B 2 F119 A120 L121 M130 I133 A153 S154 F109 A110 L111 M120 I123 A143 S144 ? 0030975 Kd~10uM remove_due_to_license_issue O34911 15451668 504 RIAGFRFSLYPMTDDFISVIKSALAATDTSKVWTKTDHISTVLRGSIDHVFDAAKAIYLHAANSEQHIVMNGTFSIGCPGDTQGDTYLSDKRVNEDAVRGLKAEAPCQFALYPMNEPDYMGLIMEAVDIAKAQGTFVQGVHYASELDGDAHDVFSTLEAVFRMAEQQTNHITMTVNLSANSP 1sc7 A 3.0 BS01 dna B 0 V410 T411 W412 I424 Y426 M428 K436 K439 K443 N722 Y723 V212 T213 W214 I226 Y228 M230 K238 K241 K245 N524 Y525 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 1 ~ 10 EEQKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLNYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1sc7 A 3.0 BS02 dna C 0 R634 K638 G717 T718 R436 K440 G519 T520 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 11 ~ 22 EEQKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLNYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1sc7 A 3.0 BS03 dna D 0 F361 R362 G363 R364 H367 K374 R488 A489 N491 K493 T501 K532 D533 N574 T585 A586 K587 K650 F163 R164 G165 R166 H169 K176 R290 A291 N293 K295 T303 K334 D335 N376 T387 A388 K389 K452 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 101 ~ 122 EEQKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLNYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1sc8 U 2.4 BS01 2IN U 1 L97B H99 D189 S190 Q192 S195 W215 G216 R217 G219 C220 L92 H94 D192 S193 Q195 S198 W218 G219 R220 G221 C222 3.4.21.73 0004252,0006508 Ki=0.036uM remove_due_to_license_issue Ki=36nM P00749 15150279 300 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1sdt A 1.3 BS01 MK1 B 1 R8 D25 G27 G48 G49 I50 V82 I84 R8 D25 G27 G48 G49 I50 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1sdt B 1.3 BS01 MK1 B 1 D125 G127 A128 D129 D130 G148 G149 P181 V182 D25 G27 A28 D29 D30 G48 G49 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=540pM remove_due_to_license_issue P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1sdu A 1.25 BS01 MK1 B 1 R8 D25 G27 G48 G49 V82 R8 D25 G27 G48 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 1sdu B 1.25 BS01 MK1 B 1 R108 D125 G127 A128 D129 D130 I147 G148 P181 R8 D25 G27 A28 D29 D30 I47 G48 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=86pM remove_due_to_license_issue P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 1sdv A 1.4 BS01 MK1 B 1 D25 G27 G48 G49 I50 I84 D25 G27 G48 G49 I50 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 1sdv B 1.4 BS01 MK1 B 1 D125 G127 A128 D129 D130 I147 G148 G149 I150 P181 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1810pM remove_due_to_license_issue P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 1seu A 3.0 BS01 dna B 0 V410 T411 W412 I424 Y426 K436 K439 K443 K532 K587 S722 Y723 V210 T211 W212 I224 Y226 K236 K239 K243 K332 K387 S522 Y523 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 1 ~ 10 QKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLSYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1seu A 3.0 BS02 dna C 0 R316 K328 R634 G717 T718 R116 K128 R434 G517 T518 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 11 ~ 22 QKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLSYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1seu A 3.0 BS03 dna D 0 F361 R362 G363 R364 H367 R488 A489 N491 K493 T501 K532 D533 T585 A586 K587 L647 K746 F161 R162 G163 R164 H167 R288 A289 N291 K293 T301 K332 D333 T385 A386 K387 L447 K546 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 101 ~ 122 QKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLSYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1sgu A 1.9 BS01 MK1 B 1 D25 G27 I47 G48 I50 P81 A82 D25 G27 I47 G48 I50 P81 A82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15379553 2632 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 1sgu B 1.9 BS01 MK1 B 1 R8 D25 G27 A28 D29 D30 I32 I47 I50 P81 R8 D25 G27 A28 D29 D30 I32 I47 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4235nM remove_due_to_license_issue P03367 15379553 2632 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 1sh9 A 2.5 BS01 RIT B 1 D25 G27 D29 I32 G48 G49 I50 P81 D25 G27 D29 I32 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15379553 301 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 1sh9 B 2.5 BS01 RIT B 1 D25 G27 D30 I47 I50 P81 D25 G27 D30 I47 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=932nM remove_due_to_license_issue P03367 15379553 301 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 1si2 A 2.6 BS01 rna B 0 K264 H269 M273 R275 R278 F292 Y309 F310 Y314 K333 T335 Y336 L337 Q348 R349 K41 H46 M50 R52 R55 F69 Y80 F81 Y85 K104 T106 Y107 L108 Q119 R120 ? 0003723 remove_due_to_license_issue Q9UL18 15152257 401 ~ 409 MAQPVIEFMCEVLDIRNIDEQPKPLTDSQRVRFTKEIKGLKVEVTHCGQMKRKYRVCNVTRRPASHQTFPLQVECTVAQYFKQKYNLQLKYPHLPCLQVGQEQKHTYLPLEVCNIVAGQR 1si3 A 2.6 BS01 rna B 0 H269 M273 R275 R278 F292 Y309 F310 Y314 K333 H334 T335 Y336 G347 Q348 H46 M50 R52 R55 F69 Y80 F81 Y85 K104 H105 T106 Y107 G118 Q119 ? 0003723 remove_due_to_license_issue Q9UL18 15152257 401 ~ 409 MAQPVIEFMCEVLDIRNIDEQPKPLTDSQRVRFTKEIKGLKVEVTHCGQMKRKYRVCNVTRRPASHQTFPLQVECTVAQYFKQKYNLQLKYPHLPCLQVGQEQKHTYLPLEVCNIVAGQR 1siv A 2.5 BS01 PSI B 1 D25 G27 D29 V47 G48 I82 D25 G27 D29 V47 G48 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P05896 8241159 100 PQFSLWRRPVVTAHIEGQPVEVLLDTGADDSIVTGIELGPHYTPKIVGGIGGFINTKEYKNVKIEVLGKRIKGTIMTGDTPINIFGRNLLTALGMSLNL 1siv B 2.5 BS01 PSI B 1 D25 G27 A28 D29 D30 G48 G49 D25 G27 A28 D29 D30 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8.4nM remove_due_to_license_issue P05896 8241159 100 PQFSLWRRPVVTAHIEGQPVEVLLDTGADDSIVTGIELGPHYTPKIVGGIGGFINTKEYKNVKIEVLGKRIKGTIMTGDTPINIFGRNLLTALGMSLNL 1sj0 A 1.9 BS01 E4D A 1 M343 L346 T347 A350 D351 E353 W383 L387 F404 G521 H524 L525 C530 M37 L40 T41 A44 D45 E47 W77 L81 F98 G215 H218 L219 C224 ? ic50=0.8nM remove_due_to_license_issue IC50=0.8nM P03372 15084115 600 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCVVPLYDLLLEMLDAHRLHA 1skj A 2.0 BS01 UR2 A 1 R32 S34 T36 C42 H58 Y59 K60 I71 G93 R30 S32 T34 C40 H56 Y57 K58 I69 G91 2.7.10.2 ic50=7uM remove_due_to_license_issue P00524 9371236 113 EEWYFGKITRRESERLLLNPENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFSSLQQLVAYYSKHADGLCHRLTNVCPT 1sl3 A 1.81 BS02 170 A 1 H57 Y60B W60E N98 L99 I174 A190 C191 S195 V213 S214 W215 G216 C220 G226 F227 H69 Y73 W76 N121 L122 I197 A218 C219 S223 V243 S244 W245 G246 C249 G256 F257 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=1.4pM remove_due_to_license_issue Ki=0.001400nM P00734 15163182 1001 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1sm2 A 2.3 BS01 STU A 1 I369 G370 V377 A389 K391 F435 F437 M438 G441 R486 L489 D500 I13 G14 V21 A33 K35 F79 F81 M82 G85 R130 L133 D144 D482 A484 R486 N487 D500 P521 D126 A128 R130 N131 D144 P147 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki<10nM remove_due_to_license_issue Q08881 14766749 301 VIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 1snk A 2.4 BS01 MYE A 1 G23 C25 N60 D61 G65 G66 Y67 L160 H162 G22 C24 N59 D60 G64 G65 Y66 L159 H161 Q19 C25 H162 N182 Q18 C24 H161 N181 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=0.250000nM P43235 15177446 1 PDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1so2 A 2.4 BS03 666 A 1 I938 G940 P941 H948 T952 L987 Q988 S990 F991 I265 G267 P268 H275 T279 L314 Q315 S317 F318 3.1.4.17 0004114,0007165,0008081 ic50=0.27nM remove_due_to_license_issue Q13370 15147193 461 LDLILVEEYDSLIEKMSNWNFPIFELVEKMGEKSGRILSQVMYTLFQDTGLLEIFKIPTQQFMNYFRALENGYRDIPYHNRIHATDVLHAVWYLTTRPVPGLQQIHNGGRIAYISSKSCSNPDESYGCLSSNIPALELMALYVAAAMHDYDHPGRTNAFLVATNAPQAVLYNDRSVLENHHAASAWNLYLSRPEYNFLLHLDHVEFKRFRFLVIEAILATDLKKHFDFLAEFNAKANDVNSNGIEWSNENDRLLVCQVCIKLADINGPAKVRDLHLKWTEGIVNEFYEQGDEEANLGLPISPFMDRSSPQLAKLQESFITHIVGPLCNSYDAAGLLPGQWLESRRRIFCQLMHHLTENHKIWK 1sqa A 2.0 BS01 UI1 A 1 H54 H106 D205 S206 C207 Q208 W231 G234 C235 H46 H94 D192 S193 C194 Q195 W218 G221 C222 H54 D109 Q208 G209 D210 S211 G212 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.00062uM remove_due_to_license_issue IC50=620nM, Ki=0.620000nM P00749 15149645 1001 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1sqb C 2.69 BS03 AZO C 1 F128 Y131 G142 A143 I146 K269 P270 E271 F274 A277 L294 F127 Y130 G141 A142 I145 K268 P269 E270 F273 A276 L293 H201 S205 K227 D228 E271 H200 S204 K226 D227 E270 1.10.2.2 0005739,0005743,0006122,0008121,0009055,0016020,0016491,0020037,0022904,0031966,0045275,0046872,0048039,1902600 remove_due_to_license_issue P00157 15312779 383 TNIRKSHPLMKIVNNAFIDLPAPSNISSWWNFGSLLGICLILQILTGLFLAMHYTSDTTTAFSSVTHICRDVNYGWIIRYMHANGASMFFICLYMHVGRGLYYGSYTFLETWNIGVILLLTVMATAFMGYVLPWGQMSFWGATVITNLLSAIPYIGTNLVEWIWGGFSVDKATLTRFFAFHFILPFIIMAIAMVHLLFLHETGSNNPTGISSDVDKIPFHPYYTIKDILGALLLILALMLLVLFAPDLLGDPDNYTPANPLNTPPHIKPEWYFLFAYAILRSIPNKLGGVLALAFSILILALIPLLHTSKQRSMMFRPLSQCLFWALVADLLTLTWIGGQPVEHPYITIGQLASVLYFLLILVLMPTAGTIENKLLKW 1sqi A 2.15 BS02 869 A 1 P239 Q251 H266 F336 F347 E349 F359 N363 F364 P221 Q228 H243 F313 F324 E326 F336 N340 F341 1.13.11.27 0000139,0003868,0005506,0005737,0005783,0005789,0005794,0006559,0006572,0009072,0016020,0016701,0042803,0046872,0051213 ic50<20nM remove_due_to_license_issue P32755 15301540 1501 GPKPERGRFLHFHSVTFWVGNAKQAASFYCNKMGFEPLAYKGLETGSREVVSHVIKQGKIVFVLCSALNPWNKEMGDHLVKHGDGVKDIAFEVEDCEHIVQKARERGAKIVREPWVEEDKFGKVKFAVLQTYGDTTHTLVEKINYTGRFLPGFEAPTYKDTLLPKLPSCNLEIIDHIVGNQPDQEMESASEWYLKNLQFHRFWSVLRSIVVANYEESIKMPINEPASQIQEYVDYNGGAGVQHIALRTEDIITTIRHLRERGMEFLAVPSSYYRLLRENLKTSKIQVKENMDVLEELKILVDYDEKGYLLQIFTKPMQDRPTLFLEVIQRHNHQGFGAGNFNS 1sqn A 1.451 BS01 NDR A 1 L718 L721 Q725 M759 Y890 C891 L35 L38 Q42 M76 Y206 C207 ? Kd=0.4nM remove_due_to_license_issue Kd=0.4nM, Ki=1.9nM, IC50=3.2nM, EC50=2.2nM P06401 15189034 1001 QLIPPLINLLMSIEPDVIYAGHDNPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 1sqo A 1.84 BS01 UI2 A 1 S157 D205 S206 C207 Q208 W231 G232 G234 C235 S145 D192 S193 C194 Q195 W218 G219 G221 C222 H54 D109 Q208 G209 D210 S211 G212 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.035uM remove_due_to_license_issue Ki=32nM P00749 15149645 1001 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1sqp C 2.7 BS03 MYX C 1 L121 F128 Y131 G142 I146 P270 E271 Y273 F274 L120 F127 Y130 G141 I145 P269 E270 Y272 F273 H201 S205 K227 D228 E271 H200 S204 K226 D227 E270 ? 0005739,0005743,0006122,0008121,0009055,0016020,0016491,0020037,0022904,0031966,0045275,0046872,0048039,1902600 remove_due_to_license_issue P00157 15312779 383 TNIRKSHPLMKIVNNAFIDLPAPSNISSWWNFGSLLGICLILQILTGLFLAMHYTSDTTTAFSSVTHICRDVNYGWIIRYMHANGASMFFICLYMHVGRGLYYGSYTFLETWNIGVILLLTVMATAFMGYVLPWGQMSFWGATVITNLLSAIPYIGTNLVEWIWGGFSVDKATLTRFFAFHFILPFIIMAIAMVHLLFLHETGSNNPTGISSDVDKIPFHPYYTIKDILGALLLILALMLLVLFAPDLLGDPDNYTPANPLNTPPHIKPEWYFLFAYAILRSIPNKLGGVLALAFSILILALIPLLHTSKQRSMMFRPLSQCLFWALVADLLTLTWIGGQPVEHPYITIGQLASVLYFLLILVLMPTAGTIENKLLKW 1sqq C 3.0 BS04 OST C 1 F128 Y131 G142 A143 I146 I268 K269 P270 E271 Y273 F274 L294 F127 Y130 G141 A142 I145 I267 K268 P269 E270 Y272 F273 L293 H201 S205 K227 D228 E271 H200 S204 K226 D227 E270 ? 0005739,0005743,0006122,0008121,0009055,0016020,0016491,0020037,0022904,0031966,0045275,0046872,0048039,1902600 remove_due_to_license_issue P00157 15312779 384 TNIRKSHPLMKIVNNAFIDLPAPSNISSWWNFGSLLGICLILQILTGLFLAMHYTSDTTTAFSSVTHICRDVNYGWIIRYMHANGASMFFICLYMHVGRGLYYGSYTFLETWNIGVILLLTVMATAFMGYVLPWGQMSFWGATVITNLLSAIPYIGTNLVEWIWGGFSVDKATLTRFFAFHFILPFIIMAIAMVHLLFLHETGSNNPTGISSDVDKIPFHPYYTIKDILGALLLILALMLLVLFAPDLLGDPDNYTPANPLNTPPHIKPEWYFLFAYAILRSIPNKLGGVLALAFSILILALIPLLHTSKQRSMMFRPLSQCLFWALVADLLTLTWIGGQPVEHPYITIGQLASVLYFLLILVLMPTAGTIENKLLKW 1sqt A 1.9 BS01 UI3 A 1 K141 S144 D191 S192 Q194 W217 G218 G220 C221 K142 S145 D192 S193 Q195 W218 G219 G221 C222 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=0.63uM remove_due_to_license_issue Ki=630nM P00749 15149645 1001 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1sr7 A 1.46 BS01 MOF A 1 L715 L718 N719 L721 Q725 M759 F778 F794 L797 C798 M801 Y890 C891 M909 L32 L35 N36 L38 Q42 M76 F95 F111 L114 C115 M118 Y207 C208 M226 ? Kd=0.08nM remove_due_to_license_issue Kd=0.08nM P06401 15189034 301 QLIPPLINLLMSIEPDVIYAGHDNPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 1sre A 1.78 BS01 HAB A 1 S27 Y43 S45 V47 N49 A50 W79 T90 W108 S13 Y29 S31 V33 N35 A36 W62 T73 W91 ? 0009374 remove_due_to_license_issue P22629 300 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPASGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1srg A 1.8 BS01 MHB B 1 S27 Y43 S45 V47 N49 A50 W79 W108 D128 S13 Y29 S31 V33 N35 A36 W62 W91 D111 ? 0009374 Ka=200000M^-1 remove_due_to_license_issue P22629 300 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPASGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1sri A 1.65 BS01 DMB B 1 S27 Y43 S45 N49 A50 W79 A86 S88 W108 L110 D128 S15 Y31 S33 N37 A38 W64 A71 S73 W93 L95 D113 ? 0009374 Ka=1200000M^-1 remove_due_to_license_issue P22629 300 AEAGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPASGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1sri B 1.65 BS01 DMB A 1 S27 Y43 S45 N49 A50 W79 A86 S88 W108 L110 D128 S15 Y31 S33 N37 A38 W67 A74 S76 W96 L98 D116 ? 0009374 Ka=1200000M^-1 remove_due_to_license_issue P22629 300 AEAGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1ssp E 1.9 BS01 dna A 0 D145 Y147 P168 S169 G246 S247 H268 S270 P271 L272 S273 R276 D64 Y66 P87 S88 G165 S166 H187 S189 P190 L191 S192 R195 3.2.2.27 0004844,0006281,0006284,0016799 remove_due_to_license_issue P13051 9724657 1 ~ 10 MEFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPLSVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 1ssq A 1.85 BS01 CYS A 1 D88 P89 D153 H154 D88 P89 D153 H154 2.3.1.30 0005737,0005829,0006535,0009001,0016740,0016746,0019344 Ki=1uM remove_due_to_license_issue P43886 15147185 2000 MNLDVWQHIRQEAKELAENEPMLASFFHSTILKHQNLGGALSYLLANKLANPIMPAISLREIIEEAYQSNPSIIDCAACDIQAVRHRDPAVELWSTPLLYLKGFHAIQSYRITHYLWNQNRKSLALYLQNQISVAFDVDIHPAAKIGHGIMFDHATGIVVGETSVIENDVSILQGVTLGGTGKESGDRHPKVREGVMIGAGAKILGNIEVGKYAKIGANSVVLNPVPEYATAAGVPARIVS 1stc E 2.3 BS02 STU E 1 L49 G50 V57 A70 M120 Y122 V123 G126 E127 E170 N171 L173 T183 D184 F327 L35 G36 V43 A56 M106 Y108 V109 G112 E113 E156 N157 L159 T169 D170 F313 D166 K168 N171 D184 T201 D152 K154 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=8nM remove_due_to_license_issue P00517 9438863 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1std A 2.9 BS01 BFS A 1 Y50 L76 V108 N131 F158 F162 Y42 L68 V100 N123 F150 F154 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 remove_due_to_license_issue Ki=47nM P56221 7866745 175 DEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFG 1stp A 2.6 BS01 BTN A 1 N23 S27 Y43 S45 V47 N49 W79 S88 T90 W108 D128 N11 S15 Y31 S33 V35 N37 W67 S76 T78 W96 D116 ? 0005576,0009374 remove_due_to_license_issue Kd=1.000000nM P22629 2911722 300 AEAGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKV 1sv3 A 1.35 BS01 ANN A 1 L2 Y22 G30 F106 L2 Y21 G29 F96 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 remove_due_to_license_issue P59071 16596639 347 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 1sve A 2.49 BS02 I01 A 1 G50 T51 G52 F54 V57 A70 K72 L74 Q84 E91 E170 L173 T183 D184 G186 F187 G44 T45 G46 F48 V51 A64 K66 L68 Q78 E85 E164 L167 T177 D178 G180 F181 D166 K168 E170 N171 D184 T201 D160 K162 E164 N165 D178 T195 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=5nM remove_due_to_license_issue IC50=5nM P00517 14998327 351 KKGSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1svg A 2.02 BS02 I04 A 1 G50 T51 G52 S53 F54 V57 A70 K72 L74 Q84 E91 E170 N171 L173 T183 D184 G186 F187 G41 T42 G43 S44 F45 V48 A61 K63 L65 Q75 E82 E161 N162 L164 T174 D175 G177 F178 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=2nM remove_due_to_license_issue IC50=2nM P00517 14998327 351 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1svh A 2.3 BS02 I08 A 1 T51 G52 S53 F54 A70 K72 L74 Q84 E91 E127 E170 N171 L173 T183 D184 G186 F187 T38 G39 S40 F41 A57 K59 L61 Q71 E78 E114 E157 N158 L160 T170 D171 G173 F174 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=360nM remove_due_to_license_issue IC50=360nM P00517 14998327 351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1sw1 A 1.9 BS03 PBE A 1 K13 Y63 T66 D109 Y111 R149 Y190 Y214 K8 Y58 T61 D104 Y106 R144 Y185 Y209 ? 0022857,0043190,0046872,0055085 Kd=50nM remove_due_to_license_issue O29280 15308642 301 ERVVIGSKPFNEQYILANMIAILLEENGYKAEVKEGLGGTLVNYEALKRNDIQLYVEYTGTAYNVILRKQPPELWDQQYIFDEVKKGLLEADGVVVAAKLGFRDDYALAVRADWAEENGVEKISDLAEFADQLVFGSDPEFASRPDGLPQIKKVYGFEFKEVKQMEPTLMYEAIKNKQVDVIPAYTTDSRVDLFNLKILEDDKGALPPYDAIIIVNGNTAKDEKLISVLKLLEDRIDTDTMRALNYQYDVEKKDAREIAMSFLKEQGLVK 1swg A 1.8 BS01 BTN A 1 W79 T90 W108 D128 N23 S27 Y43 W28 T39 W57 D77 N89 S93 Y109 ? 0009374 Kd=43.9nM remove_due_to_license_issue Kd=1.000000nM P22629 9568892 600 SRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKGITGTWYNQLGSTFIVTAGADGALTGTYESA 1swg D 1.8 BS01 BTN D 1 W79 S88 T90 W92 W108 D128 N23 L25 S27 Y43 S45 W29 S38 T40 W42 W58 D78 N91 L93 S95 Y111 S113 ? 0009374 Kd=43.9nM remove_due_to_license_issue Kd=1.000000nM P22629 9568892 900 ESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVGITGTWYNQLGSTFIVTAGADGALTGTYES 1swi C 2.6 BS01 BNZ B 1 L12 A16 L12 A16 ? 0003700,0006355 remove_due_to_license_issue P03069 8646536 100 RMKQLEDKVEELLSKAYHLENEVARLKKLV 1swk A 2.0 BS01 BTN A 1 S27 Y43 S45 V47 G48 N49 F79 A86 S88 T90 W92 W108 D128 S12 Y28 S30 V32 G33 N34 F64 A71 S73 T75 W77 W93 D113 ? 0009374 Ka=100000000000000M^-1 remove_due_to_license_issue Kd=1.000000nM P22629 9636711 5100 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAFKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTK 1swk D 2.0 BS01 BTN D 1 N23 L25 S27 Y43 S45 V47 G48 N49 F79 S88 T90 W92 W108 D128 N8 L10 S12 Y28 S30 V32 G33 N34 F64 S73 T75 W77 W93 D113 ? 0009374 Ka=100000000000000M^-1 remove_due_to_license_issue Kd=1.000000nM P22629 9636711 5400 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAFKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTK 1swn A 2.2 BS01 BTN A 1 S27 S45 V47 W79 F108 S12 S30 V32 W64 F93 ? 0009374 Ka=100000000000000M^-1 remove_due_to_license_issue Kd=1.000000nM P22629 9636711 300 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQFLLTSGTTEANAWKSTLVGHDTFTKVKP 1swn D 2.2 BS01 BTN D 1 S27 Y43 S45 V47 N49 W79 W92 F108 S12 Y28 S30 V32 N34 W64 W77 F93 ? 0009374 Ka=100000000000000M^-1 remove_due_to_license_issue Kd=1.000000nM P22629 9636711 600 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQFLLTSGTTEANAWKSTLVGHDTFTKV 1swp A 2.0 BS01 BTN A 1 L25 S27 Y43 S45 V47 W79 A86 S88 W108 D128 L10 S12 Y28 S30 V32 W64 A71 S73 W93 D113 ? 0009374 Ka=100000000M^-1 remove_due_to_license_issue Kd=1.000000nM P22629 9636711 300 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAFKSTLVGHDTFTK 1swp D 2.0 BS01 BTN D 1 L25 S27 S45 V47 N49 W79 S88 W108 D128 L10 S12 S30 V32 N34 W64 S73 W93 D113 ? 0009374 Ka=100000000M^-1 remove_due_to_license_issue Kd=1.000000nM P22629 9636711 600 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAFKSTLVGHDTFTK 1swr A 1.9 BS01 BTN A 1 N23 L25 S27 Y43 S45 V47 N49 W79 T90 W92 W108 D128 N8 L10 S12 Y28 S30 V32 N34 W64 T75 W77 W93 D113 ? 0009374 Kd=0.12uM remove_due_to_license_issue Kd=1.000000nM P22629 9636711 300 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAAKSTLVGHDTFTK 1swr D 1.9 BS01 BTN D 1 N23 L25 S27 Y43 S45 V47 G48 N49 W79 T90 W92 W108 D128 N8 L10 S12 Y28 S30 V32 G33 N34 W64 T75 W77 W93 D113 ? 0009374 Kd=0.12uM remove_due_to_license_issue Kd=1.000000nM P22629 9636711 600 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAAKSTLVGHDTFTKV 1syh A 1.8 BS01 CPW A 1 E10 Y58 P86 L87 T88 R93 L135 G138 S139 T140 L189 E190 M193 E11 Y59 P87 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 Ki=393nM remove_due_to_license_issue Ki=223nM, EC50=13900nM P19491 15591246 501 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1syi A 2.1 BS01 CPW A 1 Y58 L87 T88 R93 L135 G138 S139 T140 L189 E190 M193 Y59 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 Ki=3330nM remove_due_to_license_issue Ki=223nM, EC50=13900nM P19491 15591246 381 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1syo A 2.2 BS01 M6P A 1 Q348 C385 S386 R391 E416 C419 Y421 Q338 C375 S376 R381 E406 C409 Y411 ? 0005537,0007041,0038023 Kd~1nM remove_due_to_license_issue P08169 15169779 500 AEFPELCSYTWEAVDTKNNMLYKINICGNMGVAQCGPSSAVCMHDLKTDSFHSVGDSLLKTASRSLLEFNTTVNCKQQNHKIQSSITFLCGKTLGTPEFVTATDCVHYFEWRTTAACKKNIFKANKEVPCYAFDRELKKHDLNPLIKTSGAYLVDDSDPDTSLFINVCRDIEVLRASSPQVRVCPTGAAACLVRGDRAFDVGRPQEGLKLVSNDRLVLSYVKEGAGQPDFCDGHSPAVTITFVCPSERREGTIPKLTAKSNCRFEIEWVTEYACHRDYLESRSCSLSSAQHDVAVDLQPLSRDSLFYTSEADEYTYYLSICGGSQAPICNKKDAAVCQVKKADSTQVKVAGRPQNLTLRYSDGDLTLIYFGGEECSSGFQRMSVINFECNQTAGNNGRGAPVFTGEVDCTYFFTWDTKYACV 1syo B 2.2 BS01 M6P B 1 Y1324 Q1348 C1385 S1386 R1391 E1416 C1419 Y1421 Y300 Q324 C361 S362 R367 E392 C395 Y397 ? 0005537,0007041,0038023 Kd~1nM remove_due_to_license_issue P08169 15169779 1500 AEFPELCSYTWEAVDTKNNMLYKINICGNMGVAQCGPSSAVCMHDLKTDSFHSVGDSLLKTASRSLLEFNTTVNIQSSITFLCGKTLGTPEFVTATDCVHYFEWRTTAACKKNIFKANKEVPCYAFDRELKKHDLNPLIKTSGAYLVDDSDPDTSLFINVCRDIEVLRASSPQVRVCPTGAAACLVRGDRAFDVGRPQEGLKLVSNDRLVLSYVKFCDGHSPAVTITFVCPSERREGTIPKLTAKSNCRFEIEWVTEYACHRDYLESRSCSLSSAQHDVAVDLQPLSRVSLFYTSEADEYTYYLSICGGSQAPICNKKDAAVCQVKKADSTQVKVAGRPQNLTLRYSDGDLTLIYFGGEECSSGFQRMSVINFECNQTAGNNGRGAPVFTGEVDCTYFFTWDTKYACV 1sz0 A 2.1 BS01 M6P A 1 Y324 Q348 C385 S386 R391 E416 C419 Y421 Y309 Q333 C370 S371 R376 E401 C404 Y406 ? 0005537,0007041,0038023 Kd~1nM remove_due_to_license_issue P08169 15169779 500 AEFPELCSYTWEAVDTKNNMLYKINICGNMGVAQCGPSSAVCMHDLKTDSFHSVGDSLLKTASRSLLEFNTTVNCKIQSSITFLCGKTLGTPEFVTATDCVHYFEWRTTAACKKNIFKANKEVPCYAFDRELKKHDLNPLIKTSGAYLVDDSDPDTSLFINVCRDIEVLRASSPQVRVCPTGAAACLVRGDRAFDVGRPQEGLKLVSNDRLVLSYVKEGAGQPDFCDGHSPAVTITFVCPSERREGTIPKLTAKSNCRFEIEWVTEYACHRDYLESRSCSLSSAQHDVAVDLQPLSSDSLFYTSEADEYTYYLSICGGSQAPICNKKDAAVCQVKKADSTQVKVAGRPQNLTLRYSDGDLTLIYFGGEECSSGFQRMSVINFECNQTAGNNGRGAPVFTGEVDCTYFFTWDTKYACV 1sz0 B 2.1 BS01 M6P B 1 Y1324 Q1348 C1385 S1386 R1391 E1416 C1419 Y1421 Y308 Q332 C369 S370 R375 E400 C403 Y405 ? 0005537,0007041,0038023 Kd~1nM remove_due_to_license_issue P08169 15169779 1500 AEFPELCSYTWEAVDTKNNMLYKINICGNMGVAQCGPSSAVCMHDLKTDSFHSVGDSLLKTASRSLLEFNTTVNCKKIQSSITFLCGKTLGTPEFVTATDCVHYFEWRTTAACKKNIFKANKEVPCYAFDRELKKHDLNPLIKTSGAYLVDDSDPDTSLFINVCRDIEVLRASSPQVRVCPTGAAACLVRGDRAFDVGRPQEGLKLVSNDRLVLSYVKPDFCDGHSPAVTITFVCPSERREGTIPKLTAKSNCRFEIEWVTEYACHRDYLESRSCSLSSAQHDVAVDLQPLSRVASDSLFYTSEADEYTYYLSICGGSQAPICNKKDAAVCQVKKADSTQVKVAGRPQNLTLRYSDGDLTLIYFGGEECSSGFQRMSVINFECNQTAGNNGRGAPVFTGEVDCTYFFTWDTKYACV 1szd A 1.5 BS03 APR A 1 G32 A33 G34 F44 R45 E64 Q115 F184 G223 T224 S225 V228 N248 L249 Y269 S270 G35 A36 G37 F47 R48 E67 Q118 F187 G221 T222 S223 V226 N246 L247 Y267 S268 P42 D43 F44 R45 N116 D118 H135 P45 D46 F47 R48 N119 D121 H138 2.3.1.286 0017136,0051287,0070403 Kd=29.16uM remove_due_to_license_issue P53686 15150415 1001 MASMSVSTASTEMSVRKIAAHMKSNPNAKVIFMVGAGISTSCGIPDFRSPGTGLYHNLARLKLPYPEAVFDVDFFQSDPLPFYTLAKELYPGNFRPSKFHYLLKLFQDKDVLKRVYTQNIDTLERQAGVKDDLIIEAHGSFAHCHCIGCGKVYPPQVFKSKLAEHPIKDFVKCDVCGELVKPAIVFFGEDLPDSFSETWLNDSEWLREKITTQQPLVIVVGTSLAVYPFASLPEEIPRKVKRVLCNLETVGDFKANKRPTDLIVHQYSDEFAEQLVEELGWQEDFEKILTA 1szm A 2.5 BS01 BI4 A 1 L49 F54 A70 E121 Y122 A123 E170 M173 T183 D184 L35 F40 A56 E107 Y108 A109 E156 M159 T169 D170 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=2.94uM remove_due_to_license_issue P00517 14996846 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPEEIRVSINEKCGKEFSEF 1t13 D 2.9 BS01 INI D 1 W22 G55 A56 Y57 E58 F80 V81 I82 W12 G45 A46 Y47 E48 F70 V71 I72 R88 R78 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P61711 16165152 204 TSFKIAFIQARWHADIVDEARKSFVAELAAKTGGSVEVEIFDVPGAYEIPLHAKTLARTGRYAAIVGAAFVIDGGIYRHDFVATAVINGMMQVQLETEVPVLSVVLTPHHFHESKEHHDFFHAHFKVKGVEAAHAALQIVSERSRIAA 1t13 D 2.9 BS02 INI E 1 L112 S113 L102 S103 R88 R78 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P61711 16165152 201 TSFKIAFIQARWHADIVDEARKSFVAELAAKTGGSVEVEIFDVPGAYEIPLHAKTLARTGRYAAIVGAAFVIDGGIYRHDFVATAVINGMMQVQLETEVPVLSVVLTPHHFHESKEHHDFFHAHFKVKGVEAAHAALQIVSERSRIAA 1t13 E 2.9 BS01 INI A 1 L112 S113 L102 S103 R88 R78 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P61711 16165152 203 TSFKIAFIQARWHADIVDEARKSFVAELAAKTGGSVEVEIFDVPGAYEIPLHAKTLARTGRYAAIVGAAFVIDGGIYRHDFVATAVINGMMQVQLETEVPVLSVVLTPHHFHESKEHHDFFHAHFKVKGVEAAHAALQIVSERSRIAA 1t13 E 2.9 BS02 INI E 1 W22 G55 A56 Y57 E58 F80 V81 I82 W12 G45 A46 Y47 E48 F70 V71 I72 R88 R78 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P61711 16165152 201 TSFKIAFIQARWHADIVDEARKSFVAELAAKTGGSVEVEIFDVPGAYEIPLHAKTLARTGRYAAIVGAAFVIDGGIYRHDFVATAVINGMMQVQLETEVPVLSVVLTPHHFHESKEHHDFFHAHFKVKGVEAAHAALQIVSERSRIAA 1t1r B 2.3 BS02 IMB B 1 K124 D149 S150 E151 W211 M213 E230 P273 M275 K125 D150 S151 E152 W212 M214 E231 P274 M276 1.1.1.267 0008299,0016491,0019288,0030145,0030604,0042802,0046872,0051484,0070402,1990065 ic50=4uM remove_due_to_license_issue IC50=4000nM P45568 15339150 2001 GKQLTILGSTGSIGCSTLDVVRHNPEHFRVVALVAGKNVTRMVEQCLEFSPRYAVMDDEASAKLLKTMLQQQGSRTEVLSGQQAACDMAALEDVDQVMAAIVGAAGLLPTLAAIRAGKTILLANKESLVTCGRLFMDAVKQSKAQLLPVDSEHNAIFQSLPQPIQHNLGYADLEQNGVVSILLTGSGGPFRETPLRDLATMTPDQACRHPNWSMGRKISVDSATMMNKGLEYIEARWLFNASASQMEVLIHPQSVIHSMVRYQDGSVLAQLGEPDMRTPIAHTMAWPNRVNSGVKPLDFCKLSALTFAAPDYDRYPCLKLAMEAFEQGQAATTALNAANEITVAAFLAQQIRFTDIAALNLSVLEKMDMREPQCVDDVLSVDANAREVARKEVMRLAS 1t1s A 2.4 BS03 CBQ A 1 K124 D149 S150 E151 W211 M213 E230 P273 K125 D150 S151 E152 W212 M214 E231 P274 1.1.1.267 0008299,0016491,0019288,0030145,0030604,0042802,0046872,0051484,0070402,1990065 ic50=7uM remove_due_to_license_issue IC50=7000nM P45568 15339150 2001 GKQLTILGSTGSIGCSTLDVVRHNPEHFRVVALVAGKNVTRMVEQCLEFSPRYAVMDDEASAKLLKTMLQQQGSRTEVLSGQQAACDMAALEDVDQVMAAIVGAAGLLPTLAAIRAGKTILLANKESLVTCGRLFMDAVKQSKAQLLPVDSEHNAIFQSLPQPIQHNLGYADLEQNGVVSILLTGSGGPFRETPLRDLATMTPDQACRHPNWSMGRKISVDSATMMNKGLEYIEARWLFNASASQMEVLIHPQSVIHSMVRYQDGSVLAQLGEPDMRTPIAHTMAWPNRVNSGVKPLDFCKLSALTFAAPDYDRYPCLKLAMEAFEQGQAATTALNAANEITVAAFLAQQIRFTDIAALNLSVLEKMDMREPQCVDDVLSVDANAREVARKEVMRLAS 1t2t A 2.5 BS01 dna B 0 R170 G172 N175 F177 N179 H180 K181 H182 I190 S191 M194 K195 K197 K198 P199 N201 I202 K203 C214 A215 A216 R220 T230 Y242 R22 G24 N27 F29 N31 H32 K33 H34 I42 S43 M46 K47 K49 K50 P51 N53 I54 K55 C66 A67 A68 R72 T82 Y94 3.1.-.- 0003677,0004519 remove_due_to_license_issue P13299 15361856 1 ~ 21 KFCKCGVRIQTSAYTCSKCRNRSGENNSFFNHKHSDITKSKISEKMKGKKPSNIKKISCDGVIFDCAADAARHFKISSGLVTYRVKSDKWNWFYIN 1t2t A 2.5 BS02 dna C 0 Q158 A161 Y162 T163 C164 S165 R168 S176 F177 H182 T186 I190 K193 M194 K197 S200 N201 S225 L228 Y231 K237 Q10 A13 Y14 T15 C16 S17 R20 S28 F29 H34 T38 I42 K45 M46 K49 S52 N53 S77 L80 Y83 K89 3.1.-.- 0003677,0004519 remove_due_to_license_issue P13299 15361856 31 ~ 51 KFCKCGVRIQTSAYTCSKCRNRSGENNSFFNHKHSDITKSKISEKMKGKKPSNIKKISCDGVIFDCAADAARHFKISSGLVTYRVKSDKWNWFYIN 1t31 A 1.9 BS02 OHH A 1 K40 H57 A190 F191 K192 G193 S195 S214 Y215 G216 R217 A226 K28 H45 A177 F178 K179 G180 S182 S197 Y198 G199 R200 A207 H57 D102 K192 G193 D194 S195 G196 H45 D89 K179 G180 D181 S182 G183 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 Ki=2.3nM remove_due_to_license_issue Ki=2.3nM, IC50=4.5nM P23946 15741158 901 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPSQKNFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 1t32 A 1.85 BS01 OHH A 1 H57 F172 A190 F191 K192 G193 S195 S214 Y215 G216 E226 H44 F156 A176 F177 K178 G179 S181 S196 Y197 G198 E206 H57 D102 K192 G193 D194 S195 G196 H44 D88 K178 G179 D180 S181 G182 3.4.21.20 0002003,0002548,0004252,0005515,0005576,0005615,0005634,0005737,0005764,0005829,0005886,0006468,0006508,0006935,0006955,0008201,0008233,0008236,0010494,0016020,0016485,0016787,0019221,0019731,0022617,0030141,0030168,0032496,0035578,0035590,0042119,0042742,0048018,0050778,0050829,0050830,0050832,0050868,0051604,0062023,0070062,0070946,0071222,0089720,0098786,1901731 Ki=38nM remove_due_to_license_issue Ki=38nM P08311 15741158 901 IIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRS 1t3t A 1.9 BS07 ADP A 1 T386 G387 Y388 L652 Q668 P676 A678 N722 T394 G395 Y396 L641 Q657 P665 A667 N711 6.3.5.3 0004642,0005524,0005737,0006164,0006189,0016874,0046872 remove_due_to_license_issue P74881 15301531 2005 GLVPRGSHMMEILRGSPALSAFRINKLLARFQAANLQVHNIYAEYVHFADLNAPLNDSEQAQLTRLLQYGPALSSHTPAGKLLLVTPRPGTISPWSSKATDIAHNCGLQQVDRLERGVAYYIEASTLTAEQWRQVAAELHDRMMETVFSSLTDAEKLFIHHQPAPVSSVDLLGEGRQALIDANLRLGLALAEDEIDYLQEAFTKLGRNPNDIELYMFAQANSEHCRHKIFNADWIIDGKPQPKSLFKMIKNTFETTPDYVLSAYKDNAAVMEGSAVGRYFADHNTGRYDFHQEPAHILMKVETHNHPTAISPWPGAATGSGGEIRDEGATGRGAKPKAGLVGFSVSNLRIPGFEQPWEEDFGKPERIVTALDIMTEGPLGGAAFNNEFGRPALTGYFRTYEEKVNSHNGEELRGYHKPIMLAGGIGNIRADHVQKGEIVVGAKLIVLGGPAMNIGFASVQRDNPEMERRCQEVIDRCWQLGDANPILFIHDVGAGGLSNAMPELVSDGGRGGKFELRDILSDEPGMSPLEIWCNESQERYVLAVAADQLPLFDELCKRERAPYAVIGDATEEQHLSLHDNHFDNQPIDLPLDVLLGKTPKMTRDVQTLKAKGDALNRADITIADAVKRVLHLPTVAEKTFLVTIGDRTVTGMVARDQMVGPWQVPVADCAVTTASLDSYYGEAMSIGERAPVALLDFAASARLAVGEALTNIAATQIGDIKRIKLSANWMAAAGHPGEDAGLYDAVKAVGEELCPQLGLTIPVGKDSMSMKTRWQEGNEQREMTSPLSLVISAFARVEDVRHTLTPQLSTEDNALLLIDLGKGHNALGATALAQVYRQLGDKPADVRDVAQLKGFYDAMQALVAARKLLAWHDRSDGGLLVTLAEMAFAGHCGVQVDIAALGDDHLAALFNEELGGVIQVRAEDRDAVEALLAQYGLADCVHYLGQALAGDRFVITANDQTVFSESRTTLRVWWAETTWQMQRLRDNPQCADQEHEAKANDTDPGLNVKLSFDINEDIAAPYIATGARPKVAVLREQGVNSHVEMAAAFHRAGFDAIDVHMSDLLGGRIGLGNFHALVACGGFSYGDVLGAGEGWAKSILFNHRVRDEFETFFHRPQTLALGVCNGCQMMSNLRELIPGSELWPRFVRNHSDRFEARFSLVEVTQSPSLLLQGMVGSQMPIAVSHGEGRVEVRDDAHLAALESKGLVALRYVDNFGKVTETYPANPNGSPNGITAVTTENGRVTIMMPHPERVFRTVANSWHPENWGEDSPWMRIFRNARKQLG 1t46 A 1.6 BS01 STI A 1 L595 A621 K623 E640 L644 V668 T670 Y672 C673 I789 H790 R791 L799 C809 D810 F811 L31 A57 K59 E76 L80 V104 T106 Y108 C109 I153 H154 R155 L163 C173 D174 F175 D792 R796 N797 D810 D156 R160 N161 D174 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=100nM, Kd=15nM, Ki=14nM, EC50=100nM P10721 15123710 3 GNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFLALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISESTN 1t48 A 2.2 BS01 BB3 A 1 A189 L192 N193 F196 E200 E276 F280 W291 K292 A189 L192 N193 F196 E200 E276 F280 W285 K286 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=350uM remove_due_to_license_issue P18031 15258570 299 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGQWKELSHED 1t49 A 1.9 BS01 892 A 1 A189 L192 N193 F196 E200 E276 F280 A189 L192 N193 F196 E200 E276 F280 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=22uM remove_due_to_license_issue P18031 15258570 301 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIM 1t4e A 2.6 BS01 DIZ A 1 G16 L54 G58 I61 M62 V93 H96 Y100 G1 L39 G43 I46 M47 V78 H81 Y85 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue IC50=420nM, Kd=80nM Q00987 15715460 112 GSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 1t4j A 2.7 BS01 FRJ A 1 A189 N193 F196 E200 E276 G277 K279 F280 A189 N193 F196 E200 E276 G277 K279 F280 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue IC50=8000nM P18031 15258570 299 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIM 1t4s A 2.8 BS03 VAL A 1 H126 S137 H141 D183 H121 S132 H136 D178 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 remove_due_to_license_issue P07824 15248756 1000 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTTSSGNLHGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHKPETDYL 1t4v H 2.0 BS03 14A H 1 H79 Y83 W86 I209 D229 A230 C231 S235 W257 G258 E259 H43 Y47 W50 I171 D191 A192 C193 S197 W219 G220 E221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.021uM remove_due_to_license_issue Ki=21nM P00734 15203151 1411 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1t5f A 2.2 BS03 DHH A 1 D124 H126 D128 N130 A141 D183 E186 D232 D119 H121 D123 N125 A136 D178 E181 D227 H101 D124 H126 D128 A141 D232 D234 E277 H96 D119 H121 D123 A136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 Ki=60uM remove_due_to_license_issue P07824 15315440 1000 KPIEIIGAPFSKGCPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLAVIWVDAHTDINTPLTTSSGNLAGQPVAFLLKELKGKFPDVPGFSWVTPAISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSAFGTKREGNHKPETDYL 1t69 A 2.91 BS02 SHH A 1 Y100 H142 H143 G151 F152 D178 H180 F208 Y306 Y81 H123 H124 G132 F133 D159 H161 F189 Y287 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue IC50=243nM, Ki=480nM, Kd=1.2e+3nM Q9BY41 15242608 379 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 1t7j A 2.2 BS01 478 A 1 D25 G27 A28 D30 I50 D25 G27 A28 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.000000064M remove_due_to_license_issue P35963 15771427 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1t7j B 2.2 BS01 478 A 1 D25 G27 A28 D30 I50 T82 D25 G27 A28 D30 I50 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 15771427 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1t8i A 3.0 BS01 dna B 0 V410 T411 W412 I424 Y426 M428 K443 K532 K587 N722 Y723 V210 T211 W212 I224 Y226 M228 K243 K332 K387 N522 Y523 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 1 ~ 10 QKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLNYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1t8i A 3.0 BS02 dna C 0 T313 K324 K328 R634 A635 G717 T718 T113 K124 K128 R434 A435 G517 T518 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 11 ~ 22 QKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLNYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1t8i A 3.0 BS03 dna D 0 E356 F361 R362 G363 R364 H367 K374 R488 A489 N491 K493 T501 K532 D533 N574 T585 A586 K587 N646 E156 F161 R162 G163 R164 H167 K174 R288 A289 N291 K293 T301 K332 D333 N374 T385 A386 K387 N446 5.6.2.1 0003677,0003917,0005694,0006265 remove_due_to_license_issue P11387 15801827 101 ~ 122 QKWKWWEEERYPEGIKWKFLEHKGPVFAPPYEPLPENVKFYYDGKVMKLSPKAEEVATFFAKMLDHEYTTKEIFRKNFFKDWRKEMTNEEKNIITNLSKCDFTQMSQYFKAQTEARKQMSKEEKLKIKEENEKLLKEYGFCIMDNHKERIANFKIEPPGLFRGRGNHPKMGMLKRRIMPEDIIINCSKDAKVPSPPPGHKWKEVRHDNKVTWLVSWTENIQGSIKYIMLNPSSRIKGEKDWQKYETARRLKKCVDKIRNQYREDWKSKEMKVRQRAVALYFIDKLALRAGNEKEEGETADTVGCCSLRVEHINLHPELDGQEYVVEFDFLGKDSIRYYNKVPVEKRVFKNLQLFMENKQPEDDLFDRLNTGILNKHLQDLMEGLTAKVFRTYNASITLQQQLKELTAPDENIPAKILSYNRANRAVAILCNHQRAPPKTFEKSMMNLQTKIDAKKEQLADARRDLKSAKADAKVMKDAKTKKVVESKKKAVQRLEEQLMKLEVQATDREENKQIALGTSKLNYLDPRITVAWCKKWGVPIEKIYNKTQREKFAWAIDMADEDYEF 1t9i A 1.6 BS01 dna C 0 N20 S22 Q26 N30 Q44 T46 Q47 K48 R51 R70 V73 N136 D137 S138 R141 K142 N19 S21 Q25 N29 Q43 T45 Q46 K47 R50 R69 V72 N135 D136 S137 R140 K141 G19 N20 G18 N19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 501 ~ 524 NTKYNKEFLLYLAGFVDGNGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 1t9i A 1.6 BS02 dna D 0 S32 Y33 K34 Q38 R68 R70 E80 I81 D137 K139 S31 Y32 K33 Q37 R67 R69 E79 I80 D136 K138 G19 N20 G18 N19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 551 ~ 574 NTKYNKEFLLYLAGFVDGNGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 1t9i B 1.6 BS01 dna C 0 S332 Y333 K334 Q338 R368 R370 E380 I381 K416 D437 K439 S31 Y32 K33 Q37 R67 R69 E79 I80 K115 D136 K138 G319 N320 G18 N19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 501 ~ 524 NTKYNKEFLLYLAGFVDGNGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDSLS 1t9i B 1.6 BS02 dna D 0 N320 S322 Q326 K328 Q344 T346 Q347 K348 R370 V373 N436 D437 S438 R441 K442 N19 S21 Q25 K27 Q43 T45 Q46 K47 R69 V72 N135 D136 S137 R140 K141 G319 N320 G18 N19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 551 ~ 574 NTKYNKEFLLYLAGFVDGNGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDSLS 1t9j A 2.0 BS01 dna C 0 G19 D20 G21 S22 I24 Q26 Q44 T46 E47 K48 R70 K98 A133 N136 D137 S138 R141 K142 G17 D18 G19 S20 I22 Q24 Q42 T44 E45 K46 R68 K96 A131 N134 D135 S136 R139 K140 G19 D20 G17 D18 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 501 ~ 524 TKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1t9j A 2.0 BS02 dna D 0 S32 Y33 K34 Q38 Y66 R68 R70 E80 I81 K116 D137 K139 S30 Y31 K32 Q36 Y64 R66 R68 E78 I79 K114 D135 K137 G19 D20 G17 D18 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 551 ~ 574 TKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1t9j B 2.0 BS01 dna C 0 S332 Y333 K334 Q338 R368 R370 I381 K416 D437 K439 S30 Y31 K32 Q36 R66 R68 I79 K114 D135 K137 G319 D320 G17 D18 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 501 ~ 524 TKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1t9j B 2.0 BS02 dna D 0 G319 D320 G321 S322 I324 Q326 K328 Q344 T346 E347 K348 R370 K398 N436 D437 S438 R441 K442 G17 D18 G19 S20 I22 Q24 K26 Q42 T44 E45 K46 R68 K96 N134 D135 S136 R139 K140 G319 D320 G17 D18 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15518550 551 ~ 574 TKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1ta2 A 2.3 BS02 176 A 1 H57 Y60A L99 A190 C191 S195 V213 W215 G216 E217 H69 Y73 L122 A218 C219 S223 V243 W245 G246 E247 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=3nM remove_due_to_license_issue Ki=3nM P00734 9703466 401 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1ta6 A 1.9 BS02 177 A 1 H57 Y60A S195 V213 S214 W215 G216 G219 F227 H69 Y73 S223 V243 S244 W245 G246 G248 F257 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=0.74nM remove_due_to_license_issue Ki=0.74nM P00734 9703466 401 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1tbz H 2.3 BS03 00Q H 1 H57 Y60A W60D D189 A190 E192 G193 S195 W215 G216 H43 Y47 W50 D191 A192 E194 G195 S197 W219 G220 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 8913620 343 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1tc1 A 1.41 BS01 FMB A 1 D115 K143 F164 V165 D102 K130 F151 V152 E111 D112 D115 F164 R177 E98 D99 D102 F151 R164 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0046100,0046872,0052657 ic50>2mM remove_due_to_license_issue Q4DRC4 9790669 900 YEFAEKILFTEEEIRTRIKEVAKRIADDYKGKGLRPYVNPLVLISVLKGSFMFTADLCRALCDFNVPVRMEFICVSSYVRMLLDTRHSIEGHHVLIVEDIVDTALTLNYLYHMYFTRRPASLKTVVLLDKREGRRVPFSADYVVANIPNAFVIGYGLDYDDTYRELRDIVVLRPE 1tcw A 2.4 BS01 IM1 A 1 D29 D30 I32 V47 G48 G49 D29 D30 I32 V47 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=960nM remove_due_to_license_issue P05896 8756683 400 PQFSLWRRPVVTAHIEGQPVEVLLDTGADDSIVTGIELGPHYTPKIVGGIGGFINTKEYKNVKIEVLGKRIKGTIMTGDTPINIFGRNLLTALGMSLNL 1tcw B 2.4 BS01 IM1 A 1 R8 I50 R8 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=960nM remove_due_to_license_issue P05896 8756683 400 PQFSLWRRPVVTAHIEGQPVEVLLDTGADDSIVTGIELGPHYTPKIVGGIGGFINTKEYKNVKIEVLGKRIKGTIMTGDTPINIFGRNLLTALGMSLNL 1tcw B 2.4 BS02 IM1 B 1 A28 D29 G48 A28 D29 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=960nM remove_due_to_license_issue P05896 8756683 600 PQFSLWRRPVVTAHIEGQPVEVLLDTGADDSIVTGIELGPHYTPKIVGGIGGFINTKEYKNVKIEVLGKRIKGTIMTGDTPINIFGRNLLTALGMSLNL 1tcx A 2.3 BS01 IM1 A 1 D25 G27 D29 G48 I82 D25 G27 D29 G48 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=112nM remove_due_to_license_issue P04587 8756683 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTILEEMSLPGRWKPKMVGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 1tcx B 2.3 BS01 IM1 A 1 D25 G27 G49 D25 G27 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 8756683 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTILEEMSLPGRWKPKMVGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 1td7 A 2.5 BS02 NFL A 1 L2 F5 I9 W19 F22 G30 Y64 F101 L2 F5 I9 W18 F21 G29 Y63 F100 Y28 G30 G32 H48 D49 Y52 Y68 D94 Y27 G29 G31 H47 D48 Y51 Y67 D93 3.1.1.4 0004623,0005102,0005509,0005543,0005576,0006633,0006644,0016042,0016787,0046872,0047498,0047499,0048146,0050482 Kd=43uM remove_due_to_license_issue P60045 16301791 2001 NLYQFKNMIQCTVPSRSWQDFADYGCYCGKGGSGTPVDDLDRCCQVHDNCYNEAENISGCRPYFKTYSYECTQGTLTCKGDNNACAASVCDCDRLAAICFAGAPYNDANYNIDLKARCN 1tdz A 1.8 BS01 dna B 0 E2 E5 K57 H72 R74 M75 K129 G170 N171 I172 S217 I219 Y238 K254 K256 R260 E1 E4 K56 H71 R73 M74 K128 G169 N170 I171 S216 I218 Y232 K248 K250 R254 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 15249553 1 ~ 14 ELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSILGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1tdz A 1.8 BS02 dna C 0 K90 H91 V108 R109 K110 F111 K154 K89 H90 V107 R108 K109 F110 K153 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 15249553 15 ~ 28 ELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSILGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1tfq A -1.00 BS02 998 A 1 K297 G306 L307 T308 D309 K311 Q319 K58 G67 L68 T69 D70 K72 Q80 2.3.2.27 remove_due_to_license_issue P98170 15317454 998 MSDAVSSDRNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVRTT 1tft A -1.00 BS02 997 A 1 K297 G306 L307 T308 D309 K311 Q319 W323 K58 G67 L68 T69 D70 K72 Q80 W84 2.3.2.27 remove_due_to_license_issue Kd=5.0nM P98170 15317454 998 MSDAVSSDRNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVRTT 1tfz A 1.8 BS02 869 A 1 H205 P259 H287 M314 F360 F398 G399 N402 F403 H184 P227 H252 M279 F325 F354 G355 N358 F359 1.13.11.27 0003868,0005506,0005737,0006559,0006572,0009072,0016701,0042802,0046872,0051213 ic50=7nM remove_due_to_license_issue P93836 15301540 551 NPKSDKFKVKRFHHIEFWCGDATNVARRFSWGLGMRFSAKSDLSTGNMVHASYLLTSGDLRFLFTAPYSPSLSAGEIKPTTTASIPSFDHGSCRSFFSSHGLGVRAVAIEVEDAESAFSISVANGAIPSSPPIVLNEAVTIAEVKLYGDVVLRYVSYKEFLPGFERVEDASSFPLDYGIRRLDHAVGNVPELGPALTYVAGFTGFHQFASGLNSAVLASNDEMVLLPINEPVHGKSQIQTYLEHNEGAGLQHLALMSEDIFRTLREMRKRSSIGGFDFMPSPPPTYYQNLKKRVGDVLSDDQIKECEELGILVDRDDQGTLLQIFTKPLGDRPTIFIEIIQRVGCMQSGGCGGFGKGNFSELFK 1tg5 A 1.9 BS02 645 A 1 L244 P259 H287 F360 F371 E373 F398 G399 K400 N402 F403 L406 L216 P231 H257 F330 F341 E343 F359 G360 K361 N363 F364 L367 1.13.11.27 0003868,0005506,0005737,0006559,0006572,0009072,0016701,0042802,0046872,0051213 ic50=12nM remove_due_to_license_issue P93836 15301540 501 KNPKSDKFKVKRFHHIEFWCGDATNVARRFSWGLGMRFSAKSDLSTGNMVHASYLLTSGDLRFLFTAPYSPSLSAGEIKPTTTASIPSFDHGSCRSFFSSHGLGVRAVAIEVEDAESAFSISVANGAIPSSPPIVLNEAVTIAEVKLYGDVVLRYVSYKASEFLPGFERVEDASSFPLDYGIRRLDHAVGNVPELGPALTYVAGFTGFHQFAESGLNSAVLASNDEMVLLPINEPVHGTKSQIQTYLEHNEGAGLQHLALMSEDIFRTLREMRKRSSIGGFDFMPSPPPTYYQNLKKRVGDVLSDDQIKECEELGILVDRDDQGTLLQIFTKPLGDRPTIFIEIIQRVGCYQSGGCGGFGKGNFSELFKSI 1thl A 1.7 BS06 0DB A 1 N111 N112 A113 F130 V139 H142 E143 H146 E166 R203 H231 N111 N112 A113 F130 V139 H142 E143 H146 E166 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=0.38uM remove_due_to_license_issue P00800 8286362 320 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1thz A 1.8 BS01 326 A 1 K267 F316 K484 A486 E487 N490 K264 F313 K481 A483 E484 N487 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=7.1uM remove_due_to_license_issue P31335 15355974 4001 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1thz A 1.8 BS02 326 B 1 S451 R452 F542 P544 F545 S448 R449 F539 P541 F542 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=7.1uM remove_due_to_license_issue P31335 15355974 3001 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1thz B 1.8 BS01 326 A 1 S451 R452 P544 F545 S448 R449 P541 F542 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=7.1uM remove_due_to_license_issue P31335 15355974 4001 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1thz B 1.8 BS02 326 B 1 K267 F316 K484 A486 N490 K264 F313 K481 A483 N487 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=7.1uM remove_due_to_license_issue P31335 15355974 3001 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 1tjp A 1.5 BS01 HPF A 1 E49 D60 I64 L100 Y175 T183 G184 F212 G213 G234 S235 E49 D60 I64 L100 Y175 T183 G184 F212 G213 G234 S235 E49 D60 Y175 E49 D60 Y175 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 remove_due_to_license_issue P00929 16120446 1001 MERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGALPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 1tka A 2.7 BS02 N3T A 1 H69 G116 P117 L118 D157 G158 N187 I189 T190 I191 H263 H67 G114 P115 L116 D155 G156 N185 I187 T188 I189 H261 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tka A 2.7 BS03 N3T B 1 D382 E418 F445 Y448 D380 E416 F443 Y446 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tka B 2.7 BS01 N3T A 1 D382 I416 F445 Y448 H481 D380 I414 F443 Y446 H479 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tka B 2.7 BS03 N3T B 1 H69 L118 N187 I189 T190 I191 H263 H67 L116 N185 I187 T188 I189 H261 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkb A 2.3 BS02 N1T A 1 H69 L118 D157 G158 N187 I189 T190 I191 H263 H67 L116 D155 G156 N185 I187 T188 I189 H261 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 Kd=0.000000064M remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkb A 2.3 BS03 N1T B 1 D382 F445 Y448 D380 F443 Y446 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 Kd=0.000000064M remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkb B 2.3 BS01 N1T A 1 D382 I416 Y448 D380 I414 Y446 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 Kd=0.000000064M remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkb B 2.3 BS03 N1T B 1 H69 L118 D157 N187 I189 T190 I191 H263 H67 L116 D155 N185 I187 T188 I189 H261 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 Kd=0.000000064M remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkc A 2.7 BS02 M6T A 1 H69 G116 L118 D157 G158 N187 I189 T190 I191 H263 H67 G114 L116 D155 G156 N185 I187 T188 I189 H261 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkc A 2.7 BS03 M6T B 1 D382 L383 E418 F445 Y448 D380 L381 E416 F443 Y446 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkc B 2.7 BS01 M6T A 1 I416 E418 F445 Y448 I414 E416 F443 Y446 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkc B 2.7 BS03 M6T B 1 H69 P117 L118 G158 N187 I189 T190 I191 H263 H67 P115 L116 G156 N185 I187 T188 I189 H261 H30 I250 H263 E418 H481 H28 I248 H261 E416 H479 2.2.1.1 0003824,0004802,0005515,0005737,0005829,0006098,0016740,0046872 remove_due_to_license_issue P23254 8144674 681 QFTDIDKLAVSTIRILAVDTVSKANSGHPGAPLGMAPAAHVLWSQMRMNPTNPDWINRDRFVLSNGHAVALLYSMLHLTGYDLSIEDLKQFRQLGSRTPGHPEFELPGVEVTTGPLGQGISNAVGMAMAQANLAATYNKPGFTLSDNYTYVFLGDGCLQEGISSEASSLAGHLKLGNLIAIYDDNKITIDGATSISFDEDVAKRYEAYGWEVLYVENGNEDLAGIAKAIAQAKLSKDKPTLIKMTTTIGYGSLHAGSHSVHGAPLKADDVKQLKSKFGFNPDKSFVVPQEVYDHYQKTILKPGVEANNKWNKLFSEYQKKFPELGAELARRLSGQLPANWESKLPTYTAKDSAVATRKLSETVLEDVYNQLPELIGGSADLTPSNLTRWKEALDFQPPSSGSGNYSGRYIRYGIREHAMGAIMNGISAFGANYKPYGGTFLNFVSYAAGAVRLSALSGHPVIWVATHDSIGVGEDGPTHQPIETLAHFRSLPNIQVWRPADGNEVSAAYKNSLESKHTPSIIALSRQNLPQLEGSSIESASKGGYVLQDVANPDIILVATGSEVSLSVEAAKTLAAKNIKARVVSLPDFFTFDKQPLEYRLSVLPDNVPIMSVEVLATTCWGKYAHQSFGIDRFGASGKAPEVFKFFGFTPEGVAERAQKTIAFYKGDKLISPLKKAF 1tkt A 2.6 BS01 H12 A 1 L100 K101 V106 V179 Y181 Y188 L234 H235 P236 Y318 L90 K91 V96 V169 Y171 Y178 L224 H225 P226 Y308 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 15537346 999 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVP 1tkx A 2.85 BS01 GWB A 1 L100 K101 V179 Y181 Y188 W229 L234 Y318 L96 K97 V175 Y177 Y184 W225 L230 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 15537347 999 SPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAH 1tkz A 2.81 BS01 H16 A 1 L100 K101 Y181 Y188 L234 H235 P236 Y318 L91 K92 Y172 Y179 L225 H226 P227 Y309 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 15537346 999 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVP 1tl1 A 2.9 BS01 H18 A 1 L100 K101 V179 Y181 Y188 F227 W229 L234 H235 P236 Y318 L91 K92 V170 Y172 Y179 F218 W220 L225 H226 P227 Y309 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 15537346 999 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVP 1tl3 A 2.8 BS01 H20 A 1 L100 K101 K103 V179 Y181 Y188 W229 L234 H235 P236 Y318 L91 K92 K94 V170 Y172 Y179 W220 L225 H226 P227 Y309 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 15537346 999 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVP 1tl7 A 2.8 BS04 ONM A 1 D396 G399 F400 T401 A409 L412 L438 G439 D440 D20 G23 F24 T25 A33 L36 L62 G63 D64 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P30803 15591060 100 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1tl7 B 2.8 BS02 ONM A 1 K938 D1018 I1019 W1020 G1021 N1022 N1025 K60 D130 I131 W132 G133 N134 N137 S891 I892 S942 R1029 K1065 S13 I14 S64 R141 K177 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P26769 15591060 100 HQSYDCVCVMFASIPDFKEFYTESDVNKEGLECLRLLNEIIADFDDLLSKPKFSGVEKIKTIGSTYMAATGLSAIRQYMHIGTMVEFAYALVGKLDAINKHSFNDFKLRVGINHGPVIAGVIGAQKPQYDIWGNTVNVASRMDSTGVLDKIQVTEETSLILQTLGYTCTCRGIINVKGKGDLKTYFVNT 1tlo A 1.9 BS03 E64 A 1 Q109 G113 C115 W116 G208 C209 E212 S251 G271 H272 Q77 G81 C83 W84 G176 C177 E180 S219 G239 H240 Q109 C115 H272 N296 W298 Q77 C83 H240 N264 W266 3.4.22.52 0004198,0006508 remove_due_to_license_issue P97571 15491615 400 NAIKYLGQDYENLRARCLQNGVLFQDDAFPPVSHSLGFKELGPNSSKTYGIKWKRPTELLSNPQFIVDGATRTDICQGALGDCWLLAAIASLTLNETILHRVVPYGQSFQEGYAGIFHFQLWQFGEWVDVVVDDLLPTKDGKLVFVHSAQGNEFWSALLEKAYAKVNGSYEALSGGCTSEAFEDFTGGVTEWYDLQKAPSDLYQIILKALERGSLLGCSINISDIRDLEAITFKNLVRGHAYSVTDAKQVTYQGQRVNLIRMRNPWGEVEWKGPWSDNSYEWNKVDPYEREQLRVKMEDGEFWMSFRDFIREFTKLEICNLT 1tlp E 2.3 BS01 RDF E 1 N111 N112 A113 E143 H146 Y157 E166 R203 H231 N111 N112 A113 E143 H146 Y157 E166 R203 H231 3.4.24.27 0004222,0006508 Ki=28nM remove_due_to_license_issue Kd=28nM, IC50=33nM, Ki=28nM P00800 3709536 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1tmm A 1.25 BS04 APC A 1 Q74 R82 K85 A86 D95 D97 I98 R110 L111 T112 H115 Y116 R121 Q74 R82 K85 A86 D95 D97 I98 R110 L111 T112 H115 Y116 R121 R82 R92 D95 D97 R82 R92 D95 D97 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=0.23uM remove_due_to_license_issue P26281 15952765 171 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERAGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 1tmn E 1.9 BS01 0ZN E 1 Y110 N112 A113 H142 E143 H146 E166 L202 R203 H231 Y110 N112 A113 H142 E143 H146 E166 L202 R203 H231 3.4.24.27 0004222,0006508 Ki=50nM remove_due_to_license_issue P00800 6395881 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1tng A 1.8 BS02 AMC A 1 D189 S190 V213 G219 D171 S172 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.17mM remove_due_to_license_issue P00760 7634078 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tnh A 1.8 BS02 FBA A 1 D189 S190 C191 V213 W215 G219 D171 S172 C173 V191 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.43mM remove_due_to_license_issue P00760 7634078 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tni A 1.9 BS02 PBN A 1 D189 S190 C191 Q192 W215 G216 G219 C220 D171 S172 C173 Q174 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.1mM remove_due_to_license_issue P00760 7634078 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tnj A 1.8 BS02 PEA A 1 D189 S190 G216 G219 G226 D171 S172 G194 G196 G204 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=11mM remove_due_to_license_issue P00760 7634078 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tnk A 1.8 BS02 PRA A 1 D189 S190 C191 S195 V213 W215 G216 G219 D171 S172 C173 S177 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=32.5mM remove_due_to_license_issue P00760 7634078 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tnl A 1.9 BS02 TPA A 1 D189 S190 C191 Q192 V213 W215 G216 G219 D171 S172 C173 Q174 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=13.3mM remove_due_to_license_issue P00760 7634078 900 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tog A 2.31 BS01 HCI A 1 L18 I37 W140 X258 R386 L14 I33 W130 X246 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=0.6mM remove_due_to_license_issue P00509 15461450 410 MFENITATTADPILGLADLFRADERPGKIDLGIGVYKDETGKTPVLTSVKKAEQYLLENETTKNYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFALYNERVGACTLVAADSETVDRAFGQMKAAIRDNYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1tog B 2.31 BS01 HCI A 1 Y70 S296 Y65 S284 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=0.6mM remove_due_to_license_issue P00509 15461450 410 MFENITATTADPILGLADLFRADERPGKIDLGIGVYKDETGKTPVLTSVKKAEQYLLENETTKNYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFALYNERVGACTLVAADSETVDRAFGQMKAAIRDNYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1tog B 2.31 BS02 HCI B 1 L18 I37 G38 W140 X258 R386 L14 I33 G34 W130 X246 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=0.6mM remove_due_to_license_issue P00509 15461450 410 MFENITATTADPILGLADLFRADERPGKIDLGIGVYKDETGKTPVLTSVKKAEQYLLENETTKNYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFALYNERVGACTLVAADSETVDRAFGQMKAAIRDNYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1toi A 1.9 BS01 HCI A 1 G38 W140 X258 R386 G34 W130 X246 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=0.09mM remove_due_to_license_issue P00509 15461450 410 MFENITAAPADPILGLADLFRADERPGKINLGIGLYYDETGKIPVLTSVKKAEQYLLENETTKLYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFGLYNERVGACTLVAADSETVDRAFSQMKAAIRDNYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1toj A 1.9 BS01 HCI A 1 I17 L18 I37 G38 W140 X258 R386 I13 L14 I33 G34 W130 X246 R374 W140 D222 A224 K258 W130 D211 A213 K246 2.6.1.1 0003824,0004069,0004838,0005737,0005829,0006520,0008483,0009058,0009094,0030170,0033585,0042802,0042803 Kd=0.41mM remove_due_to_license_issue P00509 15461450 410 MFENITATTADPILGLADLFRADERPGKIDLGIGVYKDETGKTPVLTSVKKAEQYLLENETTKNYLGIDGIPEFGRCTQELLFGKGSALINDKRARTAQTPGGSGALRVAADFLAKNTSVKRVWVSNPSWPNHKSVFNSAGLEVREYAYYDAENHTLDFDALINSLNEAQAGDVVLFHGCCHNPTGIDPTLEQWQTLAQLSVEKGWLPLFDFAYQGFARGLEEDAEGLRAFAAMHKELIVASSYSKNFALYNERVGACTLVAADSETVDRAFGQMKAAIRANYSSPPAHGASVVATILSNDALRAIWEQELTDMRQRIQRMRQLFVNTLQEKGANRDFSFIIKQNGMFSFSGLTKEQVLRLREEFGVYAVASGRVNVAGMTPDNMAPLCEAIVAVL 1tom H 1.8 BS03 MIN H 1 Y60A W60D N98 L99 I174 A190 C191 W215 G216 G219 Y47 W50 N95 L96 I171 A192 C193 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 Ki=5nM remove_due_to_license_issue Ki=5nM, IC50=6nM P00734 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1tou A 2.0 BS01 B1V A 1 M20 A75 D76 R78 I104 C117 R126 Y128 M20 A75 D76 R78 I104 C117 R126 Y128 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 ic50=1uM remove_due_to_license_issue P15090 15357970 501 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 1tow A 2.0 BS01 CRZ A 1 F16 F57 D76 C117 R126 Y128 F16 F57 D76 C117 R126 Y128 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 ic50=0.57uM remove_due_to_license_issue IC50=570.0nM P15090 15357969 501 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 1tpw A 1.9 BS01 PGH A 1 K13 H95 E165 I170 G171 G210 S211 L230 G232 K10 H92 E162 I167 G168 G207 S208 L227 G229 N11 K13 H95 E97 E165 G171 S211 N8 K10 H92 E94 E162 G168 S208 4.2.3.3,5.3.1.1 0004807,0005737,0005829,0006006,0006094,0006096,0008929,0016829,0016853,0019242,0019563,0019682,0031625,0042803,0046166,0061621 Ki=0.5mM remove_due_to_license_issue P00940 10194358 250 RKFFVGGNWKMNGDKKSLGELIHTLNGAKLSADTEVVCGAPSIYLDFARQKLDAKIGVAAQNCYKVPKGAFTGEISPAMIKDIGAAWVILGHPERRHVFGESDELIGQKVAHALAEGLGVIACIGEKLDEREAGITEKVVFEQTKAIADNVKDWSKVVLAYEPVWAIGTGKTATPQQAQEVHEKLRGWLKTHVSDAVAQSTRIIYGGSVTGGNCKELASQHDVDGFLVGGASLKPEFVDIINAKH 1tpw B 1.9 BS01 PGH B 1 N11 K13 H95 E165 I170 G171 G210 S211 L230 G232 G233 N8 K10 H92 E162 I167 G168 G207 S208 L227 G229 G230 N11 K13 H95 E97 E165 G171 S211 N8 K10 H92 E94 E162 G168 S208 4.2.3.3,5.3.1.1 0004807,0005737,0005829,0006006,0006094,0006096,0008929,0016829,0016853,0019242,0019563,0019682,0031625,0042803,0046166,0061621 Ki=0.5mM remove_due_to_license_issue P00940 10194358 250 RKFFVGGNWKMNGDKKSLGELIHTLNGAKLSADTEVVCGAPSIYLDFARQKLDAKIGVAAQNCYKVPKGAFTGEISPAMIKDIGAAWVILGHPERRHVFGESDELIGQKVAHALAEGLGVIACIGEKLDEREAGITEKVVFEQTKAIADNVKDWSKVVLAYEPVWAIGTGKTATPQQAQEVHEKLRGWLKTHVSDAVAQSTRIIYGGSVTGGNCKELASQHDVDGFLVGGASLKPEFVDIINAKH 1tpz A 2.0 BS01 GDP A 1 G79 G81 K82 S83 S84 T102 G103 K184 D186 S231 N232 K233 G66 G68 K69 S70 S71 T89 G90 K171 D173 S211 N212 K213 3.6.5.- 0003924,0005515,0005525,0005634,0005737,0005783,0005789,0005794,0009617,0010506,0016020,0016787,0019003,0019221,0020005,0031965,0032580,0035458,0042802,0042832,0045087,0050829,1990606 Kd=0.64uM remove_due_to_license_issue Q9QZ85 15350217 1500 NDLPSSFTGYFKKFNTGRKIISQEILNLIELRMRKGNIQLTNSAISDALKEIDSSVLNVAVTGETGSGKSSFINTLRGIGNEEEGAAKTGVVEVTMERHPYKHPNIPNVVFWDLPGIGSTNFPPDTYLEKMKFYEYDFFIIISATRFKKNDIDIAKAISMMKKEFYFVRTKVDSDITNEADKEKVLQDIRLNCVNTFRENGIAEPPIFLLSNKNVCHYDFPVLMDKLISDLPIYKRHNFMVSLPNITDSVIEKKRQFLKQRIWLEGFAADLVNIIPSLTFLLDSDLETLKKSMKFYRTVFGVDETSLQRLARDWEIEVDQVEAMIKSPAVFKPTDEETIQERLSRYIQEFCLANGYLLPKNSFLKEIFYLKYYFLDMVTEDAKTLLKEICLKLGR 1tq4 A 1.95 BS01 GDP A 1 G79 G81 K82 S83 S84 T102 K184 D186 S231 N232 K233 G66 G68 K69 S70 S71 T89 K167 D169 S214 N215 K216 3.6.5.- 0003924,0005515,0005525,0005634,0005737,0005783,0005789,0005794,0009617,0010506,0016020,0016787,0019003,0019221,0020005,0031965,0032580,0035458,0042802,0042832,0045087,0050829,1990606 Kd=0.64uM remove_due_to_license_issue Q9QZ85 15350217 500 NDLPSSFTGYFKKFNTGRKIISQEILNLIELRMRAGNIQLTNSAISDALKEIDSSVLNVAVTGETGSGKSSFINTLRGIGNEEEGAAKTGVMERHPYKHPNIPNVVFWDLPGIGSTNFPPDTYLEKMKFYEYDFFIIISATRFKKNDIDIAKAISMMKKEFYFVRTKVDSDITNEADGEPQTFDKEKVLQDIRLNCVNTFRENGIAEPPIFLLSNKNVCHYDFPVLMDKLISDLPIYKRHNFMVSLPNITDSVIEKKRQFLKQRIWLEGFAADLVNIIPSLTFLLDSDLETLKKSMKFYRTVFGVDETSLQRLARDWEIEVDQVEAMIKSPAVFKPTDEETIQERLSRYIQEFCLANGYLLPKNSFLKEIFYLKYYFLDMVTEDAKTLLKEICLRN 1tqe P 2.7 BS01 dna C 0 G2 R3 K4 I6 K23 R24 K30 G1 R2 K3 I5 K22 R23 K29 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe P 2.7 BS02 dna D 0 G2 R3 K5 R15 K31 G1 R2 K4 R14 K30 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe Q 2.7 BS01 dna C 0 G2 R3 Q18 K31 G1 R2 Q17 K30 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe Q 2.7 BS02 dna D 0 G2 R3 K4 I6 K23 R24 K30 G1 R2 K3 I5 K22 R23 K29 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe R 2.7 BS01 dna E 0 G2 R3 K4 I6 K23 R24 K30 G1 R2 K3 I5 K22 R23 K29 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe R 2.7 BS02 dna F 0 G2 R3 K5 K31 G1 R2 K4 K30 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe S 2.7 BS01 dna E 0 G2 R3 K31 G1 R2 K30 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqe S 2.7 BS02 dna F 0 G2 R3 I6 K23 R24 K30 G1 R2 I5 K22 R23 K29 ? 0000977,0003677,0045944,0046983 remove_due_to_license_issue Q02080 15567413 1 ~ 17 GRKKIQISRILDQRNRQVTFTKRKFGLMKKAYELSVLCDCEIALIIFNSANRLFQYASTDMDRVLLKYTEYSEPHESRTNTDILETLKRR 1tqf A 1.8 BS01 32P A 1 Q12 G13 L30 Y71 T72 Q73 F108 S229 G230 T231 T232 N233 R235 A335 Q16 G17 L34 Y75 T76 Q77 F112 S220 G221 T222 T223 N224 R226 A321 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=1.4uM remove_due_to_license_issue IC50=1400nM P56817 15566281 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 1tr7 B 2.1 BS01 DEG B 1 F1 I13 N46 D47 D54 N135 D140 F1 I13 N46 D47 D54 N135 D140 ? 0007155,0009289 Kd=0.15uM remove_due_to_license_issue P08191 15659162 502 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 1trd B 2.5 BS01 PGH B 1 H95 E167 S213 L232 G234 H94 E166 S212 L231 G233 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=4uM remove_due_to_license_issue P04789 8356028 300 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 1tsi A 2.84 BS01 4PB A 1 K13 H95 I172 G211 K12 H94 I171 G210 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 remove_due_to_license_issue P04789 1304889 600 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVRGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 1tsl A 2.5 BS01 A15 A 1 T24 E84 W85 E88 H106 V316 T24 E84 W85 E88 H106 V316 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Ki=0.7uM remove_due_to_license_issue Ki=700nM P00469 9931028 318 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1tsm A 3.0 BS01 MR2 A 1 W82 E84 W85 L195 W82 E84 W85 L195 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue P00469 9931028 318 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1tsv A 2.9 BS01 UMP A 1 R23 L195 C198 H199 R218 S219 A220 D221 G225 N229 H259 Y261 R23 L195 C198 H199 R218 S219 A220 D221 G225 N229 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue P00469 9053905 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRALIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1tsy A 2.2 BS01 UMP A 1 R23 L195 C198 H199 Q217 R218 S219 A220 D221 N229 H259 Y261 R23 L195 C198 H199 Q217 R218 S219 A220 D221 N229 H259 Y261 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Kd=11uM remove_due_to_license_issue P00469 9053905 317 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRKLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKAPVAV 1tt1 A 1.93 BS01 KAI A 1 Y61 P89 A91 R96 G141 A142 T143 E191 Y59 P87 A89 R94 G139 A140 T141 E189 ? 0015276,0016020 Ki=64.6nM remove_due_to_license_issue Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 15721240 998 NRSLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWWR 1ttm A 1.95 BS02 667 A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=45nM remove_due_to_license_issue IC50=25nM, Ki=21nM, Kd=45nM P00918 15453828 264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1ttv A -1.00 BS01 IMY A 1 L50 L53 G54 I57 Q68 H69 V89 H92 L38 L41 G42 I45 Q56 H57 V77 H80 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue P56273 15557803 120 NHISTSDQEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVSANVKESSEDIFGNV 1tu6 A 1.75 BS01 FSP A 1 Q133 G137 C139 G178 G179 G180 Y181 A248 N275 H276 Q19 G23 C25 G64 G65 G66 Y67 A134 N161 H162 Q133 C139 H276 N296 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=0.832nM P43235 15341947 551 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1tu6 B 1.75 BS01 FSP A 1 N132 Q135 V204 G205 N18 Q21 V90 G91 Q133 C139 H276 N296 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=0.832nM P43235 15341947 551 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1tu6 B 1.75 BS02 FSP B 1 Q133 C136 G137 C139 G178 G179 G180 A248 N275 H276 Q19 C22 G23 C25 G64 G65 G66 A134 N161 H162 Q133 C139 H276 N296 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=0.832nM P43235 15341947 561 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1tuf A 2.4 BS01 AZ1 A 1 S227 R307 R343 Y347 S213 R293 R329 Y333 K83 H224 E304 K69 H210 E290 4.1.1.20 0003824,0008836,0009085,0009089,0016831,0030170 Ki=89uM remove_due_to_license_issue Q58497 12429091 502 FLGNDTVEIKDGRFFIDGYDAIELAEKFGTPLYVMSEEQIKINYNRYIEAFKRWEEETGKEFIVAYAYKANANLAITRLLAKLGCGADVVSGGELYIAKLSNVPSKKIVFNGNCKTKEEIIMGIEANIRAFNVDSISELILINETAKELGETANVAFRINPNVNPKTHPKISTGLKKNKFGLDVESGIAMKAIKMALEMEYVNVVGVHCHIGSQLTDISPFIEETRKVMDFVVELKEEGIEIEDVNLGGGLGIPYYKDKQIPTQKDLADAIINTMLKYKDKVEMPNLILEPGRSLVATAGYLLGKVHHIKETPVTKWVMIDAGMNDMMRPAMYEAYHHIINCKVKNEKEVVSIAGGLCESSDVFGRDRELDKVEVGDVLAIFDVGAYGISMANNYNARGRPRMVLTSKKGVFLIRERETYADLIAKDIVPPHLL 1tuf B 2.4 BS01 AZ1 B 1 R307 R343 Y347 R293 R329 Y333 K83 H224 E304 K69 H210 E290 4.1.1.20 0003824,0008836,0009085,0009089,0016831,0030170 Ki=89uM remove_due_to_license_issue Q58497 12429091 503 FLGNDTVEIKDGRFFIDGYDAIELAEKFGTPLYVMSEEQIKINYNRYIEAFKRWEEETGKEFIVAYAYKANANLAITRLLAKLGCGADVVSGGELYIAKLSNVPSKKIVFNGNCKTKEEIIMGIEANIRAFNVDSISELILINETAKELGETANVAFRINPNVNPKTHPKISTGLKKNKFGLDVESGIAMKAIKMALEMEYVNVVGVHCHIGSQLTDISPFIEETRKVMDFVVELKEEGIEIEDVNLGGGLGIPYYKDKQIPTQKDLADAIINTMLKYKDKVEMPNLILEPGRSLVATAGYLLGKVHHIKETPVTKWVMIDAGMNDMMRPAMYEAYHHIINCKVKNEKEVVSIAGGLCESSDVFGRDRELDKVEVGDVLAIFDVGAYGISMANNYNARGRPRMVLTSKKGVFLIRERETYADLIAKDIVPPHLL 1tv6 A 2.8 BS01 CP9 A 1 L100 V106 V108 Y181 Y188 P225 L234 H235 P236 Y318 L100 V106 V108 Y181 Y188 P221 L230 H231 P232 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 15249669 561 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAH 1tve A 3.0 BS01 178 A 1 S94 K117 T176 D214 D219 S93 K116 T175 D213 D218 D219 K223 D218 K222 1.1.1.3 0004412,0005634,0005737,0006520,0009067,0009086,0009088,0009090,0016491,0050661,0070403 remove_due_to_license_issue P31116 15210149 1360 STKVVNVAVIGAGVVGSAFLDQLLAMKSTITYNLVLLAEAERSLISKDFSPLNVGSDWKAALAASTTKTLPLDDLIAHLKTSPKPVILVDNTSSAYIAGFYTKFVENGISIATPNKKAFSSDLATWKALFSNKPTNGFVYHEATVGAGLPIISFLREIIQTGDEVEKIEGIFSGTLSYIFNEFSTSQANDVKFSDVVKVAKKLGYTEPDPRDDLNGLDVARKVTIVGRISGVEVESPTSFPVQSLIPKPLESVKSADEFLEKLSDYDKDLTQLKKEAATENKVLRFIGKVDVATKSVSVGIEKYDYSHPFASLKGSDNVISIKTKRYTNPVVIQGAGAGAAVTAAGVLGDVIKIAQRL 1tvo A 2.5 BS01 FRZ A 1 A52 K54 I103 Q105 M108 S153 N154 L156 C166 D167 A45 K47 I96 Q98 M101 S146 N147 L149 C159 D160 D149 K151 S153 N154 D167 T190 D142 K144 S146 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Ki=0.14uM remove_due_to_license_issue Ki=310nM, IC50=1200nM, Kd=850nM P28482 16139248 1001 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 1tvr A 3.0 BS01 TB9 A 1 L100 K101 K103 V106 V179 Y181 Y188 W229 L234 H235 Y318 L100 K101 K103 V106 V179 Y181 Y188 W229 L234 H235 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 9000632 600 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRK 1tw8 A 2.8 BS01 dna E 0 H31 Y77 G92 K93 Q109 Q138 Y199 N201 A204 K248 H30 Y76 G91 K92 Q108 Q137 Y198 N200 A203 K247 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 1tw8 A 2.8 BS02 dna F 0 G30 H31 Q109 N110 D114 D127 K129 T130 N132 S136 A137 Q138 N141 S144 Y146 K147 Q207 G29 H30 Q108 N109 D113 D126 K128 T129 N131 S135 A136 Q137 N140 S143 Y145 K146 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 1tw8 B 2.8 BS01 dna E 0 G30 H31 Q109 N110 D114 D127 T130 R131 S136 A137 Q138 A139 P140 N141 S144 Y146 K147 Q207 G29 H30 Q108 N109 D113 D126 T129 R130 S135 A136 Q137 A138 P139 N140 S143 Y145 K146 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 1tw8 B 2.8 BS02 dna F 0 Y77 S90 K93 K108 Q109 Q138 Y199 N201 A203 A204 R241 K248 Y76 S89 K92 K107 Q108 Q137 Y198 N200 A202 A203 R240 K247 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 1tw8 C 2.8 BS01 dna G 0 H31 Y77 K93 K108 Q109 Q138 Y199 N201 Q209 R241 K248 H30 Y76 K92 K107 Q108 Q137 Y198 N200 Q208 R240 K247 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 1tw8 C 2.8 BS02 dna H 0 G30 H31 Q109 N110 D111 D114 K135 A137 Q138 A139 P140 N141 S144 Y146 K147 A205 M206 Q207 G29 H30 Q108 N109 D110 D113 K134 A136 Q137 A138 P139 N140 S143 Y145 K146 A204 M205 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 1tw8 D 2.8 BS01 dna G 0 G30 H31 Q109 N110 D114 K129 T130 N132 S136 Q138 P140 N141 I143 S144 K147 Q207 G29 H30 Q108 N109 D113 K128 T129 N131 S135 Q137 P139 N140 I142 S143 K146 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKY 1tw8 D 2.8 BS02 dna H 0 H31 Y77 S90 G92 K93 Q109 Q138 Y199 N201 A203 A204 R241 H30 Y76 S89 G91 K92 Q108 Q137 Y198 N200 A202 A203 R240 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 15491133 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKY 1tx7 A 1.75 BS02 4CM A 1 H57 D189 S190 S195 S214 W215 G219 H40 D171 S172 S177 S192 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=25uM remove_due_to_license_issue P00760 11738605 247 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1txr A 2.0 BS03 BES A 1 D117 E151 E152 L155 D179 C223 Y225 C227 F244 F248 Y251 H256 D117 E151 E152 L155 D179 C223 Y225 C227 F244 F248 Y251 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=18nM remove_due_to_license_issue IC50=1.6nM, Ki=1.6nM Q01693 15274616 503 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 1tyn A 2.0 BS01 CTA A 1 H57 D189 S190 C191 Q192 G193 S195 S214 W215 G216 H40 D171 S172 C173 Q174 G175 S177 S192 W193 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1tys A 1.8 BS01 TMP A 1 R21 W80 S146 H147 R166 S167 D169 N177 H207 Y209 R21 W80 S146 H147 R166 S167 D169 N177 H207 Y209 E58 W80 Y94 S146 R166 D169 E58 W80 Y94 S146 R166 D169 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 8312270 565 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPSHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 1u0b B 2.3 BS01 rna A 0 R10 G39 H40 T43 Q158 G166 A167 R168 W205 G227 L230 F232 M259 V260 M261 M267 G296 H297 Q301 Q311 A315 R318 T321 N351 P353 E354 S357 F360 R364 N367 R427 W432 D436 R439 L449 E450 D451 R459 R10 G39 H40 T43 Q158 G166 A167 R168 W205 G227 L230 F232 M259 V260 M261 M267 G296 H297 Q301 Q311 A315 R318 T321 N351 P353 E354 S357 F360 R364 N367 R427 W432 D436 R439 L449 E450 D451 R459 H37 H40 H37 H40 6.1.1.16 0000166,0004812,0004817,0005524,0005737,0005829,0006412,0006418,0006423,0008270,0016874,0046872 remove_due_to_license_issue P21888 15489861 1 ~ 76 MLKIFNTLTRQKEEFKPIHAGEVGMYVCGITVYDLCHIGHGRTFVAFDVVARYLRFLGYKLKYVRNITDIDDKIIKRANENGESFVAMVDRMIAEMHKDFDALNILRPDMEPRATHHIAEIIELTEQLIAKGHAYVADNGDVMFDVPTDPTYGVLSRQDLDQLQAGARVDVVDDKRNPMDFVLWKMSKEGEPSWPSPWGAGRPGWHIECSAMNCKQLGNHFDIHGGGSDLMFPHHENEIAQSTCAHDGQYVNYWMHSGMVMVDREKMSKSLGNFFTVRDVLKYYDAETVRYFLMSGHYRSQLNYSEENLKQARAALERLYTALRGTDKTVAPAGGEAFEARFIEAMDDDFNTPEAYSVLFDMAREVNRLKAEDMAAANAMASHLRKLSAVLGLLEQEPEAFLQSGAQADDSEVAEIEALIQQRLDARKAKDWAAADAARDRLNEMGIVLEDGPQGTTWRRK 1u0c A 2.5 BS01 dna C 0 G19 D20 G21 S22 I24 Q26 Q44 T46 E47 K48 R51 R70 N136 D137 S138 R141 K142 G18 D19 G20 S21 I23 Q25 Q43 T45 E46 K47 R50 R69 N135 D136 S137 R140 K141 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSCKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0c A 2.5 BS02 dna D 0 S32 C33 Q38 Y66 R68 R70 E80 I81 K139 S31 C32 Q37 Y65 R67 R69 E79 I80 K138 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 551 ~ 574 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSCKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0c B 2.5 BS01 dna C 0 S332 C333 K334 Q338 Y366 R368 R370 E380 I381 K416 D437 K439 T440 S31 C32 K33 Q37 Y65 R67 R69 E79 I80 K115 D136 K138 T139 G319 D320 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSCKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0c B 2.5 BS02 dna D 0 G319 D320 G321 S322 Q326 K328 T346 E347 K348 R370 V373 K398 A433 N436 D437 S438 R441 K442 G18 D19 G20 S21 Q25 K27 T45 E46 K47 R69 V72 K97 A132 N135 D136 S137 R140 K141 G319 D320 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 551 ~ 574 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSCKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0d A 2.9 BS01 dna C 0 D20 G21 S22 I24 Q26 K28 T46 E47 K48 R70 V73 A133 N136 D137 S138 R141 K142 D19 G20 S21 I23 Q25 K27 T45 E46 K47 R69 V72 A132 N135 D136 S137 R140 K141 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSHKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0d A 2.9 BS02 dna D 0 D20 H33 K34 Q38 R68 I81 K116 D137 K139 D19 H32 K33 Q37 R67 I80 K115 D136 K138 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 551 ~ 574 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSHKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0d B 2.9 BS01 dna C 0 D320 S332 H333 K334 Q338 Y366 R368 R370 E380 D19 S31 H32 K33 Q37 Y65 R67 R69 E79 G319 D320 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSHKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0d B 2.9 BS02 dna D 0 D320 S322 I324 Q326 K328 Q344 T346 E347 K348 R370 V373 N436 D437 S438 K442 D19 S21 I23 Q25 K27 Q43 T45 E46 K47 R69 V72 N135 D136 S137 K141 G319 D320 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 15313605 551 ~ 574 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSHKFKHQLSLTFQVTEKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 1u0g A 1.7 BS01 E4P A 1 I156 G157 G158 S209 K210 T211 T214 K518 I156 G157 G158 S209 K210 T211 T214 K518 K210 E216 G271 R272 E357 H388 K518 K210 E216 G271 R272 E357 H388 K518 5.3.1.9 0001701,0001707,0002639,0004347,0005125,0005515,0005576,0005615,0005737,0005829,0005886,0006002,0006094,0006096,0007165,0007611,0008083,0010595,0016853,0031625,0032355,0032570,0033574,0034101,0035902,0035994,0042593,0043209,0043524,0046686,0048029,0051156,0060170,0061620,0061621,0097367,0141199,1901135 remove_due_to_license_issue P06745 15342241 901 AALTRNPQFQKLLEWHRANSANLKLRELFEADPERFNNFSLNLNTNHGHILVDYSKNLVNKEVMQMLVELAKSRGVEAARDNMFSGSKINYTEDRAVLHVALRNRSNTPIKVDGKDVMPEVNRVLDKMKSFCQRVRSGDWKGYTGKSITDIINIGIGGSDLGPLMVTEALKPYSKGGPRVWFVSNIDGTHIAKTLASLSPETSLFIIASKTFTTQETITNAETAKEWFLEAAKDPSAVAKHFVALSTNTAKVKEFGIDPQNMLEFWDWVGGRYSLWSAIGLSIALHVGFDHFEQLLSGAHWMDQHFLKTPLEKNAPVLLALLGIWYINCYGCETHALLPYDQYMHRFAAYFQQGDMESNGKYITKSGARVDHQTGPIVWGEPGTNGQHAFYQLIHQGTKMIPCDFLIPVQTQHPIRKGLHHKILLANFLAQTEALMKGKLPEEARKELQAAGKSPEDLEKLLPHKVFEGNRPTNSIVFTKLTPFILGALIAMYEHKIFVQGIMWDINSFDQWGVELGKQLAKKIEPELEGSSAVTSHDSSTNGLISFIKQQRDTKL 1u0g B 1.7 BS01 E4P B 1 I156 G157 G158 S209 K210 T211 T214 I156 G157 G158 S209 K210 T211 T214 K210 E216 G271 R272 E357 H388 K518 K210 E216 G271 R272 E357 H388 K518 5.3.1.9 0001701,0001707,0002639,0004347,0005125,0005515,0005576,0005615,0005737,0005829,0005886,0006002,0006094,0006096,0007165,0007611,0008083,0010595,0016853,0031625,0032355,0032570,0033574,0034101,0035902,0035994,0042593,0043209,0043524,0046686,0048029,0051156,0060170,0061620,0061621,0097367,0141199,1901135 remove_due_to_license_issue P06745 15342241 902 AALTRNPQFQKLLEWHRANSANLKLRELFEADPERFNNFSLNLNTNHGHILVDYSKNLVNKEVMQMLVELAKSRGVEAARDNMFSGSKINYTEDRAVLHVALRNRSNTPIKVDGKDVMPEVNRVLDKMKSFCQRVRSGDWKGYTGKSITDIINIGIGGSDLGPLMVTEALKPYSKGGPRVWFVSNIDGTHIAKTLASLSPETSLFIIASKTFTTQETITNAETAKEWFLEAAKDPSAVAKHFVALSTNTAKVKEFGIDPQNMLEFWDWVGGRYSLWSAIGLSIALHVGFDHFEQLLSGAHWMDQHFLKTPLEKNAPVLLALLGIWYINCYGCETHALLPYDQYMHRFAAYFQQGDMESNGKYITKSGARVDHQTGPIVWGEPGTNGQHAFYQLIHQGTKMIPCDFLIPVQTQHPIRKGLHHKILLANFLAQTEALMKGKLPEEARKELQAAGKSPEDLEKLLPHKVFEGNRPTNSIVFTKLTPFILGALIAMYEHKIFVQGIMWDINSFDQWGVELGKQLAKKIEPELEGSSAVTSHDSSTNGLISFIKQQRDTKL 1u0h A 2.9 BS04 ONM A 1 D396 G399 F400 T401 L438 G439 D440 D20 G23 F24 T25 L62 G63 D64 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P30803 15591060 100 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1u0h B 2.9 BS01 ONM A 1 D1018 N1025 D130 N137 S891 I892 S942 R1029 K1065 S13 I14 S64 R141 K177 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P26769 15591060 100 HQSYDCVCVMFASIPDFKEFYTESDVNKEGLECLRLLNEIIADFDDLLSKPKFSGVEKIKTIGSTYMAATGLSAIRQYMHIGTMVEFAYALVGKLDAINKHSFNDFKLRVGINHGPVIAGVIGAQKPQYDIWGNTVNVASRMDSTGVLDKIQVTEETSLILQTLGYTCTCRGIINVKGKGDLKTYFVNT 1u1b A 2.0 BS01 PAX A 1 K7 Q11 H12 N44 T45 Q69 N71 A109 E111 V118 H119 F120 K7 Q11 H12 N44 T45 Q69 N71 A109 E111 V118 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Kd=16nM remove_due_to_license_issue P61823 15969595 901 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1u1k A 2.0 BS01 dna B 0 K15 F17 G19 G20 D42 V44 M46 R55 G56 F57 F59 E85 K87 A89 V90 R92 S95 H101 K8 F10 G12 G13 D35 V37 M39 R48 G49 F50 F52 E78 K80 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1l A 2.0 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 V44 M46 R55 G56 F57 F59 E85 K87 A89 V90 R92 S95 H101 Q5 K8 F10 G12 G13 D35 V37 M39 R48 G49 F50 F52 E78 K80 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1m A 2.0 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 V44 M46 R55 G56 F57 F59 E85 K87 A89 V90 R92 S95 H101 Q5 K8 F10 G12 G13 D35 V37 M39 R48 G49 F50 F52 E78 K80 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1n A 2.1 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 V44 M46 R55 F57 F59 E85 A89 V90 R92 S95 H101 Q5 K8 F10 G12 G13 D35 V37 M39 R48 F50 F52 E78 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1o A 2.0 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 V44 M46 R55 F57 F59 E85 A89 V90 R92 H101 Q5 K8 F10 G12 G13 D35 V37 M39 R48 F50 F52 E78 A82 V83 R85 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1p A 1.9 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 V44 M46 R55 F57 F59 E85 K87 A89 V90 R92 H101 Q5 K8 F10 G12 G13 D35 V37 M39 R48 F50 F52 E78 K80 A82 V83 R85 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1q A 1.8 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 M46 R55 G56 F57 F59 E85 K87 A89 V90 R92 S95 H101 Q5 K8 F10 G12 G13 D35 M39 R48 G49 F50 F52 E78 K80 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1r A 1.8 BS01 dna B 0 Q12 K15 F17 G19 G20 D42 V44 M46 R55 G56 F57 F59 E85 K87 A89 V90 R92 S95 H101 Q5 K8 F10 G12 G13 D35 V37 M39 R48 G49 F50 F52 E78 K80 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 15342234 202 ~ 212 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASAS 1u1w A 1.35 BS01 3HA A 1 E45 A72 G73 H74 M198 Y203 D208 T211 G212 S213 E45 A72 G73 H74 M198 Y203 D208 T211 G212 S213 5.3.3.17 0002047,0003824,0005737,0009058,0016853,0017000,0102943 Kd=1.4uM remove_due_to_license_issue Q51792 15545603 700 MHNYVIIDAFASVPLEGNPVAVFFDADDLPPAQMQRIAREMNLSESTFVLKPRNGGDALIRIFTPVNELPFAGHPLLGTAIALGAHTDNHRLYLETQMGTIAFELERQNGSVIAASMDQPIPTWTALGRDAELLKALGISDSTFPIEIYHNGPRHVFVGLPSIDALSALHPDHRALSNFHDMAINCFAGAGRRWRSRMFSPAYGVVEDAATGSAAGPLAIHLARHGQIEFGQPVEILQGVEIGRPSLMFAKAEGRAEQLTRVEVSGNGVTFGRGTIVL 1u2r A 2.6 BS03 GDP A 1 D29 G31 K32 S33 T34 K159 D161 S213 L215 D27 G29 K30 S31 T32 K139 D141 S193 L195 3.6.5.- 0003746,0003924,0005515,0005525,0005737,0005829,0006412,0006414,0016787,0019843,0042802,0043022,0045901,0051087,1990145,1990904 remove_due_to_license_issue P32324 15316019 1920 AFTVDQMRSLMDKVTNVRNMSVIAHVDHGKSTLTDSLVQRAGIISAGITIKSTAISLYSEMSDEDVKEIKQKTDGNSFLINLIDSPGHVDFSSEVTAALRVTDGALVVVDTIEGVCVQTETVLRQALGERIKPVVVINKVDRALLELQVSKEDLYQTFARTVESVNVIVSTYADEVLGDVQVYPARGTVAFGSGLHGWAFTIRQFATRYAKKFGVDKAKMMDRLWGDSFFNPKTKKWTNKDTDAEGKPLERAFNMFILDPIFRLFTAIMNFKKDEIPVLLEKLEIVLKGDEKDLEGKALLKVVMRKFLPAADALLEMIVLHLPSPVTAQAYRAEQLYEGPADDANCIAIKNCDPKADLMLYVSKMVPTSDKGRFYAFGRVFAGTVKSGQKVRIQGPNYVPGKKDDLFIKAIQRVVLMMGRFVEPIDDCPAGNIIGLVGIDQFLLKTGTLTTSETAHNMKVMKFSVSPVVQVAVEVKNANDLPKLVEGLKRLSKSDPCVLTYMSESGEHIVAGTGELHLEICLQDLEHDHAGVPLKISPPVVAYRETVESESSQTALSKSPNKHNRIYLKAEPIDEEVSLAIENGIINPRDDFKARARIMADDYGWDVTDARKIWCFGPDGNGPNLVIDQTKAVQYLHEIKDSVVAAFQWATKEGPIFGEEMRSVRVNILDVTLHADAIHRGGGQIIPTMRRATYAGFLLADPKIQEPVFLVEIQCPEQAVGGIYSVLNKKRGQVVSEEQTPLFTVKAYLPVNESFGFTGELRQATGGQAFPQMVFDHWSTLGSDPLDPTSKAGEIVLAARKRHGMKEEVPGWQEYYDKL 1u2y A 1.95 BS02 GOX A 1 A198 H201 E233 A198 H201 E233 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 Ki=18mM remove_due_to_license_issue P04746 15304511 499 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 1u32 A 2.0 BS03 OKA A 1 R96 H125 I130 Y134 R221 Y272 L273 Y276 R91 H120 I125 Y129 R216 Y267 L268 Y271 D64 H66 D92 D95 R96 N124 H125 H173 R221 H248 D59 H61 D87 D90 R91 N119 H120 H168 R216 H243 3.1.3.16 0000070,0000165,0000775,0000776,0000781,0001824,0003723,0004721,0004722,0005515,0005521,0005634,0005654,0005694,0005730,0005737,0005739,0005741,0005815,0005829,0005856,0005925,0005977,0006338,0006357,0006470,0007283,0008157,0016607,0016787,0016791,0017018,0019901,0019903,0019904,0030182,0030496,0032154,0032922,0032991,0033192,0042752,0043153,0043197,0044877,0046822,0046872,0048511,0051301,0060252,0072357,0098793,0098794,0098978,0140791,0180004,0180005,0180006,0180007,0180008,1990439 ic50=97nM remove_due_to_license_issue IC50=>5000nM P36873 15280359 501 KLNIDSIIQRLLEVRGSKPGKNVQLQENEIRGLCLKSREIFLSQPILLELEAPLKICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFLLRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDLQSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVLGWGENDRGVSFTFGAEVVAKFLHKHDLDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYLDVYNNAGAMMSVDETLMCSFQILKP 1u33 A 1.95 BS01 LM2 A 1 W58 W59 Y62 Q63 H101 G104 T163 L165 D197 A198 E233 H299 D300 H305 W58 W59 Y62 Q63 H101 G104 T163 L165 D197 A198 E233 H299 D300 H305 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 Ki=25uM remove_due_to_license_issue P04746 15304511 500 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 1u3q A 2.4 BS01 272 A 1 E305 M340 L476 E43 M78 L205 ? 0003677,0004879,0006355 ic50=3.5nM remove_due_to_license_issue IC50=3.5nM Q92731 15456246 501 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1u3r A 2.21 BS02 338 A 1 L298 E305 L339 L343 F356 I373 H475 L476 L36 E43 L77 L81 F94 I111 H206 L207 ? 0003677,0004879,0006355 ic50=5nM remove_due_to_license_issue IC50=5nM Q92731 15456246 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMQDADSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 1u3s A 2.5 BS02 797 A 1 E305 L339 M340 F356 I376 G472 H475 E43 L77 M78 F94 I114 G202 H205 ? 0003677,0004879,0006355 ic50=1.4nM remove_due_to_license_issue IC50=1.4nM Q92731 15456246 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYADSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1u59 A 2.3 BS01 STU A 1 L344 G345 V352 A367 M414 M416 A417 G420 P421 R465 N466 L468 D479 L17 G18 V25 A37 M84 M86 A87 G90 P91 R135 N136 L138 D149 D461 A463 R465 N466 D479 W501 D131 A133 R135 N136 D149 W171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=55.8nM remove_due_to_license_issue P43403 15292186 100 KKLFLKRDNLLIADIELGCGNFGSVRQGVYRKQIDVAIKVLKQGTEKADTEEMMREAQIMHQLDNPYIVRLIGVCQAEALMLVMEMAGGGPLHKFLVGKREEIPVSNVAELLHQVSMGMKYLEEKNFVHRDLAARNVLLVNRHYAKISDFGLSKALGADDSYYTARSAGKWPLKWYAPECINFRKFSSRSDVWSYGVTMWEALSYGQKPYKKMKGPEVMAFIEQGKRMECPPECPPELYALMSDCWIYKWEDRPDFLTVEQRMRACYYSLASKVEGHHHHHH 1u63 A 3.4 BS01 rna B 0 K18 R20 N21 S25 I29 T31 R96 K100 Y159 Q161 Y200 T204 M205 G206 A208 K18 R20 N21 S25 I29 T31 R96 K100 Y159 Q161 Y200 T204 M205 G206 A208 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P54050 15659579 1 ~ 49 MDREALLQAVKEARELAKPRNFTQSFEFIATLKEIDMRKPENRIKTEVVLPHGRGKEAKIAVIGTGDLAKQAEELGLTVIRKEEIEELGKNKRKLRKIAKAHDFFIAQADLMPLIGRYMGVILGPRGKMPKPVPANANIKPLVERLKKTVVINTRDKPYFQVLVGNEKMTDEQIVDNIEAVLNVVAKKYEKGLYHIKDAYVKLTMGPAVKVKKE 1u63 A 3.4 BS02 rna D 0 K90 K92 R93 K94 K90 K92 R93 K94 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P54050 15659579 1 ~ 49 MDREALLQAVKEARELAKPRNFTQSFEFIATLKEIDMRKPENRIKTEVVLPHGRGKEAKIAVIGTGDLAKQAEELGLTVIRKEEIEELGKNKRKLRKIAKAHDFFIAQADLMPLIGRYMGVILGPRGKMPKPVPANANIKPLVERLKKTVVINTRDKPYFQVLVGNEKMTDEQIVDNIEAVLNVVAKKYEKGLYHIKDAYVKLTMGPAVKVKKE 1u63 C 3.4 BS01 rna B 0 K90 K92 R93 K90 K92 R93 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P54050 15659579 1 ~ 49 MDREALLQAVKEARELAKPRNFTQSFEFIATLKEIDMRKPENRIKTEVVLPHGRGKEAKIAVIGTGDLAKQAEELGLTVIRKEEIEELGKNKRKLRKIAKAHDFFIAQADLMPLIGRYMGVILGPRGKMPKPVPANANIKPLVERLKKTVVINTRDKPYFQVLVGNEKMTDEQIVDNIEAVLNVVAKKYEKGLYHIKDAYVKLTMGPAVKVKKE 1u63 C 3.4 BS02 rna D 0 R20 N21 F22 S25 E27 I29 R96 K100 R126 R155 Y159 Q161 Y200 K202 T204 M205 G206 A208 R20 N21 F22 S25 E27 I29 R96 K100 R126 R155 Y159 Q161 Y200 K202 T204 M205 G206 A208 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P54050 15659579 1 ~ 49 MDREALLQAVKEARELAKPRNFTQSFEFIATLKEIDMRKPENRIKTEVVLPHGRGKEAKIAVIGTGDLAKQAEELGLTVIRKEEIEELGKNKRKLRKIAKAHDFFIAQADLMPLIGRYMGVILGPRGKMPKPVPANANIKPLVERLKKTVVINTRDKPYFQVLVGNEKMTDEQIVDNIEAVLNVVAKKYEKGLYHIKDAYVKLTMGPAVKVKKE 1u65 A 2.61 BS02 CP0 A 1 Y70 W84 Y121 W279 L282 F284 D285 S286 F330 F331 Y67 W81 Y118 W276 L279 F281 D282 S283 F327 F328 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue Ki=26nM P04058 15772291 603 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNATA 1u6p A -1.00 BS01 rna B 0 R18 L21 D22 R23 Q25 A27 Y28 W35 A36 K37 K41 K42 R18 L21 D22 R23 Q25 A27 Y28 W35 A36 K37 K41 K42 ? 0003676,0008270 remove_due_to_license_issue P03332 15457265 276 ~ 376 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSLL 1u6q A 2.02 BS01 745 A 1 H45 D191 S192 Q194 G220 G228 H46 D192 S193 Q195 G221 G229 H45 D96 Q194 G195 D196 S197 G198 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue Ki=1259nM P00749 15582418 245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 1u71 A 2.2 BS01 MXA A 1 I7 V8 A9 G20 D21 R22 E30 F34 S59 P61 V115 I7 V8 A9 G20 D21 R22 E30 F34 S59 P61 V115 R22 E30 R22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 remove_due_to_license_issue IC50=0.61nM, Ki=0.025nM P00374 15681865 187 VGSLNCIVAVSQNMGIGKNGDRPWPPLRNEFRYFQRMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 1u9e A 2.4 BS02 397 A 1 E305 L339 H475 E43 L77 H201 ? 0003677,0004879,0006355 ic50=5.7nM remove_due_to_license_issue IC50=6nM Q92731 15548008 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1u9q X 2.3 BS01 186 X 1 C25 G65 G66 L67 M68 A133 D158 H159 C25 G65 G66 L67 M68 A138 D161 H162 3.4.22.51 0006508,0008234 Ki=1102.9nM remove_due_to_license_issue P25779 15727867 300 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 1u9v A 2.2 BS01 IHE A 1 G23 C25 G65 G66 Y67 A134 H162 G23 C25 G65 G66 Y67 A134 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=6nM P43235 15537340 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1u9w A 2.3 BS01 IHI A 1 G23 C25 G64 Y67 A134 N161 H162 G24 C26 G65 Y68 A135 N162 H163 Q19 C25 H162 N182 Q20 C26 H163 N183 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=3.5nM P43235 15537340 300 RAPDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1u9x A 2.1 BS01 IHJ A 1 G23 C25 G64 G66 Y67 A134 N161 H162 G24 C26 G65 G67 Y68 A135 N162 H163 Q19 C25 H162 N182 Q20 C26 H163 N183 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=7nM P43235 15537340 300 RAPDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1ua4 A 1.9 BS03 AMP A 1 N292 H342 T343 Y344 I428 V429 P432 I438 G439 N291 H341 T342 Y343 I427 V428 P431 I437 G438 2.7.1.-,2.7.1.147 0000287,0004340,0005737,0005975,0006006,0006096,0016301,0016773,0043843,0046872,0051156 Ki~0.06mM remove_due_to_license_issue Q9V2Z6 12909015 1456 PTWEELYKNAIEKAIKSVPKVKGVLLGYNTNIDAIKYLDSKDLEERIIKAGKEEVIKYSEELPDKINTVSQLLGSILWSIRRGKAAELFVESCPVRFYMKRWGWNELRMGGQAGIMANLLGGVYGVPVIVHVPQLSRLQANLFLDGPIYVPTLENGEVKLIHPKEFSGDEENCIHYIYEFPRGFRVFEFEAPRENRFIGSADDYNTTLFIREEFRESFSEVIKNVQLAILSGLQALTKENYKEPFEIVKSNLEVLNEREIPVHLEFAFTPDEKVREEILNVLGMFYSVGLNEVELASIMEILGEKKLAKELLAHDPVDPIAVTEAMLKLAKKTGVKRIHFHTYGYYLALTEYKGEHVRDALLFAALAAAAKAMKGNITSLEEIREATSVPVNEKATQVEEKLRAEYGIKEGIGEVEGYQIAFIPTKIVAKPKSTVGIGDTISSSAFIGEFSFTL 1ucn A 2.0 BS03 ADP A 1 K12 L55 W60 R88 T94 R105 N115 K11 L54 W59 R87 T93 R104 N114 K12 Y52 N115 G118 E129 K11 Y51 N114 G117 E128 2.7.4.6 0000287,0003723,0004536,0004550,0005515,0005524,0005525,0005634,0005737,0005769,0005829,0006183,0006228,0006241,0006259,0006897,0007399,0007595,0008285,0008408,0009117,0016020,0016301,0030154,0030879,0032587,0042802,0042981,0043024,0043388,0046872,0050679,0070062 Kd=6uM remove_due_to_license_issue P15531 12972261 1160 ANCERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVGLKFMQASEDLLKEHYVDLKDRPWFAGLVKYMHSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIGGSDSVESAEKEIGLWFHPEELVDYTSCAQNWIYE 1ucn B 2.0 BS02 ADP B 1 K12 L55 W60 R88 T94 R105 V112 N115 K11 L54 W59 R87 T93 R104 V111 N114 K12 Y52 N115 G118 E129 K11 Y51 N114 G117 E128 2.7.4.6 0000287,0003723,0004536,0004550,0005515,0005524,0005525,0005634,0005737,0005769,0005829,0006183,0006228,0006241,0006259,0006897,0007399,0007595,0008285,0008408,0009117,0016020,0016301,0030154,0030879,0032587,0042802,0042981,0043024,0043388,0046872,0050679,0070062 Kd=6uM remove_due_to_license_issue P15531 12972261 2160 ANCERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVGLKFMQASEDLLKEHYVDLKDRPWFAGLVKYMHSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIGGSDSVESAEKEIGLWFHPEELVDYTSCAQNWIYE 1udt A 2.3 BS02 VIA A 1 V782 A783 L804 M816 Q817 G819 F820 V235 A236 L257 M269 Q270 G272 F273 3.1.4.35 0004114,0007165,0008081 Kd~0.5nM remove_due_to_license_issue IC50=2.2nM, Ki=1.9nM, EC50=8.7nM O76074 12955149 1000 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 1udu A 2.83 BS02 CIA A 1 Y612 S663 V782 A783 F786 L804 M816 Q817 F820 Y76 S127 V235 A236 F239 L257 M269 Q270 F273 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue IC50=4nM, Ki=10nM O76074 12955149 1003 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 1ugp A 1.63 BS02 BUA A 1 A111 S112 C113 A110 S111 C112 C108 C111 S112 C113 C107 C110 S111 C112 4.2.1.84 0003824,0005515,0016829,0018822,0046872,0046914,0050897,0050899 remove_due_to_license_issue Q7SID2 14717710 1302 TENILRKSDEEIQKEITARVKALESMLIEQGILTTSMIDRMAEIYENEVGPHLGAKVVVKAWTDPEFKKRLLADGTEACKELGIGGLQGEDMMWVENTDEVHHVVVCTLCSCYPWPVLGLPPNWFKEPQYRSRVVREPRQLLKEEFGFEVPPSKEIKVWDSSSEMRFVVLPQRPAGTDGWSEEELATLVTRESMIGVEPAKAV 1ugx A 1.6 BS02 MGC C 1 G1 Y78 G121 Y122 W123 D125 G1 Y78 G121 Y122 W123 D125 ? 0019862,0030246 remove_due_to_license_issue P18670 12946359 1 GKAFDDGAFTGIREINLSYNKETAIGDFQVVYDLNGSPYVGQNHVSFITGFTPVKISLDFPSEYIMEVSGYTGNVSGYVVVRSLTFKTNKKTYGPYGVTSGTPFNLPIENGLIVGFKGSIGYWLDYFSMYLSL 1uh1 C 2.8 BS03 AMG I 1 G1 Y78 Y122 W123 D125 G1 Y78 Y122 W123 D125 ? 0019862,0030246 remove_due_to_license_issue P18670 12946359 1 GKAFDDGAFTGIREINLSYNKETAIGDFQVVYDLNGSPYVGQNHKSFITGFTPVKISLDFPSEYIMEVSGYTGNVSGYVVVRSLTFKTNKKTYGPYGVTSGTPFNLPIENGLIVGFKGSIGYWLDYFSMYLSL 1uho A 2.5 BS02 VDN A 1 H613 Y664 L804 M816 Q817 G819 F820 H77 Y128 L257 M269 Q270 G272 F273 3.1.4.35 0004114,0007165,0008081 Kd~0.6nM remove_due_to_license_issue IC50=0.890000nM, Ki=1nM O76074 12955149 1000 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 1ui0 A 1.5 BS02 URA A 1 E41 G42 E47 P53 F54 N80 H155 E40 G41 E46 P52 F53 N79 H154 3.2.2.27 0004844,0006281,0016787,0046872,0051539 Ki=88nM remove_due_to_license_issue Q5SKC5 14556741 211 TLELLQAQAQNCTACRLMEGRTRVVFGEGNPDAKLMIVGEGPGEEEDKTGRPFVGKAGQLLNRILEAAGIPREEVYITNIVKCRPPQNRAPLPDEAKICTDKWLLKQIELIAPQIIVPLGAVAAEFFLGEKVSITKVRGKWYEWHGIKVFPMFHPAYLLRNPSRAPGSPKHLTWLDIQEVKRALDALPPKER 1ui0 A 1.5 BS03 URA A 2 R64 I65 K171 W175 R63 I64 K170 W174 3.2.2.27 0004844,0006281,0016787,0046872,0051539 Ki=88nM remove_due_to_license_issue Q5SKC5 14556741 212 TLELLQAQAQNCTACRLMEGRTRVVFGEGNPDAKLMIVGEGPGEEEDKTGRPFVGKAGQLLNRILEAAGIPREEVYITNIVKCRPPQNRAPLPDEAKICTDKWLLKQIELIAPQIIVPLGAVAAEFFLGEKVSITKVRGKWYEWHGIKVFPMFHPAYLLRNPSRAPGSPKHLTWLDIQEVKRALDALPPKER 1uj5 A 2.0 BS01 5RP A 1 T30 S32 T33 G87 D89 K99 G100 G102 A104 E108 K126 T28 S30 T31 G85 D87 K97 G98 G100 A102 E106 K124 5.3.1.6 0004751,0006098,0009052,0016853 Ki=0.89mM remove_due_to_license_issue Q72J47 13679361 302 RPLESYKKEAAHAAIAYVQDGMVVGLGTGSTARYAVLELARRLREGELKGVVGVPTSRATEELAKREGIPLVDLPPEGVDLAIDGADEIAPGLALIKGMGGALLREKIVERVAKEFIVIADHTKKVPVLGRGPVPVEIVPFGYRATLKAIADLGGEPELRMDGDEFYFTDGGHLIADCRFGPIGDPLGLHRALLEIPGVVETGLFVGMATRALVAGPFGVEELLP 1uj6 A 1.74 BS01 A5P A 1 T30 S32 T33 G87 D89 K99 G100 G102 A104 E108 K126 T28 S30 T31 G85 D87 K97 G98 G100 A102 E106 K124 5.3.1.6 0004751,0006098,0009052,0016853 Ki=0.89mM remove_due_to_license_issue Q72J47 13679361 228 RPLESYKKEAAHAAIAYVQDGMVVGLGTGSTARYAVLELARRLREGELKGVVGVPTSRATEELAKREGIPLVDLPPEGVDLAIDGADEIAPGLALIKGMGGALLREKIVERVAKEFIVIADHTKKVPVLGRGPVPVEIVPFGYRATLKAIADLGGEPELRMDGDEFYFTDGGHLIADCRFGPIGDPLGLHRALLEIPGVVETGLFVGMATRALVAGPFGVEELLP 1uk0 A 3.0 BS01 FRM A 1 D105 L108 D109 H201 G202 R217 Y235 S243 Y246 D105 L108 D109 H201 G202 R217 Y235 S243 Y246 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=16nM P09874 14706823 501 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 1uk1 A 3.0 BS01 FRQ A 1 D766 L769 H862 G863 I879 A880 Y889 Y896 A898 S904 Y907 D105 L108 H201 G202 I218 A219 Y228 Y235 A237 S243 Y246 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=60nM P09874 15293985 501 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 1ukt A 2.2 BS01 GLC C 1 F259 D328 F259 D328 D135 R227 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 2.4.1.19 0003824,0004556,0005576,0005975,0016757,0030246,0043169,0043895,0046872,2001070 remove_due_to_license_issue P05618 14769878 2 APDTSVSNKQNFSTDVIYQIFTDRFSDGNPANNPTGAAFDGSCTNLRLYCGGDWQGIINKINDGYLTGMGITAIWISQPVENIYSVINYSGVNNTAYHGLWARDFKKTNPAYGTMQDFKNLIDTAHAHNIKVIIDFAPNHTSPASSDDPSFAENGRLYDNGNLLGGYTNDTQNLFHHYGGTDFSTIENGIYKNLYDLADLNHNNSSVDVYLKDAIKMWLDLGVDGIRVDAVKHMPFGWQKSFMATINNYKPVFTFGEWFLGVNEISPEYHQFANESGMSLLDFRFAQKARQVFRDNTDNMYGLKAMLEGSEVDYAQVNDQVTFIDNHDMERFHTSNGDRRKLEQALAFTLTSRGVPAIYYGSEQYMSGGNDPDNRARLPSFSTTTTAYQVIQKLAPLRKSNPAIAYGSTHERWINNDVIIYERKFGNNVAVVAINRNMNTPASITGLVTSLPRGSYNDVLGGILNGNTLTVGAGGAASNFTLAPGGTAVWQYTTDATTPIIGNVGPMMAKPGVTITIDGRGFGSGKGTVYFGTTAVTGADIVAWEDTQIQVKIPAVPGGIYDIRVANAAGAASNIYDNFEVLTGDQVTVRFVINNATTALGQNVFLTGNVSELGNWDPNNAIGPMYNQVVYQYPTWYYDVSVPAGQTIEFKFLKKQGSTVTWEGGANRTFTTPTSGTATVNVNWQP 1uml A 2.5 BS02 FR4 A 1 H17 D19 L58 F61 L62 F65 M155 G184 D185 T269 D296 H14 D16 L55 F58 L59 F62 M152 G181 D182 T266 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=30nM remove_due_to_license_issue P56658 15239652 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1ung A 2.3 BS01 ALH A 1 A31 C83 D84 Q85 L133 N144 A27 C79 D80 Q81 L129 N140 D126 K128 Q130 N131 N144 C157 T164 D122 K124 Q126 N127 N140 C153 T160 2.7.11.1 0000226,0000307,0001764,0001963,0002039,0004672,0004674,0004676,0004677,0004679,0004693,0004694,0004711,0005176,0005515,0005524,0005634,0005654,0005737,0005829,0005874,0005886,0006338,0006468,0006886,0006915,0007160,0007268,0007399,0007409,0007416,0007519,0008017,0008045,0008306,0008542,0014044,0014069,0016020,0016079,0016241,0016301,0016310,0016477,0016533,0018105,0018107,0019233,0021537,0021549,0021695,0021697,0021766,0021819,0021954,0021987,0022038,0030027,0030036,0030054,0030175,0030182,0030334,0030424,0030425,0030426,0030517,0030549,0030900,0031175,0031397,0031594,0031914,0032801,0035175,0035249,0035402,0035403,0035418,0035979,0042220,0042981,0042995,0043005,0043025,0043113,0043125,0043204,0043525,0044022,0044023,0044024,0044025,0045202,0045786,0045861,0045892,0045956,0046826,0048148,0048156,0048167,0048488,0048489,0048511,0048675,0048709,0048813,0050321,0051301,0051402,0051649,0051726,0051879,0051966,0060078,0060079,0061001,0070509,0072354,0072371,0072518,0090314,0098793,0106310,0140823,0140855,0140857,1901987,1903076,1903421,1904646,1990244 ic50=0.18uM remove_due_to_license_issue IC50=200nM Q00535 15689152 1293 MQKYEKLEKIYGTVFKAKNRETHEIVALKRVRLDDDDEGVPSSALREICLLKELKHKNIVRLHDVLHSDKKLTLVFEFCDQDLKKYFDSCNGDLDPEIVKSFLFQLLKGLGFCHSRNVLHRDLKPQNLLINRNGELKLANFGLARAFGIPVRCYSAEVVTLWYRPPDVLFGAKLYSTSIDMWSAGCIFAELANAGRPLFPGNDVDDQLKRIFRLLGTPTEEQWPSMTKLPDYKPYPMYPATTSLVNVVPKLNATGRDLLQNLLKCNPVQRISAEEALQHPYFSDFCPP 1unh A 2.35 BS01 IXM A 1 I10 A31 F80 F82 C83 D84 Q85 D86 L133 I9 A24 F69 F71 C72 D73 Q74 D75 L122 D126 K128 Q130 N131 N144 C157 T164 D115 K117 Q119 N120 N133 C146 T153 2.7.11.1 0000226,0000307,0001764,0001963,0002039,0004672,0004674,0004676,0004677,0004679,0004693,0004694,0004711,0005176,0005515,0005524,0005634,0005654,0005737,0005829,0005874,0005886,0006338,0006468,0006886,0006915,0007160,0007268,0007399,0007409,0007416,0007519,0008017,0008045,0008306,0008542,0014044,0014069,0016020,0016079,0016241,0016301,0016310,0016477,0016533,0018105,0018107,0019233,0021537,0021549,0021695,0021697,0021766,0021819,0021954,0021987,0022038,0030027,0030036,0030054,0030175,0030182,0030334,0030424,0030425,0030426,0030517,0030549,0030900,0031175,0031397,0031594,0031914,0032801,0035175,0035249,0035402,0035403,0035418,0035979,0042220,0042981,0042995,0043005,0043025,0043113,0043125,0043204,0043525,0044022,0044023,0044024,0044025,0045202,0045786,0045861,0045892,0045956,0046826,0048148,0048156,0048167,0048488,0048489,0048511,0048675,0048709,0048813,0050321,0051301,0051402,0051649,0051726,0051879,0051966,0060078,0060079,0061001,0070509,0072354,0072371,0072518,0090314,0098793,0106310,0140823,0140855,0140857,1901987,1903076,1903421,1904646,1990244 ic50=0.1uM remove_due_to_license_issue Q00535 15689152 1288 QKYEKLEKIYGTVFKAKNRHEIVALKRVRLDGVPSSALREICLLKELKHKNIVRLHDVLHSDKKLTLVFEFCDQDLKKYFDSCNGDLDPEIVKSFLFQLLKGLGFCHSRNVLHRDLKPQNLLINRNGELKLANFGLARAFGIPVRCYSAEVVTLWYRPPDVLFGAKLYSTSIDMWSAGCIFAELANAGRPLFPGNDVDDQLKRIFRLLGTPTEEQWPSMTKLPDYKPYPMYPATTSLVNVVPKLNATGRDLLQNLLKCNPVQRISAEEALQHPYFS 1unl A 2.2 BS01 RRC A 1 I10 G11 E12 V18 A31 F80 C83 D84 Q85 D86 Q130 L133 I10 G11 E12 V18 A31 F80 C83 D84 Q85 D86 Q130 L133 D126 K128 Q130 N131 N144 C157 T164 D126 K128 Q130 N131 N144 C157 T164 2.7.11.1 0000226,0000307,0001764,0001963,0002039,0004672,0004674,0004676,0004677,0004679,0004693,0004694,0004711,0005176,0005515,0005524,0005634,0005654,0005737,0005829,0005874,0005886,0006338,0006468,0006886,0006915,0007160,0007268,0007399,0007409,0007416,0007519,0008017,0008045,0008306,0008542,0014044,0014069,0016020,0016079,0016241,0016301,0016310,0016477,0016533,0018105,0018107,0019233,0021537,0021549,0021695,0021697,0021766,0021819,0021954,0021987,0022038,0030027,0030036,0030054,0030175,0030182,0030334,0030424,0030425,0030426,0030517,0030549,0030900,0031175,0031397,0031594,0031914,0032801,0035175,0035249,0035402,0035403,0035418,0035979,0042220,0042981,0042995,0043005,0043025,0043113,0043125,0043204,0043525,0044022,0044023,0044024,0044025,0045202,0045786,0045861,0045892,0045956,0046826,0048148,0048156,0048167,0048488,0048489,0048511,0048675,0048709,0048813,0050321,0051301,0051402,0051649,0051726,0051879,0051966,0060078,0060079,0061001,0070509,0072354,0072371,0072518,0090314,0098793,0106310,0140823,0140855,0140857,1901987,1903076,1903421,1904646,1990244 remove_due_to_license_issue IC50=160nM, Kd=1900nM Q00535 15689152 1293 MQKYEKLEKIGEGTYGTVFKAKNRETHEIVALKRVRLDDDDEGVPSSALREICLLKELKHKNIVRLHDVLHSDKKLTLVFEFCDQDLKKYFDSCNGDLDPEIVKSFLFQLLKGLGFCHSRNVLHRDLKPQNLLINRNGELKLANFGLARAFGIPVRCYSAEVVTLWYRPPDVLFGAKLYSTSIDMWSAGCIFAELANAGRPLFPGNDVDDQLKRIFRLLGTPTEEQWPSMTKLPDYKPYPMYPATTSLVNVVPKLNATGRDLLQNLLKCNPVQRISAEEALQHPYFSDFCPP 1uod A 1.9 BS01 G3H A 1 G62 G63 H66 F88 T89 K114 Y116 G118 D119 H230 G43 G44 H47 F69 T70 K95 Y97 G99 D100 H198 2.7.1.121 0004371,0005515,0005829,0006071,0006090,0006974,0016301,0019563,0042182,0042802,0042803,0046365,0046835,0047324,0061610,1990234 remove_due_to_license_issue P76015 15476397 1369 DVLDEQLAGLAKAHPSLTLHQDPVYVTRADAPVAGKVALLSGGGSGHEPMHCGYIGQGMLSGACPGEIFTSPTPDKIFECAMQVDGGEGVLLIIKNYTGDILNFETATELLHDSGVKVTTVVIDDDVAVKDSLYTAGRRGVANTVLIEKLVGAAAERGDSLDACAELGRKLNNQGHSIGIALGACLADNEMEFGVGIHGEPGIDRRPFSSLDQTVDEMFDTLLVNGSYHRTLRFWDYQQGSWQEEQQTKQPLQSGDRVIALVNNLGATPLSELYGVYNRLTTRCQQAGLTIERNLIGAYCTSLDMTGFSITLLKVDDETLALWDAPVHTPALNWGK 1uom A 2.28 BS01 PTI A 1 M343 L346 T347 A350 D351 E353 W383 L387 G521 H524 L525 A546 M37 L40 T41 A44 D45 E47 W77 L81 G215 H218 L219 A231 ? ic50=19nM remove_due_to_license_issue IC50=19nM, EC50=16.5nM P03372 12825935 1547 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLPLYDLLLEMLDA 1uou A 2.11 BS01 CMU A 1 H116 S117 T118 L148 Y199 R202 I214 S217 K221 H84 S85 T86 L116 Y167 R170 I182 S185 K189 D114 K115 H116 S117 T154 D195 R202 S217 K221 K222 D82 K83 H84 S85 T122 D163 R170 S185 K189 K190 2.4.2.4 0000002,0001525,0004645,0005515,0005829,0006206,0006213,0006935,0007165,0008083,0009032,0016154,0016757,0016763,0030154,0031641,0042803,0046074,0051969,1905333 Ki=20nM remove_due_to_license_issue IC50=35nM, Ki=20nM P19971 14725767 1481 PKQLPELIRMKRDGGRLSEADIRGFVAAVVNGSAQGAQIGAMLMAIRLRGMDLEETSVLTQALAQSGQQLEWPEAWRQQLVDKHSTGGVGDKVSLVLAPALAACGCKVPMISGRGLGHTGGTLDKLESIPGFNVIQSPEQMQVLLDQAGCCIVGQSEQLVPADGILYAARDVTATVDSLPLITASILSKKLVEGLSALVVDVKFGAVFPNQEQARELAKTLVGVGASLGLRVAAALTAMDKPLGRCVGHALEVEEALLCMDGAGPPDLRDLVTTLGGALLWLSGHAGTQAQGAARVAAALDDGSALGRFERMLAAQGVDPGLARALCSGSPAERRQLLPRAREQEELLAPADGTVELVRALPLALVLHELGALRLGVGAELLVDVGQRLRRGTPWLRVHRDGPALSGPQSRALQEALVLSDRAPFAAPLPFAELVLPP 1upf A 2.3 BS01 URF A 1 M166 Y228 M146 Y208 R137 T141 D235 D238 R117 T121 D215 D218 2.4.2.9 0004845,0005525,0016757,0044206 Ki=25uM remove_due_to_license_issue Q26998 9628859 999 QEESILQDIITRFPNVVLMKQTAQLRAMMTIIRDKETPKEEFVFYADRLIRLLIEEALNELPFQKKEVTTPLDVSYHGVSFYSKICGVSIVRAGESMESGLRAVCRGVRIGKILIQRDETTAEPKLIYEKLPADIRERWVMLLDPMCATAGSVCKAIEVLLRLGVKEERIIFVNILAAPQGIERVFKEYPKVRMVTAAVDICLNSRYYIVPGIGDFGDRYFGTM 1upf D 2.3 BS01 URF D 1 M166 A168 Y227 Y228 I229 M146 A148 Y207 Y208 I209 R137 T141 D235 D238 R117 T121 D215 D218 2.4.2.9 0004845,0005525,0016757,0044206 Ki=25uM remove_due_to_license_issue Q26998 9628859 999 QEESILQDIITRFPNVVLMKQTAQLRAMMTIIRDKETPKEEFVFYADRLIRLLIEEALNELPFQKKEVTTPLDVSYHGVSFYSKICGVSIVRAGESMESGLRAVCRGVRIGKILIQRDETTAEPKLIYEKLPADIRERWVMLLDPMCATAGSVCKAIEVLLRLGVKEERIIFVNILAAPQGIERVFKEYPKVRMVTAAVDICLNSRYYIVPGIGDFGDRYFGTM 1ur9 A 1.8 BS01 GDL C 1 Y10 W97 N142 E144 M212 Y214 D215 W403 Y8 W95 N140 E142 M210 Y212 D213 W401 D140 N142 E144 Y214 D138 N140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 remove_due_to_license_issue Q54276 14597613 1 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDINWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRVR 1ur9 A 1.8 BS02 PHJ A 1 W97 E144 F191 D215 W220 W95 E142 F189 D213 W218 D140 N142 E144 Y214 D138 N140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 remove_due_to_license_issue Q54276 14597613 2503 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDINWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRVR 1urw A 1.6 BS01 I1P A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A29 F67 F69 L70 H71 Q72 D73 K76 L121 D132 D127 K129 Q131 N132 D145 T165 D114 K116 Q118 N119 D132 T141 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50<0.003uM remove_due_to_license_issue IC50=<3nM P24941 15081018 1300 MENFQKVEKIGEYGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1usn A 1.8 BS06 IN9 A 1 Y155 H166 A167 Y168 A169 E202 H205 H211 Y73 H84 A85 Y86 A87 E120 H123 H129 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=0.018uM remove_due_to_license_issue Ki=18nM P08254 9792098 300 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYG 1utd L 2.1 BS01 rna 0 0 G18 F32 S35 E36 K37 D39 K56 G14 F28 S31 E32 K33 D35 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEGK 1utd M 2.1 BS01 rna 1 0 F32 E36 K37 K56 F28 E32 K33 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd N 2.1 BS01 rna 2 0 G18 F32 K37 D39 K56 G14 F28 K33 D35 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd O 2.1 BS01 rna 3 0 F32 E36 K37 D39 F28 E32 K33 D35 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEGK 1utd P 2.1 BS01 rna 4 0 G18 F32 E36 K37 D39 K56 G14 F28 E32 K33 D35 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd Q 2.1 BS01 rna 5 0 G18 F32 E36 K37 D39 K56 G14 F28 E32 K33 D35 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEGK 1utd R 2.1 BS01 rna 6 0 G18 F32 E36 K37 D39 K56 G14 F28 E32 K33 D35 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEGK 1utd S 2.1 BS01 rna 7 0 G18 F32 E36 K37 D39 K56 G14 F28 E32 K33 D35 K52 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd T 2.1 BS01 rna 8 0 G18 F32 E36 K37 D39 G14 F28 E32 K33 D35 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd T 2.1 BS02 rna 9 0 H34 E36 H30 E32 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd U 2.1 BS01 rna 9 0 G18 F32 E36 K37 D39 G14 F28 E32 K33 D35 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utd V 2.1 BS01 rna Z 0 G18 F32 E36 K37 D39 G14 F28 E32 K33 D35 ? 0003723,0005515,0006353,0006355,0042802 remove_due_to_license_issue Q9X6J6 15050822 101 ~ 106 TNSDFVVIKALEDGVNVIGLTRGADTRFHHSEKLDKGEVLIAQFTEHTSAIKVRGKAYIQTRHGVIESEG 1utj A 1.83 BS01 ABN A 1 D189 S190 C191 Q192 V213 W215 G219 D170 S171 C172 Q173 V190 W192 G195 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q173 G174 D175 S176 G177 3.4.21.4 0004252,0006508 Kd=0.144mM remove_due_to_license_issue P35031 15044735 246 IVGGYECKPYSQPHQVSLNSGYHFCGGSLVNENWVVSAAHCYKSRVEVRLGEHNIKVTEGSEQFISSSRVIRHPNYSSYNIDNDIMLIKLSKPATLNTYVQPVALPTSCAPAGTMCTVSGWGNTMSSTADSNKLQCLNIPILSYSDCNNSYPGMITNAMFCAGYLEGGKDSCQGDSGGPVVCNGELQGVVSWGYGCAEPGNPGVYAKVCIFNDWLTSTMASY 1utl M 1.7 BS01 PRA M 1 S190 S214 W215 G216 S171 S191 W192 G193 D102 G193 S195 G196 D84 G174 S176 G177 3.4.21.4 0004252,0006508 Ka=293M^-1 remove_due_to_license_issue P35031 15044735 246 IVGGYECKPYSQPHQVSLNSGYHFCGGSLVNENWVVSAAHCYKSRVEVRLGEHNIKVTEGSEQFISSSRVIRHPNYSSYNIDNDIMLIKLSKPATLNTYVQPVALPTSCAPAGTMCTVSGWGNTMSSTADSNKLQCLNIPILSYSDCNNSYPGMITNAMFCAGYLEGGKDSCQGDSGGPVVCNGELQGVVSWGYGCAEPGNPGVYAKVCIFNDWLTSTMASY 1utm A 1.5 BS01 PEA A 1 D189 S190 S195 D170 S171 S176 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q173 G174 D175 S176 G177 3.4.21.4 0004252,0006508 Ka=243M^-1 remove_due_to_license_issue P35031 15044735 246 IVGGYECKPYSQPHQVSLNSGYHFCGGSLVNENWVVSAAHCYKSRVEVRLGEHNIKVTEGSEQFISSSRVIRHPNYSSYNIDNDIMLIKLSKPATLNTYVQPVALPTSCAPAGTMCTVSGWGNTMSSTADSNKLQCLNIPILSYSDCNNSYPGMITNAMFCAGYLEGGKDSCQGDSGGPVVCNGELQGVVSWGYGCAEPGNPGVYAKVCIFNDWLTSTMASY 1utn A 1.15 BS01 ABN A 1 D189 S190 C191 Q192 S195 V213 W215 G219 D171 S172 C173 Q174 S177 V191 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Kd=0.321mM remove_due_to_license_issue P00760 15044735 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1utn A 1.15 BS02 ABN A 2 P173 G174 P153 G154 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Kd=0.321mM remove_due_to_license_issue P00760 15044735 247 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1uto A 1.15 BS01 PEA A 1 S190 Q192 S195 S214 W215 S172 Q174 S177 S192 W193 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Kd=5.32mM remove_due_to_license_issue P00760 15044735 1246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1utp A 1.3 BS01 PBN A 1 D189 S190 C191 S195 W215 D171 S172 C173 S177 W193 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 Kd=36mM remove_due_to_license_issue P00760 15044735 1246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1utr A -1.00 BS01 PCB A 1 L15 Y23 L43 I58 L61 T62 L12 Y20 L40 I55 L58 T59 ? 0007165 remove_due_to_license_issue P17559 7583672 78 ICPGFLQVLEALLLGSESNYEAALKPFNPASDLQNAGTQLKRLVDTLPQETRINIVKLTEKILTSPLC 1utr B -1.00 BS01 PCB A 1 L15 Y23 L43 I58 L61 T62 L12 Y20 L40 I55 L58 T59 ? 0007165 remove_due_to_license_issue P17559 7583672 78 ICPGFLQVLEALLLGSESNYEAALKPFNPASDLQNAGTQLKRLVDTLPQETRINIVKLTEKILTSPLC 1utt A 2.2 BS01 CP8 A 1 I180 L181 A182 L214 H218 V235 F237 P238 T239 Y240 K241 I75 L76 A77 L109 H113 V130 F132 P133 T134 Y135 K136 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=24uM remove_due_to_license_issue P39900 15289103 1266 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1utz A 2.5 BS01 PF3 A 1 G179 I180 L181 H218 E219 A234 V235 F237 T239 Y240 K241 G74 I75 L76 H113 E114 A129 V130 F132 T134 Y135 K136 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.014uM remove_due_to_license_issue IC50=14nM P39900 15289103 1265 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1utz A 2.5 BS02 PF3 A 2 S230 P232 F237 P238 S125 P127 F132 P133 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.014uM remove_due_to_license_issue IC50=14nM P39900 15289103 1266 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1utz B 2.5 BS01 PF3 A 2 D175 K177 G179 P238 D70 K72 G74 P133 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.014uM remove_due_to_license_issue IC50=14nM P39900 15289103 1266 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1utz B 2.5 BS02 PF3 B 1 I180 L181 A182 H218 E219 A234 V235 F237 T239 Y240 K241 I75 L76 A77 H113 E114 A129 V130 F132 T134 Y135 K136 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.014uM remove_due_to_license_issue IC50=14nM P39900 15289103 1265 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1uu3 A 1.7 BS01 LY4 A 1 L88 G89 A109 K111 V143 L159 S160 Y161 A162 G165 E166 E209 L212 T222 D223 L16 G17 A37 K39 V71 L87 S88 Y89 A90 G93 E94 E137 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T163 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.75uM remove_due_to_license_issue Kd=700nM, IC50=750nM O15530 14962382 1374 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 1uu7 A 1.9 BS01 BI2 A 1 L88 G89 A109 L159 S160 Y161 E166 E209 L212 T222 D223 L16 G17 A37 L87 S88 Y89 E94 E137 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T168 2.7.11.1 0004672,0004674,0005524,0006468 ic50=14uM remove_due_to_license_issue O15530 14962382 1364 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPRANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 1uu8 A 2.5 BS01 BI1 A 1 L88 G89 A109 S160 Y161 E166 E209 L212 T222 D223 L17 G18 A38 S89 Y90 E95 E138 L141 T151 D152 D205 K207 E209 N210 D223 T245 D134 K136 E138 N139 D152 T166 2.7.11.1 0004672,0004674,0005524,0006468 ic50=9uM remove_due_to_license_issue O15530 14962382 1368 PQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSNSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPK 1uu9 A 1.95 BS01 BI3 A 1 L88 G89 A109 K111 L159 S160 Y161 E166 L212 T222 D223 L17 G18 A38 K40 L88 S89 Y90 E95 L141 T151 D152 D205 K207 E209 N210 D223 T245 D134 K136 E138 N139 D152 T165 2.7.11.1 0004672,0004674,0005524,0006468 ic50=3.8uM remove_due_to_license_issue O15530 14962382 1370 PQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLNSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPK 1uv5 A 2.8 BS01 BRW A 1 I62 A83 L132 Y134 V135 P136 R141 L188 D200 A382 I28 A49 L98 Y100 V101 P102 R107 L154 D166 A348 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=1500nM P49841 14700633 1383 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQGKAFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 1uv6 C 2.5 BS01 CCE C 1 Y89 W143 Y185 C187 Y89 W143 Y185 C187 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=7575nM remove_due_to_license_issue P58154 15046723 1206 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 1uv6 D 2.5 BS01 CCE C 1 L112 M114 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=7575nM remove_due_to_license_issue P58154 15046723 1206 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 1uv6 D 2.5 BS02 CCE D 1 Y89 W143 Y185 C187 Y192 Y89 W143 Y185 C187 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=7575nM remove_due_to_license_issue P58154 15046723 1206 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 1uvr A 2.81 BS01 BI8 A 1 L88 G89 A109 L159 S160 Y161 E166 E209 L212 T222 D223 L18 G19 A39 L89 S90 Y91 E96 E139 L142 T152 D153 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T171 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 14962382 1372 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 1uvs H 2.8 BS02 I11 H 1 Y60A W60D L99 I174 D189 A190 W215 G216 G219 Y47 W50 L94 I166 D186 A187 W214 G215 G217 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 8939759 11 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRRYERNIEKISMLEKIYIHPRYNWRNLDRDIALMKLKPVAFSDYIHPVCLPDRTAASLLQAGYKGRVTGWGNLKETPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVI 1uvt H 2.5 BS02 I48 H 1 H57 Y60A W60D N98 L99 D189 A190 S195 S214 W215 G216 H43 Y47 W50 N95 L96 D192 A193 S198 S219 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.023uM remove_due_to_license_issue P00735 8939759 1 IVEGQDAEVGLSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTVDDLLVRIGKHSRTRYERKVEKISMLDKIYIHPRYNWKENLDRDIALLKLKRPIELSDYIHPVCLPDKQTAAKLLHAGFKGRVTGWGNRRETVQPSVLQVVNLPLVERPVCKASTRIRITDNMFCAGYKPGEGKRGDACEGDSGGPFVMKSPYNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIKVID 1uvu H 2.8 BS02 DCH H 1 H57 D189 A190 E192 S195 S214 W215 G216 G219 C220 H43 D192 A193 E195 S198 S219 W220 G221 G223 C224 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00735 8939759 1 IVEGQDAEVGLSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTVDDLLVRIGKHSRTRYERKVEKISMLDKIYIHPRYNWKENLDRDIALLKLKRPIELSDYIHPVCLPDKQTAAKLLHAGFKGRVTGWGNRRETVQPSVLQVVNLPLVERPVCKASTRIRITDNMFCAGYKPGEGKRGDACEGDSGGPFVMKSPYNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKWKVI 1uw6 A 2.2 BS01 NCT A 1 Y89 W143 Y192 Y90 W144 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=45.2nM remove_due_to_license_issue Ki=316.23nM, Kd=316nM P58154 15046723 1208 EFDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 1uw6 A 2.2 BS02 NCT E 1 W53 M114 W54 M115 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=45.2nM remove_due_to_license_issue Ki=316.23nM, Kd=316nM P58154 15046723 1206 EFDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 1uw6 B 2.2 BS01 NCT B 1 Y89 W143 Y192 Y90 W144 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=45.2nM remove_due_to_license_issue Ki=316.23nM, Kd=316nM P58154 15046723 1206 EFDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 1uwb A 3.2 BS01 TBO A 1 L100 K101 V106 Y188 W229 Y318 L100 K101 V106 Y188 W229 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 9000632 559 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRK 1uwf A 1.69 BS01 DEG A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 ? 0007155,0009289 Kd=0.15uM remove_due_to_license_issue P08191 15659162 1159 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 1uwh A 2.95 BS01 BAX A 1 A480 E500 L504 L513 T528 Q529 W530 C531 L566 F582 D593 F594 A34 E54 L58 L67 T82 Q83 W84 C85 L120 F136 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=22nM, Kd=260nM, Ki=22nM P15056 15035987 1723 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTAPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 1uwt A 1.95 BS01 GTL A 1 Q18 H150 E206 Y322 E387 W425 E432 W433 F441 Q18 H148 E204 Y318 E383 W421 E428 W429 F437 R79 H150 E206 V209 N320 Y322 E387 R79 H148 E204 V207 N316 Y318 E383 3.2.1.23 0004553,0004565,0005975,0008422,0016798 Ki=1.08uM remove_due_to_license_issue P22498 15147194 1490 MYSFPNSFRFGWSQAGFQSEMGTPGSEDPNTDWYKWVHDPENMAAGLVSGDLPENGPGYWGNYKTFHDNAQKMGLKIARLNVEWSRIFPNPLPRPFDESKQDVTEVEINENELKRLDEYANKDALNHYREIFKDLKSRGLYFILNMYHWPLPLWLHDPIRVRRGDFTGPSGWLSTRTVYEFARFSAYIAWKFDDLVDEYSTMNEPNVVGGLGYVGVKSGFPPGYLSFELSRRAMYNIIQAHARAYDGIKSVSKKPVGIIYANSSFQPLTDKDMEAVEMAENDNRWWFFDAIIRGEITREKIVRDDLKGRLDWIGVNYYTRTVVKRTEKGYVSLGGYGHGCERNSVSLAGLPTSDFGWEFFPEGLYDVLTKYWNRYHLYMYVTENGIADDADYQRPYYLVSHVYQVHRAINSGADVRGYLHWSLADNYEWASGFSMRFGLLKVDYNTKRLYWRPSALVYREIATNGAITDEIEHLNSVPPVKPLRH 1uwu A 1.95 BS01 GOX A 1 Q18 H150 E206 Y322 E387 W425 E432 F441 Q18 H148 E204 Y316 E381 W419 E426 F435 R79 H150 E206 V209 N320 Y322 E387 R79 H148 E204 V207 N314 Y316 E381 3.2.1.23 0004553,0004565,0005975,0008422,0016798 Ki=1.04uM remove_due_to_license_issue P22498 15147194 1490 MYSFPNSFRFGWSQAGFQSEMGTPGSEDPNTDWYKWVHDPENMAAGLVSGDLPENGPGYWGNYKTFHDNAQKMGLKIARLNVEWSRIFPNPLPRPFDESKQDVTEVEINENELKRLDEYANKDALNHYREIFKDLKSRGLYFILNMYHWPLPLWLHDPIRVRRGDFTGPSGWLSTRTVYEFARFSAYIAWKFDDLVDEYSTMNEPNVVGGLGYVGVKSGFPPGYLSFELSRRAMYNIIQAHARAYDGIKSVSKKPVGIIYANSSFQPLTDKDMEAVEMAENDNRWWFFDAIIRGEITKIVRDDLKGRLDWIGVNYYTRTVVKRTEKGYVSLGGYGHGCERNSVSLAGLPTSDFGWEFFPEGLYDVLTKYWNRYHLYMYVTENGIADDADYQRPYYLVSHVYQVHRAINSGADVRGYLHWSLADNYEWASGFSMRFGLLKVDYNTKRLYWRPSALVYREIATNGAITDEIEHLNSVPPVKPLRH 1uxa A 1.5 BS01 SIA D 1 Y312 P317 D318 K345 Y132 P137 D138 K165 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 15220447 2 YDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 1uxa B 1.5 BS01 SIA E 1 Y312 P317 D318 K345 Y130 P135 D136 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 15220447 2 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 1uxb A 1.75 BS01 SIA D 1 Y312 P317 D318 K345 Y131 P136 D137 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64822 15220447 2 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPEIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFDFSWSKTYENVEFETTSFTFSYIAQE 1uxb B 1.75 BS01 SIA E 1 Y312 P317 D318 K345 Y130 P135 D136 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64822 15220447 2 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPEIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFDFSWSKTYENVEFETTSFTFSYIAQE 1uy6 A 1.9 BS01 PU3 A 1 N51 A55 M98 L107 F138 V150 W162 T184 E223 N35 A39 M82 L91 F122 V134 W146 T168 E207 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50>200uM remove_due_to_license_issue P07900 15217611 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uy7 A 1.9 BS01 PU4 A 1 A55 M98 L107 F138 W162 T184 E223 A40 M83 L92 F123 W147 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50>200uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uy8 A 1.98 BS01 PU5 A 1 N51 A55 M98 L107 F138 V150 W162 E223 N35 A39 M82 L91 F122 V134 W146 E207 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=75uM remove_due_to_license_issue P07900 15217611 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uy9 A 2.0 BS01 PU6 A 1 N51 A55 M98 L107 F138 W162 E223 N36 A40 M83 L92 F123 W147 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=15.3uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uyc A 2.0 BS01 PU7 A 1 N51 A55 M98 L107 F138 Y139 W162 E223 N36 A40 M83 L92 F123 Y124 W147 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=41uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uyd A 2.2 BS01 PU8 A 1 N51 A55 M98 L107 F138 Y139 W162 T184 N36 A40 M83 L92 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50>200uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 1uye A 2.0 BS01 PU9 A 1 N51 A55 M98 L107 F138 Y139 W162 N36 A40 M83 L92 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50>200uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 1uyf A 2.0 BS01 PU1 A 1 N51 A55 G97 M98 L107 F138 Y139 V150 W162 T184 N36 A40 G82 M83 L92 F123 Y124 V135 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=30uM remove_due_to_license_issue EC50=1200nM P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 1uyg A 2.0 BS01 PU2 A 1 N51 A55 G97 M98 L107 F138 Y139 W162 E223 N36 A40 G82 M83 L92 F123 Y124 W147 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=53.5uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uyh A 2.2 BS01 PU0 A 1 N51 A55 G97 M98 L107 F138 W162 E223 N36 A40 G82 M83 L92 F123 W147 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=14.3uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uyi A 2.2 BS01 PUZ A 1 N51 A55 G97 M98 D102 L107 I110 F138 W162 E223 N36 A40 G82 M83 D87 L92 I95 F123 W147 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=4.1uM remove_due_to_license_issue P07900 15217611 1224 HVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uyk A 2.2 BS01 PUX A 1 N51 A55 I96 G97 M98 L107 F138 W162 T184 E223 N36 A40 I81 G82 M83 L92 F123 W147 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=17.1uM remove_due_to_license_issue P07900 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1uym A 2.45 BS01 PU3 A 1 N51 A55 D93 M98 L107 F138 Y139 V150 T184 E225 N36 A40 D78 M83 L92 F123 Y124 V135 T169 E210 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=>200000nM, EC50=3200nM P08238 15217611 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYLEKE 1uys A 2.8 BS01 H1L A 1 A1627 G1734 I1735 Y1738 L1756 A146 G253 I254 Y257 L275 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 15079078 3000 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 1uys B 2.8 BS01 H1L B 1 A1627 G1734 I1735 Y1738 A146 G253 I254 Y257 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 15079078 3000 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 1uys B 2.8 BS02 H1L C 1 W1924 F1956 V1967 L1968 G1997 G1998 V2001 V2002 W443 F475 V480 L481 G510 G511 V514 V515 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 15079078 3000 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 1uz1 A 2.0 BS01 IFL A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y292 E345 W392 E399 W400 F408 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N290 Y292 E345 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Ki=130nM remove_due_to_license_issue Q08638 15515081 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 1uz4 A 1.71 BS01 IFL A 1 W137 N214 E215 W285 E330 W376 Q403 E404 Y409 W116 N193 E194 W264 E309 W355 Q382 E383 Y388 ? 0004553,0016798,0016985 Ki=400uM remove_due_to_license_issue Q6QT42 15515081 1432 EHFVRVNGGHFELQGKPYVITGVNMWYAAYLGAPNEVGDRDRLAKELDNLKAIGVNNLRVLAVSEKSEINSAVKPAVTNGFGNYDETLLQGLDYLLVELAKRDMTVVLYFNNFWQWSGGMTQYMAWIEGEPVQDPNVTNEWEAFMAKSASFYRSEKAQQEYRKTLEKIITRVNSINGKAYVDDATIMSWQLANEPRPGNSQTTAEEKQIYIDWVHAAAAYIKTLDAHHLVSSGSEGEMGSVNDMQVFIDAHATPDIDYLTYHMWIRNWSWFDKTKPAETWPSAWEKAQNYMRAHIDVAKQLNKPLVLEEFGLDRDMGSYAMDSTTEYRDNYFRGVFELMLASLEQGEPSAGYNIWAWNGYGRTTRANYWWQEGDDFMGDPPQEEQGMYGVFDTDTSTIAIMKEFNARFQP 1uz8 A 1.8 BS01 MAG C 1 Y32 N91 L92 V94 Y37 N96 L97 V99 remove_due_to_license_issue 15242599 1 DIVMTQAAFSNPVTLGTSASISCRSSKSLLYSNGITYLYWYLQKPGQSPQLLIYQMSNLASGVPDRFSSSGSGTDFTLRISRVEAEDVGVYYCAQNLEVPWTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1uz8 A 1.8 BS02 FUC C 1 Y32 Y34 Q50 N91 Y37 Y39 Q55 N96 remove_due_to_license_issue 15242599 2 DIVMTQAAFSNPVTLGTSASISCRSSKSLLYSNGITYLYWYLQKPGQSPQLLIYQMSNLASGVPDRFSSSGSGTDFTLRISRVEAEDVGVYYCAQNLEVPWTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 1uz8 B 1.8 BS01 GAL C 1 W33 E50 T96 W33 E50 T100 remove_due_to_license_issue 15242599 3 EVKLLESGGGLVQPGGSQKLSCAASGFDFSGYWMSWVRQAPGKGLEWIGEINPDSSTINYTPSLKDKFIISRDNAKNTLYLQMSKVRSEDTALYYCARETGTRFDYWGQGTTLTVSSATTTAPSVYPLVPGGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKTELIKRIEPR 1uze A 1.82 BS05 EAL A 1 Q281 H353 A354 H383 E384 H387 E411 K511 F512 H513 V518 Y520 Y523 Q242 H314 A315 H344 E345 H348 E372 K468 F469 H470 V475 Y477 Y480 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H470 Y480 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue IC50=1.2nM P12821 15236580 3002 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWP 1v0k A 1.03 BS01 XYP A 1 E44 N45 K48 Q88 G302 E43 N44 K47 Q87 G301 E128 N170 H207 E236 D238 E127 N169 H206 E235 D237 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1303 ESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNG 1v0k A 1.03 BS02 XDN A 1 K48 H81 W85 N127 E128 Q205 E236 W266 W274 K47 H80 W84 N126 E127 Q204 E235 W265 W273 E128 N170 H207 E236 D238 E127 N169 H206 E235 D237 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1304 ESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNG 1v0l A 0.98 BS01 XIF A 1 K48 H81 W85 E128 Q205 E236 W266 W274 K47 H80 W84 E127 Q204 E235 W265 W273 E128 N170 H207 E236 D238 E127 N169 H206 E235 D237 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1304 ESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNGG 1v0l A 0.98 BS02 XYP A 1 E44 N45 K48 Q88 E43 N44 K47 Q87 E128 N170 H207 E236 D238 E127 N169 H206 E235 D237 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1305 ESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNGG 1v0m A 1.07 BS01 XDN A 1 K48 H81 W85 N127 Q205 E236 W266 W274 G302 K48 H81 W85 N127 Q205 E236 W266 W274 G302 E128 N170 H207 E236 D238 E128 N170 H207 E236 D238 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1303 AESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNG 1v0m A 1.07 BS02 XYP A 1 E44 N45 K48 Q88 E44 N45 K48 Q88 E128 N170 H207 E236 D238 E128 N170 H207 E236 D238 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1304 AESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNG 1v0n A 1.1 BS01 XIF A 1 K48 H81 W85 E128 Q205 E236 W266 W274 K48 H81 W85 E128 Q205 E236 W266 W274 E128 N170 H207 E236 D238 E128 N170 H207 E236 D238 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1305 AESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNG 1v0n A 1.1 BS02 XYP A 1 E44 N45 K48 Q88 E44 N45 K48 Q88 E128 N170 H207 E236 D238 E128 N170 H207 E236 D238 3.2.1.8 0004553,0005975 remove_due_to_license_issue P26514 15306887 1306 AESTLGAAAAQSGRYFGTAIASGRLSDSTYTSIAGREFNMVTAENEMKIDATEPQRGQFNFSSADRVYNWAVQNGKQVRGHTLAWHSQQPGWMQSLSGSALRQAMIDHINGVMAHYKGKIVQWDVVNEAFADGSSGARRDSNLQRSGNDWIEVAFRTARAADPSAKLCYNDYNVENWTWAKTQAMYNMVRDFKQRGVPIDCVGFQSHFNSGSPYNSNFRTTLQNFAALGVDVAITELDIQGAPASTYANVTNDCLAVSRCLGITVWGVRDSDSWRSEQTPLLFNNDGSKKAAYTAVLDALNG 1v0o A 1.9 BS01 INR A 1 I10 A30 K32 F79 H81 L82 D83 L132 D143 I8 A28 K30 F69 H71 L72 D73 L122 D133 D125 K127 Q129 N130 D143 K156 T163 D115 K117 Q119 N120 D133 K146 T153 2.7.11.22,2.7.11.23 0004672,0004674,0004693,0005524,0005634,0005737,0006357,0006468,0008353,0046872,0051301,0051726,0106310,0140833,0140834,0140835,0140836,0140837 ic50=5.5uM remove_due_to_license_issue Q07785 14604523 2638 KYHGLEKIGEGTYGVVYKAQNNYGETFALKKIRLSTTIREISILKELKHSNIVKLYDVIHTKKRLVLVFEHLDQDLKKLLDVCEGGLESVTAKSFLLQLLNGIAYCHDRRVLHRDLKPQNLLINREGELKIADFGLARAFGIPVRKYTHEVVTLWYRAPDVLMGSKKYSTTIDIWSVGCIFAEMVNGTPLFPGVSEADQLMRIFRILGTPNSKNWPNVTELPKYDPNFTVYEPLPWESFLKGLDESGIDLLSKMLKLDPNQRITAKQALEHAYFKE 1v0p A 2.0 BS01 PVB A 1 I10 G11 G13 V18 A30 F79 L82 D83 D85 Q129 L132 I10 G11 G13 V18 A30 F79 L82 D83 D85 Q129 L132 D125 K127 Q129 N130 D143 T163 D125 K127 Q129 N130 D143 T154 2.7.11.22,2.7.11.23 0004672,0004674,0004693,0005524,0005634,0005737,0006357,0006468,0008353,0046872,0051301,0051726,0106310,0140833,0140834,0140835,0140836,0140837 ic50=0.13uM remove_due_to_license_issue Q07785 14604523 1287 MEKYHGLEKIGEGTYGVVYKAQNNYGETFALKKIRLEKEDEGIPSTTIREISILKELKHSNIVKLYDVIHTKKRLVLVFEHLDQDLKKLLDVCEGGLESVTAKSFLLQLLNGIAYCHDRRVLHRDLKPQNLLINREGELKIADFGLARAFGIVTLWYRAPDVLMGSKKYSTTIDIWSVGCIFAEMVNGTPLFPGVSEADQLMRIFRILGTPNSKNWPNVTELPKYDPNFTVYEPLPWESFLKGLDESGIDLLSKMLKLDPNQRITAKQALEHAYFKE 1v1j A 2.2 BS01 FA3 A 1 Y28 N79 A81 A82 H85 H106 I107 S108 R117 Y28 N79 A81 A82 H85 H106 I107 S108 R117 P15 N16 R23 Y28 N79 A82 E104 H106 R113 P15 N16 R23 Y28 N79 A82 E104 H106 R113 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=15uM remove_due_to_license_issue P15474 15162210 201 PRSLANAPIMILNGPNLNLLGQRQPEIYGSDTLADVEALCVKAAAAHGGTVDFRQSNHEGELVDWIHEARLNHCGIVINPAAYSHTSVAILDALNTCDGLPVVEVHISNIHQREPFRHHSYVSQRADGVVAGCGVQGYVFGVERIAALAG 1v1j B 2.2 BS01 FA3 B 1 Y28 N79 A81 A82 H85 H106 I107 S108 R117 Y28 N79 A81 A82 H85 H106 I107 S108 R117 P15 N16 R23 Y28 N79 A82 E104 H106 R113 P15 N16 R23 Y28 N79 A82 E104 H106 R113 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=15uM remove_due_to_license_issue P15474 15162210 201 PRSLANAPIMILNGPNLNLLGQRQPEIYGSDTLADVEALCVKAAAAHGGTVDFRQSNHEGELVDWIHEARLNHCGIVINPAAYSHTSVAILDALNTCDGLPVVEVHISNIHQREPFRHHSYVSQRADGVVAGCGVQGYVFGVERIAALAG 1v1k A 2.31 BS01 3FP A 1 I10 G11 V18 A31 L83 D86 K89 N132 L134 I10 G11 V18 A31 L74 D77 K80 N123 L125 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=35uM remove_due_to_license_issue IC50=35000nM P24941 12941311 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1v2h E 2.7 BS01 GUN E 1 A117 G118 E201 M219 T242 N243 A116 G117 E200 M218 T241 N242 S33 H64 Y88 A116 M219 S220 H257 S32 H63 Y87 A115 M218 S219 H256 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 14680831 290 ENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS 1v2j T 1.9 BS02 BEN T 1 D189 S190 Q192 S195 V213 G219 D171 S172 Q174 S177 V191 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=566uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSRIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2k T 2.0 BS02 ZEN T 1 Y99 F174 A190 Q192 V213 W215 G216 G219 C220 V227 Y228 Y81 F154 A172 Q174 V191 W193 G194 G196 C197 V205 Y206 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.65uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSETYNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSFIITSNMFCAGYLEGGKDACQGDSGGPVVCSGKLQGIVSWGEGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2l T 1.6 BS02 BEN T 1 D189 A190 C191 S195 G219 D171 A172 C173 S177 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=51uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSETYNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSFIITSNMFCAGYLEGGKDACQGDSGGPVVCSGKLQGIVSWGEGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2m T 1.65 BS01 BEN T 1 D189 A190 G219 D171 A172 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=51uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSETYNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSFIITSNMFCAGYLEGGKDACQGDSGGPVVCSGKLQGIVSWGEGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2n T 1.8 BS02 BBA T 1 T98 Y99 D189 A190 Q192 W215 G216 G219 C220 T80 Y81 D171 A172 Q174 W193 G194 G196 C197 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.25uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSETYNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSFIITSNMFCAGYLEGGKDACQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2o T 1.62 BS02 ANH T 1 D189 S190 C191 Q192 S214 W215 G216 G219 C220 D171 S172 C173 Q174 S192 W193 G194 G196 C197 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=18.45uM remove_due_to_license_issue P00760 14729347 800 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSYIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2p T 1.92 BS02 ANH T 1 T98 D189 S190 W215 G216 G219 T80 D171 S172 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=18.45uM remove_due_to_license_issue P00760 14729347 800 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSYIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2q T 2.3 BS02 ANH T 1 D189 S190 C191 Q192 W215 G216 G219 D171 S172 C173 Q174 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=73.62uM remove_due_to_license_issue P00760 14729347 800 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSWIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2r T 1.7 BS02 ANH T 1 D189 S190 C191 Q192 S195 W215 G216 G219 C220 D171 S172 C173 Q174 S177 W193 G194 G196 C197 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=278.96uM remove_due_to_license_issue P00760 14729347 800 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSRIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2s T 1.72 BS02 BEN T 1 D189 S190 C191 S195 V213 G219 D171 S172 C173 S177 V191 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=68uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSFIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGEGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2t T 1.9 BS02 ANH T 1 D189 S190 C191 Q192 S195 W215 G216 G219 D171 S172 C173 Q174 S177 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=19.56uM remove_due_to_license_issue P00760 14729347 800 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSFIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGEGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2u T 1.8 BS02 BEN T 1 D189 S190 S195 V213 G219 D171 S172 S177 V191 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=427uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSAIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2v T 1.8 BS02 BEN T 1 D189 S190 C191 Q192 S195 V213 G216 G219 C220 D171 S172 C173 Q174 S177 V191 G194 G196 C197 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=427uM remove_due_to_license_issue P00760 14729347 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSAIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v2w T 1.75 BS02 ANH T 1 D189 S190 C191 Q192 S195 S214 W215 G216 G219 D171 S172 C173 Q174 S177 S192 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=97.79uM remove_due_to_license_issue P00760 14729347 800 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSASSAIITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1v3x A 2.2 BS03 D76 A 1 T98 Y99 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G218 C220 G226 I227 Y228 T84 Y85 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=24nM remove_due_to_license_issue IC50=24nM P00742 15456260 700 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 1v41 E 2.85 BS01 AZG E 1 A116 A117 G118 F200 E201 V217 M219 T242 N243 A115 A116 G117 F199 E200 V216 M218 T241 N242 S33 H64 Y88 A116 M219 S220 H257 S32 H63 Y87 A115 M218 S219 H256 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 15983407 290 ENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS 1v48 A 2.2 BS01 HA1 A 1 S33 R84 H86 A116 G118 F200 E201 V217 M219 S220 N243 S32 R77 H79 A109 G111 F193 E194 V210 M212 S213 N236 S33 H86 Y88 E89 A116 M219 S220 N243 V245 S32 H79 Y81 E82 A109 M212 S213 N236 V238 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Ki=16nM remove_due_to_license_issue Ki=2.7nM, IC50=18.7nM, Kd=0.46nM P55859 15272165 290 QNGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPESGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGENPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYEAAQKLEQFVSLLMASIPV 1v79 A 2.5 BS02 FR7 A 1 H17 D19 L62 F65 L106 W117 M155 G184 D296 H14 D16 L59 F62 L103 W114 M152 G181 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=13nM remove_due_to_license_issue P56658 15139750 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1v7a A 2.5 BS02 FRC A 1 H17 D19 F61 L62 F65 L106 M155 G184 D185 D296 H14 D16 F58 L59 F62 L103 M152 G181 D182 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=9.8nM remove_due_to_license_issue P56658 15139750 1001 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1vcj A 2.4 BS01 IBA A 1 R116 E117 D149 R150 W177 E226 E276 R292 R374 Y409 R39 E40 D72 R73 W100 E149 E199 R215 R297 Y332 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=26uM remove_due_to_license_issue P03474 15159560 1 PEWTYPRLSCQGSTFQKALLISPHRFGEIKGNSAPLIIREPFVACGPKECRHFALTHYAAQPGGYYNGTRKDRNKLRHLVSVKLGKIPTVENSIFHMAAWSGSACHDGREWTYIGVDGPDNDALVKIKYGEAYTDTYHSYAHNILRTQESACNCIGGDCYLMITDGSASGISKCRFLKIREGRIIKEILPTGRVEHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTKTYLDTPRPDDGSIAGPCESNGDKWLGGIKGGFVHQRMASKIGRWYSRTMSKTNRMGMELYVRYDGDPWTDSDALTLSGVMVSIEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKDTWHSAATAIYCLMGSGQLLWDTVTGVDMAL 1vcu A 2.85 BS01 DAN A 1 R21 D46 M85 E111 Y179 Y181 L217 R237 R304 Y334 R21 D46 M85 E111 Y179 Y181 L217 R234 R297 Y327 D46 E218 D46 E218 3.2.1.18 0004308,0005515,0005737,0005764,0005829,0006516,0006689,0009313,0016020,0016042,0016798,0046479,1902494 remove_due_to_license_issue Ki=25000nM, IC50=37000nM Q9Y3R4 15501818 381 MASLPVLQKESVFQSGAHAYRIPALLYLPGQQSLLAFAEQRASKKDEHAELIVLRRGDYDAPTHQVQWQAQEVVAQARLDGHRSMNPCPLYDAQTGTLFLFFIAIPGQVTEQQQLQTRANVTRLCQVTSTDHGRTWSSPRDLTDAAIGPAYREWSTFAVGPGHCLQLNDRARSLVVPAYAYRKLHPIQRPIPSAFCFLSHDHGRTWARGHFVAQDTLECQVAEVEQRVVTLNARSHLRARVQAQSTNDGLDFQESQLVKKLVEPPPQGCQGSVISFPSPRSPAQWLLYTHPTHSWQRADLGAYLNPRPPAPEAWSEPVLLAKGSCAYSDLQSMGTGPDGSPLFGCLYEANDYEEIVFLMFTLKQAFPAEY 1vea A 2.8 BS01 HBN B 1 G85 R88 E139 T140 F141 G80 R83 E134 T135 F136 ? 0003723,0003729,0006547,0010628 remove_due_to_license_issue P10943 15242603 1001 ERRIGRLSVLLLLNEAEESTQVEELERDGWKVCLGKVGSMDAHKVIAAIETASKKSGVIQSEGYRESHALYHATMEALHGVTRGEMLLGSLLRTVGLRFAVLRGNPYESEAEGDWIAVSLYGTIGAPIKGLEHETFGVGINHI 1vea B 2.8 BS01 HBN B 1 E81 H84 G85 V143 E77 H80 G81 V139 ? 0003723,0003729,0006547,0010628 remove_due_to_license_issue P10943 15242603 1001 KERRIGRLSVLLLLNEAEESTQVEELERDGWKVCLGKVGSMDAHKVIAAIETASKKSGVIQSEGYRESHALYHATMEALHGVTRGEMLLGSLLRTVGLRFAVLRGNPYESEAEGDWIAVSLYGTIGAPIKGLEHETFGVGINHI 1veb A 2.89 BS02 I05 A 1 G50 T51 G52 F54 A70 K72 L74 E91 M120 V123 E170 N171 L173 T183 D184 G186 G41 T42 G43 F45 A61 K63 L65 E82 M111 V114 E161 N162 L164 T174 D175 G177 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue IC50=39nM P00517 14998327 351 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1vfc A -1.00 BS01 dna B 0 K446 K447 G468 W470 A471 K488 D489 R492 K9 K10 G31 W33 A34 K51 D52 R55 ? 0000723,0000781,0005634,0031848,0042162 remove_due_to_license_issue Q15554 15608118 1 ~ 13 EDSTTNITKKQKWTVEESEWVKAGVQKYGEGNWAAISKNYPFVNRTAVMIKDRWRTMKRLGMN 1vfc A -1.00 BS02 dna C 0 K447 Q448 K449 W450 M486 D489 R490 K10 Q11 K12 W13 M49 D52 R53 ? 0000723,0000781,0005634,0031848,0042162 remove_due_to_license_issue Q15554 15608118 14 ~ 26 EDSTTNITKKQKWTVEESEWVKAGVQKYGEGNWAAISKNYPFVNRTAVMIKDRWRTMKRLGMN 1vfn A 2.15 BS01 HPA A 1 A117 G118 F200 E201 V217 N243 A107 G108 F190 E191 V207 N233 S33 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S30 H76 Y78 E79 A106 M209 S210 N233 V235 H245 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Ki=2.5uM remove_due_to_license_issue Kd=680nM P55859 9020983 300 GYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPEGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGQNPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDSQGKANHEEVLEAGKQAAQKLEQFVSLLMASI 1vgc C 1.9 BS02 V36 C 1 S190 C191 M192 G193 S195 W215 G216 S40 C41 M42 G43 S45 W65 G66 M192 G193 D194 S195 G196 M42 G43 D44 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 9425066 358 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 1vij A 2.4 BS01 BAY A 1 R8 D25 G27 D29 K45 I47 G48 G49 I50 P81 I84 R8 D25 G27 D29 K45 I47 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=0.3nM remove_due_to_license_issue P12499 9346283 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1vij B 2.4 BS01 BAY A 1 R8 D25 D29 I47 G49 I50 P81 V82 R8 D25 D29 I47 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 9346283 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1vik A 2.4 BS01 BAY B 1 D25 G27 I47 G48 G49 I50 V82 I84 D25 G27 I47 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 9346283 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1vik B 2.4 BS01 BAY B 1 R8 D25 G27 D29 I47 G48 F53 P81 V82 R8 D25 G27 D29 I47 G48 F53 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=0.3nM remove_due_to_license_issue P12499 9346283 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1vj5 A 2.35 BS03 CIU A 1 D333 W334 M337 Y381 Q382 Y465 D334 W335 M338 Y382 Q383 Y465 F265 H332 D333 W334 N357 N376 Y381 Y465 D495 H523 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.12uM remove_due_to_license_issue P34913 15096040 781 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 1vj9 U 2.4 BS01 5IN U 1 L97B H99 D189 S190 Q192 S195 S214 W215 G216 R217 G219 G226 L92 H94 D192 S193 Q195 S198 S217 W218 G219 R220 G221 G229 3.4.21.73 0004252,0006508 Ki=0.028uM remove_due_to_license_issue P00749 15150279 300 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1vja U 2.0 BS01 7IN U 1 L97B H99 D189 S190 Q192 S195 W215 G216 R217 G219 C220 G226 L92 H94 D192 S193 Q195 S198 W218 G219 R220 G221 C222 G229 3.4.21.73 0004252,0006508 Ki=0.02uM remove_due_to_license_issue IC50=20nM, Ki=20nM P00749 15150279 300 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1vjb A 3.2 BS01 OHT A 1 L268 C269 A272 D273 E275 V313 Y326 L345 L35 C36 A39 D40 E42 V80 Y93 L112 ? remove_due_to_license_issue IC50=1350nM, EC50=15nM P62508 15161930 100 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLE 1vjc A 2.1 BS01 ATP A 1 G213 K219 G238 G340 V341 E343 D374 G213 K219 G238 G340 V341 E343 D374 R38 K215 G373 G396 R38 K215 G373 G396 2.7.2.3 0004618,0005524,0005737,0005759,0005829,0006094,0006096,0016301,0043531 Kd=0.263mM remove_due_to_license_issue Q7SIB7 15035615 417 SLSNKLTLDKLDVKGKRVVMRVDFNVPMKNNQITNNQRIKAAIPSIKFCLDNGAKSVVLMSHLGRPDGIPMPDKYSLEPVAVELKSLLGKDVLFLKDCVGPEVEKACADPAAGSVILLENLRFHVEEEGKGKDASGSKVKADPAKIEAFRASLSKLGDVYVNDAFGTAHRAHSSMVGVNLPKKAGGFLMKKELNYFAKALESPERPFLAILGGAKVADKIQLINNMLDKVNEMIIGGGMAFTFLKVLNNMEIGTSLFDEEGSKIVKDLMSKAEKNGVKITLPVDFVTADKFDENAKTGQATVASGIPAGWMGLDCGPESSKKYSEAVARAKQIVWNGPVGVFEWEAFAQGTKALMDEVVKATSRGCITIIGGGDTATCCAKWNTEDKVSHVSTGGGASLELLEGKVLPGVDALSNV 1vjd A 1.9 BS01 ATP A 1 G213 A214 K219 G237 G238 G312 G337 P338 G340 V341 E343 G372 G373 D374 T375 G213 A214 K219 G237 G238 G312 G337 P338 G340 V341 E343 G372 G373 D374 T375 R38 K215 G373 G396 R38 K215 G373 G396 2.7.2.3 0004618,0005524,0005737,0005759,0005829,0006094,0006096,0016301,0043531 Kd=0.286mM remove_due_to_license_issue Q7SIB7 15035615 417 SLSNKLTLDKLDVKGKRVVMRVDFNVPMKNNQITNNQRIKAAIPSIKFCLDNGAKSVVLMSHLGRPDGIPMPDKYSLEPVAVELKSLLGKDVLFLKDCVGPEVEKACADPAAGSVILLENLRFHVEEEGKGKDASGSKVKADPAKIEAFRASLSKLGDVYVNDAFGTAHRAHSSMVGVNLPKKAGGFLMKKELNYFAKALESPERPFLAILGGAKVADKIQLINNMLDKVNEMIIGGGMAFTFLKVLNNMEIGTSLFDEEGSKIVKDLMSKAEKNGVKITLPVDFVTADKFDENAKTGQATVASGIPAGWMGLDCGPESSKKYSEAVARAKQIVWNGPVGVFEWEAFAQGTKALMDEVVKATSRGCITIIGGGDTATCCAKWNTEDKVSHVSTGGGASLELLEGKVLPGVDALSNV 1vjy A 2.0 BS01 460 A 1 I211 A230 K232 L260 L278 S280 Y282 H283 L340 D351 I11 A30 K32 L60 L78 S80 Y82 H83 L140 D151 D333 K335 N338 D351 T375 D133 K135 N138 D151 T171 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.023uM remove_due_to_license_issue P36897 15317461 999 IARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEGIKM 1vkj A 2.5 BS02 A3P A 1 K68 G70 T71 R72 A73 R151 S159 F258 L270 K274 G275 R276 K15 G17 T18 R19 A20 R98 S106 F205 L217 K221 G222 R223 2.8.2.23 0005794,0005796,0006024,0008146,0008467,0015012,0016740 Kd=14uM remove_due_to_license_issue O35310 15060080 602 STQQLPQTIIIGVRKGGTRALLEMLSLHPDVAAAENEVHFFDWEEHYSQGLGWYLTQMPFSSPHQLTVEKTPAYFTSPKVPERIHSMNPTIRLLLILRDPSERVLSDYTQVLYNHLQKHKPYPPIEDLLMRDGRLNLDYKALNRSLYHAHMLNWLRFFPLGHIHIVDGDRLIRDPFPEIQKVERFLKLSPQINASNFYFNKTKGFYCLRDSGKDRCLHESKGRAHPQVDPKLLDKLHEYFHEPNKKFFKLVGRTFDWH 1vot A 2.5 BS01 HUP A 1 W84 G118 Y121 G123 Y130 H440 W81 G115 Y118 G120 Y127 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=250nM remove_due_to_license_issue IC50=11.4nM P04058 8989325 999 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNATAC 1vru A 2.4 BS01 AAP A 1 L100 V106 Y181 Y188 G190 W229 Y318 L98 V104 Y179 Y186 G188 W227 Y316 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=0.1uM remove_due_to_license_issue P04585 7540934 999 SPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAH 1vsn A 2.0 BS01 NFT A 1 G23 C25 N60 D61 G64 G65 G66 Y67 N158 G23 C25 N60 D61 G64 G65 G66 Y67 N161 Q19 C25 H159 N175 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 16413777 283 APDSIDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKATGALLNLAPQNLVDCVSENDGCGGGYMTNAFQYVQRNRGIDSEDAYPYVGQDESCMYNPTGKAAKCRGYREIPEGNEAALKRAVAAVGPVSVAIDASLTSFQFYSAGVYYDENCSSDALNHAVLAVGYGIQAGNKHWIIKNSWGESWGNAGYILMARNKNNACGIANLASFPKM 1vso A 1.85 BS01 AT1 A 1 E13 Y61 P88 L89 T90 R95 G140 S141 E190 Y216 E9 Y57 P79 L80 T81 R86 G131 S132 E178 Y204 ? 0015276,0016020 Ki=18980nM remove_due_to_license_issue Ki=2900nM P22756 17581823 258 TLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNG 1vyf A 1.85 BS01 OLA A 1 R127 Y129 R129 Y131 ? 0005737,0008289 Kd=9nM remove_due_to_license_issue P29498 15476393 1134 GSMSSFLGKWKLSESHNFDAVMSKLGVSWATRQIGNTVTPTVTFTMDGDKMTMLTESTFKNLSCTFKFGEEFDEKTSDGRNVKSVVEKNSESKLTQTQVDPKNTTVIVREVDGDTMKTTVTVGDVTAIRNYKRLS 1vyg A 2.4 BS01 ACD A 1 F16 M20 V25 G33 S55 S75 D76 R78 I105 R107 T116 Y129 F18 M22 V27 G35 S57 S77 D78 R80 I107 R109 T118 Y131 ? 0005737,0008289 Kd=10nM remove_due_to_license_issue P29498 15476393 1134 GSMSSFLGKWKLSESHNFDAVMSKLGVSWATRQIGNTVTPTVTFTMDGDKMTMLTESTFKNLSCTFKFGEEFDEKTSDGRNVKSVVEKNSESKLTQTQVDPKNTTVIVREVDGDTMKTTVTVGDVTAIRNYKRLS 1vyq A 2.4 BS01 DUX A 1 F46 L88 N103 G106 Y112 I117 F44 L69 N84 G87 Y93 I98 S27 R91 S93 L99 D109 S25 R72 S74 L80 D90 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=4.98uM remove_due_to_license_issue Ki=5000nM Q8II92 15698576 1160 MHLKIVCLSDEVREMYKNHKTHHDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDET 1vyq A 2.4 BS02 DUX C 1 S92 S93 S95 S73 S74 S76 S27 R91 S93 L99 D109 S25 R72 S74 L80 D90 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=4.98uM remove_due_to_license_issue Ki=5000nM Q8II92 15698576 1160 MHLKIVCLSDEVREMYKNHKTHHDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDET 1vyq B 2.4 BS01 DUX A 1 S92 S93 S78 S79 S27 R91 S93 L99 D109 S27 R77 S79 L85 D95 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=4.98uM remove_due_to_license_issue Ki=5000nM Q8II92 15698576 1160 MHLKIVCLSDEVREMYKNHKTHHEGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEE 1vyq B 2.4 BS02 DUX B 1 G106 Y112 I117 G92 Y98 I103 S27 R91 S93 L99 D109 S27 R77 S79 L85 D95 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=4.98uM remove_due_to_license_issue Ki=5000nM Q8II92 15698576 1160 MHLKIVCLSDEVREMYKNHKTHHEGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEE 1vyw A 2.3 BS01 292 A 1 E8 I10 A31 F80 F82 L83 Q85 K89 L134 E12 I14 A35 F84 F86 L87 Q89 K93 L138 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=37nM remove_due_to_license_issue IC50=37nM P24941 15189033 2300 PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1vyz A 2.21 BS01 N5B A 1 I10 A31 F80 E81 F82 L83 H84 D86 L134 I10 A31 F69 E70 F71 L72 H73 D75 L123 D127 K129 Q131 N132 D145 T165 D116 K118 Q120 N121 D134 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=290nM remove_due_to_license_issue IC50=290nM P24941 15189033 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1vzq H 1.54 BS03 SHY H 1 H57 Y60A E97A N98 L99 D189 A190 E192 S214 W215 G216 H43 Y47 E94 N95 L96 D192 A193 E195 S219 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=36nM remove_due_to_license_issue P00734 1256 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTAYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1w0x C 2.2 BS01 OLO C 1 I10 A31 F82 L83 Q85 Q131 L134 I10 A31 F75 L76 Q78 Q124 L127 N132 D145 N125 D138 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=7000nM P24941 7479711 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1w0y H 2.5 BS01 771 H 1 H57 T99 D189 S190 K192 S195 S214 W215 G216 G219 H41 T87 D183 S184 K186 S189 S208 W209 G210 G212 3.4.21.21 0004252,0006508 Ki=0.38uM remove_due_to_license_issue Ki=380nM P08709 15664864 1258 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1w0z U 1.9 BS01 SI1 U 1 L97B H99 D189 S190 S195 V213 W215 G216 R217 G219 L92 H94 D192 S193 S198 V216 W218 G219 R220 G221 3.4.21.73 0004252,0006508 Ki=21nM remove_due_to_license_issue P00749 12684001 1245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1w10 U 2.0 BS01 SJ1 U 1 H57 L97B D189 S190 C191 Q192 S195 S214 W215 G216 G219 H46 L92 D192 S193 C194 Q195 S198 S217 W218 G219 G221 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 12684001 1245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1w11 U 2.0 BS01 SK1 U 1 H57 L97B H99 D189 S190 C191 Q192 S195 W215 G216 G219 C220 H46 L92 H94 D192 S193 C194 Q195 S198 W218 G219 G221 C222 3.4.21.73 0004252,0006508 Ki=6nM remove_due_to_license_issue Ki=7.7nM P00749 12684001 1247 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1w12 U 2.4 BS01 SL1 U 1 H57 T97A L97B A98 H99 D189 S190 C191 Q192 S195 S214 W215 G216 R217 H46 T91 L92 A93 H94 D192 S193 C194 Q195 S198 S217 W218 G219 R220 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 12684001 1245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1w13 U 2.0 BS01 SM1 U 1 H57 L97B H99 D189 S190 C191 Q192 S195 S214 W215 G216 G219 C220 G226 H46 L92 H94 D192 S193 C194 Q195 S198 S217 W218 G219 G221 C222 G229 3.4.21.73 0004252,0006508 Ki=2nM remove_due_to_license_issue Ki=16nM P00749 12684001 1245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1w14 U 2.2 BS01 SH1 U 1 H57 L97B D189 S190 C191 Q192 S195 S214 W215 G216 R217 G219 H46 L92 D192 S193 C194 Q195 S198 S217 W218 G219 R220 G221 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 12684001 1300 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 1w1d A 1.5 BS01 4IP A 1 K465 K467 R472 R474 Y486 K495 R521 K59 K61 R66 R68 Y80 K89 R115 2.7.11.1 Ki=0.3uM remove_due_to_license_issue O15530 15457207 1552 PLGSNIEQYIHDLDSNSFELDLQFSEDEKRLLLEKQAGGNPWHQFVENNLILKMGPVDKRKGLFARRRQLLLTEGPHLYYVDPVNKVLKGEIPWSQELRPEAKNFKTFFVHTPNRTYYLMDPSGNAHKWCRKIQEVWRQRYQS 1w1g A 1.45 BS01 4PT A 1 K465 K467 R472 R474 Y486 K495 R521 S549 K59 K61 R66 R68 Y80 K89 R115 S143 2.7.11.1 Ki=0.021uM remove_due_to_license_issue O15530 15457207 1550 PLGSNIEQYIHDLDSNSFELDLQFSEDEKRLLLEKQAGGNPWHQFVENNLILKMGPVDKRKGLFARRRQLLLTEGPHLYYVDPVNKVLKGEIPWSQELRPEAKNFKTFFVHTPNRTYYLMDPSGNAHKWCRKIQEVWRQRYQS 1w1p A 2.1 BS01 GIO A 1 Y10 F51 G96 W97 D142 E144 Y214 W403 Y9 F50 G95 W96 D141 E143 Y213 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=5mM remove_due_to_license_issue Q54276 15509170 1518 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w1t A 1.9 BS01 CHQ A 1 Y10 F51 G96 E144 M212 Y214 D215 W403 Y8 F49 G94 E142 M210 Y212 D213 W401 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=1.1mM remove_due_to_license_issue Q54276 15509170 1513 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w1t A 1.9 BS02 CHQ A 2 W97 W220 W95 W218 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=1.1mM remove_due_to_license_issue Q54276 15509170 1514 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w1v A 1.85 BS01 ALJ A 1 Y10 F51 W97 E144 Y214 W403 Y8 F49 W95 E142 Y212 W401 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=6.3mM remove_due_to_license_issue Q54276 15509170 1520 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w1y A 1.85 BS01 TYP A 1 Y10 F51 G96 Y98 E144 M212 Y214 W403 Y8 F49 G94 Y96 E142 M210 Y212 W401 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=2.4mM remove_due_to_license_issue Q54276 15509170 1507 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w1y A 1.85 BS02 TYP A 2 F12 F51 G96 W97 Y98 D336 W403 F10 F49 G94 W95 Y96 D334 W401 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=2.4mM remove_due_to_license_issue Q54276 15509170 1508 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w1y A 1.85 BS03 TYP A 3 W97 W220 W95 W218 D140 D142 E144 Y214 D138 D140 E142 Y212 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0016798,0030246 ic50=2.4mM remove_due_to_license_issue Q54276 15509170 1509 TRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPASRAKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTITDGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKVTNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPSTDYWLVGCEECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRV 1w22 A 2.5 BS04 NHB A 1 D101 H142 H143 G151 F152 D178 H180 F208 Y306 D79 H120 H121 G129 F130 D156 H158 F186 Y284 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=175.5nM remove_due_to_license_issue Q9BY41 15477595 1378 SLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLK 1w22 A 2.5 BS05 NHB B 1 F152 P273 Y306 F130 P251 Y284 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=175.5nM remove_due_to_license_issue Q9BY41 15477595 1378 SLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLK 1w25 A 2.7 BS02 C2E A 1 N335 D344 G369 E370 N334 D343 G368 E369 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 Ki=0.5uM (15569936) remove_due_to_license_issue B8GZM2 15569936 501 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAH 1w25 A 2.7 BS03 C2E A 2 R178 R359 D362 D383 I387 R390 R177 R358 D361 D382 I386 R389 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 Ki=0.5uM (15569936) remove_due_to_license_issue B8GZM2 15569936 503 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAH 1w25 A 2.7 BS04 C2E A 3 R148 V175 R178 S356 R359 A360 R390 R147 V174 R177 S355 R358 A359 R389 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 Ki=0.5uM (15569936) remove_due_to_license_issue B8GZM2 15569936 505 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAH 1w2b 1 3.5 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 K9 R10 L11 K13 Q17 P22 W24 V25 L27 K28 T29 D30 R35 N36 H37 R40 H41 W42 R43 N45 T47 G1 K2 K3 K5 A6 K8 K9 R10 L11 K13 Q17 P22 W24 V25 L27 K28 T29 D30 R32 N33 H34 R37 H38 W39 R40 N42 T44 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 15334087 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDERNHKRRHWRRNDTDE 1w2b 2 3.5 BS01 rna 0 0 M1 Q2 P4 N8 T9 Y10 N15 E16 H17 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 D49 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 D66 K68 A77 L79 R80 G82 R84 G86 Q91 M1 Q2 P4 N8 T9 Y10 N15 E16 H17 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 D49 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 D66 K68 A77 L79 R80 G82 R84 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 15334087 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 1w2b 5 3.5 BS01 rna 0 0 G43 R45 G19 R21 5.2.1.8 0006457,0015031 remove_due_to_license_issue P0A850 15334087 10 ~ 2914 ETAVKSELVNVAKKVRIDGFRKGKVPMNIVAQRYG 1w2b A 3.5 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 R17 A18 S20 H21 Y23 K24 A25 D26 K31 H47 R51 S52 S110 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 T184 K185 W186 P187 N188 V189 R190 G191 V192 A193 M194 N195 V197 D198 H199 F201 G203 G204 G205 R206 Q207 H208 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 R17 A18 S20 H21 Y23 K24 A25 D26 K31 H47 R51 S52 S110 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 T184 K185 W186 P187 N188 V189 R190 G191 V192 A193 M194 N195 V197 D198 H199 F201 G203 G204 G205 R206 Q207 H208 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 15334087 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVDAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVGGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 1w2b B 3.5 BS01 rna 0 0 P1 Q2 P3 S4 R5 P6 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 T20 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Q94 R95 P96 L97 E99 W101 R111 T112 L113 D114 P116 E117 H119 R141 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 V220 Q221 K222 K224 G225 K226 H227 R229 Q230 W232 R233 R234 R235 I236 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 K267 D281 G282 V285 N286 G288 S300 G303 K306 R307 R312 R316 N318 S334 N335 Q336 G337 P1 Q2 P3 S4 R5 P6 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 T20 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Q94 R95 P96 L97 E99 W101 R111 T112 L113 D114 P116 E117 H119 R141 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 V220 Q221 K222 K224 G225 K226 H227 R229 Q230 W232 R233 R234 R235 I236 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 K267 D281 G282 V285 N286 G288 S300 G303 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 15334087 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 1w2b C 3.5 BS01 rna 0 0 R27 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 L54 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 L73 D74 R76 A77 R78 V80 Q82 A83 V84 K85 R87 H90 P92 K93 K96 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 K173 I174 K175 A176 G177 G179 A181 R182 R184 Y186 R187 R188 P189 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 R27 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 L54 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 L73 D74 R76 A77 R78 V80 Q82 A83 V84 K85 R87 H90 P92 K93 K96 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 K173 I174 K175 A176 G177 G179 A181 R182 R184 Y186 R187 R188 P189 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 15334087 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKLDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 1w2b D 3.5 BS01 rna 0 0 K20 V22 H24 T52 A54 K55 R56 E60 Q97 D100 S105 G107 D129 Y139 R156 K11 V13 H15 T38 A40 K41 R42 E46 Q83 D86 S91 G93 D95 Y105 R122 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 15334087 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 1w2b D 3.5 BS02 rna 9 0 E12 M13 R14 R17 Q47 P49 V50 K53 K72 V73 T74 R76 P137 G138 R140 V141 R144 D145 R149 P152 K154 H155 E3 M4 R5 R8 Q33 P35 V36 K39 K58 V59 T60 R62 P103 G104 R106 V107 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 15334087 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 1w2b E 3.5 BS01 rna 0 0 N55 A56 S60 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 I138 E139 Q143 A146 Q150 R153 K157 D158 V161 F162 N55 A56 S60 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 I138 E139 Q143 A146 Q150 R153 K157 D158 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 15334087 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 1w2b F 3.5 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 15334087 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGAAATVLEEIADKVEELR 1w2b H 3.5 BS01 rna 0 0 K1 G3 M5 R7 K11 P12 A13 Y14 T15 R16 E18 Y19 D32 R57 A60 R70 R84 R86 K87 F88 F90 R94 E95 N96 M111 R112 A113 P114 F115 G116 R147 M151 K152 T154 T156 K1 G3 M5 R7 K11 P12 A13 Y14 T15 R16 E18 Y19 D32 R57 A60 R70 R84 R86 K87 F88 F90 R94 E95 N96 M100 R101 A102 P103 F104 G105 R136 M140 K141 T143 T145 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 15334087 10 ~ 2914 KPGAMYRNSSKPAYTRREYISGIPGKKIAQFDMGNNGAGPTYPAQVELVVEKPVQIRHNALEAARVAANRYVQNSGAAANYKFRIRKFPFHVIRENKDGMRAPFGKPVGTAARVHGANHIFIAWVNPDPNVEEAWRRAKMKVTPTINIDSSPAGNA 1w2b I 3.5 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 G48 R49 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R74 K80 T82 R84 M86 P88 H89 K90 K91 R95 R102 V103 K128 G140 I15 G17 R18 S21 L28 T44 G45 R46 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R71 K77 T79 R81 M83 P85 H86 K87 K88 R92 R99 V100 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 15334087 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 1w2b J 3.5 BS01 rna 0 0 M1 A3 T9 G11 E13 K14 S16 L17 K30 I32 S33 V34 H35 G36 Y37 S38 T40 K41 N42 R43 H44 T54 S56 R66 K78 R81 R87 M1 A3 T9 G11 E13 K14 S16 L17 K30 I32 S33 V34 H35 G36 Y37 S38 T40 K41 N42 R43 H44 T54 S56 R66 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 15334087 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 1w2b K 3.5 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 E71 K107 L109 G110 G112 Q113 R115 S126 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 E71 K102 L104 G105 G107 Q108 R110 S121 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 15334087 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 1w2b L 3.5 BS01 rna 0 0 A1 S3 Y5 R9 K13 W25 R32 P35 A36 R39 R42 R45 L46 R48 R50 S51 L52 K55 A56 Q58 I61 R68 G70 S71 R73 R74 T75 R76 F77 K79 G80 R81 R82 S83 K84 R85 M86 N89 R90 T92 R93 K94 K95 N96 I97 R99 I100 R104 R107 F109 P110 N111 N116 G124 K127 D135 H138 A140 Q146 W149 T153 R154 R156 L157 F160 R161 L163 S165 R168 R171 G172 R174 Q176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 A194 A1 S3 Y5 R9 K13 W25 R32 P35 A36 R39 R42 R45 L46 R48 R50 S51 L52 K55 A56 Q58 I61 R68 G70 S71 R73 R74 T75 R76 F77 K79 G80 R81 R82 S83 K84 R85 M86 N89 R90 T92 R93 K94 K95 N96 I97 R99 I100 R104 R107 F109 P110 N111 N116 G124 K127 D135 H138 A140 Q146 W149 T153 R154 R156 L157 F160 R161 L163 S165 R168 R171 G172 R174 Q176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 A194 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 15334087 10 ~ 2914 ARSAYSYIREAWKRPKEGQIAELMWHRMQEWRNEPAVVRIERPTRLDRARSLGYKAKQGIIVVRVAIRKGSSRRTRFNKGRRSKRMMVNRITRKKNIQRIAEERANRKFPNLRVLNSYSVGEDGRHKWHEVILIDPDHPAIKSDDQLSWISRTRHRLRTFRGLTSAGRRCRGLRGQGKGSEKVRPSLRVNGAKA 1w2b M 3.5 BS01 rna 0 0 P4 R5 Y6 K7 P9 R13 A16 T18 H21 R25 L26 K28 S29 V101 I104 L106 P109 F116 N132 V135 P4 R5 Y6 K7 P9 R13 A16 T18 H21 R25 L26 K28 S29 V101 I104 L106 P109 F116 N132 V135 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 15334087 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 1w2b M 3.5 BS02 rna 9 0 A1 P4 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 L158 Y159 S160 D162 A1 P4 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 L158 Y159 S160 D162 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 15334087 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 1w2b N 3.5 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 S16 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 G68 S82 G83 S109 H110 V111 R112 I114 R115 S1 K2 T3 N4 A12 K15 S16 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 G68 S82 G83 S109 H110 V111 R112 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 15334087 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 1w2b O 3.5 BS01 rna 0 0 T1 D2 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 N57 S58 R59 R61 R63 R65 Q66 K68 R69 K71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 T1 D2 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 N57 S58 R59 R61 R63 R65 Q66 K68 R69 K71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 15334087 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAKGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 1w2b P 3.5 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 L14 K15 R21 G22 T23 K38 H40 K42 S46 P48 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G78 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 L14 K15 R21 G22 T23 K38 H40 K42 S46 P48 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G78 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 15334087 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 1w2b P 3.5 BS02 rna 9 0 R19 P25 Q27 R19 P25 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 15334087 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 1w2b Q 3.5 BS01 rna 0 0 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 H27 K29 K60 H62 S64 G65 V66 G67 H68 K69 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 A116 H117 Q122 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 H27 K29 K60 H62 S64 G65 V66 G67 H68 K69 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 A116 H117 Q122 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 15334087 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 1w2b R 3.5 BS01 rna 0 0 S1 H9 T11 K13 Q21 K23 R31 S33 K34 N53 T54 Q55 N56 M58 K62 S1 H9 T11 K13 Q21 K23 R31 S33 K34 N53 T54 Q55 N56 M58 K62 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 15334087 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRIGVF 1w2b S 3.5 BS01 rna 0 0 S1 K2 Q3 P4 D5 Q7 R8 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 E80 K81 T82 R89 P90 S94 R97 D105 K107 R111 S1 K2 Q3 P4 D5 Q7 R8 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 E80 K81 T82 R89 P90 S94 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 15334087 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 1w2b T 3.5 BS01 rna 0 0 T17 S34 K35 L42 R44 E50 W51 R56 T14 S31 K32 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 15334087 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 1w2b U 3.5 BS01 rna 0 0 T1 H4 R9 Q34 P43 G44 K47 R50 K51 A54 R55 K57 T58 T1 H4 R9 Q34 P43 G44 K47 R50 K51 A54 R55 K57 T58 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 15334087 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 1w2b V 3.5 BS01 rna 0 0 R8 G9 E10 V11 N12 T15 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 R8 G9 E10 V11 N12 T15 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 15334087 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 1w2b V 3.5 BS02 rna 9 0 R8 H14 D50 K129 H130 P131 K133 E134 R8 H14 D50 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 15334087 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 1w2b W 3.5 BS01 rna 0 0 R15 R18 A19 E20 P21 N22 H23 D27 K28 M30 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 S68 R9 R12 A13 E14 P15 N16 H17 D21 K22 M24 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 15334087 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 1w2b X 3.5 BS01 rna 0 0 R115 Q119 R120 R122 K125 Q127 F128 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 K152 R154 R155 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 P231 Y233 R21 Q25 R26 R28 K31 Q33 F34 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 K58 R60 R61 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 P137 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 15334087 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 1w2b Y 3.5 BS01 rna 0 0 R10 R13 G15 P16 R17 Y18 G19 L20 K21 I22 R23 K34 C42 K46 R49 G51 T52 C60 R1 R4 G6 P7 R8 Y9 G10 L11 K12 I13 R14 K25 C33 K37 R40 G42 T43 C51 ? 0003735,0005840,0006412 remove_due_to_license_issue P60619 15334087 10 ~ 2914 RTGRFGPRYGLKIRVRVADVEIKHKKKHKCPVCGFKKLKRAGTGIWMCGHCGYKIAGGCYQPETVAGKAVMKA 1w2b Z 3.5 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 T29 K30 K31 K32 S35 K41 S42 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 T29 K30 K31 K32 S35 K41 S42 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 15334087 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 1w2g A 2.1 BS01 THM A 1 P37 F70 R74 R95 S99 N100 Y103 Y165 P37 F70 R74 R95 S99 N100 Y103 Y153 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 Ki=27uM remove_due_to_license_issue Ki=27000nM P9WKE1 15628853 1210 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAELAGERRDNYERDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLA 1w2h A 2.0 BS01 ATM A 1 D9 P37 Y39 F70 R74 R95 N100 Y103 D9 P37 Y39 F70 R74 R95 N100 Y103 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 Ki~10uM remove_due_to_license_issue P9WKE1 15628853 1209 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAELAGERDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLA 1w2h A 2.0 BS02 ATM A 2 G10 G12 K13 R14 T15 R149 G10 G12 K13 R14 T15 R149 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 Ki~10uM remove_due_to_license_issue P9WKE1 15628853 1210 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAELAGERDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLA 1w2k H 3.0 BS01 380 H 1 H57 T99 D189 S190 K192 S195 W215 G216 G219 H41 T87 D183 S184 K186 S189 W209 G210 G212 3.4.21.21 0004252,0006508 remove_due_to_license_issue Ki=350nM P08709 15664864 1258 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1w2x A 2.8 BS01 RCP A 1 T1757 A1761 K1764 M1765 T276 A280 K283 M284 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 15341732 3000 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 1w2x B 2.8 BS01 RCP B 1 T1757 I1762 K1764 M1765 T276 I281 K283 M284 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 15341732 3000 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 1w2x B 2.8 BS02 RCP C 1 R1954 G1958 L2025 E2026 G2029 R473 G477 L544 E545 G548 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 15341732 3000 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 1w31 A 1.9 BS01 SHO A 1 S179 F219 K263 Y287 V289 S290 Y329 S179 F219 K263 Y287 V289 S290 Y329 K210 K263 K210 K263 4.2.1.24 0004655,0005634,0005737,0005829,0006782,0006783,0008270,0016829,0033014,0046872 Ki=0.25mM remove_due_to_license_issue P05373 16131755 363 MHTAEFLETEPTEISSVLAGGYNHPLLRQWQSERQLTKNMLIFPLFISDNPDDFTEIDSLPNINRIGVNRLKDYLKPLVAKGLRSVILFGVPLIPGTKDPVGTAADDPAGPVIQGIKFIREYFPELYIICDVCLCEYTSHGHCGVLYDDGTINRERSVSRLAAVAVNYAKAGAHCVAPSDMIDGRIRDIKRGLINANLAHKTFVLSYAAKFSGNLYGPFRDAACSAPSNGDRKCYQLPPAGRGLARRALERDMSEGADGIIVKPSTFYLDIMRDASEICKDLPICAYHVSGEYAMLHAAAEKGVVDLKTIAFESHQGFLRAGARLIITYLAPEFLDWLDE 1w3j A 2.0 BS01 OXZ A 1 Q20 H121 E166 Y295 E351 W398 E405 W406 Q17 H118 E163 Y292 E348 W395 E402 W403 R77 H121 E166 V169 N293 Y295 E351 R74 H118 E163 V166 N290 Y292 E348 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=484nM remove_due_to_license_issue Q08638 15356002 1447 KKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLED 1w3k A 1.2 BS01 BGC A 1 H35 Y66 W262 K267 E269 H32 Y63 W259 K264 E266 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 15356002 1304 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1w3k A 1.2 BS02 OXZ A 1 Y66 H101 E139 Y202 E228 A234 T235 G236 W262 Y63 H98 E136 Y199 E225 A231 T232 G233 W259 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 15356002 1305 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1w3l A 1.04 BS01 BGC B 1 H35 W39 Y66 W262 K267 E269 H32 W36 Y63 W259 K264 E266 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 15356002 1 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1w3l A 1.04 BS02 BGC B 2 W39 K267 W36 K264 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 15356002 2 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1w3l A 1.04 BS03 OXZ A 1 Y66 H101 E139 Y202 E228 A234 T235 G236 W262 Y63 H98 E136 Y199 E225 A231 T232 G233 W259 3.2.1.4 0000272,0004553,0005975 remove_due_to_license_issue O85465 15356002 1309 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 1w4l A 2.16 BS01 GL8 A 1 Y70 W84 G117 G118 G119 Y121 E199 S200 W279 F288 F290 F330 F331 Y334 H440 Y67 W81 G114 G115 G116 Y118 E196 S197 W276 F285 F287 F327 F328 Y331 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 ic50=4nM remove_due_to_license_issue IC50=4nM P04058 15563167 1540 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1w4o A 1.6 BS01 UA3 A 1 Q11 H12 V43 N44 T45 H119 F120 Q11 H12 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=3uM remove_due_to_license_issue Ki=6000nM P61823 15670155 1125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1w4p A 1.69 BS01 UM3 A 1 H12 K41 N44 T45 H119 F120 H12 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=18uM remove_due_to_license_issue P61823 15670155 1125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1w4q A 1.68 BS01 UMF A 1 H12 K41 N44 T45 H119 F120 H12 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=5.5uM remove_due_to_license_issue P61823 15670155 1125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1w51 A 2.55 BS01 L01 A 1 G11 G13 D32 G34 S35 P70 Y71 T72 Q73 F108 R128 Y198 D228 G230 T232 G13 G15 D34 G36 S37 P72 Y73 T74 Q75 F110 R130 Y190 D220 G222 T224 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=500nM P56817 15451669 1506 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVETSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 1w5v A 1.8 BS01 BE3 A 1 R8 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 R8 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=7.1nM remove_due_to_license_issue P03366 15560801 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5v B 1.8 BS01 BE3 A 1 R8 L23 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 R8 L23 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15560801 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5w A 1.8 BS01 BE4 A 1 R8 L23 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 R8 L23 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.6nM remove_due_to_license_issue P03366 15560801 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5w B 1.8 BS01 BE4 A 1 R8 D25 G27 A28 D29 D30 V32 I47 G48 G49 I50 V82 R8 D25 G27 A28 D29 D30 V32 I47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15560801 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5x A 1.9 BS01 BE5 A 1 R8 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 I84 R8 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4nM remove_due_to_license_issue P03366 15560801 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5x B 1.9 BS01 BE5 A 1 R8 D25 G27 A28 D29 D30 V32 G48 G49 I50 P81 V82 I84 R8 D25 G27 A28 D29 D30 V32 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15560801 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5y A 1.9 BS01 BE6 A 1 R8 D25 G27 A28 D29 D30 G48 G49 I50 V82 I84 R8 D25 G27 A28 D29 D30 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.3nM remove_due_to_license_issue P03366 15560801 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w5y B 1.9 BS01 BE6 A 1 R8 D25 G27 A28 D29 D30 G48 G49 I50 V82 R8 D25 G27 A28 D29 D30 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15560801 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1w6h A 2.24 BS01 TIT A 1 D34 N76 Y77 V78 S79 F111 T114 Y192 D214 G216 T217 S218 D34 N76 Y77 V78 S79 F111 T114 Y192 D214 G216 T217 S218 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue Ki=2.2nM P46925 1330 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 1w6j A 2.2 BS01 R71 A 1 Y98 W192 W230 H232 C233 V236 W387 F444 D455 T502 I524 W581 F696 N697 Y93 W187 W225 H227 C228 V231 W382 F439 D450 T497 I519 W576 F691 N692 G107 L156 P190 H232 S339 W387 F444 D455 T457 A458 Y503 A536 W581 Y587 F696 C700 Y704 G102 L151 P185 H227 S334 W382 F439 D450 T452 A453 Y498 A531 W576 Y582 F691 C695 Y699 5.4.99.7 0000250,0005515,0005783,0005789,0005811,0006694,0006695,0008610,0016020,0016104,0016853,0016866,0031647 remove_due_to_license_issue IC50=6.5nM P48449 15525992 1733 CLRRRGGPYKTEPATDLGRWRLNCERGRQTWTYLQDERAGREQTGLEAYALGLDTKNYFKDLPKAHTAFEGALNGMTFYVGLQAEDGHWTGDYGGPLFLLPGLLITCHVARIPLPAGYREEIVRYLRSVQLPDGGWGLHIEDKSTVFGTALNYVSLRILGVGPDDPDLVRARNILHKKGGAVAIPSWGKFWLAVLNVYSWEGLNTLFPEMWLFPDWAPAHPSTLWCHCRQVYLPMSYCYAVRLSAAEDPLVQSLRQELYVEDFASIDWLAQRNNVAPDELYTPHSWLLRVVYALLNLYEHHHSAHLRQRAVQKLYEHIVADDRFTKSISIGPISKTINMLVRWYVDGPASTAFQEHVSRIPDYLWMGLDGMKMQGTNGSQIWDTAFAIQALLEAGGHHRPEFSSCLQKAHEFLRLSQVPDNPPDYQKYYRQMRKGGFSFSTLDCGWIVSDCTAEALKAVLLLQEKCPHVTEHIPRERLCDAVAVLLNMRNPDGGFATYETKRGGHLLELLNPSEVFGDIMIDYTYVECTSAVMQALKYFHKRFPEHRAAEIRETLTQGLEFCRRQQRADGSWEGSWGVCFTYGTWFGLEAFACMGQTYRDGTACAEVSRACDFLLSRQMADGGWGEDFESCEERRYLQSAQSQIHNTCWAMMGLMAVRHPDIEAQERGVRCLLEKQLPNGDWPQENIAGVFNKSCAISYTSYRNIFPIWALGRFSQLYPERALAGHP 1w6r A 2.05 BS01 GNT A 1 W84 G117 G118 G119 Y121 E199 S200 F288 F290 F330 F331 H440 W81 G114 G115 G116 Y118 E196 S197 F285 F287 F327 F328 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 ic50=702nM remove_due_to_license_issue IC50=1069nM, Ki=1.9e+2nM P04058 15563167 1536 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1w6y A 2.1 BS01 EQU A 1 Y16 D40 F86 M90 D103 W120 V127 Y15 D39 F84 M88 D101 W118 V125 Y16 D40 D100 D103 Y15 D39 D98 D101 5.3.3.1 0004769,0008202,0016853 Kd=4.4uM remove_due_to_license_issue P07445 15819891 201 NLPTAQEVQGLMARYIELVDVGDIEAIVQMYADDATVEDPFGQPPIHGREQIAAFYRQGLGGKVRACLTGPVRASHNGCGAMPFRVEMVANGQPCALDVIDVMRFDEHGRIQTMQAYWSEVNLSV 1w76 A 2.3 BS01 GNT A 1 W84 G118 Y121 E199 S200 F290 F331 H440 W81 G115 Y118 E196 S197 F281 F322 H431 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F281 F283 E318 H431 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 ic50=702nM remove_due_to_license_issue IC50=1069nM, Ki=1.9e+2nM P04058 15563167 1538 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1w7a A 2.27 BS01 dna E 0 P12 M13 M33 G34 D35 F36 R58 S61 Q95 P99 P105 V106 R108 P11 M12 M32 G33 D34 F35 R57 S60 Q94 P98 P104 V105 R107 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 15297450 1 ~ 18 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGASTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1w7a A 2.27 BS02 dna F 0 F36 E38 I53 S54 T56 M68 G70 P72 Y79 N468 L495 K496 R500 F35 E37 I52 S53 T55 M67 G69 P71 Y78 N467 L494 K495 R499 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 15297450 14 ~ 30 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGASTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1w7a B 2.27 BS01 dna E 0 N468 L495 K496 N432 L459 K460 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 15297450 1 ~ 18 MQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGAADDSGRSTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1w7g H 1.65 BS03 MIU H 1 H57 Y60A W60D K60F A190 C191 E192 W215 G216 G219 H43 Y47 W50 K52 A194 C195 E196 W221 G222 G224 3.4.21.5 0004252,0005509,0006508,0007596 Ki~13uM remove_due_to_license_issue Ki=1900nM P00734 16294249 300 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1w7h A 2.214 BS01 3IP A 1 A51 K53 L104 T106 L108 M109 D354 A48 K50 L101 T103 L105 M106 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50>1mM remove_due_to_license_issue IC50=1300000nM Q16539 15658854 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1w7x H 1.8 BS02 413 H 1 H57 K60A T99 S170H P170I D189 S190 K192 S195 S214 W215 G216 Q217 G219 C220 H41 K45 T87 S164 P165 D182 S183 K185 S188 S207 W208 G209 Q210 G211 C212 3.4.21.21 0004252,0006508 Ki=0.004uM remove_due_to_license_issue Ki=4nM P08709 16213138 1261 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1w82 A 2.2 BS01 L10 A 1 A51 K53 R67 E71 L74 L75 I84 T106 D168 D354 A48 K50 R64 E68 L71 L72 I81 T103 D165 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=196nM remove_due_to_license_issue Q16539 15658855 1356 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1w83 A 2.5 BS01 L11 A 1 V38 A51 K53 E71 L75 T106 M109 I141 H148 D168 F169 L353 D354 V35 A48 K50 E68 L72 T103 M106 I138 H145 D165 F166 L350 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.065uM remove_due_to_license_issue Q16539 15658855 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1w84 A 2.2 BS01 L12 A 1 A51 K53 L75 I84 L104 T106 M109 D354 A48 K50 L72 I81 L101 T103 M106 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=35uM remove_due_to_license_issue IC50=35000nM Q16539 15658855 1356 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1w8l A 1.8 BS01 1P3 A 1 F60 A101 N102 F113 H126 F60 A101 N102 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Ki=320mM remove_due_to_license_issue P62937 14993672 1166 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 1w8m A 1.65 BS01 E1P A 1 Q63 A101 N102 F113 H126 Q63 A101 N102 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Ki=25mM remove_due_to_license_issue P62937 14993672 1166 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 1w96 A 1.8 BS01 S1A A 1 K73 R76 S77 E392 M393 N398 W487 F510 K60 R63 S64 E379 M380 N385 W474 F497 E365 E379 N381 E387 R458 E352 E366 N368 E374 R445 6.3.4.14,6.4.1.2 0003989,0005524,0046872 Kd=3.9nM remove_due_to_license_issue Q00955 15610732 1567 MEYEITNYSERHTELPGHFIGLNTVDKLEESPLRDFVKSHGGHTVISKILIANNGIAAVKEIRSVRKWAYETFGDDRTVQFVAMATPEDLEANAEYIRMADQYIEVPGGTNNNNYANVDLIVDIAERADVDAVWAGWGHASENPLLPEKLSQSKRKVIFIGPPGNAMRSLGDKISSTIVAQSAKVPCIPWSGTGVDTVHVDEKTGLVSVDDDIYQKGCCTSPEDGLQKAKRIGFPVMIKASEGGGGKGIRQVEREEDFIALYHQAANEIPGSPIFIMKLAGRARHLEVQLLADQYGTNISLFGRDCSVQRRHQKIIEEAPVTIAKAETFHEMEKAAVRLGKLVGYVSAGTVEYLYSHDDGKFYFLELNPRLQVEHPTTEMVSGVNLPAAQLQIAMGIPMHRISDIRTLYGMNPHSASEIDFEFKTQDATKKQRRPIPKGHCTACRITSEDPNDGFKPSGGTLHELNFRSSSNVWGYFSVGNNGNIHSFSDSQFGHIFAFGENRQASRKHMVVALKELSIRGTVEYLIKLLETEDFEDNTITTGWLDDLI 1wax A 2.2 BS02 LO1 A 1 Y46 D48 D181 F182 C215 S216 A217 G220 R221 Q262 Y45 D47 D180 F181 C214 S215 A216 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=86uM remove_due_to_license_issue P18031 15658854 1300 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 1way B 2.02 BS03 L02 B 1 A190 E192 V213 W215 G219 C220 G226 F227 A192 E194 V217 W219 G222 C223 G230 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=400uM remove_due_to_license_issue P00734 15658854 1248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 1wb9 A 2.1 BS01 dna E 0 T11 P12 M13 M33 G34 D35 F36 R58 S61 Q95 P105 R108 V470 T10 P11 M12 M32 G33 D34 F35 R57 S60 Q94 P104 R107 V469 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 1 ~ 18 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYTLFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wb9 A 2.1 BS02 dna F 0 F36 I53 S54 G70 P72 Y79 N468 L495 K496 R500 F35 I52 S53 G69 P71 Y78 N467 L494 K495 R499 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 14 ~ 30 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYTLFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wb9 B 2.1 BS01 dna E 0 N468 L495 K496 R500 N432 L459 K460 R464 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 1 ~ 18 MQQYLRLKAQHPEILLFYRMGDFYTLFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wb9 B 2.1 BS02 dna F 0 T462 K464 S478 T426 K428 S442 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 14 ~ 30 MQQYLRLKAQHPEILLFYRMGDFYTLFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbb A 2.5 BS01 dna E 0 T11 P12 M13 M33 G34 D35 F36 R58 S61 P99 P105 V106 R108 V470 T10 P11 M12 M32 G33 D34 F35 R57 S60 P98 P104 V105 R107 V469 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 1 ~ 18 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYALFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbb A 2.5 BS02 dna F 0 F36 I53 S54 T56 M68 G70 P72 Y79 L495 K496 R500 F35 I52 S53 T55 M67 G69 P71 Y78 L494 K495 R499 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 14 ~ 30 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYALFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbb B 2.5 BS01 dna E 0 N468 A469 L495 K496 R500 N432 A433 L459 K460 R464 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 1 ~ 18 MQQYLRLKAQHPEILLFYRMGDFYALFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbb B 2.5 BS02 dna F 0 K464 S478 K428 S442 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 14 ~ 30 MQQYLRLKAQHPEILLFYRMGDFYALFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbd A 2.4 BS01 dna E 0 T11 P12 M13 M33 G34 D35 F36 R58 S61 Q95 P99 P105 V106 R108 V470 T10 P11 M12 M32 G33 D34 F35 R57 S60 Q94 P98 P104 V105 R107 V469 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 1 ~ 18 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYQLFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbd A 2.4 BS02 dna F 0 F36 Q38 I53 S54 T56 G70 P72 Y79 N468 L495 K496 R500 F35 Q37 I52 S53 T55 G69 P71 Y78 N467 L494 K495 R499 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 14 ~ 30 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYQLFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbd B 2.4 BS01 dna E 0 N468 L495 K496 R500 N432 L459 K460 R464 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 1 ~ 18 MQQYLRLKAQHPEILLFYRMGDFYQLFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbd B 2.4 BS02 dna F 0 K464 S478 K428 S442 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 16407973 14 ~ 30 MQQYLRLKAQHPEILLFYRMGDFYQLFYDDAKRASQLLDISLTPMAGIPYHAVENYLAKLVNQGESVAICERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 1wbg B 2.2 BS02 L03 B 1 A190 E192 V213 W215 G216 G219 C220 G226 F227 A192 E194 V217 W219 G220 G222 C223 G230 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=1mM remove_due_to_license_issue P00734 15658854 1248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCRDDGKYGFYTHVFRLKKWIQKVIDQFGE 1wbn A 2.4 BS01 L09 A 1 A51 K53 E71 L74 M78 I84 T106 M109 H148 I166 L167 D168 D354 A48 K50 E68 L71 M75 I81 T103 M106 H145 I163 L164 D165 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.35uM remove_due_to_license_issue IC50=350nM Q16539 15658855 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1wbo A 2.16 BS01 2CH A 1 V38 A51 K53 L104 T106 D168 V35 A48 K50 L101 T103 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50>1mM remove_due_to_license_issue Q16539 15658854 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1wbs A 1.8 BS01 LI2 A 1 A51 K53 E71 L75 I84 L104 T106 M109 I141 H148 L167 D168 F169 D354 A48 K50 E68 L72 I81 L101 T103 M106 I138 H145 L164 D165 F166 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.63uM remove_due_to_license_issue IC50=630nM Q16539 15658855 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1wbt A 2.0 BS01 WBT A 1 A51 K53 E71 L75 I84 T106 L108 M109 I141 H148 D168 F169 D354 A48 K50 E68 L72 I81 T103 L105 M106 I138 H145 D165 F166 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.34uM remove_due_to_license_issue IC50=340nM Q16539 15658855 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1wbv A 2.0 BS01 LI3 A 1 A51 K53 E71 L75 I84 L104 T106 H148 L167 D168 D354 A48 K50 E68 L72 I81 L101 T103 H145 L164 D165 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=162uM remove_due_to_license_issue IC50=162000nM Q16539 15658855 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1wbw A 2.41 BS01 LI4 A 1 A51 I84 L104 T106 H107 L108 M109 D354 A48 I81 L101 T103 H104 L105 M106 D351 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=44uM remove_due_to_license_issue IC50=44000nM Q16539 15658855 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1wc1 A 1.93 BS01 TAT A 1 D1017 G1020 F1021 T1022 V1059 G1060 D1061 D14 G17 F18 T19 V56 G57 D58 2.7.13.3 0009190,0035556 Ki~0.1mM remove_due_to_license_issue O32393 15619637 1500 LRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGRNEVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wc1 B 1.93 BS01 TAT B 1 G1020 F1021 T1022 V1059 G1060 D1061 G16 F17 T18 V55 G56 D57 2.7.13.3 0009190,0035556 Ki~0.1mM remove_due_to_license_issue O32393 15619637 1500 RPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGRNEVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wc1 B 1.93 BS04 TAT C 1 M1064 V1145 N1146 R1150 M60 V141 N142 R146 2.7.13.3 0009190,0035556 Ki~0.1mM remove_due_to_license_issue O32393 15619637 1500 RPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGRNEVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wc6 A 2.51 BS01 TAT A 1 D1017 I1018 V1019 G1020 F1021 T1022 V1059 G1060 D1061 R1117 D14 I15 V16 G17 F18 T19 V56 G57 D58 R111 2.7.13.3 0009190,0035556 remove_due_to_license_issue O32393 15619637 2200 LRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wc6 A 2.51 BS03 TAT C 1 F1015 K1057 M1064 T1139 A1140 V1145 N1146 A1149 F12 K54 M61 T133 A134 V139 N140 A143 2.7.13.3 0009190,0035556 remove_due_to_license_issue O32393 15619637 2200 LRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wc6 C 2.51 BS01 TAT A 1 F1015 K1057 M1064 T1139 A1140 V1145 N1146 A1149 M1199 F12 K54 M61 T133 A134 V139 N140 A143 M193 2.7.13.3 0009190,0035556 remove_due_to_license_issue O32393 15619637 2200 LRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wc6 C 2.51 BS02 TAT C 1 D1017 I1018 G1020 F1021 T1022 V1059 G1060 D1061 R1117 D14 I15 G17 F18 T19 V56 G57 D58 R111 2.7.13.3 0009190,0035556 remove_due_to_license_issue O32393 15619637 2200 LRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 1wcc A 2.2 BS01 CIG A 1 A31 K33 F80 E81 F82 L83 L134 A31 K33 F76 E77 F78 L79 L130 D127 K129 Q131 N132 D145 T165 D123 K125 Q127 N128 D141 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=350uM remove_due_to_license_issue IC50=350000nM P24941 15658854 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1wcq A 2.1 BS01 DAN A 1 R68 I69 D131 F203 D259 R276 R342 F370 R22 I23 D85 F157 D213 R230 R296 F324 D92 E260 F370 D46 E214 F324 3.2.1.18 0004308,0005576,0005737,0005975,0006689,0009313,0016020,0016798,0043231 Ki=0.55uM remove_due_to_license_issue Q02834 16206228 1651 GEPLYTEQDLAVNGREGFPNYRIPALTVTPDGDLLASYDGRPTGIDAPGPNSILQRRSTDGGRTWGEQQVVSAGQTTAPIKGFSDPSYLVDRETGTIFNFHVYSQRQGFAGSRPGTDPADPNVLHANVATSTDGGLTWSHRTITADITPDPGWRSRFAASGEGIQLRYGPHAGRLIQQYTIINAAGAFQAVSVYSDDHGRTWRAGEAVGVGMDENKTVELSDGRVLLNSRDSARSGYRKVAVSTDGGHSYGPVTIDRDLPDPTNNASIIRAFPDAPAGSARAKVLLFSNAASQTSRSQGTIRMSCDDGQTWPVSKVFQPGSMSFSTLTALPDGTYGLLYEPGTGIRYANFNLAWLGGICAPFTIPDVALEPGQQVTVPVAVTNQSGIAVPKPSLQLDASPDWQVQGSVEPLMPGRQAKGQVTITVPAGTTPGRYRVGATLRTSAGNASTTFTVTVGLLDQARMSIADVDSEETAREDGRASNVIDGNPSTFWHTEWSRADAPGYPHRISLDLGGTHTISGLQYTRRQNSANEQVADYEIYTSLNGTTWDGPVASGRFTTSLAPQRAVFPARDARYIRLVALSEQTGHKYAAVAELEVEGQR 1wdn A 1.94 BS01 GLN A 1 F13 F50 G68 T70 R75 K115 T118 H156 D157 F10 F47 G65 T67 R72 K112 T115 H153 D154 ? 0006865,0006868,0015276,0016020,0030288,0034220,0042597,0055052,0070406,1903803 Kd=0.5uM remove_due_to_license_issue P0AEQ3 9571045 227 KLVVATDTAFVPFEFKQGDLYVGFDVDLWAAIAKELKLDYELKPMDFSGIIPALQTKNVDLALAGITITDERKKAIDFSDGYYKSGLLVMVKANNNDVKSVKDLDGKVVAVKSGTGSVDYAKANIKTKDLRQFPNIDNAYMELGTNRADAVLHDTPNILYFIKTAGNGQFKAVGDSLEAQQYGIAFPKGSDELRDKVNGALKTLRENGTYNEIYKKWFGTEPK 1wdy A 1.8 BS01 25A A 1 E55 W60 Q68 K89 Y124 F126 E131 Y135 R155 E35 W40 Q48 K69 Y104 F106 E111 Y115 R135 3.1.26.- remove_due_to_license_issue IC50=20nM, EC50=0.210000nM Q05823 15385955 1001 AAVEDNHLLIKAVQNEDVDLVQQLLEGGANVNFQEEEGGWTPLHNAVQMSREDIVELLLRHGADPVLRKKNGATPFLLAAIAGSVKLLKLFLSKGADVNECDFYGFTAFMEAAVYGKVKALKFLYKRGANVNLRRKTKEDQERLRKGGATALMDAAEKGHVEVLKILLDEMGADVNACDNMGRNALIHALLSSDDSDVEAITHLLLDHGADVNVRGERGKTPLILAVEKKHLGLVQRLLEQEHIEINDTDSDGKTALLLAVELKLKKIAELLCKRGASTDCGDLV 1we2 A 2.3 BS02 DHK A 1 D34 I45 F49 G79 G80 G81 L119 R136 D33 I44 F48 G78 G79 G80 L118 R135 2.7.1.71 0000287,0004765,0005524,0005737,0005829,0008652,0009073,0009423,0016301,0019632,0019752,0046872 remove_due_to_license_issue P9WPY3 15583379 181 APKAVLVGLPGSGKSTIGRRLAKALGVGLLDTDVAIEQRTGRSIADIFATDGEQEFRRIEEDVVRAALADHDGVLSLGGGAVTSPGVRAALAGHTVVYLEISAAEGVRRTGGNTVRPLLAGPDRAEKYRALMAKRAPLYRRVATMRVDTNRRNPGAVVRHILSRL 1wet A 2.6 BS01 dna B 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S12 T14 T15 R24 V26 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 9278422 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLERNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 1wht A 2.0 BS01 BZS A 1 N51 G52 G53 C56 Y60 E145 S146 Y147 Y239 N56 G57 G58 C61 Y66 E153 S154 Y155 Y247 G53 S146 Y147 G58 S154 Y155 3.4.16.6 0004185,0006508 Ki=0.2mM remove_due_to_license_issue P08819 7727364 430 GHAADRIARLPGQPAVDFDMYSGYITVDEGAGRSLFYLLQEAPEDAQPAPLVLWLNGGPGCSSVAYGASEELGAFRVKPRGAGLVLNEYRWNKVANVLFLDSPAGVGFSYTNTSSDIYTSGDNRTAHDSYAFLAKWFERFPHYKYRDFYIAGESYAGHYVPELSQLVHRSKNPVINLKGFMVGNGLIDDYHDYVGTFEFWWNHGIVSDDTYRRLKEACLHDSFIHPSPACDAATDVATAEQGNIDMYSLYTPVCNI 1wht B 2.0 BS01 BZS A 1 H397 E398 H127 E128 D338 H397 D75 H127 3.4.16.6 0004185,0006508 remove_due_to_license_issue P08819 7727364 430 SYDPCTERYSTAYYNRRDVQMALHANVTGAMNYTWATCSDTINTHWHDAPRSMLPIYRELIAAGLRIWVFSGDTDAVVPLTATRYSIGALGLPTTTSWYPWYDDQEVGGWSQVYKGLTLVSVRGAGHEVPLHRPRQALVLFQYFLQGKPMPGQ 1wkm A 2.3 BS03 MET A 1 F50 N53 D82 D93 H161 E187 I205 F50 N53 D82 D93 H161 E187 I205 D82 D93 H153 H161 E187 E280 D82 D93 H153 H161 E187 E280 3.4.11.18 0004177,0004239,0005737,0006508,0008235,0046872,0070006 Ki=150mM remove_due_to_license_issue P56218 15628852 1298 MDTEKLMKAGEIAKKVREKAIKLARPGMLLLELAESIEKMIMELGGKPAFPVNLSINEIAAHYTPYKGDTTVLKEGDYLKIDVGVHIDGFIADTAVTVRVGMEEDELMEAAKEALNAAISVARAGVEIKELGKAIENEIRKRGFKPIVNLSGHKIERYKLHAGISIPNIYRPHDNYVLKEGDVFAIEPFATIGAGQVIEVPPTLIYMYVRDVPVRVAQARFLLAKIKREYGTLPFAYRWLQNDMPEGQLKLALKTLEKAGAIYGYPVLKEIRNGIVAQFEHTIIVEKDSVIVTTE 1wm1 A 2.1 BS01 PTB A 1 G45 G46 S113 W114 R136 F139 E204 E232 F236 H296 G42 G43 S110 W111 R133 F136 E201 E229 F233 H293 G46 S113 W114 D268 H296 G43 S110 W111 D265 H293 3.4.11.5 0004177,0005737,0006508,0008233 Ki=0.5uM remove_due_to_license_issue Ki=500nM O32449 12893291 401 LRGLYPPLAAYDSGWLDTGDGHRIYWELSGNPNGKPAVFIHGGPGGGISPHHRQLFDPERYKVLLFDQRGCGRSRPHASLDNNTTWHLVADIERLREMAGVEQWLVFGGSWGSTLALAYAQTHPERVSEMVLRGIFTLRKQRLHWYYQDGASRFFPEKWERVLSILSDDERKDVIAAYRQRLTSADPQVQLEAAKLWSVWEGETVTLLPSRESASFGEDDFALAFARIENHYFTHLGFLESDDQLLRNVPLIRHIPAVIVHGRYDMACQVQNAWDLAKAWPEAELHIVEGAGHSYDEPGILHQLMIATDRFAG 1wn6 A 1.8 BS02 BST A 1 E25 D26 S28 V29 N45 Y47 C54 A55 E56 R82 S86 P87 C88 E22 D23 S25 V26 N42 Y44 C51 A52 E53 R79 S83 P84 C85 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 1003 SQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLPSGYVWE 1wn6 B 1.8 BS02 BST B 1 E25 S28 V29 Y47 C54 E56 R82 S86 P87 E23 S26 V27 Y45 C52 E54 R80 S84 P85 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 1004 LSQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLPSGYVW 1wok A 3.0 BS01 CNQ A 1 E763 D766 H862 G863 Y896 F897 S904 Y907 E988 E102 D105 H201 G202 Y235 F236 S243 Y246 E327 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=33nM P09874 15733846 1 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 1wqv H 2.5 BS02 PSM H 1 H57 T98 T99 D189 S190 C191 K192 S195 V213 S214 W215 G216 G219 H41 T86 T87 D186 S187 C188 K189 S192 V210 S211 W212 G213 G215 3.4.21.21 0004252,0006508 ic50=130nM remove_due_to_license_issue P08709 15504346 1001 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1ws1 A 2.0 BS01 BB2 A 1 G44 V45 G46 Q51 G89 C90 L91 Y97 F125 R128 H132 E133 H136 G44 V45 G46 Q51 G89 C90 L91 Y97 F125 R128 H132 E133 H136 G46 Q51 C90 L91 H132 E133 H136 G46 Q51 C90 L91 H132 E133 H136 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=0.28nM remove_due_to_license_issue Q819U0 16049914 400 MAVLEIIKHPNEVLETPCERVINFDKKLVKLLKDMHETMLIADGVGLAAPQVGVSLQVAVVDVDDDTGKIELINPSILEKRGEQVGPEGCLSFPGLYGEVERADYIKVRAQNRRGKVFLLEAEGFLARAIQHEIDHLHGVLFTSKVTRYYE 1ws4 A 1.9 BS04 GYP A 1 G1 Y78 G121 Y122 W123 D125 G1 Y78 G121 Y122 W123 D125 ? 0019862,0030246 Kd=1mM remove_due_to_license_issue P18670 15733927 501 GKAFDDGAFTGIREINLSYNKETAIGDFQVVYDLNGSPYVGQNHVSFITGFTPVKISLDFPSEYIMEVSGYTGNVSGYVVVRSLTFKTNKKTYGPYGVTSGTPFNLPIENGLIVGFKGSIGYWLDYFSMYLSL 1wss H 2.6 BS02 3CB H 1 H57 D60 G97 T98 D189 S190 K192 S195 V213 S214 W215 G216 G219 C220 H41 D44 G85 T86 D186 S187 K189 S192 V210 S211 W212 G213 G215 C216 3.4.21.21 0004252,0006508 remove_due_to_license_issue P08709 16510984 2001 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1wsu A 2.3 BS01 rna E 0 R599 S605 R606 K607 L610 R624 R629 R89 S95 R96 K97 L100 R114 R119 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q46455 15665870 13 ~ 35 GSETQKKLLKDLEDKYRVSRWQPPSFKEVAGSFNLDPSELEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRRVGDKRVVVGN 1wsu B 2.3 BS01 rna F 0 R599 S605 R606 K607 L610 R624 R629 R89 S95 R96 K97 L100 R114 R119 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q46455 15665870 13 ~ 35 GSETQKKLLKDLEDKYRVSRWQPPSFKEVAGSFNLDPSELEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRRVGDKRVVV 1wsu C 2.3 BS01 rna G 0 R599 S605 R606 K607 L610 R73 S79 R80 K81 L84 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q46455 15665870 13 ~ 35 KLLKDLEDKYRVSRWQPPSFKEVAEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRKRVVV 1wtg H 2.2 BS02 3BP H 1 H57 D60 G97 T98 S170H P170I D189 S190 C191 K192 S195 S214 W215 G216 G219 H41 D44 G85 T86 S168 P169 D186 S187 C188 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 ic50=93nM remove_due_to_license_issue IC50=93nM P08709 15607748 2001 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1wu1 A 2.3 BS03 D91 A 1 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=18nM remove_due_to_license_issue P00742 15911309 700 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 1wug A -1.00 BS01 NP1 A 1 E750 V752 E756 A757 Y802 Y809 E36 V38 E42 A43 Y88 Y95 2.3.1.48,2.3.1.57 0004402 remove_due_to_license_issue IC50=1600nM Q92831 15724976 201 GSHMSKEPRDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLIDK 1wum A -1.00 BS01 NP2 A 1 E750 V752 E756 A757 Y802 Y809 E36 V38 E42 A43 Y88 Y95 2.3.1.48,2.3.1.57 0004402 remove_due_to_license_issue Q92831 15724976 201 GSHMSKEPRDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLIDK 1wun H 2.4 BS02 P5B H 1 H57 D60 G97 T98 S170H P170I D189 S190 C191 K192 S195 S214 W215 G216 Q217 G219 H41 D44 G85 T86 S168 P169 D186 S187 C188 K189 S192 S211 W212 G213 Q214 G215 3.4.21.21 0004252,0006508 ic50=62nM remove_due_to_license_issue P08709 15629154 2001 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1wuq A 2.0 BS02 8GT A 1 H110 H111 V148 Q149 E150 R183 H78 H79 V116 Q117 E118 R151 C108 E109 H110 H111 Q149 H177 C179 C76 E77 H78 H79 Q117 H145 C147 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 811 VDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wuq A 2.0 BS03 8GT A 2 G131 L132 S133 K134 R137 G99 L100 S101 K102 R105 C108 E109 H110 H111 Q149 H177 C179 C76 E77 H78 H79 Q117 H145 C147 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 815 VDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wuq B 2.0 BS01 8GT A 1 F89 G131 L132 S133 K134 R137 F57 G99 L100 S101 K102 R105 C108 E109 H110 H111 Q149 H177 C179 C76 E77 H78 H79 Q117 H145 C147 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 811 VDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wuq B 2.0 BS03 8GT C 1 H110 H111 V148 Q149 E150 R183 H78 H79 V116 Q117 E118 R151 C108 E109 H110 H111 Q149 H177 C179 C76 E77 H78 H79 Q117 H145 C147 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 812 VDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wur A 1.82 BS02 8DG A 1 C108 H110 H111 V148 Q149 E150 C179 R183 C77 H79 H80 V117 Q118 E119 C148 R152 C108 E109 H110 H111 Q149 H177 C179 C77 E78 H79 H80 Q118 H146 C148 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 821 EVDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wur A 1.82 BS03 8DG A 2 G131 L132 S133 K134 R137 G100 L101 S102 K103 R106 C108 E109 H110 H111 Q149 H177 C179 C77 E78 H79 H80 Q118 H146 C148 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 825 EVDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wur B 1.82 BS01 8DG A 1 G131 L132 S133 K134 R137 G100 L101 S102 K103 R106 C108 E109 H110 H111 Q149 H177 C179 C77 E78 H79 H80 Q118 H146 C148 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 821 EVDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wur B 1.82 BS03 8DG C 1 H110 H111 V148 Q149 E150 H177 C179 R183 H79 H80 V117 Q118 E119 H146 C148 R152 C108 E109 H110 H111 Q149 H177 C179 C77 E78 H79 H80 Q118 H146 C148 3.5.4.16 0003934,0005525,0005737,0006729,0006730,0008270,0009058,0016787,0046654,0046872 remove_due_to_license_issue Q5SH52 16169877 822 EVDLERLQALAAEWLQVIGEDPGREGLLKTPERVAKAWAFLTRGYRQRLEEVVGGAVFPAEGSEMVVVKGVEFYSMCEHHLLPFFGKVHIGYIPDGKILGLSKFARIVDMFARRLQVQERLAVQIAEAIQEVLEPQGVGVVVEGVHLCMMMRGVEKQHSRTVTSAMLGVFRENQKTREEFLSHLR 1wv7 H 2.7 BS02 5PI H 1 H57 D60 G97 T98 D170G S170H P170I D189 S190 C191 K192 S195 V213 S214 W215 G216 Q217 G219 H41 D44 G85 T86 D167 S168 P169 D186 S187 C188 K189 S192 V210 S211 W212 G213 Q214 G215 3.4.21.21 0004252,0006508 remove_due_to_license_issue P08709 15629154 2001 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1wva A 1.94 BS03 S2C A 1 H126 D128 H141 D183 D232 D234 E277 H122 D124 H137 D179 D228 D230 E273 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=270nM remove_due_to_license_issue P05089 16141327 1317 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHK 1wvc A 2.5 BS02 CTP A 1 L8 A9 G10 G11 G13 T14 R15 K25 S106 R111 G130 D131 L7 A8 G9 G10 G12 T13 R14 K24 S105 R110 G129 D130 2.7.7.33 0000166,0009058,0009103,0009243,0016779,0046872,0047343 remove_due_to_license_issue Q8Z5I4 15634670 401 ASKAVILAGGLGTRLSEETIVKPKPMVEIGGKPILWHIMKMYSVHGIKDFIICCGYKGYVIKEYFANYFLHMSDVTFHMAENRMEVHHKRVEPWNVTLVDTGDSSMTGGRLKRVAEYVKDDEAFLFTYGDGVADLDIKATIDFHKAHGKKATLTATFPPGRGALDIQAGQVRSFQKGDGAMINGGFFVLNPSVIDLIDNDATTWEQEPLMTLAQQGELMAFEHPGFWQPMDTLRDKVYLEGLWEKGKAPWKTWE 1wvj A 1.75 BS01 IBC A 1 E13 Y61 L90 T91 R96 G141 S142 T143 L192 E193 M196 E13 Y61 L90 T91 R96 G141 S142 T143 L192 E193 M196 ? 0015276,0016020 Ki=185nM remove_due_to_license_issue P19491 15794751 1001 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1wwd A -1.00 BS01 rna B 0 L21 D22 R23 Q25 A27 Y28 K30 A36 K42 L21 D22 R23 Q25 A27 Y28 K30 A36 K42 ? 0003676,0008270 remove_due_to_license_issue P03332 15751950 493 ~ 498 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSLL 1wwe A -1.00 BS01 rna B 0 G14 E15 L21 D22 R23 Q25 A27 Y28 A36 K41 K42 G14 E15 L21 D22 R23 Q25 A27 Y28 A36 K41 K42 ? 0003676,0008270 remove_due_to_license_issue P03332 15751950 517 ~ 523 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSLL 1wwf A -1.00 BS01 rna B 0 R16 L21 D22 R23 Q25 A27 Y28 A36 K37 K41 K42 P43 R16 L21 D22 R23 Q25 A27 Y28 A36 K37 K41 K42 P43 ? 0003676,0008270 remove_due_to_license_issue P03332 15751950 504 ~ 510 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSLL 1wwg A -1.00 BS01 rna B 0 R18 L21 D22 R23 Q25 A27 Y28 W35 A36 K37 K41 K42 R18 L21 D22 R23 Q25 A27 Y28 W35 A36 K37 K41 K42 ? 0003676,0008270 remove_due_to_license_issue P03332 15751950 304 ~ 309 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSLL 1wxz A 2.8 BS02 FRL A 1 H17 D19 L58 F61 L62 F65 L106 W117 G184 D185 D296 H14 D16 L55 F58 L59 F62 L103 W114 G181 D182 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 remove_due_to_license_issue P56658 16033254 401 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 1wzy A 2.5 BS01 F29 A 1 A52 I53 K54 I103 Q105 M108 E109 T110 N154 L156 D167 A45 I46 K47 I96 Q98 M101 E102 T103 N147 L149 D160 D149 K151 S153 N154 D167 T190 D142 K144 S146 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.56uM remove_due_to_license_issue IC50=560nM P28482 16242327 1001 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 1x07 A 2.2 BS02 IPE A 1 M25 D26 G27 N28 G29 R30 R39 H43 A69 R77 M16 D17 G18 N19 G20 R21 R30 H34 A60 R68 D26 H43 L137 D17 H34 L128 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 Kd=520uM remove_due_to_license_issue P60472 15788389 901 SEKLPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 1x0n A -1.00 BS01 DTF A 1 R67 R86 Q106 H107 F108 K109 L111 W121 R8 R27 Q47 H48 F49 K50 L52 W62 ? remove_due_to_license_issue IC50=20nM P62993 174 WFFGKIPRAKAEEMLSKQRHDGAFLIRESESAPGDFSLSVKFGNDVQHFKVLRDGAGKYFLWVVKFNSLNELVDYHRSTSVSRNQQIFLRDIEQVPQQPT 1x1z A 1.45 BS01 BMP A 1 D20 K42 K72 M126 S127 P180 Q185 G202 R203 D10 K32 K62 M116 S117 P170 Q175 G192 R193 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=8.8pM remove_due_to_license_issue O26232 16248642 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 1x1z A 1.45 BS02 BMP A 2 D75 I76 T79 D65 I66 T69 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=8.8pM remove_due_to_license_issue O26232 16248642 302 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 1x1z B 1.45 BS01 BMP A 1 D1075 I1076 T1079 D65 I66 T69 K1042 D1070 K1072 D1075 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue O26232 16248642 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 1x1z B 1.45 BS02 BMP A 2 D1020 K1042 K1072 M1126 S1127 P1180 Q1185 G1202 R1203 D10 K32 K62 M116 S117 P170 Q175 G192 R193 K1042 D1070 K1072 D1075 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue O26232 16248642 302 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 1x38 A 1.698 BS02 IDD A 1 D95 R158 K206 H207 M250 Y253 D285 W286 W434 E491 D95 R158 K206 H207 M250 Y253 D285 W286 W434 E491 D285 E491 D285 E491 3.2.1.21 0004553,0005975,0016798 Ki=1.7nM remove_due_to_license_issue Q9XEI3 16342944 1001 DYVLYKDATKPVEDRVADLLGRMTLAEKIGQMTQIERLVATPDVLRDNFIGSLLSGGGSVPRKGATAKEWQDMVDGFQKACMSTRLGIPMIYGIDAVHGQNNVYGATIFPHNVGLGATRDPYLVKRIGEATALEVRATGIQYAFAPCIAVCRDPRWGRCYESYSEDRRIVQSMTELIPGLQGDVPKDFTSGMPFVAGKNKVAACAKHFVGDGGTVDGINENNTIINREGLMNIHMPAYKNAMDKGVSTVMISYSSWNGVKMHANQDLVTGYLKDTLKFKGFVISDWEGIDRITTPAGSDYSYSVKASILAGLDMIMVPNKYQQFISILTGHVNGGVIPMSRIDDAVTRILRVKFTMGLFENPYADPAMAEQLGKQEHRDLAREAARKSLVLLKNGKTSTDAPLLPLPKKAPKILVAGSHADNLGYQCGGWTIEWQGDTGRTTVGTTILEAVKAAVDPSTVVVFAENPDAEFVKSGGFSYAIVAVGEHPYTETKGDNLNLTIPEPGLSTVQAVCGGVRCATVLISGRPVVVQPLLAASDALVAAWLPGSEGQGVTDALFGDFGFTGRLPRTWFKSVDQLPMNVGDAHYDPLFRLGYGLTTNAT 1x39 A 1.8 BS02 IDE A 1 D95 R158 K206 H207 M250 Y253 D285 W286 R291 E491 D95 R158 K206 H207 M250 Y253 D285 W286 R291 E491 D285 E491 D285 E491 3.2.1.21 0004553,0005975,0016798 Ki=0.6nM remove_due_to_license_issue Q9XEI3 16342944 1001 DYVLYKDATKPVEDRVADLLGRMTLAEKIGQMTQIERLVATPDVLRDNFIGSLLSGGGSVPRKGATAKEWQDMVDGFQKACMSTRLGIPMIYGIDAVHGQNNVYGATIFPHNVGLGATRDPYLVKRIGEATALEVRATGIQYAFAPCIAVCRDPRWGRCYESYSEDRRIVQSMTELIPGLQGDVPKDFTSGMPFVAGKNKVAACAKHFVGDGGTVDGINENNTIINREGLMNIHMPAYKNAMDKGVSTVMISYSSWNGVKMHANQDLVTGYLKDTLKFKGFVISDWEGIDRITTPAGSDYSYSVKASILAGLDMIMVPNKYQQFISILTGHVNGGVIPMSRIDDAVTRILRVKFTMGLFENPYADPAMAEQLGKQEHRDLAREAARKSLVLLKNGKTSTDAPLLPLPKKAPKILVAGSHADNLGYQCGGWTIEWQGDTGRTTVGTTILEAVKAAVDPSTVVVFAENPDAEFVKSGGFSYAIVAVGEHPYTETKGDNLNLTIPEPGLSTVQAVCGGVRCATVLISGRPVVVQPLLAASDALVAAWLPGSEGQGVTDALFGDFGFTGRLPRTWFKSVDQLPMNVGDAHYDPLFRLGYGLTTNAT 1x6u A 2.7 BS01 DO8 A 1 N26 K55 N62 Q113 F117 K138 D199 H202 F237 E239 P252 N26 K55 N62 Q113 F117 K138 D199 H202 F225 E227 P240 N26 K60 D250 N26 K60 D238 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0032991,0042802 remove_due_to_license_issue P0A715 16023668 2634 MKQKVVSIGDINVANDLPFVLFGGMNVLESRDLAMRICEHYVTVTQKLGIPYVFKASFDKANRSSIHSYRGPGLEEGMKIFQELKQTFGVKIITDVHEPSQAQPVADVVDVIQLPAFLARQTDLVEAMAKTGAVINVKKPQFVSPGQMGNIVDKFKEGGNEKVILCDRGANFGYDNLVVDMLGFSIMKKVSGNSPVIFDVTHALQRAQVAELARAGMAVGLAGLFIEAHPDPEHAKCDGPSALPLAKLEPFLKQMKAIDDLVKGFEELDTSK 1x70 A 2.1 BS01 715 A 1 E205 E206 V207 S209 F357 R358 S630 Y631 Y662 Y666 N710 V711 E167 E168 V169 S171 F319 R320 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=18nM remove_due_to_license_issue IC50=18nM, Kd=1.3nM P27487 15634008 801 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 1x76 A 2.2 BS02 697 A 1 M295 E305 L339 I376 H475 L476 M33 E43 L77 I114 H203 L204 ? 0003677,0004879,0006355 ic50=1.9nM remove_due_to_license_issue IC50=2.2nM Q92731 15548008 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1x78 A 2.3 BS02 244 A 1 M295 L298 L301 E305 L339 I376 F377 H475 L476 M33 L36 L39 E43 L77 I114 F115 H203 L204 ? 0003677,0004879,0006355 ic50=14nM remove_due_to_license_issue IC50=14nM Q92731 15548008 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 1x7a C 2.9 BS01 187 C 1 N97 Y99 R143 F174 D189 S190 C191 Q192 I213 S214 W215 G216 E217 E219 C220 G226 N84 Y86 R132 F162 D179 S180 C181 Q182 I203 S204 W205 G206 E207 E208 C209 G216 H57 H41 3.4.21.22 0004252,0006508 remove_due_to_license_issue P16293 15454208 298 IVGGENAKPGQFPWQVLLNGKIDAFCGGSIINEKWVVTAAHCIEPGVKITVVAGEYNTEETEPTEQRRNVIRAIPHHSYNATVNKYSHDIALLELDEPLTLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFNRGRSATILQYLKVPLVDRATCLRSTKFTIYSNMFCAGFHEGGKDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAVKGKYGIYTKVSRYVNWIKEKTKLT 1x7b A 2.3 BS02 041 A 1 M295 E305 L339 M340 L343 I373 I376 H475 L476 M33 E43 L77 M78 L81 I111 I114 H203 L204 ? 0003677,0004879,0006355 ic50=4.1nM remove_due_to_license_issue IC50=5nM Q92731 15548008 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 1x7e A 2.8 BS02 244 A 1 L346 E353 F404 M421 I424 L428 H524 L525 L42 E49 F100 M117 I120 L124 H213 L214 ? remove_due_to_license_issue IC50=1152nM P03372 15548008 201 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPVKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRL 1x7r A 2.0 BS02 GEN A 1 M343 L346 E353 L387 I424 H524 L525 M31 L34 E41 L75 I112 H212 L213 ? ic50=360nM remove_due_to_license_issue IC50=395nM, EC50=240nM, Ki=370nM P03372 15576033 201 LALSLTADQMVSALLDAEPPILYSESEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPVKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAH 1x81 B 3.5 BS02 JAN B 1 L96 W102 W106 D359 Y361 L75 W81 W85 D338 Y340 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H227 R270 K273 D276 C278 Y279 D331 D338 H341 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 15454228 1 PLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQK 1x8b A 1.81 BS03 824 A 1 I305 A326 K328 V360 N376 E377 Y378 C379 G382 F433 D463 I15 A36 K38 V70 N86 E87 Y88 C89 G92 F143 D153 D426 K428 D136 K138 2.7.10.2 0004672,0005524,0006468 ic50=97nM remove_due_to_license_issue IC50=97nM P30291 15837193 901 MKSRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVL 1x8d A 1.8 BS01 RNS A 1 Y18 H22 Y41 W76 W77 Y18 H22 Y41 W76 W77 5.1.3.32 0005737,0016853,0016857,0019299,0019301,0042803,0062192 Kd=6.16mM remove_due_to_license_issue P32156 15876375 1105 MIRKAFVMQVNPDAHEEYQRRHNPIWPELEAVLKSHGAHNYAIYLDKARNLLFAMVEIESEERWNAVASTDVCQRWWKYMTDVMPANPDNSPVSSELQEVFYLP 1x8d B 1.8 BS01 RNS B 1 Y18 H22 Y41 W76 W77 Y18 H22 Y41 W76 W77 5.1.3.32 0005737,0016853,0016857,0019299,0019301,0042803,0062192 Kd=6.16mM remove_due_to_license_issue P32156 15876375 1106 MIRKAFVMQVNPDAHEEYQRRHNPIWPELEAVLKSHGAHNYAIYLDKARNLLFAMVEIESEERWNAVASTDVCQRWWKYMTDVMPANPDNSPVSSELQEVFYLP 1x8j A 2.35 BS03 AOI A 1 I111 Y298 I105 Y292 R73 H164 S193 R67 H158 S187 ? 0008146,0016740,0046872 Ki=0.11uM remove_due_to_license_issue Q26490 15608121 400 LPFPYEFRELNPEEDKLVKANLGAFPTTYVKLGPKGYMVYRPYLKDAANIYNMPLRPTDVFVASYQRSGTTMTQELVWLIENDLNFEAAKTYMSLRYIYLDGFMIYDPEKQEEYNDILPNPENLDMERYLGLLEYSSRPGSSLLAAVPPTEKRFVKTHLPLSLMPPNMLDTVKMVYLARDPRDVAVSSFHHARLLYLLNKQSNFKDFWEMFHRGLYTLTPYFEHVKEAWAKRHDPNMLFLFYEDYLKDLPGSIARIADFLGKKLSEEQIQRLSEHLNFEKFKNNGAVNMEDYREIGILADGEHFIRKGKAGCWRDYFDEEMTKQAEKWIKDNLKDTDLRYPNM 1x8r A 1.5 BS01 SC1 A 1 K22 S23 R27 G96 T97 R124 S169 S170 Q171 S197 Y200 D313 N336 K340 E341 H385 K411 K22 S23 R27 G96 T97 R124 S169 S170 Q171 S197 Y200 D313 N336 K340 E341 H385 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 Ki=2.9uM remove_due_to_license_issue Kd=15nM, Ki=15nM P0A6D3 15736934 601 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 1x8t A 1.9 BS01 RC1 A 1 K22 S23 R27 T97 S169 S170 Q171 S197 Y200 D313 N336 K340 R344 H385 R386 K22 S23 R27 T97 S169 S170 Q171 S197 Y200 D313 N336 K340 R344 H385 R386 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 Ki=16nM remove_due_to_license_issue P0A6D3 15736934 501 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 1xa5 A 2.12 BS05 KAR A 1 L18 L39 F68 M71 M72 I85 M109 M145 L16 L37 F66 M69 M70 I81 M105 M141 V35 V33 ? 0000922,0002027,0005509,0005513,0005515,0005737,0005813,0005819,0005829,0005856,0005876,0008179,0010856,0010880,0019901,0019904,0030017,0031432,0032465,0032991,0034704,0043209,0043539,0044325,0046872,0051592,0055117,0060315,0060316,0072542,0097720,0098901,1902494 Kd=316nM remove_due_to_license_issue P62157 15596444 153 QLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAK 1xap A 2.1 BS01 TTB A 1 F221 L224 L259 L262 F279 S280 R387 L407 F47 L50 L85 L88 F105 S106 R210 L230 ? 0003677,0004879,0005634,0006355,0048384 Kd=2.5nM remove_due_to_license_issue EC50=4nM, Ki=0.500000nM, Kd=5nM, IC50=5nM P10826 15319780 1 AELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALKIYIRKRRPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLEN 1xbb A 1.57 BS01 STI A 1 L377 V385 A400 M448 E449 M450 A451 E452 G454 L501 L15 V23 A38 M81 E82 M83 A84 E85 G87 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 Ki=5uM remove_due_to_license_issue Ki=5000nM, Kd=>10000nM, IC50=>10000nM P43405 15507431 1 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 1xbc A 2.0 BS01 STU A 1 L377 G378 A400 M448 M450 A451 G454 P455 R498 N499 L501 D512 L15 G16 A38 M80 M82 A83 G86 P87 R130 N131 L133 D144 D494 A496 R498 N499 D512 K533 D126 A128 R130 N131 D144 K165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.012uM remove_due_to_license_issue P43405 15507431 1 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNE 1xbo A 2.5 BS01 IX1 A 1 Y20 R24 Y46 D48 V49 D181 C215 S216 A217 I219 G220 R221 R254 G259 Q262 L299 Y19 R23 Y45 D47 V48 D180 C214 S215 A216 I218 G219 R220 R253 G258 Q261 L298 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.92uM remove_due_to_license_issue IC50=920nM P18031 15482920 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 1xc8 A 1.95 BS01 dna B 0 E2 E5 K57 H72 R74 M75 G170 N171 I172 S217 I219 R220 T221 Y222 Y238 K254 K256 R260 E2 E5 K57 H72 R74 M75 G170 N171 I172 S217 I219 R220 T221 Y222 Y238 K254 K256 R260 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 15249553 1 ~ 14 PELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSIRTYSALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1xc8 A 1.95 BS02 dna C 0 H91 V108 R109 K110 F111 H91 V108 R109 K110 F111 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 15249553 15 ~ 28 PELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSIRTYSALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 1xd0 A 2.0 BS01 ARE A 1 W58 W59 Y62 Q63 H101 Y151 T163 D197 K200 H201 E233 E240 H299 D300 H305 W58 W59 Y62 Q63 H101 Y151 T163 D197 K200 H201 E233 E240 H299 D300 H305 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 Ki=0.075uM remove_due_to_license_issue P04746 15736945 501 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 1xdd A 2.2 BS02 AAY A 1 Y166 I235 Y257 Y39 I108 Y130 ? ic50=0.2uM remove_due_to_license_issue P20701 15304496 401 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 1xdd A 2.2 BS03 AAY B 1 K304 Y307 K177 Y180 ? ic50=0.2uM remove_due_to_license_issue P20701 15304496 501 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 1xdg A 2.1 BS02 AB8 A 1 L132 I235 I255 Y257 L302 L5 I108 I128 Y130 L175 ? ic50=0.05uM remove_due_to_license_issue IC50=50nM P20701 15304496 401 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 1xdg A 2.1 BS03 AB8 B 1 V308 I309 V181 I182 ? ic50=0.05uM remove_due_to_license_issue IC50=50nM P20701 15304496 501 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 1xff A 1.8 BS01 GLU A 1 C1 R73 W74 T76 H86 N98 G99 D123 C1 R73 W74 T76 H86 N98 G99 D123 C1 R26 G27 W74 N98 G99 C1 R26 G27 W74 N98 G99 2.6.1.16 Ki=15uM remove_due_to_license_issue P17169 8805567 5300 CGIVGAIAQRDVAEILLEGLRRLEYRGYDSAGLAVVDAEGHMTRLRRLGKVQMLAQAAEEHPLHGGTGIAHTRWATHGEPSEVNAHPHVSEHIVVVHNGIIENHEPLREELKARGYTFVSETDTEVIAHLVNWELKQGGTLREAVLRAIPQLRGAYGTVIMDSRHPDTLLAARSGSPLVIGLGMGENFIASDQLALLPVTRRFIFLEEGDIAEITRRSVNIFDKTGAEVKRQDIESNL 1xfv A 3.35 BS02 3AT A 1 R329 K353 G547 T548 G578 E588 R266 K290 G484 T485 G515 E525 Y626 Y627 R630 Y679 D686 Y563 Y564 R567 Y616 D623 4.6.1.1 0003824,0005576,0008237,0008294,0046872 remove_due_to_license_issue P40136 15719022 903 NNLVKTEFTNETLDKIQQTQDLLKKIPKDVLEIYSELGGEIYFTDIDLVEHKELQDLSEEEKNSMNSRGEKVPFASRFVFEKKRETPKLIINIKDYAINSEQSKEVYYEIGKGISLDIISKDKSLDPEFLNLIKSLSDDSDSSDLLFSQKFKEKLELNNKSIDINFIKENLTEFQHAFSLAFSYYFAPDHRTVLELYAPDMFEYMNKLEKGGFEKISESLKKEGVEKDRIDVLKGEKALKASGLVPEHADAFKKIARELNTYILFRPVNKLATNLIKSGVATKGLNVHGKSSDWGPVAGYIPFDQDLSKKHGQQLAVEKGNLENKKSITEHEGEIGKIPLKLDHLRIEELKENGIILKGKKEIDNGKKYYLLESNNQVYEFRISDENNEVQYKTKEGKITVLGEKFNWRNIEVMAKNVEGVLKPLTADYDLFALAPSLTEIKKQIPQKEWDKVVNTPNSLEKQKGVTNLLIKYGIERKPDSTKGTLSNWQKQMLDRLNEAVKYTGYTGGDVVNHGTEQDNEEFPEKDNEIFIINPEGEFILTKNWEMTGRFIEKNITGKDYLYYFNRSYNKIAPGNKAYIEWTDPITKAKINTIPTSAEFIKNLSSIRRSSNVGVYKDSGDKDEFAKKESVKKIAGYLSDYYNSANHIFSQEKKRKISIFRGIQAYNEIENVLKSKQIAPEYKNYFQYLKERITNQVQLLLTHQKSNIEFKLLYKQLNFTENETDNFEVFQKIID 1xge A 1.9 BS03 DOR A 1 H18 R20 H139 C221 L222 A252 H254 A266 G267 H15 R17 H136 C218 L219 A249 H251 A263 G264 H16 H18 K102 H139 H177 D250 H13 H15 K99 H136 H174 D247 3.5.2.3 0004151,0005737,0005829,0006207,0006221,0008270,0016787,0016812,0019856,0042803,0044205,0046872 Kd=20.8uM remove_due_to_license_issue P05020 15826651 1410 SQVLKIRRPDDWHLHLRDGDMLKTVVPYTSEIYGRAIVMPNLAPPVTTVEAAVAYRQRILDAVPAGHDFTPLMTCYLTDSLDPNELERGFNEGVFTAAKLYPANATTNSSHGVTSVDAIMPVLERMEKIGMPLLVHGEVTHADIDIFDREARFIESVMEPLRQRLTALKVVFEHITTKDAADYVRDGNERLAATITPQHLMFNRNHMLVGGVRPHLYCLPILKRNIHQQALRELVASGFNRVFLGTDSAPHARHRKESSCGCAGCFNAPTALGSYATVFEEMNALQHFEAFCSVNGPQFYGLPVNDTFIELVREEQQVAESIALTDDTLVPFLAGETVRWSVK 1xgi B 1.96 BS01 NST B 1 S64 Q120 N152 Y221 G317 A318 T319 G320 S61 Q117 N149 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=14uM remove_due_to_license_issue P00811 15796528 416 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1xgj A 1.97 BS01 HTC A 1 S64 L119 N152 Y221 G317 A318 T319 G320 S61 L116 N149 Y218 G307 A308 T309 G310 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K305 A308 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1uM remove_due_to_license_issue Ki=1000nM P00811 15796528 777 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1xh4 A 2.45 BS02 R69 A 1 G50 T51 G52 S53 F54 R56 V57 A70 K72 L74 Q84 E91 V123 E127 E170 N171 L173 T183 D184 G186 F327 G37 T38 G39 S40 F41 R43 V44 A57 K59 L61 Q71 E78 V110 E114 E157 N158 L160 T170 D171 G173 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=34nM remove_due_to_license_issue IC50=30nM P00517 15634010 351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1xh5 A 2.05 BS02 R68 A 1 G50 T51 G52 S53 F54 G55 V57 A70 K72 V123 E127 E170 N171 L173 T183 D184 F327 G37 T38 G39 S40 F41 G42 V44 A57 K59 V110 E114 E157 N158 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=3400nM remove_due_to_license_issue P00517 15634010 1001 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1xh6 A 1.9 BS02 R94 A 1 G50 T51 G52 S53 F54 V57 A70 K72 Q84 E127 E170 N171 L173 T183 D184 F187 G33 T34 G35 S36 F37 V40 A53 K55 Q67 E110 E153 N154 L156 T166 D167 F170 D166 K168 E170 N171 D184 T201 D149 K151 E153 N154 D167 T184 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=48nM remove_due_to_license_issue IC50=400nM P00517 15634010 351 FLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1xh7 A 2.47 BS02 R96 A 1 G50 T51 G52 S53 F54 V57 A70 K72 L74 Q84 E91 V123 E127 E170 N171 L173 T183 D184 F187 F327 G41 T42 G43 S44 F45 V48 A61 K63 L65 Q75 E82 V114 E118 E161 N162 L164 T174 D175 F178 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=150nM remove_due_to_license_issue IC50=1900nM P00517 15634010 351 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1xh8 A 1.6 BS02 R55 A 1 G50 T51 G52 S53 F54 V57 K72 L74 Q84 E91 V123 E170 N171 L173 T183 D184 G186 F327 G39 T40 G41 S42 F43 V46 K61 L63 Q73 E80 V112 E159 N160 L162 T172 D173 G175 F316 D166 K168 E170 N171 D184 T201 D155 K157 E159 N160 D173 T190 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=1700nM remove_due_to_license_issue IC50=1700nM P00517 15634010 351 QESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1xh9 A 1.64 BS02 R69 A 1 G50 T51 G52 F54 V57 A70 K72 L74 E84 E91 A123 E127 E170 N171 M173 T183 D184 G186 F327 G38 T39 G40 F42 V45 A58 K60 L62 E72 E79 A111 E115 E158 N159 M161 T171 D172 G174 F315 D166 K168 E170 N171 D184 T201 D154 K156 E158 N159 D172 T189 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=17nM remove_due_to_license_issue IC50=30nM P00517 15634010 351 ESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKEIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGLAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1xhy A 1.85 BS01 KAI A 1 Y58 P86 T88 R93 G138 S139 T140 E190 Y58 P86 T88 R93 G138 S139 T140 E190 ? 0015276,0016020 Ki=624nM remove_due_to_license_issue EC50=380000nM, Ki=3690nM P19491 15591246 1001 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 1xjd A 2.0 BS01 STU A 1 L386 G387 K388 G389 V394 A407 M458 E459 Y460 L461 G464 D465 D508 N509 L511 D522 L10 G11 K12 G13 V18 A31 M82 E83 Y84 L85 G88 D89 D132 N133 L135 D146 D504 K506 D508 N509 D522 T542 D128 K130 D132 N133 D146 T166 2.7.11.13 0004672,0004674,0004697,0005524,0006468 Ki=0.33nM remove_due_to_license_issue Q04759 15364937 200 IEDFILHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNTFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPQNMFRNFSF 1xjv A 1.73 BS01 dna B 0 F31 K33 Y36 S38 K39 G40 T41 D42 T48 L60 F62 Y89 Q94 Y161 Y223 D224 S243 H245 H266 G267 S270 Y271 R273 F26 K28 Y31 S33 K34 G35 T36 D37 T43 L55 F57 Y84 Q89 Y153 Y215 D216 S235 H237 H258 G259 S262 Y263 R265 ? 0000723,0000781,0003677,0043047 remove_due_to_license_issue Q9NUX5 15558049 1 ~ 10 ATNYIYTPLNQLKGGTIVNVYGVVKFFKPPYLSKGTDYCSVVTIVDQTNVKLTCLLFSGNYEALPIIYKNGDIVRFHRLKIQVYKKETQGITSSGFASLTFEGTLGAPIIPRTSSKYFNFTTEDHKMVEALRVWASTHMSTLLKLCDVQPMQYFDLTCQLLGKAEVDGASFLLKVWDGTRTPFPSWRVLIQDLVLEGDLSHIHRLQNLTIDILVYDNHVHVARSLKVGSFLRIYSLHTKLQSMNSENQTMLSLEFHLHGGTSYGRGIRVLPESNSDVDQLKKDLESANLTA 1xk5 A 2.4 BS01 TPG A 1 S105 E106 W107 G127 K128 R129 K144 D255 W276 S9 E10 W11 G31 K32 R33 K48 D159 W180 ? 0005634,0005737,0061015 Kd=1uM remove_due_to_license_issue O95149 15920472 400 HYANQLMLSEWLIDVPSDLGQEWIVVVCPVGKRALIVASRGSTSAYTKSGYCVNRFSSLLPGGNRRNSTAKDYTILDCIYNEVNQTYYVLDVMCWRGHPFYDCQTDFRFYWMHSKLPEEEGLGEKTKLNPFKFVGLKNFPCTPESLCDVLSMDFPFEVDGLLFYHKQTHYSPGSTPLVGWLRPYMVSDVLGVAVPAGPLTTKPD 1xk9 A 2.1 BS01 P34 A 1 H440 G441 Y470 I471 A478 Y481 Q485 H42 G43 Y72 I73 A80 Y83 Q87 E553 E155 2.4.2.36 0047286 Ki=140nM remove_due_to_license_issue P11439 15458385 1001 EFLGDGGDVSFSTRGTQNWTVERLLQAHRQLEERGYVFVGYHGTFLEAAQSIVFGGVRARSQDLDAIWRGFYIAGDPALAYGYAQDQEPDARGRIRNGALLRVYVPRSSLPGFYRTSLTLAAPEAAGEVERLIGHPLPLRLDAITGPEEEGGRLETILGWPLAERTVVIPSAIPTDPRNVGGDLDPSSIPDKEQAISALPDYAS 1xka C 2.3 BS02 4PP C 1 T98 Y99 F174 D189 A190 Q192 S195 V213 W215 G216 G218 T84 Y85 F162 D179 A180 Q182 S185 V203 W205 G206 G208 G193 S195 G196 G183 S185 G186 3.4.21.6 0004252,0006508 Ki=131nM remove_due_to_license_issue IC50=270nM P00742 9618463 500 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTR 1xkk A 2.4 BS01 FMM A 1 A743 K745 M766 C775 R776 L788 T790 M793 L799 D800 L844 T854 D855 F856 A38 K40 M57 C66 R67 L79 T81 M84 L90 D91 L135 T145 D146 F147 N756 I759 D837 A839 R841 N842 V843 D855 G911 N47 I50 D128 A130 R132 N133 V134 D146 G194 2.7.10.1 0004672,0004713,0005524,0006468 Ki=3nM remove_due_to_license_issue IC50=11nM, Kd=1.2nM, Ki=3.0nM P00533 15374980 91 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPVKIPVAIKELREKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMSNFYRALMDEVVDADEYLI 1xlx A 2.19 BS02 CIO A 1 M347 I410 M411 S442 Q443 F446 M185 I248 M249 S280 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.025uM remove_due_to_license_issue IC50=100nM, Ki=38nM Q07343 15576036 101 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xlz A 2.06 BS02 FIL A 1 T407 I410 M411 F414 M431 S442 Q443 F446 T245 I248 M249 F252 M269 S280 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.96uM remove_due_to_license_issue Q07343 15576036 1003 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xm4 A 2.31 BS02 PIL A 1 H234 M347 D392 L393 T407 I410 F414 S442 Q443 F446 H72 M185 D230 L231 T245 I248 F252 S280 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.041nM remove_due_to_license_issue IC50=1nM, Ki=1.5nM Q07343 15576036 1003 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xm6 A 1.92 BS02 5RM A 1 T407 I410 F414 S442 Q443 F446 T245 I248 F252 S280 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.42uM remove_due_to_license_issue IC50=420nM Q07343 15576036 1003 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPCQGLMEKFQFELTLD 1xmu A 2.3 BS02 ROF A 1 T345 M347 D392 L393 N395 Y403 W406 T407 I410 S442 Q443 F446 T191 M193 D238 L239 N241 Y249 W252 T253 I256 S288 Q289 F292 3.1.4.53 0004114,0007165,0008081 ic50=0.84nM remove_due_to_license_issue IC50=0.398nM, Ki=0.398107nM Q07343 15576036 101 RFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xmy A 2.4 BS02 ROL A 1 N395 M431 Q443 F446 N233 M269 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.57uM remove_due_to_license_issue Q07343 15576036 101 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xn0 A 2.31 BS02 ROL A 1 Y233 H234 T407 I410 M411 F414 Q443 F446 Y71 H72 T245 I248 M249 F252 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.57uM remove_due_to_license_issue Q07343 15576036 1003 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xn0 A 2.31 BS03 ROL A 2 I410 M411 F414 M431 Q443 F446 I248 M249 F252 M269 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.57uM remove_due_to_license_issue Q07343 15576036 1004 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xns A 2.8 BS01 dna C 0 F37 S38 H40 T41 I174 A175 K244 N245 R259 E262 K276 R282 Y283 S287 G288 H289 F18 S19 H21 T22 I155 A156 K225 N226 R240 E243 K257 R263 Y264 S268 G269 H270 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 15591069 1 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 1xns A 2.8 BS02 dna D 0 K43 M44 S47 R50 R81 A84 K86 T87 Q90 K132 R159 R173 T202 R241 V242 R243 K244 L256 S257 R259 R282 W315 Y324 K24 M25 S28 R31 R62 A65 K67 T68 Q71 K113 R140 R154 T183 R222 V223 R224 K225 L237 S238 R240 R263 W296 Y305 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 15591069 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 1xns B 2.8 BS01 dna C 0 R118 K122 R99 K103 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 15591069 1 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 1xns B 2.8 BS02 dna D 0 F37 S38 H40 T41 Q90 M97 R100 R101 R106 R121 I174 A175 K201 R243 K244 N245 R259 E262 R282 Y283 S287 G288 H289 F18 S19 H21 T22 Q71 M78 R81 R82 R87 R102 I155 A156 K182 R224 K225 N226 R240 E243 R263 Y264 S268 G269 H270 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 15591069 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTKTLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 1xnx A 2.9 BS01 ATE A 1 F171 N175 F227 K235 L253 F58 N62 F114 K122 L140 ? 0003677,0004879,0006355 remove_due_to_license_issue IC50=250nM O35627 15610734 500 LQLNQQQKELVQILLGAHTRHVGPLFDQFVQFKPPAYLFMHHRPFQPRGPVLPLLTHFADINTFMVQQIIKFTKDLPLFRSLTMEDQISLLKGAAVEILHISLNTTFCLQTENFFCGPLCYKMEDAVHAGFQYEFLESILHFHKNLKGLHLQEPEYVLMAATALFSPDRPGVTQREEIDQLQEEMALILNNHIMEQQSRLQSRFLYAKLMGLLADLRSINNAYSYELQRLEE 1xnz A 1.52 BS03 FCD A 1 Y62 H63 Y65 H79 D97 D108 H171 H178 E204 W221 E235 Y61 H62 Y64 H78 D96 D107 H170 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.24uM remove_due_to_license_issue IC50=116000nM P0AE18 15506752 268 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 1xo2 B 2.9 BS01 FSE B 1 I19 A41 K43 E61 F98 D104 Q149 L152 D163 I9 A31 K33 E51 F85 D91 Q136 L139 D150 D145 K147 Q149 N150 D163 A175 T182 D132 K134 Q136 N137 D150 A162 T169 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue IC50=850nM Q00534 15689157 309 QQYECVAEIGEGAYGKVFKARDLKNGGRFVALKRVRVQTGEEGMPLSTIREVAVLRHLETFEHPNVVRLFDVCTVSRETKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLARIYSFQMALTSVVVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPRDVALPRQAFHAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQDLER 1xoe A 2.2 BS01 ABX A 1 R119 E120 D152 R153 W180 R226 A248 E278 R294 R372 Y406 R36 E37 D69 R70 W97 R143 A165 E195 R211 R289 Y323 D152 E279 R294 R372 Y406 D69 E196 R211 R289 Y323 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=41nM remove_due_to_license_issue P03472 15582424 500 DFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1xog A 2.8 BS01 ABW A 1 E120 D152 R153 W180 E278 R294 R372 Y406 E37 D69 R70 W97 E195 R211 R289 Y323 D152 E279 R294 R372 Y406 D69 E196 R211 R289 Y323 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue P03472 15582424 1000 DFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 1xom A 1.55 BS02 CIO A 1 M273 I336 M337 F340 M357 Q369 F372 M188 I251 M252 F255 M272 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=0.011uM remove_due_to_license_issue IC50=11nM Q08499 15576036 603 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1xon A 1.72 BS02 PIL A 1 M273 D318 L319 T333 I336 M337 F340 M357 S368 Q369 F372 M188 D229 L230 T244 I247 M248 F251 M268 S279 Q280 F283 3.1.4.53 0004114,0007165,0008081 ic50=0.021nM remove_due_to_license_issue IC50=21nM Q08499 15576036 501 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1xoq A 1.83 BS02 ROF A 1 M273 D318 L319 N321 Y329 W332 T333 I336 M357 S368 Q369 F372 M188 D233 L234 N236 Y244 W247 T248 I251 M272 S283 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=0.68nM remove_due_to_license_issue IC50=0.400000nM Q08499 15576036 502 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1xor A 1.54 BS02 ZAR A 1 Y159 H160 H164 D318 I336 M357 Q369 F372 Y72 H73 H77 D228 I246 M267 Q279 F282 3.1.4.53 0004114,0007165,0008081 ic50=0.39uM remove_due_to_license_issue IC50=390nM Q08499 15576036 701 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1xos A 2.28 BS02 VIA A 1 M347 N395 I410 S429 M431 C432 Q443 F446 M186 N232 I247 S266 M268 C269 Q280 F283 3.1.4.53 0004114,0007165,0008081 ic50=20uM remove_due_to_license_issue IC50=20000nM Q07343 15576036 1 NEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1xow A 1.8 BS02 R18 A 1 L704 N705 Q711 M745 M749 F764 T877 L34 N35 Q41 M75 M79 F94 T201 ? remove_due_to_license_issue Kd=0.99nM, IC50=0.302000nM, EC50=0.013000nM, Ki=0.400000nM P10275 15525515 1001 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIATSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 1xoz A 1.37 BS02 CIA A 1 A767 Q775 V782 F786 L804 M816 Q817 F820 A235 Q243 V250 F254 L272 M284 Q285 F288 3.1.4.35 0004114,0007165,0008081 ic50=0.0012uM remove_due_to_license_issue IC50=4nM, Ki=10nM O76074 15576036 501 EEETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHPGVSNQFLINTNSELALMYNDESVLEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 1xp0 A 1.79 BS02 VDN A 1 Q817 F820 Q285 F288 3.1.4.35 0004114,0007165,0008081 ic50=0.001uM remove_due_to_license_issue IC50=0.890000nM, Ki=1nM O76074 15576036 201 EEETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHPGVSNQFLINTNSELALMYNDESVLEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 1xp1 A 1.8 BS01 AIH A 1 A350 D351 E353 L354 W383 F404 G521 H524 L525 A44 D45 E47 L48 W77 F98 G215 H218 L219 ? ic50=0.5nM remove_due_to_license_issue IC50=0.5nM P03372 15582421 600 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLHA 1xp6 A 1.7 BS01 AIU A 1 L346 T347 A350 D351 E353 W383 F404 G521 H524 K531 L40 T41 A44 D45 E47 W77 F98 G215 H218 K225 ? ic50=0.4nM remove_due_to_license_issue IC50=0.4nM P03372 15582421 600 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLHA 1xp9 A 1.8 BS01 AIJ A 1 L346 T347 A350 D351 E353 L354 W383 F404 G521 H524 L525 L40 T41 A44 D45 E47 L48 W77 F98 G215 H218 L219 ? ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P03372 15582421 600 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLHA 1xpc A 1.6 BS01 AIT A 1 L346 T347 A350 D351 E353 L354 W383 F404 G521 H524 C530 K531 L40 T41 A44 D45 E47 L48 W77 F98 G215 H218 C224 K225 ? ic50=1.7nM remove_due_to_license_issue IC50=1.7nM P03372 15582421 600 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLHA 1xpz A 2.02 BS02 4TZ A 1 N62 H94 L198 T199 T200 P202 W209 N60 H92 L195 T196 T197 P199 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=84nM remove_due_to_license_issue IC50=27nM P00918 15865431 270 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1xq0 A 1.76 BS02 4TR A 1 H94 V121 F131 L198 T199 P202 W209 H92 V119 F128 L195 T196 P199 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=454nM remove_due_to_license_issue IC50=137nM P00918 15865431 270 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1xqc A 2.05 BS01 AEJ A 1 M343 A350 D351 E353 W383 L387 F404 I424 L525 M27 A34 D35 E37 W67 L71 F88 I108 L207 ? ic50=63nM remove_due_to_license_issue EC50=23.2nM, IC50=63nM P03372 15658851 1001 ALSLTADQMVSALLDAEPPILYSESMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMPLYDLLLEMLDAHR 1xs7 D 2.8 BS01 MMI D 1 Y71 T72 Q73 W115 Y198 G230 T231 T232 N233 R235 Y75 T76 Q77 W119 Y202 G234 T235 T236 N237 R239 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue Ki=25nM P56817 15582402 386 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 1xsc A -1.00 BS01 ATP A 1 H42 Y87 A89 F133 E135 H42 Y87 A89 F133 E135 3.6.1.17 0004081,0005515,0005525,0005759,0006139,0006167,0006754,0006915,0008796,0008803,0016787,0034599 remove_due_to_license_issue P50583 15596429 154 GPLGSMALRACGLIIFRRCLIPKVDNNAIEFLLLQASDGIHHWTPPKGHVEPGEDDLETALRATQEEAGIEAGQLTIIEGFKRELNYVARNKPKTVIYWLAEVKDYDVEIRLSHEHQAYRWLGLEEACQLAQFKEMKAALQEGHQFLCSIEAL 1xt3 A 2.4 BS01 IDS C 1 L6 K12 K35 R36 G37 L6 K12 K35 R36 G37 ? 0005576,0016020,0031640,0035821,0044218,0090729 remove_due_to_license_issue P60301 15590643 6 LKCNKLVPLFYKTCPAGKNLCYKMFMVATPKVPVKRGCIDVCPKSSLLVKYVCCNTDRCN 1xt8 A 2.0 BS01 CYS A 1 F27 K30 R74 N89 T91 R96 T138 T139 H176 D177 F18 K21 R65 N80 T82 R87 T129 T130 H167 D168 ? Kd=0.14uM remove_due_to_license_issue Q0P9S0 15948956 401 LNSLDKIKQNGVVRIGVFGDKPPFGYVDEKGNNQGYDIALAKRIAKELFGDENKVQFVLVEAANRVEFLKSNKVDIILANFTQTPQRAEQVDFCSPYMKVALGVAVPKDSNITSVEDLKDKTLLLNKGTTADAYFTQNYPNIKTLKYDQNTETFAALMDKRGDALSHDNTLLFAWVKDHPDFKMGIKELGNKDVIAPAVKKGDKELKEFIDNLIIKLGQEQFFHKAYDETLKAHFGDDVKADDVVIEG 1xuc A 1.7 BS05 PB3 A 1 F217 L218 H222 L239 F241 I243 Y244 T245 Y246 T247 S250 F252 F114 L115 H119 L136 F138 I140 Y141 T142 Y143 T144 S147 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=72nM remove_due_to_license_issue IC50=72nM P45452 15734645 2001 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDED 1xud A 1.8 BS05 PB4 A 1 F217 L218 V219 H222 L239 F241 I243 Y244 T245 Y246 T247 S250 F252 F114 L115 V116 H119 L136 F138 I140 Y141 T142 Y143 T144 S147 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=8nM remove_due_to_license_issue IC50=8nM P45452 15734640 2001 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDED 1xug A 1.5 BS03 BAB A 1 F41 D189 S190 C191 Q192 V213 W215 G219 F24 D171 S172 C173 Q174 V191 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.09uM remove_due_to_license_issue P00760 9468142 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1xuo A 1.8 BS02 LA1 A 1 F153 Y166 V233 Y257 L302 I306 V308 F26 Y39 V106 Y130 L175 I179 V181 ? ic50=69nM remove_due_to_license_issue IC50=69nM P20701 15686945 401 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYV 1xur A 1.85 BS05 PB5 A 1 F217 L218 H222 L239 F241 I243 Y244 T245 Y246 T247 K249 S250 F252 F114 L115 H119 L136 F138 I140 Y141 T142 Y143 T144 K146 S147 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=6600nM remove_due_to_license_issue IC50=6600nM P45452 15734640 2001 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDED 1xws A 1.8 BS01 BI1 A 1 L44 G45 F49 V52 A65 E89 L120 E121 R122 L174 I185 D186 L12 G13 F17 V20 A33 E57 L88 E89 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=150nM, Kd=10.0nM P11309 1001 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 1xxe A -1.00 BS02 TUX A 1 H58 T179 F180 C181 I186 I189 G195 G198 Y212 K227 H56 T177 F178 C179 I184 I187 G193 G196 Y210 K225 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue O67648 15667205 320 LEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFCFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQKLT 1xxh D 3.45 BS02 AGS D 1 A7 R11 P12 V19 R47 G48 V49 G50 K51 T52 S53 L214 R215 A3 R7 P8 V15 R43 G44 V45 G46 K47 T48 S49 L210 R211 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 15556993 801 VLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 1xxi D 4.1 BS02 ADP D 1 A7 W10 R11 P12 V19 G48 V49 G50 K51 T52 S53 L214 R215 A3 W6 R7 P8 V15 G44 V45 G46 K47 T48 S49 L210 R211 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 15556993 801 VLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 1xz8 B 2.8 BS02 U5P B 1 D104 V106 F108 T109 G110 R111 T112 R137 L160 I161 D86 V88 F90 T91 G92 R93 T94 R119 L142 I143 2.4.2.9 0003723,0004845,0006353,0016757 remove_due_to_license_issue P41007 15716449 400 MQKAVVMDEQAIRRALTRIAHEIIERNKGIDGCVLVGIKTRGIYLARRLAERIEQIEGASVPVGELDITLYRVPFPVTERNVILVDDVLFTGRTVRAAMDAVMDLGRPARIQLAVLVDRGHRELPIRADFVGKNVPTSRSELIVVELSEVDGIDQVSIHEK 1xzx X 2.5 BS01 T3 X 1 F269 F272 I275 I276 A279 R282 M310 M313 R316 L330 L346 H435 M442 F455 F58 F61 I64 I65 A68 R71 M99 M102 R105 L119 L135 H224 M231 F244 ? 0003677,0004879,0006355 Kd=0.06nM remove_due_to_license_issue P10828 15466465 500 HMEELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 1y0l H 2.5 BS01 HAN H 1 E50 L95 Y100D E50 L99 Y108 Kd~1nM remove_due_to_license_issue 15788533 501 EVKLLESGGGLAQPGGSLKLSCAASGFDFRRYWMTWVRQAPGKGLEWIGEINPDSRTINYMPSLKDKFIISRDNAKNSLYLQLSRLRSEDSALYYCVRLDFDVYNHYYVLDYWGQGTSVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 1y0l L 2.5 BS01 HAN H 1 Y32 W91 L96 Y34 W93 L98 remove_due_to_license_issue 15788533 501 ELVVTQESALTTSPGETVTLTCRSSSGAVTTSNYATWVQEKPDHLFTGLIGGTNKRAPGVPARFSGSLIGDRAALTITGAQTEDEAIYFCALWNSNHLVFGGGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 1y0x X 3.1 BS01 T44 X 1 F272 I276 A279 R282 M310 M313 R316 L346 H435 M442 F455 F459 F62 I66 A69 R72 M100 M103 R106 L136 H225 M232 F245 F249 ? 0003677,0004879,0006355 remove_due_to_license_issue EC50=240nM P10828 15466465 500 SHMEELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 1y1m A 1.8 BS01 AC5 A 1 F92 L125 T126 R131 S180 W223 D224 F78 L111 T112 R117 S166 W209 D210 ? 0015276,0016020 Ki=15.3mM remove_due_to_license_issue P35439 15996549 1001 RLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWV 1y1z A 1.5 BS01 192 A 1 F92 L125 T126 R131 S179 S180 W223 D224 F83 L116 T117 R122 S170 S171 W214 D215 ? 0015276,0016020 Ki=0.831mM remove_due_to_license_issue P35439 15996549 293 RLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPNSPRHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQECD 1y20 A 1.4 BS01 1AC A 1 F92 L125 T126 R131 S179 S180 W223 D224 F88 L121 T122 R127 S175 S176 W219 D220 ? 0015276,0016020 Ki=4.8uM remove_due_to_license_issue P35439 15996549 1001 RLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPNDTSPGSPRHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQECD 1y2b A 1.4 BS02 DEE A 1 Y159 T333 I336 Q369 F372 Y74 T248 I251 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=82uM remove_due_to_license_issue IC50=82000nM Q08499 15685167 502 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1y2c A 1.67 BS02 3DE A 1 Y159 M273 W332 T333 I336 Q369 F372 Y74 M188 W247 T248 I251 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=0.27uM remove_due_to_license_issue Q08499 15685167 1003 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1y2d A 1.7 BS02 4DE A 1 M273 T333 M357 F372 M188 T248 M272 F287 3.1.4.53 0004114,0007165,0008081 ic50=2uM remove_due_to_license_issue IC50=2000nM Q08499 15685167 601 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1y2e A 2.1 BS02 5DE A 1 Y159 M273 L319 N321 W332 T333 I336 M357 Q369 F372 Y74 M188 L234 N236 W247 T248 I251 M272 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=0.16uM remove_due_to_license_issue IC50=160nM Q08499 15685167 1003 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1y2f A 2.0 BS01 WAI A 1 M42 A62 T83 F85 M37 A57 T78 F80 ? 0016020,0090529 Kd=12uM remove_due_to_license_issue Ki=12000nM, Kd=12000nM P77173 15743191 300 RKEAVIIMNVAAHHGSELNGELLLNSIQQAGFIFGDMNIYHRHLSPDGSGPALFSLANMVKPGTFDPEMKDFTTPGVTIFMQVPSYGDELQNFKLMLQSAQHIADEVGGVVLDDQRRMMTPQKLREYQDIIREVKDANA 1y2g A 1.9 BS01 CL3 A 1 I12 M42 I44 A62 G68 F85 I7 M37 I39 A57 G63 F80 ? 0016020,0090529 Kd=83.1uM remove_due_to_license_issue Kd=83100nM P77173 15743191 301 RKEAVIIMNVAAHHGSELNGELLLNSIQQAGFIFGDMNIYHRHLSPDGSGPALFSLANMVKPGTFDPEMKDFTTPGVTIFMQVPSYGDELQNFKLMLQSAQHIADEVGGVVLDDQRRMMTPQKLREYQDIIREVKDA 1y2h A 2.4 BS02 6DE A 1 H234 M347 N395 I410 F414 Q443 F446 H72 M185 N233 I248 F252 Q281 F284 3.1.4.53 0004114,0007165,0008081 ic50=0.056uM remove_due_to_license_issue IC50=56nM Q07343 15685167 101 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1y2j A 2.55 BS02 7DE A 1 D392 L393 T407 I410 F414 M431 Q443 F446 D230 L231 T245 I248 F252 M269 Q281 F284 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=33nM Q07343 15685167 101 EDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 1y2k A 1.36 BS02 7DE A 1 Y159 M273 D318 L319 N321 W332 T333 I336 Q369 F372 Y74 M188 D233 L234 N236 W247 T248 I251 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=0.021uM remove_due_to_license_issue IC50=21nM Q08499 15685167 602 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 1y3g E 2.1 BS06 AMM E 1 A113 E143 H146 E166 L202 R203 H231 A113 E143 H146 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 16342943 804 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1y3g E 2.1 BS07 LEU E 1 N112 H231 N112 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 16342943 805 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1y3n A 1.6 BS01 MAV B 1 R20 Y129 W270 R20 Y129 W270 ? 0030313,0046872 remove_due_to_license_issue Q9KWT6 15794643 1 REATWVTEKPLTLKIHMHFRDKWVWDENWPVAREVARLTNVKLVGVANRAATNSQEQFNLMMASGQLPDIVGGDNLKDKFIRYGMEGAFIPLNKLIDQNAPNLKAFFKTHPEVQRAITAPDGNIYYLPYVPDGLVSRGYFIRQDWLDKLHLKTPQTVDELYTVLKAFKEKDPNGNGKADEIPFINRDPEEVFRLVNFWGARSTGSNTWMDFYVENGKIKHPFAEVAFKDGIKHVAQWYKEGLIDPEIFTRKARSREQTFGNNIGGMTHDWFASTALFNDALSKNIPGFKLVPMAPPINSKGQRWEEDARQIPRPDGWAITATNKNPVETIKLFDFYFGPKGRELSNFGVPGLTYDIKNGKPVYKDTVLKAAQPVNNQMYDIGAQIPIGFWQDYEYERQWTNDVALQGIDMYIKNKYVLPQFTGVNLTVEEREIYDKYWPDVKTYMFEMGQSWVMGTKDPEKTWNDYQQQLKNRGFYQVMIVMQKAYDRQY 1y3n A 1.6 BS02 BEM B 1 W270 S273 N375 Y395 E396 W270 S273 N375 Y395 E396 ? 0030313,0046872 remove_due_to_license_issue Q9KWT6 15794643 2 REATWVTEKPLTLKIHMHFRDKWVWDENWPVAREVARLTNVKLVGVANRAATNSQEQFNLMMASGQLPDIVGGDNLKDKFIRYGMEGAFIPLNKLIDQNAPNLKAFFKTHPEVQRAITAPDGNIYYLPYVPDGLVSRGYFIRQDWLDKLHLKTPQTVDELYTVLKAFKEKDPNGNGKADEIPFINRDPEEVFRLVNFWGARSTGSNTWMDFYVENGKIKHPFAEVAFKDGIKHVAQWYKEGLIDPEIFTRKARSREQTFGNNIGGMTHDWFASTALFNDALSKNIPGFKLVPMAPPINSKGQRWEEDARQIPRPDGWAITATNKNPVETIKLFDFYFGPKGRELSNFGVPGLTYDIKNGKPVYKDTVLKAAQPVNNQMYDIGAQIPIGFWQDYEYERQWTNDVALQGIDMYIKNKYVLPQFTGVNLTVEEREIYDKYWPDVKTYMFEMGQSWVMGTKDPEKTWNDYQQQLKNRGFYQVMIVMQKAYDRQY 1y3p A 2.0 BS01 MAV B 1 R20 D21 D74 N75 W208 R20 D21 D74 N75 W208 ? 0030313,0046872 remove_due_to_license_issue Q9KWT6 15794643 1 REATWVTEKPLTLKIHMHFRDKWVWDENWPVAREVARLTNVKLVGVANRAATNSQEQFNLMMASGQLPDIVGGDNLKDKFIRYGMEGAFIPLNKLIDQNAPNLKAFFKTHPEVQRAITAPDGNIYYLPYVPDGLVSRGYFIRQDWLDKLHLKTPQTVDELYTVLKAFKEKDPNGNGKADEIPFINRDPEEVFRLVNFWGARSTGSNTWMDFYVENGKIKHPFAEVAFKDGIKHVAQWYKEGLIDPEIFTRKARSREQTFGNNIGGMTHDWFASTALFNDALSKNIPGFKLVPMAPPINSKGQRWEEDARQIPRPDGWAITATNKNPVETIKLFDFYFGPKGRELSNFGVPGLTYDIKNGKPVYKDTVLKAAQPVNNQMYDIGAQIPIGFWQDYEYERQWTNDVALQGIDMYIKNKYVLPQFTGVNLTVEEREIYDKYWPDVKTYMFEMGQSWVMGTKDPEKTWNDYQQQLKNRGFYQVMIVMQKAYDRQY 1y3p A 2.0 BS02 MAV B 2 R20 Y129 R186 W270 R20 Y129 R186 W270 ? 0030313,0046872 remove_due_to_license_issue Q9KWT6 15794643 3 REATWVTEKPLTLKIHMHFRDKWVWDENWPVAREVARLTNVKLVGVANRAATNSQEQFNLMMASGQLPDIVGGDNLKDKFIRYGMEGAFIPLNKLIDQNAPNLKAFFKTHPEVQRAITAPDGNIYYLPYVPDGLVSRGYFIRQDWLDKLHLKTPQTVDELYTVLKAFKEKDPNGNGKADEIPFINRDPEEVFRLVNFWGARSTGSNTWMDFYVENGKIKHPFAEVAFKDGIKHVAQWYKEGLIDPEIFTRKARSREQTFGNNIGGMTHDWFASTALFNDALSKNIPGFKLVPMAPPINSKGQRWEEDARQIPRPDGWAITATNKNPVETIKLFDFYFGPKGRELSNFGVPGLTYDIKNGKPVYKDTVLKAAQPVNNQMYDIGAQIPIGFWQDYEYERQWTNDVALQGIDMYIKNKYVLPQFTGVNLTVEEREIYDKYWPDVKTYMFEMGQSWVMGTKDPEKTWNDYQQQLKNRGFYQVMIVMQKAYDRQY 1y3p A 2.0 BS03 BEM B 1 W270 S273 N375 Y395 E396 W270 S273 N375 Y395 E396 ? 0030313,0046872 remove_due_to_license_issue Q9KWT6 15794643 4 REATWVTEKPLTLKIHMHFRDKWVWDENWPVAREVARLTNVKLVGVANRAATNSQEQFNLMMASGQLPDIVGGDNLKDKFIRYGMEGAFIPLNKLIDQNAPNLKAFFKTHPEVQRAITAPDGNIYYLPYVPDGLVSRGYFIRQDWLDKLHLKTPQTVDELYTVLKAFKEKDPNGNGKADEIPFINRDPEEVFRLVNFWGARSTGSNTWMDFYVENGKIKHPFAEVAFKDGIKHVAQWYKEGLIDPEIFTRKARSREQTFGNNIGGMTHDWFASTALFNDALSKNIPGFKLVPMAPPINSKGQRWEEDARQIPRPDGWAITATNKNPVETIKLFDFYFGPKGRELSNFGVPGLTYDIKNGKPVYKDTVLKAAQPVNNQMYDIGAQIPIGFWQDYEYERQWTNDVALQGIDMYIKNKYVLPQFTGVNLTVEEREIYDKYWPDVKTYMFEMGQSWVMGTKDPEKTWNDYQQQLKNRGFYQVMIVMQKAYDRQY 1y3v A 1.6 BS02 UIR A 1 H57 N97 T98 L99 D189 S190 Q192 S214 W215 G216 G219 H40 N79 T80 L81 D171 S172 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=2300nM remove_due_to_license_issue P00760 16374786 1994 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1y3w A 1.8 BS02 UIP A 1 N97 L99 D189 S190 Q192 S214 W215 G216 G219 N79 L81 D171 S172 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1680nM remove_due_to_license_issue P00760 16374786 1994 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1y3x A 1.7 BS02 UIB A 1 N97 T98 L99 D189 S190 Q192 S214 W215 G216 G219 N79 T80 L81 D171 S172 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=7315nM remove_due_to_license_issue P00760 16374786 1994 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1y3y A 1.75 BS02 UIR A 1 H57 D189 S190 Q192 S195 S214 W215 G216 G219 H40 D171 S172 Q174 S177 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=2300nM remove_due_to_license_issue P00760 16374786 2222 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1y4z C 2.0 BS03 PCI C 1 G65 H66 G69 K86 A90 M156 G65 H66 G69 K78 A82 M148 1.7.5.1 0005886,0008940,0009055,0009061,0009325,0016020,0016491,0019645,0020037,0042126,0042128,0044799,0046872,0160182 Ki=57nM remove_due_to_license_issue P11350 15615728 1808 MQFLNMFFFDIYPYIAGAVFLIGSWLRYDYGQYTWRAASSQMLDRKGMNLASNLFHIGILGIFVGHFFGMLTLPIEVKQKMAMFAGGASGVLCLIGGVLLLKRRLFSPRVRATTTGADILILSLLVIQCALGLLTIPFSAQHMDGSEMMKLVGWAQSVVTFHGGASQHLDGVAFIFRLHLVLGMTLFLLFPFSRLIHIWSVPVEYLTRKYQLVRARH 1y57 A 1.91 BS01 MPZ A 1 L273 Q275 V281 A293 Y340 M341 G344 L393 L192 Q194 V200 A212 Y259 M260 G263 L312 D386 R388 A390 N391 D404 F424 D305 R307 A309 N310 D323 F343 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1633nM remove_due_to_license_issue IC50=7800nM P12931 15939018 600 MVTTFVALYDYESRTETDLSFKKGERLQIVNNTEGDWWLAHSLSTGQTGYIPSNYVAPSDSIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPTSKPQTQGLAKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGETGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEDNEYTARQGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKEPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 1y69 8 3.33 BS01 rna 0 0 E50 V54 R57 R60 R61 D65 K66 S77 E78 D79 R82 E50 V54 R57 R60 R61 D65 K66 S77 E78 D79 R82 ? 0006412 remove_due_to_license_issue P0A805 15616575 1 ~ 2877 MISDIRKDAEVRMDKCVEAFKTQISKIRTGGGGTEERRKDLTKIVRGEAEQARVAVRNVRRDANDKVKALLKDKEISEDDDRRSQDDVQKLTDAAIKKIEAALADKEAELMQF 1y69 K 3.33 BS01 rna 0 0 R11 K12 Q13 F14 R15 R17 M18 D21 K23 N46 A50 I53 R60 R61 Y66 I67 R68 F70 K78 E81 R83 M84 G85 K86 G87 K88 H124 K125 E140 A141 R6 K7 Q8 F9 R10 R12 M13 D16 K18 N41 A45 I48 R55 R56 Y61 I62 R63 F65 K73 E76 R78 M79 G80 K81 G82 K83 H119 K120 E135 A136 ? 0000049,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue Q9RXJ5 15616575 1 ~ 2877 KRTKFRKQFRGRMTGDAKGGDYVAFGDYGLIAMEPAWIKSNQIEACRIVMSRHFRRGGKIYIRIFPDKPVTKKPAETRMGKGKGAVEYWVSVVKPGRVMFEVAGVTEEQAKEAFRLAGHKLPIQTKMVKREVYDEA 1y69 K 3.33 BS02 rna 9 0 T19 D21 E39 P40 K99 T14 D16 E34 P35 K94 ? 0000049,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue Q9RXJ5 15616575 4 ~ 121 KRTKFRKQFRGRMTGDAKGGDYVAFGDYGLIAMEPAWIKSNQIEACRIVMSRHFRRGGKIYIRIFPDKPVTKKPAETRMGKGKGAVEYWVSVVKPGRVMFEVAGVTEEQAKEAFRLAGHKLPIQTKMVKREVYDEA 1y69 U 3.33 BS01 rna 0 0 G13 N17 P18 K19 Y20 V23 K24 F26 G27 E29 K32 A33 G34 I36 R39 R41 G42 T43 K44 F45 G54 R55 D56 T58 F60 F69 G12 N16 P17 K18 Y19 V22 K23 F25 G26 E28 K31 A32 G33 I35 R38 R40 G41 T42 K43 F44 G53 R54 D55 T57 F59 F68 ? 0000049,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue Q9RY65 15616575 1 ~ 2877 AHKKGVGSSKNGRDSNPKYLGVKKFGGEVVKAGNILVRQRGTKFKAGQGVGMGRDHTLFALSDGKVVFINKGKGARFISIEAAQ 1y6a A 2.1 BS01 AAZ A 1 L838 V846 F916 C917 G920 N921 L1033 F1045 L21 V25 F91 C92 G95 N96 L149 F161 D1026 R1030 N1031 D1044 D142 R146 N147 D160 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=0.022uM remove_due_to_license_issue IC50=22nM P35968 15743202 201 LPYDASKWEFPRDRLKLGKPLGRQVIEADAFGIDKTATCRTVAVKMLTHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQAN 1y6b A 2.1 BS01 AAX A 1 L838 V846 A864 K866 E883 V912 V914 F916 C917 G920 N921 L1033 F1045 L22 V28 A46 K48 E63 V92 V94 F96 C97 G100 N101 L153 F165 D1026 R1030 N1031 D1044 D146 R150 N151 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=38nM remove_due_to_license_issue IC50=38nM P35968 15743202 201 RLPYDASKWEFPRDRLKLGKPLGRGGQVIEADAFGIDKTATCRTVAVKMLKATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 1y6q A 2.2 BS01 TDI A 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I52 S78 A79 G80 F153 I154 E174 M175 E176 D199 F209 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=2pM remove_due_to_license_issue Kd=0.002nM, Ki=0.048nM P0AF12 15746096 233 FSMKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1y6q B 2.2 BS01 TDI B 1 I50 S76 A77 G78 F151 I152 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 M173 E174 D197 F207 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=2pM remove_due_to_license_issue Kd=0.002nM, Ki=0.048nM P0AF12 15746096 234 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1y6r A 2.2 BS01 MTM A 1 I50 S76 A77 F151 I152 E172 M173 E174 D197 F207 I52 S78 A79 F153 I154 E174 M175 E176 D199 F209 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=77pM remove_due_to_license_issue P0AF12 15746096 233 FSMKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1y6r B 2.2 BS01 MTM B 1 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=77pM remove_due_to_license_issue P0AF12 15746096 234 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 1y8o A 2.48 BS01 ADP A 1 N251 R254 A255 V292 L300 G325 L328 N239 R242 A243 V280 L288 G298 L301 H243 E247 K250 N251 H231 E235 K238 N239 2.7.11.2 0004672,0004674,0004740,0005515,0005524,0005730,0005739,0005759,0010510,0010906,0016301,0018105,0035357,0071333,0071398,0097411,2000377 Kd=1.3uM remove_due_to_license_issue Q15120 15861126 504 PKQIERYSRFSPSPLSIKQFLDFGRDNACEKTSYMFLRKELPVRLANTMREVNLLPDNLLNRPSVGLVQSWYMQSFLELLEYENKSPEDPQVLDNFLQVLIKVRNRHNDVVPTMAQGVIEYKEKFGFDPFISTNIQYFLDRFYTNRISFRMLINQHTLLFGGDTNPVHPKHIGSIDPTCNVADVVKDAYETAKMLCEQYYLVAPELEVEEFNAKAPDKPIQVVYVPSHLFHMLFELFKNSMRATVELYEDRKEGYPAVKTLVTLGKEDLSIKISDLGGGVPLRKIDRLFNYMYSPLFGYGLPISRLYARYFQGDLKLYSMEGVGTDAVIYLKALSSESFERLPVFNKSAWRHYKTTPEADDWSNPSSEPRDASK 1y8p A 2.63 BS01 ATP A 1 E247 N251 A255 V292 S306 T307 A322 F324 G325 G327 L328 E236 N240 A244 V281 S295 T296 A302 F304 G305 G307 L308 H243 E247 K250 N251 H232 E236 K239 N240 2.7.11.2 0004672,0004674,0004740,0005515,0005524,0005730,0005739,0005759,0010510,0010906,0016301,0018105,0035357,0071333,0071398,0097411,2000377 remove_due_to_license_issue Q15120 15861126 504 VPKQIERYSRFSPSPLSIKQFLDFGRDNACEKTSYMFLRKELPVRLANTMREVNLLPDNLLNRPSVGLVQSWYMQSFLELLEYENKSPEDPQVLDNFLQVLIKVRNRHNDVVPTMAQGVIEYKEKFGFDPFISTNIQYFLDRFYTNRISFRMLINQHTLLFGGDTNPVHPKHIGSIDPTCNVADVVKDAYETAKMLCEQYYLVAPELEVEEFNAKAPDKPIQVVYVPSHLFHMLFELFKNSMRATVELYEDRKEGYPAVKTLVTLGKEDLSIKISDLGGGVPLRKIDRLFNYMYSTAPRPLAGFGYGLPISRLYARYFQGDLKLYSMEGVGTDAVIYLKALSSESFERLPVFNKSAWRHYKTTPEADDWSNPSSEPRDASK 1y91 A 2.15 BS01 CT9 A 1 I10 V18 A31 F80 L83 H84 Q85 K89 N132 L134 D145 I10 V18 A31 F73 L76 H77 Q78 K82 N125 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T153 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.059uM remove_due_to_license_issue IC50=59nM P24941 15686876 401 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1ya4 A 3.2 BS02 CTX A 1 F101 S221 L304 S305 L318 L363 M364 L388 H468 F80 S200 L283 S284 L297 L341 M342 L366 H446 G142 G143 G173 S221 A222 L319 E354 H468 G121 G122 G152 S200 A201 L298 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 remove_due_to_license_issue P23141 16081098 1 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1ya4 A 3.2 BS03 CTX A 2 W357 P360 M361 L368 S369 G371 K414 W336 P339 M340 L346 S347 G349 K392 G142 G143 G173 S221 A222 L319 E354 H468 G121 G122 G152 S200 A201 L298 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 remove_due_to_license_issue P23141 16081098 11 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1ybg A 2.6 BS01 TAV A 1 K22 N23 L26 R91 A92 I94 W95 P121 H125 G164 F328 K22 N23 L26 R91 A92 I94 W95 P121 H125 G164 F328 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 15701635 550 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 1ybg D 2.6 BS01 TAV D 1 K22 N23 R91 A92 I94 W95 P121 H125 V163 G164 F328 K22 N23 R91 A92 I94 W95 P121 H125 V163 G164 F328 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 15701635 850 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 1yc1 A 1.7 BS01 4BC A 1 N51 A55 K58 D93 I96 G97 M98 F138 T184 N37 A41 K44 D79 I82 G83 M84 F124 T170 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.68uM remove_due_to_license_issue Kd=680nM P07900 15713410 401 EEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 1yc4 A 1.81 BS01 43P A 1 N51 A55 K58 D93 I96 G97 M98 F138 T184 N37 A41 K44 D79 I82 G83 M84 F124 T170 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.28uM remove_due_to_license_issue Kd=280nM P07900 15713410 301 EEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 1yc5 A 1.4 BS03 NCA A 1 P31 F33 N99 I100 D101 P31 F33 N88 I89 D90 P31 D32 F33 N99 D101 H116 P31 D32 F33 N88 D90 H105 2.3.1.286 0005737,0008270,0016740,0017136,0032041,0034979,0046872,0046969,0046970,0051287,0070403,0097372,0140765,0141222 ic50=1mM remove_due_to_license_issue Q9WYW0 15780941 2001 MKMKEFLDLLNESRLTVTLTGAGISTPSGIPDFQNVFDIDFFYSHPEEFYRFAKEGIFPMLQAKPNLAHVLLAKLEEKGLIEAVITQNIDRLHQRAGSKKVIELHGNVEEYYCVRCEKKYTVEDVIKKLESSDVPLCDDCNSLIRPNIVFFGENLPQDALREAIGLSSRASLMIVLGSSLVVYPAAELPLITVRSGGKLVIVNLGETPFDDIATLKYNMDVVEFARRVMEEGGI 1yci A 2.7 BS02 NDF A 1 Y145 L188 T196 H199 N205 F207 K214 I281 Y132 L175 T183 H186 N192 F194 K201 I268 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 remove_due_to_license_issue Kd=83000nM Q9NWT6 15913349 400 GEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 1yci A 2.7 BS03 NDF A 2 D222 F224 E225 K315 M319 D209 F211 E212 K302 M306 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 remove_due_to_license_issue Kd=83000nM Q9NWT6 15913349 401 GEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 1ycm A -1.00 BS06 NGH A 1 L181 A182 T215 H218 E219 P238 T239 Y240 L77 A78 T111 H114 E115 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=4.3nM P39900 15809432 269 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 1yda A 2.1 BS02 AZM A 1 Q92 H94 H119 V121 F131 E198 T199 T200 Q88 H90 H115 V117 F126 E193 T194 T195 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=280nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 7696263 264 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSETTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1ydb A 1.9 BS02 AZM A 1 Q92 H94 F198 T199 T200 Q88 H90 F193 T194 T195 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=5.8nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 7696263 264 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSFTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1ydd A 2.1 BS02 AZM A 1 H94 H119 V121 F131 R198 T199 T200 H91 H116 V118 F127 R194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=86nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 7696263 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSRTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1ydk A 1.95 BS01 GTX A 1 R15 R45 Q54 V55 Q67 T68 L107 R13 R43 Q52 V53 Q65 T66 L105 Y9 R15 R20 Y7 R13 R18 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM remove_due_to_license_issue P08263 15893769 5100 EKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMD 1ydk A 1.95 BS02 GTX B 1 D101 R131 D99 R129 Y9 R15 R20 Y7 R13 R18 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM remove_due_to_license_issue P08263 15893769 5200 EKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMD 1ydk B 1.95 BS01 GTX A 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM remove_due_to_license_issue P08263 15893769 5100 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKAFRF 1ydk B 1.95 BS02 GTX B 1 R15 Q54 V55 Q67 T68 L107 F220 R12 Q51 V52 Q64 T65 L104 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM remove_due_to_license_issue P08263 15893769 5200 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKAFRF 1ydr E 2.2 BS02 IQP E 1 G50 V57 A70 Y122 V123 E170 L173 T183 F327 G36 V43 A56 Y108 V109 E156 L159 T169 F313 N171 D184 N157 D170 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=3uM remove_due_to_license_issue P00517 8824261 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1yds E 2.2 BS02 IQS E 1 L49 V57 A70 M120 Y122 V123 L173 T183 D184 F327 L35 V43 A56 M106 Y108 V109 L159 T169 D170 F313 N171 D184 N157 D170 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=1.2uM remove_due_to_license_issue IC50=5300nM P00517 8824261 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1ydt E 2.3 BS02 IQB E 1 L49 T51 G52 G55 V57 A70 Y122 V123 E170 L173 T183 F327 L35 T37 G38 G41 V43 A56 Y108 V109 E156 L159 T169 F313 N171 D184 N157 D170 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=48nM remove_due_to_license_issue IC50=73nM P00517 8824261 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1yei H 1.9 BS01 PGG L 1 H35 W95 F97 Y100D H35 W99 F101 Y108 remove_due_to_license_issue 9826512 551 EMQLQQSGAELLRPGTSVKLSCKTSGYIFTSYWIHWVKQRSGQGLEWIARIYPGTGSTYYNEKFKGKATLTADKSSSTAYMQLSTLKSEDSAVYFCTRWGFIPVREDYVMDYWGQGTLVTVSSAKTTAPSVYPLAPVCGDTTGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEP 1yei L 1.9 BS02 PGG L 1 Y27D Y32 G91 Y96 F98 Y31 Y37 G96 Y101 F103 ? 0046872 Kd=35nM remove_due_to_license_issue Q58EU8 9826512 551 DIVMTQSPLTLSVTIGQPASISCKSSQSLLYSNGKTYLNWLLQRPGQSPKRLIHLVSKLDSGVPDRITGSGSGTDFTLKISRVEAADLGVYYCVQGTHFPYTFGGGTKLEILRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 1yej H 1.85 BS01 PNF L 1 H35 W95 Y100D H35 W99 Y108 remove_due_to_license_issue 9826512 551 EMQLQQSGAELLRPGTSVKLSCKTSGYIFTSYWIHWVKQRSGQGLEWIARIYPGTGSTYYNEKFKGKATLTADKSSSTAYMQLSTLKSEDSAVYFCTRWGFIPVREDYVMDYWGQGTLVTVSSAKTTAPSVYPLAPVCGDTTGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEP 1yej L 1.85 BS03 PNF L 1 G91 T92 H93 F94 Y96 F98 G96 T97 H98 F99 Y101 F103 ? 0046872 Kd=35nM remove_due_to_license_issue Q58EU8 9826512 551 DIVMTQSPLTLSVTIGQPASISCKSSQSLLYSNGKTYLNWLLQRPGQSPKRLIHLVSKLDSGVPDRITGSGSGTDFTLKISRVEAADLGVYYCVQGTHFPYTFGGGTKLEILRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 1yet A 1.9 BS01 GDM A 1 N51 D54 A55 K58 M98 D102 N106 L107 K112 G135 V136 F138 N41 D44 A45 K48 M88 D92 N96 L97 K102 G125 V126 F128 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=42nM, Kd=714nM P07900 9108479 275 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 1yfh A 3.01 BS01 dna F 0 Y114 Q115 A127 R128 G131 M134 R135 N137 P140 C145 S151 Y158 S159 G160 Y100 Q101 A113 R114 G117 M120 R121 N123 P126 C131 S137 Y144 S145 G146 2.1.1.63 0003824,0003908,0006281 remove_due_to_license_issue P16455 15964013 1 ~ 16 CEMKRTTLDSPLGKLELSGCEQGLHEIKLLGVPAPAAVLGGPEPLMQCTAWLNAYFHQPEAIEEFPVPALHHPVFQQESFTRQVLWKLLKVVKFGEVISYQQLAALAGNPKAARAVGGAMRGNPVPILIPCHRVVCSSGAVGNYSGGLAVKEWLLAHEGHRLGKP 1yfh A 3.01 BS02 dna G 0 F94 T95 R128 A129 F80 T81 R114 A115 2.1.1.63 0003824,0003908,0006281 remove_due_to_license_issue P16455 15964013 15 ~ -1 CEMKRTTLDSPLGKLELSGCEQGLHEIKLLGVPAPAAVLGGPEPLMQCTAWLNAYFHQPEAIEEFPVPALHHPVFQQESFTRQVLWKLLKVVKFGEVISYQQLAALAGNPKAARAVGGAMRGNPVPILIPCHRVVCSSGAVGNYSGGLAVKEWLLAHEGHRLGKP 1yfh B 3.01 BS01 dna F 0 Y114 R128 G131 R135 S159 Y100 R114 G117 R121 S145 2.1.1.63 0003824,0003908,0006281 remove_due_to_license_issue P16455 15964013 1 ~ 16 CEMKRTTLDSPLGKLELSGCEQGLHEIKLLGVPAPAAVLGGPEPLMQCTAWLNAYFHQPEAIEEFPVPALHHPVFQQESFTRQVLWKLLKVVKFGEVISYQQLAALAGNPKAARAVGGAMRGNPVPILIPCHRVVCSSGAVGNYSGGLAVKEWLLAHEGHR 1yfh B 3.01 BS02 dna G 0 F94 N123 K125 A129 F80 N109 K111 A115 2.1.1.63 0003824,0003908,0006281 remove_due_to_license_issue P16455 15964013 15 ~ -1 CEMKRTTLDSPLGKLELSGCEQGLHEIKLLGVPAPAAVLGGPEPLMQCTAWLNAYFHQPEAIEEFPVPALHHPVFQQESFTRQVLWKLLKVVKFGEVISYQQLAALAGNPKAARAVGGAMRGNPVPILIPCHRVVCSSGAVGNYSGGLAVKEWLLAHEGHR 1yfh C 3.01 BS01 dna D 0 Y114 Q115 A127 R128 G131 M134 R135 P140 C150 S151 Y91 Q92 A104 R105 G108 M111 R112 P117 C127 S128 2.1.1.63 0003824,0003908,0006281 remove_due_to_license_issue P16455 15964013 1 ~ 16 CEMKRTTLDSPLGKLELSGCEQGLHEIKLLGGPEPLMQCTAWLNAYFHQPEAIEEFPVPALHHPVFQQESFTRQVLWKLLKVVKFGEVISYQQLAALAGNPKAARAVGGAMRGNPVPILIPCHRVVCSSGAVGLAVKEWLLAHEGHRLG 1yfh C 3.01 BS02 dna E 0 F94 T95 K125 R128 F71 T72 K102 R105 2.1.1.63 0003824,0003908,0006281 remove_due_to_license_issue P16455 15964013 15 ~ -1 CEMKRTTLDSPLGKLELSGCEQGLHEIKLLGGPEPLMQCTAWLNAYFHQPEAIEEFPVPALHHPVFQQESFTRQVLWKLLKVVKFGEVISYQQLAALAGNPKAARAVGGAMRGNPVPILIPCHRVVCSSGAVGLAVKEWLLAHEGHRLG 1yfz A 2.2 BS02 IMP A 1 K45 G46 F154 V155 D161 R167 K43 G44 F152 V153 D159 R165 E101 D102 D105 F154 R167 E99 D100 D103 F152 R165 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0046100,0046872,0052657 Ki=45uM remove_due_to_license_issue Q8R7L0 15854655 1210 SPMEDIEEILITEEQLKAKVKELGEMITRDYEGKDLVLIGVLKGAIMFMSGLSRAIDLPLSIDFLAVSSYGSSTKSSGIVKIIKDHDIDIEGKDVLIVEDIIDSGLTLAYLRETLLGRKPRSLKICTILDKPERREADVKVDYCGFKIPDKFVVGYGLDYAEKYRNLPFIGVLKPELY 1yhm A 2.5 BS03 AHD A 1 D98 R107 K207 D250 K264 D98 R107 K207 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.10 0004659,0008299,0016765 ic50=147uM remove_due_to_license_issue Q8WS26 16288456 901 MASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKRKK 1yhs A 2.15 BS01 STU A 1 L44 G45 F49 V52 A65 L120 E121 R122 V126 D128 E171 L174 I185 D186 L12 G13 F17 V20 A33 L84 E85 R86 V90 D92 E135 L138 I149 D150 D167 K169 N172 D186 L193 T204 D131 K133 N136 D150 L157 T168 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.01uM remove_due_to_license_issue P11309 15657054 306 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGETRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 1yi3 A 2.5 BS01 LY2 A 1 L44 F49 V52 A65 I104 L120 E121 R122 L174 L12 F17 V20 A33 I68 L84 E85 R86 L138 D167 K169 N172 D186 L193 T204 D131 K133 N136 D150 L157 T168 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=4uM remove_due_to_license_issue IC50=820nM P11309 15657054 306 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGETRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 1yid B 2.4 BS01 ATP B 1 D29 R30 H39 R206 L207 M216 S217 S219 D9 R10 H19 R186 L187 M196 S197 S199 E133 K215 K218 E113 K195 K198 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0006412,0006418,0006436 Kd=10uM remove_due_to_license_issue Q9RVD6 15998643 3000 ARPRVLTGDRPTGALHLGHLAGSLQNRVRLQDEAELFVLLADVQALTDHFDRPEQVRENVLAVALDYLAAGLDPQKTTCVVQSAVPELAELTVYFLNLVTVSHLRQNPTVKAEIAQKGYGERVPAGFFVYPVSQAADIAAFGATLVPVGDDQLPMLEQTREIVRRFNALYAPVLAEPQAQLSRVPRLPGLDGQAKMSKSLGNAIALGDSADEVARKVMGMYTDPGHLRASDPGRVEGNPVFTFLDAFDPDPARVQALKDQYRAGGLGDVKVKKHLIDVLNGVLAPIRTRRAEYERDPDAVLRFVTEGTARGREVAAQTLGQVRRAMRLFGH 1yk7 A 2.5 BS01 NBL A 1 G23 C25 E59 G65 G66 Y67 L160 N161 G23 C25 E59 G65 G66 Y67 L160 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 15780613 216 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1ykr A 1.8 BS01 628 A 1 V18 A31 K33 V64 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 V18 A31 K33 V64 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.56uM remove_due_to_license_issue IC50=560nM P24941 15780638 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 1ylv A 2.15 BS02 SHF A 1 K210 Y216 F219 K263 Y287 S290 K210 Y216 F219 K263 Y287 S290 K210 K263 K210 K263 4.2.1.24 0004655,0005634,0005737,0005829,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue P05373 10386874 363 MHTAEFLETEPTEISSVLAGGYNHPLLRQWQSERQLTKNMLIFPLFISDNPDDFTEIDSLPNINRIGVNRLKDYLKPLVAKGLRSVILFGVPLIPGTKDPVGTAADDPAGPVIQGIKFIREKFPELYIICDVCLCEYTSHGHCGVLYDDGTINRERSVSRLAAVAVNYAKAGAHCVAPSDMIDGRIRDIKRGLINANLAHKTFVLSYAAKFSGNLYGPFRDAACSAPSNGDRKCYQLPPAGRGLARRALERDMSEGADGIIVKPSTFYLDIMRDASEICKDLPICAYHVSGEYAMLHAAAEKGVVDLKTIAFESHTGFLRAGARLIITYLAPEFLDWLDEE 1yly A 1.25 BS01 CB4 A 1 S70 Y105 S130 N132 G236 S237 G238 D240 S45 Y80 S105 N107 G211 S212 G213 D214 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677,0046872 remove_due_to_license_issue Q9L5C7 15826180 2001 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 1ym1 A 1.12 BS01 SM2 A 1 C69 S70 N104 Y105 S130 N132 E166 N170 T235 S237 G238 D240 C44 S45 N79 Y80 S105 N107 E141 N145 T210 S212 G213 D214 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9L5C8 15826180 2001 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 1yms A 1.6 BS01 NBF A 1 S70 N104 Y105 S130 N132 N170 G236 S237 G238 D240 S45 N79 Y80 S105 N107 N145 G211 S212 G213 D214 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9L5C8 15826180 1001 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 1ynd A 1.6 BS01 SFA A 1 R55 G59 F60 Q63 T73 A101 N102 Q111 F113 W121 H126 R54 G58 F59 Q62 T72 A100 N101 Q110 F112 W120 H125 R55 F60 Q63 N102 F113 L122 H126 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 ic50=3.6nM remove_due_to_license_issue IC50=1.000000nM, Kd=3.3nM P62937 15772070 401 VNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 1yon A 1.95 BS01 A2R A 1 G9 A10 L11 L71 K72 H97 N98 T118 S244 R253 E256 G9 A10 L11 L71 K72 H97 N98 T118 S244 R253 E256 K176 K176 1.1.1.169 0005737,0008677,0015940,0016491,0016616,0050661 Kd=61uM remove_due_to_license_issue P0A9J4 17242510 501 MKITVLGCGALGQLWLTALCKQGHEVQGWLRVPQPYCSVNLVETDGSIFNESLTANDPDFLATSDLLLVTLKAWQVSDAVKSLASTLPVTTPILLIHNGMGTIEELQNIQQPLLMGTTTHAARRDGNVIIHVANGITHIGPARQQDGDYSYLADILQTVLPDVAWHNNIRAELWRKLAVNCVINPLTAIWNCPNGELRHHPQEIMQICEEVAAVIEREGHHTSAEDLRDYVMQVIDATAENISSMLQDIRALRHTEIDYINGFLLRRARAHGIAVPENTRLFEMVKRKESEY 1you A 2.3 BS04 PFD A 1 L184 A186 H222 E223 H232 L239 F241 I243 Y244 L81 A83 H119 E120 H129 L136 F138 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.87nM remove_due_to_license_issue IC50=0.6nM P45452 15780611 998 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDE 1yp9 A 2.1 BS02 UIZ A 1 H57 T98 L99 D189 S190 Q192 S214 W215 G216 G219 H40 T80 L81 D171 S172 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=7700nM remove_due_to_license_issue P00760 16374786 2222 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1ype H 1.81 BS03 UIP H 1 H57 Y60A E97A N98 L99 D189 A190 E192 W215 G216 G219 H43 Y47 E94 N95 L96 D192 A193 E195 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=8nM remove_due_to_license_issue P00734 16374786 5555 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1ypg H 1.8 BS03 UIR H 1 H57 Y60A E97A N98 D189 A190 W215 G216 G219 H43 Y47 E94 N95 D193 A194 W221 G222 G224 3.4.21.5 0004252,0005509,0006508,0007596 Ki=10nM remove_due_to_license_issue P00734 16374786 5555 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1ypj H 1.78 BS03 UIB H 1 H57 Y60A W60D E97A N98 L99 D189 A190 E192 S195 S214 W215 G216 G219 H43 Y47 W50 E94 N95 L96 D193 A194 E196 S199 S220 W221 G222 G224 3.4.21.5 0004252,0005509,0006508,0007596 Ki=95nM remove_due_to_license_issue P00734 16374786 5555 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1yq7 A 2.2 BS03 RIS A 1 D117 R126 Q185 K214 T215 Q254 D257 K271 D88 R97 Q156 K185 T186 Q225 D228 K242 K71 F112 D117 D121 R126 D188 K214 F253 D257 D258 K42 F83 D88 D92 R97 D159 K185 F224 D228 D229 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=11nM, Ki=82.2nM P14324 901 EKQDFVQHFSQIVRVLTEDEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 1yqj A 2.0 BS01 6NP A 1 Y35 V38 A51 K53 I84 L104 V105 T106 M109 A111 D112 S154 Y39 V42 A55 K57 I88 L108 V109 T110 M113 A115 D116 S158 D150 K152 N155 D168 T185 D154 K156 N159 D172 T189 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=7.3nM remove_due_to_license_issue Q16539 15837335 362 HMLEMSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1yqy A 2.3 BS02 915 A 1 D328 S655 K656 G657 L677 H686 E687 H690 Y728 E735 E739 D64 S391 K392 G393 L413 H422 E423 H426 Y464 E471 E475 H686 E687 H690 Y728 E735 H422 E423 H426 Y464 E471 3.4.24.83 0008237 Ki=24nM remove_due_to_license_issue Ki=24nM, IC50=54nM P15917 15911756 782 LSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEEEKELLNRIQVDSSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINSLV 1yrs A 2.5 BS02 L47 A 1 E116 E118 R119 W127 D130 A133 I136 P137 L214 R221 F239 E99 E101 R102 W110 D113 A116 I119 P120 L197 R204 F222 ? 0003777,0005524,0007018,0008017 ic50=450nM remove_due_to_license_issue IC50=450nM P52732 15808464 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 1ysg A -1.00 BS01 4FC A 1 F101 Y105 A108 F109 L134 G142 R143 A146 F61 Y65 A68 F69 L94 G102 R103 A106 ? 0042981 remove_due_to_license_issue Kd=300000nM, EC50=>31500nM, IC50=>99200nM Q07817 15902208 1000 MSMAMSQSNRELVVDFLSYKLSQKGYSWSQFSDVEENRTEAPEGTESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGNNAAAESRKGQERLEHHHHHH 1ysi A -1.00 BS01 N3B A 1 F101 Y105 A108 L134 G142 V145 Y199 F61 Y65 A68 L94 G102 V105 Y159 ? 0042981 remove_due_to_license_issue IC50=>10000nM, Ki=36nM, Kd=1900nM Q07817 15902208 1000 MSMAMSQSNRELVVDFLSYKLSQKGYSWSQFSDVEENRTEAPEGTESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGNNAAAESRKGQERLEHHHHHH 1yt7 A 2.3 BS01 3FC A 1 Q19 G20 Q21 G23 C25 D61 G64 G65 G66 Y67 N161 H162 A163 W184 Q18 G19 Q20 G22 C24 D60 G63 G64 G65 Y66 N160 H161 A162 W183 Q19 C25 H162 N182 Q18 C24 H161 N181 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=130nM P43235 15982880 301 PDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 1yt9 A 3.0 BS01 OIS A 1 R8 D25 G27 D29 D30 I47 P81 V82 R8 D25 G27 D29 D30 I47 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15837308 1000 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1yt9 B 3.0 BS01 OIS A 1 D25 G27 A28 D29 G48 G49 I84 D25 G27 A28 D29 G48 G49 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 15837308 1000 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ytf A 2.5 BS01 dna E 0 V71 F116 S118 K120 Q158 N159 L189 F190 R196 T215 V11 F56 S58 K60 Q98 N99 L129 F130 R136 T155 ? 0003677,0006352 remove_due_to_license_issue P13393 8610010 1 ~ 16 SGIVPTLQNIVATVTLGCRLDLKTVALHARNAEYNPKRFAAVIMRIREPKTTALIFASGKMVVTGAKSEDDSKLASRKYARIIQKIGFAAKFTDFKIQNIVGSCDVKFPIRLEGLAFSHGTFSSYEPELFPGLIYRMVKPKIVLLIFVSGKIVLTGAKQREEIYQAFEAIYPVLSEFRKM 1ytf A 2.5 BS02 dna F 0 Q68 N69 R98 F99 I103 R105 T112 T124 F190 P191 F207 S209 K211 V213 Q8 N9 R38 F39 I43 R45 T52 T64 F130 P131 F147 S149 K151 V153 ? 0003677,0006352 remove_due_to_license_issue P13393 8610010 1 ~ 16 SGIVPTLQNIVATVTLGCRLDLKTVALHARNAEYNPKRFAAVIMRIREPKTTALIFASGKMVVTGAKSEDDSKLASRKYARIIQKIGFAAKFTDFKIQNIVGSCDVKFPIRLEGLAFSHGTFSSYEPELFPGLIYRMVKPKIVLLIFVSGKIVLTGAKQREEIYQAFEAIYPVLSEFRKM 1ytf C 2.5 BS01 dna E 0 R257 K259 R17 K19 ? 0005672,0006367 remove_due_to_license_issue P32773 8610010 1 ~ 16 ENLMLCLYDKVTRTKARWKCSLKDGVVTINRNDYTFQKAQVEAEWV 1ytu A 2.5 BS01 rna C 0 Y118 N119 T120 Y123 K127 Q137 F138 M139 R140 R147 Y152 N155 Q159 K163 R380 R383 R385 N386 L427 Y117 N118 T119 Y122 K126 Q136 F137 M138 R139 R146 Y151 N154 Q158 K162 R363 R366 R368 N369 L410 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 15800629 1 ~ 5 MEYKIVENGLTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDILSNRNLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGDPYEGTKVKLSSKRYLLTLLQPYPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPINPEGNRSLQTNPWFL 1ytu A 2.5 BS02 rna D 0 F151 R383 F150 R366 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 15800629 15 ~ 18 MEYKIVENGLTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDILSNRNLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGDPYEGTKVKLSSKRYLLTLLQPYPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPINPEGNRSLQTNPWFL 1ytu B 2.5 BS01 rna E 0 Y118 N119 T120 Y123 K127 Q137 F138 M139 R140 I143 R147 Y152 N155 Q159 K163 R380 R385 L427 Y118 N119 T120 Y123 K127 Q137 F138 M139 R140 I143 R147 Y152 N155 Q159 K163 R380 R385 L427 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 15800629 1 ~ 6 MMEYKIVENGLTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDILSNRNLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGDPNNRFHPYEGTKVKLSSKRYLLTLLQPYLKRNGLEMVTPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPINPEGNRSLQTNPWFL 1ytu B 2.5 BS02 rna F 0 F151 R334 R383 F151 R334 R383 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 15800629 15 ~ 18 MMEYKIVENGLTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDILSNRNLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGDPNNRFHPYEGTKVKLSSKRYLLTLLQPYLKRNGLEMVTPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPINPEGNRSLQTNPWFL 1yvf A 2.5 BS01 PH7 A 1 F193 P197 R200 N316 C366 S368 L384 M414 Y448 F194 P198 R201 N317 C367 S369 L385 M415 Y449 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.1uM remove_due_to_license_issue O93077 15863301 800 MSMSYTWTGALITPCAAEESKLPINALSNSLLRHHNLVYSTTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRSLSSRAVNHIRSVWKDLLEDTDTPIQTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKAKKCPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYVGGPMTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTVPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRAKLLSQGGRAAICGKYLFNWAVRTKLKLTPIPAASRLLLSGWFVAGYSGGDIYHS 1yvm A 1.6 BS03 TMG A 1 C59 Y62 Y65 C70 H79 H178 C58 Y61 Y64 C69 H78 H177 H79 D97 D108 H171 Q175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 Q174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 Ki=0.4uM remove_due_to_license_issue IC50=472nM P0AE18 15880695 501 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGQGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 1yvp A 2.2 BS01 rna C 0 K108 Q109 K133 G142 W144 G145 R146 A147 R149 W177 D181 R184 L185 H187 K104 Q105 K129 G138 W140 G141 R142 A143 R145 W173 D177 R180 L181 H183 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 15907467 1 ~ 10 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKEGMKCGMWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 1yvp A 2.2 BS02 rna D 0 R146 R149 H187 I188 K189 P190 A199 K200 S203 K204 R142 R145 H183 I184 K185 P186 A195 K196 S199 K200 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 15907467 1 ~ 10 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKEGMKCGMWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 1yvp A 2.2 BS03 rna G 0 R120 I121 T123 K170 Y171 R174 R252 V254 R255 E256 P277 T279 A280 R283 L313 K316 R318 R116 I117 T119 K166 Y167 R170 R248 V250 R251 E252 P273 T275 A276 R279 L309 K312 R314 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 15907467 6 ~ 10 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKEGMKCGMWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 1yvp B 2.2 BS01 rna E 0 K108 Q109 K133 G142 W144 G145 R146 A147 R149 W177 D181 R184 L185 H187 K105 Q106 K130 G139 W141 G142 R143 A144 R146 W174 D178 R181 L182 H184 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 15907467 1 ~ 10 TMDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKEGMKCGMWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 1yvp B 2.2 BS02 rna F 0 R146 R149 H187 I188 K189 P190 K200 S203 K204 R143 R146 H184 I185 K186 P187 K197 S200 K201 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 15907467 1 ~ 10 TMDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKEGMKCGMWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 1yvp B 2.2 BS03 rna H 0 R120 I121 T123 M166 K170 Y171 R174 R252 R255 E256 D275 P277 L278 T279 A280 R283 K316 A317 R318 R117 I118 T120 M163 K167 Y168 R171 R249 R252 E253 D272 P274 L275 T276 A277 R280 K313 A314 R315 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 15907467 4 ~ 10 TMDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKEGMKCGMWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 1yvx A 2.0 BS01 IPC A 1 R422 M423 L474 H475 T476 Y477 L497 R498 W528 R422 M423 L474 H475 T476 Y477 L497 R498 W528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=8uM remove_due_to_license_issue P26660 15746101 580 SMSYSWTGALITPCSPEEEKLPINPLSNSLLRYHNKVYCTTSKSASLRAKKVTFDRMQVLDAYYDSVLKDIKLAASKVSARLLTLEEACQLTPPHSARSKYGFGAKEVRSLSGRAVNHIKSVWKDLLEDSQTPIPTTIMAKNEVFCVDPTKGGKKAARLIVYPDLGVRVCEKMALYDVTQKLPQAVMGASYGFQYSPAQRVEFLLKAWAEKKDPMGFSYDTRCFDSTVTERDIRTEESIYQACSLPEEARTAIHSLTERLYVGGPMFNSKGQSCGYRRCRASGVLTTSMGNTITCYVKALAACKAAGIVAPTMLVCGDDLVVISESQGTEEDERNLRAFTEAMTRYSAPPGDPPRPEYDLELITSCSSNVSVALGPQGRRRYYLTRDPTTPIARAAWETVRHSPVNSWLGNIIQYAPTIWVRMVLMTHFFSILMAQDTLDQNLNFEMYGSVYSVSPLDLPAIIERLHGLDAFSLHTYTPHELTRVASALRKLGAPPLRAWKSRARAVRASLISRGGRAAVCGRYLFNWAVKTKLKLTPLPEARLLDLS 1yvz A 2.2 BS01 JPC A 1 R422 M423 H475 T476 Y477 L497 R498 K501 W528 R422 M423 H475 T476 Y477 L497 R498 K501 W528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=4.4uM remove_due_to_license_issue P26660 15746101 578 SMSYSWTGALITPCSPEEEKLPINPLSNSLLRYHNKVYCTTSKSASLRAKKVTFDRMQVLDAYYDSVLKDIKLAASKVSARLLTLEEACQLTPPHSARSKYGFGAKEVRSLSGRAVNHIKSVWKDLLEDSQTPIPTTIMAKNEVFCVDPTKGGKKAARLIVYPDLGVRVCEKMALYDVTQKLPQAVMGASYGFQYSPAQRVEFLLKAWAEKKDPMGFSYDTRCFDSTVTERDIRTEESIYQACSLPEEARTAIHSLTERLYVGGPMFNSKGQSCGYRRCRASGVLTTSMGNTITCYVKALAACKAAGIVAPTMLVCGDDLVVISESQGTEEDERNLRAFTEAMTRYSAPPGDPPRPEYDLELITSCSSNVSVALGPQGRRRYYLTRDPTTPIARAAWETVRHSPVNSWLGNIIQYAPTIWVRMVLMTHFFSILMAQDTLDQNLNFEMYGSVYSVSPLDLPAIIERLHGLDAFSLHTYTPHELTRVASALRKLGAPPLRAWKSRARAVRASLISRGGRAAVCGRYLFNWAVKTKLKLTPLPEARLLDLS 1yw2 A 2.01 BS01 PGJ A 1 A1051 K1053 L1104 V1105 T1106 L1108 M1109 G1110 A1111 A48 K50 L101 V102 T103 L105 M106 G107 A108 D1150 K1152 N1155 D1168 T1185 D147 K149 N152 D165 T173 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=141nM remove_due_to_license_issue P47811 15837333 2001 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGARHVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 1yw7 A 1.85 BS03 A41 A 1 H231 L328 N329 H331 E364 Y444 H122 L219 N220 H222 E255 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 ic50=1.4uM remove_due_to_license_issue IC50=1400nM P50579 16789740 482 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 1yw8 A 2.65 BS03 A75 A 1 H231 L328 N329 H331 I338 E364 F366 Y444 H122 L219 N220 H222 I229 E255 F257 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 remove_due_to_license_issue IC50=10nM P50579 16789740 104 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 1ywr A 1.95 BS01 LI9 A 1 V30 Y35 A51 K53 L104 V105 T106 M109 D112 D168 V26 Y31 A47 K49 L100 V101 T102 M105 D108 D163 D150 K152 N155 D168 T185 D145 K147 N150 D163 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=32nM remove_due_to_license_issue P47811 15837310 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1yxd A 2.0 BS01 LYS B 1 A49 L51 H53 H56 Y106 A49 L51 H53 H56 Y106 T44 Y107 Y133 R138 K161 I203 T44 Y107 Y133 R138 K161 I203 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0042802,0044281 remove_due_to_license_issue P0A6L2 16041077 1300 MFTGSIVAIVTPMDEKGNVCRASLKKLIDYHVASGTSAIVSVGTTGESATLNHDEHADVVMMTLDLADGRIPVIAGTGANATAEAISLTQRFNDSGIVGCLTVTPYYNRPSQEGLYQHFKAIAEHTDLPQILYNVPSRTGCDLLPETVGRLAKVKNIIGIKEATGNLTRVNQIKELVSDDFVLLSGDDASALDFMQLGGHGVISVTANVAARDMAQMCKLAAEGHFAEARVINQRLMPLHNKLFVEPNPIPVKWACKELGLVATDTLRLPMTPITDSGRETVRAALKHAGLL 1yxd A 2.0 BS02 LYS B 2 N80 E84 N80 E84 T44 Y107 Y133 R138 K161 I203 T44 Y107 Y133 R138 K161 I203 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0042802,0044281 remove_due_to_license_issue P0A6L2 16041077 2300 MFTGSIVAIVTPMDEKGNVCRASLKKLIDYHVASGTSAIVSVGTTGESATLNHDEHADVVMMTLDLADGRIPVIAGTGANATAEAISLTQRFNDSGIVGCLTVTPYYNRPSQEGLYQHFKAIAEHTDLPQILYNVPSRTGCDLLPETVGRLAKVKNIIGIKEATGNLTRVNQIKELVSDDFVLLSGDDASALDFMQLGGHGVISVTANVAARDMAQMCKLAAEGHFAEARVINQRLMPLHNKLFVEPNPIPVKWACKELGLVATDTLRLPMTPITDSGRETVRAALKHAGLL 1yxd B 2.0 BS01 LYS B 1 N80 E84 N80 E84 T44 Y107 Y133 R138 K161 I203 T44 Y107 Y133 R138 K161 I203 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0042802,0044281 Ki~22uM remove_due_to_license_issue P0A6L2 16041077 1300 MFTGSIVAIVTPMDEKGNVCRASLKKLIDYHVASGTSAIVSVGTTGESATLNHDEHADVVMMTLDLADGRIPVIAGTGANATAEAISLTQRFNDSGIVGCLTVTPYYNRPSQEGLYQHFKAIAEHTDLPQILYNVPSRTGCDLLPETVGRLAKVKNIIGIKEATGNLTRVNQIKELVSDDFVLLSGDDASALDFMQLGGHGVISVTANVAARDMAQMCKLAAEGHFAEARVINQRLMPLHNKLFVEPNPIPVKWACKELGLVATDTLRLPMTPITDSGRETVRAALKHAGLL 1yxd B 2.0 BS02 LYS B 2 S48 A49 L51 H53 H56 Y106 S48 A49 L51 H53 H56 Y106 T44 Y107 Y133 R138 K161 I203 T44 Y107 Y133 R138 K161 I203 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0042802,0044281 Ki~22uM remove_due_to_license_issue P0A6L2 16041077 2300 MFTGSIVAIVTPMDEKGNVCRASLKKLIDYHVASGTSAIVSVGTTGESATLNHDEHADVVMMTLDLADGRIPVIAGTGANATAEAISLTQRFNDSGIVGCLTVTPYYNRPSQEGLYQHFKAIAEHTDLPQILYNVPSRTGCDLLPETVGRLAKVKNIIGIKEATGNLTRVNQIKELVSDDFVLLSGDDASALDFMQLGGHGVISVTANVAARDMAQMCKLAAEGHFAEARVINQRLMPLHNKLFVEPNPIPVKWACKELGLVATDTLRLPMTPITDSGRETVRAALKHAGLL 1yy4 A 2.7 BS02 4NA A 1 M295 E305 L339 I373 H475 L476 M33 E43 L77 I111 H203 L204 ? remove_due_to_license_issue IC50=2.52nM Q92731 15943471 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNA 1yye A 2.03 BS02 196 A 1 M295 L298 T299 E305 L339 M340 F356 I376 H475 L476 M33 L36 T37 E43 L77 M78 F94 I114 H203 L204 ? ic50=2.7nM remove_due_to_license_issue IC50=2.7nM Q92731 15943471 531 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 1yyr B 2.5 BS02 SAZ B 1 M73 W78 T96 L97 G186 V191 M221 Y295 M71 W76 T94 L95 G184 V189 M219 Y293 Y93 T96 L97 D100 R182 K232 R304 F305 Y91 T94 L95 D98 R180 K230 R302 F303 4.2.3.6 0016106,0016829,0016838,0045482,0046872 remove_due_to_license_issue P13513 15835903 704 NFPTEYFLNTTVRLLEYIRYRDSNYTREERIENLHYAYNKAAHHFAQPRQQQLLKVDPKRLQASLQTIVGMVVYSWAKVSKECMADLSIHYTYTLVLDDSKDDPYPTMVNYFDDLQAGREQAHPWWALVNEHFPNVLRHFGPFCSLNLIRSTLDFFEGCWIEQYNFGGFPGSHDYPQFLRRMNGLGHCVGASLWPKEQFNERSLFLEITSAIAQMENWMVWVNDLMSFYKEFDDERDQISLVKNYVVSDEISLHEALEKLTQDTLHSSKQMVAVFSDKDPQVMDTIECFMHGYVTWHLCDRRFRLSEIYEKVKEEKTEDAQKFCKFYEQAANVGAVSPSEWAYPPVAQLANV 1yys A 2.75 BS01 SAZ A 1 I70 L187 N225 Y295 W298 I69 L186 N224 Y294 W297 Y93 T96 L97 D100 R182 K232 R304 F305 Y92 T95 L96 D99 R181 K231 R303 F304 4.2.3.6 0016106,0016829,0016838,0045482,0046872 remove_due_to_license_issue P13513 15835903 709 ENFPTEYFLNTTVRLLEYIRYRDSNYTREERIENLHYAYNKAAHHFAQPRQQQLLKVDPKRLQASLQTIVGMVVYSWAKVSKECMADLSIHYTYTLVLDDSKDDPYPTMVNYFDDLQAGREQAHPWWALVNEHFPNVLRHFGPFCSLNLIRSTLDFFEGCWIEQYNFGGFPGSHDYPQFLRRMNGLGHCVGASLWPKEQFNERSLFLEITSAIAQMENWMVWVNDLMSFYKEFDDERDQISLVKNYVVSDEISLHEALEKLTQDTLHSSKQMVAVFSDKDPQVMDTIECFMHGYVTWHLCDRRFRLSEIYEKVKEEKTEDAQKFCKFYEQAANVGAVSPSEWAYPPVAQLANV 1yyy 1 2.1 BS02 0KV 1 1 H57 D189 S190 C191 S195 S214 W215 G216 S217 G219 H40 D171 S172 C173 S177 S192 W193 G194 S195 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 9724521 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 1yz3 A 2.4 BS01 SKA A 1 Y35 N39 Y40 V53 K57 F182 E219 V269 Y18 N22 Y23 V36 K40 F165 E202 V252 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=1.55nM remove_due_to_license_issue Ki=3.1nM, IC50=10nM P11086 16279783 3001 PGQAAVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 1z1h A 1.85 BS01 HBB A 1 D25 G27 A28 D29 G48 I50 I84 D25 G27 A28 D29 G48 I50 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4nM remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1z1h B 1.85 BS01 HBB A 1 D125 G127 D130 V182 I184 D25 G27 D30 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1z1r A 1.85 BS01 HBH A 1 D25 G27 A28 D29 D30 G48 G49 I50 V82 D25 G27 A28 D29 D30 G48 G49 I50 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1z1r B 1.85 BS01 HBH A 1 D125 A128 D130 V182 I184 D25 A28 D30 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 10387041 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1z2b B 4.1 BS03 VLB C 1 K176 V177 Y210 T221 P222 T223 Y224 K173 V174 Y207 T218 P219 T220 Y221 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Ki=>100000nM Q6B856 15917812 800 REIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVVPSPKVSDTVVEPYNATLSVHQLVENTDETYSIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSLTVPELTQQMFDSKNMMAACDPRHGRYLTVAAVFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 1z2b C 4.1 BS03 VLB C 1 P325 V328 N329 V353 I355 P315 V318 N319 V343 I345 3.6.5.- 0000226,0000278,0005200,0005525,0005737,0005856,0005874,0007017,0016787,0046872 remove_due_to_license_issue Q2HJ86 15917812 800 RECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLIGQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGI 1z34 A 2.4 BS01 2FD A 1 M64 T90 C91 G92 F159 V178 M180 E181 M64 T90 C91 G92 F159 V178 M180 E181 0003824,0004731,0006139,0009116 ic50=0.42mM remove_due_to_license_issue 15817485 300 ATPHNSAQVGDFAETVLMCGDPLRAKLIAETYLENPKLVNNVRGIQGYTGTYKGKPISVMGHGMGLPSICIYAEELYSTYKVKTIIRVGTCGAIDMDIHTRDIVIFTSAGTNSKINRIRFMDHDYPATASFDVVCALVDAAKELNIPAKVGKGFSTDLFYNPQTELAQLMNKFHFLAVEMESAGLFPIADLYGARAGCICTVSDHILHHEERQNSFQNMMKIALEAAIKL 1z3c A 2.2 BS01 SA8 A 1 K54 G72 D94 I95 D122 S123 Y124 Q140 F141 S142 Y145 K14 G32 D54 I55 D82 S83 Y84 Q100 F101 S102 Y105 2.1.1.56 0003723,0004482,0005634,0006370,0008168,0032259,0106005 ic50=100uM remove_due_to_license_issue Q8SR66 15760890 299 SKTINIRNANNFIKACLIRLYTKRGDSVLDLGCGKGGDLLKYERAGIGEYYGVDIAEVSINDARVRARNMKRRFKVFFRAQDSYGRHMDLGKEFDVISSQFSFHYAFSTSESLDIAQRNIARHLRPGGYFIMTVPSRDVILERYKQGRMSNDFYKIELEKMEDVPMESVREYRFTLLDSVNNCIEYFVDFTRMVDGFKRLGLSLVERKGFIDFYEDEGRRNPELSKKMGLGCLTREESEVVGIYEVVVFRKL 1z3j A -1.00 BS06 NGH A 1 G179 I180 L181 A182 L214 T215 H218 E219 H222 P238 T239 Y240 G75 I76 L77 A78 L110 T111 H114 E115 H118 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=4.3nM P39900 15809432 269 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 1z4n A 1.97 BS02 GL1 A 1 H20 W24 V47 R49 S116 K117 N118 H20 W24 V47 R49 S116 K117 N118 D8 L9 D10 T16 K45 S114 A115 K145 E169 D170 D8 L9 D10 T16 K45 S114 A115 K145 E169 D170 5.4.2.6 0000287,0003824,0005737,0005975,0008801,0016853,0046872 Ki=30uM remove_due_to_license_issue P71447 15826149 1220 MFKAVLFDLDGVITDTAEYHFRAWKALAEEIGINGVDRQFNEQLKGVSREDSLQKILDLADKKVSAEEFKELAKRKNDNYVKMIQDVSPADVYPGILQLLKDLRSNKIKIALASASKNGPFLLERMNLTGYFDAIADPAEVAASKPAPDIFIAAAHAVGVAPSESIGLEDSQAGIQAIKDSGALPIGVGRPEDLGDDIVIVPDTSHYTLEFLKEVWLQK 1z4o A 1.9 BS02 GL1 A 1 D10 H20 W24 G46 V47 R49 S116 K117 N118 D10 H20 W24 G46 V47 R49 S116 K117 N118 D8 L9 D10 T16 K45 S114 A115 K145 E169 D170 D8 L9 D10 T16 K45 S114 A115 K144 E168 D169 5.4.2.6 0000287,0003824,0005737,0005975,0008801,0016853,0046872 Ki=30uM remove_due_to_license_issue P71447 15826149 1220 MFKAVLFDLDGVITDTAEYHFRAWKALAEEIGINGVDRQFNEQLKGVSREDSLQKILDLADKKVSAEEFKELAKRKNDNYVKMIQDVSPADVYPGILQLLKDLRSNKIKIALASASKNGPFLLERMNLTGYFDAIADPAVAASKPAPDIFIAAAHAVGVAPSESIGLEDSQAGIQAIKDSGALPIGVGRPEDLGDDIVIVPDTSHYTLEFLKEVWLQKQ 1z4u A 2.8 BS01 PH9 A 1 P197 R200 N316 S368 L384 G410 M414 Y415 I447 Y448 S556 P198 R201 N317 S369 L385 G411 M415 Y416 I448 Y449 S557 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O93077 15911260 600 MSMSYTWTGALITPCAAEESKLPINALSNSLLRHHNLVYSTTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRSLSSRAVNHIRSVWKDLLEDTDTPIQTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKAKKCPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYVGGPMTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTVPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRAKLLSQGGRAAICGKYLFNWAVRTKLKLTPIPAASRLLLSGWFVAGYSGGDIYHS 1z5m A 2.17 BS01 LI8 A 1 L88 G89 E90 G91 V96 A109 L159 S160 A162 G165 E166 L212 L15 G16 E17 G18 V23 A36 L86 S87 A89 G92 E93 L139 D205 K207 E209 N210 D223 T245 D132 K134 E136 N137 D150 T162 2.7.11.1 0004672,0004674,0005524,0006468 ic50=30nM remove_due_to_license_issue IC50=39nM O15530 15772071 501 PRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 1z63 A 3.0 BS01 dna C 0 H524 R527 T541 A543 R547 R728 H93 R96 T110 A112 R116 R297 ? 0005524 remove_due_to_license_issue Q97XQ7 15882619 7 ~ 25 FQLLEPYNIKANLRPYQIKGFSWMRFMNKLGFGICLADDMGLGKTLQTIAVFSDAKKENELTPSLVICPLSVLKNWEEELSKFAPHLRFAVFHEDRSKIKLEDYDIILTTYAVLLRDTRLKEVEWKYIVIDEAQNIKNPQTKIFKAVKELKSKYRIALTGTPIENKVDDLWSIMTFLNPGLLGSYSEFKSKFATPIKKGDNMAKEELKAIISPFILRRTKYDKAIINDLPDKIETNVYCNLTPEQAAMYKAEVENLFNNIDSVTGIKRKGMILSTLLKLKQIVDHPALLKGGEQSVRRSGKMIRTMEIIEEALDEGDKIAIFTQFVDMGKIIRNIIEKELNTEVPFLYGELSKKERDDIISKFQNNPSVKFIVLSVKAGFGINLTSANRVIHFDRWWNPDQATDRVYRIGQTRNVIVHKLISVGTLEEKIDQLLAFKRSLFKDIISSGDSWITELSTEELRKVIELSV 1z63 A 3.0 BS02 dna D 0 K573 I574 K681 K142 I143 K250 ? 0005524 remove_due_to_license_issue Q97XQ7 15882619 1 ~ 20 FQLLEPYNIKANLRPYQIKGFSWMRFMNKLGFGICLADDMGLGKTLQTIAVFSDAKKENELTPSLVICPLSVLKNWEEELSKFAPHLRFAVFHEDRSKIKLEDYDIILTTYAVLLRDTRLKEVEWKYIVIDEAQNIKNPQTKIFKAVKELKSKYRIALTGTPIENKVDDLWSIMTFLNPGLLGSYSEFKSKFATPIKKGDNMAKEELKAIISPFILRRTKYDKAIINDLPDKIETNVYCNLTPEQAAMYKAEVENLFNNIDSVTGIKRKGMILSTLLKLKQIVDHPALLKGGEQSVRRSGKMIRTMEIIEEALDEGDKIAIFTQFVDMGKIIRNIIEKELNTEVPFLYGELSKKERDDIISKFQNNPSVKFIVLSVKAGFGINLTSANRVIHFDRWWNPDQATDRVYRIGQTRNVIVHKLISVGTLEEKIDQLLAFKRSLFKDIISSGDSWITELSTEELRKVIELSV 1z63 B 3.0 BS01 dna E 0 H524 R527 T541 A543 R547 R728 H93 R96 T110 A112 R116 R297 ? 0005524 remove_due_to_license_issue Q97XQ7 15882619 7 ~ 25 FQLLEPYNIKANLRPYQIKGFSWMRFMNKLGFGICLADDMGLGKTLQTIAVFSDAKKENELTPSLVICPLSVLKNWEEELSKFAPHLRFAVFHEDRSKIKLEDYDIILTTYAVLLRDTRLKEVEWKYIVIDEAQNIKNPQTKIFKAVKELKSKYRIALTGTPIENKVDDLWSIMTFLNPGLLGSYSEFKSKFATPIKKGDNMAKEELKAIISPFILRRTKYDKAIINDLPDKIETNVYCNLTPEQAAMYKAEVENLFNNIDSVTGIKRKGMILSTLLKLKQIVDHPALLKGGEQSVRRSGKMIRTMEIIEEALDEGDKIAIFTQFVDMGKIIRNIIEKELNTEVPFLYGELSKKERDDIISKFQNNPSVKFIVLSVKAGFGINLTSANRVIHFDRWWNPDQATDRVYRIGQTRNVIVHKLISVGTLEEKIDQLLAFKRSLFKDIISSGDSWITELSTEELRKVIELSV 1z63 B 3.0 BS02 dna F 0 K573 I574 K681 K142 I143 K250 ? 0005524 remove_due_to_license_issue Q97XQ7 15882619 1 ~ 20 FQLLEPYNIKANLRPYQIKGFSWMRFMNKLGFGICLADDMGLGKTLQTIAVFSDAKKENELTPSLVICPLSVLKNWEEELSKFAPHLRFAVFHEDRSKIKLEDYDIILTTYAVLLRDTRLKEVEWKYIVIDEAQNIKNPQTKIFKAVKELKSKYRIALTGTPIENKVDDLWSIMTFLNPGLLGSYSEFKSKFATPIKKGDNMAKEELKAIISPFILRRTKYDKAIINDLPDKIETNVYCNLTPEQAAMYKAEVENLFNNIDSVTGIKRKGMILSTLLKLKQIVDHPALLKGGEQSVRRSGKMIRTMEIIEEALDEGDKIAIFTQFVDMGKIIRNIIEKELNTEVPFLYGELSKKERDDIISKFQNNPSVKFIVLSVKAGFGINLTSANRVIHFDRWWNPDQATDRVYRIGQTRNVIVHKLISVGTLEEKIDQLLAFKRSLFKDIISSGDSWITELSTEELRKVIELSV 1z6d A 1.54 BS01 IMP A 1 K7 Q11 H12 K41 V118 H119 K7 Q11 H12 K41 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=4.6mM remove_due_to_license_issue P61823 16045769 919 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1z6d A 1.54 BS02 IMP A 2 H12 V43 N44 T45 R85 F120 H12 V43 N44 T45 R85 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=4.6mM remove_due_to_license_issue P61823 16045769 920 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1z6d A 1.54 BS03 IMP A 3 K66 S123 V124 K66 S123 V124 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=4.6mM remove_due_to_license_issue P61823 16045769 921 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1z6e A 1.8 BS01 IK8 A 1 K96 T98 Y99 E146 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G218 C220 G226 K82 T84 Y85 E135 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.19nM remove_due_to_license_issue Ki=0.19nM P00742 15771420 711 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 1z6f A 1.6 BS01 BO9 A 1 A43 S44 K47 P81 K84 G85 S86 S87 F90 L153 R198 G215 H216 A40 S41 K44 P78 K81 G82 S83 S84 F87 L150 R195 G212 H213 3.4.16.4,3.5.2.6 0000270,0004180,0005515,0005886,0006508,0008233,0008360,0008658,0008800,0009002,0009252,0030288,0042803,0051301,0071555 remove_due_to_license_issue P0AEB2 15938610 401 NIKTMIPGVPQIDAESYILIDYNSGKVLAEQNADVRRDPASLTKMMTSYVIGQAMKAGKFKETDLVTIGNDAWATGNPVFKGSSLMFLKPGMQVPVSQLIRGINLQSGNDACVAMADFAAGSQDAFVGLMNSYVNALGLKNTHFQTVHGLDADGQYSSARDMALIGQALIRDVPNEYSIYKEKEFTFNGIRQLNRNGLLWDNSLNVDGIKTGHTDKAGYNLVASATEGQMRLISAVMGGRTFKGREAESKKLLTWGFRFFETVNPLKVGKEFASEPVWFGDSDRASLGVDKDVYLTIPRGRMKDLKASYVLNSSELHAPLQKNQVVGTINFQLDGKTIEQRPLVVLQEIPEGNF 1z6j H 2.0 BS02 PY3 H 1 H57 C58 D60 G97 T98 D189 S190 C191 K192 S195 S214 W215 G216 G219 C220 H41 C42 D44 G85 T86 D186 S187 C188 K189 S192 S211 W212 G213 G215 C216 3.4.21.21 0004252,0006508 ic50=0.0094uM remove_due_to_license_issue IC50=9.4nM P08709 15913999 403 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 1z6p A 2.4 BS01 194 A 1 W67 I68 Q71 Q72 Y75 R81 Y155 R193 R310 W61 I62 Q65 Q66 Y69 R75 Y149 R187 R294 H377 K568 R569 K574 T676 K680 H355 K546 R547 K552 T654 K658 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=0.9uM remove_due_to_license_issue P00489 15214781 843 QEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 1z6q A 2.03 BS01 195 A 1 W67 I68 Q71 Q72 Y75 R81 R193 R309 R310 W61 I62 Q65 Q66 Y69 R75 R187 R293 R294 H377 K568 R569 K574 T676 K680 H355 K546 R547 K552 T654 K658 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=74nM remove_due_to_license_issue P00489 15214781 843 QEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 1z6s A 1.5 BS01 AMP A 1 Q11 H12 N67 Q69 N71 A109 H119 Q11 H12 N67 Q69 N71 A109 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=46uM remove_due_to_license_issue P61823 16045769 1101 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1z71 A 1.8 BS02 L17 A 1 H57 Y60A W60D E97A N98 L99 I174 A190 C191 S195 V213 S214 W215 G216 G226 F227 H69 Y73 W76 E120 N121 L122 I197 A218 C219 S223 V243 S244 W245 G246 G256 F257 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=0.66nM remove_due_to_license_issue P00734 15911253 1001 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1z95 A 1.8 BS01 198 A 1 L704 N705 L707 Q711 M742 M745 V746 M749 F764 T877 M895 I899 L33 N34 L36 Q40 M71 M74 V75 M78 F93 T198 M216 I220 ? Ki=76nM remove_due_to_license_issue IC50=248nM, Ki=509nM P10275 15833816 501 IFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSLMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 1z9c A 2.64 BS01 dna G 0 Y19 R23 V57 K58 S68 T72 R94 S95 V96 Y11 R15 V49 K50 S60 T64 R86 S87 V88 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 29 KLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLHQ 1z9c A 2.64 BS02 dna H 0 T39 P41 G69 T70 R77 E93 R94 T31 P33 G61 T62 R69 E85 R86 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 29 KLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLHQ 1z9c B 2.64 BS01 dna G 0 T39 P41 Q42 G69 T70 M74 R77 D92 E93 R94 T32 P34 Q35 G62 T63 M67 R70 D85 E86 R87 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 29 MKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c B 2.64 BS02 dna H 0 Y19 R23 K27 V57 K58 S68 T72 R94 S95 V96 Y12 R16 K20 V50 K51 S61 T65 R87 S88 V89 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 29 MKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c C 2.64 BS01 dna I 0 Y19 R23 V57 K58 S68 T72 R94 S95 V96 Y13 R17 V51 K52 S62 T66 R88 S89 V90 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 2 ~ 29 HMKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c C 2.64 BS02 dna J 0 T39 L66 G69 T70 R77 E93 R94 T33 L60 G63 T64 R71 E87 R88 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 28 HMKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c D 2.64 BS01 dna I 0 T39 P41 Q42 T70 R77 D92 E93 R94 T32 P34 Q35 T63 R70 D85 E86 R87 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 2 ~ 29 MKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c D 2.64 BS02 dna J 0 Y19 R23 V57 K58 S68 G69 T72 R86 R94 S95 V96 Y12 R16 V50 K51 S61 G62 T65 R79 R87 S88 V89 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 28 MKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c E 2.64 BS01 dna K 0 Y19 K27 V57 K58 S68 T72 R86 R94 S95 Y12 K20 V50 K51 S61 T65 R79 R87 S88 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 29 MKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c E 2.64 BS02 dna L 0 T39 P41 Q42 L66 G69 T70 R77 D92 E93 R94 T32 P34 Q35 L59 G62 T63 R70 D85 E86 R87 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 28 MKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c F 2.64 BS01 dna K 0 T39 P41 Q42 G69 T70 R77 D92 E93 R94 T33 P35 Q36 G63 T64 R71 D86 E87 R88 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 29 HMKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9c F 2.64 BS02 dna L 0 Y19 R23 K30 V57 K58 S68 G69 T72 K76 R94 S95 Y13 R17 K24 V51 K52 S62 G63 T66 K70 R88 S89 ? 0000122,0000977,0001227,0003677,0003700,0005737,0006355,0006950,0042542,0042802,0042803,0045892 remove_due_to_license_issue O34777 16209951 1 ~ 28 HMKLENQLSFLLYASSREMTKQYKPLLDKLNITYPQYLALLLLWEHETLTVKKMGEQLYLDSGTLTPMLKRMEQQGLITRKRSEEDERSVLISLTEDGALLKEKAVDIPGTILGLSKQSGEDLKQLKSALYTLLETLH 1z9g E 1.7 BS06 RRT E 1 N112 A113 V139 E143 I188 L202 R203 H231 N112 A113 V139 E143 I188 L202 R203 H231 3.4.24.27 0004222,0006508 Ki=2.3uM remove_due_to_license_issue Ki=2300nM P00800 2719912 1006 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1z9h A 2.6 BS01 IMN A 1 T109 C110 P111 F112 P134 I246 Y251 S260 Y263 V343 T10 C11 P12 F13 P35 I147 Y152 S161 Y164 V244 Y107 C110 F112 C113 Y8 C11 F13 C14 5.3.99.3 0050220 remove_due_to_license_issue Q9N0A4 15854652 379 LQLTLYQYKTCPFCSKVRAFLDFHALPYQVVEVNPVLRAEIKFSSYRKVPILVAQEGESSQQLNDSSVIISALKTYLVSGQPLEEIITYYPAMKAVNDQGKEVTEFGNKYWLMLNEKEAQQVYSGKEARTEEMKWRQWADDWLVHLISPNVYRTPTEALASFDYIVREGKFGAVEGAVAKYMGAAAMYLISKRLKSRHRLQDNVREDLYEAADKWVAAVGKDRPFMGGQKPNLADLAVYGVLRVMEGLDAFDDLMQHTHIQPWYLRVERAITEA 1z9y A 1.66 BS02 FUN A 1 H64 H94 H119 V121 F131 L198 T199 T200 H61 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=6.5e+4nM P00918 500 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1zaf A 2.2 BS02 789 A 1 M295 E305 L339 F356 H475 L476 M33 E43 L77 F94 H203 L204 ? ic50=20nM remove_due_to_license_issue IC50=20nM Q92731 15876535 201 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSAMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 1zaj A 1.89 BS01 M2P A 1 D33 S35 S38 K107 K146 E187 K229 S271 G272 Y301 G302 R303 D33 S35 S38 K107 K146 E187 K229 S271 G272 Y301 G302 R303 D33 K146 E187 E189 K229 S300 Y363 D33 K146 E187 E189 K229 S300 Y363 4.1.2.13 0004332,0005515,0005737,0006096,0016829,0030335,0031430,0031674,0034316,0051289 remove_due_to_license_issue IC50=8000nM P00883 15870069 3001 PHSHPALTPEQKKELSDIAHRIVAPGKGILAADESTGSIAKRLQSIGTENTEENRRFYRQLLLTADDRVNPCIGGVILFHETLYQKADDGRPFPQVIKSKGGVVGIKVDKGVVPLAGTNGETTTQGLDGLSERCAQYKKDGADFAKWRCVLKIGEHTPSALAIMENANVLARYASICQQNGIVPIVEPEILPDGDHDLKRCQYVTEKVLAAVYKALSDHHIYLEGTLLKPNMVTPGHACTQKYSHEEIAMATVTALRRTVPPAVTGVTFLSGGQSEEEASINLNAINKCPLLKPWALTFSYGRALQASALKAWGGKKENLKAAQEEYVKRALANSLACQGKYTPSGQAGAAASESLFISNHAY 1zc9 A 2.0 BS01 PMP A 1 G111 A112 W138 H139 E210 D243 A245 Q246 K272 G109 A110 W136 H137 E208 D241 A243 Q244 K270 G21 W138 E210 D243 Q246 K272 T303 R406 G19 W136 E208 D241 Q244 K270 T301 R404 4.1.1.64 0008483,0016831,0030170,0047432 Kd=0.6mM remove_due_to_license_issue P16932 16342932 502 LNDDATFWRNARHHLVRYGGTFEPMIIERAKGSFVYDADGRAILDFTSGQMSAVLGHCHPEIVSVIGEYAGKLDHLFSEMLSRPVVDLATRLANITPPGLDRALLLSTGAESNEAAIRMAKLVTGKYEIVGFAQSWHGMTGAAASATYSAGRKGVGPAAVGSFAIPAPFTYRPRFERNGAYDYLAELDYAFDLIDRQSSGNLAAFIAEPILSSGGIIELPDGYMAALKRKCEARGMLLILDEAQTGVGRTGTMFACQRDGVTPDILTLSKTLGAGLPLAAIVTSAAIEERAHELGYLFYTTHVSDPLPAAVGLRVLDVVQRDGLVARANVMGDRLRRGLLDLMERFDCIGDVRGRGLLLGVEIVKDRRTKEPADGLGAKITRECMNLGLSMNIVQLPGMGGVFRIAPPLTVSEDEIDLGLSLLGQAIERAL 1zd2 P 3.0 BS02 NC3 P 1 F265 D333 W334 Y381 M418 Y465 H523 W524 F266 D334 W335 Y382 M418 Y465 H523 W524 F265 W334 N376 Y381 D495 H523 F266 W335 N377 Y382 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=>500000nM P34913 16322563 700 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 1zd3 A 2.3 BS02 NC4 A 1 D333 W334 Y381 Q382 M418 Y465 H523 W524 D334 W335 Y382 Q383 M418 Y465 H523 W524 F265 H332 D333 W334 N357 N376 Y381 Y465 D495 H523 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50>500uM remove_due_to_license_issue IC50=36000nM P34913 16322563 790 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 1zd4 A 2.7 BS02 NC6 A 1 D333 W334 M337 Y381 M418 Y465 H523 D334 W335 M338 Y382 M418 Y465 H523 F265 H332 D333 W334 N357 N376 Y381 Y465 D495 H523 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=>100000nM P34913 16322563 700 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 1zd5 A 2.6 BS02 NC7 A 1 F265 D333 W334 F379 Y381 Q382 M418 Y465 H523 F266 D334 W335 F380 Y382 Q383 M418 Y465 H523 F265 H332 D333 W334 N357 N376 Y381 Y465 D495 H523 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue P34913 16322563 700 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 1zdp E 1.7 BS06 TIO E 1 N112 A113 V139 E143 I188 L202 R203 H231 N112 A113 V139 E143 I188 L202 R203 H231 3.4.24.27 0004222,0006508 Ki=1.8uM remove_due_to_license_issue Ki=1800nM, IC50=9500nM P00800 2719912 1006 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 1ze8 A 2.0 BS03 PIU A 1 I91 H94 H119 F131 L198 T199 T200 I89 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=21nM remove_due_to_license_issue Ki=21nM P00918 16134940 1 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1zeo A 2.5 BS01 C01 A 1 F282 C285 S289 H323 I326 L330 F363 M364 H449 Y473 F68 C71 S75 H109 I112 L116 F149 M150 H235 Y259 ? 0003677,0004879,0005634,0006355 ic50=0.21uM remove_due_to_license_issue P37231 15974597 478 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 1zfk A 1.56 BS02 NR2 A 1 H1094 H1119 L1198 T1199 T1200 P1202 H91 H116 L194 T195 T196 P198 H1064 H1094 H1096 E1106 H1119 T1199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=12nM P00918 1400 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1zfk A 1.56 BS03 NR2 A 2 L1057 F1070 D1071 D1072 I1091 L54 F67 D68 D69 I88 H1064 H1094 H1096 E1106 H1119 T1199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=12nM P00918 1500 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1zfq A 1.55 BS02 ZEC A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=30nM, IC50=4nM P00918 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1zfq A 1.55 BS03 ZEC A 2 H4 W5 N11 H15 W16 D19 H1 W2 N8 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=30nM, IC50=4nM P00918 400 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1zg1 A 2.3 BS01 dna C 0 P172 N173 K188 S202 R203 P22 N23 K38 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 A 2.3 BS02 dna D 0 T157 R159 I182 T183 S185 T186 V189 H190 T7 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 B 2.3 BS01 dna C 0 T157 R159 I182 T183 S185 T186 H190 T7 R9 I32 T33 S35 T36 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 B 2.3 BS02 dna D 0 P172 N173 K192 S202 R203 P22 N23 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 E 2.3 BS01 dna G 0 P172 N173 S202 R203 P22 N23 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 E 2.3 BS02 dna H 0 T157 R159 I182 T183 S185 T186 H190 T7 R9 I32 T33 S35 T36 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 F 2.3 BS01 dna G 0 T157 R159 I182 T183 S185 T186 V189 H190 T7 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg1 F 2.3 BS02 dna H 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 A 2.3 BS01 dna C 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 A 2.3 BS02 dna D 0 T157 R159 I182 T183 S185 T186 V189 H190 T7 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 B 2.3 BS01 dna C 0 T157 R159 I182 T183 S185 T186 V189 H190 T7 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 B 2.3 BS02 dna D 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 E 2.3 BS01 dna G 0 P172 N173 K188 K192 S202 R203 P23 N24 K39 K43 S53 R54 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 ERDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 E 2.3 BS02 dna H 0 T157 R159 I182 T183 S185 T186 V189 H190 T8 R10 I33 T34 S36 T37 V40 H41 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 ERDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 F 2.3 BS01 dna G 0 T157 R159 I182 T183 S185 T186 V189 H190 T7 R9 I32 T33 S35 T36 V39 H40 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 1 ~ 20 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zg5 F 2.3 BS02 dna H 0 P172 N173 K188 K192 S202 R203 P22 N23 K38 K42 S52 R53 ? 0003677,0006355 remove_due_to_license_issue P0AF28 16262254 21 ~ 40 RDVNQLTPRERDILKLIAQGLPNKMIARRLDITESTVKVHVKHMLKKMKLKSRVEAAVWVHQERIF 1zgb A 2.3 BS01 A1E A 1 W84 G118 Y121 E199 W279 F330 Y334 W432 H440 W81 G115 Y118 E196 W276 F327 Y331 W429 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 ic50=8.8nM remove_due_to_license_issue P04058 16076210 1001 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 1zge A 1.65 BS02 SDA A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=50nM P00918 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 1zgi A 2.2 BS02 382 A 1 H57 Y60A W60D E97A N98 L99 A190 E192 S195 V213 W215 G216 G219 C220 H69 Y73 W76 E120 N121 L122 A218 E220 S223 V243 W245 G246 G248 C249 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=4.6uM remove_due_to_license_issue Ki=4.6nM P00734 16137886 1001 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1zgv A 2.2 BS02 501 A 1 Y60A A190 C191 S195 V213 W215 G216 G219 G226 F227 Y73 A218 C219 S223 V243 W245 G246 G248 G256 F257 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 ic50~1uM remove_due_to_license_issue IC50=1000nM P00734 16137886 1001 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 1zh5 A 1.85 BS01 rna C 0 F28 V108 Q141 K185 F24 V104 Q137 K181 ? 0003676,0003723,0005634,0006396,1990904 remove_due_to_license_issue P05455 16387655 1 ~ 9 GDNEKMAALEAKICHQIEYYFGDFNLPRDKFLKEQIKLDEGWVPLEIMIKFNRLNRLTTDFNVIVEALSKSKAELMEISEDKTKIRRSPSKPLPEVTDEYKNDVKNRSVYIKGFPTDATLDDIKEWLEDKGQVLNIQMRRTLHKAFKGSIFVVFDSIESAKKFVETPGQKYKETDLLILFKDDYF 1zh5 A 1.85 BS02 rna D 0 Y23 Y24 D33 F55 N56 R57 I140 Y19 Y20 D29 F51 N52 R53 I136 ? 0003676,0003723,0005634,0006396,1990904 remove_due_to_license_issue P05455 16387655 1 ~ 9 GDNEKMAALEAKICHQIEYYFGDFNLPRDKFLKEQIKLDEGWVPLEIMIKFNRLNRLTTDFNVIVEALSKSKAELMEISEDKTKIRRSPSKPLPEVTDEYKNDVKNRSVYIKGFPTDATLDDIKEWLEDKGQVLNIQMRRTLHKAFKGSIFVVFDSIESAKKFVETPGQKYKETDLLILFKDDYF 1zh5 B 1.85 BS01 rna C 0 Y23 Y24 D33 F35 K54 F55 R57 L124 I140 Y18 Y19 D28 F30 K49 F50 R52 L119 I135 ? 0003676,0003723,0005634,0006396,1990904 remove_due_to_license_issue P05455 16387655 1 ~ 9 DNEKMAALEAKICHQIEYYFGDFNLPRDKFLKEQIKLDEGWVPLEIMIKFNRLNRLTTDFNVIVEALSKSKAELMEISEDKTKIRRSPSKPLPEVTDEYKNDVKNRSVYIKGFPTDATLDDIKEWLEDKGQVLNIQMRRTLHKAFKGSIFVVFDSIESAKKFVETPGQKYKETDLLILFKDDYF 1zh5 B 1.85 BS02 rna D 0 F28 R32 V108 Q141 K185 F23 R27 V103 Q136 K180 ? 0003676,0003723,0005634,0006396,1990904 remove_due_to_license_issue P05455 16387655 1 ~ 9 DNEKMAALEAKICHQIEYYFGDFNLPRDKFLKEQIKLDEGWVPLEIMIKFNRLNRLTTDFNVIVEALSKSKAELMEISEDKTKIRRSPSKPLPEVTDEYKNDVKNRSVYIKGFPTDATLDDIKEWLEDKGQVLNIQMRRTLHKAFKGSIFVVFDSIESAKKFVETPGQKYKETDLLILFKDDYF 1zho A 2.6 BS01 rna B 0 P1 H3 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 K70 P133 R134 D166 K167 T168 H172 P174 Y213 T217 M218 G219 P220 S221 P1 H3 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 K70 P133 R134 D166 K167 T168 H172 P174 Y213 T217 M218 G219 P220 S221 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 16330048 1 ~ 38 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 1zho A 2.6 BS02 rna H 0 S54 D55 N57 G124 S125 K126 R129 L137 K141 F147 S54 D55 N57 G124 S125 K126 R129 L137 K141 F147 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 16330048 1 ~ 38 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 1zho C 2.6 BS01 rna B 0 S54 D55 N57 P117 D118 V119 G121 G128 R129 P133 K141 F147 S54 D55 N57 P117 D118 V119 G121 G128 R129 P133 K141 F147 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 16330048 1 ~ 38 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 1zho C 2.6 BS02 rna D 0 H3 G4 K5 R6 Y7 K36 F37 T40 E42 H44 K46 D166 K167 T168 H172 Y213 T217 M218 G219 P220 S221 H3 G4 K5 R6 Y7 K36 F37 T40 E42 H44 K46 D166 K167 T168 H172 Y213 T217 M218 G219 P220 S221 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 16330048 1 ~ 38 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 1zho E 2.6 BS01 rna F 0 P1 H3 G4 K5 R6 Y7 A35 K36 F37 E42 H44 K46 R134 D166 K167 T168 H172 S211 Y213 T217 M218 G219 P220 S221 P1 H3 G4 K5 R6 Y7 A35 K36 F37 E42 H44 K46 R134 D166 K167 T168 H172 S211 Y213 T217 M218 G219 P220 S221 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 16330048 1 ~ 38 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 1zho G 2.6 BS01 rna H 0 P1 H3 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 D166 K167 T168 H172 P174 Y213 T215 T217 M218 G219 P220 S221 P1 H3 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 D166 K167 T168 H172 P174 Y213 T215 T217 M218 G219 P220 S221 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 16330048 1 ~ 38 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 1zhy A 1.6 BS01 CLR A 1 Q96 Y97 E107 N165 Q181 Q98 Y99 E109 N167 Q183 ? 0000139,0005546,0005737,0005794,0005829,0006665,0006869,0006887,0006892,0006897,0008142,0008289,0015248,0015918,0016020,0030011,0034727,0035621,0070273,0070300,0120015 Kd=300nM remove_due_to_license_issue P35844 16136145 1001 MDPSQYASSSSWTSFLKSIASFNGDLSSLSAPPFILSPISLTEFSQYWAEHPELFLEPSFINDDNYKEHCLIDPEVESPELARMLAVTKWFISTLKSQYCSRNESLGSEKKPLNPFLGELFVGKWENKEHPEFGETVLLSEQVSHHPPVTAFSIFNDKNKVKLQGYNQIKASFTKSLMLTVKQFGHTMLDIKDESYLVTPPPLHIEGILVASPFVELEGKSYIQSSTGLLCVIEFSGRGYFSGKKNSFKARIYKDSKDSKDKEKALYTISGQWSGSSKIIKANKKEESRLFYDAARIPAEHLNVKPLEEQHPLESRKAWYDVAGAIKLGDFNLIAKTKTELEETQRELRKEEEAKGISWQRRWFKDFDYSVTPEEGALVPEKDDTFLKLASALNLSTKNAPSGTLVGDKEDRKEDLSSIHWRFQRELWDEEKEIVL 1zjm A 2.1 BS01 dna T 0 H34 S229 K230 G231 T233 K234 Y271 Y296 H25 S217 K218 G219 T221 K222 Y259 Y284 D190 D192 D256 D181 D183 D244 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 16084394 1 ~ 16 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 1zjm A 2.1 BS02 dna P 0 S104 G105 I106 G107 P108 S109 A110 R254 D256 S95 G96 I97 G98 P99 S100 A101 R242 D244 D190 D192 D256 D181 D183 D244 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 16084394 1 ~ 10 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 1zjm A 2.1 BS03 dna D 0 K35 A38 Y39 G64 G66 K68 I69 K26 A29 Y30 G55 G57 K59 I60 D190 D192 D256 D181 D183 D244 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 16084394 1 ~ 5 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 1zjn A 2.61 BS01 dna T 0 H34 S229 K230 G231 T233 K234 K280 R283 I293 N294 E295 Y296 H25 S220 K221 G222 T224 K225 K271 R274 I284 N285 E286 Y287 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 16084394 1 ~ 16 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRS 1zjn A 2.61 BS02 dna P 0 S104 G105 G107 P108 S109 A110 S95 G96 G98 P99 S100 A101 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 16084394 1 ~ 10 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRS 1zjn A 2.61 BS03 dna D 0 K35 A38 Y39 P63 G64 G66 K68 I69 K26 A29 Y30 P54 G55 G57 K59 I60 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 16084394 1 ~ 5 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRS 1zkl A 1.67 BS02 IBM A 1 Y211 F384 Q413 F416 Y73 F246 Q275 F278 3.1.4.53 0004114,0007165,0008081 ic50=8.1uM remove_due_to_license_issue IC50=85600nM, Ki=4000nM Q13946 15994308 503 DYNGQAKCMLEKVGNWNFDIFLFDRLTNGNSLVSLTFHLFSLHGLIEYFHLDMMKLRRFLVMIQEDYHSQNPYHNAVHAADVTQAMHCYLKEPKLANSVTPWDILLSLIAAATHDLDHPGVNQPFLIKTNHYLATLYKNTSVLENHHWRSAVGLLRESGLFSHLPLESRQQMETQIGALILATDISRQNEYLSLFRSHLDRGDLCLEDTRHRHLVLQMALKCADICNPCRTWELSKQWSEKVTEEFFHQGDIEKKYHLGVSPLCDRHTESIANIQIGFMTYLVEPLFTEWARFSNTRLSQTMLGHVGLNKASWKGLQ 1zkn A 2.1 BS02 IBM A 1 I336 F340 M357 F372 I258 F262 M279 F294 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=31000nM Q08499 14668322 603 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 1zky A 2.25 BS02 689 A 1 M343 E353 L387 F404 M421 H524 M40 E50 L84 F101 M118 H214 ? Ki=560nM remove_due_to_license_issue P03372 16648639 700 NSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL 1zm7 A 2.2 BS01 TTP A 1 I29 G30 S31 G32 K33 T34 W57 Y70 F80 Q81 E104 R105 A110 F114 R167 R169 E172 I18 G19 S20 G21 K22 T23 W46 Y59 F69 Q70 E93 R94 A99 F103 R156 R158 E161 E52 R105 E41 R94 2.7.1.145 0004136,0004137,0004138,0004797,0004849,0005524,0005737,0005739,0006139,0006170,0006222,0009157,0009224,0016301,0019136,0043174,0043771,0071897,1901293 ic50>1000uM remove_due_to_license_issue Q9XZT6 16008571 300 TKYAEGTQPFTVLIEGNIGSGKTTYLNHFEKYKNDICLLTEPVEKWRNVNGVDLLELMYKDPKKWAMPFQSYVTLTMLQSHTAPTNKKLKIMERSIFSARYCFVENMRRNGSLEQGMYNTLEEWYKFIEESIHVQADLIIYLRTSPEVAYERIRQRARSEESCVPLKYLQELHELHEDWLIHQRRPQSCKVLVLDAD 1zoe A 1.77 BS01 K25 A 1 R47 V53 I66 F113 V116 M163 I174 R41 V47 I60 F107 V110 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.04uM remove_due_to_license_issue P28523 16298300 501 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 1zog A 2.3 BS01 K37 A 1 V45 V53 I66 F113 V116 M163 I174 V39 V47 I60 F107 V110 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.07uM remove_due_to_license_issue P28523 16298300 501 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 1zog A 2.3 BS02 K37 A 2 V53 I66 V95 F113 V116 M163 I174 V47 I60 V89 F107 V110 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.07uM remove_due_to_license_issue P28523 16298300 502 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 1zoh A 1.81 BS01 K44 A 1 I66 K68 V95 F113 V116 M163 I174 I61 K63 V90 F108 V111 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.1uM remove_due_to_license_issue P28523 16298300 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 1zom A 2.25 BS01 339 A 1 H57 E98 H174 D189 A190 C191 K192 G193 D194 S195 W215 G216 E217 H44 E89 H165 D182 A183 C184 K185 G186 D187 S188 W208 G209 E210 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 17181160 1001 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQA 1zp5 A 1.8 BS05 2NI A 1 I159 L160 A161 V194 H197 E198 L214 Y216 P217 N218 Y219 I80 L81 A82 V115 H118 E119 L135 Y137 P138 N139 Y140 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=1200uM remove_due_to_license_issue IC50=1200000nM P22894 16242329 1000 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1zp8 A 2.02 BS01 AB2 A 1 D25 D29 D30 G48 G49 I50 I84 D25 D29 D30 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=1.7nM remove_due_to_license_issue O92139 15934050 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1zpa A 2.02 BS01 A83 A 1 D25 A28 D29 G48 G49 I50 D25 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4nM remove_due_to_license_issue P03366 15934050 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1zpb A 2.1 BS01 995 A 1 H57 D189 A190 C191 K192 G193 D194 S195 S214 W215 G216 E217 H44 D182 A183 C184 K185 G186 D187 S188 S207 W208 G209 E210 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 16524727 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQA 1zpc A 2.6 BS01 716 A 1 H57 E98 H174 D189 A190 C191 K192 G193 D194 S195 S214 W215 G216 E217 H44 E89 H165 D182 A183 C184 K185 G186 D187 S188 S207 W208 G209 E210 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 16524727 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQA 1zq3 P -1.00 BS01 dna A 0 G1 R4 T5 R6 F9 N52 R56 G1 R4 T5 R6 F9 N52 R56 ? 0000981,0003677,0006355 remove_due_to_license_issue P09081 16406070 69 ~ 81 GPRRTRTTFTSSQIAELEQHFLQGRYLTAPRLADLSAKLALGTAQVKIWFKNRRRRHKIQSDQHKDQS 1zq3 P -1.00 BS02 dna B 0 R3 R4 T5 L27 K47 K51 R54 R55 K58 R3 R4 T5 L27 K47 K51 R54 R55 K58 ? 0000981,0003677,0006355 remove_due_to_license_issue P09081 16406070 82 ~ 94 GPRRTRTTFTSSQIAELEQHFLQGRYLTAPRLADLSAKLALGTAQVKIWFKNRRRRHKIQSDQHKDQS 1zrz A 3.0 BS01 BI1 A 1 I251 G252 V259 A272 K274 E324 Y325 V326 D373 L376 T386 D387 I12 G13 V20 A33 K35 E85 Y86 V87 D134 L137 T147 D148 D369 K371 N374 D387 T407 D130 K132 N135 D148 T168 2.7.11.13 0004672,0004674,0004697,0005524,0006468 remove_due_to_license_issue IC50=3463nM P41743 16125198 1000 LGLQDFDLLRVIGRGSYAKVLLVRLKKTDRIYAMKVVKKELVNDDEDIDWVQTEKHVFEQASNHPFLVGLHSCFQTESRLFFVIEYVNGGDLMFHMQRQRKLPEEHARFYSAEISLALNYLHERGIIYRDLKLDNVLLDSEGHIKLTDYGMCKEGLRPGDTTSTFCGTPNYIAPEILRGEDYGFSVDWWALGVLMFEMMAGRSPFDQNTEDYLFQVILEKQIRIPRSMSVKAASVLKSFLNKDPKERLGCLPQTGFADIQGHPFFRNVDWDMMEQKQVVPPFKPVQLTPDDDDIVRKIDQSEFEGFEYINPL 1zs0 A 1.56 BS05 EIN A 1 I159 L160 A161 L193 V194 H197 E198 H201 H207 L214 Y216 P217 N218 Y219 I80 L81 A82 L114 V115 H118 E119 H122 H128 L135 Y137 P138 N139 Y140 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 Ki=0.7uM remove_due_to_license_issue Ki=700nM, IC50=810nM P22894 16451058 994 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1zsb A 2.0 BS02 AZM A 1 Q92 H94 H119 V121 F131 L198 T199 T200 Q89 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=250mM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 8639494 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAQLHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 1zsf A 1.98 BS01 0ZS B 1 D25 G27 A28 D29 D30 I47 G48 P81 V82 D25 G27 A28 D29 D30 I47 G48 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 16627941 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1zsf B 1.98 BS01 0ZS B 1 D125 G127 A128 G148 G149 V182 I184 D25 G27 A28 G48 G49 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.12nM remove_due_to_license_issue P03366 16627941 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1zsh A 2.9 BS02 IHP A 1 R236 K250 K324 K326 R231 K245 K319 K321 ? 0000822,0001664,0001934,0002029,0002031,0002092,0005515,0005547,0005634,0005737,0005829,0005886,0005905,0006511,0007165,0007601,0009968,0015031,0030132,0030276,0031143,0031410,0031623,0032050,0033130,0035612,0036094,0042995,0045746,0060090,0070374,0072583 remove_due_to_license_issue P17870 16439357 601 TRVFKKASPNGKLTVYLGKRDFVDHIDLVEPVDGVVLVDPEYLKERRVYVTLTCAFRYGREDLDVLGLTFRKDLFVANVQSFPPAPEDKKPLTRLQERLIKKLGEHAYPFTFEIPPNLPCSVTLQPGPEDTGKACGVDYEVKAFCAENLEEKIHKRNSVRLVIRKVQYAPERPGPQPTAETTRQFLMSDKPLHLEASLDKEIYYHGEPISVNVHVTNNTNKTVKKIKISVRQYADICLFNTAQYKCPVAMEEADDTVAPSSTFCKVYTLTPFLANNREKRGLALDGKLKHEDTNLASSTLLREGANREILGIIVSYKVKVKLVVSSSDVAVELPFTLMHPKDIVFEDFARQRLK 1zsr A 2.06 BS01 0ZT A 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 V82 D25 G27 A28 D29 D30 I47 G48 G49 I50 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.15nM remove_due_to_license_issue P03366 16627941 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1zsr B 2.06 BS01 0ZT A 1 D125 G127 G148 P181 V182 I184 D25 G27 G48 P81 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 16627941 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1ztq A 2.0 BS06 033 A 1 L159 L160 A161 H197 E198 H201 H207 G212 L214 F216 P217 I218 Y219 T220 F227 P230 L78 L79 A80 H116 E117 H120 H126 G131 L133 F135 P136 I137 Y138 T139 F146 P149 H197 E198 H201 H207 H116 E117 H120 H126 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P45452 16005220 601 YNVFLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGP 1zuc A 2.0 BS01 T98 A 1 L718 N719 Q725 M759 F778 L797 T894 L37 N38 Q44 M78 F97 L116 T213 ? ic50=1.7nM remove_due_to_license_issue IC50=0.5nM, EC50=0.15nM P06401 15937332 201 QLIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 1zvx A 1.87 BS05 FIN A 1 I159 L160 A161 H162 H197 E198 H207 L214 Y216 P217 N218 Y219 I80 L81 A82 H83 H118 E119 H128 L135 Y137 P138 N139 Y140 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 Ki=0.6nM remove_due_to_license_issue Ki=0.6nM, IC50=1.4nM P22894 16451058 994 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 1zxc A 2.28 BS02 IH6 A 1 T347 L348 G349 L401 H405 E406 H409 H415 P437 A439 V440 T131 L132 G133 L185 H189 E190 H193 H199 P221 A223 V224 3.4.24.86 0004222,0006508,0008237 ic50=8nM remove_due_to_license_issue IC50=8nM P78536 16084720 478 DPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYVGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERSN 1zxv A 2.67 BS02 MFM A 1 G657 L658 P661 E687 H690 Y728 G609 L610 P613 E639 H642 Y680 H686 E687 H690 Y728 E735 H638 E639 H642 Y680 E687 3.4.24.83 0003824,0005576,0008237,0046872 remove_due_to_license_issue IC50=1700nM, Ki=800nM Q52NH3 15983377 9002 ERNKTQEEHLKEIMKHIVKIEVKGEEAVKKEAAEKLLEKVPSDVLEMYKAIGGKIYIVDGDITKHISLEALSEDKKKIKDIYGKDALLHEHYVYAKEGYEPVLVIQSSEDYVENTEKALNVYYEIGKILSRDILSKINQPYQKFLDVLNTIKNASDSDGQDLLFTNQLKEHPTDFSVEFLEQNSNEVQEVFAKAFAYYIEPQHRDVLQLYAPEAFNYMDKFNEQEINLSLEELKDQRMLSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDILSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 1zyj A 2.0 BS01 BI5 A 1 A51 K53 L104 T106 L108 M109 G110 A111 L167 A43 K45 L96 T98 L100 M101 G102 A103 L159 D150 K152 N155 D168 T185 D142 K144 N147 D160 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=1.5uM remove_due_to_license_issue IC50=1500nM Q16539 16169718 362 RPTFYRQELNKTIWEVPERYQNLSPVGGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1zyr C 3.0 BS01 STD D 1 A423 F425 R428 A423 F425 R428 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue Q8RQE9 16122422 1525 MEIKRFGRIREVIPLPPLTEIQVESYRRALQADVPPEKRENVGIQAAFRETFPIEEEDKGKGGLVLDFLEYRLGEPPFPQDECREKDLTYQAPLYARLQLIHKDTGLIKEDEVFLGHIPLMTEDGSFIINGADRVIVSQIHRSPGVYFTPDPARPGRYIASIIPLPKRGPWIDLEVEPNGVVSMKVNKRKFPLVLLLRVLGYDQETLARELGAYGELVQGLMDESVFAMRPEEALIRLFTLLRPGDPPKRDKAVAYVYGLIADPRRYDLGEAGRYKAEEKLGIRLSGRTLARFEDGEFKDEVFLPTLRYLFALTAGVPGHEVDDIDHLGNRRIRTVGELMTDQFRVGLARLARGVRERMLMGSEDSLTPAKLVNSRPLEAAIREFFSRSQLSQFKDETNPLSSLRHKRRISALGPGGLTRERAGFDVRDVHRTHYGRICPVETPEGANIGLITSLAAYARVDELGFIRTPYRRVVGGVVTDEVVYMTATEEDRYTIAQANTPLEGNRIAAERVVARRKGEPVIVSPEEVEFMDVSPKQVFSVNTNLIPFLEHDDANRALMGSNMQTQAVPLIRAQAPVVMTGLEERVVRDSLAALYAEEDGEVAKVDGNRIVVRYEDGRLVEYPLRRFYRSNQGTALDQRPRVVVGQRVRKGDLLADGPASENGFLALGQNVLVAIMPFDGYNFEDAIVISEELLKRDFYTSIHIERYEIEARDTKLGPERITRDIPHLSEAALRDLDEEGVVRIGAEVKPGDILVGRTSFKGESEPTPEERLLRSIFGEKARDVKDTSLRVPPGEGGIVVRTVRLRRGDPGVELKPGVREVVRVYVAQKRKLQVGDKLANRHGNKGVVAKILPVEDMPHLPDGTPVDVILNPLGVPSRMNLGQILETHLGLAGYFLGQRYISPIFDGAKEPEIKELLAQAFEVYFGKRKGEGFGVDKREVEVLRRAEKLGLVTPGKTPEEQLKELFLQGKVVLYDGRTGEPIEGPIVVGQMFIMKLYHMVEDKMHARSTGPYSLITQQPLGGKAQFGGQRFGEMEVWALEAYGAAHTLQEMLTLKSDDIEGRNAAYEAIIKGEDVPEPSVPESFRVLVKELQALALDVQTLDEKDNPVDIFEGLASKR 1zyr D 3.0 BS01 STD D 1 A1082 A1085 L1086 D1090 P1257 A969 A972 L973 D977 P1144 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0006351,0006360,0006366,0006383,0008270,0016779,0034062,0042793,0046872 remove_due_to_license_issue Q8RQE8 16122422 1525 KKEVRKVRIALASPEKIRSWSYGEVEKPETINYRTLKPERDGLFDERIFGPIKDYECACGKYKRQRFEGKVCERCGVEVTKSIVRRYRMGHIELATPAAHIWFVKDVPSKIGTLLDLSATELEQVLYFSKYIVLDPKGAILNGVPVEKRQLLTDEEYRELRYGKQETYPLPPGVDALVKDGEEVVKGQELAPGVVSRLDGVALYRFPRRVRVEYVKKERAGLRLPLAAWVEKEAYKPGEILAELPEPYLFGDKIVAAIDPEEEVIAEAEGVVHLHEPASILVVKARVYPFEDDVEVSTGDRVAPGDVLADGGKVKSDVYGRVEVDLVRNVVRVVESYDIDARMGAEAIQQLLKELDLEALEKELLEEMKHPSRARRAKARKRLEVVRAFLDSGNRPEWMILEAVPVLPPDLRPMVQVDGGRFATSDLNDLYRRLINRNNRLKKLLAQGAPEIIIRNEKRMLQEAVDALLDNGRRGAPVTNPGSDRPLRSLTDILSGKQGRFRQNLLGKRVDYSGRSVIVVGPQLKLHQCGLPKRMALELFKPFLLKKMEEKGIAPNVKAARRMLERQRDIKDEVWDALEEVIHGKVVLLNRAPTLHRLGIQAFQPVLVEGQSIQLHPLVCEAFNADFDGDQMAVHVPLSSFAQAEARIQMLSAHNLLSPASGEPLAKPSRDIILGLYYITQVRKEKKGAGLEFATPEEALAAHERGEVALNAPIKVAGRETSVGRLKYVFANPDEALLAVAHGIVDLQDVVTVRYMGKRLETSPGRILFARIVAEAVEDEKVAWELIQLDVPQEKNSLKDLVYQAFLRLGMEKTARLLDALKYYGFTFSTTSGITIGIDDAVIPEEKKQYLEEADRKLLQIEQAYEMGFLTDRERYDQILQLWTETTEKVTQAVFKNFEENYPFNPLYVMAQSGARGNPQQIRQLCGLRGLMQKPSGETFEVPVRSSFREGLTVLEYFISSHGARKGGADTALRTADSGYLTRKLVDVTHEIVVREADCGTTNYISVPLFQPDEVTRSLRLRKRADIEAGLYGRVLAREVEVLGVRLEEGRYLSMDDVHLLIKAAEAGEIQEVPVRSPLTCQTRYGVCQKCYGYDLSMARPVSIGEAVGIVAAQSIGEPGTQLTMRTFHTGGVAGAADITQGLPRVIELFEARRPKAKAVISEIDGVVRIEETEEKLSVFVESEGFSKEYKLPKEARLLVKDGDYVEAGQPLTRGAIDPHQLLEAKGPEAVERYLVEEIQKVYRAQGVKLHDKHIEIVVRQMMKYVEVTDPGDSRLLEGQVLEKWDVEALNERLIAEGKTPVAWKPLLMGVTKSALSTKSWLSAASFQNTTHVLTEAAIAGKKDELIGLKENVILGRLIPAGTGSDFVRFTQVVDQKTLKAIEEARKEAVEA 1zz1 A 1.57 BS02 SHH A 1 D98 I100 H142 H143 F152 D180 H182 F208 Y312 D97 I99 H141 H142 F151 D179 H181 F207 Y311 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.95uM remove_due_to_license_issue Ki=1000nM, Kd=300nM, IC50=1000nM Q70I53 16242151 2452 AIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADI 1zz2 A 2.0 BS01 B11 A 1 Y35 V38 A51 K53 L75 I84 L104 V105 T106 D150 S154 N155 L167 D168 L171 Y31 V34 A47 K49 L71 I80 L100 V101 T102 D146 S150 N151 L163 D164 L167 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=6uM remove_due_to_license_issue IC50=6000nM Q16539 16169718 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 1zz3 A 1.76 BS01 3YP A 1 H142 H143 G151 F152 D180 H182 F208 Y312 H141 H142 G150 F151 D179 H181 F207 Y311 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.29uM remove_due_to_license_issue Q70I53 16242151 1452 AIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADI 1zzi A 1.8 BS01 dna C 0 G26 S27 I29 G30 K31 G32 G33 R40 E51 R59 Y84 S85 G19 S20 I22 G23 K24 G25 G26 R33 E44 R52 Y77 S78 ? 0003676,0003723 remove_due_to_license_issue P61978 16004877 1 ~ 6 GAMGPIITTQVTIPKDLAGSIIGKGGQRIKQIRHESGASIKIDEPLEGSEDRIITITGTQDQIQNAQYLLQNSVKQYSGKFF 1zzi B 1.8 BS01 dna D 0 G26 S27 I29 G30 K31 G32 I36 R40 R59 Y84 S85 G16 S17 I19 G20 K21 G22 I26 R30 R49 Y74 S75 ? 0003676,0003723 remove_due_to_license_issue P61978 16004877 1 ~ 6 GPIITTQVTIPKDLAGSIIGKGGQRIKQIRHESGASIKIDEPLEGSEDRIITITGTQDQIQNAQYLLQNSVKQYSGKFF 1zzl A 2.0 BS01 TZY A 1 Y35 A51 K53 L104 V105 T106 L108 M109 G110 Y32 A48 K50 L101 V102 T103 L105 M106 G107 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=5nM remove_due_to_license_issue IC50=5nM Q16539 16134941 999 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 1zzz A 1.9 BS01 0IV A 1 H57 D189 S190 C191 S195 S214 W215 G216 S217 G219 H40 D171 S172 C173 S177 S192 W193 G194 S195 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004252,0006508 remove_due_to_license_issue P00760 9724521 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 220l A 1.85 BS01 BNZ A 1 A102 M106 V111 F114 L133 F153 A102 M106 V111 F114 L133 F153 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=0.4mM remove_due_to_license_issue P00720 9514755 169 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINAVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYK 223l A 1.9 BS01 BNZ A 1 M102 S117 L121 F153 M102 S117 L121 F153 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=0.4mM remove_due_to_license_issue P00720 9514755 169 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNGAKSRWYNQTPNRAKRVITTFRTGTWDAYK 2a0c X 1.95 BS01 CK9 X 1 I10 G11 V18 A31 F80 L83 H84 K89 N132 L134 I10 G11 V18 A31 F76 L79 H80 K85 N128 L130 N132 D145 T158 N128 D141 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 16003486 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2a0i A 2.72 BS01 dna B 0 M1 M2 S3 I4 A5 S12 A13 F16 S85 A86 P87 K88 H146 S149 R150 Q155 H157 H159 I186 E187 Y190 Q193 R201 H221 M223 R237 S238 R242 L251 R254 D255 K265 M1 M2 S3 I4 A5 S12 A13 F16 S79 A80 P81 K82 H133 S136 R137 Q142 H144 H146 I173 E174 Y177 Q180 R188 H208 M210 R224 S225 R229 L238 R241 D242 K252 3.6.4.12,5.6.2.1 remove_due_to_license_issue P14565 16216584 1 ~ 10 MMSIAQVRSAGSAGNFYTDVLGSGERWAGRGAEQLGLQGSVDKDVFTRLLEGRLPDGADLSRMQDGSNRHRPGYDLTFSAPKSVSMMAMLGGDKRLIDAHNQAVDFAVRQVEALASTRVTVLTGNLVMALFNHDTSRDQEPQLHTHAVVANVTQHNGEWKTLSSDKVGKTGFIENVYANQIAFGRLYREKLKEQVEALGYETEVVGKHGMWEMPGVPVEAFSGRSQTIREAVGEDASLKSRDVAALDTRKSKQHVDPEIKMAEWMQTLKETGFDIRAYRDAADQRADLRTLTP 2a14 A 1.7 BS01 SAH A 1 Y11 Y20 Y25 G63 S64 G65 T67 Y69 D85 F86 T87 N90 D142 V143 L163 L164 A165 A169 Y7 Y16 Y21 G59 S60 G61 T63 Y65 D81 F82 T83 N86 D138 V139 L159 L160 A161 A165 2.1.1.49,2.1.1.96 0004790,0005515,0005737,0005829,0008168,0008170,0008757,0009308,0009636,0030748,0032259 remove_due_to_license_issue Ki=2000nM O95050 4001 FTGGDEYQKHFLPRDYLATYYSFDGSPSPEAEMLKFNLECLHKTFGPGGLQGDTLIDIGSGPTIYQVLAACDSFQDITLSDFTDRNREELEKWLKKEPGAYDWTPAVKFACELEGNSGRWEEKEEKLRAAVKRVLKCDVHLGNPLAPAVLPLADCVLTLLAMECACCSLDAYRAALCNLASLLKPGGHLVTTVTLRLPSYMVGKREFSCVALEKGEVEQAVLDAGFDIEQLLHSPQSYSVTNAANNGVCCIVARKKP 2a29 A -1.00 BS01 ANP A 1 D344 E348 G349 F377 A379 R382 S384 K395 L431 D29 E33 G34 F62 A64 R67 S69 K80 L116 7.2.2.6 0000166,0005524,0006813,0008556,0016020 remove_due_to_license_issue P03960 16354672 1001 NRQASEFIPAQGVDEKTLADAAQLASLADETPEGRSIVILAKQRFNLRERDVQSLHATFVPFTAQSRMSGINIDNRMIRKGSVDAIRRHVEANGGHFPTDVDQKVDQVARQGATPLVVVEGSRVLGVIALKDIVKG 2a2g A 2.9 BS01 LEO A 1 F54 L105 Y120 F54 L105 Y120 ? 0036094 remove_due_to_license_issue P02761 10089305 201 EEASSTRGNLDVAKLNGDWFSIVVASNKREKIEENGSMRVFMQHIDVLENSLGFKFRIKENGECRELYLVAYKTPEDGEYFVEYDGGNTFTILKTDYDRYVMFHLINFKNGETFQLMVLYGRTKDLSSDIKEKFAKLCEAHGITRDNIIDLTKTDRCL 2a2x H 2.44 BS02 NA9 H 1 W60D L99 D189 A190 S214 W215 G216 E217 G219 W50 L96 D192 A193 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=20.2nM remove_due_to_license_issue IC50=20.2nM P00734 16460939 501 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2a3a A 2.1 BS01 TEP A 1 F76 G136 E177 M243 Y245 W384 F38 G98 E139 M205 Y207 W346 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 ic50=1500uM remove_due_to_license_issue IC50=1500000nM Q873X9 16183021 1433 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQ 2a3a A 2.1 BS02 TEP A 2 W52 Y139 W14 Y101 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 ic50=1500uM remove_due_to_license_issue IC50=1500000nM Q873X9 16183021 1434 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQ 2a3a A 2.1 BS03 TEP A 3 F251 R301 F213 R263 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 ic50=1500uM remove_due_to_license_issue IC50=1500000nM Q873X9 16183021 1436 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQ 2a3c A 2.07 BS01 PNX A 1 W52 F76 G136 W137 D175 M243 Y245 W384 W14 F38 G98 W99 D137 M205 Y207 W346 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 Kd=43uM remove_due_to_license_issue Kd=43000nM, Ki=37000nM, IC50=126000nM Q873X9 16183021 1434 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQT 2a3c A 2.07 BS02 PNX A 2 W137 Y178 D246 A248 G249 F251 R301 W99 Y140 D208 A210 G211 F213 R263 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 Kd=43uM remove_due_to_license_issue Kd=43000nM, Ki=37000nM, IC50=126000nM Q873X9 16183021 1435 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQT 2a3w A 2.2 BS03 CPJ A 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 ic50=3.8uM remove_due_to_license_issue P02743 16036920 341 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2a3w J 2.2 BS01 CPJ A 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 remove_due_to_license_issue P02743 16036920 341 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2a3x D 3.0 BS03 CPK I 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 remove_due_to_license_issue P02743 16036920 401 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2a3x I 3.0 BS03 CPK I 1 N59 Y74 E136 Q148 N59 Y74 E136 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 remove_due_to_license_issue P02743 16036920 401 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2a4g A 2.5 BS04 UNH A 1 Q41 T42 H57 R123 K136 G137 S139 R155 A156 A157 D168 Q41 T42 H57 R123 K136 G137 S139 R155 A156 A157 D168 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P26664 16087332 401 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2a4l A 2.4 BS01 RRC A 1 I10 A31 F82 L83 H84 K89 L134 D145 I10 A31 F70 L71 H72 K77 L122 D133 D127 K129 Q131 N132 D145 T158 T165 D115 K117 Q119 N120 D133 T146 T153 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.4uM remove_due_to_license_issue IC50=700nM, Kd=3400nM, Ki=250nM P24941 9030780 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2a4m C 2.3 BS01 TRP C 1 R30 Q64 Q154 R10 Q44 Q134 E133 K215 K218 E113 K195 K198 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0006412,0006418,0006436 Kd=30uM remove_due_to_license_issue Q9RVD6 15998643 500 ARPRVLTGDRPTGALHLGHLAGSLQNRVRLQDEAELFVLLADVQALTDHFDRPEQVRENVLAVALDYLAAGLDPQKTTCVVQSAVPELAELTVYFLNLVTVSHLRQNPTVKAEIAQKGYGERVPAGFFVYPVSQAADIAAFGATLVPVGDDQLPMLEQTREIVRRFNALYAPVLAEPQAQLSRVPRLPGLDGQAKMSKSLGNAIALGDSADEVARKVMGMYTDPGHLRASDPGRVEGNPVFTFLDAFDPDPARVQALKDQYRAGGLGDVKVKKHLIDVLNGVLAPIRTRRAEYERDPDAVLRFVTEGTARGREVAAQTLGQVRRAMRLFGH 2a4q A 2.45 BS04 FNH A 1 Q41 T42 H57 K136 G137 S139 R155 A156 A157 C159 D168 Q41 T42 H57 K136 G137 S139 R155 A156 A157 C159 D168 H57 D81 G137 S139 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036,0097264 remove_due_to_license_issue Q91RS4 16112859 401 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2a4r A 2.4 BS04 BNH A 1 Q41 T42 H57 R123 I132 K136 G137 S139 R155 A156 A157 C159 Q41 T42 H57 R123 I132 K136 G137 S139 R155 A156 A157 C159 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 16112862 401 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2a4w A 1.5 BS01 BLM A 1 V107 W108 G109 Y112 V106 W107 G108 Y111 ? remove_due_to_license_issue O05205 16756991 750 SARISLFAVVVEDMAKSLEFYRKLGVEIPAEADSAPHTEAVLDGGIRLAWDTVETVRSYDPEWQAPTGGHRFAIAFEFPDTASVDKKYAELVDAGYEGHLKPWNAVWGQRYAIVKDPDGNVVDLFAPL 2a4w B 1.5 BS01 BLM A 1 H238 D252 Y260 H37 D51 Y59 ? remove_due_to_license_issue O05205 16756991 750 SARISLFAVVVEDMAKSLEFYRKLGVEIPAEADSAPHTEAVLDGGIRLAWDTVETVRSYDPEWQAPTGGHRFAIAFEFPDTASVDKKYAELVDAGYEGHLKPWNAVWGQRYAIVKDPDGNVVDLFAPLPL 2a4z A 2.9 BS01 BYM A 1 K833 Y867 I879 V882 M953 I963 D964 K573 Y607 I619 V622 M693 I703 D704 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 16127437 101 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHSQTIKVSPDDTPGAILQSFFTEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISFNADKLTSATNPDKENSMSISILLDNYCHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 2a58 A 2.8 BS01 RBF A 1 S62 W63 E64 V86 L87 H94 S50 W51 E52 V74 L75 H82 H94 H82 2.5.1.78 0000906,0004746,0005515,0005634,0005737,0005758,0009231,0009349,0016740,1902444 remove_due_to_license_issue Q9UUB1 15265040 300 LKGPELRILIVHARYNLQAIEPLVKGAVETMIEKHDVKLENIDIESVPGSWELPQGIRASIARNTYDAVIGIGVLIKGSTMHFEYISEAVVHGLMRVGLDSGVPVILGLLTVLNEEQALYRAGLNGGHNHGNDWGSAAVEMGLKAL 2a58 E 2.8 BS01 RBF E 1 S62 W63 E64 V86 L87 H94 S50 W51 E52 V74 L75 H82 H94 H82 2.5.1.78 0000906,0004746,0005515,0005634,0005737,0005758,0009231,0009349,0016740,1902444 remove_due_to_license_issue Q9UUB1 15265040 304 LKGPELRILIVHARYNLQAIEPLVKGAVETMIEKHDVKLENIDIESVPGSWELPQGIRASIARNTYDAVIGIGVLIKGSTMHFEYISEAVVHGLMRVGLDSGVPVILGLLTVLNEEQALYRAGLNGGHNHGNDWGSAAVEMGLKAL 2a5b A 2.49 BS01 8HG A 1 T35 W70 F72 T77 T35 W70 F72 T77 ? 0005576,0009374,0019731 Kd=117uM remove_due_to_license_issue P02701 16413579 255 ARKCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYTTAVTATSNEIKESPLHGTENTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRLR 2a5c A 2.5 BS01 8DA A 1 L14 W70 T77 N118 L14 W70 T77 N118 ? 0005576,0009374,0019731 Kd=24uM remove_due_to_license_issue P02701 16413579 303 ARKCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYTTAVTATSNEIKESPLHGTENTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 2a5s A 1.7 BS01 GLU A 1 H88 T116 R121 G172 S173 T174 Y214 D215 H81 T109 R114 G165 S166 T167 Y207 D208 ? 0015276,0016020 remove_due_to_license_issue Q00959 16281028 1001 NHLSIVTLEEAPFVIVEDIDPLETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGICH 2a5u A 2.7 BS01 QYT A 1 I831 K833 I879 I881 V882 M953 F961 I963 D964 I592 K594 I640 I642 V643 M713 F721 I723 D724 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=8.0nM P48736 16127437 101 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 2a66 A 2.2 BS01 dna B 0 Y96 H97 Y98 K107 K111 V156 R157 M161 R162 R165 N166 Y172 Y13 H14 Y15 K24 K28 V73 R74 M78 R79 R82 N83 Y89 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue O00482 16289203 201 ~ 212 ELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRYTCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRAL 2a66 A 2.2 BS02 dna C 0 E104 S105 R112 R135 K136 R142 R162 G163 G164 E21 S22 R29 R52 K53 R59 R79 G80 G81 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue O00482 16289203 301 ~ 312 ELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRYTCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRAL 2a8g B 1.99 BS01 GNG B 1 S16 Y33 W70 F72 T77 W97 N118 S14 Y31 W68 F70 T75 W95 N116 ? 0005576,0009374,0019731 Kd=205uM remove_due_to_license_issue P02701 16413579 201 KCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYTTAVTATSNEIKESPLHGTENTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 2a8h A 2.3 BS02 4NH A 1 T347 E398 L401 H405 E406 H409 H415 P437 A439 V440 T131 E182 L185 H189 E190 H193 H199 P221 A223 V224 3.4.24.86 0004222,0006508,0008237 ic50=67nM remove_due_to_license_issue IC50=67nM P78536 16426848 158 DPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYVGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERSN 2aa6 A 1.95 BS01 STR A 1 L769 N770 Q776 M807 F829 M845 M852 F941 C942 T945 L48 N49 Q55 M86 F108 M124 M131 F219 C220 T223 ? remove_due_to_license_issue IC50=14nM, Kd=0.390000nM P08235 15967794 401 ALVPQLSTISRALTPSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKCNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFH 2aa9 A 1.5 BS01 SKM A 1 K22 S23 R27 T97 Q171 Y200 D313 K340 K22 S23 R27 T97 Q171 Y200 D313 K340 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 remove_due_to_license_issue IC50=>90000000nM P0A6D3 16225867 501 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 2aac B 1.6 BS01 FCB B 1 P8 L9 F15 T24 R38 Y82 H93 W95 P3 L4 F10 T19 R33 Y77 H88 W90 ? 0006355 Kd=6mM remove_due_to_license_issue P0A9E0 9367758 179 NDPLLPGYSFNAHLVAGLTPIEANGYLDFFIDRPLGMKGYILNLTIRGQGVVKNQGREFVCRPGDILLFPPGEIHHYGRHPEAREWYHQWVYFRPRAYWHEWLNWPSIFANTGFFRPDEAHQPHFSDLFGQIINAGQGEGRYSELLAINLLEQLLLRRMEAIN 2aay A 1.55 BS01 SKM A 1 K22 S23 R27 T97 Q171 Y200 D313 K340 K22 S23 R27 T97 Q171 Y200 D313 K340 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 ic50=1.2mM remove_due_to_license_issue IC50=>90000000nM P0A6D3 16225867 701 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 2ac0 A 1.8 BS01 dna E 0 A119 K120 S121 R248 A26 K27 S28 R155 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ac0 A 1.8 BS02 dna F 0 S241 R248 R273 C275 A276 R280 S148 R155 R180 C182 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ac0 B 1.8 BS01 dna E 0 S241 R248 R273 C275 A276 C277 R280 S148 R155 R180 C182 A183 C184 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ac0 B 1.8 BS02 dna F 0 T118 K120 G279 R280 R283 T25 K27 G186 R187 R190 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ac0 C 1.8 BS01 dna G 0 S241 R248 R273 C275 A276 C277 R280 S146 R153 R178 C180 A181 C182 R185 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLR 2ac0 C 1.8 BS02 dna H 0 A119 K120 S121 A24 K25 S26 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLR 2ac0 D 1.8 BS01 dna G 0 A119 K120 A24 K25 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRKKG 2ac0 D 1.8 BS02 dna H 0 S241 R248 R273 C275 A276 R280 S146 R153 R178 C180 A181 R185 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRKKG 2ad5 A 2.8 BS03 CTP A 1 S14 D147 I148 E149 S14 D147 I148 E149 6.3.4.2 0000287,0003883,0004359,0005524,0005737,0005829,0006221,0006241,0016874,0019856,0032991,0042802,0044210,0046872,0051289,0097268 remove_due_to_license_issue P0A7E5 16216072 602 MTTNYIFVTGGVVSSLGKGIAAASLAAILEARGLNVTIMKLDPYINVDPGTMSPIQHGEVFVTEDGAETDLDLGHYERFIRTKMSRRNNFTTGRIYSDVLRKERRGDYLGATVQVIPHITNAIKERVLEGGEGHDVVLVEIGGTVGDIESLPFLEAIRQMAVEIGREHTLFMHLTLVPYMAASGEVKTKPTQHSVKELLSIGIQPDILICRSDRAVPANERAKIALFCNVPEKAVISLKDVDSIYKIPGLLKSQGLDDYICKRFSLNCPEANLSEWEQVIFEEANPVSEVTIGMVGKYIELPDAYKSVIEALKHGGLKNRVSVNIKLIDSQDVETRGVEILKGLDAILVPGGFGYRGVEGMITTARFARENNIPYLGICLGMQVALIDYARHVANMENANSTEFVPDCKYPVVALITEWRDENGNVETMRLGAQQCQLVDDSLVRQLYNAPTIVERHRHRYEVNNMLLKQIEDAGLRVAGRSGDDQLVEIIEVPNHPWFVACQFHPEFTSTPRDGHPLFAGFVKAASEFQKRQA 2ad5 A 2.8 BS04 CTP B 1 K187 T188 K189 Q192 K223 K187 T188 K189 Q192 K223 6.3.4.2 0000287,0003883,0004359,0005524,0005737,0005829,0006221,0006241,0016874,0019856,0032991,0042802,0044210,0046872,0051289,0097268 remove_due_to_license_issue P0A7E5 16216072 1602 MTTNYIFVTGGVVSSLGKGIAAASLAAILEARGLNVTIMKLDPYINVDPGTMSPIQHGEVFVTEDGAETDLDLGHYERFIRTKMSRRNNFTTGRIYSDVLRKERRGDYLGATVQVIPHITNAIKERVLEGGEGHDVVLVEIGGTVGDIESLPFLEAIRQMAVEIGREHTLFMHLTLVPYMAASGEVKTKPTQHSVKELLSIGIQPDILICRSDRAVPANERAKIALFCNVPEKAVISLKDVDSIYKIPGLLKSQGLDDYICKRFSLNCPEANLSEWEQVIFEEANPVSEVTIGMVGKYIELPDAYKSVIEALKHGGLKNRVSVNIKLIDSQDVETRGVEILKGLDAILVPGGFGYRGVEGMITTARFARENNIPYLGICLGMQVALIDYARHVANMENANSTEFVPDCKYPVVALITEWRDENGNVETMRLGAQQCQLVDDSLVRQLYNAPTIVERHRHRYEVNNMLLKQIEDAGLRVAGRSGDDQLVEIIEVPNHPWFVACQFHPEFTSTPRDGHPLFAGFVKAASEFQKRQA 2ad5 B 2.8 BS01 CTP A 1 K187 T188 K189 Q192 K223 K187 T188 K189 Q192 K223 6.3.4.2 0000287,0003883,0004359,0005524,0005737,0005829,0006221,0006241,0016874,0019856,0032991,0042802,0044210,0046872,0051289,0097268 remove_due_to_license_issue P0A7E5 16216072 602 MTTNYIFVTGGVVSSLGKGIAAASLAAILEARGLNVTIMKLDPYINVDPGTMSPIQHGEVFVTEDGAETDLDLGHYERFIRTKMSRRNNFTTGRIYSDVLRKERRGDYLGATVQVIPHITNAIKERVLEGGEGHDVVLVEIGGTVGDIESLPFLEAIRQMAVEIGREHTLFMHLTLVPYMAASGEVKTKPTQHSVKELLSIGIQPDILICRSDRAVPANERAKIALFCNVPEKAVISLKDVDSIYKIPGLLKSQGLDDYICKRFSLNCPEANLSEWEQVIFEEANPVSEVTIGMVGKYIELPDAYKSVIEALKHGGLKNRVSVNIKLIDSQDVETRGVEILKGLDAILVPGGFGYRGVEGMITTARFARENNIPYLGICLGMQVALIDYARHVANMENANSTEFVPDCKYPVVALITEWRDENGNVEVTMRLGAQQCQLVDDSLVRQLYNAPTIVERHRHRYEVNNMLLKQIEDAGLRVAGRSGDDQLVEIIEVPNHPWFVACQFHPEFTSTPRDGHPLFAGFVKAASEFQKRQAK 2ad5 B 2.8 BS04 CTP B 1 S14 D147 I148 E149 S14 D147 I148 E149 6.3.4.2 0000287,0003883,0004359,0005524,0005737,0005829,0006221,0006241,0016874,0019856,0032991,0042802,0044210,0046872,0051289,0097268 remove_due_to_license_issue P0A7E5 16216072 1602 MTTNYIFVTGGVVSSLGKGIAAASLAAILEARGLNVTIMKLDPYINVDPGTMSPIQHGEVFVTEDGAETDLDLGHYERFIRTKMSRRNNFTTGRIYSDVLRKERRGDYLGATVQVIPHITNAIKERVLEGGEGHDVVLVEIGGTVGDIESLPFLEAIRQMAVEIGREHTLFMHLTLVPYMAASGEVKTKPTQHSVKELLSIGIQPDILICRSDRAVPANERAKIALFCNVPEKAVISLKDVDSIYKIPGLLKSQGLDDYICKRFSLNCPEANLSEWEQVIFEEANPVSEVTIGMVGKYIELPDAYKSVIEALKHGGLKNRVSVNIKLIDSQDVETRGVEILKGLDAILVPGGFGYRGVEGMITTARFARENNIPYLGICLGMQVALIDYARHVANMENANSTEFVPDCKYPVVALITEWRDENGNVEVTMRLGAQQCQLVDDSLVRQLYNAPTIVERHRHRYEVNNMLLKQIEDAGLRVAGRSGDDQLVEIIEVPNHPWFVACQFHPEFTSTPRDGHPLFAGFVKAASEFQKRQAK 2ada A 2.4 BS02 HPR A 1 H17 D19 F61 L62 F65 M155 A183 G184 H214 E217 D295 D296 H14 D16 F58 L59 F62 M152 A180 G181 H211 E214 D292 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0000255,0001666,0001701,0001829,0001889,0001890,0002314,0002467,0002636,0002686,0002901,0002906,0004000,0005737,0005764,0005829,0005886,0006154,0006157,0006196,0006915,0006939,0007155,0008270,0009117,0009168,0009897,0009986,0010460,0014074,0016020,0016787,0019239,0019722,0030217,0030324,0030890,0031410,0032261,0032263,0032264,0033077,0033089,0033632,0042100,0042110,0043066,0043084,0043605,0044209,0045580,0045582,0045987,0046059,0046061,0046085,0046101,0046103,0046111,0046632,0046638,0046872,0046936,0048286,0048541,0048566,0050728,0050850,0050852,0050862,0050870,0050900,0060169,0060205,0060407,0070161,0070242,0070244,0070254,0070256,0140928 Ki~0.1pM remove_due_to_license_issue P03958 1925539 353 TPAFNKPKVELHVHLDGAIKPETILYFGKKRGIALPADTVEELRNIIGMDKPLSLPGFLAKFDYYMPVIAGCREAIKRIAYEFVEMKAKEGVVYVEVRYSPHLLANSKVDPMPWNQTEGDVTPDDVVDLVNQGLQEGEQAFGIKVRSILCCMRHQPSWSLEVLELCKKYNQKTVVAMDLAGDETIEGSSLFPGHVEAYEGAVKNGIHRTVHAGEVGSPEVVREAVDILKTERVGHGYHTIEDEALYNRLLKENMHFEVCPWSSYLTGAWDPKTTHAVVRFKNDKANYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEEEKKELLERLYREYQ 2adm B 2.6 BS01 SAM B 1 A47 P52 E71 I72 D89 N105 P107 A27 P32 E51 I52 D69 N85 P87 N105 P106 Y108 F196 N85 P86 Y88 F168 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 8995524 500 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTGYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSTLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2adu A 1.9 BS03 R20 A 1 F219 H231 D251 D262 H331 H339 Y444 E459 F96 H108 D128 D139 H208 H216 Y321 E336 D251 D262 H331 H339 E364 E459 D128 D139 H208 H216 E241 E336 3.4.11.18 0006508,0070006 Ki=18nM remove_due_to_license_issue IC50=18nM, Ki=18nM P50579 16134930 906 KVQTDPPSVPICDLYPNGVFPKGQECEYPEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 2ady A 2.5 BS01 dna E 0 K120 S121 R248 K26 S27 R154 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ady A 2.5 BS02 dna F 0 S241 R273 C275 A276 R280 S147 R179 C181 A182 R186 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ady B 2.5 BS01 dna E 0 S241 R248 R273 C275 A276 R280 S148 R155 R180 C182 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ady B 2.5 BS02 dna F 0 T118 A119 K120 R248 R283 T25 A26 K27 R155 R190 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2aeb A 1.29 BS03 ABH A 1 H101 D124 H126 D128 S137 H141 D183 D232 H97 D120 H122 D124 S133 H137 D179 D228 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=5nM remove_due_to_license_issue P05089 16141327 551 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 2aei H 2.52 BS02 03R H 1 H57 T98 P170I D189 S190 C191 K192 G193 S195 S214 W215 G216 Q217 G219 C220 H41 T86 P169 D186 S187 C188 K189 G190 S192 S211 W212 G213 Q214 G215 C216 3.4.21.21 0004252,0006508 remove_due_to_license_issue IC50=86.0nM P08709 16125385 500 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2ael B 2.5 BS03 SAZ B 1 T96 L97 F157 L187 M221 N225 Y295 W298 Y305 T95 L96 F156 L186 M220 N224 Y294 W297 Y304 Y93 T96 L97 D100 R182 K232 K304 Y305 Y92 T95 L96 D99 R181 K231 K303 Y304 4.2.3.6 0016106,0016829,0016838,0045482,0046872 Ki=0.51uM remove_due_to_license_issue P13513 16171386 704 ENFPTEYFLNTTVRLLEYIRYRDSNYTREERIENLHYAYNKAAHHFAQPRQQQLLKVDPKRLQASLQTIVGMVVYSWAKVSKECMADLSIHYTYTLVLDDSKDDPYPTMVNYFDDLQAGREQAHPWWALVNEHFPNVLRHFGPFCSLNLIRSTLDFFEGCWIEQYNFGGFPGSHDYPQFLRRMNGLGHCVGASLWPKEQFNERSLFLEITSAIAQMENWMVWVNDLMSFYKEFDDERDQISLVKNYVVSDEISLHEALEKLTQDTLHSSKQMVAVFSDKDPQVMDTIECFMHGYVTWHLCDRKYRLSEIYEKVKEEKTEDAQKFCKFYEQAANVGAVSPSEWAYPPVAQLANV 2afw A 1.56 BS02 AHN A 1 D159 E201 E202 D248 Q304 H330 D127 E163 E164 D210 Q266 H292 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Ki=17uM remove_due_to_license_issue Q16769 16135565 1501 ASAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPYGYRSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 2afx A 1.64 BS02 1BN A 1 D159 E201 E202 D248 Q304 F325 W329 H330 D127 E163 E164 D210 Q266 F287 W291 H292 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 remove_due_to_license_issue Ki=262nM Q16769 16135565 1501 ASAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPYGYRSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 2agv A 2.4 BS02 BHQ A 1 D59 L61 V62 L65 F256 P308 L311 P312 D59 L61 V62 L65 F256 P308 L311 P312 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 Kd=20nM remove_due_to_license_issue IC50=2000nM P04191 16150713 1004 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 2ahi A 1.85 BS01 dna E 0 A119 K120 S121 R248 A25 K26 S27 R154 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 10 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRKK 2ahi A 1.85 BS02 dna F 0 S241 R248 R273 C275 A276 R280 S147 R154 R179 C181 A182 R186 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 2 ~ 12 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRKK 2ahi B 1.85 BS01 dna E 0 S241 R248 R273 C275 A276 R280 S148 R155 R180 C182 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 10 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ahi B 1.85 BS02 dna F 0 K120 R248 K27 R155 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 2 ~ 12 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ahi C 1.85 BS01 dna G 0 S241 R273 C275 A276 R280 S146 R178 C180 A181 R185 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEEN 2ahi D 1.85 BS01 dna G 0 A119 K120 R248 A24 K25 R153 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ahi D 1.85 BS02 dna H 0 S241 R248 R273 C275 A276 R280 S146 R153 R178 C180 A181 R185 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ai7 A 2.0 BS01 SB7 A 1 G71 Q76 E128 C130 L131 H173 E174 H177 G71 Q76 E119 C121 L122 H164 E165 H168 G71 Q76 C130 L131 H173 E174 H177 G71 Q76 C121 L122 H164 E165 H168 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=0.4uM remove_due_to_license_issue Q8DP79 12538898 300 SAIERISKAAHLIDMCDIIREGNPSLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNIEAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLILE 2ai8 A 1.7 BS01 SB7 A 1 I44 G45 Q50 E88 G89 L91 H132 E133 H136 I44 G45 Q50 E88 G89 L91 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 G45 Q50 C90 L91 H132 E133 H136 3.5.1.88 0005515,0005829,0006412,0008198,0008270,0016787,0042586,0043022,0043686,0046872 ic50=0.16uM remove_due_to_license_issue P0A6K3 12538898 501 SVLQVLHIPDERLRKVAKPVEEVNAEIQRIVDDMFETMYAEEGIGLAATQVDIHQRIIVIDVSENRDERLVLINPELLEKSGETGIEEGCLSIPEQRALVPRAEKVKIRALDRDGKPFELEADGLLAICIQHEMDHLVGKLFMDYLSPLKQQRIRQKVEKLDRLKA 2aia A 1.7 BS01 SB8 A 1 G71 Q76 L123 G126 E128 G129 C130 L131 Y166 V170 H173 E174 H177 G71 Q76 L113 G116 E117 G118 C119 L120 Y155 V159 H162 E163 H166 G71 Q76 C130 L131 H173 E174 H177 G71 Q76 C119 L120 H162 E163 H166 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=3.9uM remove_due_to_license_issue IC50=3900nM Q8DP79 12538898 501 SAIERISKAAHLIDMCDIIREGNPSLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLILE 2aie P 1.7 BS01 SB9 P 1 G71 Q76 L123 E128 C130 L131 Y166 H173 E174 H177 G71 Q76 L115 E119 C121 L122 Y157 H164 E165 H168 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=2.2uM remove_due_to_license_issue IC50=2200nM Q8DP79 12538898 501 SAIERIVKAAHLIDMCDIIREGNPSLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNIEAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLILE 2aig P 2.6 BS01 0GR P 1 G105 K106 I107 I108 T139 H142 E143 I165 R167 P168 G169 L170 G104 K105 I106 I107 T138 H141 E142 I164 R166 P167 G168 L169 3.4.24.46 0004222,0005576,0005886,0006508,0008237,0046872 remove_due_to_license_issue P34179 9521103 203 NLPQRYIELVVVADRRVFMKYNSDLNIIRTRVHEIVNIINEFYRSLNIRVSLTDLEIWSGQDFITIQSSSSNTLNSFGEWRERVLLTRKRHDNAQLLTAINFEGKIIGKAYTSSMCNPRSSVGIVKDHSPINLLVAVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTPGRSYEFSDDSMGYYQKFLNQYKPQCILNKP 2aj8 A 2.11 BS01 SC3 A 1 E205 E206 Y547 S630 Y631 V656 Y662 Y666 V711 E167 E168 Y509 S592 Y593 V618 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 Ki=638nM remove_due_to_license_issue P22411 16330047 1601 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 2aj8 A 2.11 BS02 SC3 A 2 W187 A280 S281 W149 A242 S243 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 Ki=638nM remove_due_to_license_issue P22411 16330047 1608 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 2ajb A 2.75 BS01 0QG A 1 R125 E205 E206 Y547 S630 Y631 Y662 Y666 N710 H740 R87 E167 E168 Y509 S592 Y593 Y624 Y628 N672 H702 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P22411 16330047 802 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 2ajd A 2.56 BS01 BPR A 1 E205 E206 Y547 S630 Y631 Y662 Y666 H740 E167 E168 Y509 S592 Y593 Y624 Y628 H702 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P22411 16330047 801 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 2ajl I 2.5 BS01 JNH I 1 E205 E206 S209 F357 Y547 S630 Y631 Y662 Y666 E165 E166 S169 F317 Y507 S590 Y591 Y622 Y626 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 16236500 1 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2al5 A 1.65 BS01 FWD A 1 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y59 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 remove_due_to_license_issue Ki=4nM, EC50=460nM P19491 16192394 901 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 2alv A 1.9 BS01 CY6 A 1 T26 H41 F140 L141 N142 G143 C145 H163 H164 M165 E166 P168 D187 Q189 T190 A191 Q192 T25 H40 F139 L140 N141 G142 C144 H162 H163 M164 E165 P167 D186 Q188 T189 A190 Q191 H41 G143 C145 H40 G142 C144 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue IC50=800000nM P0C6X7 16250632 1145 GFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGV 2am1 A 2.5 BS01 1LG A 1 F31 D32 R34 A48 F54 Y135 G140 N326 N328 P329 T330 A331 L334 L367 F31 D32 R34 A48 F54 Y135 G140 N326 N328 P329 T330 A331 L334 L367 6.3.2.10 0005524,0005737,0008360,0008766,0009058,0009252,0016874,0016881,0047480,0051301,0071555 ic50=1uM remove_due_to_license_issue IC50=1000nM Q8DNV6 16322581 1000 MKLTIHEIAQVVGAKNDISIFEDTQLEKAEFDSRLIGTGDLFVPLKGARDGHDFIETAFENGAAVTLSEKEVSNHPYILVDDVLTAFQSLASYYLEKTTVDVFAVTGSNGKTTTKDMLAHLLSTRYKTYKTQGNYNNEIGLPYTVLHMPEGTEKLVLEMGQDHLGDIHLLSELARPKTAIVTLVGEAHLAFFKDRSEIAKGKMQIADGMASGSLLLAPADPIVEDYLPIDKKVVRFGQGAELEITDLVERKDSLTFKANFLEQALDLPVTGKYNATNAMIASYVALQEGVSEEQIRLAFQHLELTRNRTEWKKAANGADILSDVYNANPTAMKLILETFSAIPANEGGKKIAVLADMKELGDQSVQLHNQMILSLSPDVLDIVIFYGEDIAQLAQLASQMFPIGHVYYFKKTEDQDQFEDLVKQVKESLGAHDQILLKGSNSMNLAKLVESLEN 2am2 A 2.8 BS01 2LG A 1 F31 R34 A48 R49 Y135 N137 N326 N328 T330 L367 F31 R34 A48 R49 Y135 N137 N326 N328 T330 L367 6.3.2.10 0005524,0005737,0008360,0008766,0009058,0009252,0016874,0016881,0047480,0051301,0071555 remove_due_to_license_issue IC50=8000nM Q8DNV6 16322581 1000 MKLTIHEIAQVVGAKNDISIFEDTQLEKAEFDSRLIGTGDLFVPLKGARDGHDFIETAFENGAAVTLSEKEVSNHPYILVDDVLTAFQSLASYYLEKTTVDVFAVTGSNGKTTTKDMLAHLLSTRYKTYKTQGNYNNEIGLPYTVLHMPEGTEKLVLEMGQDHLGDIHLLSELARPKTAIVTLVGEAHLAFFKDRSEIAKGKMQIADGMASGSLLLAPADPIVEDYLPIDKKVVRFGQGAELEITDLVERKDSLTFKANFLEQALDLPVTGKYNATNAMIASYVALQEGVSEEQIRLAFQHLELTRNRTEWKKAANGADILSDVYNANPTAMKLILETFSAIPANEGGKKIAVLADMKELGDQSVQLHNQMILSLSPDVLDIVIFYGEDIAQLAQLASQMFPIGHVYYFKKTEDQDQFEDLVKQVKESLGAHDQILLKGSNSMNLAKLVESLEN 2am4 A 1.7 BS01 U2F A 1 I113 A114 C115 R117 D144 C145 Y184 I187 H190 E211 D212 D291 G320 V321 S322 I8 A9 C10 R12 D39 C40 Y79 I82 H85 E106 D107 D186 G215 V216 S217 D213 D291 D108 D186 2.4.1.101 0006486,0008375 Ki=190uM remove_due_to_license_issue P27115 16769084 449 AVIPILVIACDRSTVRRCLDKLLHYRPSAELFPIIVSQDCGHEETAQVIASYGSAVTHIRQPDLSNIAVQPDHRKFQGYYKIARHYRWALGQIFHNFNYPAAVVVEDDLEVAPDFFEYFQATYPLLKADPSLWCVSAWNDNGKEQMVDSSKPELLYRTDFFPGLGWLLLAELWAELEPKWPKAFWDDWMRRPEQRKGRACVRPEISRTMTFGRKGVSHGQFFDQHLKFIKLNQQFVPFTQLDLSYLQQEAYDRDFLARVYGAPQLQVEKVRTNDRKELGEVRVQYTGRDSFKAFAKALGVMDDLKSGVPRAGYRGIVTFLFRGRRVHLAPPQTWDGYDPSWT 2am9 A 1.64 BS01 TES A 1 L704 N705 M745 M749 F764 T877 M895 L35 N36 M76 M80 F95 T208 M226 ? remove_due_to_license_issue IC50=2.7nM, Ki=3.2nM, EC50=1.1nM P10275 16641486 1000 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ama A 1.9 BS01 DHT A 1 L704 N705 M745 M749 F764 T877 M895 L34 N35 M75 M79 F94 T201 M219 ? remove_due_to_license_issue IC50=>10000nM, EC50=6nM, Ki=0.2nM P10275 16641486 1001 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIATSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2amt A 2.3 BS02 1AA A 1 H34 D56 I57 G58 F61 P62 H34 D56 I57 G58 F61 P62 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=36uM remove_due_to_license_issue P62617 16392111 1901 MRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 2amt A 2.3 BS04 1AA C 2 A100 K104 M105 L106 A131 T132 T133 E135 A100 K104 M105 L106 A131 T132 T133 E135 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=36uM remove_due_to_license_issue P62617 16392111 3901 MRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 2amt B 2.3 BS01 1AA A 1 A100 K104 M105 L106 A131 T132 T133 E135 A100 K104 M105 L106 A131 T132 T133 E135 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 remove_due_to_license_issue P62617 16392111 1901 MRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 2amt B 2.3 BS04 1AA C 1 H34 S35 H42 D56 I57 G58 L76 H34 S35 H42 D56 I57 G58 L76 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 remove_due_to_license_issue P62617 16392111 2901 MRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 2amv A 2.3 BS02 BIN A 1 I68 Q71 Q72 Y75 R193 E195 F196 R309 R310 I56 Q59 Q60 Y63 R181 E183 F184 R297 R298 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=1.6nM remove_due_to_license_issue P00489 9384557 930 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKI 2an5 A 2.5 BS02 TTL A 1 Y35 R44 K57 F182 E219 V269 Y13 R22 K35 F160 E197 V247 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=2.1uM remove_due_to_license_issue P11086 16363801 1401 VASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2ank H 2.46 BS02 N12 H 1 L99 D189 A190 S195 S214 W215 G216 E217 G219 L96 D192 A193 S198 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=47.3nM remove_due_to_license_issue IC50=47.3nM P00734 16460939 501 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2anl A 3.3 BS01 JE2 A 1 D34 G36 Y77 G78 S79 L131 F192 D214 T217 V292 D34 G36 Y77 G78 S79 L131 F192 D214 T217 V292 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 ? 0004190,0006508 remove_due_to_license_issue O60990 16510971 3151 SENDVIELDDVANLMFYGEGEVGDNHQKFMLIFDTGSANLWVPSKKCNSIGCSTKHLYDSSKSKSYEKDGTKVEITYGSGTVRGFFSKDLVTLGYLSLPYKFIEVTDTDDLEPLYTAAEFDGILGLGWKDLSIGSIDPIVVELKNQNKIDQALFTFYLPVHDKHSGYLTIGGIEEKFYEGELTYEKLNHDLFWQVDLDVNFGKTSMEKANVIVDSGTSTITAPTSFINKFFKDLNVIKVPFLPFYITTCNNKDMPTLEFKSANNTYTLEPEYYMEPLLDIDDTLCMLYILPVDIDKNTFILGDPFMRKYFTVFDYDKESIGFAVAKN 2anm H 2.4 BS01 CDO H 1 H57 Y60A D189 A190 S195 W215 G216 E217 G219 H43 Y47 D192 A193 S198 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=1.8nM remove_due_to_license_issue IC50=1nM P00734 16460939 1001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2ans A 2.5 BS01 2AN A 1 F16 F57 R78 V115 C117 R126 Y128 F16 F57 R78 V115 C117 R126 Y128 ? 0005324,0005634,0005654,0005737,0008289,0009617,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0071285,0071356,0120162 Kd=1.2uM remove_due_to_license_issue P04117 10423455 201 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDLVTIRSESTFKNTEISFKLGVEFDEITADDRKVKSIITLDGGALVQVQKWDGKSTTIKRKRDGDKLVVECVMKGVTSTRVYERA 2ao6 A 1.89 BS02 R18 A 1 L704 N705 Q711 M745 M749 F764 T877 L34 N35 Q41 M75 M79 F94 T201 ? remove_due_to_license_issue Kd=0.99nM, IC50=0.302000nM, EC50=0.013000nM, Ki=0.400000nM P10275 15525515 1001 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIATSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 2aoc A 1.3 BS01 2NC B 1 R8 D25 G27 A28 D29 G48 I50 V82 R8 D25 G27 A28 D29 G48 I50 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16218957 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2aoc B 1.3 BS01 2NC B 1 D125 G127 A128 D129 D130 I147 G148 I150 V182 D25 G27 A28 D29 D30 I47 G48 I50 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16218957 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2aod A 1.4 BS01 2NC B 1 R8 D25 G27 A28 D29 D30 G48 V82 I84 R8 D25 G27 A28 D29 D30 G48 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16218957 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2aod B 1.4 BS01 2NC B 1 D125 G127 A128 D129 D130 I147 G148 P181 V182 D25 G27 A28 D29 D30 I47 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16218957 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2aoe A 1.54 BS01 0Q4 B 1 R8 D25 G27 A28 D29 G48 G49 P81 I84 R8 D25 G27 A28 D29 G48 G49 P81 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16218957 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2aoe B 1.54 BS01 0Q4 B 1 D125 G127 A128 D129 D130 M146 I147 G148 G149 I150 D25 G27 A28 D29 D30 M46 I47 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.024uM remove_due_to_license_issue P04587 16218957 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2aog A 1.1 BS01 2NC A 1 R8 D25 G27 A28 D29 G48 I50 I84 R8 D25 G27 A28 D29 G48 I50 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.53uM remove_due_to_license_issue P04587 16218957 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2aog B 1.1 BS01 2NC A 1 D125 G127 A128 D129 D130 I147 G148 G149 P181 D25 G27 A28 D29 D30 I47 G48 G49 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16218957 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2aoq A 2.2 BS01 dna B 0 R46 K48 T174 A175 R176 R184 G187 A188 N189 S190 R214 K215 R38 K40 T166 A167 R168 R176 G179 A180 N181 S182 R206 K207 ? 0003677,0004519,0005737,0006281,0006298,0006304 remove_due_to_license_issue P44688 16209953 1 ~ 12 MIPQTLEQLLSQAQSIAGLTFGELADELHIPVPIDLKRDKGWVGMLLERALGATAGSKAEQDFSHLGVELKTLPINAEGYPLETTFVSLAPLVQNSGVKWENSHVRHKLSCVLWMPIEGSRHIPLRERHIGAPIFWKPTAEQERQLKQDWEELMDLIVLGKLDQITARIGEVMQLRPKGANSRAVTKGIGKNGEIIDTLPLGFYLRKEFTAQILNAFLET 2aoq A 2.2 BS02 dna C 0 K48 G49 G52 E56 G64 S65 E68 D70 T80 P82 E91 F94 L97 K116 R129 K186 T194 K40 G41 G44 E48 G56 S57 E60 D62 T72 P74 E83 F86 L89 K108 R121 K178 T186 ? 0003677,0004519,0005737,0006281,0006298,0006304 remove_due_to_license_issue P44688 16209953 1 ~ 12 MIPQTLEQLLSQAQSIAGLTFGELADELHIPVPIDLKRDKGWVGMLLERALGATAGSKAEQDFSHLGVELKTLPINAEGYPLETTFVSLAPLVQNSGVKWENSHVRHKLSCVLWMPIEGSRHIPLRERHIGAPIFWKPTAEQERQLKQDWEELMDLIVLGKLDQITARIGEVMQLRPKGANSRAVTKGIGKNGEIIDTLPLGFYLRKEFTAQILNAFLET 2aor A 2.0 BS01 dna C 0 R46 K48 M53 T174 A175 R184 P185 G187 A188 N189 S190 R38 K40 M45 T166 A167 R176 P177 G179 A180 N181 S182 ? 0003677,0004519,0005737,0006281,0006298,0006304 remove_due_to_license_issue P44688 16209953 1 ~ 22 MIPQTLEQLLSQAQSIAGLTFGELADELHIPVPIDLKRDKGWVGMLLERALGATAGSKAEQDFSHLGVELKTLPINAEGYPLETTFVSLAPLVQNSGVKWENSHVRHKLSCVLWMPIEGSRHIPLRERHIGAPIFWKPTAEQERQLKQDWEELMDLIVLGKLDQITARIGEVMQLRPKGANSRAVTKGIGKNGEIIDTLPLGFYLRKEFTAQILNAFLET 2aor A 2.0 BS02 dna D 0 K45 K48 G49 G52 S65 K66 T80 P82 E91 F94 K186 K37 K40 G41 G44 S57 K58 T72 P74 E83 F86 K178 ? 0003677,0004519,0005737,0006281,0006298,0006304 remove_due_to_license_issue P44688 16209953 1 ~ 22 MIPQTLEQLLSQAQSIAGLTFGELADELHIPVPIDLKRDKGWVGMLLERALGATAGSKAEQDFSHLGVELKTLPINAEGYPLETTFVSLAPLVQNSGVKWENSHVRHKLSCVLWMPIEGSRHIPLRERHIGAPIFWKPTAEQERQLKQDWEELMDLIVLGKLDQITARIGEVMQLRPKGANSRAVTKGIGKNGEIIDTLPLGFYLRKEFTAQILNAFLET 2aor B 2.0 BS01 dna C 0 K45 K48 G49 G52 M53 K66 T80 P82 E91 F94 K186 K37 K40 G41 G44 M45 K58 T72 P74 E83 F86 K178 ? 0003677,0004519,0005737,0006281,0006298,0006304 remove_due_to_license_issue P44688 16209953 1 ~ 22 MIPQTLEQLLSQAQSIAGLTFGELADELHIPVPIDLKRDKGWVGMLLERALGATAGSKAEQDFSHLGVELKTLPINAEGYPLETTFVSLAPLVQNSGVKWENSHVRHKLSCVLWMPIEGSRHIPLRERHIGAPIFWKPTAEQERQLKQDWEELMDLIVLGKLDQITARIGEVMQLRPKGANSRAVTKGIGKNGEIIDTLPLGFYLRKEFTAQILNAFLETK 2aor B 2.0 BS02 dna D 0 R46 K48 T174 A175 R184 P185 G187 A188 N189 S190 R38 K40 T166 A167 R176 P177 G179 A180 N181 S182 ? 0003677,0004519,0005737,0006281,0006298,0006304 remove_due_to_license_issue P44688 16209953 1 ~ 22 MIPQTLEQLLSQAQSIAGLTFGELADELHIPVPIDLKRDKGWVGMLLERALGATAGSKAEQDFSHLGVELKTLPINAEGYPLETTFVSLAPLVQNSGVKWENSHVRHKLSCVLWMPIEGSRHIPLRERHIGAPIFWKPTAEQERQLKQDWEELMDLIVLGKLDQITARIGEVMQLRPKGANSRAVTKGIGKNGEIIDTLPLGFYLRKEFTAQILNAFLETK 2aou A 2.3 BS01 CQA A 1 Y15 F19 Q94 Q143 Y146 V173 W179 W183 F243 E246 Y11 F15 Q90 Q139 Y142 V169 W175 W179 F239 E242 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 Ki=18.6nM remove_due_to_license_issue Ki=19nM P50135 16168438 402 MRSLFSDHGKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKTSNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 2aou A 2.3 BS02 CQA A 2 D180 W183 G187 F190 P191 D193 Y198 T245 T247 D176 W179 G183 F186 P187 D189 Y194 T241 T243 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 Ki=18.6nM remove_due_to_license_issue Ki=19nM P50135 16168438 403 MRSLFSDHGKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKTSNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 2aov A 2.48 BS01 C2M A 1 E28 Q143 Y146 W179 W183 Q197 Y198 E24 Q139 Y142 W175 W179 Q193 Y194 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 Ki=91nM remove_due_to_license_issue P50135 16168438 401 MRSLFSDHGKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKTSNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 2aow A 2.97 BS01 THA A 1 F22 E28 Q143 W179 W183 F18 E24 Q139 W175 W179 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 remove_due_to_license_issue P50135 16168438 400 MRSLFSDHGKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKISNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 2aox A 3.12 BS01 THA A 1 F19 F22 E28 Q143 W179 W183 F15 F18 E24 Q139 W175 W179 2.1.1.8 0001692,0001695,0005654,0005737,0005813,0005829,0006548,0007585,0008168,0008170,0032259,0046539,0070062 remove_due_to_license_issue P50135 16168438 400 MRSLFSDHGKYVESFRRFLNHSTEHQCMQEFMDKKLPGIIGRIGDTKSEIKILSIGGGAGEIDLQILSKVQAQYPGVCINNEVVEPSAEQIAKYKELVAKTSNLENVKFAWHKETSSEYQSRMLEKKELQKWDFIHMIQMLYYVKDIPATLKFFHSLLGTNAKMLIIVVSGSSGWDKLWKKYGSRFPQDDLCQYITSDDLTQMLDNLGLKYECYDLLSTMDISDCFIDGNENGDLLWDFLTETCNFNATAPPDLRAELGKDLQEPEFSAKKEGKVLFNNTLSFIVIEA 2aq7 A 2.3 BS01 TL5 A 1 C163 F229 D268 M269 V270 A271 P272 H298 T300 H333 F390 G391 F392 G394 C163 F229 D268 M269 V270 A271 P272 H298 T300 H333 F390 G391 F392 G394 C163 H298 E309 K328 H333 F390 F392 C163 H298 E309 K328 H333 F390 F392 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 ic50=500uM remove_due_to_license_issue P0A953 16392800 600 MKRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2aq7 B 2.3 BS01 TL5 B 1 C163 F229 D268 M269 V270 A271 P272 H298 H333 F390 G391 F392 G394 C162 F228 D267 M268 V269 A270 P271 H297 H332 F389 G390 F391 G393 C163 H298 E309 K328 H333 F390 F392 C162 H297 E308 K327 H332 F389 F391 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 ic50=500uM remove_due_to_license_issue P0A953 16392800 601 KRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2aqb A 2.19 BS01 TL6 A 1 C163 F229 V270 A271 P272 H298 T300 H333 F390 G391 F392 G394 C163 F229 V270 A271 P272 H298 T300 H333 F390 G391 F392 G394 C163 H298 E309 K328 H333 F390 F392 C163 H298 E309 K328 H333 F390 F392 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 ic50=500uM remove_due_to_license_issue P0A953 16392800 600 MKRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2aqb B 2.19 BS01 TL6 B 1 C163 F229 V270 A271 P272 H298 T300 F390 G391 F392 G394 C162 F228 V269 A270 P271 H297 T299 F389 G390 F391 G393 C163 H298 E309 K328 H333 F390 F392 C162 H297 E308 K327 H332 F389 F391 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 ic50=500uM remove_due_to_license_issue P0A953 16392800 601 KRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2aqu A 2.0 BS01 DR7 B 1 D25 G27 D29 G48 G49 P81 V82 I84 D25 G27 D29 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 16634628 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2aqu B 2.0 BS01 DR7 B 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.48nM remove_due_to_license_issue P03366 16634628 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2arm A 1.23 BS01 OIN A 1 Y28 G30 W31 H48 D49 Y52 P68 K69 Y27 G29 W30 H47 D48 Y51 P59 K60 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 Kd=0.000000064M remove_due_to_license_issue P59071 16596639 401 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 2ata A 2.2 BS01 dna E 0 K120 S121 R248 K25 S26 R153 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 10 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRKK 2ata A 2.2 BS02 dna F 0 S241 R273 C275 A276 R280 S146 R178 C180 A181 R185 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 2 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRKK 2ata B 2.2 BS01 dna E 0 S241 R248 R273 C275 A276 C277 R280 S148 R155 R180 C182 A183 C184 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 10 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLRK 2ata C 2.2 BS01 dna F 0 A119 T123 A24 T28 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 2 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLR 2ata C 2.2 BS02 dna G 0 S241 R248 R273 C275 A276 R280 S146 R153 R178 C180 A181 R185 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 12 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLR 2ata C 2.2 BS03 dna H 0 A119 K120 A24 K25 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 11 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLR 2ata D 2.2 BS01 dna H 0 N239 S241 R248 R273 C275 A276 R280 N146 S148 R155 R180 C182 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 16793544 1 ~ 11 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRVEYLDDRNTFRHSVVVPYEPPEVGSDCTTIHYNYMCNSSCMGGMNRRPILTIITLEDSSGNLLGRNSFEVRVCACPGRDRRTEEENLR 2ate A 1.8 BS01 NIA A 1 G15 S16 D19 S43 A44 H45 R46 A70 G71 G8 S9 D12 S36 A37 H38 R39 A63 G64 5.4.99.18 0003824,0005829,0006164,0006189,0016853,0034023,0042802 remove_due_to_license_issue P0AG18 17298082 400 ARVAIVMGSKSDWATMQFAAEIFEILNVPHHVEVVSAHRTPDKLFSFAESAEENGYQVIIAGAGGAAHLPGMIAAKTLVPVLGVPVQSAALSGVDSLYSIVQMPRGIPVGTLAIGKAGAANAALLAAQILATHDKELHQRLNDWRKAQTDEVLENPDPRGAA 2ath A 2.28 BS01 3EA A 1 F282 G284 C285 R288 S289 H323 L330 I341 M364 H449 Y473 F76 G78 C79 R82 S83 H117 L124 I135 M158 H243 Y267 ? 0003677,0004879,0005634,0006355 ic50=0.152uM remove_due_to_license_issue IC50=152nM, EC50=230nM P37231 16366601 1001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2aux A 2.4 BS01 CT1 A 1 G23 C25 G64 G65 G66 L160 N161 H162 G21 C23 G62 G63 G64 L158 N159 H160 Q19 C25 H162 N182 Q17 C23 H160 N180 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=0.500000nM P43235 16290936 216 DSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 2auz A 2.3 BS01 CT2 A 1 G23 C25 G65 G66 A134 N161 G23 C25 G65 G66 A134 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=0.350000nM P43235 16290936 216 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 2avi A 3.0 BS01 BTN A 1 L14 T35 V37 T38 A39 T40 W70 F72 S73 S75 T77 W97 N118 L12 T33 V35 T36 A37 T38 W68 F70 S71 S73 T75 W95 N116 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 8506353 150 KCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYTTAVTATSNEIKESPLHGTENTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 2avm A 1.1 BS01 2NC B 1 D25 G27 A28 D29 G48 P81 V82 I84 D25 G27 A28 D29 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16277992 300 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avm B 1.1 BS01 2NC B 1 D25 G27 A28 D29 D30 I47 G48 I50 D25 G27 A28 D29 D30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2uM remove_due_to_license_issue P04587 16277992 300 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avo A 1.1 BS01 MK1 B 1 R8 D25 G48 G49 V82 I84 R8 D25 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 16277992 902 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avo B 1.1 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 I47 G48 G49 P81 V82 D25 G27 A28 D29 D30 V32 I47 G48 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508,0042802 Ki=1.4nM remove_due_to_license_issue P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avq A 1.3 BS01 2NC B 1 R8 D25 G27 A28 D29 D30 G48 I84 R8 D25 G27 A28 D29 D30 G48 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16277992 300 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avq B 1.3 BS01 2NC B 1 D25 G27 A28 D29 D30 I47 G48 G49 V50 P81 V82 D25 G27 A28 D29 D30 I47 G48 G49 V50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=41uM remove_due_to_license_issue P04587 16277992 300 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avs A 1.1 BS01 MK1 B 1 R8 D25 G27 G48 G49 P81 V82 I84 R8 D25 G27 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avs B 1.1 BS01 MK1 B 1 R8 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 R8 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=27nM remove_due_to_license_issue P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avv A 1.5 BS01 MK1 A 1 R8 D25 G27 A28 G48 G49 V82 I84 R8 D25 G27 A28 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.55nM remove_due_to_license_issue P04587 16277992 901 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAISTVLVGPTPVNIIGRNLLTQIGATLNF 2avv B 1.5 BS01 MK1 A 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 I84 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16277992 901 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAISTVLVGPTPVNIIGRNLLTQIGATLNF 2aw1 A 1.46 BS03 COX A 1 H94 H96 H119 F131 L141 L198 T199 T200 H92 H94 H117 F128 L138 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=43nM remove_due_to_license_issue Ki=43nM, IC50=43nM P00918 16290146 264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2ax6 A 1.5 BS01 HFT A 1 L704 N705 L707 Q711 M745 V746 M749 F764 M895 L34 N35 L37 Q41 M75 V76 M79 F94 M220 ? remove_due_to_license_issue IC50=26nM, Ki=43nM P10275 16129672 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIAPTSCSRRFYQLTKLLDSVQPIARELHQFAFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 2ax9 A 1.65 BS01 BHM A 1 L704 N705 L707 G708 Q711 W741 M745 V746 M749 F764 T877 L33 N34 L36 G37 Q40 W70 M74 V75 M78 F93 T198 ? Ki=0.3nM remove_due_to_license_issue Ki=0.3nM P10275 16129672 1 IFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 2ay1 A 2.2 BS02 AHC B 1 Y70 S296 Y65 S281 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay1 B 2.2 BS02 AHC B 1 G38 W140 N142 R386 G28 W121 N123 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=5.14mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay2 B 2.4 BS02 CXP B 1 G38 W140 R386 G28 W121 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=13.1mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay3 A 2.4 BS02 MPP A 1 G38 W140 N142 N194 R386 G34 W127 N129 N180 R371 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=0.28mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay3 B 2.4 BS01 MPP A 1 Y70 S296 Y59 S275 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=0.28mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay3 B 2.4 BS03 MPP B 1 D15 I17 L18 G38 W140 N142 R386 D11 I13 L14 G28 W121 N123 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=0.28mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay4 B 2.2 BS02 PPT B 1 I17 G38 W140 N142 R386 I13 G28 W121 N123 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=1.24mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay5 A 2.4 BS02 IOP B 1 Y70 S296 Y65 S281 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay5 B 2.4 BS02 IOP B 1 G38 W140 N142 R386 G28 W121 N123 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=2.6mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay6 A 2.2 BS02 3IB B 1 Y70 S296 Y65 S281 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay6 B 2.2 BS02 3IB B 1 D15 I17 G38 W140 N142 K258 R386 D11 I13 G28 W121 N123 K237 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=0.78mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay7 A 2.4 BS02 CLT B 1 Y70 S296 Y65 S281 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay7 B 2.4 BS02 CLT B 1 G38 W140 N142 N194 R386 G28 W121 N123 N174 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=5mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay8 A 2.2 BS02 4TB A 1 G38 W140 N194 F360 R386 G34 W127 N180 F345 R371 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=5.8mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay8 A 2.2 BS03 4TB B 1 Y70 S296 F297 Y65 S281 F282 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=5.8mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay8 B 2.2 BS01 4TB A 1 Y70 S296 F297 Y59 S275 F276 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=5.8mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay8 B 2.2 BS03 4TB B 1 G38 W140 N194 R386 G28 W121 N174 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=5.8mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay9 A 2.5 BS02 5PV A 1 W140 N142 N194 R386 W127 N129 N180 R371 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=6.9mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay9 A 2.5 BS03 5PV B 1 Y70 S296 F297 Y65 S281 F282 W140 D222 A224 K258 W127 D208 A210 K243 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=6.9mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFRADPRQGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay9 B 2.5 BS01 5PV A 1 Y70 S296 Y59 S275 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=6.9mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ay9 B 2.5 BS03 5PV B 1 D15 G38 W140 N142 N194 K258 R386 D11 G28 W121 N123 N174 K237 R365 W140 D222 A224 K258 W121 D202 A204 K237 2.6.1.57 0004069,0004838,0005737,0005829,0006520,0008483,0008652,0008793,0009058,0009073,0030170,0033585,0042802,0080130 Kd=6.9mM remove_due_to_license_issue P95468 9930977 414 MLGNLKPQAPDKILALMGEFGKIDLGVGVYKDATGHTPIMRAVHAAEQRMLETETTKTYAGLSGEPEFQKAMGELILGDGLKSETTATLATVGGTGALRQALELARMANPDLRVFVSDPTWPNHVSIMNFMGLPVQTYRYFDAETRGVDFEGMKADLAAAKKGDMVLLHGCCHNPTGANLTLDQWAEIASILEKTGALPLIDLAYQGFGDGLEEDAAGTRLIASRIPEVLIAASCSKNFGIYRERTGCLLALCADAATRELAQGAMAFLNRQTYSFPPFHGAKIVSTVLTTPELRADWMAELEAVRSGMLRLREQLAGELRDLSGSDRFGFVAEHRGMFSRLGATPEQVKRIKEEFGIYMVGDSRINIAGLNDNTIPILARAIIEVGV 2ayb A 3.2 BS01 dna C 0 S293 K297 R300 Y301 T316 H318 S13 K17 R20 Y21 T37 H39 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 16 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayb A 3.2 BS02 dna D 0 N294 R302 P351 T353 N14 R22 P72 T74 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 16 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayb B 3.2 BS01 dna C 0 N294 R302 P351 T353 N14 R22 P72 T74 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 16 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayb B 3.2 BS02 dna D 0 S293 K297 R300 Y301 T316 H318 S13 K17 R20 Y21 T37 H39 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 16 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayg A 3.1 BS01 dna C 0 S293 K297 R300 Y301 T316 S13 K17 R20 Y21 T37 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 18 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayg A 3.1 BS02 dna D 0 N294 R302 P351 T353 N14 R22 P72 T74 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 18 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayg B 3.1 BS01 dna C 0 R302 K349 P351 T353 R22 K70 P72 T74 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 18 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayg B 3.1 BS02 dna D 0 S293 K297 R300 Y301 S315 T316 S13 K17 R20 Y21 S36 T37 ? 0003677,0003700,0006275,0006355,0042025 remove_due_to_license_issue Q84294 16914454 1 ~ 18 SSATPIVQFQGESNCLKCFRYRLNDKHRHLFDLISSTWHWASPKAPHKHAIVTVTYHSEEQRQQFLNVVKIPPTIRHKLGFMSMHLL 2ayp A 2.9 BS01 43A A 1 L15 A36 K38 E55 N59 V68 L84 C87 G90 L137 S147 D148 F149 L14 A35 K37 E54 N58 V67 L83 C86 G89 L136 S146 D147 F148 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=7nM O14757 16242328 270 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2ayr A 1.9 BS01 L4G A 1 M343 L346 T347 A350 D351 E353 W383 L387 R394 M421 I424 H524 L525 K529 M38 L41 T42 A45 D46 E48 W78 L82 R89 M116 I119 H219 L220 K224 ? Ki=0.51nM remove_due_to_license_issue Ki=0.47nM, EC50=10.7nM P03372 16250633 201 LALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKSKNVVPLYDLLLEMLDAHRLHA 2az0 A 2.6 BS01 rna C 0 N40 K47 K62 N39 K46 K61 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEG 2az0 A 2.6 BS02 rna D 0 N33 R36 D37 R54 M55 S58 N32 R35 D36 R53 M54 S57 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEG 2az0 B 2.6 BS01 rna C 0 N33 R36 D37 R54 M55 S58 N32 R35 D36 R53 M54 S57 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEGK 2az0 B 2.6 BS02 rna D 0 N40 C44 K47 K62 P63 N39 C43 K46 K61 P62 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEGK 2az2 A 2.6 BS01 rna C 0 N40 K47 K62 N39 K46 K61 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEG 2az2 A 2.6 BS02 rna D 0 R36 D37 R54 M55 S58 R35 D36 R53 M54 S57 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEG 2az2 B 2.6 BS01 rna C 0 N33 R36 D37 R54 M55 S58 N32 R35 D36 R53 M54 S57 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEG 2az2 B 2.6 BS02 rna D 0 N40 C44 K47 K62 P63 N39 C43 K46 K61 P62 ? remove_due_to_license_issue P68831 16228003 1 ~ 18 PSKLALIQELPDRIQTAVEAAMGMSYQDAPNNVRRDLDNLHACLNKAKLTVSRMVTSLLEKPSVVAYLEG 2az5 A 2.1 BS01 307 A 1 L57 Y59 S60 Y119 L120 G121 G122 Y151 L43 Y45 S46 Y94 L95 G96 G97 Y126 ? 0005164,0006955,0016020 ic50=22uM remove_due_to_license_issue Kd=5360nM, IC50=1300nM P01375 16284179 1 DKPVAHVVANPQAEGQLQWLNLLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 2az5 B 2.1 BS01 307 A 1 Y59 Y119 L120 G121 Y151 Y50 Y102 L103 G104 Y134 ? 0005164,0006955,0016020 remove_due_to_license_issue Kd=5360nM, IC50=1300nM P01375 16284179 1 DKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCQRKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 2az5 D 2.1 BS01 307 C 1 Y59 Y119 L120 G121 Y50 Y103 L104 G105 ? 0005164,0006955,0016020 remove_due_to_license_issue Kd=5360nM, IC50=1300nM P01375 16284179 2 DKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCQRAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 2az8 A 2.0 BS01 3TL A 1 G27 A28 D29 I47 G48 G49 I50 G27 A28 D29 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=6nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2az9 A 2.5 BS01 3TL A 1 D25 G27 A28 D29 M46 I47 G48 G49 I50 D25 G27 A28 D29 M46 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=22nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 2azb A 2.03 BS01 3TL A 1 D25 G27 D29 I47 G48 G49 I50 D25 G27 D29 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=64nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKIIGGIGIKVRQYDQILIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 2azc A 2.01 BS01 3TL A 1 D25 G27 A28 D29 K45 I46 I47 G48 G49 I50 D25 G27 A28 D29 K45 I46 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=183nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVLEEMNLPGRWKPKIIGGIGGLIKVRQYDQIPIEICGHKAIGTVLIGPTPANIIGRNLLTQIGCTLNF 2azc A 2.01 BS02 3TL B 1 D25 P81 D25 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=183nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVLEEMNLPGRWKPKIIGGIGGLIKVRQYDQIPIEICGHKAIGTVLIGPTPANIIGRNLLTQIGCTLNF 2azc B 2.01 BS01 3TL A 1 D25 I50 I84 D25 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=183nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVLEEMNLPGRWKPKIIGGIGGLIKVRQYDQIPIEICGHKAIGTVLIGPTPANIIGRNLLTQIGCTLNF 2azc B 2.01 BS02 3TL B 1 G27 G48 G49 I50 G27 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=183nM remove_due_to_license_issue P03367 16403521 200 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVLEEMNLPGRWKPKIIGGIGGLIKVRQYDQIPIEICGHKAIGTVLIGPTPANIIGRNLLTQIGCTLNF 2azr A 2.0 BS01 982 A 1 Y46 V49 K120 D181 F182 S216 A217 I219 G220 R221 Q262 Y45 V48 K119 D180 F181 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=230uM remove_due_to_license_issue P18031 16303309 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2b07 A 2.1 BS01 598 A 1 Y46 D48 V49 K120 F182 S216 I219 R221 G259 Q262 Y45 D47 V48 K119 F181 S215 I218 R220 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.37uM remove_due_to_license_issue P18031 16303309 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2b0d A 2.0 BS01 dna C 0 T37 N70 K92 T93 T94 Y95 T106 T111 S112 K119 S183 T186 N188 T36 N69 K91 T92 T93 Y94 T103 T108 S109 K116 S174 T177 N179 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0d A 2.0 BS02 dna D 0 S183 G184 N185 T222 S223 R226 S174 G175 N176 T213 S214 R217 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0d B 2.0 BS01 dna C 0 Q69 N70 L180 S183 G184 N185 T222 S223 Q68 N69 L174 S177 G178 N179 T216 S217 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVATSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0d B 2.0 BS02 dna D 0 T37 N70 K92 T94 Y95 T106 T111 S112 K119 N120 G182 S183 T186 N188 T36 N69 K91 T93 Y94 T103 T108 S109 K116 N117 G176 S177 T180 N182 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVATSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0e A 1.9 BS01 dna C 0 T37 N70 K92 T93 T94 Y95 T106 T111 S112 K119 N120 S183 T186 N188 T36 N69 K91 T92 T93 Y94 T100 T105 S106 K113 N114 S171 T174 N176 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0e A 1.9 BS02 dna D 0 S183 G184 N185 T222 S223 R226 S171 G172 N173 T210 S211 R214 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0e B 1.9 BS01 dna C 0 L180 S183 G184 N185 T222 S223 N231 L171 S174 G175 N176 T213 S214 N222 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b0e B 1.9 BS02 dna D 0 T37 N70 K92 T93 T94 Y95 T106 T111 S112 K119 N120 S183 T186 N188 T36 N69 K91 T92 T93 Y94 T102 T107 S108 K115 N116 S174 T177 N179 3.1.21.4 0003677,0004519,0009036,0009307,0046872 remove_due_to_license_issue P04390 16236314 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYERTSQLRNDKYNNISEYRNWIYRGRK 2b17 A 2.71 BS01 DIF A 1 L2 F5 I19 G30 C45 L2 F5 I18 G29 C44 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 remove_due_to_license_issue P59071 16552142 701 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 2b1g A 2.1 BS01 13A A 1 S11 V12 S13 R65 K67 T68 N103 Y105 D126 I127 G128 S8 V9 S10 R62 K64 T65 N100 Y102 D123 I124 G125 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.23uM remove_due_to_license_issue P31335 17324932 600 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1i A 2.02 BS01 93A A 1 S11 V12 S13 S35 G37 T38 G64 R65 K67 T68 L69 C102 N103 L104 Y105 D126 I127 G128 G129 S8 V9 S10 S32 G34 T35 G61 R62 K64 T65 L66 C99 N100 L101 Y102 D123 I124 G125 G126 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.15uM remove_due_to_license_issue P31335 17324932 600 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1i A 2.02 BS02 93A A 2 R208 Y209 I239 K267 H268 G317 D340 R205 Y206 I236 K264 H265 G314 D337 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.15uM remove_due_to_license_issue P31335 17324932 701 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1i A 2.02 BS03 93A B 2 N432 A541 R589 F591 N429 A538 R586 F588 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.15uM remove_due_to_license_issue P31335 17324932 700 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1i B 2.02 BS01 93A A 2 N432 A541 R589 F591 N429 A538 R586 F588 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.15uM remove_due_to_license_issue P31335 17324932 701 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1i B 2.02 BS02 93A B 1 S11 V12 S13 K15 S35 G37 T38 G64 R65 K67 T68 L69 C102 N103 L104 Y105 D126 I127 G128 G129 S8 V9 S10 K12 S32 G34 T35 G61 R62 K64 T65 L66 C99 N100 L101 Y102 D123 I124 G125 G126 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.15uM remove_due_to_license_issue P31335 17324932 601 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1i B 2.02 BS03 93A B 2 R208 Y209 I239 K267 H268 G317 D340 R205 Y206 I236 K264 H265 G314 D337 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 Ki=0.15uM remove_due_to_license_issue P31335 17324932 700 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2b1p A 1.9 BS01 AIZ A 1 A91 K93 L144 M146 M149 D150 A151 N152 Q155 A44 K46 L97 M99 M102 D103 A104 N105 Q108 D189 K191 N194 D207 T226 D142 K144 N147 D160 T164 2.7.11.24 0004672,0004707,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=3nM P53779 16140012 501 NQFYSVEVGDSTFTVLKRYQNLKPIGSGGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPDEREHTIEEWKELIYKEVMN 2b1v A 1.8 BS02 458 A 1 E353 L391 F404 M421 H524 E49 L87 F100 M117 H212 ? Ki=1.8uM remove_due_to_license_issue P03372 16648639 201 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 2b1z A 1.78 BS02 17M A 1 E353 L387 M388 F404 H524 L525 E49 L83 M84 F100 H211 L212 ? ic50=79nM remove_due_to_license_issue P03372 17949766 201 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 2b4m A 2.8 BS01 PBE A 1 S25 G26 I27 W72 W178 W225 T229 S17 G18 I19 W64 W170 W217 T221 ? 0005886,0006865,0022857,0043190,0045121,0055085 remove_due_to_license_issue P46922 16445940 311 SAAEQVNKTIIGIDPGSGIMSLTDKAMKDYDLNDWTLISASSAAMTATLKKSYDRKKPIIITGWTPHWMFSRYKLKYLDDPKQSYGSAEEIHTITRKGFSKEQPNAAKLLSQFKWTQDEMGEIMIKVEEGEKPAKVAAEYVNKHKDQIAEWTKGVQKVKGDKINLAYVAWDSEIASTNVIGKVLEDLGYEVTLTQVEAGPMWTAIATGSADASLSAWLPNTHKAYAAKYKGKYDDIGTSMTGVKMGLVVPQYMKNVNSIEDLKK 2b52 A 1.88 BS01 D42 A 1 I10 G13 V18 A31 V64 F80 F82 L83 H84 D86 K89 Q131 N132 L134 D145 I10 G13 V18 A31 V60 F76 F78 L79 H80 D82 K85 Q127 N128 L130 D141 D127 K129 Q131 N132 D145 T165 D123 K125 Q127 N128 D141 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=8nM remove_due_to_license_issue IC50=8nM P24941 14698155 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2b53 A 2.0 BS01 D23 A 1 I10 F80 L83 D86 K89 D145 I10 F76 L79 D82 K85 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.6uM remove_due_to_license_issue IC50=600nM P24941 11354366 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2b54 A 1.85 BS01 D05 A 1 I10 G11 V18 F82 L83 H84 Q131 N132 L134 I10 G11 V18 F82 L83 H84 Q131 N132 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=20nM P24941 15537345 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2b55 A 1.85 BS01 D31 A 1 I10 E12 V18 A31 F80 F82 L83 D86 K89 Q131 L134 D145 I10 E12 V18 A31 F73 F75 L76 D79 K82 Q124 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T143 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=96nM remove_due_to_license_issue IC50=96nM P24941 12431051 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2b5j A 2.9 BS02 3AC A 1 L100 K101 V106 Y188 G190 F227 W229 L234 Y318 L100 K101 V106 Y188 G190 F227 W229 L234 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 16302798 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 2b63 A 3.8 BS01 rna R 0 Q316 S318 R320 K323 K332 R337 E833 R1386 E1403 Q307 S309 R311 K314 K323 R328 E824 R1347 E1364 D481 D483 D485 D472 D474 D476 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001065,0001066,0001172,0003677,0003899,0003968,0005515,0005634,0005665,0005739,0006351,0006360,0006366,0006367,0006368,0006383,0006390,0008270,0010494,0016779,0019985,0034062,0042793,0046872 remove_due_to_license_issue P04050 16341226 2 ~ 32 VGQQYSSAPLRTVKEVQFGLFSPEEVRAISVAKIRFPETMDETQTRAKIGGLNDPRLGSIDRNLKCQTCQEGMNECPGHFGHIDLAKPVFHVGFIAKIKKVCECVCMHCGKLLLDEHNELMRQALAIKDSKKRFAAIWTLCKTKMVCETDVPSEDDPTQLVSRGGCGNTQPTIRKDGLKLVGSWKDEPELRVLSTEEILNIFKHISVKDFTSLGFNEVFSRPEWMILTCLPVPPPPVRPSISFNESQRGEDDLTFKLADILKANISLETLEHNGAPHHAIEEAESLLQFHVATYMDNDIAGQPQALQKSGRPVKSIRARLKGKEGRIRGNLMGKRVDFSARTVISGDPNLELDQVGVPKSIAKTLTYPEVVTPYNIDRLTQLVRNGPNEHPGAKYVIRDSGDRIDLRYSKRAGDIQLQYGWKVERHIMDNDPVLFNRQPSLHKMSMMAHRVKVIPYSTFRLNLSVTSPYNADFDGDEMNLHVPQSEETRAELSQLCAVPLQIVSPQSNKPCMGIVQDTLCGIRKLTLRDTFIELDQVLNMLYWVPDWDGVIPTPAIIKPKPLWSGKQILSVAIPNGIHLQRFDEGTTLLSPKDNGMLIIDGQIIFGVVEKKTVGSSNGGLIHVVTREKGPQVCAKLFGNIQKVVNFWLLHNGFSTGIGDTIADGPTMREITETIAEAKKKVLDVTKEAQANLLTAKHGMTLRESFEDNVVRFLNEARDKAGRLAEVNLKDLNNVKQMVMAGSKGSFINIAQMSACVGQQSVEGKRIAFGFVDRTLPHFSKDDYSPESKGFVENSYLRGLTPQEFFFHAMGGREGLIDTAVKTAETGYIQRRLVKALEDIMVHYDNTTRNSLGNVIQFIYGEDGMDAAHIEKQSLDTIGGSDAAFEKRYRVDLLNTDHTLDPSLLESGSEILGDLKLQVLLDEEYKQLVKDRKFLREVFVDGEANWPLPVNIRRIIQNAQQTFHIDHTKPSDLTIKDIVLGVKDLQENLLVLRGKNEIIQNAQRDAVTLFCCLLRSRLATRRVLQEYRLTKQAFDWVLSNIEAQFLRSVVHPGEMVGVLAAQSIGEPATQMTLKKVTSGVPRLKEILNVAKNMKTPSLTVYLEPGHAADQEQAKLIRSAIEHTTLKSVTIASEIYYDPDPRSTVIPEDEEIIQLHFSLQQSPWLLRLELDRAAMNDKDLTMGQVGERIKQTFKNDLFVIWSEDNDEKLIIRCRVVAEEDHMLKKIENTMLENITLRGVENIERVVMMKYDRKVPSPTGEYVKEPEWVLETDGVNLSEVMTVPGIDPTRIYTNSFIDIMEVLGIEAGRAALYKEVYNVIASDGSYVNYRHMALLVDVMTTQGGLTSVTRHGFNRSNTGALMRCSFEETVEILFEAGASAELDDCRGVSENVILGQMAPIGTGAFDVMIDEESLVKYMP 2b63 B 3.8 BS01 rna R 0 Y459 T463 N465 S474 S475 R476 Q481 V482 R512 Q531 R1124 Y375 T379 N381 S390 S391 R392 Q397 V398 R428 Q447 R1012 D837 D738 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001065,0001066,0001172,0003677,0003729,0003899,0003968,0005515,0005634,0005665,0005739,0006351,0006360,0006366,0006367,0006368,0006383,0006390,0008270,0010494,0016779,0032549,0034062,0042793,0046872 remove_due_to_license_issue P08518 16341226 2 ~ 32 DESAPITAEDSWAVISAFFREKGLVSQQLDSFNQFVDYTLQDIICEDSTLIISFGKIYVTKPMVNESDGVTHALYPQEARLRNLTYSSGLFVDVKKKVFIGRLPIMLRSKNCYLSEATESDLYKLKECPFDMGGYFIINGSEKVLIAQERSAGNIVQVFKKAAPSPISHVAEIRSALEKGSRFISTLQVKLYGREGSSARTIKATLPYIKQDIPIVIIFRALGIIPDGEILEHICYDVNDWQMLEMLKPCVEDGFVIQDRETALDFIGKEKRIQYAKDILQKEFLPHITQLEGFESRKAFFLGYMINRLLLCALDRKDQDDRDHFGKKRLDLAGPLLAQLFKTLFKKLTKDIFRYMQRTVELAINAKTITSGLKYALATGNWGEQKKAMSSRAGVSQVLNRYTYSSTLSHLRRTNTPIGRDGKLAKPRQLHNTHWGLVCPAETPEGQACGLVKNLSLMSCISVGTDPMPIITFLSEWGMEPLEDYVPHQSPDATRVFVNGVWHGVHRNPARLMETLRTLRRKGDINPEVSMIRDIREKELKIFTDAGRVYRPLFIVEDDESLGHKELKVRKGHIAKLMATEYQDEYTWSSLLNEGLVEYIDAEEEESILIAMQPEDLEPAEADVDPAKRIRVSHHATTFTHCEIHPSMILGVAASIIPFPDHNQSPRNTYQSAMGKQAMGVFLTNYNVRMDTMANILYYPQKPLGTTRAMEYLKFRELPAGQNAIVAIACYSGYNQEDSMIMNQSSIDRGLFRSLFFRSYMDQEKKYGMSITETFEKPQRTNTLRMKHGTYDKLDDDGLIAPGVRVSGEDVIIGKTTPISSKRDASTPLRSTENGIVDQVLVTTNQDGLKFVKVRVRTTKIPQIGDKFASRHGQKGTIGITYRREDMPFTAEGIVPDLIINPHAIPSRMTVAHLIECLLSKVAALSGNEGDASPFTDITVEGISKLLREHGYQSRGFEVMYNGHTGKKLMAQIFFGPTYYQRLRHMVDDKIHARARGPMQVLTRQPVEGRSRDGGLRFGEMERDCMIAHGAASFLKERLMEASDAFRVHICGICGLMTVIAKLNHNQFECKGCDNKIDIYQIHIPYAAKLLFQELMAMNITPRLYTDRSRDF 2b6g A -1.00 BS01 rna B 0 Y468 A495 L496 G497 A498 Y26 A53 L54 G55 A56 ? 0003729,0043488 remove_due_to_license_issue Q08831 16429155 1 ~ 19 NPKSLTDPKLLKNIPMWLKSLRLHKYSDALSGTPWIELIYLDDETLEKKGVLALGARRKLLKAFGIVIDYKERDLIDRSAY 2b7a A 2.0 BS01 IZA A 1 L855 G856 K857 V863 A880 M929 Y931 L932 G935 L983 L13 G14 K15 V21 A38 M83 Y85 L86 G89 L137 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1nM O60674 16174768 2001 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG 2b7d H 2.24 BS01 C1B H 1 H57 D60 K60A D189 S190 C191 K192 S195 V213 W215 G219 H41 D44 K45 D186 S187 C188 K189 S192 V210 W212 G215 3.4.21.21 0004252,0006508 Ki=0.002uM remove_due_to_license_issue Ki=2nM P08709 16412633 258 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2b8l A 1.7 BS01 5HA A 1 G11 Q12 G13 L30 D32 G34 Y71 T72 Q73 F108 W115 I118 D228 G230 T232 N233 R235 A335 G17 Q18 G19 L36 D38 G40 Y77 T78 Q79 F114 W121 I124 D222 G224 T226 N227 R229 A329 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=15nM remove_due_to_license_issue IC50=15nM, EC50=43nM, Ki=233nM P56817 16263281 386 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2b8v A 1.8 BS01 3BN A 1 Q12 G13 L30 D32 G34 Y71 T72 Q73 F108 I110 W115 I226 D228 G230 T231 T232 N233 R235 Q18 G19 L36 D38 G40 Y77 T78 Q79 F114 I116 W121 I219 D221 G223 T224 T225 N226 R228 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=98nM remove_due_to_license_issue IC50=98nM P56817 16263281 1001 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2b9a A 1.54 BS01 FBC A 1 L17 A108 L110 S117 L8 A93 L95 S102 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 14711308 301 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTARYTIAALLSPYSYSTTAVVT 2b9a B 1.54 BS01 FBC B 1 A108 L110 S117 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 14711308 302 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 2baj A 2.25 BS01 1PP A 1 A51 E71 L104 T106 L167 D168 A50 E70 L103 T105 L156 D157 D150 K152 N155 D168 T185 D139 K141 N144 D157 T174 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=4nM remove_due_to_license_issue IC50=30nM Q16539 16342939 401 HHHSQERPTFYRQELIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESRNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 2bak A 2.2 BS01 AQZ A 1 V30 A51 K53 E71 M78 T106 H107 M109 H148 I166 L167 D168 F169 V26 A47 K49 E67 M74 T102 H103 M105 H141 I159 L160 D161 F162 D150 K152 N155 D168 T185 D143 K145 N148 D161 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=37nM remove_due_to_license_issue IC50=39nM Q16539 16342939 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 2bal A 2.1 BS01 PQA A 1 A51 L104 T106 L108 M109 G110 A111 A47 L100 T102 L104 M105 G106 A107 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=490nM remove_due_to_license_issue Q16539 16342939 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 2ban A 2.95 BS02 357 A 1 L100 K101 K103 V179 Y181 Y188 G190 W229 L234 Y318 L100 K101 K103 V179 Y181 Y188 G190 W229 L234 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 16302798 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 2bb7 A 1.7 BS03 QMS A 1 C59 Y62 C70 H79 F177 H178 W221 C55 Y58 C66 H75 F173 H174 W217 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H75 D93 D104 H167 R171 H174 Q178 E200 N204 Q229 E231 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=2.14uM remove_due_to_license_issue P0AE18 16300729 305 IKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISH 2bbb A 1.7 BS01 HH1 A 1 D25 G27 A28 D29 D30 G48 G49 P81 D25 G27 A28 D29 D30 G48 G49 P81 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=2.4nM remove_due_to_license_issue P03366 16298527 301 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bbb B 1.7 BS01 HH1 A 1 D225 G227 A228 D230 G249 P281 D25 G27 A28 D30 G49 P81 D225 T226 G227 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 16298527 301 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bdf A 2.1 BS01 24A A 1 L273 V281 A293 T338 Y340 M341 G344 L393 L17 V25 A37 T82 Y84 M85 G88 L137 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F157 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.067uM remove_due_to_license_issue P12931 16492148 600 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGETGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKEPEERPTFEYLQAFLEDYFTSTEPQYQ 2bdj A 2.5 BS01 HET A 1 L273 G274 V281 A293 K295 E310 T338 Y340 M341 S342 G344 L393 D404 L17 G18 V25 A37 K39 E54 T82 Y84 M85 S86 G88 L137 D148 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F157 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.00045uM remove_due_to_license_issue IC50=0.450000nM P12931 16492148 800 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGETGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKEPEERPTFEYLQAFLEDYFT 2bdl A 2.0 BS01 4PR A 1 Q19 C22 G23 C25 G64 G65 G66 Y67 N161 H162 W184 Q19 C22 G23 C25 G64 G65 G66 Y67 N161 H162 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 16376075 301 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 2bdy A 1.61 BS02 UNB A 1 H79 Y83 W86 E130 L132 I209 D229 A230 C231 S235 V255 S256 W257 G258 G260 H70 Y74 W77 E121 L123 I199 D219 A220 C221 S225 V245 S246 W247 G248 G250 H79 D135 E232 G233 D234 S235 G236 H70 D126 E222 G223 D224 S225 G226 3.4.21.5 0004252,0005509,0005576,0006508,0007596 ic50=0.017uM remove_due_to_license_issue IC50=17nM P00734 16290930 401 ADCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 2be2 A 2.43 BS03 R22 A 1 L100 K101 K103 V106 Y181 Y188 G190 F227 L234 H235 P236 Y318 L100 K101 K103 V106 Y181 Y188 G190 F227 L234 H235 P236 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=0.002uM remove_due_to_license_issue P03366 16302798 4002 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 2bed A 2.7 BS01 736 B 1 K164 Y166 H201 K111 Y113 H148 K164 K111 2.5.1.58,2.5.1.59 0008318,0018342 remove_due_to_license_issue Q04631 16298128 2001 GFLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSEKFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVWHFRRVLLRSLQKDLQEEMNYITAIIEEQPKNYQVWHHRRVLVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFRLWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRAVLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPNLLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDILNKALELCEILAKEKDTIRKEYWRYIGRSLQSK 2bed B 2.7 BS03 736 B 1 W102 W106 Y300 D359 Y361 W80 W84 Y278 D337 Y339 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 16298128 2001 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 2bes A 2.1 BS01 RES A 1 D11 H12 G70 S71 G74 E75 D9 H10 G68 S69 G72 E73 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=0.057mM remove_due_to_license_issue Ki=57000nM P9WKD7 15590681 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVPG 2bes A 2.1 BS02 RES B 1 H102 N103 R137 R141 H100 N101 R135 R139 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=0.057mM remove_due_to_license_issue Ki=57000nM P9WKD7 15590681 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVPG 2bes B 2.1 BS01 RES A 1 H102 N103 R137 R141 H101 N102 R136 R140 D11 G69 S71 H102 H138 D10 G68 S70 H101 H137 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=0.057mM remove_due_to_license_issue Ki=57000nM P9WKD7 15590681 200 SGMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVP 2bes B 2.1 BS02 RES B 1 D11 H12 G70 S71 G74 E75 R113 D10 H11 G69 S70 G73 E74 R112 D11 G69 S71 H102 H138 D10 G68 S70 H101 H137 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=0.057mM remove_due_to_license_issue Ki=57000nM P9WKD7 15590681 200 SGMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVP 2bet A 2.2 BS01 DEZ A 1 D11 H12 G70 S71 G74 E75 D9 H10 G68 S69 G72 E73 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=1.7mM remove_due_to_license_issue P9WKD7 15590681 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVPG 2bet A 2.2 BS02 DEZ B 1 H102 R137 R141 H100 R135 R139 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=1.7mM remove_due_to_license_issue P9WKD7 15590681 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVPG 2bet B 2.2 BS01 DEZ A 1 R137 R141 R135 R139 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=1.7mM remove_due_to_license_issue P9WKD7 15590681 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVPG 2bet B 2.2 BS02 DEZ B 1 D11 H12 S71 G74 E75 R113 D9 H10 S69 G72 E73 R111 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 Ki=1.7mM remove_due_to_license_issue P9WKD7 15590681 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVPG 2bfq A 1.5 BS01 AR6 A 1 D20 I21 A32 N34 G41 G42 V43 A44 A139 S141 G143 I144 Y145 Y176 D20 I21 A32 N34 G41 G42 V43 A44 A139 S141 G143 I144 Y145 Y176 3.2.2.- 0016787,0140291,0140293 remove_due_to_license_issue O28751 15902274 1193 MEVLFEAKVGDITLKLAQGDITQYPAKAIVNAANKRLEHGGGVAYAIAKACAGDAGLYTEISKKAMREQFGRDYIDHGEVVVTPAMNLEERGIKYVFHTVGPICSGMWSEELKEKLYKAFLGPLEKAEEMGVESIAFPAVSAGIYGCDLEKVVETFLEAVKNFKGSAVKEVALVIYDRKSAEVALKVFERSL 2bfr A 2.5 BS01 ADP A 1 D20 I21 G42 V43 A139 S141 G143 I144 Y145 Y176 D20 I21 G42 V43 A139 S141 G143 I144 Y145 Y176 3.2.2.- 0016787,0140291,0140293 Kd=5.63uM remove_due_to_license_issue O28751 15902274 1193 MEVLFEAKVGDITLKLAQGDITQYPAKAIVNAANKRLEHGGGVAYAIAKACAGDAGLYTEISKKAMREQFGRDYIDHGEVVVTPAMNLEERGIKYVFHTVGPICSGMWSEELKEKLYKAFLGPLEKAEEMGVESIAFPAVSAGIYGCDLEKVVETFLEAVKNFKGSAVKEVALVIYDRKSAEVALKVFERSL 2bgd A 2.4 BS01 T1D A 1 Y46 V49 K150 F182 C215 S216 A217 I219 G220 R221 E297 Y46 V49 K147 F179 C212 S213 A214 I216 G217 R218 E294 D181 C215 R221 S222 Q262 D178 C212 R218 S219 Q259 3.1.3.48 0004725,0006470,0016311 ic50=2.47uM remove_due_to_license_issue IC50=2500nM P18031 15863305 1298 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHE 2bge A 1.8 BS01 T2D A 1 Y46 S151 D181 F182 C215 S216 A217 I219 G220 R221 Q262 E297 Y46 S151 D181 F182 C215 S216 A217 I219 G220 R221 Q262 E297 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=1608uM remove_due_to_license_issue IC50=1600000nM P18031 15863305 1298 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHE 2bjc A -1.00 BS01 dna C 0 V15 S16 A18 T19 H29 V30 S31 T34 L56 A57 K59 Q60 V15 S16 A18 T19 H29 V30 S31 T34 L56 A57 K59 Q60 ? 0003677,0006355 remove_due_to_license_issue P03023 16094693 1 ~ 22 MKPVTLYDVAEYAGVSVATVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2bjc A -1.00 BS02 dna D 0 K2 T5 L6 Y7 V17 A18 S21 N25 Y47 P49 N50 A53 Q54 A57 K2 T5 L6 Y7 V17 A18 S21 N25 Y47 P49 N50 A53 Q54 A57 ? 0003677,0006355 remove_due_to_license_issue P03023 16094693 101 ~ 122 MKPVTLYDVAEYAGVSVATVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2bjc B -1.00 BS01 dna C 0 T105 L106 Y107 V117 A118 S121 N125 Y147 P149 A153 Q154 A157 Q160 T5 L6 Y7 V17 A18 S21 N25 Y47 P49 A53 Q54 A57 Q60 ? 0003677,0006355 remove_due_to_license_issue P03023 16094693 1 ~ 22 MKPVTLYDVAEYAGVSVATVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2bjc B -1.00 BS02 dna D 0 V115 S116 A118 T119 H129 V130 S131 T134 L156 A157 K159 Q160 V15 S16 A18 T19 H29 V30 S31 T34 L56 A57 K59 Q60 ? 0003677,0006355 remove_due_to_license_issue P03023 16094693 101 ~ 122 MKPVTLYDVAEYAGVSVATVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2bjm H 2.15 BS01 ANF H 1 W33 Y101 W33 Y101 Ka<100000M^-1 remove_due_to_license_issue 16129832 500 EVQLQQSGAELVKPGASVKLSCKASGYTFTSYWMHWVKQRPGRGLEWIGRIDPNGGGTKYNEKFKSKATLTVDKPSSTAYMQLSSLTSEDSAVYYCARMWYYGTYYFDYWGQGTTLTVSS 2bjm L 2.15 BS01 ANF H 1 Y34 W93 L98 Y34 W93 L98 ? 0002250,0006955,0019814 remove_due_to_license_issue P01724 16129832 500 QAVVTQESALTTSPGETVTLTCRSSTGAVTTSNYANWVQEKPDHLFTGLIGGTNNRAPGVPARFSGSLIGNKAALTITGAQTEDEAIYFCALWYSNHLVFGGGTKLTVLE 2bks B 2.2 BS01 PZ1 B 1 T13 Q14 Y15 D33 G35 W40 P42 H56 V106 M109 F114 F119 D120 G121 V122 D219 G221 T11 Q12 Y13 D31 G33 W38 P40 H54 V104 M107 F112 F117 D118 G119 V120 D215 G217 D33 S36 N38 W40 Y78 D219 A222 D31 S34 N36 W38 Y76 D215 A218 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=37nM P00797 15837327 401 SSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSELGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2bkt A 2.3 BS01 RPF A 1 Q14 D33 G35 W40 P42 H56 V106 M109 F114 A117 F119 D120 G121 V122 D219 G221 Q13 D32 G34 W39 P41 H55 V105 M108 F113 A116 F118 D119 G120 V121 D215 G217 D33 S36 N38 W40 Y78 D219 A222 D32 S35 N37 W39 Y77 D215 A218 3.4.23.15 0004190,0006508 ic50=23nM remove_due_to_license_issue IC50=23nM P00797 15837327 567 TSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2bkz A 2.6 BS01 SBC A 1 I10 A31 K33 F80 L83 H84 Q85 D86 L134 D145 I14 A35 K37 F84 L87 H88 Q89 D90 L138 D149 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=0.3nM P24941 15713378 1299 PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2bmc A 2.6 BS01 MPY A 1 G140 K141 V147 K162 Y212 A213 P214 G216 L263 G14 K15 V21 K36 Y86 A87 P88 G90 L137 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T154 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 15828847 1395 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPSNCQ 2bmg B 2.7 BS02 I1H B 1 T98 Y99 F174 D189 A190 C191 W215 G216 G219 C220 G226 I227 Y228 T84 Y85 F162 D179 A180 C181 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=18nM P00742 15857135 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2bmk A 2.3 BS01 PDD B 1 H34 R91 Y94 F96 H33 R90 Y93 F95 remove_due_to_license_issue 16790434 1217 DIELTQSPAIMAASPGEKVTITCSATSGVNYMHWFQQKPGTSPKLWIYSTSNLASAVPARFSGSGSGTSYSLTISRMEAEDAATYYCQQRSTYPFTFGGGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 2bmk B 2.3 BS01 PDD B 1 Y33 R52 D95 K96 Y33 R52 D101 K102 Kd=2.4uM remove_due_to_license_issue 16790434 1217 EVKLQESGGGLVQPGHSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGLIRNKANGYTKEYSASVKGRFTISRDNSQSILYLQMNALRAEDSATYYCVRDKGSYGNYEAWFAYWGQGTTVTVSSAKTTPPSVYPLAPGSQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPR 2bnw A 2.45 BS01 dna E 0 N50 V51 K52 N28 V29 K30 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 DIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw A 2.45 BS02 dna F 0 K28 T29 V30 R31 K6 T7 V8 R9 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 DIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw B 2.45 BS01 dna E 0 T29 R31 T11 R13 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw B 2.45 BS02 dna F 0 H37 K41 V51 K52 H19 K23 V33 K34 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw C 2.45 BS01 dna E 0 H37 K41 N50 V51 K52 H19 K23 N32 V33 K34 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw C 2.45 BS02 dna F 0 T29 V30 R31 T11 V12 R13 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw D 2.45 BS01 dna E 0 T29 R31 T5 R7 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 MGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnw D 2.45 BS02 dna F 0 K41 V51 K52 K17 V27 K28 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 MGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz A 2.6 BS01 dna E 0 K28 T29 R31 K7 T8 R10 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 17 KDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz A 2.6 BS02 dna F 0 H37 K41 N50 V51 K52 H16 K20 N29 V30 K31 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 KDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz B 2.6 BS01 dna E 0 N50 V51 K52 N29 V30 K31 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 17 KDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz B 2.6 BS02 dna F 0 K28 T29 V30 R31 K7 T8 V9 R10 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 KDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz C 2.6 BS01 dna E 0 R31 H37 K41 V51 K52 R12 H18 K22 V32 K33 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 17 AKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz C 2.6 BS02 dna F 0 T29 R31 T10 R12 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 AKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz D 2.6 BS01 dna E 0 K28 T29 V30 R31 K4 T5 V6 R7 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 17 MGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2bnz D 2.6 BS02 dna F 0 K41 N50 V51 K52 K17 N26 V27 K28 ? 0006355 remove_due_to_license_issue Q57468 16528102 19 ~ 36 MGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2boh B 2.2 BS02 IIA B 1 Y99 E147 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G219 G226 Y228 Y85 E135 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=3nM remove_due_to_license_issue Ki=3nM P00742 15999990 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2boi A 1.1 BS03 MFU A 1 S22 A23 D95 D98 D100 D103 S22 A23 D95 D98 D100 D103 ? 0046872 ic50=48uM remove_due_to_license_issue Q7NX84 16768446 400 AQQGVFTLPARINFGVTVLVNSAATQHVEIFVDNEPRAAFSGVGTGDNNLGTKVINSGSGNVRVQITANGRQSDLVSSQLVLANKLNLAVVGSEDGTDMDYNDSIVILNWPLG 2boi B 1.1 BS03 MFU B 1 S22 A23 D95 D98 D100 D103 S22 A23 D95 D98 D100 D103 ? 0046872 ic50=48uM remove_due_to_license_issue Q7NX84 16768446 700 AQQGVFTLPARINFGVTVLVNSAATQHVEIFVDNEPRAAFSGVGTGDNNLGTKVINSGSGNVRVQITANGRQSDLVSSQLVLANKLNLAVVGSEDGTDMDYNDSIVILNWPLG 2boj A 1.8 BS01 ARW A 1 N21 S22 S23 D96 D99 D101 D104 N21 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=1.7uM remove_due_to_license_issue Q9HYN5 16438968 1115 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2boj C 1.8 BS01 ARW C 1 N21 S22 S23 D96 D99 D101 D104 N21 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=1.7uM remove_due_to_license_issue Q9HYN5 16438968 1115 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2bok A 1.64 BS01 784 A 1 H57 Q61 Y99 F174 D189 A190 S195 S214 W215 G216 C220 H42 Q46 Y74 F151 D168 A169 S174 S193 W194 G195 C198 H57 D102 Q192 G193 D194 S195 G196 H42 D77 Q171 G172 D173 S174 G175 3.4.21.6 0004252,0006508 Ki=0.28uM remove_due_to_license_issue P00742 15952226 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2bow A 2.8 BS02 P4P A 1 V28 Y51 G52 A53 Y68 V27 Y34 G35 A36 Y51 ? remove_due_to_license_issue P39075 10025401 162 LGEVFVLDEEEIRIIQTEAEGIGPENVLNASYSYGATFSFQPYTSIDEMTYRHIFTPVLTISSITPDMEITTIPKGRYACIAYNFSPEHYFLNLQKLIKYIADRQLTVVSDVYELIIPIHYRVEMKIRIL 2bpm A 2.4 BS01 529 A 1 E8 I10 A31 F80 F82 L83 Q85 D86 L134 E12 I14 A35 F84 F86 L87 Q89 D90 L138 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=2nM remove_due_to_license_issue P24941 15828833 1299 PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2bpv A 1.9 BS01 1IN B 1 R8 D25 G27 F53 R8 D25 G27 F53 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bpv B 1.9 BS01 1IN B 1 D25 G27 A28 D29 G48 P81 D25 G27 A28 D29 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=21.2nM remove_due_to_license_issue P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bpx A 2.8 BS01 MK1 B 1 R8 D25 G27 G48 V82 I84 R8 D25 G27 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bpx B 2.8 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 I47 P81 I84 D25 G27 A28 D29 D30 V32 I47 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bpy A 1.9 BS01 3IN B 1 R8 D25 G48 V82 I84 R8 D25 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bpy B 1.9 BS01 3IN B 1 R8 D25 G27 A28 D29 G48 G49 R8 D25 G27 A28 D29 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=39.8nM remove_due_to_license_issue P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bq6 B 3.0 BS02 IIB B 1 Y99 E147 F174 D189 A190 C191 Q192 W215 G216 E217 G219 G226 Y228 Y85 E135 F162 D179 A180 C181 Q182 W205 G206 E207 G208 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=0.07nM P00742 15999990 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2bq7 B 2.2 BS01 IID A 1 T98 Y99 R143 F174 D189 A190 C191 Q192 W215 G216 G219 T84 Y85 R132 F162 D179 A180 C181 Q182 W205 G206 G208 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=89nM P00742 15999990 1001 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2bqv A 2.1 BS01 A1A A 1 D25 G27 A28 D30 G48 G49 D25 G27 A28 D30 G48 G49 3.4.23.16 0004190,0006508 Ki=9nM remove_due_to_license_issue O92139 16335934 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bqv B 2.1 BS01 A1A A 1 L123 D125 G127 A128 D129 G148 G149 I150 V182 I184 L23 D25 G27 A28 D29 G48 G49 I50 V82 I84 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue O92139 16335934 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bqw B 2.95 BS02 IIE B 1 E97 Y99 R143 F174 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 E83 Y85 R132 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=3nM P00742 15999990 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2br1 A 2.0 BS01 PFP A 1 L15 G16 V23 A36 E85 Y86 C87 G90 L137 L14 G15 V22 A35 E81 Y82 C83 G86 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=7.2uM remove_due_to_license_issue IC50=15400nM O14757 15974586 1277 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP 2br6 A 1.7 BS03 HSL A 1 H106 D108 H169 D191 Y194 H235 H96 D98 H159 D181 Y184 H225 3.1.1.81 0016787,0046872,0102007 Ki=1.1mM remove_due_to_license_issue P0CJ63 16314577 1255 MDMTVKKLYFIPAGRCMLDHSSVNSALTPGKLLNLPVWCYLLETEEGPILVDTGMPESAVNNILPKMTEEDRIVNILKRVGYEPDDLLYIISSHLHFDHAGGNGAFTNTPIIVQRTEYEAALHREEYMKECILPHLNYKIIEGDYEVVPGVQLLYTPGHSPGHQSLFIKTEQSGSVLLTIDASYTKENFEDEVPFAGFDPELALSSIKRLKEVVKKEKPIIFFGHDIEQEKSCRVFPEYI 2brb A 2.1 BS01 PFQ A 1 L15 G16 V23 A36 E85 C87 L137 L14 G15 V22 A35 E81 C83 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=13.7uM remove_due_to_license_issue IC50=20900nM O14757 15974586 1277 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP 2brc A 1.6 BS01 CT5 A 1 N37 A41 D79 I82 G83 M84 F124 T171 L173 N37 A41 D79 I82 G83 M84 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 ic50=7.1uM remove_due_to_license_issue P02829 15955698 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2brg A 2.1 BS01 DFY A 1 L15 G16 A36 E85 Y86 C87 G90 E91 L9 G10 A30 E73 Y74 C75 G78 E79 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=6.1uM remove_due_to_license_issue IC50=6100nM O14757 15974586 1270 EDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2brh A 2.1 BS01 DFW A 1 L15 G16 V23 E85 C87 G90 E91 L137 L10 G11 V18 E71 C73 G76 E77 L123 D130 K132 E134 N135 D148 T170 D116 K118 E120 N121 D134 T156 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=22.9uM remove_due_to_license_issue IC50=22900nM O14757 15974586 1272 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 2brm A 2.2 BS01 DFZ A 1 L15 G16 V23 A36 E85 C87 G90 L137 S147 L9 G10 V17 A30 E74 C76 G79 L126 S136 D130 K132 E134 N135 D148 T170 D119 K121 E123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=1.3uM remove_due_to_license_issue IC50=2300nM O14757 15974586 1275 EDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAK 2brn A 2.8 BS01 DF1 A 1 L15 G16 V23 A36 E85 C87 G90 L137 S147 L10 G11 V18 A31 E77 C79 G82 L129 S139 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=5500nM O14757 15974586 1277 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP 2bro A 2.2 BS01 DF2 A 1 L15 G16 V23 E85 C87 G90 L137 L14 G15 V22 E81 C83 G86 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.4uM remove_due_to_license_issue IC50=1400nM O14757 15974586 1277 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP 2brp A 2.0 BS01 SIE A 1 N290 W291 E388 H399 Y408 R462 R466 N580 N121 W122 E219 H230 Y239 R293 R297 N411 N349 H399 Y408 R462 E577 N180 H230 Y239 R293 E408 4.2.2.1 0003824,0005576,0005975,0016829,0030246 ic50>100uM remove_due_to_license_issue Q54873 16638841 1000 VKDTYTDRLDDWNGIIAGNQYYDSKNDQMAKLNQELEGKVADSLSSISSQADRIYLWEKFSNYKTSANLTATYRKLEEMAKQVTNPSSRYYQDETVVRTVRDSMEWMHKHVYNSEKSIVGNWWDYEIGTPRAINNTLSLMKEYFSDEEIKKYTDVIEKFVPDPEHFRKTTDNPFKALGGNLVDMGRVKVIAGLLRKDDQEISSTIRSIEQVFKLVDQGEGFYQDGSYIDHTNVAYTGAYGNVLIDGLSQLLPVIQKTKNPIDKDKMQTMYHWIDKSFAPLLVNGELMDMSRGRSISRANSEGHVAAVEVLRGIHRIADMSEGETKQRLQSLVKTIVQSDSYYDVFKNLKTYKDISLMQSLLSDAGVASVPRTSYLSAFNKMDKTAMYNAEKGFGFGLSLFSSRTLNYEHMNKENKRGWYTSDGMFYLYNGDLSHYSDGYWPTVNPYKMPGTTETDAKRADSDTGKVLPSAFVGTSKLDDANATATMDFTNWNQTLTAHKSWFMLKDKIAFLGSNIQNTSTDTAATTIDQRKLESSNPYKVYVNDKEASLTEQEKDYPETQSVFLESSDSKKNIGYFFFKKSSISMSKALQKGAWKDINEGQSDKEVENEFLTISQAHKQNGDSYGYMLIPNVDRATFNQMIKELESSLIENNETLQSVYDAKQGVWGIVKYDDSVSTISNQFQVLKRGVYTIRKEGDEYKIAYYNPETQESAPDQEVFKKL 2bsq A 3.0 BS01 dna I 0 H142 H143 H142 H143 3.1.-.- 0000287,0003677,0004518,0004540,0005515,0044001,0046872 remove_due_to_license_issue Q5F882 16982615 1 ~ 36 MILLDTNVISEPLRPQPNERVVAWLDSLILEDVYLSAITVAEMRLGVALLLNGKKKNVLHERMEQSILPLFAGRILPFDEPVAAIYAQIRSYAKTHGKEIAAADGYIAATAKQHSMTVATRDTGSFFAADVAVFNPWHLEHHH 2bsq E 3.0 BS01 dna I 0 S3 V5 R7 S2 V4 R6 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 1 ~ 36 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVELEDVRG 2bsq E 3.0 BS02 dna J 0 S27 T28 E29 R33 S26 T27 E28 R32 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 37 ~ 72 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVELEDVRG 2bsq F 3.0 BS01 dna I 0 V5 R7 V4 R6 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 1 ~ 36 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVELE 2bsq F 3.0 BS02 dna J 0 R22 S27 T28 E29 R33 R21 S26 T27 E28 R32 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 37 ~ 72 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVELE 2bsq G 3.0 BS01 dna I 0 T28 E29 R33 T27 E28 R32 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 1 ~ 36 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVELEDVR 2bsq G 3.0 BS02 dna J 0 S3 R7 S2 R6 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 37 ~ 72 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVELEDVR 2bsq H 3.0 BS01 dna I 0 S27 T28 E29 R33 L64 S26 T27 E28 R32 L63 ? 0003677,0005515,0006355,0042803,0043565,0044001 remove_due_to_license_issue Q5F881 16982615 1 ~ 36 ASVVIRNLSEATHNAIKFRARAAGRSTEAEIRLILDNIAKAQQTVRLGSMLASIGQEIGGVEL 2bt9 A 0.94 BS01 MFU A 1 R17 E28 G39 A40 W76 W81 R17 E28 G39 A40 W76 W81 ? Kd=0.64uM remove_due_to_license_issue Q8XXK6 15923179 1091 SSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSTN 2bt9 A 0.94 BS02 MFU A 2 R62 E73 G84 A85 R62 E73 G84 A85 ? Kd=0.64uM remove_due_to_license_issue Q8XXK6 15923179 1092 SSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSTN 2bt9 A 0.94 BS03 MFU C 2 I16 W31 W36 I16 W31 W36 ? Kd=0.64uM remove_due_to_license_issue Q8XXK6 15923179 1091 SSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSTN 2btr A 1.85 BS01 U73 A 1 I10 A31 F80 F82 L83 H84 L134 I10 A31 F69 F71 L72 H73 L123 D127 K129 Q131 N132 D145 T165 D116 K118 Q120 N121 D134 T142 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=95nM remove_due_to_license_issue P24941 16260160 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2bts A 1.99 BS01 U32 A 1 I10 A31 L83 H84 Q85 D86 K89 L134 I10 A31 L74 H75 Q76 D77 K80 L125 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T141 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=20nM remove_due_to_license_issue P24941 16260160 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2bu1 A 2.2 BS01 rna R 0 T45 C46 S47 R49 S51 T59 K61 E63 Y85 N87 T45 C46 S47 R49 S51 T59 K61 E63 Y85 N87 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2bu1 B 2.2 BS01 rna R 0 T45 S47 R49 S51 S52 N55 K57 T59 K61 T91 T45 S47 R49 S51 S52 N55 K57 T59 K61 T91 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2bu1 C 2.2 BS01 rna S 0 T45 C46 S47 S51 T59 K61 E63 Y85 N87 T45 C46 S47 S51 T59 K61 E63 Y85 N87 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2bu5 A 2.35 BS01 TF1 A 1 L23 Q27 F31 S41 F44 L45 L160 Q163 C384 L18 Q22 F26 S34 F37 L38 L153 Q156 C355 H239 E243 K246 N247 H224 E228 K231 N232 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 remove_due_to_license_issue EC50=57nM, IC50=17nM Q15119 16401071 1386 GSAPKYIEHFSKFSPSPLSMKQFLDFSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTAPGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWC 2bua A 2.56 BS01 007 A 1 E205 E206 Y547 S630 Y662 Y666 E167 E168 Y509 S592 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue IC50=30000nM P22411 16376544 1767 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 2bub A 2.66 BS01 FPB A 1 R125 E205 E206 S209 F357 Y547 Y662 Y666 N710 R87 E167 E168 S171 F319 Y509 Y624 Y628 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=90nM P27487 16376544 1771 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2buc A 2.5 BS01 008 A 1 E205 E206 S209 F357 R358 Y547 Y662 Y666 N710 E167 E168 S171 F319 R320 Y509 Y624 Y628 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 ic50=23nM remove_due_to_license_issue P22411 16376544 1767 SRRTYTLTDYLKSTFRVKFYTLQWISDHEYLYKQENNILLFNAEYGNSSIFLENSTFDELGYSTNDYSVSPDRQFILFEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWITWSPVGHKLAYVWNNDIYVKNEPNLSSQRITWTGKENVIYNGVTDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRIPYPKAGAENPTVKFFVVDTRTLSPNASVTSYQIVPPASVLIGDHYLCGVTWVTEERISLQWIRRAQNYSIIDICDYDESTGRWISSVARQHIEISTTGWVGRFRPAEPHFTSDGNSFYKIISNEEGYKHICHFQTDKSNCTFITKGAWEVIGIEALTSDYLYYISNEHKGMPGGRNLYRIQLNDYTKVTCLSCELNPERCQYYSASFSNKAKYYQLRCFGPGLPLYTLHSSSSDKELRVLEDNSALDKMLQDVQMPSKKLDVINLHGTKFWYQMILPPHFDKSKKYPLLIEVYAGPCSQKVDTVFRLSWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEATRQFSKMGFVDDKRIAIWGWSYGGYVTSMVLGAGSGVFKCGIAVAPVSKWEYYDSVYTERYMGLPTPEDNLDYYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQLSKALVDAGVDFQTMWYTDEDHGIASNMAHQHIYTHMSHFLKQCFSLP 2bvd A 1.6 BS01 ISX A 1 W14 F41 E70 E109 Y115 Y185 W187 E222 F256 E258 K260 E261 W7 F34 E63 E102 Y108 Y178 W180 E215 F249 E251 K253 E254 3.2.1.4 0004553,0006080,0016985 Ki=1uM remove_due_to_license_issue P16218 15987675 1284 GLKIGAWVGTQPSESAIKSFQELQGRKLDIVHQFINWSTDFSWVRPYADAVYNNGSILMITWEPWEYNTVDIKNGKADAYITRMAQDMKAYGKEIWLRPLHEANGDWYPWAIGYSSRVNTNETYIAAFRHIVDIFRANGATNVKWVFNVNCDNVGNGTSYLGHYPGDNYVDYTSIDGYNWGTTQSWGSQWQSFDQVFSRAYQALASINKPIIIAEFASAEIGGNKARWITEAYNSIRTSYNKVIAAVWFHENKETDWRINSSPEALAAYREAIGAL 2bve A 2.2 BS01 PH5 A 1 W2 R97 S103 R105 W106 L107 W2 R97 S103 R105 W106 L107 ? ic50=215uM remove_due_to_license_issue Q62230 17137591 1120 TWGVSSPKNVQGLSGSCLLIPCIFSYPADVPVSNGITAIWYYDYSGKRQVVIHSGDPKLVDKRFRGRAELMGNMDHKVCNLLLKDLKPEDSGTYNFRFEISDSNRWLDVKGTTVTVTTD 2bvr H 1.25 BS03 4CP H 1 W60D A190 C191 E192 V213 W215 G216 G219 C220 G226 F227 W50 A193 C194 E195 V218 W220 G221 G223 C224 G231 F232 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2bvs H 1.4 BS03 2CE H 1 H57 Y60A W60D Y134 A190 C191 E192 V213 W215 G216 G219 G226 F227 H43 Y47 W50 Y134 A194 C195 E196 V219 W221 G222 G224 G232 F233 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2bvx H 3.2 BS03 5CB H 1 H57 Y60A W60D N98 L99 I174 A190 C191 E192 V213 S214 W215 G216 F227 H43 Y47 W50 N95 L96 I173 A194 C195 E196 V219 S220 W221 G222 F233 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2bw7 A 2.3 BS03 ECS A 1 F1015 D1017 N1146 A1149 R1150 E1153 F14 D16 N145 A148 R149 E152 2.7.13.3 0009190,0035556 ic50~2uM remove_due_to_license_issue O32393 16002394 2203 SHMRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGRNEVPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 2bw7 B 2.3 BS04 ECS B 1 F1015 D1017 A1062 N1146 A1149 R1150 E1153 F12 D14 A59 N140 A143 R144 E147 2.7.13.3 0009190,0035556 ic50~2uM remove_due_to_license_issue O32393 16002394 2203 MRPEPRLITILFSDIVGFTRMSNALQSQGVAELLNEYLGEMTRAVFENQGTVDKFVGDAIMALYGAPEEMSPSEQVRRAIATARQMLVALEKLNQGWQERGLVGRPPVRFRCGIHQGMAVVGLFGSQERSDFTAIGPSVNIAARLQEATAPNSIMVSAMVAQYVPDEEIIKREFLELKGIDEPVMTCVINPNM 2bxt H 1.83 BS03 C2D H 1 H57 Y60A E97A N98 L99 Y134 I174 D189 A190 E192 S195 S214 W215 G216 E217 G219 G226 F227 H43 Y47 E94 N95 L96 Y134 I173 D193 A194 E196 S199 S220 W221 G222 E223 G224 G232 F233 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2bxu H 2.8 BS03 C1D H 1 H57 Y60A W60D N98 Y134 D189 A190 E192 S195 W215 G216 H43 Y47 W50 N95 Y134 D193 A194 E196 S199 W221 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2byh A 1.9 BS01 2D7 A 1 N51 A55 D93 G97 M98 N106 G135 V136 F138 T184 N41 A45 D83 G87 M88 N96 G125 V126 F128 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.258uM remove_due_to_license_issue P07900 16213716 1226 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 2byi A 1.6 BS01 2DD A 1 N51 A55 D93 G97 M98 L107 V136 F138 T184 N41 A45 D83 G87 M88 L97 V126 F128 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.461uM remove_due_to_license_issue P07900 16213716 1226 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 2byr A 2.45 BS01 MLK A 1 Y93 S94 K143 W147 V148 Y188 C190 Y195 Y98 S99 K148 W152 V153 Y193 C195 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=2.8nM remove_due_to_license_issue Q8WSF8 16193063 301 DDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2byr A 2.45 BS02 MLK B 1 M116 I118 S167 M121 I123 S172 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=2.8nM remove_due_to_license_issue Q8WSF8 16193063 301 DDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2byr E 2.45 BS01 MLK A 1 I118 S167 I124 S173 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=2.8nM remove_due_to_license_issue Q8WSF8 16193063 301 DDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2byr E 2.45 BS02 MLK E 1 Y93 S94 K143 W147 V148 Y188 C190 Y195 Y99 S100 K149 W153 V154 Y194 C196 Y201 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=2.8nM remove_due_to_license_issue Q8WSF8 16193063 301 DDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2bys A 2.05 BS01 LOB A 1 Y93 G145 S146 W147 Y188 C190 C191 Y195 Y90 G142 S143 W144 Y185 C187 C188 Y192 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.3nM remove_due_to_license_issue Q8WSF8 16193063 301 SQANLMRLKSDLFNRSYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2bys A 2.05 BS02 LOB B 1 Y55 V108 M116 I118 Y52 V105 M113 I115 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.3nM remove_due_to_license_issue Q8WSF8 16193063 301 SQANLMRLKSDLFNRSYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2bys E 2.05 BS01 LOB A 1 Y55 V108 M116 I118 Y53 V106 M114 I116 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.3nM remove_due_to_license_issue Q8WSF8 16193063 301 KLHSQANLMRLKSDLFNYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2bys E 2.05 BS02 LOB E 1 Y93 G145 S146 W147 Y188 C191 Y195 Y91 G143 S144 W145 Y186 C189 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.3nM remove_due_to_license_issue Q8WSF8 16193063 301 KLHSQANLMRLKSDLFNYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2bz5 A 1.9 BS01 AB4 A 1 N51 D54 A55 D93 I96 G97 M98 N106 L107 F138 T184 N36 D39 A40 D78 I81 G82 M83 N91 L92 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 16202589 1226 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 2bz6 H 1.6 BS01 346 H 1 H57 D102 D189 S190 K192 S195 S214 W215 G216 G219 H41 D90 D186 S187 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=0.081uM remove_due_to_license_issue Ki=88nM P08709 16621574 1258 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2bza A 1.9 BS02 ABN A 1 D189 S190 C191 Q192 W215 G219 D171 S172 C173 Q174 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=1.58mM remove_due_to_license_issue P00760 10651279 703 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2bzz A 0.98 BS01 AP5 A 1 Q1014 H1015 K1038 Q1040 N1070 H1082 A1110 V1128 H1129 L1130 Q15 H16 K39 Q41 N71 H83 A111 V129 H130 L131 H1015 K1038 H1129 H16 K39 H130 4.6.1.18 0003676 Ki=0.37uM remove_due_to_license_issue P10153 16401072 2135 MKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII 2c02 A 2.0 BS01 ADP A 1 Q14 H15 K38 R68 N70 A110 H129 Q15 H16 K39 R69 N71 A111 H130 H15 K38 H129 H16 K39 H130 4.6.1.18 0003676 Ki=70uM remove_due_to_license_issue P10153 16401072 1135 MKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII 2c0o A 2.85 BS01 L2G A 1 L247 V255 A267 V268 K269 F281 I310 T312 F314 M315 S319 D322 L367 D378 F379 L381 L189 V197 A209 V210 K211 F223 I252 T254 F256 M257 S261 D264 L309 D320 F321 L323 D360 R362 A364 N365 D378 D302 R304 A306 N307 D320 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1220nM P08631 16216497 1506 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 2c1a A 1.95 BS02 I5S A 1 G50 T51 G52 G55 R56 V57 A70 M120 Y122 V123 E127 E170 N171 L173 T183 D184 F327 G37 T38 G39 G42 R43 V44 A57 M107 Y109 V110 E114 E157 N158 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=0.17uM remove_due_to_license_issue IC50=170nM P00517 16249095 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2c1b A 2.0 BS02 CQP A 1 L49 T51 G52 R56 V57 A70 K72 M120 Y122 V123 E127 E170 N171 L173 T183 F327 L36 T38 G39 R43 V44 A57 K59 M107 Y109 V110 E114 E157 N158 L160 T170 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=0.4uM remove_due_to_license_issue IC50=400nM P00517 16249095 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2c1p A 2.0 BS01 FNZ B 1 G91 F94 G96 F99 ? 0046872 remove_due_to_license_issue Q58EU8 16427081 1215 ELVMTQSPLTLSVTIGQPASISCKSSQSLLYSNGKTYLNWLLQRPGQSPKRLIYLVSKLDSGDPDRFTGSGSGTDFTLKISRVEAEDLGIYYCVQGSHFPPTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRN 2c1p B 2.0 BS01 FNZ B 1 N35 W47 M50 D95 N34 W46 M49 D98 remove_due_to_license_issue 16427081 1215 VQLQQSGAELVRPGTSVKLSCKASGYSFTNYWMNWLRQRPGQGLDWIGMIHPSDSETRLNQKFKDKATLTVDRSSSTAYIQLSSPTSEDSAVYYCARDDYDGAFWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPAPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRD 2c1q A 2.1 BS01 BTN A 1 L14 S16 Y33 T35 V37 T38 W71 S76 T78 F80 W98 N119 L14 S16 Y33 T35 V37 T38 W69 S74 T76 F78 W96 N117 0009374 Kd~0.1pM remove_due_to_license_issue 17343730 1126 TRKCELQGLWRNELGSNMTISALDVAGTFSGSYQTAVTATNKQILVSPLKGAQQPPKGQQPTFGFTVQWQFADSTTVFVGQCFVDRRGKEMLEMAWLLREEVPSRKDTWKATRVGTNVFTRVK 2c2e A 2.61 BS01 dna P 0 A102 E106 G185 G187 I189 T190 K193 I295 R298 R300 T301 I341 A102 E106 G185 G187 I189 T190 K193 I295 R298 R300 T301 I341 2.7.7.7 0000287,0003677,0003684,0003887,0005737,0006260,0006261,0006281,0006974,0034061,0042276,0046872 remove_due_to_license_issue Q97W02 16306039 1 ~ 14 MIVLFVDFDYFYAQVEEVLNPSLKGKPVVVCVFSGRFEDSGAVATANYEARKFGVKAGIPIVEAKKILPNAVYLPMRKEVYQQVSSRIMNLLREYSEKIEIASIDEAYLDISDKVRDYREAYNLGLEIKNKILEKEKITVTVGISKNKVFAKIAADMAKPNGIKVIDDEEVKRLIRELDIADVPGIGNITAEKLKKLGINKLVDTLSIEFDKLKGMIGEAKAKYLISLARDEYNEPIRTRVRKSIGRIVTMKRNSRNLEEIKPYLFRAIEESYYKLDKRIPKAIHVVAVTEDLDIVSRGRTFPHGISKETAYSESVKLLQKILEEDERKIRRIGVRFSKFI 2c2e A 2.61 BS02 dna T 0 V32 S34 S40 G41 A42 G218 A220 K221 R240 R242 S244 I245 G246 R247 I248 T250 R331 R332 R336 V32 S34 S40 G41 A42 G218 A220 K221 R240 R242 S244 I245 G246 R247 I248 T250 R331 R332 R336 2.7.7.7 0000287,0003677,0003684,0003887,0005737,0006260,0006261,0006281,0006974,0034061,0042276,0046872 remove_due_to_license_issue Q97W02 16306039 4 ~ 18 MIVLFVDFDYFYAQVEEVLNPSLKGKPVVVCVFSGRFEDSGAVATANYEARKFGVKAGIPIVEAKKILPNAVYLPMRKEVYQQVSSRIMNLLREYSEKIEIASIDEAYLDISDKVRDYREAYNLGLEIKNKILEKEKITVTVGISKNKVFAKIAADMAKPNGIKVIDDEEVKRLIRELDIADVPGIGNITAEKLKKLGINKLVDTLSIEFDKLKGMIGEAKAKYLISLARDEYNEPIRTRVRKSIGRIVTMKRNSRNLEEIKPYLFRAIEESYYKLDKRIPKAIHVVAVTEDLDIVSRGRTFPHGISKETAYSESVKLLQKILEEDERKIRRIGVRFSKFI 2c3i B 1.9 BS02 IYZ B 1 F49 A65 K67 L174 I185 D186 F13 A29 K31 L135 I146 D147 D167 K169 N172 D186 L193 T204 D128 K130 N133 D147 L154 T165 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Kd=25nM remove_due_to_license_issue IC50=61nM, Kd=25nM P11309 17638903 1306 QYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGEGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 2c3j A 2.1 BS01 DBQ A 1 V23 A36 K38 E85 Y86 C87 L137 S147 D148 V15 A28 K30 E72 Y73 C74 L124 S134 D135 D130 K132 E134 N135 D148 T170 D117 K119 E121 N122 D135 T157 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.659uM remove_due_to_license_issue IC50=725nM O14757 16289938 1271 VEDWDLVQTLGEGEVQLAVNRVTEEAVAVKIVDMKRENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2c3k A 2.6 BS01 ABO A 1 L15 A36 E55 N59 V68 L84 E85 Y86 C87 G90 L137 D148 F149 L10 A31 E47 N51 V60 L76 E77 Y78 C79 G82 L129 D140 F141 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=42nM, Ki=26nM O14757 16289938 1271 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2c3l A 2.35 BS01 IDZ A 1 L15 A36 E85 Y86 C87 G90 L137 L14 A35 E77 Y78 C79 G82 L129 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=8.58uM remove_due_to_license_issue Ki=8580nM, IC50=6296nM O14757 16289938 1274 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 2c4f H 1.72 BS02 GIL H 1 H57 T99 D189 S190 K192 G193 S195 V213 S214 W215 G216 H41 T87 D186 S187 K189 G190 S192 V210 S211 W212 G213 3.4.21.21 0004252,0006508 remove_due_to_license_issue IC50=20nM P08709 16289811 302 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2c4g A 2.7 BS01 514 A 1 I10 A31 K33 F80 L83 H84 Q85 D86 L134 I14 A35 K37 F84 L87 H88 Q89 D90 L138 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 16290148 306 PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 2c4q A 2.38 BS01 rna R 0 T45 C46 S47 R49 S51 T59 K61 E63 Y85 T45 C46 S47 R49 S51 T59 K61 E63 Y85 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c4q B 2.38 BS01 rna R 0 V29 T45 S47 R49 S51 S52 N55 K57 T59 K61 V29 T45 S47 R49 S51 S52 N55 K57 T59 K61 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c4q C 2.38 BS01 rna S 0 T45 C46 S47 S51 T59 K61 E63 Y85 T45 C46 S47 S51 T59 K61 E63 Y85 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c4w A 1.55 BS01 GAJ A 1 L11 L14 D18 G78 H82 H102 L103 T104 I106 R113 L20 L23 D27 G87 H91 H111 L112 T113 I115 R122 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P18 N19 R26 Y31 N85 A88 E109 H111 R118 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=20uM remove_due_to_license_issue Q48255 16480265 1160 AGLVPRGSHMKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSEYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKNNP 2c4y A 2.68 BS01 rna R 0 T45 C46 S47 S51 T59 E63 Y85 T45 C46 S47 S51 T59 E63 Y85 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c4y B 2.68 BS01 rna R 0 T45 S47 R49 S51 S52 N55 K57 T59 K61 T45 S47 R49 S51 S52 N55 K57 T59 K61 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 2 ~ 18 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c4y C 2.68 BS01 rna S 0 T45 C46 S47 T59 K61 E63 Y85 T45 C46 S47 T59 K61 E63 Y85 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 4 ~ 16 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c50 A 2.65 BS01 rna R 0 T45 C46 S47 T59 Y85 T45 C46 S47 T59 Y85 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 3 ~ 16 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c50 B 2.65 BS01 rna R 0 T45 S47 R49 S51 S52 N55 K57 T59 K61 T45 S47 R49 S51 S52 N55 K57 T59 K61 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 3 ~ 16 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c50 C 2.65 BS01 rna S 0 K43 T45 S47 T59 Y85 K43 T45 S47 T59 Y85 ? 0003723,0005198,0006417,0019028,0039617,0042802,1904972 remove_due_to_license_issue P03612 11720290 4 ~ 16 ASNFTQFVLVDNGGTGDVTVAPSNFANGVAEWISSNSRSQAYKVTCSVRQSSAQNRKYTIKVEVPKVATQTVGGVELPVAAWRSYLNMELTIPIFATNSDCELIVKAMQGLLKDGNPIPSAIAANSGIY 2c57 A 3.1 BS01 FA1 A 1 N76 G78 A79 H82 H102 L103 T104 R113 N82 G84 A85 H88 H108 L109 T110 R119 P9 N10 N76 A79 E100 H102 R109 P22 N23 N82 A85 E106 H108 R115 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue Kd=370000nM Q48255 16480265 1159 GSSHHHHHHSSSHMKILVIQGPNLNMLGGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKNN 2c57 B 3.1 BS01 FA1 B 1 N76 G78 A79 H82 H102 L103 T104 R113 N71 G73 A74 H77 H97 L98 T99 R108 P9 N10 R17 N76 A79 E100 H102 R109 P9 N10 R17 N71 A74 E95 H97 R104 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue Kd=370000nM Q48255 16480265 1159 MKILVIQGPNLNMLGHRGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKNN 2c5n A 2.1 BS01 CK8 A 1 Y15 A31 F80 E81 L83 H84 Q85 K89 L134 Y15 A31 F80 E81 L83 H84 Q85 K89 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.22uM remove_due_to_license_issue IC50=2.2e+2nM, Ki=220nM P24941 16492568 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2c5o A 2.1 BS01 CK2 A 1 A31 F82 L83 L134 A31 F82 L83 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=6.5uM remove_due_to_license_issue Ki=6500nM, Kd=30300nM, IC50=6.50e+3nM, kon=8.22E+04M-1-s-1, koff=1.42E+00s-1 P24941 16492568 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2c5x A 2.9 BS01 MTW A 1 V18 A31 F80 E81 F82 L83 H84 N132 L134 D145 V18 A31 F80 E81 F82 L83 H84 N132 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 16492568 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2c5y A 2.25 BS01 MTW A 1 I10 G11 E12 G13 V18 A31 K33 V64 E81 F82 L83 H84 Q85 L134 D145 I10 G11 E12 G13 V18 A31 K33 V57 E74 F75 L76 H77 Q78 L127 D138 D127 K129 Q131 N132 D145 T158 T165 D120 K122 Q124 N125 D138 T151 T158 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.25uM remove_due_to_license_issue P24941 16492568 1298 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 2c68 A 1.95 BS01 CT6 A 1 I10 G11 E12 G13 A31 K33 F82 L83 H84 K89 Q131 L134 I10 G11 E12 G13 A31 K33 F76 L77 H78 K83 Q125 L128 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1.8uM remove_due_to_license_issue P24941 16325401 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2c69 A 2.1 BS01 CT8 A 1 G11 E12 G13 V18 A31 K33 F82 L83 H84 Q131 L134 G11 E12 G13 V18 A31 K33 F76 L77 H78 Q125 L128 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=26uM remove_due_to_license_issue IC50=26000nM P24941 16325401 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2c6c A 2.0 BS04 24I A 1 R210 N257 D387 E424 E425 D453 S454 G518 Y552 H553 K699 Y700 R154 N201 D327 E364 E365 D393 S394 G458 Y486 H487 K631 Y632 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=30nM remove_due_to_license_issue Q04609 16467855 1767 NMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2c6e A 2.1 BS01 HPM A 1 K161 Q184 L209 A212 P213 G215 L262 D273 F274 W276 K36 Q59 L84 A87 P88 G90 L137 D148 F149 W151 D255 K257 E259 N260 D273 T291 D130 K132 E134 N135 D148 T154 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=0.80nM O14965 16337122 1389 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2c6g A 2.2 BS01 GLU A 1 R210 E424 G518 Y552 K699 Y700 R154 E362 G456 Y483 K628 Y629 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Q04609 16467855 1766 NMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2c6i A 1.8 BS01 DT1 A 1 I10 E12 G13 A31 K33 L83 H84 Q85 D86 K89 Q131 N132 L134 I10 E12 G13 A31 K33 L77 H78 Q79 D80 K83 Q125 N126 L128 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=11uM remove_due_to_license_issue IC50=11000nM P24941 16325401 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2c6k A 1.9 BS01 DT2 A 1 I10 A31 K33 L83 H84 Q85 D86 K89 L134 I10 A31 K33 L77 H78 Q79 D80 K83 L128 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.73uM remove_due_to_license_issue IC50=730nM P24941 16325401 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2c6l A 2.3 BS01 DT4 A 1 A31 K33 L83 H84 Q85 D86 K89 L134 D145 A31 K33 L76 H77 Q78 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T158 T165 D120 K122 Q124 N125 D138 T151 T158 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.27uM remove_due_to_license_issue IC50=270nM P24941 16325401 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2c6m A 1.9 BS01 DT5 A 1 I10 V18 A31 K33 E81 L83 H84 Q85 D86 K89 L134 I10 V18 A31 K33 E75 L77 H78 Q79 D80 K83 L128 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.35uM remove_due_to_license_issue IC50=350nM P24941 16325401 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2c6n A 3.0 BS02 LPR A 1 Q259 H331 A332 S333 H361 E362 K489 H491 T496 Y501 Q259 H331 A332 S333 H361 E362 K489 H491 T496 Y501 H331 A332 H361 E362 H365 E389 H491 Y501 H331 A332 H361 E362 H365 E389 H491 Y501 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue IC50=1.2nM P12821 16476442 705 LDPGLQPGNFSADEAGAQLFAQSYNSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQNFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSNMSRIYSTAKVCLPNKTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWNATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLQAGSSRPWQEVLKDMVGLDALDAQPLLKYFQPVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEGID 2c6o A 2.1 BS01 4SP A 1 I10 G13 V18 A31 L83 H84 D86 K89 Q131 L134 I10 G13 V18 A31 L77 H78 D80 K83 Q125 L128 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=6.0nM, Ki=6.0nM, Kd=1310nM P24941 16325401 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2c7a A 2.5 BS01 dna C 0 C577 H578 Y579 K588 K592 K617 G635 R637 K638 C15 H16 Y17 K26 K30 K55 G73 R75 K76 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 16931575 1 ~ 18 PQKICLICGDEASGCHYGVLTCGSCKVFFKRAMEGQHNYLCAGRNDCIVDKIRRKNCPACRLRKCCQAGMVLGGRKFK 2c7a A 2.5 BS02 dna D 0 G585 S586 R593 R616 R623 G23 S24 R31 R54 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 16931575 1 ~ 18 PQKICLICGDEASGCHYGVLTCGSCKVFFKRAMEGQHNYLCAGRNDCIVDKIRRKNCPACRLRKCCQAGMVLGGRKFK 2c7a B 2.5 BS01 dna C 0 S586 R593 R616 R623 K638 S24 R31 R54 R61 K76 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 16931575 1 ~ 18 PQKICLICGDEASGCHYGVLTCGSCKVFFKRAMEGQHNYLCAGRNDCIVDKIRRKNCPACRLRKCCQAGMVLGGRK 2c7a B 2.5 BS02 dna D 0 C577 H578 Y579 K588 K592 K617 G636 R637 C15 H16 Y17 K26 K30 K55 G74 R75 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 16931575 1 ~ 18 PQKICLICGDEASGCHYGVLTCGSCKVFFKRAMEGQHNYLCAGRNDCIVDKIRRKNCPACRLRKCCQAGMVLGGRK 2c80 A 2.3 BS01 GTX A 1 Y10 R16 W41 K45 R52 L53 E70 S71 Y110 L113 Y7 R13 W38 K42 R49 L50 E67 S68 Y107 L110 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=4.7uM remove_due_to_license_issue P30113 16777141 1212 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRAATPF 2c80 B 2.3 BS01 GTX B 1 Y10 F11 R16 W41 K45 R52 L53 E70 S71 Y110 F211 Y7 F8 R13 W38 K42 R49 L50 E67 S68 Y107 F208 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=4.7uM remove_due_to_license_issue P30113 16777141 1213 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRAATPF 2c8w B 1.96 BS03 C7M B 1 H57 Y60A W60D E97A N98 L99 A190 C191 E192 V213 W215 G216 G219 C220 G226 F227 H43 Y47 W50 E94 N95 L96 A192 C193 E194 V217 W219 G220 G222 C223 G230 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=3.7nM remove_due_to_license_issue P00734 16480269 1249 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 2c8x B 2.17 BS03 C5M B 1 H57 Y60A W60D L99 D189 A190 S195 V213 W215 G216 G226 F227 H43 Y47 W50 L96 D191 A192 S197 V217 W219 G220 G230 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=220nM remove_due_to_license_issue IC50=220nM P00734 16480269 1251 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 2c8y B 2.2 BS03 C3M B 1 H57 Y60A W60D N98 L99 W215 G216 H43 Y47 W50 N95 L96 W219 G220 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue IC50=100000nM P00734 16480269 1252 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 2c90 B 2.25 BS03 C1M B 1 A190 C191 E192 V213 W215 C220 G226 F227 A192 C193 E194 V217 W219 C223 G230 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=330uM remove_due_to_license_issue IC50=330000nM P00734 16480269 1250 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 2c92 A 1.6 BS01 TP6 A 1 W27 G58 A59 I60 E61 V81 V82 I83 G85 Q86 T87 W14 G45 A46 I47 E48 V68 V69 I70 G72 Q73 T74 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=474900M^-1 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c92 A 1.6 BS02 TP6 E 1 A113 N114 R128 A100 N101 R115 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=474900M^-1 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c92 B 1.6 BS01 TP6 A 1 A113 N114 R128 K138 A100 N101 R115 K125 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=474900M^-1 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c92 B 1.6 BS02 TP6 B 1 W27 G58 A59 I60 E61 V81 V82 I83 G85 Q86 T87 W14 G45 A46 I47 E48 V68 V69 I70 G72 Q73 T74 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=474900M^-1 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c93 B 2.2 BS03 C4M B 1 H57 Y60A W60D L99 E192 W215 G216 H43 Y47 W50 L96 E194 W219 G220 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=12uM remove_due_to_license_issue IC50=12000nM P00734 16480269 1251 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 2c94 A 1.9 BS01 TSF A 1 W27 G58 A59 I60 E61 V81 V82 G85 Q86 T87 W13 G44 A45 I46 E47 V67 V68 G71 Q72 T73 H89 H75 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=6540000M^-1 remove_due_to_license_issue P9WHE9 16984393 701 ASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c94 A 1.9 BS02 TSF E 1 A113 N114 R128 A99 N100 R114 H89 H75 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=6540000M^-1 remove_due_to_license_issue P9WHE9 16984393 701 ASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c94 B 1.9 BS01 TSF A 1 A113 N114 R128 K138 A99 N100 R114 K124 H89 H75 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=6540000M^-1 remove_due_to_license_issue P9WHE9 16984393 701 ASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c94 B 1.9 BS02 TSF B 1 W27 G58 A59 I60 E61 V81 V82 I83 G85 T87 W13 G44 A45 I46 E47 V67 V68 I69 G71 T73 H89 H75 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=6540000M^-1 remove_due_to_license_issue P9WHE9 16984393 701 ASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c97 A 2.0 BS01 JCL A 1 W27 H28 G58 A59 V81 V82 I83 G85 Q86 T87 W14 H15 G45 A46 V68 V69 I70 G72 Q73 T74 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=1380000M^-1 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c97 B 2.0 BS01 JCL B 1 W27 H28 G58 A59 V81 V82 I83 G85 Q86 T87 W14 H15 G45 A46 V68 V69 I70 G72 Q73 T74 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ka=1380000M^-1 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9b A 2.75 BS01 PUG A 1 W27 G58 A59 I60 E61 V81 V82 H89 W14 G45 A46 I47 E48 V68 V69 H76 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9b A 2.75 BS02 PUG E 1 A113 N114 K138 A100 N101 K125 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9b B 2.75 BS01 PUG A 1 A113 N114 A100 N101 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9b B 2.75 BS02 PUG B 1 W27 A59 I60 E61 V81 V82 H89 W14 A46 I47 E48 V68 V69 H76 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 701 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9d A 2.8 BS01 PHR A 1 W27 A59 I60 E61 V81 V82 I83 G85 Q86 T87 H89 F90 W14 A46 I47 E48 V68 V69 I70 G72 Q73 T74 H76 F77 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 791 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9d A 2.8 BS02 PHR E 1 N114 R128 N101 R115 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 791 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9d B 2.8 BS01 PHR A 1 N114 R128 N101 R115 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 791 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2c9d B 2.8 BS02 PHR B 1 W27 G58 A59 I60 E61 V81 G85 Q86 T87 H89 W14 G45 A46 I47 E48 V68 G72 Q73 T74 H76 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 remove_due_to_license_issue P9WHE9 16984393 791 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2ca8 A 2.49 BS01 GSH A 1 Y10 R16 W41 K45 R52 L53 E70 S71 Y7 R13 W38 K42 R49 L50 E67 S68 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=22uM remove_due_to_license_issue P30113 16777141 1212 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRAATPF 2cax A 2.9 BS01 dna Y 0 H37 K41 N50 V51 K52 H19 K23 N32 V33 K34 ? 0006355 remove_due_to_license_issue Q57468 16528102 21 ~ 38 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cax B 2.9 BS01 dna U 0 N50 V51 K52 N29 V30 K31 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 KDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cax B 2.9 BS02 dna Y 0 K28 T29 V30 R31 K7 T8 V9 R10 ? 0006355 remove_due_to_license_issue Q57468 16528102 21 ~ 38 KDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cax C 2.9 BS01 dna U 0 K41 N50 V51 K52 K23 N32 V33 K34 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cax C 2.9 BS02 dna Y 0 K28 T29 R31 K10 T11 R13 ? 0006355 remove_due_to_license_issue Q57468 16528102 21 ~ 38 MAKKDIMGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cax D 2.9 BS01 dna U 0 K28 T29 R31 K4 T5 R7 ? 0006355 remove_due_to_license_issue Q57468 16528102 1 ~ 18 MGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cax D 2.9 BS02 dna Y 0 H37 K41 N50 V51 K52 H13 K17 N26 V27 K28 ? 0006355 remove_due_to_license_issue Q57468 16528102 21 ~ 38 MGDKTVRVRADLHHIIKIETAKNGGNVKEVMDQALEEYIRKYLPDKL 2cbj A 2.35 BS01 OAN A 1 G187 K218 D297 D298 Y335 V370 W394 N396 D401 Y402 W490 G148 K179 D258 D259 Y296 V331 W355 N357 D362 Y363 W451 3.2.1.169 Ki=5.4nM remove_due_to_license_issue Q0TR53 16541109 1625 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYNRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2cbj A 2.35 BS02 OAN B 1 L512 S513 L473 S474 3.2.1.169 Ki=5.4nM remove_due_to_license_issue Q0TR53 16541109 1625 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYNRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2cbr A 2.8 BS01 A80 A 1 T54 T56 R59 D77 L120 R131 Y133 T54 T56 R59 D77 L120 R131 Y133 ? 0001972,0005501,0005504,0005634,0005737,0005829,0008289,0015908,0016918,0019841,0032991,0042802 remove_due_to_license_issue P62964 10531482 201 PNFAGTWKMRSSENFDELLKALGVNAMLRKVAVAAASKPHVEIRQDGDQFYIKTSTTVRTTEINFKVGEGFEEETVDGRKCRSLPTWENENKIHCTQTLLEGDGPKTYWTRELANDELILTFGADDVVCTRIYVRE 2cbs A 2.1 BS01 R13 A 1 V24 A32 T56 R59 V76 L121 R132 Y134 V24 A32 T56 R59 V76 L121 R132 Y134 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 ic50=6nM remove_due_to_license_issue P29373 10531482 200 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKTSTTVRTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTRELTNDGELILTMTADDVVCTRVYVRE 2cbu A 1.85 BS01 CTS A 1 Q20 H121 N165 E166 Y295 W324 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y291 W318 E345 W392 E399 W400 F408 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N289 Y291 E345 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=2.1uM remove_due_to_license_issue Q08638 16628756 1447 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLED 2cbv A 1.95 BS01 CGB A 1 Q20 H121 W122 N165 E166 E351 W398 E405 W406 Q18 H119 W120 N163 E164 E348 W395 E402 W403 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N290 Y292 E348 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=3.3uM remove_due_to_license_issue Q08638 16628756 1447 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLED 2cbz A 1.5 BS02 ATP A 1 W653 T660 V680 G681 C682 G683 K684 S685 S686 Q713 W12 T19 V39 G40 C41 G42 K43 S44 S45 Q72 7.6.2.2,7.6.2.3 0005524,0016887 Kd=118uM remove_due_to_license_issue P33527 16697012 1873 NSITVRNATFTWARSDPPTLNGITFSIPEGALVAVVGQVGCGKSSLLSALLAEMDKVEGHVAIKGSVAYVPQQAWIQNDSLRENILFGCQLEEPYYRSVIQACALLPDLEILPSGDRTEIGEKGVNLSGGQKQRVSLARAVYSNADIYLFDDPLSAVDAHVGKHIFENVIGPKGMLKNKTRILVTHSMSYLPQVDVIIVMSGGKISEMGSYQELLARDGAFAEFLRTYAS 2ccb A 1.65 BS01 RBF A 1 F3 V35 W36 F2 V34 W35 ? 0005737,0005829 Kd=35.76nM remove_due_to_license_issue B0R5M0 16460756 1067 VFKKVLLTGTSEESFTAAADDAIDRAEDTLDNVVWAEVVDQGVEIGAVEERTYQTEVQVAFELD 2ccs A 1.79 BS01 4BH A 1 N51 A55 D93 I96 G97 M98 L107 G108 F138 T184 E223 N36 A40 D78 I81 G82 M83 L92 G93 F123 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=2uM remove_due_to_license_issue P07900 16480864 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2cct A 2.3 BS01 2E1 A 1 N51 A55 K58 D93 I96 G97 M98 L107 G108 F138 T184 V186 E223 N36 A40 K43 D78 I81 G82 M83 L92 G93 F123 T169 V171 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=6.3uM remove_due_to_license_issue P07900 16480864 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2ccu A 2.7 BS01 2D9 A 1 S50 N51 D54 A55 D93 G97 M98 F138 T184 E223 S35 N36 D39 A40 D78 G82 M83 F123 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 16480864 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2ccz A 2.7 BS01 dna C 0 E32 R34 W47 Q49 N85 G86 K89 E38 R40 W53 Q55 N91 G92 K95 ? 0003677,0003697,0005515,0006260,0006268,0006269,0006270,0006276,0009314,0030894,0031297,0042802,1990077,1990099,1990158 remove_due_to_license_issue P07013 16899446 1 ~ 15 MDPNSLMTNRLVLSGTVCRAPLRKVSPSGIPHCQFVLEHRSVQEEAGFHRQAWCQMPVIVSGHENQAITHSITVGSRITVQGFISCHKAKNGLSKMVLHAEQIELIDSVDKLAAALEHHHH 2ccz B 2.7 BS01 dna C 0 W47 K82 H113 H114 W51 K86 H117 H118 ? 0003677,0003697,0005515,0006260,0006268,0006269,0006270,0006276,0009314,0030894,0031297,0042802,1990077,1990099,1990158 remove_due_to_license_issue P07013 16899446 1 ~ 15 PNSLMTNRLVLSGTVCRAPLRKVSPSGIPHCQFVLEHRSVQEEAGFHRQAWCQMPVIVSGHENQAITHSITVGSRITVQGFISCHKAKNGLSKMVLHAEQIELIDSVDKLAAALEHHH 2cej A 2.5 BS01 1AH B 1 R8 L23 D25 G27 D29 G48 V82 I84 R8 L23 D25 G27 D29 G48 V82 I84 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q8Q3H0 16509598 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2cej B 2.5 BS01 1AH B 1 R108 G127 A128 D129 D130 V132 I147 G148 G149 I150 V182 R8 G27 A28 D29 D30 V32 I47 G48 G49 I50 V82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=2.4nM remove_due_to_license_issue Q8Q3H0 16509598 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2cem A 1.8 BS01 2AH B 1 L23 D25 G27 D29 G48 G49 I50 V82 I84 L23 D25 G27 D29 G48 G49 I50 V82 I84 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q8Q3H0 16509598 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2cem B 1.8 BS01 2AH B 1 D125 G127 A128 D129 D130 V132 G148 G149 I150 P181 V182 D25 G27 A28 D29 D30 V32 G48 G49 I50 P81 V82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=12nM remove_due_to_license_issue Q8Q3H0 16509598 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2cen A 1.7 BS01 4AH B 1 L23 D25 G27 A28 D29 G48 G49 I50 V82 I84 L23 D25 G27 A28 D29 G48 G49 I50 V82 I84 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q5RZ09 16509598 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2cen B 1.7 BS01 4AH B 1 D125 G127 A128 D129 D130 V132 G148 G149 I150 P181 V182 D25 G27 A28 D29 D30 V32 G48 G49 I50 P81 V82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=5nM remove_due_to_license_issue Q5RZ09 16509598 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2ceo A 2.8 BS01 T44 A 1 S23 L246 L269 N273 R378 R381 S4 L227 L250 N254 R351 R354 ? 0004867,0005576,0005615,0070062,0070327 remove_due_to_license_issue P05543 16938877 1395 YKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMEQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAAVPENTFLHPIIQIDRSFMLLILERSTRSILFLGKVVNPTE 2ceq A 2.14 BS01 GIM A 1 Q18 H150 W151 E206 Y322 E387 W425 E432 W433 F441 Q18 H150 W151 E206 Y322 E387 W425 E432 W433 F441 R79 H150 E206 V209 N320 Y322 E387 R79 H150 E206 V209 N320 Y322 E387 3.2.1.23 0004553,0004565,0005975,0008422,0016798 Ki=53nM remove_due_to_license_issue P22498 17002288 1492 MYSFPNSFRFGWSQAGFQSEMGTPGSEDPNTDWYKWVHDPENMAAGLVSGDLPENGPGYWGNYKTFHDNAQKMGLKIARLNVEWSRIFPNPLPRPQNFDESKQDVTEVEINENELKRLDEYANKDALNHYREIFKDLKSRGLYFILNMYHWPLPLWLHDPIRVRRGDFTGPSGWLSTRTVYEFARFSAYIAWKFDDLVDEYSTMNEPNVVGGLGYVGVKSGFPPGYLSFELSRRAMYNIIQAHARAYDGIKSVSKKPVGIIYANSSFQPLTDKDMEAVEMAENDNRWWFFDAIIRGEITRGNEKIVRDDLKGRLDWIGVNYYTRTVVKRTEKGYVSLGGYGHGCERNSVSLAGLPTSDFGWEFFPEGLYDVLTKYWNRYHLYMYVTENGIADDADYQRPYYLVSHVYQVHRAINSGADVRGYLHWSLADNYEWASGFSMRFGLLKVDYNTKRLYWRPSALVYREIATNGAITDEIEHLNSVPPVKPLRH 2cer A 2.29 BS01 PGI A 1 Q18 H150 W151 E206 Y322 E387 W425 E432 F441 Q18 H150 W151 E206 Y322 E387 W425 E432 F441 R79 H150 E206 V209 N320 Y322 E387 R79 H150 E206 V209 N320 Y322 E387 3.2.1.23 0004553,0004565,0005975,0008422,0016798 Ki<0.6nM remove_due_to_license_issue P22498 17002288 1490 MYSFPNSFRFGWSQAGFQSEMGTPGSEDPNTDWYKWVHDPENMAAGLVSGDLPENGPGYWGNYKTFHDNAQKMGLKIARLNVEWSRIFPNPLPRPQNFDESKQDVTEVEINENELKRLDEYANKDALNHYREIFKDLKSRGLYFILNMYHWPLPLWLHDPIRVRRGDFTGPSGWLSTRTVYEFARFSAYIAWKFDDLVDEYSTMNEPNVVGGLGYVGVKSGFPPGYLSFELSRRAMYNIIQAHARAYDGIKSVSKKPVGIIYANSSFQPLTDKDMEAVEMAENDNRWWFFDAIIRGEITRGNEKIVRDDLKGRLDWIGVNYYTRTVVKRTEKGYVSLGGYGHGCERNSVSLAGLPTSDFGWEFFPEGLYDVLTKYWNRYHLYMYVTENGIADDADYQRPYYLVSHVYQVHRAINSGADVRGYLHWSLADNYEWASGFSMRFGLLKVDYNTKRLYWRPSALVYREIATNGAITDEIEHLNSVPPVKPLRH 2ces A 2.15 BS01 GIM A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y293 E346 W393 E400 W401 F409 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E346 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=56nM remove_due_to_license_issue Q08638 17002288 1447 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2cet A 1.97 BS01 PGI A 1 Q20 H121 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 E164 Y288 E341 W388 E395 W396 F404 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N286 Y288 E341 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=9.6nM remove_due_to_license_issue Q08638 17002288 1447 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASERAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2cex B 2.2 BS01 DAN B 1 N10 E67 R147 F170 N187 N9 E66 R146 F169 N186 ? 0030288,0042597,0055085 Kd=20uM remove_due_to_license_issue P44542 16702222 1307 DYDLKFGMNAGTSSNEYKAAEMFAKEVKEKSQGKIEISLYPSSQLGDDRAMLKQLKDGSLDFTFAESARFQLFYPEAAVFALPYVISNYNVAQKALFDTEFGKDLIKKMDKDLGVTLLSQAYNGTRQTTSNRAINSIADMKGLKLRVPNAATNLAYAKYVGASPTPMAFSEVYLALQTNAVDGQENPLAAVQAQKFYEVQKFLAMTNHILNDQLYLVSNETYKELPEDLQKVVKDAAENAAKYHTKLFVDGEKDLVTFFEKQGVKITHPDLVPFKESMKPYYAEFVKQTGQKGESALKQIEAINP 2cf8 H 1.3 BS03 ESH H 1 H57 Y60A W60D L99 D189 A190 S214 W215 G216 G219 H43 Y47 W50 L96 D192 A193 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.008uM remove_due_to_license_issue P00734 16763681 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2cf9 H 1.79 BS03 348 H 1 H57 Y60A N98 D189 A190 S214 W215 G216 G219 H43 Y47 N95 D192 A193 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.015uM remove_due_to_license_issue P00734 16763681 1247 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2cfd A 1.6 BS02 R4A A 1 E102 F105 P136 L137 Y296 Y302 Q306 Y307 R336 G380 A382 E94 F97 P128 L129 Y288 Y294 Q298 Y299 R328 G372 A374 Y284 D298 Y382 H431 H433 H592 Y276 D290 Y374 H423 H425 H584 1.4.3.21 0005507,0008131,0009308,0016491,0016641,0046872,0048038,0052595 Ki=32nM remove_due_to_license_issue P46881 18507382 705 ASPFRLASAGEISEVQGILRTAGLLGPEKRIAYLGVLDPARGAGSEAEDRRFRVFIHDVSGARPQEVTVSVTNGTVISAVELDTAATGELPVLEEEFEVVEQLLATDERWLKALAARNLDVSKVRVAPLSAGVFEYAEERGRRILRGLAFVQDFPEDSAWAHPVDGLVAYVDVVSKEVTRVIDTGVFPVPAEHGNYTDPELTGPLRTTQKPISITQPEGPSFTVTGGNHIEWEKWSLDVGFDVREGVVLHNIAFRDGDRLRPIINRASIAEMVVPYGDPSPIRSWQNYFDTGEYLVGQYANSLELGCDCLGDITYLSPVISDAFGNPREIRNGICMHEEDWGILAKHSDLWSGINYTRRNRRMVISFFTTIGNYDYGFYWYLYLDGTIEFEAKATGVVFTSAFPEGGSDNISQLAPGLGAPFHQHIFSARLDMAIDGFTNRVEEEDVVRQTMGPGNERGNAFSRKRTVLTRESEAVREADARTGRTWIISNPESKNRLNEPVGYKLHAHNQPTLLADPGSSIARRAAFATKDLWVTRYADDERYPTGDFVNQHSGGAGLPSYIAQDRDIDGQDIVVWHTFGLTHFPRVEDWPIMPVDTVGFKLRPEGFFDRSPVLDVPA 2cfd B 1.6 BS02 R4A B 1 E102 F105 P136 L137 W168 Y296 Y302 Q306 Y307 R336 T378 G380 A382 E94 F97 P128 L129 W160 Y288 Y294 Q298 Y299 R328 T370 G372 A374 Y284 D298 Y382 H431 H433 H592 Y276 D290 Y374 H423 H425 H584 1.4.3.21 0005507,0008131,0009308,0016491,0016641,0046872,0048038,0052595 Ki=32nM remove_due_to_license_issue P46881 18507382 705 ASPFRLASAGEISEVQGILRTAGLLGPEKRIAYLGVLDPARGAGSEAEDRRFRVFIHDVSGARPQEVTVSVTNGTVISAVELDTAATGELPVLEEEFEVVEQLLATDERWLKALAARNLDVSKVRVAPLSAGVFEYAEERGRRILRGLAFVQDFPEDSAWAHPVDGLVAYVDVVSKEVTRVIDTGVFPVPAEHGNYTDPELTGPLRTTQKPISITQPEGPSFTVTGGNHIEWEKWSLDVGFDVREGVVLHNIAFRDGDRLRPIINRASIAEMVVPYGDPSPIRSWQNYFDTGEYLVGQYANSLELGCDCLGDITYLSPVISDAFGNPREIRNGICMHEEDWGILAKHSDLWSGINYTRRNRRMVISFFTTIGNYDYGFYWYLYLDGTIEFEAKATGVVFTSAFPEGGSDNISQLAPGLGAPFHQHIFSARLDMAIDGFTNRVEEEDVVRQTMGPGNERGNAFSRKRTVLTRESEAVREADARTGRTWIISNPESKNRLNEPVGYKLHAHNQPTLLADPGSSIARRAAFATKDLWVTRYADDERYPTGDFVNQHSGGAGLPSYIAQDRDIDGQDIVVWHTFGLTHFPRVEDWPIMPVDTVGFKLRPEGFFDRSPVLDVPA 2cfg A 1.55 BS02 R4A A 1 E102 F105 P136 L137 W168 Y296 Y302 Y307 I379 G380 A382 F407 E94 F97 P128 L129 W160 Y288 Y294 Y299 I371 G372 A374 F399 Y284 D298 Y382 H431 H433 H592 Y276 D290 Y374 H423 H425 H584 1.4.3.21 0005507,0008131,0009308,0016491,0016641,0046872,0048038,0052595 remove_due_to_license_issue P46881 18507382 1630 ASPFRLASAGEISEVQGILRTAGLLGPEKRIAYLGVLDPARGAGSEAEDRRFRVFIHDVSGARPQEVTVSVTNGTVISAVELDTAATGELPVLEEEFEVVEQLLATDERWLKALAARNLDVSKVRVAPLSAGVFEYAEERGRRILRGLAFVQDFPEDSAWAHPVDGLVAYVDVVSKEVTRVIDTGVFPVPAEHGNYTDPELTGPLRTTQKPISITQPEGPSFTVTGGNHIEWEKWSLDVGFDVREGVVLHNIAFRDGDRLRPIINRASIAEMVVPYGDPSPIRSWQNYFDTGEYLVGQYANSLELGCDCLGDITYLSPVISDAFGNPREIRNGICMHEEDWGILAKHSDLWSGINYTRRNRRMVISFFTTIGNYDYGFYWYLYLDGTIEFEAKATGVVFTSAFPEGGSDNISQLAPGLGAPFHQHIFSARLDMAIDGFTNRVEEEDVVRQTMGPGNERGNAFSRKRTVLTRESEAVREADARTGRTWIISNPESKNRLNEPVGYKLHAHNQPTLLADPGSSIARRAAFATKDLWVTRYADDERYPTGDFVNQHSGGAGLPSYIAQDRDIDGQDIVVWHTFGLTHFPRVEDWPIMPVDTVGFKLRPEGFFDRSPVLDVPA 2cfg A 1.55 BS03 R4A B 1 S356 D357 L358 S348 D349 L350 Y284 D298 Y382 H431 H433 H592 Y276 D290 Y374 H423 H425 H584 1.4.3.21 0005507,0008131,0009308,0016491,0016641,0046872,0048038,0052595 remove_due_to_license_issue P46881 18507382 1632 ASPFRLASAGEISEVQGILRTAGLLGPEKRIAYLGVLDPARGAGSEAEDRRFRVFIHDVSGARPQEVTVSVTNGTVISAVELDTAATGELPVLEEEFEVVEQLLATDERWLKALAARNLDVSKVRVAPLSAGVFEYAEERGRRILRGLAFVQDFPEDSAWAHPVDGLVAYVDVVSKEVTRVIDTGVFPVPAEHGNYTDPELTGPLRTTQKPISITQPEGPSFTVTGGNHIEWEKWSLDVGFDVREGVVLHNIAFRDGDRLRPIINRASIAEMVVPYGDPSPIRSWQNYFDTGEYLVGQYANSLELGCDCLGDITYLSPVISDAFGNPREIRNGICMHEEDWGILAKHSDLWSGINYTRRNRRMVISFFTTIGNYDYGFYWYLYLDGTIEFEAKATGVVFTSAFPEGGSDNISQLAPGLGAPFHQHIFSARLDMAIDGFTNRVEEEDVVRQTMGPGNERGNAFSRKRTVLTRESEAVREADARTGRTWIISNPESKNRLNEPVGYKLHAHNQPTLLADPGSSIARRAAFATKDLWVTRYADDERYPTGDFVNQHSGGAGLPSYIAQDRDIDGQDIVVWHTFGLTHFPRVEDWPIMPVDTVGFKLRPEGFFDRSPVLDVPA 2cfg B 1.55 BS01 R4A A 1 S356 D357 L358 S348 D349 L350 Y284 D298 Y382 H431 H433 H592 Y276 D290 Y374 H423 H425 H584 1.4.3.21 0005507,0008131,0009308,0016491,0016641,0046872,0048038,0052595 remove_due_to_license_issue P46881 18507382 1630 ASPFRLASAGEISEVQGILRTAGLLGPEKRIAYLGVLDPARGAGSEAEDRRFRVFIHDVSGARPQEVTVSVTNGTVISAVELDTAATGELPVLEEEFEVVEQLLATDERWLKALAARNLDVSKVRVAPLSAGVFEYAEERGRRILRGLAFVQDFPEDSAWAHPVDGLVAYVDVVSKEVTRVIDTGVFPVPAEHGNYTDPELTGPLRTTQKPISITQPEGPSFTVTGGNHIEWEKWSLDVGFDVREGVVLHNIAFRDGDRLRPIINRASIAEMVVPYGDPSPIRSWQNYFDTGEYLVGQYANSLELGCDCLGDITYLSPVISDAFGNPREIRNGICMHEEDWGILAKHSDLWSGINYTRRNRRMVISFFTTIGNYDYGFYWYLYLDGTIEFEAKATGVVFTSAFPEGGSDNISQLAPGLGAPFHQHIFSARLDMAIDGFTNRVEEEDVVRQTMGPGNERGNAFSRKRTVLTRESEAVREADARTGRTWIISNPESKNRLNEPVGYKLHAHNQPTLLADPGSSIARRAAFATKDLWVTRYADDERYPTGDFVNQHSGGAGLPSYIAQDRDIDGQDIVVWHTFGLTHFPRVEDWPIMPVDTVGFKLRPEGFFDRSPVLDVPA 2cfg B 1.55 BS03 R4A B 1 E102 F105 P136 L137 W168 Y296 Y302 Y307 G380 N381 A382 F407 E94 F97 P128 L129 W160 Y288 Y294 Y299 G372 N373 A374 F399 Y284 D298 Y382 H431 H433 H592 Y276 D290 Y374 H423 H425 H584 1.4.3.21 0005507,0008131,0009308,0016491,0016641,0046872,0048038,0052595 remove_due_to_license_issue P46881 18507382 1632 ASPFRLASAGEISEVQGILRTAGLLGPEKRIAYLGVLDPARGAGSEAEDRRFRVFIHDVSGARPQEVTVSVTNGTVISAVELDTAATGELPVLEEEFEVVEQLLATDERWLKALAARNLDVSKVRVAPLSAGVFEYAEERGRRILRGLAFVQDFPEDSAWAHPVDGLVAYVDVVSKEVTRVIDTGVFPVPAEHGNYTDPELTGPLRTTQKPISITQPEGPSFTVTGGNHIEWEKWSLDVGFDVREGVVLHNIAFRDGDRLRPIINRASIAEMVVPYGDPSPIRSWQNYFDTGEYLVGQYANSLELGCDCLGDITYLSPVISDAFGNPREIRNGICMHEEDWGILAKHSDLWSGINYTRRNRRMVISFFTTIGNYDYGFYWYLYLDGTIEFEAKATGVVFTSAFPEGGSDNISQLAPGLGAPFHQHIFSARLDMAIDGFTNRVEEEDVVRQTMGPGNERGNAFSRKRTVLTRESEAVREADARTGRTWIISNPESKNRLNEPVGYKLHAHNQPTLLADPGSSIARRAAFATKDLWVTRYADDERYPTGDFVNQHSGGAGLPSYIAQDRDIDGQDIVVWHTFGLTHFPRVEDWPIMPVDTVGFKLRPEGFFDRSPVLDVPA 2cgf A 2.2 BS01 P2N A 1 N37 A41 D79 M84 F124 T171 L173 N36 A40 D78 M83 F123 T170 L172 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.39uM remove_due_to_license_issue IC50=1.2e+2nM P02829 17114002 1214 ASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKKHSEFVAYPIQLVVTKEV 2cgr H 2.2 BS01 GAS H 1 W33 E35 E50 R57 N59 Y100 S101 S102 W33 E35 E50 R57 N59 Y100 S101 S102 Kd=53nM remove_due_to_license_issue 7893280 215 RVQLLESGAELMKPGASVQISCKATGYTFSEYWIEWVKERPGHGLEWIGEILPGSGRTNYREKFKGKATFTADTSSNTAYMQLSSLTSEDSAVYYCTRGYSSMDYWGQGTSVTVSAAKTTPPSVYPLAPGCGDTTGSSVTLGCLVKGYFPESVTVTWNSGSLSSSVHTFPALLQSGLYTMSSSVTVPSSTWPSQTVTCSVAHPASSTTVDKKLE 2cgr L 2.2 BS01 GAS H 1 Y37 G96 Y101 Y37 G96 Y101 ? remove_due_to_license_issue A2P1G9 7893280 215 ELVMTQSPLSLPVSLGDQASISCRPSQSLVHSNGNTYLHWYLQKPGQSPKLLIYRVSNRFSGVPDRFSGSGSGTAFTLKISRVEAEDLGVYFCSQGTHVPYTFGGGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 2cgu A 2.5 BS01 3A3 A 1 L15 V23 K38 Y86 C87 L137 D148 L10 V18 K33 Y78 C79 L129 D140 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=13.4uM remove_due_to_license_issue O14757 16574416 1272 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 2cgv A 2.6 BS01 3B3 A 1 L15 V23 C87 E91 E134 N135 L137 S147 L10 V18 C79 E83 E126 N127 L129 S139 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=27300nM O14757 16574416 1273 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKG 2cgw A 2.2 BS01 3C3 A 1 V23 A36 K38 E85 Y86 C87 L137 D148 V18 A31 K33 E76 Y77 C78 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=17.3uM remove_due_to_license_issue O14757 16574416 1272 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 2cgx A 2.2 BS01 3D3 A 1 G16 Y20 V23 A36 E85 Y86 C87 L137 G11 Y15 V18 A31 E77 Y78 C79 L129 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=15.6uM remove_due_to_license_issue IC50=15600nM O14757 16574416 1274 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 2chm A 1.6 BS02 3P4 A 1 L725 L765 A767 I768 A779 V782 A783 L804 Q817 F820 L190 L230 A232 I233 A244 V247 A248 L269 Q282 F285 3.1.4.35,3.1.4.53 0004114,0007165,0008081 ic50=5.5nM remove_due_to_license_issue O76074,Q07343 16759100 1861 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHPGVSNQFLINTNSELALMYNDESVLEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHEKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 2chw A 2.6 BS01 039 A 1 V803 M804 P810 L811 W812 I831 E880 I881 T887 M953 I963 V564 M565 P571 L572 W573 I592 E641 I642 T648 M714 I724 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 16647110 2093 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 2chx A 2.5 BS01 090 A 1 W812 I831 K833 Y867 I879 E880 V882 M953 I963 D964 L1092 W575 I594 K596 Y630 I642 E643 V645 M716 I726 D727 L842 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 16647110 2093 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEWCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 2chz A 2.6 BS01 093 A 1 W812 I831 Y867 I879 V882 M953 I963 D964 L1092 W573 I592 Y628 I640 V643 M713 I723 D724 L839 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=16nM, Ki=7.0nM P48736 16647110 2093 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 2cji A 2.1 BS02 GSK A 1 E97 T98 A190 Q192 W215 G216 G219 C220 G226 I227 Y228 E83 T84 A180 Q182 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=6nM remove_due_to_license_issue Ki=6nM P00742 16697194 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2ckm A 2.15 BS01 AA7 A 1 Y70 W84 G118 Y121 E199 E278 W279 F330 W432 H440 Y67 W81 G115 Y118 E196 E275 W276 F327 W429 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Kd=77fM remove_due_to_license_issue P04058 16942022 1536 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 2cle A 1.5 BS01 F6F A 1 E49 A59 D60 L100 I153 Y175 F212 G234 S235 E48 A58 D59 L99 I152 Y174 F196 G218 S219 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 Kd=280uM remove_due_to_license_issue P00929 17559195 1268 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 2clf A 1.7 BS01 F6F A 1 E49 A59 L100 A129 I153 Y175 F212 G213 G234 S235 E49 A59 L100 A129 I153 Y175 F197 G198 G219 S220 E49 D60 Y175 E49 D60 Y175 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 Kd=280uM remove_due_to_license_issue P00929 17559195 1269 MERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASRA 2clf B 1.7 BS01 F6F A 1 P18 G395 P17 G394 K87 E109 S377 K86 E108 S376 4.2.1.20 0000162,0004834,0005515,0005737,0006568,0016829,0042802 Kd=280uM remove_due_to_license_issue P0A2K1 17559195 1269 TTLLNPYFGEFGGMYVPQILMPALNQLEEAFVRAQKDPEFQAQFADLLKNYAGRPTALTKCQNITAGTRTTLYLKREDLLHGGAHKTNQVLGQALLAKRMGKSEIIAETGAGQHGVASALASALLGLKCRIYMGAKDVERQSPNVFRMRLMGAEVIPVHSGSATLKDACNEALRDWSGSYETAHYMLGTAAGPHPYPTIVREFQRMIGEETKAQILDKEGRLPDAVIACVGGGSNAIGMFADFINDTSVGLIGVEPGGHGIETGEHGAPLKHGRVGIYFGMKAPMMQTADGQIEESYSISAGLDFPSVGPQHAYLNSIGRADYVSITDDEALEAFKTLCRHEGIIPALESSHALAHALKMMREQPEKEQLLVVNLSGRGDKDIFTVHDILKARG 2clf B 1.7 BS02 F6F B 1 E109 T110 G111 H115 L166 C170 L188 G189 T190 F280 E108 T109 G110 H114 L165 C169 L187 G188 T189 F279 K87 E109 S377 K86 E108 S376 4.2.1.20 0000162,0004834,0005515,0005737,0006568,0016829,0042802 Kd=280uM remove_due_to_license_issue P0A2K1 17559195 1396 TTLLNPYFGEFGGMYVPQILMPALNQLEEAFVRAQKDPEFQAQFADLLKNYAGRPTALTKCQNITAGTRTTLYLKREDLLHGGAHKTNQVLGQALLAKRMGKSEIIAETGAGQHGVASALASALLGLKCRIYMGAKDVERQSPNVFRMRLMGAEVIPVHSGSATLKDACNEALRDWSGSYETAHYMLGTAAGPHPYPTIVREFQRMIGEETKAQILDKEGRLPDAVIACVGGGSNAIGMFADFINDTSVGLIGVEPGGHGIETGEHGAPLKHGRVGIYFGMKAPMMQTADGQIEESYSISAGLDFPSVGPQHAYLNSIGRADYVSITDDEALEAFKTLCRHEGIIPALESSHALAHALKMMREQPEKEQLLVVNLSGRGDKDIFTVHDILKARG 2clh A 1.7 BS01 F19 A 1 F22 L100 L127 I153 Y175 T183 G184 F212 G213 G234 S235 F22 L100 L127 I153 Y175 T183 G184 F203 G204 G225 S226 E49 D60 Y175 E49 D60 Y175 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 Kd=87.6uM remove_due_to_license_issue P00929 17559195 1268 MERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 2cli A 1.7 BS01 F9F A 1 F22 L100 L127 A129 I153 Y175 T183 G184 F212 G234 S235 F22 L100 L127 A129 I153 Y175 T183 G184 F202 G224 S225 E49 D60 Y175 E49 D60 Y175 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 Kd=50uM remove_due_to_license_issue P00929 17559195 1269 MERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASRA 2clk A 1.5 BS01 G3H A 1 F22 I64 L100 Y175 T183 G184 F212 G213 G234 S235 F22 I64 L100 Y175 T183 G184 F212 G213 G234 S235 E49 D60 Y175 E49 D60 Y175 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 Kd=164uM remove_due_to_license_issue P00929 17559195 1268 MERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLAIIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGAENRGALPLHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 2cll A 1.6 BS01 F9F A 1 F22 L100 L127 A129 I153 Y175 T183 G184 F212 G234 S235 F21 L99 L126 A128 I152 Y174 T182 G183 F202 G224 S225 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 remove_due_to_license_issue P00929 17559232 1268 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 2clm A 1.51 BS01 F6F A 1 E49 A59 I64 L100 A129 I153 Y175 F212 G213 S235 E48 A58 I63 L99 A128 I152 Y174 F196 G197 S219 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 remove_due_to_license_issue P00929 17559232 1268 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 2clm B 1.51 BS01 F6F A 1 P18 L391 K392 A393 P17 L390 K391 A392 K87 E109 S377 K86 E108 S376 4.2.1.20 0000162,0004834,0005515,0005737,0006568,0016829,0042802 remove_due_to_license_issue P0A2K1 17559232 1268 TTLLNPYFGEFGGMYVPQILMPALNQLEEAFVRAQKDPEFQAQFADLLKNYAGRPTALTKCQNITAGTRTTLYLKREDLLHGGAHKTNQVLGQALLAKRMGKSEIIAETGAGQHGVASALASALLGLKCRIYMGAKDVERQSPNVFRMRLMGAEVIPVHSGSATLKDACNEALRDWSGSYETAHYMLGTAAGPHPYPTIVREFQRMIGEETKAQILDKEGRLPDAVIACVGGGSNAIGMFADFINDTSVGLIGVEPGGHGIETGEHGAPLKHGRVGIYFGMKAPMMQTADGQIEESYSISAGLDFPSVGPQHAYLNSIGRADYVSITDDEALEAFKTLCRHEGIIPALESSHALAHALKMMREQPEKEQLLVVNLSGRGDKDIFTVHDILKA 2clo A 1.5 BS01 F19 A 1 F22 L100 I153 Y175 T183 G184 F212 S235 F21 L99 I152 Y174 T182 G183 F202 S225 E49 D60 Y175 E48 D59 Y174 4.2.1.20 0000162,0004834,0005515,0005829,0006568,0016829 remove_due_to_license_issue P00929 17559232 1268 ERYENLFAQLNDRREGAFVPFVTLGDPGIEQSLKIIDTLIDAGADALELGVPFSDPLADGPTIQNANLRAFAAGVTPAQCFEMLALIREKHPTIPIGLLMYANLVFNNGIDAFYARCEQVGVDSVLVADVPVEESAPFRQAALRHNIAPIFICPPNADDDLLRQVASYGRGYTYLLSRSGVTGHHLIEKLKEYHAAPALQGFGISSPEQVSAAVRAGAAGAISGSAIVKIIEKNLASPKQMLAELRSFVSAMKAASR 2clx A 1.8 BS01 F18 A 1 A31 F80 E81 F82 L83 L134 D145 A31 F75 E76 F77 L78 L129 D140 D127 K129 Q131 N132 D145 T158 T165 D122 K124 Q126 N127 D140 T153 T160 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=69000nM P24941 17064068 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2cm7 A 2.1 BS01 IZD A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 D298 Y44 R45 D46 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=210nM remove_due_to_license_issue IC50=190nM, Ki=180nM P18031 16916797 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2cm8 A 2.1 BS01 F16 A 1 Y46 D181 F182 C215 S216 A217 I219 G220 R221 Q262 D298 Y45 D180 F181 C214 S215 A216 I218 G219 R220 Q261 D297 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=1350nM remove_due_to_license_issue P18031 16916797 1299 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2cma A 2.3 BS01 F20 A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 D298 Y44 R45 D46 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=185nM remove_due_to_license_issue P18031 16916797 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2cmb A 1.7 BS01 F17 A 1 K41 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 F280 K47 Y52 R53 D54 D187 F188 C221 S222 A223 I225 G226 R227 F286 D181 C215 R221 S222 Q262 D187 C221 R227 S228 Q268 3.1.3.48 0004725,0006470,0016311 ic50=65nM remove_due_to_license_issue P18031 16916797 1282 MHHHHHHEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKF 2cmc A 2.2 BS01 DFM A 1 Y46 R47 D48 V49 F182 C215 S216 A217 I219 G220 R221 Q262 K279 F280 Y51 R52 D53 V54 F187 C220 S221 A222 I224 G225 R226 Q267 K284 F285 D181 C215 R221 S222 Q262 D186 C220 R226 S227 Q267 3.1.3.48 0004725,0006470,0016311 ic50=1750nM remove_due_to_license_issue IC50=1750nM P18031 16916797 1281 HHHHHHEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKF 2cmf A 2.5 BS01 F11 A 1 Y70 W84 G118 Y121 E199 F330 F331 Y334 W432 H440 Y67 W81 G115 Y118 E196 F327 F328 Y331 W429 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 16942022 1536 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 2cmo A 2.65 BS01 M1L A 1 E13 Y16 Y61 G62 P89 T91 R96 L138 G141 T173 T174 E193 M196 Y220 E9 Y12 Y57 G58 P85 T87 R92 L134 G137 T169 T170 E189 M192 Y216 ? 0015276,0016020 remove_due_to_license_issue P19491 16483599 1112 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 2cn0 H 1.3 BS03 F25 H 1 H57 Y60A L99 D189 A190 S214 W215 G216 G219 H43 Y47 L96 D192 A193 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=22nM remove_due_to_license_issue P00734 17001711 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2cn8 A 2.7 BS02 DBQ A 1 L226 V234 A247 L301 L303 M304 E308 L354 T367 L15 V19 A32 L71 L73 M74 E78 L124 T137 D347 K349 N352 D368 D117 K119 N122 D138 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=183nM O96017 16794575 1506 YPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEEN 2cne A 1.8 BS01 DFJ A 1 K41 Y46 R47 D48 F182 C215 S216 A217 I219 G220 R221 F280 K47 Y52 R53 D54 F188 C221 S222 A223 I225 G226 R227 F286 D181 C215 R221 S222 Q262 D187 C221 R227 S228 Q268 3.1.3.48 0004725,0006470,0016311 ic50=1.7nM remove_due_to_license_issue Ki=1.7nM P18031 17028182 1281 MHHHHHHEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKF 2cnf A 2.2 BS01 F32 A 1 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 D298 Y44 D46 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=240nM remove_due_to_license_issue IC50=270nM P18031 17028182 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2cng A 1.9 BS01 IZE A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 D298 Y44 R45 D46 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=110nM remove_due_to_license_issue P18031 17028182 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2cnh A 1.8 BS01 IZB A 1 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y44 D46 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=59nM remove_due_to_license_issue P18031 17028182 1300 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2cni A 2.0 BS01 IZF A 1 Y20 R24 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 L299 Y20 R24 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 L299 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=21nM remove_due_to_license_issue P18031 17028182 1301 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 2csm A 2.8 BS01 TYR A 1 I74 R75 R76 I74 R75 R76 R16 R157 K168 N194 E198 T242 E246 R16 R157 K168 N194 E198 T233 E237 5.4.99.5 0004106,0005515,0005634,0005737,0006571,0009073,0009094,0016853,0046417,0072545,0120284 remove_due_to_license_issue P32178 8622937 300 MDFTKPETVLNLQNIRDELVRMEDSIIFKFIERSHFATCPSVYEANHPGLEIPNFKGSFLDWALSNLEIAHSRIRRFESPDETPFFPDKIQKSFLPSINYPQILAPYAPEVNYNDKIKKVYIEKIIPLISKRDGDDKNNFGSVATRDIECLQSLSRRIHFGKFVAEAKFQSDIPLYTKLIKSKDVEGIMKNITNSAVEEKILERLTKKAEVYGVRITPEYLVKIYKEIVIPITKEVEVEYLLRRL 2csn A 2.5 BS01 CKI A 1 I18 I26 L88 L138 I13 I21 L83 L133 2.7.11.1 0004672,0005524,0006468 Ki=39uM remove_due_to_license_issue P40233 8692811 300 NVVGVHYKVGRRIGEGSFGVIFEGTNLLNNQQVAIKFEPRRSDAPQLRDEYRTYKLLAGCTGIPNVYYFGQEGLHNVLVIDLLGPSLEDLLDLCGRKFSVKTVAMAAKQMLARVQSIHEKSLVYRDIKPDNFLIGRPNSKNANMIYVVDFGMVKFYRDPVTKQHIPYREKKNLSGTARYMSINTHLGREQSRRDDLEALGHVFMYFLRGSLPWQGLKAATNKQKYERIGEKKQSTPLRELCAGFPEEFYKYMHYARNLAFDATPDYDYLQGLFSKVLERLNTTEDENFDWNLL 2ctc A 1.4 BS02 HFA A 1 H69 N144 R145 I243 Y248 A250 E270 H69 N144 R145 I243 Y248 A250 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=0.13mM remove_due_to_license_issue P00730 15299490 309 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVEALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTLNN 2cvd A 1.45 BS02 HQL A 1 M11 G13 R14 M99 F102 W104 Y152 T159 M10 G12 R13 M98 F101 W103 Y151 T158 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.8uM remove_due_to_license_issue IC50=3800nM O60760 16547010 2201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2d06 A 2.3 BS02 EST A 1 P47 K106 H108 F142 V148 F247 P40 K99 H101 F135 V141 F240 K48 H108 S138 K41 H101 S131 2.8.2.1 0004062,0005515,0005737,0005829,0006068,0006584,0006805,0008146,0008202,0008210,0009308,0009812,0016740,0047894,0050294,0050427,0050656,0051923 Ki=83.2uM remove_due_to_license_issue Kd=1200nM P50225 16221673 304 SRPPLEYVKGVPLIKYFAEALGPLQSFQARPDDLLISTYPKSGTTWVSQILDMIYQGGDLEKCHRAPIFMRVPFLEFKAPGIPSGMETLKDTPAPRLLKTHLPLALLPQTLLDQKVKVVYVARNAKDVAVSYYHFYHMAKVHPEPGTWDSFLEKFMVGEVSYGSWYQHVQEWWELSRTHPVLYLFYEDMKENPKREIQKILEFVGHSLPEETVDFMVQHTSFKEMKKNPMTNYTTVPQEFMDHSISPFMRKGMAGDWKTTFTVAQNERFDADYAEKMAGCSLSFRSEL 2d1n A 2.37 BS06 FA4 A 1 Y176 L184 L185 A186 H222 E223 H226 H232 P236 A238 L239 F241 P242 I243 Y244 T245 F252 Y73 L81 L82 A83 H119 E120 H123 H129 P133 A135 L136 F138 P139 I140 Y141 T142 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.007uM remove_due_to_license_issue P45452 16603129 1001 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 2d1o A 2.02 BS06 FA4 A 1 V163 L164 A165 H201 E202 H205 H211 T215 A217 L218 Y220 P221 L222 Y223 F232 V81 L82 A83 H119 E120 H123 H129 T133 A135 L136 Y138 P139 L140 Y141 F150 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=0.02uM remove_due_to_license_issue P08254 16603129 1001 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPPDSP 2d3u A 2.0 BS01 CCT A 1 L419 R422 M423 H475 S476 Y477 I482 W528 L414 R417 M418 H470 S471 Y472 I477 W523 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Ki=0.12uM remove_due_to_license_issue Q99AU2 16828488 1001 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 2d3z A 1.8 BS01 FIH A 1 L419 R422 M423 H475 S476 Y477 I482 L497 W528 L416 R419 M420 H472 S473 Y474 I479 L494 W525 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Ki=0.23uM remove_due_to_license_issue Q99AU2 16828488 2001 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPERKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 2d41 A 2.1 BS01 SNH A 1 L419 M423 H475 S476 Y477 I482 L497 R501 W528 L414 M418 H470 S471 Y472 I477 L492 R496 W523 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Ki=0.15uM remove_due_to_license_issue Q99AU2 16828488 1001 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 2dbl H 2.9 BS01 S5H L 1 G33 N35 W50 G95 D96 Y97 W100 F100B G33 N35 W50 G99 D100 Y101 W104 F106 ? remove_due_to_license_issue P01868 8413674 212 QIQLVQSGPELKKPGETVKISCKASGYAFTNYGVNWVKEAPGKELKWMGWINIYTGEPTYVDDFKGRFAFSLETSASTAYLEINNLKNEDTATYFCTRGDYVNWYFDVWGAGTTVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPR 2dbl L 2.9 BS01 S5H L 1 H27D S92 H93 V94 H31 S97 H98 V99 remove_due_to_license_issue 8413674 212 DVVMTQIPLSLPVNLGDQASISCRSSQSLIHSNGNTYLHWYLQKPGQSPKLLMYKVSNRFYGVPDRFSGSGSGTDFTLKISRVEAEDLGIYFCSQSSHVPPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 2ddf A 1.7 BS03 INN A 1 G346 T347 Y390 H405 E406 H409 H415 P437 I438 A439 G129 T130 Y169 H184 E185 H188 H194 P216 I217 A218 3.4.24.86 0004222,0006508,0008237 ic50=41nM remove_due_to_license_issue P78536 16459338 3 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 2doo A 2.43 BS03 C4H A 1 W28 H79 H139 K161 Y163 G164 H197 W25 H76 H136 K158 Y160 G161 H194 H77 H79 D81 H139 C158 K161 N167 H197 H74 H76 D78 H136 C155 K158 N164 H194 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Kd=67nM remove_due_to_license_issue P52699 16937423 601 LPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNE 2doo A 2.43 BS04 C4H B 1 E211 Q212 E208 Q209 H77 H79 D81 H139 C158 K161 N167 H197 H74 H76 D78 H136 C155 K158 N164 H194 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Kd=67nM remove_due_to_license_issue P52699 16937423 602 LPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNE 2doo B 2.43 BS01 C4H A 1 E211 Q212 K215 E208 Q209 K212 H77 H79 D81 H139 C158 K161 N167 H197 H74 H76 D78 H136 C155 K158 N164 H194 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Kd=67nM remove_due_to_license_issue P52699 16937423 601 LPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNE 2doo B 2.43 BS04 C4H B 1 W28 H79 D81 H139 K161 Y163 G164 H197 W25 H76 D78 H136 K158 Y160 G161 H194 H77 H79 D81 H139 C158 K161 N167 H197 H74 H76 D78 H136 C155 K158 N164 H194 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Kd=67nM remove_due_to_license_issue P52699 16937423 602 LPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNE 2dq7 X 2.8 BS01 STU X 1 L17 V25 A37 K39 T82 Y84 M85 G88 A134 L137 D148 L17 V25 A37 K39 T82 Y84 M85 G88 A134 L137 D148 N135 D148 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P06241 16782058 902 KDVWEIPRESLQLIKRLGNGQFGEVWMGTWNGNTKVAIKTLKPGTMSPESFLEEAQIMKKLKHDKLVQLYAVVSEEPIYIVTEYMNKGSLLDFLKDGEGRALKLPNLVDMAAQVAAGMAYIERMNYIHRDLRSANILVGNGLICKIADFGLARLIEDNEYTARQGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELVTKGRVPYPGMNNREVLEQVERGYRMPCPQDCPISLHELMIHCWKKDPEERPTFEYLQSFLEDY 2drc A 1.9 BS01 MTX A 1 I5 A6 D27 F31 I50 R57 I94 I5 A6 D27 F31 I50 R57 I94 I5 M20 F22 D27 L28 F31 L54 I91 T113 I5 M20 F22 D27 L28 F31 L54 I91 T113 1.5.1.3 0004146,0005515,0005542,0005829,0006730,0009257,0009410,0016491,0031427,0046452,0046654,0046655,0046656,0046677,0050661,0051870,0051871,0070401,0070402 Kd=0.13nM remove_due_to_license_issue IC50=8.8nM, EC50=1nM P0ABQ4 1932031 161 MISLIAALAVDRVIGMENAMPFNLPADLAWFKRNTLDKPVIMGRHTWESIGRPLPGRKNIILSSQPGTDDRVTWVKSVDEAIAACGDVPEIMVIGGGRVYEQFLPKAQKLYLTHIDAEVEGDTHFPDYEPDDWESVFSEFHDADAQNSHSYCFEILERR 2drc B 1.9 BS01 MTX B 1 I5 A6 D27 L28 F31 K32 I50 R52 R57 I94 I5 A6 D27 L28 F31 K32 I50 R52 R57 I94 I5 M20 F22 D27 L28 F31 L54 I91 T113 I5 M20 F22 D27 L28 F31 L54 I91 T113 1.5.1.3 0004146,0005515,0005542,0005829,0006730,0009257,0009410,0016491,0031427,0046452,0046654,0046655,0046656,0046677,0050661,0051870,0051871,0070401,0070402 Kd=0.13nM remove_due_to_license_issue IC50=8.8nM, EC50=1nM P0ABQ4 1932031 161 MISLIAALAVDRVIGMENAMPFNLPADLAWFKRNTLDKPVIMGRHTWESIGRPLPGRKNIILSSQPGTDDRVTWVKSVDEAIAACGDVPEIMVIGGGRVYEQFLPKAQKLYLTHIDAEVEGDTHFPDYEPDDWESVFSEFHDADAQNSHSYCFEILERR 2dri A 1.6 BS01 RIP A 1 N13 F15 F16 D89 R90 R141 F164 N190 D215 N13 F15 F16 D89 R90 R141 F164 N190 D215 ? 0005515,0006935,0015752,0016020,0030246,0030288,0042597,0048029,0050918,0055052,0055085 Kd=0.13uM remove_due_to_license_issue P02925 7982928 272 KDTIALVVSTLNNPFFVSLKDGAQKEADKLGYNLVVLDSQNNPAKELANVQDLTVRGTKILLINPTDSDAVGNAVKMANQANIPVITLDRQATKGEVVSHIASDNVLGGKIAGDYIAKKAGEGAKVIELQGIAGTSAARERGEGFQQAVAAHKFNVLASQPADFDRIKGLNVMQNLLTAHPDVQAVFAQNDEMALGALRALQTAGKSDVMVVGFDGTPDGEKAVNDGKLAATIAQLPDQIGAKGVETADKVLKGEKVQAKYPVDLKLVVKQ 2ds1 A 2.0 BS01 1CD A 1 I10 G13 V18 A31 K33 V64 F80 H82 V83 Q131 L134 D145 I10 G13 V18 A31 K33 V56 F72 H74 V75 Q123 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=3.4nM remove_due_to_license_issue IC50=3.4nM P24941 16876403 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEHVHQDLKTFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2duv A 2.2 BS01 371 A 1 I10 G11 V18 A31 K33 F80 F82 L83 Q131 L134 D145 I10 G11 V18 A31 K33 F67 F69 L70 Q118 L121 D132 D127 K129 Q131 N132 D145 T165 D114 K116 Q118 N119 D132 T139 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.087uM remove_due_to_license_issue IC50=87nM P24941 17178224 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2dxs A 2.2 BS01 JTP A 1 V37 L392 A393 A395 A396 L425 H428 F429 L492 G493 V494 P495 W500 R503 V15 L365 A366 A368 A369 L398 H401 F402 L465 G466 V467 P468 W473 R476 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.046uM remove_due_to_license_issue P26663 17125247 1000 SMSYTWTGALITPCVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQ 2e1w A 2.5 BS02 FR6 A 1 H17 D19 L62 F65 M155 G184 D185 D296 H14 D16 L59 F62 M152 G181 D182 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 Ki=11nM remove_due_to_license_issue P56658 15139750 1 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 2e27 H 1.7 BS01 AB0 H 1 W33 Q35 A50 S99 D100 Y1001 W33 Q35 A50 S99 D100 Y101 Ka=2220000000M^-1 remove_due_to_license_issue 18326040 6001 QVQLLESGAELARPGASVKLSCKASGYTFTTYWMQWVRQRPGQGLEWIGAIYPGNGDTRYSQKFKGKATLTADTSSSTASMQLSSLASEDSAVYYCARSDYGGDYWGQGTSVTVSS 2e27 L 1.7 BS01 AB0 H 1 Y49 Y91 F94 T95 W96 Y48 Y90 F93 T94 W95 remove_due_to_license_issue 18326040 6001 IQMTQSPSSLSASLGGKVTITCKANQDIKKKIAWYQHKPGKGPRLLIYYTSTLKSGISSRFSGSGSGRDYSFSISNLEPEDAATYYCLQYDNFTWTFGGGTKLEIKR 2e2b A 2.2 BS01 406 A 1 L248 Y253 A269 K271 E286 V289 M290 L298 I313 T315 F317 M318 I360 H361 V379 A380 D381 F382 L24 Y29 A45 K47 E58 V61 M62 L70 I85 T87 F89 M90 I132 H133 V151 A152 D153 F154 D363 A365 R367 N368 D381 P402 D135 A137 R139 N140 D153 P170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=11nM remove_due_to_license_issue IC50=4.0nM P00519 17376680 1001 MDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSI 2e2p A 2.0 BS01 ADP A 1 G115 T116 A199 A202 K203 D206 G248 R251 G115 T116 A199 A202 K203 D206 G248 R251 2.7.1.1 0000166,0004396,0016740,0046835 Ki=18uM remove_due_to_license_issue Q96Y14 17229727 600 MMIIVGVDAGGTKTKAVAYDCEGNFIGEGSSGPGNYHNVGLTRAIENIKEAVKIAAKGEADVVGMGVAGLDSKFDWENFTPLASLIAPKVIIQHDGVIALFAETLGEPGVVVIAGTGSVVEGYNGKEFLRVGGRGWLLSDDGSAYWVGRKALRKVLKMMDGLENKTILYNKVLKTINVKDLDELVMWSYTSSCQIDLVASIAKAVDEAANEGDTVAMDILKQGAELLASQAVYLARKIGTNKVYLKGGMFRSNIYHKFFTLYLEKEGIISDLGKRSPEIGAVILAYKEVGCDIKKLIS 2e2r A 1.6 BS01 2OH A 1 L268 E275 M306 L309 Y326 N346 I349 F435 V458 L37 E44 M75 L78 Y95 N115 I118 F204 V227 ? Kd=5.5nM remove_due_to_license_issue IC50=13.1nM P62508 17761695 1401 KPYNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAKV 2e5y A 1.92 BS01 ATP A 1 E83 I88 D89 R92 A93 R122 R126 E83 I88 D89 R92 A93 R122 R126 3.6.3.14 0015986,0045261,0046933 Kd=22mM remove_due_to_license_issue P07678 17581881 1001 MKTIHVSVVTPDGPVYEDDVEMVSVKAKSGELGILPGHIPLVAPLEISAARLKKGGKTQYIAVSGGFLEVRPDKVTILAQAAERAEDIDVLRAKAAKERAERRLQSQQDDIDFKRAELALKRAMNRLSVAEMK 2e5y B 1.92 BS01 ATP B 1 E83 I88 D89 R92 A93 R122 R126 E83 I88 D89 R92 A93 R122 R126 3.6.3.14 0015986,0045261,0046933 Kd=22mM remove_due_to_license_issue P07678 17581881 1002 MKTIHVSVVTPDGPVYEDDVEMVSVKAKSGELGILPGHIPLVAPLEISAARLKKGGKTQYIAVSGGFLEVRPDKVTILAQAAERAEDIDVLRAKAAKERAERRLQSQQDDIDFKRAELALKRAMNRLSVAEMK 2e7f A 2.2 BS02 C2F A 1 E6 M11 F12 D75 N96 D160 G196 S198 N199 Q202 R207 I227 E6 M11 F12 D75 N96 D160 G196 S198 N199 Q202 R207 I227 2.1.1.258 0005509,0005515,0005829,0008168,0008705,0009086,0015977,0031419,0032259,0042558,0044237,0046653,0046872,0050667,0102036 Kd=0.79uM remove_due_to_license_issue Q46389 17172470 3000 MLIIGERINGMFGDIKRAIQERDPAPVQEWARRQEEGGARALDLNVGPAVQDKVSAMEWLVEVTQEVSNLTLCLDSTNIKAIEAGLKKCKNRAMINSTNAEREKVEKLFPLAVEHGAALIGLTMNKTGIPKDSDTRLAFAMELVAAADEFGLPMEDLYIDPLILPANVAQDHAPEVLKTLQQIKMLADPAPKTVLGLSNVSQNCQNRPLINRTFLAMAMACGLDAAIADACDEALIETAATAEILLNQTVYCDSFVKMFKTR 2e91 A 2.14 BS03 ZOL A 1 D80 R89 Q147 K174 D214 K238 D77 R86 Q144 K171 D207 K228 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue IC50=6.6e+2nM, Ki=260nM Q12051 17535895 901 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQMSGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN 2e92 A 2.31 BS03 M0N A 1 S76 D80 R89 L143 Q147 K174 D214 K238 S69 D73 R82 L136 Q140 K167 D201 K222 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue IC50=340nM, Ki=130nM Q12051 17535895 901 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQMSGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2e92 B 2.31 BS03 M0N B 1 D80 R89 L143 Q147 K174 Q211 D214 K238 D74 R83 L137 Q141 K168 Q199 D202 K222 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue IC50=340nM, Ki=130nM Q12051 17535895 902 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQMGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN 2e93 A 2.12 BS01 B29 A 1 S76 D80 R89 Y112 L140 Q147 K174 Q211 D214 S73 D77 R86 Y109 L137 Q144 K171 Q203 D206 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Ki=110nM, IC50=280nM Q12051 17535895 901 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPHSLVPFINLLGIIYQIRDDYLNLKDEKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDYIIDH 2e93 A 2.12 BS02 B29 A 2 G40 K41 R44 V69 E70 H73 L77 R89 R90 F179 Y210 K228 G37 K38 R41 V66 E67 H70 L74 R86 R87 F176 Y202 K215 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Ki=110nM, IC50=280nM Q12051 17535895 902 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPHSLVPFINLLGIIYQIRDDYLNLKDEKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDYIIDH 2e93 B 2.12 BS01 B29 B 1 G40 K41 R44 H73 R89 R90 F179 G37 K38 R41 H70 R86 R87 F176 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Ki=110nM, IC50=280nM Q12051 17535895 903 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQMFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPDELLYIIDHLSE 2e93 B 2.12 BS02 B29 B 2 S76 D80 R89 Y112 L140 L143 Q147 K174 Y210 Q211 D214 S73 D77 R86 Y109 L137 L140 Q144 K171 Y203 Q204 D207 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Ki=110nM, IC50=280nM Q12051 17535895 904 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQMFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPDELLYIIDHLSE 2e94 A 2.18 BS02 364 A 1 V69 H73 D80 R89 L178 F179 Y210 Q211 K238 V68 H72 D79 R88 L177 F178 Y207 Q208 K235 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Q12051 17535895 1101 TKNKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSGHSLVPFINLLGIIYQIRDDYLNLKDFQMSSEKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN 2e95 B 2.2 BS03 B75 B 1 R44 H73 D80 R89 K174 T175 L178 F179 T182 D214 K238 R41 H70 D77 R86 K171 T172 L175 F176 T179 D207 K228 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue IC50=200nM, Ki=80nM Q12051 17535895 1002 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQMSGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPYIIDHLS 2e98 A 1.9 BS01 B29 A 1 M25 N28 G29 H43 A47 A69 F70 S71 S72 E73 R77 I141 M11 N14 G15 H29 A33 A55 F56 S57 S58 E59 R63 I127 D26 H43 L137 D12 H29 L123 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 501 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e98 A 1.9 BS02 B29 A 2 R39 H43 R77 E81 L85 R25 H29 R63 E67 L71 D26 H43 L137 D12 H29 L123 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 502 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e98 A 1.9 BS03 B29 A 3 Y68 A69 L85 M86 F89 A143 N144 Y145 Y54 A55 L71 M72 F75 A129 N130 Y131 D26 H43 L137 D12 H29 L123 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 503 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e98 A 1.9 BS04 B29 A 4 R51 S55 L93 E96 S99 L100 H103 I141 R37 S41 L79 E82 S85 L86 H89 I127 D26 H43 L137 D12 H29 L123 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 504 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e99 A 2.0 BS01 B08 A 1 M25 N28 G29 R39 H43 V50 A69 F70 S71 S72 E73 R77 F89 M12 N15 G16 R26 H30 V37 A56 F57 S58 S59 E60 R64 F76 D26 H43 L137 D13 H30 L124 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 505 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e99 A 2.0 BS02 B08 A 2 V54 S55 N59 S99 L100 H103 V41 S42 N46 S86 L87 H90 D26 H43 L137 D13 H30 L124 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 506 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e99 A 2.0 BS03 B08 A 3 R39 H43 A69 R77 E81 L85 F89 R26 H30 A56 R64 E68 L72 F76 D26 H43 L137 D13 H30 L124 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 507 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e9a A 2.1 BS01 B28 A 1 M25 N28 G29 R39 H43 A47 A69 F70 S71 S72 F89 M12 N15 G16 R26 H30 A34 A56 F57 S58 S59 F67 D26 H43 L137 D13 H30 L115 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 701 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e9a A 2.1 BS02 B28 A 2 A40 H43 A69 S71 M86 F89 A27 H30 A56 S58 M64 F67 D26 H43 L137 D13 H30 L115 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 702 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e9c B 2.05 BS01 B75 B 1 M25 N28 G29 R39 H43 V50 A69 F70 S71 M9 N12 G13 R23 H27 V34 A53 F54 S55 D26 H43 L137 D10 H27 L111 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 703 GCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 2e9d A 2.5 BS01 B76 A 1 N28 H43 F70 S71 N13 H28 F55 S56 D26 H43 L137 D11 H28 L115 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 701 HGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e9d A 2.5 BS02 B76 A 2 V50 R51 V54 S55 E96 S99 L100 H103 V35 R36 V39 S40 E74 S77 L78 H81 D26 H43 L137 D11 H28 L115 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 17535895 702 HGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 2e9n A 2.5 BS01 76A A 1 L15 K38 E55 L84 Y86 C87 E91 D94 L137 D148 F149 L14 K37 E54 L83 Y85 C86 E90 D93 L136 D147 F148 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=6.2nM remove_due_to_license_issue EC50=>10000nM, IC50=4nM O14757 17287122 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2e9o A 2.1 BS01 A58 A 1 Q13 L15 A36 K38 L84 E85 Y86 C87 G90 L137 D148 Q12 L14 A35 K37 L83 E84 Y85 C86 G89 L136 D147 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=20nM remove_due_to_license_issue IC50=20nM O14757 17287122 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2e9u A 2.0 BS01 A25 A 1 L15 A36 V68 L84 E85 Y86 C87 G90 L137 S147 L14 A35 V67 L83 E84 Y85 C86 G89 L136 S146 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=10nM O14757 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2e9v A 2.0 BS01 85A A 1 L15 A36 K38 L84 E85 Y86 C87 G90 E91 L137 D148 L14 A35 K37 L83 E84 Y85 C86 G89 E90 L136 D147 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=13nM O14757 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2ea2 A 2.5 BS03 F77 A 1 H231 L328 N329 H331 I338 E364 F366 Y444 H122 L219 N220 H222 I229 E255 F257 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 ic50=0.016uM remove_due_to_license_issue IC50=16nM P50579 17350258 482 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 2ea4 A 2.35 BS03 F79 A 1 F219 H231 D251 D262 L328 N329 H331 H339 E364 F366 Y444 F110 H122 D142 D153 L219 N220 H222 H230 E255 F257 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 ic50=0.046uM remove_due_to_license_issue IC50=46nM P50579 17350258 482 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 2eep A 2.2 BS01 AIO A 1 Q203 E205 Y518 S603 Y604 Y635 E636 Y639 H710 Q137 E139 Y447 S530 Y531 Y562 E563 Y566 H637 Y518 S603 Y604 D678 H710 Y447 S530 Y531 D605 H637 3.4.14.12 0004177,0006508,0008236,0008239 remove_due_to_license_issue Q7MUW6 18042490 801 YPEYVVGLQWMGDNYVFIEGDDLVFNKTTRFSAADLNALMPFPSFRTLDAGRGLVVLFTQGGLVGFDMLARKVTYLFDTNEETASLDFSPVGDRVAYVRNHNLYIARGGKLGEGMSRAIAVTIDGTETLVYGQAVHQREFGIEKGTFWSPKGSCLAFYRMDQSMVKPTPIVDYHPLEAESKPLYYPMAGTPSHHVTVGIYHLATGKTVYLQTGEPKEKFLTNLSWSPDENILYVAEVNRAQNECKVNAYDAETGRFVRTLFVETDKHYVEPLHPLTFLPGSNNQFIWQSRRDGWNHLYLYDTTGRLIRQVTKGEWEVTNFAGFDPKGTRLYFESTEASPLERHFYCIDIKGGKTKDLTPESGMHRTQLSPDGSAIIDIFQSPTVPRKVTVTNIGKGSHTLLEAKNAMPEIRTGTIMAADGQTPLYYKLTMPLHFDPAKKYPVIVYVYGGPHAQLVTKTWRVGGWDIYMAQKGYAVFTVDSRGSANRGAAFEQVIHRRLGQTEMADQMCGVDFLKSQSWVDADRIGVHGWSYGGFMTTNLMLTHGDVFKVGVAGGPVIDWNRYEIMYGERYFDAPQENPEGYDAANLLKRAGDLKGRLMLIHGAIDPVVVWQHSLLFLDACVKARTYPDYYVYPSHEHNVMGPDRVHLYETITRYFTDHL 2efw A 2.5 BS01 dna D 0 K14 Q15 R16 R59 L82 Q83 K7 Q8 R9 R52 L75 Q76 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 3 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw A 2.5 BS02 dna E 0 T9 Y33 L35 H54 T55 Y58 H62 K77 Q83 T2 Y26 L28 H47 T48 Y51 H55 K70 Q76 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 1 ~ 19 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw B 2.5 BS01 dna D 0 T9 L35 K36 H54 T55 Y58 T2 L28 K29 H47 T48 Y51 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 3 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw B 2.5 BS02 dna E 0 R16 H54 T55 E56 R59 R9 H47 T48 E49 R52 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 1 ~ 19 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw F 2.5 BS01 dna I 0 Q15 T55 R59 K81 L82 Q83 Q8 T48 R52 K74 L75 Q76 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 3 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw F 2.5 BS02 dna J 0 Y33 L35 H54 Y58 R59 H62 V85 Y26 L28 H47 Y51 R52 H55 V78 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 1 ~ 19 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKKEGAKLQEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw G 2.5 BS01 dna I 0 T9 L35 H54 Y58 T2 L28 H47 Y51 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 3 ~ 21 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2efw G 2.5 BS02 dna J 0 T55 R59 T48 R52 ? 0003677,0006274 remove_due_to_license_issue P0CI76 17521668 1 ~ 19 STGFLVKQRAFLKLYMITMTEQERLYGLKLLEVLRSEFKEIGFKPNHTEVYRSLHELLDDGILKQIKVKEVVLYQFKDYEAAKLYKKQLKVELDRSKKLIEKALSDNF 2eg7 A 2.0 BS03 OTD A 1 H18 R20 K102 H139 H177 C221 L222 D250 H254 A266 G267 H15 R17 K99 H136 H174 C218 L219 D247 H251 A263 G264 H16 H18 K102 H139 H177 D250 H13 H15 K99 H136 H174 D247 3.5.2.3 0004151,0005737,0005829,0006207,0006221,0008270,0016787,0016812,0019856,0042803,0044205,0046872 Ki=1.3uM remove_due_to_license_issue P05020 17550785 410 SQVLKIRRPDDWHLHLRDGDMLKTVVPYTSEIYGRAIVMPNLAPPVTTVEAAVAYRQRILDAVPAGHDFTPLMTCYLTDSLDPNELERGFNEGVFTAAKLYPANATTNSSHGVTSVDAIMPVLERMEKIGMPLLVHGEVTHADIDIFDREARFIESVMEPLRQRLTALKVVFEHITTKDAADYVRDGNERLAATITPQHLMFNRNHMLVGGVRPHLYCLPILKRNIHQQALRELVASGFNRVFLGTDSAPHARHRKESSCGCAGCFNAPTALGSYATVFEEMNALQHFEAFCSVNGPQFYGLPVNDTFIELVREEQQVAESIALTDDTLVPFLAGETVRWSVK 2eg8 A 2.2 BS03 FOT A 1 R20 N44 H139 C221 L222 H254 A266 G267 R17 N41 H136 C218 L219 H251 A263 G264 H16 H18 K102 H139 H177 D250 H13 H15 K99 H136 H174 D247 3.5.2.3 0004151,0005737,0005829,0006207,0006221,0008270,0016787,0016812,0019856,0042803,0044205,0046872 Ki=31.8uM remove_due_to_license_issue P05020 17550785 410 SQVLKIRRPDDWHLHLRDGDMLKTVVPYTSEIYGRAIVMPNLAPPVTTVEAAVAYRQRILDAVPAGHDFTPLMTCYLTDSLDPNELERGFNEGVFTAAKLYPANATTNSSHGVTSVDAIMPVLERMEKIGMPLLVHGEVTHADIDIFDREARFIESVMEPLRQRLTALKVVFEHITTKDAADYVRDGNERLAATITPQHLMFNRNHMLVGGVRPHLYCLPILKRNIHQQALRELVASGFNRVFLGTDSAPHARHRKESSCGCAGCFNAPTALGSYATVFEEMNALQHFEAFCSVNGPQFYGLPVNDTFIELVREEQQVAESIALTDDTLVPFLAGETVRWSVK 2ei6 A 2.3 BS03 D92 A 1 T98 Y99 F174 A190 C191 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 T84 Y85 F162 A180 C181 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=16nM remove_due_to_license_issue IC50=16nM P00742 17555959 700 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2epn A 1.61 BS01 NGT A 1 R95 H170 D223 E224 W267 W307 Y309 W340 W374 D376 R91 H166 D219 E220 W263 W303 Y305 W336 W370 D372 3.2.1.52 0015929,0016231,0016798 Ki=60nM remove_due_to_license_issue Q6ST21 18237743 1650 ATFLGLSSKQEKALVRLDKYLNLGEIAVSLVATSIKVEGRQGYYQVSYKQPHQLYRALALLSAALRSGQDEVQIEEEAAYEDLAYMADCSRNAVLNLSSAKKMIEVLALMGYSTFELYMEDTYEIENQPYFGYFRGRYTVAELQEIEDYAADFDMSFVPCIQTLAHLSAFVKWGIKEVQELRDVEDILLIGEEKVYDLIEGMFQTMAHLHTRKINIGMDEAHLVGLGRYLIKHGFQNRSLLMCQHLERVLDIADKYGFNCQMWSDMFFKLMSADGQYDRDVEIPEETRVYLDRLKERVTLVYWDYYQDSEEKYNRNFQNHHKISQDIAFAGGAWKWIGFTPHNHFSRLVAIEANKACRKNQVKEVIVTGWGDNGGETSQFSVLPALQIWAELAYRNDLKKVSEHFLVSTGLDFDDFMKIDLANLLPDLPDNLSGINPNRYVLYQDVLCPLLEQHIRPEKDKQHFASSAQQLGEISKRAGEYAYIFETQAQLNALLALKISITSGIQKAYRNGDKEHLSALAEKDFPQLYQMVEDFSDQFSRQWQQENKIFGLDTIDIRFGGLLKRIKRAQERLEQFISGQIDCVEELEQEILPFNDFYKDQGLTATTANQWHLIATASTIYTT 2epn B 1.61 BS01 NGT B 1 R95 H170 D223 E224 W267 W307 Y309 W340 W374 D376 R91 H166 D219 E220 W263 W303 Y305 W336 W370 D372 3.2.1.52 0015929,0016231,0016798 Ki=60nM remove_due_to_license_issue Q6ST21 18237743 2650 ATFLGLSSKQEKALVRLDKYLNLGEIAVSLVATSIKVEGRQGYYQVSYKQPHQLYRALALLSAALRSGQDEVQIEEEAAYEDLAYMADCSRNAVLNLSSAKKMIEVLALMGYSTFELYMEDTYEIENQPYFGYFRGRYTVAELQEIEDYAADFDMSFVPCIQTLAHLSAFVKWGIKEVQELRDVEDILLIGEEKVYDLIEGMFQTMAHLHTRKINIGMDEAHLVGLGRYLIKHGFQNRSLLMCQHLERVLDIADKYGFNCQMWSDMFFKLMSADGQYDRDVEIPEETRVYLDRLKERVTLVYWDYYQDSEEKYNRNFQNHHKISQDIAFAGGAWKWIGFTPHNHFSRLVAIEANKACRKNQVKEVIVTGWGDNGGETSQFSVLPALQIWAELAYRNDLKKVSEHFLVSTGLDFDDFMKIDLANLLPDLPDNLSGINPNRYVLYQDVLCPLLEQHIRPEKDKQHFASSAQQLGEISKRAGEYAYIFETQAQLNALLALKISITSGIQKAYRNGDKEHLSALAEKDFPQLYQMVEDFSDQFSRQWQQENKIFGLDTIDIRFGGLLKRIKRAQERLEQFISGQIDCVEELEQEILPFNDFYKDQGLTATTANQWHLIATASTIYTT 2ere A 3.0 BS01 dna C 0 A36 R41 K44 K46 R79 A2 R7 K10 K12 R40 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 1 ~ 15 FACVECRQQKSKCDAHPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2ere A 3.0 BS02 dna D 0 Q43 K44 R75 Y77 K78 R79 Q9 K10 R36 Y38 K39 R40 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 16 ~ 30 FACVECRQQKSKCDAHPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2ere B 3.0 BS01 dna C 0 Q43 K44 R75 Y77 K78 R79 Q9 K10 R36 Y38 K39 R40 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 1 ~ 15 FACVECRQQKSKCDAHPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2ere B 3.0 BS02 dna D 0 F35 A36 R41 K44 K46 R79 F1 A2 R7 K10 K12 R40 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 16 ~ 30 FACVECRQQKSKCDAHPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2erg A 3.15 BS01 dna C 0 F35 A36 R41 K44 R79 F1 A2 R7 K10 R45 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 1 ~ 15 FACVECRQQKSKCDACERAPEPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2erg A 3.15 BS02 dna D 0 Q43 K44 R75 Y77 K78 R79 Q9 K10 R41 Y43 K44 R45 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 16 ~ 30 FACVECRQQKSKCDACERAPEPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2erg B 3.15 BS01 dna C 0 Q43 K44 R75 Y77 K78 R79 Q9 K10 R41 Y43 K44 R45 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 1 ~ 15 FACVECRQQKSKCDACERAPEPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2erg B 3.15 BS02 dna D 0 F35 A36 R41 K44 R79 F1 A2 R7 K10 R45 ? 0000981,0006355,0008270 remove_due_to_license_issue P08638 16615914 16 ~ 30 FACVECRQQKSKCDACERAPEPCTKCAKKNVPCILKRDFRRTYKRARNEAIEKRFKELTRTLTNL 2err A -1.00 BS01 rna B 0 R118 H120 S122 N123 I124 F126 E147 I148 I149 N151 R153 G154 K156 G157 F158 F160 R184 N189 N190 A191 T192 A193 R194 R10 H12 S14 N15 I16 F18 E39 I40 I41 N43 R45 G46 K48 G49 F50 F52 R76 N81 N82 A83 T84 A85 R86 ? 0000381,0003676,0003723,0007399 remove_due_to_license_issue Q9NWB1 16362037 197 ~ 203 NTENKSQPKRLHVSNIPFRFRDPDLRQMFGQFGKILDVEIIFNERGSKGFGFVTFENSADADRAREKLHGTVVEGRKIEVNNATARVM 2erz E 2.2 BS02 HFS E 1 L49 T51 V57 A70 E121 Y122 N171 L173 T183 F327 L35 T37 V43 A56 E107 Y108 N157 L159 T169 F313 N171 D184 N157 D170 2.7.11.11 0000122,0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,0141156,1904262,1904539,1990044,2000810 Ki=2.2uM remove_due_to_license_issue P05132 16249185 351 VKEFLAKAKEDFLKKWETPSQNTAQLDQFDRIKTLGTGSFGRVMLVKHKESGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 2es2 A 1.78 BS01 dna B 0 K7 W8 F15 F17 D25 F27 H29 R56 Q59 K7 W8 F15 F17 D25 F27 H29 R56 Q59 ? 0003676,0003677,0005737,0009295,0010468 remove_due_to_license_issue P32081 16780871 1 ~ 6 MLEGKVKWFNSEKGFGFIEVEGQDDVFVHFSAIQGEGFKTLEEGQAVSFEIVEGNRGPQAANVTKEA 2etk A 2.96 BS01 HFS A 1 V90 A103 M153 E154 Y155 M156 D202 D216 F368 V85 A98 M148 E149 Y150 M151 D197 D211 F363 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=150nM Q13464 16249185 416 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSNRRY 2etm A 2.3 BS01 7PY A 1 I428 V436 A452 L501 C502 G505 L553 I14 V22 A38 L87 C88 G91 L139 D546 A548 R550 N551 D564 K583 D132 A134 R136 N137 D150 K159 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=200nM Q05397 131 YEIQRERIELGRCIGEGQFGDVHQGIYMSPENPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSRYMEKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 2etr A 2.6 BS01 Y27 A 1 I82 A103 M156 N203 D216 F368 I77 A98 M151 N198 D211 F363 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=150nM, IC50=200nM Q13464 16249185 416 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSNRRY 2euf B 3.0 BS01 LQQ B 1 I19 F98 E99 V101 D102 Q103 D104 T107 L152 A162 D163 I10 F89 E90 V92 D93 Q94 D95 T98 L143 A153 D154 D145 K147 Q149 N150 D163 A175 T182 D136 K138 Q140 N141 D154 A166 T173 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue IC50=16nM, Ki=27nM Q00534 16789739 401 DQQYECVAEIGEGAYGKVFKARDLKNGGRFVALKRVRVQTGEEGMPLSTIREVAVLRHLETFEHPNVVRLFDVCTVSRTDRETKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLARIYSFQMALTSVVVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQDLER 2euk A 1.85 BS01 GAL A 1 D48 N52 K55 W96 Y207 D45 N49 K52 W93 Y202 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 300 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2euk A 1.85 BS02 SPH A 1 D48 W96 D45 W93 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 301 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2eum A 2.3 BS02 SPH A 1 D48 W96 D45 W93 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 301 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSKQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2eum A 2.3 BS03 OCA A 1 I45 D48 W96 F103 L136 H140 I42 D45 W93 F100 L133 H137 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 302 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSKQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2evc A 1.6 BS03 FC3 A 1 C59 Y62 H63 Y65 C70 H79 D97 D108 H171 H178 E204 W221 E235 C56 Y59 H60 Y62 C67 H76 D94 D105 H168 H175 E201 W218 E232 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H76 D94 D105 H168 R172 H175 Q179 E201 N205 Q230 E232 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.29uM remove_due_to_license_issue IC50=158000nM P0AE18 16552144 999 SIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISH 2evl A 2.2 BS01 GAL A 1 D48 N52 W96 Y207 D45 N49 W93 Y203 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 300 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSKQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2evl A 2.2 BS02 SPH A 1 D48 W96 I147 D45 W93 I144 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 301 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSKQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2evl A 2.2 BS03 EIC A 1 F34 I45 D48 W96 F103 F107 L136 F148 F31 I42 D45 W93 F100 F104 L133 F145 ? 0005515,0005737,0005829,0006869,0008289,0017089,0035627,0035902,0042802,0046836,0051861,0120009,0120013,1902387,1902388,1902389 remove_due_to_license_issue Q9NZD2 17105344 302 LAEHLLKPLPADKQIETGPFLEAVSHLPPFFDCLGSPVFTPIKADISGNITKIKAVYDTNPAKFRTLQNILEVEKEMYGAEWPKVGATLALMWLKRGLRFIQVFLQSICDGERDENHPNLIRVNATKAYEMALKKYHGWIVQKIFQAALYAAPYKSDFLKALSKQNVTEEECLEKIRLFLVNYTATIDVIYEMYTQMNAELNYKV 2evm A 1.7 BS03 FC2 A 1 Y62 H63 Y65 C70 H79 D97 D108 H171 H178 E204 W221 E235 Y59 H60 Y62 C67 H76 D94 D105 H168 H175 E201 W218 E232 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H76 D94 D105 H168 R172 H175 Q179 E201 N205 Q230 E232 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.693uM remove_due_to_license_issue IC50=84000nM P0AE18 16552144 999 SIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISH 2ew5 A 2.2 BS02 Y12 A 1 S42 G44 I45 G46 E94 G95 C96 L97 Y103 L131 H138 E139 S41 G43 I44 G45 E93 G94 C95 L96 Y102 L130 H137 E138 G46 Q51 C96 L97 H138 E139 H142 G45 Q50 C95 L96 H137 E138 H141 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=1.25uM remove_due_to_license_issue Q672W7 16882991 200 ALLEIIHYPSKILRTISKEVVSFDAKLHQQLDDMYETMIASEGIGLAAIQVGLPLRMLIINLPQEDGVQHKEDCLEIINPKFIETGGSMMYKEGCLSVPGFYEEVERFEKVKIEYQNRFAEVKVLEASELLAVAIQHEIDHLNGVLFVDKLSILKRKKFEKELKEL 2ew6 A 2.2 BS02 Y13 A 1 G44 I45 G46 Y92 E94 G95 C96 L97 P100 Y103 L131 V134 A135 H138 E139 G43 I44 G45 Y91 E93 G94 C95 L96 P99 Y102 L130 V133 A134 H137 E138 G46 Q51 C96 L97 H138 E139 H142 G45 Q50 C95 L96 H137 E138 H141 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=10.8uM remove_due_to_license_issue Q672W7 16882991 200 ALLEIIHYPSKILRTISKEVVSFDAKLHQQLDDMYETMIASEGIGLAAIQVGLPLRMLIINLPQEDGVQHKEDCLEIINPKFIETGGSMMYKEGCLSVPGFYEEVERFEKVKIEYQNRFAEVKVLEASELLAVAIQHEIDHLNGVLFVDKLSILKRKKFEKELKEL 2ewa A 2.1 BS01 SB2 A 1 Y35 V38 A51 K53 I84 L104 V105 T106 M109 F169 G170 Y31 V34 A47 K49 I80 L100 V101 T102 M105 F160 G161 D150 K152 N155 D168 T185 D141 K143 N146 D159 T162 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 remove_due_to_license_issue P47811 16374788 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNILTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGTRWYRAPEIMLNMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 2ewb A 1.85 BS04 ZED A 1 K250 D255 K262 N330 D332 E334 L360 T361 I421 K250 D255 K262 N330 D332 E334 L360 T361 I421 K262 R336 K262 R336 3.4.11.1,3.4.11.5,3.4.13.23 0004177,0004180,0005737,0005739,0006508,0008233,0016805,0019538,0030145,0046872,0070006,0097718 Ki=0.8uM remove_due_to_license_issue P00727 16519517 2000 TKGLVLGIYSKEKEEDEPQFTSAGENFNKLVSGKLREILNISGPPLKAGKTRTFYGLHEDFPSVVVVGLGKKTAGIDEQENWHEGKENIRAAVAAGCRQIQDLEIPSVEVDPCGDAQAAAEGAVLGLYEYDDLKQKRKVVVSAKLHGSEDQEAWQRGVLFASGQNLARRLMETPANEMTPTKFAEIVEENLKSASIKTDVFIRPKSWIEEQEMGSFLSVAKGSEEPPVFLEIHYKGSPNASEPPLVFVGKGITFDSGGISIKAAANMDLMRADMGGAATICSAIVSAAKLDLPINIVGLAPLCENMPSGKANKPGDVVRARNGKTIQVDNTDAEGRLILADALCYAHTFNPKVIINAATLTGAMDIALGSGATGVFTNSSWLWNKLFEASIETGDRVWRMPLFEHYTRQVIDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHLDIAGVMTNKDEVPYLRKGMAGRPTRTLIEFLFRFSQDS 2ewp A 2.3 BS01 TXF A 1 C269 A272 D273 E275 L309 V313 Y326 N346 F435 L440 E441 C37 A40 D41 E43 L77 V81 Y94 N114 F203 L208 E209 ? ic50=0.079uM remove_due_to_license_issue IC50=77nM P62508 16307879 501 PYNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEA 2ews A 2.05 BS01 ANP A 1 G8 G9 T10 L11 K13 G98 T99 G121 Q125 Y137 S225 S226 G8 G9 T10 L11 K13 G98 T99 G121 Q125 Y137 S218 S219 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q6G7I0 16905099 1001 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLEK 2ews B 2.05 BS01 ANP B 1 G8 G9 T10 L11 K13 G98 T99 G121 Q125 Y137 S225 S226 G8 G9 T10 L11 K13 G98 T99 G121 Q125 Y137 S217 S218 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q6G7I0 16905099 1002 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLE 2ewy A 3.1 BS01 DBO A 1 L46 D48 G50 Y87 T88 F124 W131 Y211 D241 G243 T244 T245 R248 L31 D33 G35 Y72 T73 F109 W116 Y187 D217 G219 T220 T221 R224 D48 S51 N53 A55 Y87 D241 T244 D33 S36 N38 A40 Y72 D217 T220 3.4.23.45 0004190,0006508,0016020 remove_due_to_license_issue Q9Y5Z0 16305800 1001 LAMVDNLQGDSGRGYYLEMLIGTPPQKLQILVDTGSSNFAVAGTPHSYIDTYFDTERSSTYRSKGFDVTVKYTQGSWTGFVGEDLVTIPKGFNTSFLVNIATIFESENFFLPGIKWNGILGLAYATLAKPSSSLETFFDSLVTQANIPNVFSMQMCGANGGSLVLGGIEPSLYKGDIWYTPIKEEWYYQIEILKLEIGGQSLNLDCREYNADKAIVDSGTTLLRLPQKVFDAVVEAVARASLIPEFSDGFWTGSQLACWTNSETPWSYFPKISIYLRDENSSRSFRITILPQLYIQPMMGAGLNYECYRFGISPSTNALVIGATVMEGFYVIFDRAQKRVGFAASPCAEIAGAAVSEISGPFSTEDVASNCVPA 2exc X 2.75 BS01 JNK X 1 I70 V78 K93 L144 V145 M146 M149 D150 V196 L206 I26 V31 K46 L97 V98 M99 M102 D103 V149 L159 N194 D207 N147 D160 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=235nM P53779 600 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLAVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQLDEREHTIEEWKELIYKEVMN 2exg A -1.00 BS01 STF A 1 M23 G24 L25 I27 M83 M23 G24 L25 I27 M83 ? 0005911 remove_due_to_license_issue P55196 16671149 102 GPLGSLRKEPEIITVTLKKQNGMGLSIVAAKGAGQDKLGIYVKSVVKGGAADVDGRLAAGDQLLSVDGRSLVGLSQERAAELMTRTSSVVTLEVAKQGAIY 2exm A 1.8 BS01 ZIP A 1 I10 G11 V18 A31 K33 E81 L83 L134 I10 G11 V18 A31 K33 E81 L83 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 7479711 400 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2ez7 A 2.0 BS02 DHI A 1 W5 H64 P201 W3 H62 P198 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=43.5uM remove_due_to_license_issue P00918 16807956 301 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2f01 A 0.85 BS01 BTN A 1 L25 S27 Y43 S45 V47 N49 W79 S88 T90 W108 D128 L12 S14 Y30 S32 V34 N36 W66 S75 T77 W95 D115 ? 0009374 Kd~0.1pM remove_due_to_license_issue Kd=1.000000nM P22629 16699183 5100 EAGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVK 2f0z A 2.8 BS01 ZMR A 1 R21 I22 E39 M85 N86 E111 Y179 Y181 E218 R237 R304 Y334 R19 I20 E37 M76 N77 E102 Y170 Y172 E205 R221 R283 Y313 E218 E205 3.2.1.18 0004308,0005515,0005737,0005764,0005829,0006516,0006689,0009313,0016020,0016042,0016798,0046479,1902494 remove_due_to_license_issue IC50=7800nM, Ki=5700nM Q9Y3R4 381 SLPVLQKESVFQSGAHAYRIPALLYLPGQQSLLAFAEQRAELIVLRRGDYDAPTHQVQWQAQEVVAQARLDGHRSMNPCPLYDAQTGTLFLFFIAIPGQVTEQQQLQTRANVTRLCQVTSTDHGRTWSSPRDLTDAAIGPAYREWSTFAVGPGHCLQLNDRARSLVVPAYAYRKLRPIPSAFCFLSHDHGRTWARGHFVAQDTLECQVAEVEQRVVTLNARSHLRARVQAQSTNDGLDFQESQLVKKLVEPPPQGCQGSVISFPSPRPAQWLLYTHPTHSWQRADLGAYLNPRPPAPEAWSEPVLLAKGSCAYSDLQSMGTGPDGSPLFGCLYEANDYEEIVFLMFTLKQAFPAEY 2f10 A 2.9 BS01 BCZ A 1 R21 E218 R237 R304 Y334 R19 E199 R215 R276 Y306 E218 E199 3.2.1.18 0004308,0005515,0005737,0005764,0005829,0006516,0006689,0009313,0016020,0016042,0016798,0046479,1902494 remove_due_to_license_issue Ki=56000nM, IC50=70000nM Q9Y3R4 382 SLPVLQKESVFQSGAHAYRIPALLYLPGQQSLLAFAEQRAAELIVLRRGDYDAPTHQVQWQAQEVVAQARLDGHRSMNPCPLYDAQTGTLFLFFIAIPGRANVTRLCQVTSTDHGRTWSSPRDLTDAAIGPAYREWSTFAVGPGHCLQLNDRARSLVVPAYAYRKLHIQRPIPSAFCFLSHDHGRTWARGHFVAQDTLECQVAEVEQRVVTLNARSHLRARVQAQSTNDGLDFQESQLVKKLVEPPPQGCQGSVISFPSPRAQWLLYTHPTHSWQRADLGAYLNPRPPAPEAWSEPVLLAKGSCAYSDLQSMGTGPDGSPLFGCLYEANDYEEIVFLMFTLKQAFPAEY 2f14 A 1.71 BS03 FL1 A 1 H94 H119 D130 F131 G132 L198 T199 T200 P202 H91 H116 D126 F127 G128 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.64nM remove_due_to_license_issue Ki=45nM P00918 16787097 1270 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2f18 A 1.3 BS02 GB1 A 1 H90 D92 W95 D204 Y269 D340 D341 H471 D472 G877 H60 D62 W65 D174 Y239 D310 D311 H441 D442 G847 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=80uM remove_due_to_license_issue Q24451 17557336 1804 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 2f1a A 1.45 BS02 GB2 A 1 H90 D92 W95 D204 Y269 D341 H471 D472 G877 H60 D62 W65 D174 Y239 D311 H441 D442 G847 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=720uM remove_due_to_license_issue Q24451 17557336 1804 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 2f1b A 1.45 BS02 GB3 A 1 H90 D92 W95 D204 F206 Y269 D340 D341 H471 D472 Y727 G877 H60 D62 W65 D174 F176 Y239 D310 D311 H441 D442 Y697 G847 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=1000uM remove_due_to_license_issue Q24451 17557336 1803 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 2f1g A 1.9 BS01 GNF A 1 Q19 G23 C25 G62 K64 G68 G69 F70 M71 G137 N163 H164 G165 W186 Q22 G26 C28 G65 K67 G71 G72 F73 M74 G140 N166 H167 G168 W189 Q19 C25 H164 N184 Q22 C28 H167 N187 3.4.22.27 0006508,0008234 Ki=0.029uM remove_due_to_license_issue Ki=29nM P25774 16446091 1002 NRILPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 2f2c B 2.8 BS01 AP9 B 1 V27 A41 F98 V101 D102 Q103 D104 T107 Q149 L152 V14 A28 F84 V87 D88 Q89 D90 T93 Q135 L138 D145 K147 Q149 N150 D163 A175 T182 D131 K133 Q135 N136 D149 A161 T168 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue Q00534 16789739 401 ADQQYECAEIGGKVFKARDLKNGGRFVALKRVRVQTGEEGMPLSTIREVAVLRHLETFEHPNVVRLFDVCTVSTDRETKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLARIYSFQMALTSVVVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPQAFAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQDLER 2f2h A 1.95 BS01 XTG A 1 D185 F277 D306 K414 R466 W479 D482 F515 H540 D185 F277 D306 K414 R466 W479 D482 F515 H540 3.2.1.177 0003824,0004553,0005975,0016798,0030246,0042802,0061634,0080176 Ki=2uM remove_due_to_license_issue P31434 16478160 3015 MKISDGNWLIQPGLNLIHPLQVFEVEQQDNEMVVYAAPRDVRERTWQLDTPLFTLRFFSPQEGIVGVRIEHFQGALNNGPHYPLNILQDVKVTIENTERYAEFKSGNLSARVSKGEFWSLDFLRNGERITGSQVKNNGYVQDTNNQRNYMFERLDLGVGETVYGLGERFTALVRNGQTVETWNRDGGTSTEQAYKNIPFYMTNRGYGVLVNHPQCVSFEVGSEKVSKVQFSVESEYLEYFVIDGPTPKAVLDRYTRFTGRPALPPAWSFGLWLTTSFTTNYDEATVNSFIDGMAERNLPLHVFHFDCFWMKAFQWCDFEWDPLTFPDPEGMIRRLKAKGLKICVWINPYIGQKSPVFKELQEKGYLLKRPDGSLWQWDKWQPGLAIYDFTNPDACKWYADKLKGLVAMGVDCFKTDFGERIPTDVQWFDGSDPQKMHNHYAYIYNELVWNVLKDTVGEEEAVLFARSASVGAQKFPVHWGGDCYANYESMAESLRGGLSIGLSGFGFWSHDIGGFENTAPAHVYKRWCAFGLLSSHSRLHGSKSYRVPWAYDDESCDVVRFFTQLKCRMMPYLYREAARANARGTPMMRAMMMEFPDDPACDYLDRQYMLGDNVMVAPVFTEAGDVQFYLPEGRWTHLWHNDELDGSRWHKQQHGFLSLPVYVRDNTLLALGNNDQRPDYVWHEGTAFHLFNLQDGHEAVCEVPAADGSVIFTLKAARTGNTITVTGAGEAKNWTLCLRNVVKVNGLQDGSQAESEQGLVVKPQGNALTITLH 2f2h B 1.95 BS01 XTG A 1 T45 D49 T45 D49 3.2.1.177 0003824,0004553,0005975,0016798,0030246,0042802,0061634,0080176 Ki=2uM remove_due_to_license_issue P31434 16478160 3015 MKISDGNWLIQPGLNLIHPLQVFEVEQQDNEMVVYAAPRDVRERTWQLDTPLFTLRFFSPQEGIVGVRIEHFQGALNNGPHYPLNILQDVKVTIENTERYAEFKSGNLSARVSKGEFWSLDFLRNGERITGSQVKNNGYVQDTNNQRNYMFERLDLGVGETVYGLGERFTALVRNGQTVETWNRDGGTSTEQAYKNIPFYMTNRGYGVLVNHPQCVSFEVGSEKVSKVQFSVESEYLEYFVIDGPTPKAVLDRYTRFTGRPALPPAWSFGLWLTTSFTTNYDEATVNSFIDGMAERNLPLHVFHFDCFWMKAFQWCDFEWDPLTFPDPEGMIRRLKAKGLKICVWINPYIGQKSPVFKELQEKGYLLKRPDGSLWQWDKWQPGLAIYDFTNPDACKWYADKLKGLVAMGVDCFKTDFGERIPTDVQWFDGSDPQKMHNHYAYIYNELVWNVLKDTVGEEEAVLFARSASVGAQKFPVHWGGDCYANYESMAESLRGGLSIGLSGFGFWSHDIGGFENTAPAHVYKRWCAFGLLSSHSRLHGSKSYRVPWAYDDESCDVVRFFTQLKCRMMPYLYREAARANARGTPMMRAMMMEFPDDPACDYLDRQYMLGDNVMVAPVFTEAGDVQFYLPEGRWTHLWHNDELDGSRWHKQQHGFLSLPVYVRDNTLLALGNNDQRPDYVWHEGTAFHLFNLQDGHEAVCEVPAADGSVIFTLKAARTGNTITVTGAGEAKNWTLCLRNVVKVNGLQDGSQAESEQGLVVKPQGNALTITLH 2f2h B 1.95 BS02 XTG B 1 D185 D306 K414 D416 R466 W479 D482 F515 H540 D185 D306 K414 D416 R466 W479 D482 F515 H540 3.2.1.177 0003824,0004553,0005975,0016798,0030246,0042802,0061634,0080176 Ki=2uM remove_due_to_license_issue P31434 16478160 3016 MKISDGNWLIQPGLNLIHPLQVFEVEQQDNEMVVYAAPRDVRERTWQLDTPLFTLRFFSPQEGIVGVRIEHFQGALNNGPHYPLNILQDVKVTIENTERYAEFKSGNLSARVSKGEFWSLDFLRNGERITGSQVKNNGYVQDTNNQRNYMFERLDLGVGETVYGLGERFTALVRNGQTVETWNRDGGTSTEQAYKNIPFYMTNRGYGVLVNHPQCVSFEVGSEKVSKVQFSVESEYLEYFVIDGPTPKAVLDRYTRFTGRPALPPAWSFGLWLTTSFTTNYDEATVNSFIDGMAERNLPLHVFHFDCFWMKAFQWCDFEWDPLTFPDPEGMIRRLKAKGLKICVWINPYIGQKSPVFKELQEKGYLLKRPDGSLWQWDKWQPGLAIYDFTNPDACKWYADKLKGLVAMGVDCFKTDFGERIPTDVQWFDGSDPQKMHNHYAYIYNELVWNVLKDTVGEEEAVLFARSASVGAQKFPVHWGGDCYANYESMAESLRGGLSIGLSGFGFWSHDIGGFENTAPAHVYKRWCAFGLLSSHSRLHGSKSYRVPWAYDDESCDVVRFFTQLKCRMMPYLYREAARANARGTPMMRAMMMEFPDDPACDYLDRQYMLGDNVMVAPVFTEAGDVQFYLPEGRWTHLWHNDELDGSRWHKQQHGFLSLPVYVRDNTLLALGNNDQRPDYVWHEGTAFHLFNLQDGHEAVCEVPAADGSVIFTLKAARTGNTITVTGAGEAKNWTLCLRNVVKVNGLQDGSQAESEQGLVVKPQGNALTITLH 2f2h D 1.95 BS01 XTG D 1 D185 D306 C307 K414 D416 R466 W479 D482 F515 H540 D185 D306 C307 K414 D416 R466 W479 D482 F515 H540 3.2.1.177 0003824,0004553,0005975,0016798,0030246,0042802,0061634,0080176 Ki=2uM remove_due_to_license_issue P31434 16478160 3018 MKISDGNWLIQPGLNLIHPLQVFEVEQQDNEMVVYAAPRDVRERTWQLDTPLFTLRFFSPQEGIVGVRIEHFQGALNNGPHYPLNILQDVKVTIENTERYAEFKSGNLSARVSKGEFWSLDFLRNGERITGSQVKNNGYVQDTNNQRNYMFERLDLGVGETVYGLGERFTALVRNGQTVETWNRDGGTSTEQAYKNIPFYMTNRGYGVLVNHPQCVSFEVGSEKVSKVQFSVESEYLEYFVIDGPTPKAVLDRYTRFTGRPALPPAWSFGLWLTTSFTTNYDEATVNSFIDGMAERNLPLHVFHFDCFWMKAFQWCDFEWDPLTFPDPEGMIRRLKAKGLKICVWINPYIGQKSPVFKELQEKGYLLKRPDGSLWQWDKWQPGLAIYDFTNPDACKWYADKLKGLVAMGVDCFKTDFGERIPTDVQWFDGSDPQKMHNHYAYIYNELVWNVLKDTVGEEEAVLFARSASVGAQKFPVHWGGDCYANYESMAESLRGGLSIGLSGFGFWSHDIGGFENTAPAHVYKRWCAFGLLSSHSRLHGSKSYRVPWAYDDESCDVVRFFTQLKCRMMPYLYREAARANARGTPMMRAMMMEFPDDPACDYLDRQYMLGDNVMVAPVFTEAGDVQFYLPEGRWTHLWHNDELDGSRWHKQQHGFLSLPVYVRDNTLLALGNNDQRPDYVWHEGTAFHLFNLQDGHEAVCEVPAADGSVIFTLKAARTGNTITVTGAGEAKNWTLCLRNVVKVNGLQDGSQAESEQGLVVKPQGNALTITLH 2f34 A 1.74 BS01 UBA A 1 Y61 P88 L89 T90 R95 V137 G140 S141 T142 Y216 Y58 P85 L86 T87 R92 V134 G137 S138 T139 Y213 ? 0015276,0016020 Kd=0.13uM remove_due_to_license_issue Kd=18nM P22756 16540562 801 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGN 2f35 A 1.87 BS01 UBC A 1 Y61 P88 L89 T90 R95 V137 G140 S141 T142 Y216 Y58 P85 L86 T87 R92 V134 G137 S138 T139 Y213 ? 0015276,0016020 Kd=3.94uM remove_due_to_license_issue Kd=402nM P22756 16540562 801 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGN 2f3e A 2.11 BS01 AXQ A 1 Q12 G13 L30 D32 G34 P70 Y71 T72 Q73 Y198 D228 G230 T231 T232 Q15 G16 L33 D35 G37 P73 Y74 T75 Q76 Y190 D220 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=156nM remove_due_to_license_issue P56817 16854060 601 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2f3f A 2.3 BS01 AXF A 1 G11 Q12 D32 G34 Y71 T72 Q73 F108 D228 G230 T232 G14 Q15 D35 G37 Y74 T75 Q76 F111 D218 G220 T222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=190nM remove_due_to_license_issue P56817 16854060 601 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2f3k A 1.599 BS01 RO1 A 1 D25 I47 G49 I50 P81 D25 I47 G49 I50 P81 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Kd=0.95nM remove_due_to_license_issue O38708 16569872 506 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2f3k B 1.599 BS01 RO1 A 1 D25 G27 A28 D29 D30 G48 P81 I84 D25 G27 A28 D29 D30 G48 P81 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue O38708 16569872 506 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2f3r A 2.5 BS01 G5P A 1 S13 G14 G16 K17 S18 S19 S38 R42 R45 Y54 E73 Y82 G83 D102 I103 D104 R134 G137 S12 G13 G15 K16 S17 S18 S37 R41 R44 Y53 E72 Y81 G82 D101 I102 D103 R133 G136 2.7.4.8 0004385,0005524,0005737,0005829,0006163,0016301,0042802,0046037,0046710 ic50=0.5uM remove_due_to_license_issue P60546 16690197 601 AQGTLYIVSAPSGAGKSSLIQALLKTQPLYDTQVSVSHTTRQPRPGEVHGEHYFFVNHDEFKEMISRDAFLEHAEVFGNYYGTSREAIEQVLATGVDVFLDIDWQGAQQIRQKMPHARSIFILPPSKIELDRRLRGSEEVIAKRMAQAVAEMSHYAEYDYLIVNDDFDTALTDLKTIIRAERLRMSRQKQRHDALISKLLA 2f4b A 2.07 BS01 EHA A 1 L255 E259 F282 G284 C285 I341 M348 M364 K367 H449 Y473 L49 E53 F76 G78 C79 I135 M142 M158 K161 H243 Y267 ? 0003677,0004879,0005634,0006355 ic50=50nM remove_due_to_license_issue IC50=50nM, EC50=70nM P37231 16451087 201 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2f4j A 1.91 BS01 VX6 A 1 G249 Y253 V256 A269 T315 E316 F317 M318 T319 G321 L370 D381 G23 Y27 V30 A43 T89 E90 F91 M92 T93 G95 L144 D155 D363 A365 R367 N368 D381 P402 D137 A139 R141 N142 D155 P176 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=420nM, Kd=9.4nM, Ki=42nM P00519 16424036 514 GMSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAPAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELGKQ 2f4v B 3.8 BS01 rna A 0 P26 R96 L98 G99 G100 T103 N104 R111 K133 I172 R175 K179 P20 R90 L92 G93 G94 T97 N98 R105 K127 I166 R169 K173 ? 0003735,0005840,0006412,0015935,0019843,0022627,1990904 remove_due_to_license_issue P80371 16492561 5 ~ 1534 VKELLEAGVHFGHERKRWNPKFARYIYAERNGIHIIDLQKTMEELERTFRFIEDLAMRGGTILFVGTKKQAQDIVRMEAERAGMPYVNQRWLGGMLTNFKTISQRVHRLEELEALFASPEIEERPKKEQVRLKHELERLQKYLSGFRLLKRLPDAIFVVDPTKEAIAVREARKLFIPVIALADTDSDPDLVDYIIPGNDDAIRSIQLILSRAVDLIIQARGGVVEPSPSYALVQEAE 2f4v C 3.8 BS01 rna A 0 G2 N3 K4 I5 R127 S154 R156 E161 A163 R172 H176 T177 L178 R179 T192 Y193 G194 V195 G197 K199 G1 N2 K3 I4 R126 S153 R155 E160 A162 R171 H175 T176 L177 R178 T191 Y192 G193 V194 G196 K198 ? 0003676,0003723,0003729,0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P80372 16492561 5 ~ 1534 GNKIHPIGFRLGITRDWESRWYAGKKQYRHLLLEDQRIRGLLEKELYSAGLARVDIERAADNVAVTVHVAKPGVVIGRGGERIRVLREELAKLTGKNVALNVQEVQNPNLSAPLVAQRVAEQIERRFAVRRAIKQAVQRVMESGAKGAKVIVSGRIGGAEQARTEWAAQGRVPLHTLRANIDYGFALARTTYGVLGVKAYIFLGEV 2f4v D 3.8 BS01 rna A 0 G2 R3 V8 C9 R10 R13 R14 K22 R25 K30 R35 R36 Y38 P40 G41 Q42 H43 K46 S52 Y54 Q62 R66 E72 R73 Q74 K84 S113 R115 Q116 R118 Q119 R122 H123 H125 D134 L135 S137 L155 E205 S208 G1 R2 V7 C8 R9 R12 R13 K21 R24 K29 R34 R35 Y37 P39 G40 Q41 H42 K45 S51 Y53 Q61 R65 E71 R72 Q73 K83 S112 R114 Q115 R117 Q118 R121 H122 H124 D133 L134 S136 L154 E204 S207 ? 0003723,0003735,0005840,0006412,0015935,0019843,0042274,0046872,1990904 remove_due_to_license_issue P80373 16492561 5 ~ 1534 GRYIGPVCRLCRREGVKLYLKGERCYSPKCAMERRPYPPGQHGQKRARRPSDYAVRLREKQKLRRIYGISERQFRNLFEEASKKKGVTGSVFLGLLESRLDNVVYRLGFAVSRRQARQLVRHGHITVNGRRVDLPSYRVRPGDEIAVAEKSRNLELIRQNLEAMKGRKVGPWLSLDVEGMKGKFLRLPDREDLALPVQENLVIEFYSR 2f4v E 3.8 BS01 rna A 0 R14 T16 A17 R18 M19 Q20 A21 G22 R24 R25 K47 Y61 K92 A94 A95 T98 I101 A102 G103 R107 T120 K121 E122 L123 S125 R126 N127 N130 R10 T12 A13 R14 M15 Q16 A17 G18 R20 R21 K43 Y57 K88 A90 A91 T94 I97 A98 G99 R103 T116 K117 E118 L119 S121 R122 N123 N126 ? 0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHQ5 16492561 5 ~ 1534 DFEEKMILIRRTARMQAGGRRFRFGALVVVGDRQGRVGLGFGKAPEVPLAVQKAGYYARRNMVEVPLQNGTIPHEIEVEFGASKIVLKPAAPGTGVIAGAVPRAILELAGVTDILTKELGSRNPINIAYATMEALRQLRTKADVERLRKG 2f4v F 3.8 BS01 rna A 0 R2 Y4 Y50 E69 N73 R87 V91 K92 R2 Y4 Y50 E69 N73 R87 V91 K92 ? 0003735,0005737,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLP8 16492561 5 ~ 1534 MRRYEVNIVLNPNLDQSQLALEKEIIQRALENYGARVEKVEELGLRRLAYPIAKDPQGYFLWYQVEMPEDRVNDLARELRIRDNVRRVMVVKSQEPFLANA 2f4v G 3.8 BS01 rna A 0 A2 R3 R4 R6 R10 L12 K29 I30 M31 R32 D33 L38 R41 I42 R94 R95 S98 R102 N109 R114 A116 R119 A1 R2 R3 R5 R9 L11 K28 I29 M30 R31 D32 L37 R40 I41 R93 R94 S97 R101 N108 R113 A115 R118 ? 0000049,0003723,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P17291 16492561 5 ~ 1534 ARRRRAEVRQLQPDLVYGDVLVTAFINKIMRDGKKNLAARIFYDACKIIQEKTGQEPLKVFKQAVENVKPRMEVRSRRVGGANYQVPMEVSPRRQQSLALRWLVQAANQRPERRAAVRIAHELMDAAEGKGGAVKKKEDVERMAEANRAYAHYRW 2f4v H 3.8 BS01 rna A 0 M1 T3 D8 T11 R12 R14 N15 S29 R30 K56 R75 K88 P89 G90 R92 Y94 G96 S113 T114 S115 G130 E132 M1 T3 D8 T11 R12 R14 N15 S29 R30 K56 R75 K88 P89 G90 R92 Y94 G96 S113 T114 S115 G130 E132 ? 0003735,0005737,0005840,0006412,0019843,1990904 remove_due_to_license_issue P0DOY9 16492561 5 ~ 1534 MLTDPIADMLTRIRNATRVYKESTDVPASRFKEEILRILAREGFIKGYERVDVDGKPYLRVYLKYGPRRQGPDPRPEQVIHHIRRISKPGRRVYVGVKEIPRVRRGLGIAILSTSKGVLTDREARKLGVGGELICEVW 2f4v I 3.8 BS01 rna A 0 Q3 Y5 T7 R9 R10 K11 E12 V14 R16 F18 R20 Y36 Q38 G39 Y62 G67 G68 G69 K70 S71 Q73 R83 R93 K97 T103 R104 R107 V108 R111 K112 K113 Y114 K118 R120 R121 A122 Q124 Y125 S126 K127 R128 Q2 Y4 T6 R8 R9 K10 E11 V13 R15 F17 R19 Y35 Q37 G38 Y61 G66 G67 G68 K69 S70 Q72 R82 R92 K96 T102 R103 R106 V107 R110 K111 K112 Y113 K117 R119 R120 A121 Q123 Y124 S125 K126 R127 ? 0000049,0003723,0003735,0005737,0005840,0006412,0019843,0022627,0043232,1990904 remove_due_to_license_issue P80374 16492561 5 ~ 1534 EQYYGTGRRKEAVARVFLRPGNGKVTVNGQDFNEYFQGLVRAVAALEPLRAVDALGRFDAYITVRGGGKSGQIDAIKLGIARALVQYNPDYRAKLKPLGFLTRDARVVERKKYGKHKARRAPQYSKR 2f4v J 3.8 BS01 rna A 0 R5 H13 D17 S35 G36 P37 I38 P39 L40 P41 T42 R43 R45 T48 R51 F54 K55 H56 K57 R60 H62 H68 D73 R3 H11 D15 S33 G34 P35 I36 P37 L38 P39 T40 R41 R43 T46 R49 F52 K53 H54 K55 R58 H60 H66 D71 ? 0000049,0003723,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q5SHN7 16492561 5 ~ 1534 KIRIKLRGFDHKTLDASAQKIVEAARRSGAQVSGPIPLPTRVRRFTVIRGPFKHKDSREHFELRTHNRLVDIINPNRKTIEQLMTLDLPTGVEIEIKT 2f4v K 3.8 BS01 rna A 0 Y20 N26 N27 I29 T31 G37 N38 P39 W42 S44 G46 G52 S53 K55 R85 P115 H116 N117 C119 R120 K122 K123 K124 Y10 N16 N17 I19 T21 G27 N28 P29 W32 S34 G36 G42 S43 K45 R75 P105 H106 N107 C109 R110 K112 K113 K114 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P80376 16492561 5 ~ 1534 KRQVASGRAYIHASYNNTIVTITDPDGNPITWSSGGVIGYKGSRKGTPYAAQLAALDAAKKAMAYGMQSVDVIVRGTGAGREQAIRALQASGLQVKSIVDDTPVPHNGCRPKKKFRKAS 2f4v L 3.8 BS01 rna A 0 P5 T6 N8 Q9 L10 R12 R15 E16 K17 K28 G29 A30 P31 F32 R33 R34 K46 K47 N49 S50 L52 R53 K54 T61 Y69 P71 G72 E73 R86 K91 D92 P94 G95 R97 V104 R113 K114 K115 S116 R117 S118 K119 Y120 G121 T122 K123 K124 P1 T2 N4 Q5 L6 R8 R11 E12 K13 K24 G25 A26 P27 F28 R29 R30 K42 K43 N45 S46 L48 R49 K50 T57 Y65 P67 G68 E69 R82 K87 D88 P90 G91 R93 V100 R109 K110 K111 S112 R113 S114 K115 Y116 G117 T118 K119 K120 ? 0000049,0003735,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHN3 16492561 5 ~ 1534 PTINQLVRKGREKVRKKSKVPALKGAPFRRGVCTVVRTVTPKKPNSALRKVAKVRLTSGYEVTAYIPGEGHNLQEHSVVLIRGGRVKDLPGVRYHIVRGVYDAAGVKDRKKSRSKYGTKKPKEAA 2f4v M 3.8 BS01 rna A 0 K13 R14 Y23 G24 I25 G26 A28 R29 R44 N77 Y87 R91 H92 P97 V98 R99 Q101 R102 T103 R104 T105 N106 A107 R108 T109 R110 K111 R114 K115 T116 V117 R125 K126 K12 R13 Y22 G23 I24 G25 A27 R28 R43 N76 Y86 R90 H91 P96 V97 R98 Q100 R101 T102 R103 T104 N105 A106 R107 T108 R109 K110 R113 K114 T115 V116 R124 K125 ? 0000049,0003676,0003723,0003735,0005829,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue P80377 16492561 5 ~ 1534 ARIAGVEIPRNKRVDVALTYIYGIGKARAKEALEKTGINPATRVKDLTEAEVVRLREYVENTWKLEGELRAEVAANIKRLMDIGCYRGLRHRRGLPVRGQRTRTNARTRKGPRKTVAGKKKAPRK 2f4v N 3.8 BS01 rna A 0 A2 R3 K4 A5 L6 E8 K15 F16 K17 V18 R19 Y21 T22 C27 R29 R31 S32 R35 R41 I42 R45 K58 S60 W61 A1 R2 K3 A4 L5 E7 K14 F15 K16 V17 R18 Y20 T21 C26 R28 R30 S31 R34 R40 I41 R44 K57 S59 W60 ? 0003735,0005737,0005840,0006412,0008270,0015935,0019843,0046872,1990904 remove_due_to_license_issue P0DOY6 16492561 5 ~ 1534 ARKALIEKAKRTPKFKVRAYTRCVRCGRARSVYRFFGLCRICLRELAHKGQLPGVRKASW 2f4v O 3.8 BS01 rna A 0 P2 K8 F18 D21 T22 G23 S24 T25 Q28 R35 L39 H42 H46 K48 D49 H50 H51 S52 R54 L57 R64 R65 Y69 P1 K7 F17 D20 T21 G22 S23 T24 Q27 R34 L38 H41 H45 K47 D48 H49 H50 S51 R53 L56 R63 R64 Y68 ? 0003735,0005737,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue Q5SJ76 16492561 5 ~ 1534 PITKEEKQKVIQEFARFPGDTGSTEVQVALLTLRINRLSEHLKVHKKDHHSHRGLLMMVGQRRRLLRYLQREDPERYRALIEKLGIRG 2f4v P 3.8 BS01 rna A 0 M1 K3 R5 L6 R8 F9 S11 K12 H13 H16 Y17 R18 D23 R25 R26 K27 R28 K31 Y38 P41 R42 K43 W59 V62 G63 Q65 T67 T69 R72 R75 F80 R81 Q82 M1 K3 R5 L6 R8 F9 S11 K12 H13 H16 Y17 R18 D23 R25 R26 K27 R28 K31 Y38 P41 R42 K43 W59 V62 G63 Q65 T67 T69 R72 R75 F80 R81 Q82 ? 0003735,0005737,0005840,0006412,0015935,1990904 remove_due_to_license_issue Q5SJH3 16492561 5 ~ 1534 MVKIRLARFGSKHNPHYRIVVTDARRKRDGKYIEKIGYYDPRKTTPDWLKVDVERARYWLSVGAQPTDTARRLLRQAGVFRQE 2f4v Q 3.8 BS01 rna A 0 P2 K3 K4 S12 K14 M15 Q16 K17 T18 R25 L31 Y32 K34 R38 S39 K40 K41 Y42 E61 S62 R63 P64 I65 S66 K67 R68 K69 R70 K87 N94 Y95 Q96 L98 S99 R101 K104 A105 P1 K2 K3 S11 K13 M14 Q15 K16 T17 R24 L30 Y31 K33 R37 S38 K39 K40 Y41 E60 S61 R62 P63 I64 S65 K66 R67 K68 R69 K86 N93 Y94 Q95 L97 S98 R100 K103 A104 ? 0003735,0005840,0006412,0019843,0022627,1990904 remove_due_to_license_issue P0DOY7 16492561 5 ~ 1534 PKKVLTGVVVSDKMQKTVTVLVERQFPHPLYGKVIKRSKKYLAHDPEEKYKLGDVVEIIESRPISKRKRFRVLRLVESGRMDLVEKYLIRRQNYQSLSKRGGKA 2f4v R 3.8 BS01 rna A 0 K49 I50 P52 K61 R64 K68 K71 R72 R74 I75 F81 K34 I35 P37 K46 R49 K53 K56 R57 R59 I60 F66 ? 0003735,0005840,0006412,0019843,0070181,1990904 remove_due_to_license_issue Q5SLQ0 16492561 5 ~ 1534 PSRKAKVKATLGEFDLRDYRNVEVLKRFLSETGKILPRRRTGLSGKEQRILAKTIKRARILGLLPFTEKLVRK 2f4v S 3.8 BS01 rna A 0 P2 R3 S4 L5 K6 F10 H14 K18 W34 R36 R37 Y52 N53 G54 K55 K70 E73 T77 R78 T79 Y80 H83 P1 R2 S3 L4 K5 F9 H13 K17 W33 R35 R36 Y51 N52 G53 K54 K69 E72 T76 R77 T78 Y79 H82 ? 0000028,0003723,0003735,0005737,0005840,0006412,0015935,0019843,1990904 remove_due_to_license_issue Q5SHP2 16492561 5 ~ 1534 PRSLKKGVFVDDHLLEKVLELNAKGEKRLIKTWSRRSTIVPEMVGHTIAVYNGKQHVPVYITENMVGHKLGEFAPTRTYRGHGK 2f4v T 3.8 BS01 rna A 0 L10 K14 R15 H16 R17 S19 R22 R23 R25 N26 A28 K29 S31 T35 K38 R57 E60 S61 D64 K65 K68 S70 K74 R79 K81 S82 R83 M85 R89 G102 G103 S105 L3 K7 R8 H9 R10 S12 R15 R16 R18 N19 A21 K22 S24 T28 K31 R50 E53 S54 D57 K58 K61 S63 K67 R72 K74 S75 R76 M78 R82 G95 G96 S98 ? 0003723,0003735,0005840,0006412,0015935,0019843,0070181,1990904 remove_due_to_license_issue P80380 16492561 5 ~ 1534 RNLSALKRHRQSLKRRLRNKAKKSAIKTLSKKAVQLAQEGKAEEALKIMRKAESLIDKAAKGSTLHKNAAARRKSRLMRKVRQLLEAAGAPLIGGGLSA 2f6t A 1.7 BS01 1C2 A 1 Y46 D48 V49 D181 F182 C215 S216 A217 I219 G220 R221 Y45 D47 V48 D180 F181 C214 S215 A216 I218 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=24uM remove_due_to_license_issue P18031 16386905 608 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2f6v A 1.7 BS01 SK2 A 1 Y46 D48 V49 D181 F182 C215 S216 A217 I219 G220 R221 M258 G259 Q262 Y45 D47 V48 D180 F181 C214 S215 A216 I218 G219 R220 M257 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=37uM remove_due_to_license_issue P18031 16386905 608 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2f6y A 2.15 BS01 ENT A 1 Y46 D181 F182 C215 S216 A217 I219 G220 R221 Y45 D180 F181 C214 S215 A216 I218 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=134.8uM remove_due_to_license_issue P18031 16386905 608 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2f6z A 1.7 BS01 UN5 A 1 Y20 R24 Y46 D48 V49 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 Y19 R23 Y45 D47 V48 D180 F181 C214 S215 A216 I218 G219 R220 R253 M257 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=4.8uM remove_due_to_license_issue IC50=4800nM P18031 16386905 608 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2f70 A 2.12 BS01 UN6 A 1 R24 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 R23 Y45 D47 D180 F181 C214 S215 A216 I218 G219 R220 R253 M257 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=33.5uM remove_due_to_license_issue P18031 16386905 608 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2f71 A 1.55 BS01 UN7 A 1 R24 Y46 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 R23 Y45 D180 F181 C214 S215 A216 I218 G219 R220 R253 M257 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=2.5uM remove_due_to_license_issue P18031 16386905 608 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2f7o A 1.43 BS02 MSN A 1 H90 D92 W95 D204 D341 H471 D472 Y727 H60 D62 W65 D174 D311 H441 D442 Y697 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=0.036uM remove_due_to_license_issue Ki=36nM Q24451 16787095 5002 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 2f7p A 1.28 BS02 2SK A 1 H90 D92 W95 D204 R228 Y269 D341 H471 D472 Y727 R876 H60 D62 W65 D174 R198 Y239 D311 H441 D442 Y697 R846 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=0.249uM remove_due_to_license_issue Q24451 16787095 5009 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 2f80 A 1.45 BS01 017 B 1 D25 G27 A28 N30 V32 P81 V82 I84 D25 G27 A28 N30 V32 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16480273 301 PQITLWKRPLVTIKIGGQLKEALLDTGADNTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2f80 B 1.45 BS01 017 B 1 D25 G27 A28 D29 N30 G48 G49 I50 D25 G27 A28 D29 N30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=6.6nM remove_due_to_license_issue P04587 16480273 301 PQITLWKRPLVTIKIGGQLKEALLDTGADNTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2f81 A 1.25 BS01 017 A 1 D25 G27 A28 D30 G49 P81 V82 I84 D25 G27 A28 D30 G49 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.03nM remove_due_to_license_issue P04587 16480273 302 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 2f81 B 1.25 BS01 017 A 1 D125 G127 A128 D129 D130 G148 G149 I150 D25 G27 A28 D29 D30 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16480273 302 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 2f89 F 2.6 BS04 210 F 1 D103 R112 K200 D243 K257 D96 R105 K193 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=200nM, Ki=55.9nM P14324 16892359 9001 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 2f8g A 1.22 BS01 017 B 1 D25 G27 A28 D29 G48 G49 V50 D25 G27 A28 D29 G48 G49 V50 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 16480273 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2f8g B 1.22 BS01 017 B 1 D125 G127 A128 D130 G149 V150 P181 I184 D25 G27 A28 D30 G49 V50 P81 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2nM remove_due_to_license_issue P04587 16480273 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2f8i A 1.541 BS01 205 A 1 K15 L17 A108 A109 L110 S117 K6 L8 A99 A100 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 12820260 1002 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 2f8i B 1.541 BS01 205 B 1 K15 L17 A108 A109 L110 S117 K6 L8 A95 A96 L97 S104 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 12820260 1001 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDRYTIAALLSPYSYSTTAVVT 2f8k A 2.0 BS01 rna B 0 K461 R464 L465 H466 K467 A495 L496 G497 R500 K22 R25 L26 H27 K28 A56 L57 G58 R61 ? 0003729,0043488 remove_due_to_license_issue Q08831 16429151 0 ~ 15 SSMNPKSLTDPKLLKNIPMWLKSLRLHKYSDALSGTPWIELIYLDDETLEKKGVLALGARRKLLKAFGIVIDYKERDLIDRSAY 2f94 F 1.94 BS04 BFQ F 1 F99 D103 R112 K200 Q240 D243 K257 F92 D96 R105 K193 Q233 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=20nM, Ki=46nM P14324 16892359 9001 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 2f9b H 2.54 BS01 N1H H 1 H57 C58 K60A S190 C191 K192 S195 V213 S214 W215 G219 H41 C42 K45 S187 C188 K189 S192 V210 S211 W212 G215 3.4.21.21 0004252,0006508 remove_due_to_license_issue Ki=300nM P08709 16460932 258 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2f9k F 2.06 BS04 ZOL F 1 D103 R112 Q171 K200 T201 D243 K257 D96 R105 Q164 K193 T194 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=100nM, Ki=85.9nM P14324 16892359 9001 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 2f9u A 2.6 BS04 5NH A 1 Q41 T42 H57 K136 G137 S139 R155 A156 A157 C159 D168 Q41 T42 H57 K136 G137 S139 R155 A156 A157 C159 D168 H57 D81 G137 S139 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036,0097264 remove_due_to_license_issue Q91RS4 16413182 999 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRSGS 2f9v A 2.6 BS04 BN6 A 1 Q41 T42 H57 I132 L135 K136 G137 S139 R155 A156 A157 C159 Q43 T44 H59 I134 L137 K138 G139 S141 R157 A158 A159 C161 H57 D81 G137 S139 H59 D83 G139 S141 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 16387495 999 MGAPITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2fai A 2.1 BS02 459 A 1 M343 L346 E353 H524 M39 L42 E49 H212 ? Ki=570nM remove_due_to_license_issue P03372 16648639 101 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 2fb8 A 2.9 BS01 215 A 1 I463 G464 V471 A481 K483 T529 C532 F583 D594 I15 G16 V23 A33 K35 T81 C84 F135 D146 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 17145850 102 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 2fda A 2.0 BS01 682 A 1 H57 D189 A190 C191 K192 G193 D194 S195 S214 W215 G216 H44 D182 A183 C184 K185 G186 D187 S188 S207 W208 G209 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 16524727 1 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQA 2fdd A 1.58 BS01 385 B 1 D25 G27 A28 D29 G48 G49 V50 D25 G27 A28 D29 G48 G49 V50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q7SPG9 16458505 501 PQITLWQRPIVTIKIGGQQREALLDTGADDTVLEDINLPGRWKPKIIGGVGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPANIIGRNLMTQIGCTLNF 2fdd B 1.58 BS01 385 B 1 D25 G27 A28 D30 P81 A82 I84 D25 G27 A28 D30 P81 A82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 ic50=4.8nM remove_due_to_license_issue Q7SPG9 16458505 501 PQITLWQRPIVTIKIGGQQREALLDTGADDTVLEDINLPGRWKPKIIGGVGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPANIIGRNLMTQIGCTLNF 2fde A 2.7 BS01 385 A 1 D25 G27 D29 D30 G48 G49 I50 F53 D25 G27 D29 D30 G48 G49 I50 F53 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 16458505 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2fde B 2.7 BS01 385 A 1 D25 G27 A28 D30 P81 D25 G27 A28 D30 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 16458505 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2fdp A 2.5 BS01 FRP A 1 G11 Q12 G13 D32 G34 S35 P70 Y71 T72 Q73 F108 I110 W115 I118 I126 R128 D228 G230 T231 T232 G14 Q15 G16 D35 G37 S38 P73 Y74 T75 Q76 F111 I113 W118 I121 I129 R131 D220 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 Ki=0.026uM remove_due_to_license_issue P56817 16451048 386 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2feq H 2.44 BS03 34P H 1 D189 A190 S195 S214 W215 G216 E217 G219 D192 A193 S198 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=1.39nM remove_due_to_license_issue P00734 16517159 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2fes H 2.42 BS02 3SP H 1 H57 Y60A D189 A190 S195 W215 G216 E217 G219 H43 Y47 D192 A193 S198 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 ic50=0.98nM remove_due_to_license_issue IC50=1nM P00734 16517159 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2ff1 A 2.07 BS02 IMH A 1 N12 D14 D40 W83 M164 E184 N186 W260 D261 N12 D14 D40 W83 M164 E184 N186 W247 D248 D10 D15 D40 W83 T137 W185 N186 W260 D261 D10 D15 D40 W83 T137 W185 N186 W247 D248 3.2.2.1 0005829,0006139,0006152,0008477,0016798,0016799,0046872 Ki=6.2nM remove_due_to_license_issue Q9GPQ4 16630632 401 SAKNVVLDHDGNLDDFVAMVLLASNTEKVRLIGALCTDADCFVENGFNVTGKIMCLMHNNMNLPLFPIGKSAATAVNPFPKEWRCLAKNMDDMPILNIPENVELWDKIKAENEKYEGQQLLADLVMNSEEKVTICVTGPLSNVAWCIDKYGEKFTSKVEECVIMGGAVDVRGNVFLPSTDGTAEWNIYWDPASAKTVFGCPGLRRIMFSLDSTNTVPVRSPYVQRFGEQTNFLLSILVGTMWAMYAWDALTAAYVVDQKVANVDPVPIDVVVDKQPNEGATVRTDAENYPLTFVARNPEAEFFLDMLLRSARAC 2ff2 A 2.2 BS02 IMH A 1 N12 D14 D40 W83 M164 E184 N186 R252 Y257 W260 D261 N11 D13 D39 W82 M163 E183 N185 R251 Y256 W259 D260 D10 D15 D40 W83 T137 W185 N186 W260 D261 D9 D14 D39 W82 T136 W184 N185 W259 D260 3.2.2.1 0005829,0006139,0006152,0008477,0016798,0016799,0046872 Ki=6.2nM remove_due_to_license_issue Q9GPQ4 16630632 501 AKNVVLDHDGNLDDFVAMVLLASNTEKVRLIGALCTDADCFVENGFNVTGKIMCLMHNNMNLPLFPIGKSAATAVNPFPKEWRCLAKNMDDMPILNIPENVELWDKIKAENEKYEGQQLLADLVMNSEEKVTICVTGPLSNVAWCIDKYGEKFTSKVEECVIMGGAVDVRGNVFLPSTDGTAEWNIYWDPASAKTVFGCPGLRRIMFSLDSTNTVPVRSPYVQRFGEQTNFLLSILVGTMWAMCTHCELLRDGDGYYAWDALTAAYVVDQKVANVDPVPIDVVVDKQPNEGATVRTDAENYPLTFVARNPEAEFFLDMLLRSARAC 2fgh A 2.8 BS01 ATP A 1 N368 W369 R370 D371 K503 R542 R629 L630 N334 W335 R336 D337 K469 R508 R595 L596 ? 0003779,0005546,0005615,0005737,0005856,0007417,0008154,0015629,0030030,0030031,0046872,0051014,0051015,0051016,0051693,0060271 remove_due_to_license_issue Q28372 16469333 5380 VEHPEFLKAGKEPGLQIWRVEKFDLVPVPPNLYGDFFTGDAYVILKTVQLRNGILQYDLHYWLGNECSQDESGAAAIFTVQLDDYLNGRAVQHREVQGFESATFLGYFKSGLKYKKGGVASGFKHVVPNEVVVQRLLQVKGRRVVRATEVPVSWESFNNGDCFILDLGNNIYQWCGSKSNRFERLKATQVSKGIRDNERSGRAQVSVFEEGAEPEAMLQVLGPKPTLPEATENRKLAKLYKVSNGAGPMVVSLVADENPFAQGALRSEDCFILDHGKDGKIFVWKGKQANMEERKAALKTASDFISKMDYPKQTQVSVLPEGGETPLFRQFFKNWRDPDQTEGLGLAYLSSHIAHVERVPFDAATLHTSTAMAAQHGMDDDGTGQKQIWRVEGSNKVPVDPATYGQFYGGDSYIILYNYRHGSRQGQIIYNWQGAQSTQDEVAASAILTAQLDEELGGTPVQSRVVQGKEPAHLMSLFGGKPMIVYKGGTSREGGQTAPASTRLFQVRASSSGATRAVEIIPKAGALNSNDAFVLKTPSAAYLWVGAGASEAEKTGAQELLRVLRAQPVQVAEGSEPDSFWEALGGKATYRTSPRLKDKKMDAHPPRLFACSNKIGRFVIEEVPGEFMQEDLATDDVMLLDTWDQVFVWVGKDSQDEEKTEALTSAKRYIDTDPAHRDRRTPITVVKQGFEPPSFVGWFLGWDDSYWSVDPLDRALAELAA 2fgi A 2.5 BS01 PD1 A 1 L484 G485 V492 A512 K514 M535 I545 V561 Y563 A564 S565 G567 L630 A640 D641 L21 G22 V24 A40 K42 M63 I73 V89 Y91 A92 S93 G95 L144 A154 D155 D623 A625 R627 N628 D641 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Ki=36.4nM remove_due_to_license_issue IC50=22nM, EC50=21nM P11362 9774334 1001 ELPEDPRWELPRDRLVLGKPLGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLADIHHIDYYKKTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS 2fgu A 2.0 BS01 ASN A 1 D30 G48 D30 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 505 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPSPVNIIGRNLLTQIGCTLNF 2fgu A 2.0 BS02 HPH A 1 D25 G27 G49 I50 D25 G27 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 506 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPSPVNIIGRNLLTQIGCTLNF 2fgu A 2.0 BS03 DIQ A 1 D25 I84 D25 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 507 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPSPVNIIGRNLLTQIGCTLNF 2fgu B 2.0 BS01 QNC A 1 R8 P81 R8 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 504 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPSPVNIIGRNLLTQIGCTLNF 2fgu B 2.0 BS02 HPH A 1 D25 I84 D25 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 506 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPSPVNIIGRNLLTQIGCTLNF 2fgu B 2.0 BS03 DIQ A 1 G27 I50 G27 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 507 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPSPVNIIGRNLLTQIGCTLNF 2fgv A 1.5 BS01 QNC A 1 D29 G48 D29 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 508 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPNPVNIIGRNLLTQIGCTLNF 2fgv A 1.5 BS02 ASN A 1 A28 D30 G48 A28 D30 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 509 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPNPVNIIGRNLLTQIGCTLNF 2fgv A 1.5 BS03 HPH A 1 D25 G27 G49 I50 D25 G27 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 510 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPNPVNIIGRNLLTQIGCTLNF 2fgv B 1.5 BS01 QNC A 1 R8 P81 R8 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 508 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPNPVNIIGRNLLTQIGCTLNF 2fgv B 1.5 BS02 HPH A 1 D25 I84 D25 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 16809296 510 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPNPVNIIGRNLLTQIGCTLNF 2fhy A 2.95 BS02 A37 A 1 V17 M18 E20 G21 R22 G26 T27 G28 L30 T31 M177 V9 M10 E12 G13 R14 G18 T19 G20 L22 T23 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=3400nM P09467 16442285 502 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKH 2fhy L 2.95 BS03 A37 L 1 V17 M18 E20 G21 R22 G26 T27 G28 L30 T31 M177 V9 M10 E12 G13 R14 G18 T19 G20 L22 T23 M160 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=3400nM P09467 16442285 802 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKH 2fie A 2.81 BS01 A74 A 1 V17 M18 G21 R22 A24 R25 G26 G28 L30 T31 M177 V9 M10 G13 R14 A16 R17 G18 G20 L22 T23 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue P09467 16446092 701 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fie L 2.81 BS01 A74 A 1 G26 S335 G18 S318 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue P09467 16446092 701 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fie L 2.81 BS02 A74 L 1 V17 G21 R22 A24 R25 G26 G28 L30 T31 V9 G13 R14 A16 R17 G18 G20 L22 T23 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue P09467 16446092 1001 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fix A 3.5 BS01 870 A 1 V17 E20 G21 R22 A24 R25 G26 L30 T31 M177 V9 E12 G13 R14 A16 R17 G18 L22 T23 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=570nM P09467 16446092 701 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fix A 3.5 BS02 870 L 1 G26 T27 T31 G18 T19 T23 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=570nM P09467 16446092 1001 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fix L 3.5 BS01 870 A 1 G26 T27 G28 S335 G18 T19 G20 S318 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=570nM P09467 16446092 701 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fix L 3.5 BS02 870 L 1 V17 G21 A24 R25 G26 L30 T31 M177 V9 G13 A16 R17 G18 L22 T23 M160 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=570nM P09467 16446092 1001 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGSKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2fj0 A 2.7 BS01 TFC A 1 G146 G147 S226 A227 F259 L313 Y424 H471 G111 G112 S191 A192 F224 L278 Y389 H436 G146 G147 N178 S226 A227 V265 T314 F316 E357 H471 G111 G112 N143 S191 A192 V230 T279 F281 E322 H436 3.1.1.- 0052689 remove_due_to_license_issue IC50=22nM Q9GPG0 16566578 600 EEVVVRTESGWIRGLKRRAEGNKSYASFRGVPYAKQPLGELRFKELQPLEPWQDELDATQEGPVCQQTDVLYGRIMRPRGMSEACIHANIHVPYYALPRDGLPVLVFIHGGGFAFGSGDSDLHGPEYLVSKDVIVITFNYRLNVYGFLSLNSTSVPGNAGLRDMVTLLKWVQRNAHFFGGRPDDVTLMGQSAGAAATHILSLSKAADGLFRRAILMSGTSSSAFFTTNPVFAQYINKLFVTNIGITATDPEEIHQKLIEMPAEKLNEANRFLLEQFGLTTFFPVVESPINGVTTILDGDPEQLIAKGRGKHIPLIIGFTDAECEIFRRQFEQIDIVSKIKENPGILVPLSVLFSSAPDTVAEITKAMHEKYFKKSVDMEGYIELCTDSYFMYPAISLAIKRARSNGAPVYLYQFSFDGDYSVFREVNHLNFEGAGHIEDLTYVFRTNSMLGGHASFPPHDKDDHMKYWMTSFITNFMKYSNPVTDAKLWPEVRADNLRYQDIDTPDVYQNVKPHSEQRDMLDFFDSIYNW 2fjm A 2.1 BS01 073 A 1 Y546 R547 D548 V549 F682 C715 S716 A717 I719 G720 R721 M758 Q762 Y50 R51 D52 V53 F182 C215 S216 A217 I219 G220 R221 M258 Q262 D681 C715 R721 S722 Q762 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=142nM remove_due_to_license_issue IC50=39nM P18031 16407290 800 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 2fjm A 2.1 BS02 073 B 1 A518 H525 E526 A22 H29 E30 D681 C715 R721 S722 Q762 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=142nM remove_due_to_license_issue IC50=39nM P18031 16407290 801 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 2fjn A 2.2 BS01 073 A 1 Y546 R547 D548 V549 L619 F682 C715 S716 A717 I719 G720 R721 Q762 Y50 R51 D52 V53 L123 F186 C219 S220 A221 I223 G224 R225 Q266 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=39nM remove_due_to_license_issue IC50=39nM P18031 16407290 401 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 2fjn A 2.2 BS02 073 B 1 A518 D522 H525 E526 A22 D26 H29 E30 D681 C715 R721 S722 Q762 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 ic50=39nM remove_due_to_license_issue IC50=39nM P18031 16407290 402 KLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 2fjp A 2.4 BS01 S14 A 1 R125 E205 E206 F357 R358 Y631 Y662 Y666 N710 V711 R87 E167 E168 F319 R320 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=4.3nM remove_due_to_license_issue IC50=4nM, Ki=4.3nM P27487 16759103 1001 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2fkf A 2.0 BS01 G16 A 1 R15 H109 S327 R421 S423 N424 T425 R7 H101 S319 R413 S415 N416 T417 R20 S108 H109 K118 D242 D244 D246 R247 H329 D340 R12 S100 H101 K110 D234 D236 D238 R239 H321 D332 5.4.2.2,5.4.2.8 0000287,0004614,0004615,0005975,0009103,0009243,0009244,0009298,0016853,0016868,0042121,0046872 Kd=1.2mM remove_due_to_license_issue P26276 16595672 465 LPASIFRAYDIRGVVGDTLTAETAYWIGRAIGSESLARGEPCVAVGRDGRLSGPELVKQLIQGLVDCGCQVSDVGMVPTPVLYYAANVLEGKSGVMLTGSHNPPDYNGFKIVVAGETLANEQIQALRERIEKNDLASGVGSVEQVDILPRYFKQIRDDIAMAKPMKVVVDCGNGVAGVIAPQLIEALGCSVIPLYCEVDGNFPNHHPDPGKPENLKDLIAKVKAENADLGLAFDGDGDRVGVVTNTGTIIYPDRLLMLFAKDVVSRNPGADIIFDVKCTRRLIALISGYGGRPVMWKTGHSLIKKKMKETGALLAGEMSGHVFFKERWFGFDDGIYSAARLLEILSQDQRDSEHVFSAFPSDISTPEINITVTEDSKFAIIEALQRDAQWGEGNITTLDGVRVDYPKGWGLVRASNTTPVLVLRFEADTEEELERIKTVFRNQLKAVDSSLPVPF 2fky A 2.3 BS02 N2T A 1 E116 E118 R119 W127 A133 I136 P137 L160 Y211 L214 G217 R221 F239 E99 E101 R102 W110 A116 I119 P120 L143 Y194 L197 G200 R204 F222 ? 0003777,0005524,0007018,0008017 ic50=2.6nM remove_due_to_license_issue P52732 16439123 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2fl2 A 2.5 BS02 N4T A 1 E116 E118 R119 A133 I136 P137 L160 Y211 L214 E215 G217 F239 E99 E101 R102 A116 I119 P120 L143 Y194 L197 E198 G200 F222 ? 0003777,0005524,0007018,0008017 ic50=2nM remove_due_to_license_issue IC50=2nM P52732 16439123 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2fl5 H 3.0 BS01 RBF H 1 Y33 N50 R52 E56 F58 Y100A Y33 N50 R52 E57 F59 Y105 remove_due_to_license_issue 16537445 201 EVQLVESGGGLVQPGESLKLSCTASGFSLSNYYMTWVRQAPGKGLEWVTNIRPDETEKFYSDSVKGRFTVSRDNARNSLFNSMSLQRVEDTATYYCARVSDFGDYGPDFWGQGTLVSVTSASTKGPSVFPLAPCSRSTSESTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTKTYTCNVNHKPSNTKVDKKVEP 2fl5 L 3.0 BS01 RBF H 1 G95 Y95A G94 Y95 ? remove_due_to_license_issue Q5FWF9 16537445 201 SYELKQPPSVSVSPGQTARITCSGDVLPKKYAYWYQERSGQAPVLVVYEDSGRPSEIPERFSGSSSGTKATLTISGAQVEDEADYYCYSDISNGYPLFGGGTKLSVGQPKAAPSVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADSSPIKAGVETTTPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAPT 2fl6 A 2.5 BS02 N5T A 1 E116 E118 R119 A133 I136 P137 L160 R221 F239 E99 E101 R102 A116 I119 P120 L143 R204 F222 ? 0003777,0005524,0007018,0008017 ic50=38nM remove_due_to_license_issue P52732 16439123 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2flb H 1.95 BS01 6NH H 1 C42 H57 D189 S190 C191 K192 S195 V213 W215 G216 C26 H41 D186 S187 C188 K189 S192 V210 W212 G213 3.4.21.21 0004252,0006508 remove_due_to_license_issue P08709 16487703 1246 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2fle A 1.9 BS01 AI B 1 R8 L23 D25 G27 A28 D29 G48 G49 I50 P81 I84 R8 L23 D25 G27 A28 D29 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q9J2R0 18215016 845 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGKWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 2fle B 1.9 BS01 AI B 1 R8 D25 G27 A28 D29 G48 G49 I50 P81 I84 R8 D25 G27 A28 D29 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=14nM remove_due_to_license_issue Q9J2R0 18215016 845 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGKWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 2flh A 1.2 BS01 ZEA A 1 L22 F26 E69 T139 Y142 L22 F26 E69 T132 Y135 ? 0004864,0005634,0005737,0006952,0009738,0010331,0010427,0038023,0044373 Kd=106uM remove_due_to_license_issue A0A1S3THR8 16998071 701 MVKEFNTQTELSVRLEALWAVLSKDFITVVPKVLPHIVKDVQLIEGDGGVGTILIFNFLPEVSPSYQREEITEFDESSHEIGLQVIEGGYLSQGLSYYKTTFKLSEIEEDKTLVNVKISYDHVTPTKTSQSTLMYLRRLERYLS 2flh A 1.2 BS02 ZEA A 2 L34 F58 V62 Q67 G89 Y90 Q93 L34 F58 V62 Q67 G89 Y90 Q93 ? 0004864,0005634,0005737,0006952,0009738,0010331,0010427,0038023,0044373 Kd=106uM remove_due_to_license_issue A0A1S3THR8 16998071 702 MVKEFNTQTELSVRLEALWAVLSKDFITVVPKVLPHIVKDVQLIEGDGGVGTILIFNFLPEVSPSYQREEITEFDESSHEIGLQVIEGGYLSQGLSYYKTTFKLSEIEEDKTLVNVKISYDHVTPTKTSQSTLMYLRRLERYLS 2flh A 1.2 BS03 ZEA A 3 K24 I27 L43 D47 G48 K24 I27 L43 D47 G48 ? 0004864,0005634,0005737,0006952,0009738,0010331,0010427,0038023,0044373 Kd=106uM remove_due_to_license_issue A0A1S3THR8 16998071 708 MVKEFNTQTELSVRLEALWAVLSKDFITVVPKVLPHIVKDVQLIEGDGGVGTILIFNFLPEVSPSYQREEITEFDESSHEIGLQVIEGGYLSQGLSYYKTTFKLSEIEEDKTLVNVKISYDHVTPTKTSQSTLMYLRRLERYLS 2flr H 2.35 BS01 7NH H 1 C42 H57 C58 D60 K60A C191 K192 S195 V213 S214 W215 C26 H41 C42 D44 K45 C188 K189 S192 V210 S211 W212 3.4.21.21 0004252,0006508 Ki=0.8uM remove_due_to_license_issue Ki=800nM P08709 16621549 258 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2fm0 A 2.0 BS02 M98 A 1 M273 N321 Y329 W332 T333 I336 M357 Q369 F372 M195 N243 Y251 W254 T255 I258 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=0.4nM remove_due_to_license_issue IC50=0.4nM Q08499 16539372 601 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 2fm2 A 2.7 BS04 3BC A 1 Q41 T42 H57 I132 K136 G137 S139 F154 R155 A156 A157 D168 Q41 T42 H57 I132 K136 G137 S139 F154 R155 A156 A157 D168 H57 D81 G137 S139 H57 D81 G137 S139 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue Q9ELS8 16352601 900 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2fm5 A 2.03 BS02 M99 A 1 M273 D318 N321 Y329 W332 T333 I336 M357 Q369 F372 M195 D240 N243 Y251 W254 T255 I258 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=43nM remove_due_to_license_issue IC50=43nM Q08499 16539372 601 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 2fmb A 1.8 BS01 LP1 A 1 D25 G27 A28 D29 G54 P86 D25 G27 A28 D29 G54 P86 3.4.23.16 0004190,0006508 Ki=2nM remove_due_to_license_issue Q66729 9827997 201 VTYNLEKRPTTIVLINDTPLNVLLDTGADTSVLTTAHYNRLKYRGRKYQGTGIGGVGGNVETFSTPVTIKKKGRHIKTRMLVADIPVTILGRDILQDLGAKLVL 2fme A 2.1 BS01 3QC A 1 E116 E118 R119 W127 D130 A133 I136 P137 Y211 L214 E215 E96 E98 R99 W107 D110 A113 I116 P117 Y191 L194 E195 ? 0003777,0005524,0007018,0008017 ic50=104nM remove_due_to_license_issue IC50=306nM P52732 16458511 370 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKVKIGKLNLVDLAGSENIGRINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2fou A 0.99 BS03 B22 A 1 H94 H119 F131 L198 T199 T200 P202 H94 H119 F130 L197 T198 T199 P201 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=80nM remove_due_to_license_issue P00918 16506782 301 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2fou A 0.99 BS04 B22 A 2 H4 W5 N11 W16 D19 H4 W5 N11 W16 D19 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=80nM remove_due_to_license_issue P00918 16506782 303 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2fov A 1.15 BS03 B30 A 1 H64 H94 H119 F131 L198 T199 T200 H63 H93 H118 F129 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=28nM remove_due_to_license_issue P00918 16506782 301 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2fov A 1.15 BS04 B30 A 2 H4 H15 W16 D19 H3 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=28nM remove_due_to_license_issue P00918 16506782 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2foy A 1.55 BS02 B30 A 1 H67 H94 L198 T199 H200 H63 H90 L194 T195 H196 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=120nM remove_due_to_license_issue P00915 16506782 311 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2foy A 1.55 BS03 B30 A 2 Y7 P240 M241 Q242 H243 Y3 P236 M237 Q238 H239 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=120nM remove_due_to_license_issue P00915 16506782 313 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2foy A 1.55 BS04 B30 A 3 S99 E102 H103 H243 N245 S95 E98 H99 H239 N241 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=120nM remove_due_to_license_issue P00915 16506782 315 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2fpz A 2.0 BS01 270 A 1 D189 S190 C191 Q192 G216 G219 D188 S189 C190 Q191 G215 G217 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=110uM remove_due_to_license_issue P20231 16681368 1000 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2fq6 A 1.78 BS01 P3F A 1 C85 G86 A87 Y111 P113 D185 A207 T209 K210 M219 Y338 S339 W340 R372 C81 G82 A83 Y107 P109 D181 A203 T205 K206 M215 Y334 S335 W336 R368 R58 Y111 D185 K210 R54 Y107 D181 K206 4.4.1.13,4.4.1.28 0003824,0005737,0006520,0008784,0009086,0016829,0019346,0019450,0030170,0032991,0042802,0047804,0051289,0080146 remove_due_to_license_issue P06721 17300162 700 KLDTQLVNAGRSKKYTLGAVNSVIQRASSLVFDSVEAKKHATRNRANGELFYGRRGTLTHFSLQQAMCELEGGAGCVLFPCGAAAVANSILAFIEQGDHVLMTNTAYEPSQDFCSKILSKLGVTTSWFDPLIGADIVKHLQPNTKIVFLESPGSITMEVHDVPAIVAAVRSVVPDAIIMIDNTWAAGVLFKALDFGIDVSIQAATKYLVGHSDAMIGTAVCNARCWEQLRENAYLMGQMVDADTAYITSRGLRTLGVRLRQHHESSLKVAEWLAEHPQVARVNHPALPGSKGHEFWKRDFTGSSGLFSFVLKKKLNNEELANYLDNFSLFSMAYSWGGYESLILANQPEHIAAIRPQGEIDFSGTLIRLHIGLEDVDDLIADLDAGFARIV 2fqo A 1.87 BS02 HYI A 1 H54 E57 H58 A61 D78 I79 C126 G127 H51 E54 H55 A58 D75 I76 C123 G124 4.4.1.21 0005506,0009372,0016829,0043768,0046872 Ki=0.37uM remove_due_to_license_issue Ki=370nM O34667 16686542 703 VESFELDHNAVVAPYVRHCGVHKVGTDGVVNKFDIRFCQPNKQAMKPDTIHTLEHLLAFTIRSHAEKYDHFDIIDISPMGCQTGYYLVVSGEPTSAEIVDLLEDTMKEAVEITEIPAANEKQCGQAKLHDLEGAKRLMRFWLSQDKEELLKVFG 2fqt A 1.79 BS02 H1D A 1 H54 E57 H58 A61 D78 I79 C126 G127 H51 E54 H55 A58 D75 I76 C123 G124 4.4.1.21 0005506,0009372,0016829,0043768,0046872 Ki=0.72uM remove_due_to_license_issue Ki=720nM O34667 16686542 4398 VESFELDHNAVVAPYVRHCGVHKVGTDGVVNKFDIRFCQPNKQAMKPDTIHTLEHLLAFTIRSHAEKYDHFDIIDISPMGCQTGYYLVVSGEPTSAEIVDLLEDTMKEAVEITEIPAANEKQCGQAKLHDLEGAKRLMRFWLSQDKEELLKVFG 2fqw A 1.71 BS01 NOS A 1 D27 F36 D108 M158 F186 V210 G212 D238 K260 D10 F19 D91 M141 F169 V193 G195 D221 K243 ? 0005886 Kd=210nM remove_due_to_license_issue P29724 16418175 400 GDFVVGMVTDSGDIDDKSFNQQVWEGISRFAQENNAKCKYVTASTDAEYVPSLSAFADENMGLVVACGSFLVEAVIETSARFPKQKFLVIDAVVQDRDNVVSAVFGQNEGSFLVGVAAALKAKEAGKSAVGFIVGMELGMMPLFEAGFEAGVKAVDPDIQVVVEVANTFSDPQKGQALAAKLYDSGVNVIFQVAGGTGNGVIKEARDRRLNGQDVWVIGVDRDQYMDGVYDGSKSVVLTSMVKRADVAAERISKMAYDGSFPGGQSIMFGLEDKAVGIPEENPNLSSAVMEKIRSFEEKIVSKEIVVPVRSARMMN 2fqx A 1.7 BS01 GMP A 1 D27 F36 N37 D108 M158 F186 V210 G212 V237 D238 K260 D10 F19 N20 D91 M141 F169 V193 G195 V220 D221 K243 ? 0005886 Kd=71nM remove_due_to_license_issue P29724 16418175 400 GDFVVGMVTDSGDIDDKSFNQQVWEGISRFAQENNAKCKYVTASTDAEYVPSLSAFADENMGLVVACGSFLVEAVIETSARFPKQKFLVIDAVVQDRDNVVSAVFGQNEGSFLVGVAAALKAKEAGKSAVGFIVGMELGMMPLFEAGFEAGVKAVDPDIQVVVEVANTFSDPQKGQALAAKLYDSGVNVIFQVAGGTGNGVIKEARDRRLNGQDVWVIGVDRDQYMDGVYDGSKSVVLTSMVKRADVAAERISKMAYDGSFPGGQSIMFGLEDKAVGIPEENPNLSSAVMEKIRSFEEKIVSKEIVVPVRSARMMN 2fqy A 1.9 BS01 ADN A 1 D27 S28 F36 D108 M158 F186 V210 G212 V237 D238 K260 D10 S11 F19 D91 M141 F169 V193 G195 V220 D221 K243 ? 0005886 Kd=270nM remove_due_to_license_issue P29724 16418175 400 GDFVVGMVTDSGDIDDKSFNQQVWEGISRFAQENNAKCKYVTASTDAEYVPSLSAFADENMGLVVACGSFLVEAVIETSARFPKQKFLVIDAVVQDRDNVVSAVFGQNEGSFLVGVAAALKAKEAGKSAVGFIVGMELGMMPLFEAGFEAGVKAVDPDIQVVVEVANTFSDPQKGQALAAKLYDSGVNVIFQVAGGTGNGVIKEARDRRLNGQDVWVIGVDRDQYMDGVYDGSKSVVLTSMVKRADVAAERISKMAYDGSFPGGQSIMFGLEDKAVGIPEENPNLSSAVMEKIRSFEEKIVSKEIVVPVRSARMMN 2fr3 A 1.48 BS01 REA A 1 A32 L121 R132 Y134 A32 L121 R132 Y134 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 Kd=2nM remove_due_to_license_issue P29373 16979656 300 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKTSTTVRTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTRELTNDGELILTMTADDVVCTRVYVRE 2fr4 A 1.95 BS01 dna M 0 Y32 Y49 N50 H91 Y32 Y49 N50 H91 remove_due_to_license_issue 18028946 5 ~ 14 ELQMTQSPASLSASVGETVTITCRASENIYSYLAWYQQKQGKSPQLLVYNAKTLAEGVPSRFSGSGSGTQFSLKINSLQPEDFGSYYCQHHYGTPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 2fr4 B 1.95 BS01 dna M 0 Y97 R98 Y100 Y100A A100B Y101 R102 Y104 Y105 A106 remove_due_to_license_issue 18028946 5 ~ 14 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPGSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 2fr4 B 1.95 BS02 dna N 0 S31 Y53 Y97 R98 S31 Y54 Y101 R102 remove_due_to_license_issue 18028946 5 ~ 14 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPGSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 2fr4 H 1.95 BS01 dna M 0 T30 S31 Y53 Y97 R98 T30 S31 Y54 Y101 R102 remove_due_to_license_issue 18028946 5 ~ 14 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 2fr4 H 1.95 BS02 dna N 0 Y97 R98 Y100 Y100A A100B Y101 R102 Y104 Y105 A106 remove_due_to_license_issue 18028946 5 ~ 14 QVKLLESGPELVKPGASVKMSCKASGYTFTSYVMHWVKQKPGQGLEWIGYINPYNDGTKYNEKFKGKATLTSDKSSSTAYMELSSLTSEDSAVYYCVRGGYRPYYAMDYWGQGTSVTVSSAKTTPPSVYPLAPNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 2fr4 L 1.95 BS01 dna N 0 Y32 Y49 N50 E56 H91 Y92 Y31 Y48 N49 E55 H90 Y91 remove_due_to_license_issue 18028946 5 ~ 14 LQMTQSPASLSASVGETVTITCRASENIYSYLAWYQQKQGKSPQLLVYNAKTLAEGVPSRFSGSGSGTQFSLKINSLQPEDFGSYYCQHHYGTPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 2fs8 A 2.5 BS01 C3A A 1 V35 F41 H57 C58 S190 C191 Q192 G193 S195 V213 S214 W215 V20 F28 H44 C45 S189 C190 Q191 G192 S194 V212 S213 W214 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 remove_due_to_license_issue P20231 16681368 999 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2fs8 D 2.5 BS01 C3A D 1 V35 F41 H57 C58 A63 S190 C191 Q192 G193 S195 S214 W215 C220 V20 F28 H44 C45 A55 S189 C190 Q191 G192 S194 S213 W214 C218 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 remove_due_to_license_issue P20231 16681368 996 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2fs9 A 2.3 BS01 C4A A 1 F41 H57 C58 K60D A63 D189 S190 C191 Q192 G193 S195 V213 S214 F28 H44 C45 K51 A55 D188 S189 C190 Q191 G192 S194 V212 S213 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 remove_due_to_license_issue Ki=3nM P20231 16681368 999 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2fs9 D 2.3 BS01 C4A D 1 F41 H57 C58 K60D D189 S190 Q192 G193 D194 S195 S214 F28 H44 C45 K51 D188 S189 Q191 G192 D193 S194 S213 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 remove_due_to_license_issue Ki=3nM P20231 16681368 996 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2ftd A 2.55 BS01 ILI A 1 Q19 C22 G23 C25 D61 G65 G66 Y67 M68 N161 W184 Q19 C22 G23 C25 D61 G65 G66 Y67 M68 N161 W184 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P61277 16509577 300 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 2fu8 A 1.8 BS03 MCO A 1 Y33 W39 D120 H196 S225 P227 H263 Y10 W16 D87 H159 S186 P188 H224 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=20uM remove_due_to_license_issue P52700 17999929 1410 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 2fum A 2.89 BS01 MIX A 1 L17 A38 V95 G97 A142 N143 M145 L15 A36 V93 G95 A140 N141 M143 D138 K140 A142 N143 D156 T179 D136 K138 A140 N141 D154 T165 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P9WI81 16674948 539 TPSHLSDRYELGEILGFGGMSEVHLARDLRLHRDVAVKVLRADLARDPSFYLRFRREAQNAAALNHPAIVAVYDTGEAETPAGPLPYIVMEYVDGVTLRDIVHTEGPMTPKRAIEVIADACQALNFSHQNGIIHRDVKPANIMISATNAVKVMDFGIARAIADGTAQYLSPEQARGDSVDARSDVYSLGCVLYEVLTGEPPFTGDSPVSVAYQHVREDPIPPSARHEGLSADLDAVVLKALAKNPENRYQTAAEMRADLVRVH 2fv5 A 2.1 BS02 541 A 1 T347 L348 G349 E398 L401 H405 E406 H409 H415 Y433 P437 V440 S441 N447 T132 L133 G134 E183 L186 H190 E191 H194 H200 Y218 P222 V225 S226 N232 3.4.24.86 0004222,0006508,0008237 Ki~0.033nM remove_due_to_license_issue IC50=1nM P78536 16762314 1 ADPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERSNA 2fvc A 2.0 BS01 888 A 1 F193 P197 N316 C366 L384 G410 M414 Y415 Y448 F193 P197 N316 C366 L384 G410 M414 Y415 Y448 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=32nM remove_due_to_license_issue Q99AU2 16451063 901 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 2fvd A 1.85 BS01 LIA A 1 V18 A31 K33 F80 L83 H84 Q85 D86 K89 L134 D145 V18 A31 K33 F68 L71 H72 Q73 D74 K77 L122 D133 D127 K129 Q131 N132 D145 T158 T165 D115 K117 Q119 N120 D133 T144 T151 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.003uM remove_due_to_license_issue Ki=3nM, Kd=0.530000nM P24941 17064073 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2fw3 A 2.5 BS01 BUI A 1 H372 Y486 S488 T499 S590 F602 A613 G622 C623 H341 Y455 S457 T468 S559 F571 A582 G591 C592 Y120 P133 H372 S590 Y89 P102 H341 S559 2.3.1.21 0001676,0001701,0004095,0005739,0005743,0006631,0006635,0008374,0008458,0009437,0015909,0016746,0070542,0120162 remove_due_to_license_issue IC50=380nM P18886 16615901 900 DDYLQHSIVPTMHYQDSLPRLPIPKLEDTMKRYLNAQKPLLDDSQFRRTEALCKNFETGVGKELHAHLLAQDKQNKHTSYISGPWFDMYLTARDSIVLNFNPFMAFNPDPKSEYNDQLTRATNLTVSAVRFLKTLQAGLLEPEVFHLNPSKSDTDAFKRLIRFVPPSLSWYGAYLVNAYPLDMSQYFRLFNSTRIPRPNRDELFTDTKARHLLVLRKGHFYVFDVLDQDGNIVNPLEIQAHLKYILSDSSPVPEFPVAYLTSENRDVWAELRQKLIFDGNEETLKKVDSAVFCLCLDDFPMKDLIHLSHTMLHGDGTNRWFDKSFNLIVAEDGTAAVHFEHSWGDGVAVLRFFNEVFRDSTQTPAITPQSQPAATNSSASVETLSFNLSGALKAGITAAKEKFDTTVKTLSIDSIQFQRGGKEFLKKKQLSPDAVAQLAFQMAFLRQYGQTVATYESCSTAAFKHGRTETIRPASIFTKRCSEAFVRDPSKHSVGELQHMMAECSKYHGQLTKEAAMGQGFDRHLYALRYLATARGLNLPELYLDPAYQQMNHNILSTSTLNSPAVSLGGFAPVVPDGFGIAYAVHDDWIGCNVSSYSGRNAREFLHCVQKCLEDIFDALEGK 2fwy A 2.1 BS01 H64 A 1 N51 A55 M98 L107 F138 W162 N35 A39 M82 L91 F122 W146 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=200nM remove_due_to_license_issue EC50=38.8nM P07900 16884307 1001 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2fwz A 2.1 BS01 H71 A 1 N51 A55 M98 L107 F138 W162 N36 A40 M83 L92 F123 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=50nM remove_due_to_license_issue IC50=51nM, EC50=10.00nM P07900 16884307 1001 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2fx6 A 1.57 BS02 270 A 1 D189 S190 C191 Q192 G216 D171 S172 C173 Q174 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=200uM remove_due_to_license_issue P00760 16681368 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2fxr A 2.5 BS01 C3A A 1 V35 F41 H57 C58 K60D A63 Q98 D189 S190 C191 Q192 G193 D194 S195 W215 V20 F28 H44 C45 K51 A55 Q87 D188 S189 C190 Q191 G192 D193 S194 W214 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 remove_due_to_license_issue P20231 16681368 999 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2fxr D 2.5 BS01 C3A D 1 V35 F41 H57 C58 K60D A63 Q98 S190 C191 Q192 G193 S195 W215 V20 F28 H44 C45 K51 A55 Q87 S189 C190 Q191 G192 S194 W214 H57 D102 Q192 G193 D194 S195 G196 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 remove_due_to_license_issue P20231 16681368 996 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVPK 2fxs A 2.0 BS01 RDA A 1 N37 A41 K44 D79 M84 N92 F124 T171 L173 N36 A40 K43 D78 M83 N91 F123 T170 L172 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.87uM remove_due_to_license_issue P02829 19361515 1001 ASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2fxu A 1.35 BS04 BID A 1 Y133 A135 I136 Y143 Y169 A170 P172 T351 F352 M355 Y123 A125 I126 Y133 Y159 A160 P162 T341 F342 M345 3.6.4.- 0000287,0001725,0003785,0005509,0005515,0005523,0005524,0005737,0005856,0005865,0005884,0010628,0016787,0019904,0030027,0030041,0030175,0030240,0031013,0031432,0031941,0032036,0032432,0042802,0044297,0048306,0048741,0051017,0090131,0098723,0140660 Kd=7nM remove_due_to_license_issue P68135 16551075 402 ETTALVCDNGSGLVKAGFAGDDAPRAVFPSIVGRPRHQGVDSYVGDEAQSKRGILTLKYPIEHGIITNWDDMEKIWHHTFYNELRVAPEEHPTLLTEAPLNPKANREKMTQIMFETFNVPAMYVAIQAVLSLYASGRTTGIVLDSGDGVTHNVPIYEGYALPHAIMRLDLAGRDLTDYLMKILTERGYSFVTTAEREIVRDIKEKLCYVALDFENEMATAASSSSLEKSYELPDGQVITIGNERFRCPETLFQPSFIGMESAGIHETTYNSIMKCDIDIRKDLYANNVMSGGTTMYPGIADRMQKEITALAPSTMKIKIIAPPERKYSVWIGGSILASLSTFQQMWITKQEYDEAGPSIVH 2fxv A 2.05 BS01 5GP A 1 V19 L20 F99 T100 F126 A128 N129 G130 Q131 A132 K156 V19 L20 F99 T100 F126 A128 N129 G130 Q131 A132 K156 2.4.2.22 0000310,0005737,0006166,0016757,0016763,0032265,0043101,0046110 Kd=4.5uM remove_due_to_license_issue P42085 16716072 200 MEALKRKIEEEGVVLSDQVLKVDSFLNHQIDPLLMQRIGDEFASRFAKDGITKIVTIESSGIAPAVMTGLKLGVPVVFARKHKSLTLTDNLLTASVYSFTKQTESQIAVSGTHLSDQDHVLIIDDFLANGQAAHGLVSIVKQAGASIAGIGIVIEKSFQPGRDELVKLGYRVESLARIQSLEEGKVSFVQ 2fxv B 2.05 BS01 5GP B 1 V19 L20 F99 T100 D124 D125 F126 A128 N129 G130 Q131 A132 K156 V19 L20 F99 T100 D124 D125 F126 A128 N129 G130 Q131 A132 K156 2.4.2.22 0000310,0005737,0006166,0016757,0016763,0032265,0043101,0046110 Kd=4.5uM remove_due_to_license_issue P42085 16716072 201 MEALKRKIEEEGVVLSDQVLKVDSFLNHQIDPLLMQRIGDEFASRFAKDGITKIVTIESSGIAPAVMTGLKLGVPVVFARKHKSLTLTDNLLTASVYSFTKQTESQIAVSGTHLSDQDHVLIIDDFLANGQAAHGLVSIVKQAGASIAGIGIVIEKSFQPGRDELVKLGYRVESLARIQSLEEGKVSFVQ 2fyv A 1.9 BS02 W72 A 1 D92 W95 D204 F206 S268 Y269 D340 D341 H471 D472 Y727 R876 D62 W65 D174 F176 S238 Y239 D310 D311 H441 D442 Y697 R846 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=0.3mM remove_due_to_license_issue Q24451 17010621 2000 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHS 2fzc A 2.1 BS01 EOP A 1 S52 R54 T55 R105 R167 T168 P266 L267 S52 R54 T55 R105 R167 T168 P266 L267 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=1900uM remove_due_to_license_issue P0A786 16906764 811 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 2fzg A 2.25 BS01 EOB A 1 S52 R54 T55 R105 H134 R167 T168 R229 P266 L267 S52 R54 T55 R105 H134 R167 T168 R229 P266 L267 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=420uM remove_due_to_license_issue P0A786 16906764 611 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 2fzk A 2.5 BS01 EOZ A 1 T55 H134 Q137 T168 R229 P266 L267 R296 T55 H134 Q137 T168 R229 P266 L267 R296 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 Ki=310uM remove_due_to_license_issue P0A786 16906764 611 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 2fzz A 2.2 BS01 5QC A 1 K96 E97 T98 Y99 E146 F174 D189 A190 C191 Q192 W215 G216 G218 C220 G226 K82 E83 T84 Y85 E135 F162 D179 A180 C181 Q182 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=30pM remove_due_to_license_issue Ki=0.03nM P00742 16730984 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2g00 A 2.1 BS01 4QC A 1 K96 E97 T98 Y99 E146 F174 D189 A190 C191 Q192 V213 W215 G216 G218 C220 K82 E83 T84 Y85 E135 F162 D179 A180 C181 Q182 V203 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.18nM remove_due_to_license_issue Ki=0.18nM P00742 16963264 711 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2g01 A 3.5 BS02 73Q A 1 I32 A53 M108 M111 A113 N114 L168 I23 A44 M99 M102 A104 N105 L159 D151 K153 N156 D169 T188 D142 K144 N147 D160 T179 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=1220nM P45983 16527482 901 FYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 2g0g A 2.54 BS01 SP0 A 1 F282 C285 Q286 S289 F363 M364 K367 H449 F76 C79 Q80 S83 F157 M158 K161 H243 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=512nM, EC50=1750nM P37231 16640330 101 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2g0h A 2.3 BS01 SP3 A 1 F282 C285 Q286 R288 S289 L330 V339 F360 F363 M364 K367 H449 L453 Y473 F76 C79 Q80 R82 S83 L124 V133 F154 F157 M158 K161 H243 L247 Y267 ? 0003677,0004879,0005634,0006355 ic50=22.7nM remove_due_to_license_issue IC50=23nM, EC50=0.78nM P37231 16640330 101 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2g19 A 1.7 BS02 4HG A 1 D254 M299 Y303 Y310 H313 Y329 H374 V376 R383 D67 M112 Y116 Y123 H126 Y142 H187 V189 R196 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=1400nM Q9GZT9 16782814 801 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKY 2g1q A 2.51 BS02 N9H A 1 E116 G117 E118 R119 W127 A133 I136 P137 L160 L214 G217 F239 E99 G100 E101 R102 W110 A116 I119 P120 L143 L197 G200 F222 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue P52732 16603356 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2g1r A 2.42 BS01 3IG A 1 T13 Q14 Y15 V31 D33 G35 Y78 T80 A117 V122 D221 G223 T11 Q12 Y13 V29 D31 G33 Y76 T78 A115 V120 D219 G221 D33 S36 N38 W40 Y78 D221 A224 D31 S34 N36 W38 Y76 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=20nM P00797 16480874 885 SSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2g1y A 2.5 BS01 5IG A 1 T13 Q14 Y15 V31 D33 G35 Y78 T80 A117 V122 D221 G223 T11 Q12 Y13 V29 D31 G33 Y76 T78 A115 V120 D219 G221 D33 S36 N38 W40 Y78 D221 A224 D31 S34 N36 W38 Y76 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=90nM P00797 16480874 885 SSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2g24 A 1.9 BS01 7IG A 1 V31 D33 Y78 T80 P113 F114 L116 F119 V122 D219 G221 V29 D31 Y76 T78 P111 F112 L114 F117 V120 D215 G217 D33 S36 N38 W40 Y78 D219 A222 D31 S34 N36 W38 Y76 D215 A218 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=4000nM P00797 16480874 334 SSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSELGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2g2r H 2.75 BS01 TNS L 1 Y33 N35 Y95 V101 W103 Y33 N35 Y99 V106 W108 ? 0002250,0003823,0005576,0016064,0019814 remove_due_to_license_issue P84751 17089439 1006 QVQLQQSGPVLVKPGTSLKMSCKASGYTFTAYYMNWMKQSHGKRLEWIAVINPYNGFTTYNQKFKGKATLTVDKSSNTAYMDLNSLTSEDSAVYYCVPYDYAADRVYWGHGTLVTVSTAKTTAPSVYPLAPVCGGTTGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPALLQSGLYTLSSSVTVTSNTWPSQTITCNVAHPASSTKVDKKIEPRG 2g2r L 2.75 BS01 TNS L 1 L89 F94 L94 F99 remove_due_to_license_issue 17089439 1006 DVVMTQTPLTLSVTIGQPASISCRSSQSLLYINGKTHLNWLLQRPGQSPKRLIYLVSKLDSGVPDRFSGSGSGTDFTLKISRVEAEDLGIYFCLQSTHFPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPRDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 2g4b A 2.5 BS01 rna B 0 R150 Y152 K195 N196 F199 K225 R227 P229 H230 D231 R6 Y8 K51 N52 F55 K81 R83 P85 H86 D87 ? 0003676,0003723 remove_due_to_license_issue P26368 16818232 1 ~ 7 LGSARRLYVGNIPFGITEEAMMDFFNAQMRLGGLTQAPGNPVLAVQINQDKNFAFLEFRSVDETTQAMAFDGIIFQGQSLKIRRPHDYQPLPGAHKLFIGGLPNYLNDDQVKELLTSFGPLKAFNLVKDSATGLSKGYAFCEYVDINVTDQAIAGLNGMQLGDKKLLVQRAS 2g5p A 2.4 BS01 ADF A 1 E205 E206 S209 F357 Y547 S630 Y631 Y662 Y666 E167 E168 S171 F319 Y509 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue Ki=3.8nM P27487 16759095 800 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2g5t A 2.3 BS01 ACF A 1 R125 H126 E205 E206 Y547 S630 Y631 Y662 Y666 R87 H88 E167 E168 Y509 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue Ki=0.820000nM P27487 16759095 800 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2g5u A 1.8 BS01 PCQ A 1 K15 A108 L110 S117 K6 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.2nM remove_due_to_license_issue P02766 15610856 240 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 2g5u B 1.8 BS01 PCQ B 1 K15 A108 K6 A96 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.2nM remove_due_to_license_issue P02766 15610856 239 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSRYTIAALLSPYSYSTTAVVTN 2g63 B 2.0 BS01 AAF B 1 R125 E205 E206 Y547 S630 Y631 Y662 Y666 R87 E167 E168 Y509 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue Ki=6.7nM P27487 16759095 800 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2g6p A 1.9 BS03 HM2 A 1 Y195 C203 H212 Y300 H310 W353 Y106 C114 H123 Y211 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=0.6uM remove_due_to_license_issue EC50=190nM, IC50=860nM P53582 16724298 410 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 2g70 A 2.4 BS02 HNT A 1 Y35 N39 Y40 V53 F182 E219 Y222 M258 Y16 N20 Y21 V34 F163 E200 Y203 M239 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=17nM remove_due_to_license_issue Ki=17nM P11086 17845018 5001 QAAVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2g70 A 2.4 BS03 HNT A 2 V250 R251 L253 V231 R232 L234 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=17nM remove_due_to_license_issue Ki=17nM P11086 17845018 5003 QAAVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2g71 A 2.2 BS02 FTS A 1 Y35 N39 Y40 R44 V53 G54 K57 Y126 F182 E219 Y222 Y15 N19 Y20 R24 V33 G34 K37 Y106 F162 E199 Y202 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=35nM remove_due_to_license_issue Ki=220nM P11086 17845018 3001 AAVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKVG 2g72 A 2.0 BS02 F21 A 1 Y35 N39 Y40 R44 V53 F182 E219 Y222 M258 Y19 N23 Y24 R28 V37 F166 E203 Y206 M242 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=315nM remove_due_to_license_issue Ki=1200nM P11086 17845018 4001 APGQAAVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2g78 A 1.7 BS01 REA A 1 F15 A32 T54 V58 L121 M123 K132 F15 A32 T54 V58 L121 M123 K132 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 remove_due_to_license_issue P29373 17447762 200 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKTSTTVRTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTRELTNDGELILTMTADDVVCTKVFVRE 2g79 A 1.69 BS01 RET A 1 F15 L28 A32 P39 L121 M123 K132 F15 L28 A32 P39 L121 M123 K132 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 Kd=120nM remove_due_to_license_issue P29373 17447762 200 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKTSTTVRTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTRELTNDGELILTMTADDVVCTKVFVRE 2g83 A 2.8 BS04 GDP A 1 E43 G45 K46 S47 T48 R176 T177 R178 K270 D272 L273 C325 A326 E11 G13 K14 S15 T16 R134 T135 R136 K228 D230 L231 C283 A284 E43 T48 R178 D200 Q204 E11 T16 R136 D158 Q162 ? 0003924,0005525,0007165,0007186,0007188,0019001,0031683 remove_due_to_license_issue P63096 16981699 355 EVKLLLLGAGESGKSTIVKQMKIIHEAGYSEEECKQYKAVVYSNTIQSIIAIIRAMGRLKIDFGDSARADDARQLFVLAELAGVIKRLWKDSGVQACFNRSREYQLNDSAAYYLNDLDRIAQPNYIPTQQDVLRTRVKTTGIVETHFTFKDLHFKMFDVGGQRSERKKWIHCFEGVTAIIFCVALSDYDLVLAEDEEMNRMHESMKLFDSICNNKWFTDTSIILFLNKKDLFEEKIKKSPLTICYPEYAGSNTYEEAAAYIQCQFEDLNKRKDTKEIYTHFTCATDTKNVQFVFDAVTDVIIK 2g8n A 2.15 BS01 F83 A 1 Y35 N39 Y40 R44 V53 G54 L58 Y126 F182 E219 Y222 Y13 N17 Y18 R22 V31 G32 L36 Y104 F160 E197 Y200 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=0.063uM remove_due_to_license_issue Ki=63nM P11086 16942016 2001 VASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2g94 A 1.86 BS01 ZPQ A 1 G13 D32 G34 P70 Y71 T72 Q73 Y198 D228 G230 T231 T232 R235 G17 D36 G38 P74 Y75 T76 Q77 Y202 D232 G234 T235 T236 R239 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=0.3nM remove_due_to_license_issue Ki=0.300000nM P56817 16620080 1001 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2g96 A 2.9 BS01 NMN A 1 F193 R196 D219 R311 D313 G353 G383 G384 F173 R176 D199 R291 D293 G333 G363 G364 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 16901503 1001 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 2g96 A 2.9 BS02 NMN B 1 Y18 R392 Y10 R372 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 16901503 1002 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 2g96 B 2.9 BS01 NMN A 1 D16 Y18 R392 D8 Y10 R372 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 16901503 1001 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 2g96 B 2.9 BS02 NMN B 1 F193 R196 D219 R311 D313 G353 G383 G384 F173 R176 D199 R291 D293 G333 G363 G364 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 16901503 1002 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 2g97 A 2.9 BS01 DGB A 1 H191 F193 D219 V242 A244 I309 R311 R349 E376 S379 H171 F173 D199 V222 A224 I289 R291 R329 E356 S359 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 16901503 1001 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 2g97 B 2.9 BS01 DGB B 1 F193 R196 D219 V242 A244 S275 R311 R349 E376 S379 F173 R176 D199 V222 A224 S255 R291 R329 E356 S359 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 16901503 1002 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 2g9q A 2.5 BS03 1AB A 1 H377 N484 E672 A673 S674 G675 H345 N452 E640 A641 S642 G643 H377 K568 R569 K574 T676 K680 H345 K536 R537 K542 T644 K648 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=0.84uM remove_due_to_license_issue Ki=400nM P00489 16970395 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFGYIQAVLDRNLAENISRVLYPFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2g9r A 2.07 BS01 G27 A 1 H377 N484 H571 E672 S674 G675 H351 N458 H545 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=0.84uM remove_due_to_license_issue IC50=840nM P00489 16970395 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2g9u A 2.15 BS02 G27 A 1 H377 N484 R569 H571 E672 S674 G675 H344 N451 R536 H538 E639 S641 G642 H377 K568 R569 K574 T676 K680 H344 K535 R536 K541 T643 K647 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=0.84uM remove_due_to_license_issue IC50=840nM P00489 16970395 998 SVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2g9v A 2.15 BS02 IFM A 1 H377 N484 E672 S674 G675 H348 N455 E643 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=5.2uM remove_due_to_license_issue IC50=1210nM, Ki=5200nM P00489 16970395 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2g9x A 2.5 BS01 NU5 A 1 I10 E12 G13 A31 F80 E81 L83 H84 Q85 D86 K89 L134 I11 E13 G14 A32 F81 E82 L84 H85 Q86 D87 K90 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=45nM remove_due_to_license_issue P24941 16669651 299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2ga2 A 1.95 BS03 A19 A 1 H231 L328 N329 H331 I338 H339 E364 F366 Y444 H122 L219 N220 H222 I229 H230 E255 F257 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 ic50=3uM remove_due_to_license_issue IC50=9100nM P50579 16632353 482 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 2gbf A 3.1 BS01 AIA A 1 E203 E204 Y548 S631 Y632 Y663 Y667 E166 E167 Y511 S594 Y595 Y626 Y630 Y548 S631 Y632 D709 H741 Y511 S594 Y595 D672 H704 3.4.14.5 0001618,0001662,0001666,0002020,0002337,0002709,0002717,0004177,0004252,0005102,0005518,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0030163,0031258,0031295,0033632,0035641,0036343,0042110,0042277,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P14740 16768443 768 RRTYTLADYLKNTFRVKSYSLRWVSDSEYLYKQENNILLFNAEHGNSSIFLENSTFEIFGDSISDYSVSPDRLFVLLEYNYVKQWRHSYTASYSIYDLNKRQLITEEKIPNNTQWITWSQEGHKLAYVWKNDIYVKIEPHLPSHRITSTGKENVIFNGINDWVYEEEIFGAYSALWWSPNGTFLAYAQFNDTGVPLIEYSFYSDESLQYPKTVWIPYPKAGAVNPTVKFFIVNTDSLSSTTTTIPMQITAPASVTTGDHYLCDVAWVSEDRISLQWLRRIQNYSVMAICDYDKTTLVWNCPTTQEHIETSATGWCGRFRPAEPHFTSDGSSFYKIVSDKDGYKHICQFQKDRKPEQVCTFITKGAWEVISIEALTSDYLYYISNEYKEMPGGRNLYKIQLTDHTNKKCLSCDLNPERCQYYSVSLSKEAKYYQLGCRGPGLPLYTLHRSTDQKELRVLEDNSALDKMLQDVQMPSKKLDFIVLNETRFWYQMILPPHFDKSKKYPLLIDVYAGPCSQKADAAFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINKRLGTLEVEDQIEAARQFLKMGFVDSKRVAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDAGVDFQAMWYTDEDHGIASSTAHQHIYSHMSHFLQQCFSLR 2gbg A 3.0 BS01 1AD A 1 E203 E204 F355 Y548 S631 Y632 Y663 Y667 E166 E167 F318 Y511 S594 Y595 Y626 Y630 Y548 S631 Y632 D709 H741 Y511 S594 Y595 D672 H704 3.4.14.5 0001618,0001662,0001666,0002020,0002337,0002709,0002717,0004177,0004252,0005102,0005518,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0030163,0031258,0031295,0033632,0035641,0036343,0042110,0042277,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P14740 16768443 768 RRTYTLADYLKNTFRVKSYSLRWVSDSEYLYKQENNILLFNAEHGNSSIFLENSTFEIFGDSISDYSVSPDRLFVLLEYNYVKQWRHSYTASYSIYDLNKRQLITEEKIPNNTQWITWSQEGHKLAYVWKNDIYVKIEPHLPSHRITSTGKENVIFNGINDWVYEEEIFGAYSALWWSPNGTFLAYAQFNDTGVPLIEYSFYSDESLQYPKTVWIPYPKAGAVNPTVKFFIVNTDSLSSTTTTIPMQITAPASVTTGDHYLCDVAWVSEDRISLQWLRRIQNYSVMAICDYDKTTLVWNCPTTQEHIETSATGWCGRFRPAEPHFTSDGSSFYKIVSDKDGYKHICQFQKDRKPEQVCTFITKGAWEVISIEALTSDYLYYISNEYKEMPGGRNLYKIQLTDHTNKKCLSCDLNPERCQYYSVSLSKEAKYYQLGCRGPGLPLYTLHRSTDQKELRVLEDNSALDKMLQDVQMPSKKLDFIVLNETRFWYQMILPPHFDKSKKYPLLIDVYAGPCSQKADAAFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINKRLGTLEVEDQIEAARQFLKMGFVDSKRVAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDAGVDFQAMWYTDEDHGIASSTAHQHIYSHMSHFLQQCFSLR 2gbi A 3.3 BS01 XIH A 1 R123 E203 E204 Y548 S631 Y632 Y663 V712 R86 E166 E167 Y511 S594 Y595 Y626 V675 Y548 S631 Y632 D709 H741 Y511 S594 Y595 D672 H704 3.4.14.5 0001618,0001662,0001666,0002020,0002337,0002709,0002717,0004177,0004252,0005102,0005518,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0030163,0031258,0031295,0033632,0035641,0036343,0042110,0042277,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue Ki=3nM P14740 16768443 901 RRTYTLADYLKNTFRVKSYSLRWVSDSEYLYKQENNILLFNAEHGNSSIFLENSTFEIFGDSISDYSVSPDRLFVLLEYNYVKQWRHSYTASYSIYDLNKRQLITEEKIPNNTQWITWSQEGHKLAYVWKNDIYVKIEPHLPSHRITSTGKENVIFNGINDWVYEEEIFGAYSALWWSPNGTFLAYAQFNDTGVPLIEYSFYSDESLQYPKTVWIPYPKAGAVNPTVKFFIVNTDSLSSTTTTIPMQITAPASVTTGDHYLCDVAWVSEDRISLQWLRRIQNYSVMAICDYDKTTLVWNCPTTQEHIETSATGWCGRFRPAEPHFTSDGSSFYKIVSDKDGYKHICQFQKDRKPEQVCTFITKGAWEVISIEALTSDYLYYISNEYKEMPGGRNLYKIQLTDHTNKKCLSCDLNPERCQYYSVSLSKEAKYYQLGCRGPGLPLYTLHRSTDQKELRVLEDNSALDKMLQDVQMPSKKLDFIVLNETRFWYQMILPPHFDKSKKYPLLIDVYAGPCSQKADAAFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINKRLGTLEVEDQIEAARQFLKMGFVDSKRVAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDAGVDFQAMWYTDEDHGIASSTAHQHIYSHMSHFLQQCFSLR 2gc8 A 2.2 BS01 885 A 1 R200 C366 L384 M414 Y415 Q446 Y448 G449 R200 C366 L384 M414 Y415 Q446 Y448 G449 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=3.1uM remove_due_to_license_issue Q99AU2 16722622 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPDLSGWFVAGYSGGDIYH 2gcd A 2.55 BS01 STU A 1 I34 V42 A55 M105 Y107 C108 L109 G110 G155 L158 D169 K314 I23 V31 A44 M94 Y96 C97 L98 G99 G144 L147 D158 K303 D151 K153 G155 N156 D169 P178 T185 D140 K142 G144 N145 D158 P167 T174 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9JLS3 16761096 400 DPDVAELFFKDDPEKLFSDLREIGHGSFGAVYFARDVRNSEVVAIKKMSYSGKQSNEKWQDIIKEVRFLQKLRHPNTIQYRGCYLREHTAWLVMEYCLGSASDLLEVHKKPLQEVEIAAVTHGALQGLAYLHSHNMIHRDVKAGNILLSEPGLVKLGDFGSASIMAPANSFVGTPYWMAPEVILAMDEGQYDGKVDVWSLGITCIELAERKPPLFNMNAMSALYHIAQNESPALQSGHWSEYFRNFVDSCLQKIPQDRPTSEVLLKHRFVLRERPPTVIMDLIQRTKDAVRELDNLQYRKMKKILFQEA 2gd8 A 1.46 BS02 PO1 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=379nM remove_due_to_license_issue IC50=379nM, Ki=270nM, Kd=3750nM P00918 17181151 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2gd8 A 1.46 BS03 PO1 A 2 N62 N67 I91 Q92 D130 F131 G132 N59 N64 I88 Q89 D126 F127 G128 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=379nM remove_due_to_license_issue IC50=379nM, Ki=270nM, Kd=3750nM P00918 17181151 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2gde H 2.0 BS03 SN3 H 1 Y60A W60D I174 D189 A190 C191 S195 W215 G216 E217 G219 R221A Y47 W50 I172 D192 A193 C194 S198 W220 G221 E222 G223 R226 3.4.21.5 0004252,0005509,0006508,0007596 ic50=5.7nM remove_due_to_license_issue P00734 16895415 401 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 2gdo A 3.0 BS01 12C A 1 L15 G16 E17 G18 A36 L84 E85 Y86 C87 G90 E91 E134 L137 D148 L15 G16 E17 G18 A36 L80 E81 Y82 C83 G86 E87 E130 L133 D144 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=0.320000nM O14757 16603354 298 MAVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 2ge5 A 2.4 BS01 dna C 0 T37 N70 D90 K92 T93 T94 Y95 G109 T111 S112 K119 G182 S183 T186 T36 N69 D89 K91 T92 T93 Y94 G108 T110 S111 K118 G181 S182 T185 3.1.21.4 0003677,0004519 remove_due_to_license_issue P04390 16981705 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKENEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVATRKSSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYE 2ge5 A 2.4 BS02 dna D 0 Q69 N70 L180 S183 G184 N185 Q68 N69 L179 S182 G183 N184 3.1.21.4 0003677,0004519 remove_due_to_license_issue P04390 16981705 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKENEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVATRKSSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYE 2ge5 B 2.4 BS01 dna C 0 Q69 N70 S183 G184 N185 Q68 N69 S182 G183 N184 3.1.21.4 0003677,0004519 remove_due_to_license_issue P04390 16981705 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKENEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVATRKSSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYE 2ge5 B 2.4 BS02 dna D 0 T37 N70 D90 K92 T93 T94 Y95 T106 G109 K119 N120 S183 T186 N188 T36 N69 D89 K91 T92 T93 Y94 T105 G108 K118 N119 S182 T185 N187 3.1.21.4 0003677,0004519 remove_due_to_license_issue P04390 16981705 1 ~ 11 SLRSDLINALYDENQKYDVCGIISAEGKIYPLGSDTKVLSTIFELFSRPIINKIAEKHGYIVEEPKQQNHYPDFTLYKPSEPNKKIAIDIKTTYTNKENEKIKFTLGGYTSFIRNNTKNIVYPFDQYIAHWIIGYVYTRVATRKSSLKTYNINELNEIPKPYKGVKVFLQDKWVIAGDLAGSGNTTNIGSIHAHYKDFVEGKGIFDSEDEFLDYWRNYE 2gej A 2.6 BS01 GDD A 1 P14 G15 G16 L194 R196 K202 Q250 V251 D252 D253 K256 E274 S275 F276 I278 E282 P14 G15 G16 L182 R184 K190 Q238 V239 D240 D241 K244 E262 S263 F264 I266 E270 2.4.1.345 0004377,0005886,0008654,0009247,0016757,0043750,0046488 remove_due_to_license_issue A0QWG6 17510062 2567 MRIGMVCPYSFDVPGGVQSHVLQLAEVLRDAGHEVSVLAPASPHVKLPDYVVSGGKAVFGPATHRKVKKWIAEGDFDVLHIHEPNAPSLSMLALQAAEGPIVATFHTSTTKSLTLSVFQGILRPYHEKIIGRIAVSDLARRWQMEALGSDAVEIPNGVDVASFADAPLLDGYPREGRTVLFLGRYDEPRKGMAVLLAALPKLVARFPDVEILIVGRGDEDELREQAGDLAGHLRFLGQVDDATKASAMRSADVYCAPHLGGESFGIVLVEAMAAGTAVVASDLDAFRRVLADGDAGRLVPVDDADGMAAALIGILEDDQLRAGYVARASERVHRYDWSVVSAQIMRVYETVSGAGIKVQVS 2gek A 2.4 BS01 GDP A 1 P14 G15 G16 L194 K202 Q250 V251 D252 D253 K256 V279 E282 P14 G15 G16 L182 K190 Q238 V239 D240 D241 K244 V267 E270 2.4.1.345 0004377,0005886,0008654,0009247,0016757,0043750,0046488 remove_due_to_license_issue A0QWG6 17510062 2567 MRIGMVCPYSFDVPGGVQSHVLQLAEVLRDAGHEVSVLAPASPHVKLPDYVVSGGKAVFGPATHRKVKKWIAEGDFDVLHIHEPNAPSLSMLALQAAEGPIVATFHTSTTKSLTLSVFQGILRPYHEKIIGRIAVSDLARRWQMEALGSDAVEIPNGVDVASFADAPLLDGYPREGRTVLFLGRYDEPRKGMAVLLAALPKLVARFPDVEILIVGRGDEDELREQAGDLAGHLRFLGQVDDATKASAMRSADVYCAPHLGGESFGIVLVEAMAAGTAVVASDLDAFRRVLADGDAGRLVPVDDADGMAAALIGILEDDQLRAGYVARASERVHRYDWSVVSAQIMRVYETVSGAGIKVQVS 2gfd A 2.3 BS01 RDA A 1 N107 A111 D149 M154 N162 V197 F199 I247 N34 A38 D76 M81 N89 V116 F118 I166 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.52uM remove_due_to_license_issue P41148 19361515 1001 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIKGTSEFLNKMTESTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 2gfj A 1.8 BS03 VI A 1 W39 H118 D120 I162 H196 S225 H263 W16 H85 D87 I127 H159 S186 H224 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=150uM remove_due_to_license_issue P52700 17999929 1410 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 2gfk A 1.9 BS03 VII A 1 W39 D120 F156 I162 H196 S225 W16 D87 F123 I127 H159 S186 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=30uM remove_due_to_license_issue P52700 17999929 1410 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 2gfs A 1.752 BS01 PQB A 1 Y35 K53 L104 T106 H107 L108 M109 G110 A111 Y31 K49 L100 T102 H103 L104 M105 G106 A107 D150 K152 N155 D168 T185 D146 K148 N151 D164 T177 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.7uM remove_due_to_license_issue IC50=400nM Q16539 16509574 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2gg0 A 1.28 BS03 U11 A 1 Y62 H79 D97 D108 Y168 H171 F177 H178 E204 E235 Y60 H77 D95 D106 Y166 H169 F175 H176 E202 E233 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H77 D95 D106 H169 R173 H176 Q180 E202 N206 Q231 E233 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=1.7uM remove_due_to_license_issue IC50=1700nM P0AE18 17120228 601 ISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg2 A 1.0 BS03 U12 A 1 Y62 Y65 H79 D97 D108 H171 F177 H178 E204 W221 E235 Y61 Y64 H78 D96 D107 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.25uM remove_due_to_license_issue IC50=250nM P0AE18 17120228 801 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg3 A 1.45 BS03 U13 A 1 Y62 H63 H79 D97 D108 H171 F177 H178 E204 W221 E235 Y61 H62 H78 D96 D107 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.58uM remove_due_to_license_issue IC50=580nM P0AE18 17120228 501 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg5 A 2.12 BS03 U19 A 1 Y62 Y65 D97 H171 F177 H178 E204 W221 Y61 Y64 D96 H170 F176 H177 E203 W220 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.25uM remove_due_to_license_issue IC50=250nM P0AE18 17120228 501 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg7 A 1.12 BS03 U14 A 1 C59 Y62 H63 Y65 H79 D97 D108 H171 F177 H178 E204 W221 C58 Y61 H62 Y64 H78 D96 D107 H170 F176 H177 E203 W220 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=1.75uM remove_due_to_license_issue IC50=1750nM P0AE18 17120228 701 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg8 A 1.8 BS03 U15 A 1 Y62 C70 H79 D97 D108 Y168 H171 F177 H178 E204 W221 E235 Y61 C69 H78 D96 D107 Y167 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=25uM remove_due_to_license_issue P0AE18 17120228 501 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg9 A 1.05 BS03 U16 A 1 Y62 Y65 C70 H79 D97 D108 Y168 H171 F177 H178 E204 W221 E235 Y61 Y64 C69 H78 D96 D107 Y167 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=3.5uM remove_due_to_license_issue IC50=3500nM P0AE18 17120228 801 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gga A 1.7 BS02 GPJ A 1 K28 A99 A100 T101 R128 D326 E354 R357 R405 K23 A94 A95 T96 R123 D321 E349 R352 R400 K28 S29 D55 N98 R128 D326 E354 H404 R405 T431 K23 S24 D50 N93 R123 D321 E349 H399 R400 T426 2.5.1.19 0003824,0003866,0005737,0008652,0009073,0009423,0009635,0016740,0016765 Ki=6mM remove_due_to_license_issue Q9R4E4 16916934 701 SSRPATARKSSGLSGTVRIPGDKSISHRSFMFGGLASGETRITGLLEGEDVINTGKAMQAMGARIRKEGDTWIIDGVGNGGLLAPEAPLDFGNAATGCRLTMGLVGVYDFDSTFIGDASLTKRPMGRVLNPLREMGVQVKSEDGDRLPVTLRGPKTPTPITYRVPMASAQVKSAVLLAGLNTPGITTVIEPIMTRDHTEKMLQGFGANLTVETDADGVRTIRLEGRGKLTGQVIDVPGDPSSTAFPLVAALLVPGSDVTILNVLMNPTRTGLILTLQEMGADIEVINPRLAGGEDVADLRVRSSTLKGVTVPEDRAPSMIDEYPILAVAAAFAEGATVMNGLEELRVKESDRLSAVANGLKLNGVDCDEGETSLVVRGRPDGKGLGNASGAAVATHLDHRIAMSFLVMGLVSENPVTVDDATMIATSFPEFMDLMAGLGAKIELS 2ggb A 2.13 BS03 U17 A 1 Y62 H63 H79 D97 D108 Y168 C169 H171 F177 H178 E204 E235 Y61 H62 H78 D96 D107 Y167 C168 H170 F176 H177 E203 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=12uM remove_due_to_license_issue IC50=12000nM P0AE18 17120228 304 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2ggd A 1.7 BS02 GPJ A 1 K28 G100 T101 R128 Q175 D326 E354 R357 H404 R405 K23 G95 T96 R123 Q170 D321 E349 R352 H399 R400 K28 S29 D55 N98 R128 D326 E354 H404 R405 T431 K23 S24 D50 N93 R123 D321 E349 H399 R400 T426 2.5.1.19 0003824,0003866,0005737,0008652,0009073,0009423,0009635,0016740,0016765 ic50=160uM remove_due_to_license_issue Q9R4E4 16916934 601 SSRPATARKSSGLSGTVRIPGDKSISHRSFMFGGLASGETRITGLLEGEDVINTGKAMQAMGARIRKEGDTWIIDGVGNGGLLAPEAPLDFGNAGTGCRLTMGLVGVYDFDSTFIGDASLTKRPMGRVLNPLREMGVQVKSEDGDRLPVTLRGPKTPTPITYRVPMASAQVKSAVLLAGLNTPGITTVIEPIMTRDHTEKMLQGFGANLTVETDADGVRTIRLEGRGKLTGQVIDVPGDPSSTAFPLVAALLVPGSDVTILNVLMNPTRTGLILTLQEMGADIEVINPRLAGGEDVADLRVRSSTLKGVTVPEDRAPSMIDEYPILAVAAAFAEGATVMNGLEELRVKESDRLSAVANGLKLNGVDCDEGETSLVVRGRPDGKGLGNASGAAVATHLDHRIAMSFLVMGLVSENPVTVDDATMIATSFPEFMDLMAGLGAKIELS 2ggx A 1.9 BS04 NPJ A 1 E321 N323 E329 F335 T336 N337 N341 R343 E117 N119 E125 F131 T132 N133 N137 R139 ? ic50=0.32mM remove_due_to_license_issue P35247 16636058 700 ASLRQQVEALQGQVQHLQAAFSQYKKVELFPNGQSVGEKIFKTAGFVKPFTEAQLLCTQAGGQLASPRSAAENAALQQLVVAKNEAAFLSMTDSKTEGKFTYPTGESLVYSNWAPGEPNDDGGSEDCVEIFTNGKWNDRACGEKRLVVCEF 2gh6 A 2.203 BS02 CF3 A 1 I100 P140 H142 H143 G151 F152 D180 H182 F208 G310 Y312 I99 P139 H141 H142 G150 F151 D179 H181 F207 G309 Y311 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 17401192 9452 AIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADI 2gh7 A 1.0 BS01 BTN A 1 L25 S27 Y43 S45 V47 N49 W79 S88 T90 W108 D128 L12 S14 Y30 S32 V34 N36 W66 S75 T77 W95 D115 ? 0009374 Kd~0.1pM remove_due_to_license_issue Kd=1.000000nM P22629 16699183 5100 EAGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVK 2ghg A 3.5 BS01 A53 A 1 L15 E17 G18 A19 Y20 A36 L84 Y86 C87 G90 L137 S147 D148 L14 E16 G17 A18 Y19 A35 L83 Y85 C86 G89 L136 S146 D147 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=126nM O14757 16644221 1 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2gie A 2.6 BS01 dna E 0 H73 Y77 S90 K93 Q109 Q138 Y199 N201 A204 R241 K248 H72 Y76 S89 K92 Q108 Q137 Y198 N200 A203 R240 K247 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gie A 2.6 BS02 dna F 0 G30 H31 Q109 N110 D114 D127 K129 T130 N132 S136 A137 Q138 P140 N141 S144 Y146 K147 A205 M206 Q207 G29 H30 Q108 N109 D113 D126 K128 T129 N131 S135 A136 Q137 P139 N140 S143 Y145 K146 A204 M205 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gie B 2.6 BS01 dna E 0 G30 H31 Q109 N110 D127 K129 T130 R131 N132 K135 S136 A137 Q138 A139 P140 N141 S144 K147 A205 Q207 G29 H30 Q108 N109 D126 K128 T129 R130 N131 K134 S135 A136 Q137 A138 P139 N140 S143 K146 A204 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gie B 2.6 BS02 dna F 0 Y77 L86 S90 G92 K93 K108 Q109 Q138 Y199 N201 A204 Y76 L85 S89 G91 K92 K107 Q108 Q137 Y198 N200 A203 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gie C 2.6 BS01 dna G 0 Y77 R91 G92 K93 A94 K108 Q109 Q138 Y199 N201 A204 Y76 R90 G91 K92 A93 K107 Q108 Q137 Y198 N200 A203 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gie C 2.6 BS02 dna H 0 G30 H31 Q109 N110 D114 D127 K129 T130 N132 K135 A137 Q138 P140 N141 I143 S144 Y146 K147 A205 Q207 G29 H30 Q108 N109 D113 D126 K128 T129 N131 K134 A136 Q137 P139 N140 I142 S143 Y145 K146 A204 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gie D 2.6 BS01 dna G 0 G30 H31 A33 Q109 N110 D111 D114 T130 N132 K135 S136 A137 Q138 P140 N141 S144 K147 A205 G29 H30 A32 Q108 N109 D110 D113 T129 N131 K134 S135 A136 Q137 P139 N140 S143 K146 A204 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gie D 2.6 BS02 dna H 0 Y77 G92 K93 K108 Q109 Q138 Y199 N201 K248 Y76 G91 K92 K107 Q108 Q137 Y198 N200 K247 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 13 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAQAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gig A 1.83 BS01 dna E 0 H31 G92 K93 K108 Q109 F138 Y199 N201 A203 A204 R241 K248 H23 G84 K85 K100 Q101 F130 Y191 N193 A195 A196 R233 K240 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKRPHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gig A 1.83 BS02 dna F 0 Q109 N110 D111 D114 D127 K129 T130 R131 S136 A137 F138 A139 P140 N141 S144 K147 A205 M206 Q207 Q101 N102 D103 D106 D119 K121 T122 R123 S128 A129 F130 A131 P132 N133 S136 K139 A197 M198 Q199 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKRPHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gig B 1.83 BS01 dna E 0 A137 F138 A139 P140 N141 S144 K147 A205 Q207 A120 F121 A122 P123 N124 S127 K130 A188 Q190 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gig B 1.83 BS02 dna F 0 G92 K93 F138 Y199 N201 A203 A204 R241 K248 G75 K76 F121 Y182 N184 A186 A187 R224 K231 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gih A 2.5 BS01 dna E 0 R91 K93 K108 Q109 F138 Y199 A203 A204 R241 K248 R90 K92 K107 Q108 F137 Y198 A202 A203 R240 K247 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gih A 2.5 BS02 dna F 0 G30 H31 Q109 N110 A137 F138 A139 N141 S144 K147 A205 M206 Q207 G29 H30 Q108 N109 A136 F137 A138 N140 S143 K146 A204 M205 Q206 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKRPKSGTLSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gih B 2.5 BS01 dna E 0 Q109 N110 D127 T130 K135 A137 F138 A139 P140 N141 S144 K147 A205 M206 Q207 Q102 N103 D120 T123 K128 A130 F131 A132 P133 N134 S137 K140 A198 M199 Q200 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKRSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gih B 2.5 BS02 dna F 0 G92 K93 Q109 F138 Y199 N201 A204 R241 K248 G85 K86 Q102 F131 Y192 N194 A197 R234 K241 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKRSGHAAGEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gii A 2.3 BS01 dna E 0 G92 K93 F138 Y199 N201 A203 A204 R241 G76 K77 F122 Y179 N181 A183 A184 R221 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gii A 2.3 BS02 dna F 0 E35 Q109 A137 F138 P140 N141 S144 A205 Q207 E19 Q93 A121 F122 P124 N125 S128 A185 Q187 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gii B 2.3 BS01 dna E 0 Q109 K135 F138 N141 S144 A205 M206 Q87 K113 F116 N119 S122 A176 M177 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWECVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKY 2gii B 2.3 BS02 dna F 0 K93 F138 Y199 N201 A203 A204 R241 K248 K74 F116 Y170 N172 A174 A175 R212 K219 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIEPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWECVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKY 2gij A 1.93 BS01 dna E 0 G92 K93 Q109 F138 Y199 N201 A203 A204 G79 K80 Q96 F125 Y186 N188 A190 A191 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKREPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gij A 1.93 BS02 dna F 0 Q109 N110 D111 D114 D127 V128 K129 T130 R131 N132 S136 A137 F138 A139 P140 N141 S144 K147 A205 Q207 Q96 N97 D98 D101 D114 V115 K116 T117 R118 N119 S123 A124 F125 A126 P127 N128 S131 K134 A192 Q194 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQKVKREPFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWELNGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYIL 2gij B 1.93 BS01 dna E 0 Q109 N110 S136 A137 F138 P140 N141 S144 K147 A205 Q207 Q90 N91 S117 A118 F119 P121 N122 S125 K128 A184 Q186 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWEGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2gij B 1.93 BS02 dna F 0 G92 K93 K108 F138 Y199 N201 A203 A204 R241 K248 G73 K74 K89 F119 Y178 N180 A182 A183 R220 K227 3.1.21.4 0003677,0004519,0009036,0009307 remove_due_to_license_issue P17743 16675462 1 ~ 14 SFIKPIYQDINSILIGQFEKLVYKFLKENLSDLTFKQYEYLNDLFMKNPAIIGHEARYKLFNSPTLLFLLSRGKAATENWSIENLFEEKQNDTADILLVKDQFYELLDVKTRNISKSAFAPNIISAYKLAQTCAKMIDNKEFDLFDINYLEVDWEGEDLVCVSTSFAELFKSEPSELYINWAAAMQIQFHVRDLDQGFNGTREEWAKSYLKHFVTQAEQRAISMIDKFVKPFKKYI 2giu A 2.2 BS01 FBR A 1 L298 E305 I373 I376 F377 L33 E40 I107 I110 F111 ? 0003677,0004879,0006355 ic50=1.5nM remove_due_to_license_issue IC50=1.8nM, EC50=4nM Q92731 16632357 600 LDALSPEQLVLTLLEAEPPHVLISRPASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVADSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMVVPVYDLLLEMLNAHVL 2gj4 A 1.6 BS02 2TH A 1 R60 W67 E190 K191 R49 W56 E179 K180 H377 K568 R569 K574 T676 K680 H345 K536 R537 K542 T644 K648 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=319nM remove_due_to_license_issue P00489 16945526 949 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 2gj5 A 2.4 BS01 VD3 A 1 L39 I56 K60 E62 I71 I84 F105 M107 L38 I55 K59 E61 I70 I83 F104 M106 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=4.74nM remove_due_to_license_issue P02754 18004750 163 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 2gj5 A 2.4 BS02 VD3 A 2 D137 L140 K141 M145 H146 I147 R148 D136 L139 K140 M144 H145 I146 R147 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=4.74nM remove_due_to_license_issue P02754 18004750 164 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 2gje A 3.37 BS01 rna R 0 R67 R92 R96 E114 K117 R3 R28 R32 E50 K53 ? 0003677,0006355 remove_due_to_license_issue Q952G2 16923390 11 ~ 23 RARRAQLPPAFDVVHWNDEDISRGHLLRVLHRDTFVVLDYHRQARMLTEEGNKAERVVSVMLPAVYTARFLAVLEGRSEKVEVHSRYTNATFTPNPAAPYTFTLKCTSTRPDETFEWTVEFDVAESLMLQRFLTQALHYNTGFAR 2gje D 3.37 BS01 rna R 0 Y61 A80 R83 Y35 A54 R57 ? 0003677,0003723,0003729,0005515,0005739,0006355,0010608,0016556,0031019,0031981 remove_due_to_license_issue P90629 16923390 11 ~ 23 QSLPKFEIHDVRDDPAEGTMTRVAVDGKLLLISQYPQLGPRKVDPNDLSPQFDADRRISVRLRHVDLAYLVGVCKERVPRHRMETKAYTLDFEKSAQGYHLHGKVHRVASQRMEDWSVKFDNHFAVTLEHFLESALDESFGFRQHYA 2gkd A -1.00 BS01 dna B 0 G87 R130 N131 G87 R130 N131 ? remove_due_to_license_issue Q8KNF0 17168523 1 ~ 11 NYDPFVRHSVTVKADRKTAFKTFLEGFPEWWPNNFRTTKVGAPLGVDKKGGRWYEIDEQGEEHTFGLIRKVDEPDTLVIGWRLNGFGRIDPDNSSEFTVTFVADGQKKTRVDVEHTHFDRMGTKHAKRVRNGMDKGWPTILQSFQDKIDEEGAKK 2gkd A -1.00 BS02 dna C 0 K124 K127 R128 K124 K127 R128 ? remove_due_to_license_issue Q8KNF0 17168523 12 ~ 22 NYDPFVRHSVTVKADRKTAFKTFLEGFPEWWPNNFRTTKVGAPLGVDKKGGRWYEIDEQGEEHTFGLIRKVDEPDTLVIGWRLNGFGRIDPDNSSEFTVTFVADGQKKTRVDVEHTHFDRMGTKHAKRVRNGMDKGWPTILQSFQDKIDEEGAKK 2gkl A 1.86 BS02 PD2 A 1 V67 W87 D120 H196 C221 K224 N233 H263 V21 W41 D72 H147 C166 K169 N174 H204 N116 H118 D120 H196 C221 K224 N233 H263 N68 H70 D72 H147 C166 K169 N174 H204 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=4.5uM remove_due_to_license_issue P26918 17307979 2 AGMSLTQVSGPVYVVEDNYYVQENSMVYFGAKGVTVVGATWTPDTARELHKLIKRVSRKPVLEVINTNYHTDRAGGNAYWKSIGAKVVSTRQTRDLMKSDWAEIVAFTRKGLPEYPDLPLVLPNVVHDGDFTLQEGKVRAFYAGPAHTPDGIFVYFPDEQVLYGNCILKEKLGNLSFADVKAYPQTLERLKAMKLPIKTVIGGHDSPLHGPELIDHYEALIKAA 2gl0 A 2.25 BS01 ADN C 1 N20 W95 T116 A117 Y165 N16 W91 T112 A113 Y161 2.7.1.20 0000166 Kd=15uM remove_due_to_license_issue Q8ZVF7 16737961 903 SIKFELIDVPIPQGTNVIIGQAHFIKTVEDLYEALVTSVPGVKFGIAFCEASGKRLVRHEANDEELRNLAIDLCKKIAAGHVFVIYIRNAWPINVLNAIKNVPEVVRIFAATANPLKVIVAEVEPERRGVVGVVDGHSPLGVETEKDREERKKFLREVVKYKL 2gl0 B 2.25 BS01 ADN A 1 N20 W95 I97 A117 Y165 N16 W91 I93 A113 Y161 2.7.1.20 0000166 Kd=15uM remove_due_to_license_issue Q8ZVF7 16737961 901 SIKFELIDVPIPQGTNVIIGQAHFIKTVEDLYEALVTSVPGVKFGIAFCEASGKRLVRHEANDEELRNLAIDLCKKIAAGHVFVIYIRNAWPINVLNAIKNVPEVVRIFAATANPLKVIVAEVEPERRGVVGVVDGHSPLGVETEKDREERKKFLREVVKYKL 2gl0 E 2.25 BS01 ADN D 1 N20 W95 A117 Y165 N16 W91 A113 Y161 2.7.1.20 0000166 Kd=15uM remove_due_to_license_issue Q8ZVF7 16737961 904 SIKFELIDVPIPQGTNVIIGQAHFIKTVEDLYEALVTSVPGVKFGIAFCEASGKRLVRHEANDEELRNLAIDLCKKIAAGHVFVIYIRNAWPINVLNAIKNVPEVVRIFAATANPLKVIVAEVEPERRGVVGVVDGHSPLGVETEKDREERKKFLREVVKYKL 2glm A 2.6 BS01 SCB A 1 F59 P60 K62 I64 P112 F52 P53 K55 I57 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue O25928 18093984 3001 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 2glm B 2.6 BS01 SCB A 1 I98 Y100 F101 R158 I90 Y92 F93 R150 H58 I64 G67 V68 E72 H50 I56 G59 V60 E64 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue O25928 18093984 3001 QSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 2glo A -1.00 BS01 dna B 0 R45 N69 Q70 R71 R81 R82 Q85 K86 R3 N27 Q28 R29 R39 R40 Q43 K44 ? remove_due_to_license_issue Q9XTN4 16876822 1 ~ 12 GSRRIFTPHFKLQVLESYRNDNDCKGNQRATARKYNIHRRQIQKWLQCESNLRSSVANN 2glo A -1.00 BS02 dna C 0 S44 R45 F48 K53 H80 R82 Q83 W87 S2 R3 F6 K11 H38 R40 Q41 W45 ? remove_due_to_license_issue Q9XTN4 16876822 13 ~ 24 GSRRIFTPHFKLQVLESYRNDNDCKGNQRATARKYNIHRRQIQKWLQCESNLRSSVANN 2glp C 2.42 BS01 BDE C 1 I20 L21 P22 F83 A94 K97 I98 V99 R158 I12 L13 P14 F75 A86 K89 I90 V91 R150 H58 I64 G67 V68 E72 H50 I56 G59 V60 E64 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 Ki=9.7uM remove_due_to_license_issue IC50=39800nM O25928 18093984 3002 QSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 2glp D 2.42 BS01 BDE C 1 F59 I64 F52 I57 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue IC50=39800nM O25928 18093984 3002 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 2gm1 A 2.3 BS02 2AZ A 1 E116 G117 E118 W127 I136 P137 Y211 L214 E215 R221 E98 G99 E100 W109 I118 P119 Y193 L196 E197 R203 ? 0003777,0005524,0007018,0008017 ic50=0.1uM remove_due_to_license_issue IC50=100nM P52732 16730979 371 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKEVKIGKLNLVDLAGSENIGRINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 2gm9 A 2.3 BS02 3TH A 1 R60 W67 W189 E190 K191 R49 W56 W178 E179 K180 H377 K568 R569 K574 T676 K680 H346 K537 R538 K543 T645 K649 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=41nM remove_due_to_license_issue P00489 16945526 1 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2gmk A 1.65 BS01 AMP A 1 K9 K31 K9 K31 3.1.27.- 0003676,0004519,0004540,0050830 Ki=590uM remove_due_to_license_issue P22069 18001769 940 QDWLTFQKKHITNTRDVDCDNIMSTNLFHCKDKNTFIYSRPEPVKAICKGIIASKNVLTTSEFYLSDCNVTSRPCKYKLKKSTNKFCVNCANQAPVHFVGVGSC 2gmk A 1.65 BS02 AMP A 2 K9 H10 H97 F98 K9 H10 H97 F98 3.1.27.- 0003676,0004519,0004540,0050830 Ki=590uM remove_due_to_license_issue P22069 18001769 941 QDWLTFQKKHITNTRDVDCDNIMSTNLFHCKDKNTFIYSRPEPVKAICKGIIASKNVLTTSEFYLSDCNVTSRPCKYKLKKSTNKFCVNCANQAPVHFVGVGSC 2gmv A 2.3 BS03 UN8 A 1 A287 N292 L293 M296 T343 W516 F517 F525 F530 N533 A278 N283 L284 M287 T334 W499 F500 F508 F513 N516 R87 Y235 K244 H264 S286 C288 D311 R405 R78 Y226 K235 H255 S277 C279 D302 R396 2.7.11.-,4.1.1.32 0000287,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0016301,0016831,0017076,0018105,0019543,0030145,0031406,0032868,0032869,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070062,0070365,0071333,0071549,0072350,0106264 ic50=0.63uM remove_due_to_license_issue IC50=630nM P35558 17532214 703 NLSAKVVQGSLDSLPQAVREFLENNAELCQPDHIHICDGSEEENGRLLGQMEEEGILRRLKKYDNCWLALTDPRDVARIESKTVIVTQEQRDTVPIPKTGLSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLSKIGIELTDSPYVVASMRIMTRMGTPVLEALGDGEFVKCLHSVGCPLPLQKPLVNNWPCNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRMASRLAKEEGWLAEHMLVLGITNPEGEKKYLAAAFPSACGKTNLAMMNPSLPGWKVECVGDDIAWMKFDAQGHLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLASGVTITSWKNKEWSSEDGEPCAHPNSRFCTPASQCPIIDAAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEAKIIMHDPFAMRPFFGYNFGKYLAHWLSMAQHPAAKLPKIFHVNWFRKDKEGKFLWPGFGENSRVLEWMFNRIDGTKLTPIGYIPKEDALNLKGLGHINMMELFSISKEFWDKEVEDIEKYLVDQVNADLPCEIEREILALKQRISQM 2gmx A 3.5 BS02 877 A 1 I32 M108 L110 M111 D112 A113 I25 M101 L103 M104 D105 A106 D151 K153 N156 D169 T188 D144 K146 N149 D162 T181 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=77nM P45983 16759099 901 NNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 2gnf A 2.28 BS02 Y27 A 1 A70 E121 Y122 M123 N171 L173 D184 A61 E112 Y113 M114 N162 L164 D175 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=6uM remove_due_to_license_issue IC50=42000nM P00517 16699172 501 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYMPGGDMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2gnh A 2.05 BS02 H52 A 1 V57 A70 M120 Y122 E170 L173 A183 F327 V48 A61 M111 Y113 E161 L164 A174 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=149nM remove_due_to_license_issue IC50=394nM P00517 16699172 501 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYMPGGDMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2gnh A 2.05 BS03 H52 A 2 E86 K189 T197 E77 K180 T188 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=149nM remove_due_to_license_issue IC50=394nM P00517 16699172 502 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYMPGGDMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2gni A 2.27 BS02 M77 A 1 I49 V57 A70 M120 Y122 M123 D127 E170 L173 A183 F327 I40 V48 A61 M111 Y113 M114 D118 E161 L164 A174 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=2280nM remove_due_to_license_issue IC50=1494nM P00517 16699172 601 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYMPGGDMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2gnj A 2.28 BS02 Y27 A 1 I49 T51 G52 S53 V57 A70 Y122 V123 N171 L173 D184 F327 I36 T38 G39 S40 V44 A57 Y109 V110 N158 L160 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=6uM remove_due_to_license_issue IC50=42000nM P00517 16699172 501 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2gnl A 2.6 BS02 H52 A 1 I49 T51 A70 E170 L173 A183 F327 I39 T41 A60 E160 L163 A173 F317 D166 K168 E170 N171 D184 T201 D156 K158 E160 N161 D174 T191 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue IC50=394nM P00517 16699172 501 EQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2go4 A 2.7 BS04 TUX A 1 H58 E78 H79 T191 E197 I198 L212 V217 H238 D242 H265 H57 E72 H73 T178 E184 I185 L199 V204 H225 D229 H252 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue O67648 16800620 901 GLEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFAFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQ 2gpp A 2.6 BS02 1BA A 1 E247 I249 L268 A272 E275 L309 V313 R316 Y326 D328 F435 E15 I17 L36 A40 E43 L77 V81 R84 Y94 D96 F203 ? remove_due_to_license_issue P62508 16990259 459 PYNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAK 2gqn A 1.8 BS01 BLP A 1 C85 G86 A87 Y111 E112 D185 A207 T209 K210 M219 Y338 S339 W340 R372 C81 G82 A83 Y107 E108 D181 A203 T205 K206 M215 Y334 S335 W336 R368 R58 Y111 D185 K210 R54 Y107 D181 K206 4.4.1.13,4.4.1.28 0003824,0005737,0006520,0008784,0009086,0016829,0019346,0019450,0030170,0032991,0042802,0047804,0051289,0080146 remove_due_to_license_issue P06721 17300162 700 KLDTQLVNAGRSKKYTLGAVNSVIQRASSLVFDSVEAKKHATRNRANGELFYGRRGTLTHFSLQQAMCELEGGAGCVLFPCGAAAVANSILAFIEQGDHVLMTNTAYEPSQDFCSKILSKLGVTTSWFDPLIGADIVKHLQPNTKIVFLESPGSITMEVHDVPAIVAAVRSVVPDAIIMIDNTWAAGVLFKALDFGIDVSIQAATKYLVGHSDAMIGTAVCNARCWEQLRENAYLMGQMVDADTAYITSRGLRTLGVRLRQHHESSLKVAEWLAEHPQVARVNHPALPGSKGHEFWKRDFTGSSGLFSFVLKKKLNNEELANYLDNFSLFSMAYSWGGYESLILANQPEHIAAIRPQGEIDFSGTLIRLHIGLEDVDDLIADLDAGFARIV 2gss A 1.9 BS01 EAA A 1 Y7 F8 R13 I104 Y108 Y6 F7 R12 I103 Y107 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=11.5uM remove_due_to_license_issue IC50=2.6e+4nM P09211 9012673 0 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 2gss B 1.9 BS01 EAA B 1 Y7 F8 R13 I104 Y108 Y6 F7 R12 I103 Y107 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=11.5uM remove_due_to_license_issue IC50=2.6e+4nM P09211 9012673 0 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 2gst A 1.8 BS01 GPS A 1 Y6 W7 V9 G11 L12 R42 W45 K49 N58 L59 Q71 S72 I111 Y115 F208 S209 Y6 W7 V9 G11 L12 R42 W45 K49 N58 L59 Q71 S72 I111 Y115 F208 S209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005496,0005576,0005737,0005829,0006629,0006693,0006749,0007608,0009410,0010038,0010288,0016151,0016740,0018916,0019899,0019901,0032991,0042178,0042802,0042803,0043200,0043295,0045471,0048678,0051122,0070458,0071466,1901687 Ki=0.85uM remove_due_to_license_issue P04905 8110735 220 PMILGYWNVRGLTHPIRLLLEYTDSSYEEKRYAMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGSRKITQSNAIMRYLARKHHLCGETEEERIRADIVENQVMDNRMQLIMLCYNPDFEKQKPEFLKTIPEKMKLYSEFLGKRPWFAGDKVTYVDFLAYDILDQYHIFEPKCLDAFPNLKDFLARFEGLKKISAYMKSSRYLSTPIFSKLAQWSNK 2gst B 1.8 BS01 GPS B 1 Y6 W7 V9 G11 L12 W45 K49 N58 L59 Q71 S72 I111 F208 Y6 W7 V9 G11 L12 W45 K49 N58 L59 Q71 S72 I111 F208 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005496,0005576,0005737,0005829,0006629,0006693,0006749,0007608,0009410,0010038,0010288,0016151,0016740,0018916,0019899,0019901,0032991,0042178,0042802,0042803,0043200,0043295,0045471,0048678,0051122,0070458,0071466,1901687 Ki=0.85uM remove_due_to_license_issue P04905 8110735 218 PMILGYWNVRGLTHPIRLLLEYTDSSYEEKRYAMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGSRKITQSNAIMRYLARKHHLCGETEEERIRADIVENQVMDNRMQLIMLCYNPDFEKQKPEFLKTIPEKMKLYSEFLGKRPWFAGDKVTYVDFLAYDILDQYHIFEPKCLDAFPNLKDFLARFEGLKKISAYMKSSRYLSTPIFSKLAQWSNK 2gsu A 2.0 BS03 AMP A 1 T90 F91 L123 Y174 Y205 D210 E211 H363 T47 F48 L80 Y131 Y162 D167 E168 H320 Ki=268uM remove_due_to_license_issue 16893180 1004 TPHALLLISIDGLRADMLDRGITPNLSHLAREGVRARWMAPSYPSLTFPNHYTLVTGLRPDHHGIVHNSMRDPTLGGFWLSKSEAVGDARWWGGEPVWVGVENTGQHAATWSWPGSEAAIKGVRPSQWRHYQKGVRLDTRVDAVRGWLATDGAQRNRLVTLYFEHVDEAGHDHGPESRQYADAVRAVDAAIGRLLAGMQRDGTRARTNIIVVSDHGMAEVAPGHAISVEDIAPPQIATAITDGQVIGFEPLPGQQAAAEASVLGAHDHYDCWRKAELPARWQYGSHPRIPSLVCQMHEGWDALFPDKLAKRAQRGTRGSHGYDPALPSMRAVFLAQGPDLAQGKTLPGFDNVDVYALMSRLLGIPAAPNDGNPATLLPALRM 2gtk A 2.1 BS02 208 A 1 I281 F282 C285 R288 S289 H323 L330 M364 H449 L469 Y473 I62 F63 C66 R69 S70 H104 L111 M145 H230 L250 Y254 ? 0003677,0004879,0005634,0006355 ic50=0.251uM remove_due_to_license_issue EC50=760nM, IC50=251nM P37231 16737814 1001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2gtv X -1.00 BS01 TSA X 1 R9 R34 V41 K45 D54 R57 E58 N90 Q94 R9 R34 V41 K45 D54 R57 E58 N90 Q94 5.4.99.5 0046417 remove_due_to_license_issue Q57696 17994104 501 MIEKLAEIRKKIDEIDNKILKARWPWAEKLIAERNSLAKDVAEIKNQLGIPINDPEREKYIYDRIRKLCKEHNVDENIGIKIFQRLIEHNKALQKQYLEETLEH 2gu8 A 2.2 BS02 796 A 1 L49 G50 T51 G52 G55 R56 A70 K72 E121 Y122 V123 N171 L173 T183 D184 F327 L36 G37 T38 G39 G42 R43 A57 K59 E108 Y109 V110 N158 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM P17612 16765046 1001 SVKEFLAKAKEDFLKKWETPSQNTAQLDQFDRIKTLGTGSFGRVMLVKHKESGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDEQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 2gv6 A 2.1 BS01 730 A 1 F99 D189 S190 C191 Q192 S195 W215 G216 G219 C220 F94 D185 S186 C187 Q188 S191 W212 G213 G215 C216 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 Ki=0.046uM remove_due_to_license_issue Q9Y5Y6 16821772 1 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 2gv7 A 2.2 BS01 672 A 1 H57 I60 Y60G F99 D189 S190 C191 Q192 S195 V213 S214 W215 G216 G219 C220 H42 I45 Y52 F94 D185 S186 C187 Q188 S191 V210 S211 W212 G213 G215 C216 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 Ki=0.014uM remove_due_to_license_issue Ki=14nM Q9Y5Y6 16821772 245 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 2gvd A 2.9 BS04 128 A 1 I397 G399 F400 A409 L412 G439 D440 R484 I22 G24 F25 A34 L37 G64 D65 R109 D396 I397 D440 H516 D21 I22 D65 H141 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P30803 16766715 584 DMMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 2gvd B 2.9 BS02 128 A 1 F889 N1022 N1025 S1028 K1065 F11 N134 N137 S140 K177 S891 I892 S942 R1029 K1065 S13 I14 S64 R141 K177 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P26769 16766715 584 HQSYDCVCVMFASIPDFKEFYTESDVNKEGLECLRLLNEIIADFDDLLSKPKFSGVEKIKTIGSTYMAATGLSAIRQYMHIGTMVEFAYALVGKLDAINKHSFNDFKLRVGINHGPVIAGVIGAQKPQYDIWGNTVNVASRMDSTGVLDKIQVTEETSLILQTLGYTCTCRGIINVKGKGDLKTYFVNT 2gvf A 2.5 BS04 NHN A 1 Q41 T42 H57 I132 K136 G137 S139 R155 A156 A157 C159 D168 Q43 T44 H59 I134 K138 G139 S141 R157 A158 A159 C161 D170 H57 D81 G137 S139 H59 D83 G139 S141 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P26664 16730985 999 MGAPITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2gvj A 2.1 BS01 DGB A 1 K189 H191 F193 R196 D219 V242 A244 S275 R311 R349 E376 N377 I378 A379 K169 H171 F173 R176 D199 V222 A224 S255 R291 R329 E356 N357 I358 A359 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Ki=0.3nM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 16783377 502 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIE 2gvj B 2.1 BS01 DGB B 1 F193 R196 D219 V242 A244 S275 R311 R349 E376 I378 A379 F173 R176 D199 V222 A224 S255 R291 R329 E356 I358 A359 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Ki=0.3nM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 16783377 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 2gvv A 1.73 BS03 DI9 A 1 E21 P36 N120 N175 D229 W244 E19 P34 N118 N173 D227 W242 E21 E37 N120 N175 D229 H287 E19 E35 N118 N173 D227 H285 3.8.2.2 0005509,0016787,0046872,0047862 Kd=400uM remove_due_to_license_issue Q7SIG4 17002369 502 IPVIEPLFTKVTEDIPGAEGPVFDKNGDFYIVAPEVEVNGKPAGEILRIDLKTGKKTVICKPEVNGYGGIPAGCQCDRDANQLFVADMRLGLLVVQTDGTFEEIAKKDSEGRRMQGCNDCAFDYEGNLWITAPAGEVAPADYTRSMQEKFGSIYCFTTDGQMIQVDTAFQFPNGIAVRHMNDGRPYQLIVAETPTKKLWSYDIKGPAKIENKKVWGHIPGTHEGGADGMDFDEDNNLLVANWGSSHIEVFGPDGGQPKMRIRCPFEKPSNLHFKPQTKTIFVTEHENNAVWKFEWQRNGKKQYCETLKF 2gvz A 3.27 BS03 ONA A 1 D396 G399 F400 T401 A404 G439 D440 D20 G23 F24 T25 A28 G63 D64 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P30803 16766715 100 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 2gvz B 3.27 BS02 ONA A 1 N1022 N1025 N133 N136 S891 I892 S942 R1029 K1065 S12 I13 S63 R140 K176 4.6.1.1 0009190,0016849,0035556 remove_due_to_license_issue P26769 16766715 100 QSYDCVCVMFASIPDFKEFYTESDVNKEGLECLRLLNEIIADFDDLLSKPKFSGVEKIKTIGSTYMAATGLSAIRQYMHIGTMVEFAYALVGKLDAINKHSFNDFKLRVGINHGPVIAGVIGAQKPQYDIWGNTVNVASRMDSTGVLDKIQVTEETSLILQTLGYTCTCRGIINVKGKGDLKTYFVNT 2gyi A 1.6 BS03 HYA A 1 H53 W136 E180 K182 H219 D286 H52 W135 E179 K181 H218 D285 H53 D56 M87 E180 K182 E216 H219 D244 D254 D256 D286 H52 D55 M86 E179 K181 E215 H218 D243 D253 D255 D285 5.3.1.5 0000287,0005737,0005975,0009045,0016853,0042732,0046872 Ki<100nM remove_due_to_license_issue P15587 7893671 960 YQPTPEDRFTFGLWTVGWQGRDPFGDATRPALDPVETVQRLAELGAHGVTFHDDDLIPFGSSDTERESHIKRFRQALDATGMTVPMATTNLFTHPVFKDGGFTANDRDVRRYALRKTIRNIDLAVELGAKTYVAWGGREGAESGAAKDVRVALDRMKEAFDLLGEYVTSQGYDTRFAIEPKPNEPRGDILLPTVGHALAFIERLERPELYGVNPEVGHEQMAGLNFPHGIAQALWAGKLFHIDLNGQSGIKYDQDLRFGAGDLRAAFWLVDLLESAGYEGPRHFDFKPPRTEDIDGVWASAAGCMRNYLILKERAAAFRADPEVQEALRASRLDELAQPTAADGVQELLADRTAFEDFDVDAAAARGMAFERLDQLAMDHLLGAR 2gyi B 1.6 BS03 HYA B 1 H53 F93 W136 E180 D286 H52 F92 W135 E179 D285 H53 D56 M87 E180 K182 E216 H219 D244 D254 D256 D286 H52 D55 M86 E179 K181 E215 H218 D243 D253 D255 D285 5.3.1.5 0000287,0005737,0005975,0009045,0016853,0042732,0046872 Ki<100nM remove_due_to_license_issue P15587 7893671 970 YQPTPEDRFTFGLWTVGWQGRDPFGDATRPALDPVETVQRLAELGAHGVTFHDDDLIPFGSSDTERESHIKRFRQALDATGMTVPMATTNLFTHPVFKDGGFTANDRDVRRYALRKTIRNIDLAVELGAKTYVAWGGREGAESGAAKDVRVALDRMKEAFDLLGEYVTSQGYDTRFAIEPKPNEPRGDILLPTVGHALAFIERLERPELYGVNPEVGHEQMAGLNFPHGIAQALWAGKLFHIDLNGQSGIKYDQDLRFGAGDLRAAFWLVDLLESAGYEGPRHFDFKPPRTEDIDGVWASAAGCMRNYLILKERAAAFRADPEVQEALRASRLDELAQPTAADGVQELLADRTAFEDFDVDAAAARGMAFERLDQLAMDHLLGAR 2gz2 A 2.1 BS01 A2P A 1 G9 T11 G12 A36 S37 R39 S40 T57 A72 T76 G8 T10 G11 A35 S36 R38 S39 T56 A71 T75 C128 Q155 R245 H252 C127 Q154 R244 H251 1.2.1.11 0000166,0004073,0008652,0009085,0009086,0009088,0009089,0009097,0016491,0016620,0019877,0046983,0050661,0051287,0071266 Kd=6uM remove_due_to_license_issue A0A0H2UPS5 16895909 502 GYTVAVVGATGAVGAQMIKMLEESTLPIDKIRYLASARSAGKSLKFKDQDITIEETTETAFEGVDIALFSAGSSTSAKYAPYAVKAGVVVVDNTSYFRQNPDVPLVVPEVNAHALDAHNGIIACPNCSTIQMMVALEPVRQKWGLDRIIVSTYQAVSGAGMGAILETQRELREVLNDGVKPCDLHAEILPSGGDKKHYPIAFNALPQIDVFTDNDYTYEEMKMTKETKKIMEDDSIAVSATCVRIPVLSAHSESVYIETKEVAPIEEVKAAIAAFPGAVLEDDVAHQIYPQAINAVGSRDTFVGRIRKDLDAEKGIHMWVVSDNLLKGAAWNSVQIAETLHERGLVRPTAELKFELK 2gz7 A 1.856 BS01 D3F A 1 P39 H41 C145 H164 M165 E166 Q192 P39 H41 C145 H164 M165 E166 Q192 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=0.3uM remove_due_to_license_issue IC50=300nM P0C6X7 16913704 307 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 2gz8 A 1.97 BS01 F3F A 1 N142 G143 C145 E166 P168 Q189 N142 G143 C145 E166 P168 Q189 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=3uM remove_due_to_license_issue IC50=3000nM P0C6X7 16913704 307 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 2gzk A -1.00 BS01 dna B 0 R4 K6 R7 M9 N10 I13 R17 R20 R21 M30 N32 Y74 K76 G77 E78 T79 K81 R91 F96 F97 G117 A120 K121 Y149 I153 R157 R4 K6 R7 M9 N10 I13 R17 R20 R21 M30 N32 Y74 K76 G77 E78 T79 K81 R91 F96 F97 G117 A120 K121 Y149 I153 R157 ? remove_due_to_license_issue P63159,Q05066 16813837 201 ~ 216 VQDRVKRPMNAFIVWSRDQRRKMALENPRMRNSEISKQLGYQWKMLTEAEKWPFFQEAQKLQAMHREKYPNYKYRKGETKKKFKDPNAPKRPPSAFFLFCSEYRPKIKGEHPGLSIGDVAKKLGEMWNNTAADDKQPYEKKAAKLKEKYEKDIAAYRAK 2gzk A -1.00 BS02 dna C 0 R7 N10 F12 N32 S36 K37 G40 W43 K44 F55 Q62 Y74 K76 K84 K90 R91 F97 R104 I116 R7 N10 F12 N32 S36 K37 G40 W43 K44 F55 Q62 Y74 K76 K84 K90 R91 F97 R104 I116 ? remove_due_to_license_issue P63159,Q05066 16813837 217 ~ 232 VQDRVKRPMNAFIVWSRDQRRKMALENPRMRNSEISKQLGYQWKMLTEAEKWPFFQEAQKLQAMHREKYPNYKYRKGETKKKFKDPNAPKRPPSAFFLFCSEYRPKIKGEHPGLSIGDVAKKLGEMWNNTAADDKQPYEKKAAKLKEKYEKDIAAYRAK 2gzl A 2.5 BS02 2AA A 1 H10 D56 G58 F68 A71 D72 L76 H12 D58 G60 F70 A73 D74 L78 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=15uM remove_due_to_license_issue P62617 16392111 901 LEMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIKA 2h02 A 2.3 BS01 2UN A 1 Y1733 N1735 D1870 H1871 C1904 S1905 A1906 V1908 G1909 R1910 Q1948 Y56 N58 D181 H182 C215 S216 A217 V219 G220 R221 Q259 D1870 C1904 R1910 T1911 Q1948 D181 C215 R221 T222 Q259 3.1.3.48 0004725,0006470,0016311 ic50=0.32uM remove_due_to_license_issue IC50=320nM P23467 16759857 402 KTSCPIKINQFEGHFMKLQADSNYLLSKEYEELKDVGRNQSCDIALLPENRGKNRYNNILPYDATRVKLSSDYINASYIPGNNFRREYIVTQGPLPGTKDDFWKMVWEQNVHNIVMVTQCVEKGRVKCDHYWPADQDSLYYGDLILQMLSESVLPEWTIREFKICGEHRLIRHFHYTVWPDHGVPETTQSLIQFVRTVRDYINRSPGAGPTVVHCSAGVGRTGTFIALDRILQQLDSKDSVDIYGAVHDLRLHRVHMVQTECQYVYLHQCVRDVLRAR 2h03 A 1.65 BS01 3UN A 1 Y1733 N1735 K1811 D1870 H1871 C1904 S1905 A1906 V1908 G1909 R1910 H1945 Y56 N58 K129 D188 H189 C222 S223 A224 V226 G227 R228 H263 D1870 C1904 R1910 T1911 Q1948 D188 C222 R228 T229 Q266 3.1.3.48 0004725,0006470,0016311 ic50=0.09uM remove_due_to_license_issue P23467 16759857 401 KTSCPIKINQFEGHFMKLQADSNYLLSKEYEELKDVGRNQSCDIALLPENRGKNRYNNILPYDATRVKLSGGSDYINASYIPGNNFRREYIVTQGPLPGTKDDFWKMVWEQNVHNIVMVTQCVEKGRVKCDHYWPADQDSLYYGDLILQMLSESVLPEWTIREFKICGEEQLDAHRLIRHFHYTVWPDHGVPETTQSLIQFVRTVRDYINRSPGAGPTVVHCSAGVGRTGTFIALDRILQQLDSKDSVDIYGAVHDLRLHRVHMVQTECQYVYLHQCVRDVLRARKLR 2h15 A 1.9 BS02 B19 A 1 N62 N67 Q92 H94 H96 L198 T199 T200 N59 N64 Q89 H91 H93 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2135nM remove_due_to_license_issue Ki=2135nM, Kd=25000nM P00918 17125255 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2h1h A 2.4 BS01 AFH A 1 A186 T187 T188 K192 W217 G218 E222 D261 T262 G263 L264 H266 I287 A186 T187 T188 K192 W217 G218 E222 D261 T262 G263 L264 H266 I287 2.4.99.23 0005515,0005829,0005886,0008713,0008920,0009103,0009244,0016757 ic50=30uM remove_due_to_license_issue P24173 16963083 400 MRVLIVKTSSMGDVLHTLPALTDAQQAIPGIKFDWVVEEGFAQIPSWHAAVERVIPVAIRRWRKAWFSAPIKAERKAFREALQAKNYDAVIDAQGLVKSAALVTRLAHGVKHGMDWQTAREPLASLFYNRKHHIAKQQHAVERTRELFAKSLGYSKPQTQGDYAIAQHFLTNLPTDAGEYAVFLHATTRDDKHWPEEHWRELIGLLADSGIRIKLPWGAPHEEERAKRLAEGFAYVEVLPKMSLEGVARVLAGAKFVVSVDTGLSHLTAALDRPNITVYGPTDPGLIGGYGKNQMVCRAPGNELSQLTANAVKQFIEENAEK 2h1k A 2.42 BS01 dna C 0 R5 Y25 R31 K46 Q50 R53 M54 K57 R3 Y23 R29 K44 Q48 R51 M52 K55 ? 0000981,0003677,0006355 remove_due_to_license_issue P70118 17315980 100 ~ 114 RTRTAYTRAQLLELEKEFLFNKYISRPRRVELAVMLNLTERHIKIWFQNRRMKWKKEE 2h1k A 2.42 BS02 dna D 0 R3 R5 T6 Y8 I47 N51 K55 R1 R3 T4 Y6 I45 N49 K53 ? 0000981,0003677,0006355 remove_due_to_license_issue P70118 17315980 214 ~ 228 RTRTAYTRAQLLELEKEFLFNKYISRPRRVELAVMLNLTERHIKIWFQNRRMKWKKEE 2h1k B 2.42 BS01 dna E 0 R5 Y25 R31 Q50 R53 M54 R5 Y25 R31 Q50 R53 M54 ? 0000981,0003677,0006355 remove_due_to_license_issue P70118 17315980 100 ~ 114 NKRTRTAYTRAQLLELEKEFLFNKYISRPRRVELAVMLNLTERHIKIWFQNRRMKWKKEE 2h1k B 2.42 BS02 dna F 0 K2 R3 R5 T6 Y8 R43 I47 N51 K55 K2 R3 R5 T6 Y8 R43 I47 N51 K55 ? 0000981,0003677,0006355 remove_due_to_license_issue P70118 17315980 214 ~ 228 NKRTRTAYTRAQLLELEKEFLFNKYISRPRRVELAVMLNLTERHIKIWFQNRRMKWKKEE 2h21 A 2.45 BS01 SAM A 1 E80 L82 S221 R222 D239 N242 H243 Y287 Y300 F302 E31 L33 S172 R173 D187 N190 H191 Y225 Y238 F240 Y287 Y225 2.1.1.127,2.1.1.259 0009507,0016279,0018022,0030785 Kd=0.29uM remove_due_to_license_issue Q43088 16682405 801 LSPAVQTFWKWLQEEGVITAKTPVKASVVTEGLGLVALKDISRNDVILQVPKRLWINPDAVAASEIGRVCSELKPWLSVILFLIRERSREDSVWKHYFGILPQETDSTIYWSEEELQELQGSQLLKTTVSVKEYVKNECLKLEQEIILPNKRLFPDPVTLDDFFWAFGILRSRAFSRLNLVVVPMADLINHSAGVTTEDHAYEVYLFSLKSPLSVKAGEQVYIQYDLNKSNAELALDYGFIEPNENRHAYTLTLEISESDPFFDDKLDVAESNGFAQTAYFDIFYNRTLPPGLLPYLRLVALGGTDAFLLESLFRDTIWGHLELSVSRDNEELLCKAVREACKSALAGYHTTIEQDRELKEGNLDSRLAIAVGIREGEKMVLQQIDGIFEQKELELDQLEYYQERRLKDLGLCGENGDILENLY 2h23 A 2.45 BS01 SAH A 1 E80 L82 P151 S221 R222 D239 N242 H243 Y287 Y300 F302 E31 L33 P102 S172 R173 D187 N190 H191 Y225 Y238 F240 Y287 Y225 2.1.1.127,2.1.1.259 0009507,0016279,0018022,0030785 Kd=21.2uM remove_due_to_license_issue Q43088 16682405 800 LSPAVQTFWKWLQEEGVITAKTPVKASVVTEGLGLVALKDISRNDVILQVPKRLWINPDAVAASEIGRVCSELKPWLSVILFLIRERSREDSVWKHYFGILPQETDSTIYWSEEELQELQGSQLLKTTVSVKEYVKNECLKLEQEIILPNKRLFPDPVTLDDFFWAFGILRSRAFSRLNLVVVPMADLINHSAGVTTEDHAYEVYLFSLKSPLSVKAGEQVYIQYDLNKSNAELALDYGFIEPNENRHAYTLTLEISESDPFFDDKLDVAESNGFAQTAYFDIFYNRTLPPGLLPYLRLVALGGTDAFLLESLFRDTIWGHLELSVSRDNEELLCKAVREACKSALAGYHTTIEQDRELKEGNLDSRLAIAVGIREGEKMVLQQIDGIFEQKELELDQLEYYQERRLKDLGLCGENGDILENLY 2h2e A 2.6 BS01 SA8 A 1 E80 L82 S221 R222 L240 N242 H243 Y287 F302 E31 L33 S172 R173 L188 N190 H191 Y225 F240 Y287 Y225 2.1.1.127,2.1.1.259 0009507,0016279,0018022,0030785 remove_due_to_license_issue Q43088 16682405 800 LSPAVQTFWKWLQEEGVITAKTPVKASVVTEGLGLVALKDISRNDVILQVPKRLWINPDAVAASEIGRVCSELKPWLSVILFLIRERSREDSVWKHYFGILPQETDSTIYWSEEELQELQGSQLLKTTVSVKEYVKNECLKLEQEIILPNKRLFPDPVTLDDFFWAFGILRSRAFSRLNLVVVPMADLINHSAGVTTEDHAYEVYLFSLKSPLSVKAGEQVYIQYDLNKSNAELALDYGFIEPNENRHAYTLTLEISESDPFFDDKLDVAESNGFAQTAYFDIFYNRTLPPGLLPYLRLVALGGTDAFLLESLFRDTIWGHLELSVSRDNEELLCKAVREACKSALAGYHTTIEQDRELKEGNLDSRLAIAVGIREGEKMVLQQIDGIFEQKELELDQLEYYQERRLKDLGLCGENGDILENLY 2h2j A 2.45 BS01 SFG A 1 E80 G81 L82 P151 T154 S221 R222 D239 N242 H243 Y287 F302 E31 G32 L33 P102 T105 S172 R173 D187 N190 H191 Y224 F239 Y287 Y224 2.1.1.127,2.1.1.259 0009507,0016279,0018022,0030785 Kd=4.2uM remove_due_to_license_issue Q43088 16682405 800 LSPAVQTFWKWLQEEGVITAKTPVKASVVTEGLGLVALKDISRNDVILQVPKRLWINPDAVAASEIGRVCSELKPWLSVILFLIRERSREDSVWKHYFGILPQETDSTIYWSEEELQELQGSQLLKTTVSVKEYVKNECLKLEQEIILPNKRLFPDPVTLDDFFWAFGILRSRAFSRLNLVVVPMADLINHSAGVTTEDHAYEYLFSLKSPLSVKAGEQVYIQYDLNKSNAELALDYGFIEPNENRHAYTLTLEISESDPFFDDKLDVAESNGFAQTAYFDIFYNRTLPPGLLPYLRLVALGGTDAFLLESLFRDTIWGHLELSVSRDNEELLCKAVREACKSALAGYHTTIEQDRELKEGNLDSRLAIAVGIREGEKMVLQQIDGIFEQKELELDQLEYYQERRLKDLGLCGENGDILENLY 2h3a A -1.00 BS01 dna C 0 R4 I5 T6 V7 T8 R4 I5 T6 V7 T8 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 173 ~ 185 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h3a A -1.00 BS02 dna D 0 M1 K2 R4 N23 S25 M1 K2 R4 N23 S25 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 186 ~ 198 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h3a B -1.00 BS01 dna C 0 K102 R104 Y114 N123 S125 E160 S164 F165 K2 R4 Y14 N23 S25 E60 S64 F65 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 173 ~ 185 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h3a B -1.00 BS02 dna D 0 Q103 R104 I105 T106 T108 N162 F165 D167 K170 Q3 R4 I5 T6 T8 N62 F65 D67 K70 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 186 ~ 198 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h3c A -1.00 BS01 dna C 0 R4 T6 R4 T6 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 173 ~ 185 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h3c A -1.00 BS02 dna D 0 K2 R4 Y14 N23 S25 K2 R4 Y14 N23 S25 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 186 ~ 198 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h3c B -1.00 BS01 dna D 0 Q103 R104 I105 T106 Q3 R4 I5 T6 ? 0003677,0005515,0017053,0032984,0045892,0097351,0110001 remove_due_to_license_issue P62552 17007877 186 ~ 198 MKQRITVTVDSDSYQLLKAYDVNISGLVSTTMQNEARRLRAERWKVENQEGMVEVARFIEMNGSFADENKDW 2h42 A 2.3 BS03 VIA A 1 F786 L804 Q817 F820 F252 L270 Q283 F286 3.1.4.35 0004114,0007165,0008081 ic50=2.4nM remove_due_to_license_issue IC50=2.2nM, Ki=1.9nM, EC50=8.7nM O76074 16735511 901 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 2h44 A 1.8 BS03 7CA A 1 H613 Y664 I665 S668 D764 A767 I768 Q775 A779 F786 L804 M816 Q817 F820 H79 Y130 I131 S134 D230 A233 I234 Q241 A245 F252 L270 M282 Q283 F286 3.1.4.35 0004114,0007165,0008081 ic50=1.7uM remove_due_to_license_issue O76074 16735511 301 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 2h4g A 2.5 BS01 694 A 1 Y46 D48 K120 F182 A217 I219 G220 R221 Q262 Y45 D47 K119 F181 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.3uM remove_due_to_license_issue P18031 16806920 300 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2h4k A 2.3 BS01 509 A 1 Y46 V49 K120 F182 A217 I219 G220 R221 Q262 Y45 V48 K119 F181 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=3.2uM remove_due_to_license_issue Ki=3200nM P18031 16806920 300 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2h4n A 1.9 BS03 AZM A 1 Q92 N94 H96 H119 V121 F131 T199 T200 Q89 N91 H93 H116 V118 F127 T195 T196 H64 N94 H96 E106 H119 T199 H61 N91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.002nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 9398308 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFNFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2h5a X 1.72 BS02 X1P X 1 Y17 T306 G307 H308 E325 S327 H329 R421 S423 N424 T425 Y9 T298 G299 H300 E317 S319 H321 R413 S415 N416 T417 H109 D242 D244 D246 R247 D340 H101 D234 D236 D238 R239 D332 5.4.2.2,5.4.2.8 0000287,0004614,0004615,0005975,0009103,0009243,0009244,0009298,0016853,0016868,0042121,0046872 remove_due_to_license_issue P26276 16880541 600 LPASIFRAYDIRGVVGDTLTAETAYWIGRAIGSESLARGEPCVAVGRDGRLSGPELVKQLIQGLVDCGCQVSDVGMVPTPVLYYAANVLEGKSGVMLTGSHNPPDYNGFKIVVAGETLANEQIQALRERIEKNDLASGVGSVEQVDILPRYFKQIRDDIAMAKPMKVVVDCGNGVAGVIAPQLIEALGCSVIPLYCEVDGNFPNHHPDPGKPENLKDLIAKVKAENADLGLAFDGDGDRVGVVTNTGTIIYPDRLLMLFAKDVVSRNPGADIIFDVKCTRRLIALISGYGGRPVMWKTGHSLIKKKMKETGALLAGEMSGHVFFKERWFGFDDGIYSAARLLEILSQDQRDSEHVFSAFPSDISTPEINITVTEDSKFAIIEALQRDAQWGEGNITTLDGVRVDYPKGWGLVRASNTTPVLVLRFEADTEEELERIKTVFRNQLKAVDSSLPVPF 2h5e A 2.8 BS01 GDP A 1 D23 G25 K26 T27 T28 H92 N142 K143 D145 T258 L260 D21 G23 K24 T25 T26 H59 N109 K110 D112 T225 L227 D23 D21 ? 0003924,0005515,0005525,0005737,0005829,0006412,0006415,0006449,0016149,0016150,0019003,0097216,1990145 remove_due_to_license_issue P0A7I4 17540173 2567 LSPYLQEVAKRRTFAIISHPDAGKTTITEKVLLFGQITTSVMQFPYHDCLVNLLDTPGHEDFSEDTYRTLTAVDCCLMVIDAAKGVEDRTRKLMEVTRLRDTPILTFMNKLDRDIRDPMELLDEVENELKIGCAPITWPIGCGKLFKGVYHLYKDETYLYQSGKGHTIQEVRIVKGLNNPDLDAAVGEDLAQQLRDELELVKGASNEFDKELFLAGEITPVFFGTALGNFGVDHMLDGLVEWAPAPMPRQTDTRTVEASEDKFTGFVFKIQANMDPKHRDRVAFMRVVSGKYEKGMKLRQVRTAKDVVISDALTFMAVEEAYPGDILGLHNHGTIQIGDTFTQGEMMKFTGIPNFAPELFRRIRLKDPKQLLKGLVQLSEEGAVQVFRPISNNDLIVGAVGVLQFDVVVARLKSEYNVEAVYESVNVATARWVECADAKKFEEFKRKNESQLALDGGDNLAYIATSMVNLRLAQERYPDVQFHQTREH 2h6b A 2.2 BS01 3C4 A 1 Y76 I84 G85 K86 T90 N92 K133 Y74 I82 G83 K84 T88 N90 K131 ? 0003677,0006355 Kd=4.1uM remove_due_to_license_issue Q8RPJ2 16803881 302 VEGLGKDFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLACLKRENILDKKKNKIIVYNLGELKHLSEQTSVDKLAAALDHH 2h6b B 2.2 BS01 3C4 A 1 L131 V134 L123 V126 ? 0003677,0006355 Kd=4.1uM remove_due_to_license_issue Q8RPJ2 16803881 302 DFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLACLKRENILDKKKNKIIVYNLGELKHLSEQTSYYSDPNSSSVDKL 2h6b B 2.2 BS02 3C4 B 1 Y76 I84 G85 K86 T90 N92 I94 K133 Y68 I76 G77 K78 T82 N84 I86 K125 ? 0003677,0006355 Kd=4.1uM remove_due_to_license_issue Q8RPJ2 16803881 301 DFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLACLKRENILDKKKNKIIVYNLGELKHLSEQTSYYSDPNSSSVDKL 2h8h A 2.2 BS01 H8H A 1 L273 V281 A293 K295 T338 Y340 M341 S342 G344 L393 D404 L189 V197 A209 K211 T254 Y256 M257 S258 G260 L309 D320 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0000122,0001545,0001819,0002102,0002223,0002376,0002862,0004672,0004713,0004715,0005080,0005102,0005158,0005178,0005515,0005524,0005634,0005654,0005737,0005739,0005743,0005764,0005770,0005829,0005856,0005884,0005886,0005901,0005911,0005925,0006338,0006468,0007155,0007165,0007172,0007173,0007179,0007229,0007283,0007611,0008284,0009410,0009612,0010447,0010628,0010629,0010632,0010634,0010907,0010954,0014856,0014911,0016004,0016020,0016236,0016301,0016477,0018108,0019899,0019901,0019904,0020037,0022407,0030054,0030154,0030168,0030296,0030331,0030900,0031295,0031333,0031648,0031667,0032205,0032587,0032869,0033146,0033625,0034139,0034332,0034446,0034614,0035306,0035331,0035401,0035556,0036035,0036120,0038096,0038128,0038166,0042169,0042476,0042542,0043025,0043065,0043066,0043114,0043149,0043274,0044294,0044325,0044877,0045056,0045087,0045121,0045124,0045296,0045453,0045747,0045780,0045785,0045821,0046579,0046628,0046718,0046777,0046875,0048008,0048010,0048011,0048013,0048041,0048471,0048477,0050731,0050839,0050847,0050900,0051057,0051117,0051219,0051222,0051385,0051450,0051602,0051895,0051897,0051902,0060065,0060444,0060491,0060576,0070062,0070102,0070161,0070301,0070374,0070542,0070555,0070700,0071222,0071253,0071375,0071393,0071398,0071456,0071498,0071560,0071803,0071897,0071902,0086091,0090263,0097060,0097110,0098609,0098978,0099091,0140801,1900182,1902533,1902564,1902737,1904263,1904385,1904707,1990646,2000117,2000256,2000386,2000394,2000588,2000641,2000811,2001237,2001243,2001286 ic50=2.7nM remove_due_to_license_issue IC50=2.7nM P12931 17064066 534 TFVALYDYESRTETDLSFKKGERLQIVNNTEGDWWLAHSLSTGQTGYIPSNYVAPSDSIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPTSKPQTQGLAKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGETGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEDNEYTARQGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKEPEERPTFEYLQAFLEDYFTSTEPQYQP 2h96 A 3.0 BS02 893 A 1 V40 M108 L110 M111 D112 A113 V158 L168 V34 M102 L104 M105 D106 A107 V152 L162 D151 K153 N156 D169 T188 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=230nM P45983 16854050 901 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 2h9t H 2.4 BS03 SVR H 1 P92 R93 R101 W237 K240 V241 D243 Q244 G246 E247 P88 R89 R98 W240 K243 V244 D246 Q247 G249 E250 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 19332154 301 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 2ha0 A 2.2 BS02 NWA A 1 W86 G120 G121 G122 S203 A204 F297 H447 W84 G118 G119 G120 S201 A202 F289 H439 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G119 G120 G152 S201 A202 G240 F289 F291 E326 H439 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 16837465 709 REDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 2ha2 A 2.05 BS01 SCK A 1 Y72 W86 Y124 W286 Y337 F338 Y341 Y72 W86 Y124 W280 Y331 F332 Y335 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd=0.022mM remove_due_to_license_issue Ki=21000nM P21836 16837465 901 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2ha3 A 2.25 BS01 CHT A 1 W86 G121 E202 H447 W86 G121 E202 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd=0.93mM remove_due_to_license_issue P21836 16837465 951 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 2ha3 A 2.25 BS02 CHT A 2 Y72 W286 Y341 Y72 W281 Y336 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd=0.93mM remove_due_to_license_issue P21836 16837465 952 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 2ha4 A 2.56 BS01 ACH A 1 Y72 Y124 W286 Y341 Y72 Y124 W280 Y335 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 16837465 545 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 2ha4 A 2.56 BS02 ACH A 2 W86 Y124 Y337 F338 W86 Y124 Y331 F332 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 16837465 546 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 2ha5 A 2.15 BS01 AT3 A 1 W86 Y124 F297 F338 W86 Y124 F290 F331 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 16837465 1901 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2ha5 A 2.15 BS03 AT3 A 2 E81 M85 D131 E452 Y465 E81 M85 D131 E445 Y458 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 16837465 1902 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2ha6 A 2.25 BS01 SCK A 1 Y72 W86 Y124 W286 Y337 F338 Y341 Y72 W86 Y124 W280 Y331 F332 Y335 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Ki=21000nM P21836 16837465 901 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2ha6 A 2.25 BS02 SCK A 2 E81 E84 M85 Y465 E81 E84 M85 Y459 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Ki=21000nM P21836 16837465 902 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2ha7 A 2.66 BS03 BCH A 1 Y72 Y124 W286 Y341 Y72 Y124 W280 Y335 G121 G122 G154 A203 A204 G242 F297 F299 E334 H447 G121 G122 G154 A203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 16837465 910 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGEAAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2hah A 1.7 BS01 3TL A 1 G32 A33 D34 Q54 I56 G57 G58 I59 G28 A29 D30 Q50 I52 G53 G54 I55 D30 T31 G32 D26 T27 G28 3.1.13.2,3.1.26.13 0004190,0006508 Ki=10nM remove_due_to_license_issue Q66972 17212810 201 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMIGGIGGFIRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSTPVNILGRDNMIKFNIRLVM 2hai A 1.58 BS01 PFI A 1 L419 R422 M423 H475 S476 I482 A486 L497 W528 L419 R422 M423 H475 S476 I482 A486 L497 W528 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.53uM remove_due_to_license_issue Q99AU2 16824756 601 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 2haw A 1.75 BS05 2PN A 1 D13 D75 H97 H98 K205 R295 K296 D12 D74 H96 H97 K204 R294 K295 3.6.1.1 0004427,0005737,0016462,0016787,0030145,0046872 Kd=12uM remove_due_to_license_issue P37487 17095506 2001 EKILIFGHQNPDTDTICSAIAYADLKNKLGFNAEPVRLGQVNGETQYALDYFKQESPRLVETAANEVNGVILVDHNERQQSIKDIEEVQVLEVIDHHRIANFETAEPLYYRAEPVGCTATILNKMYKENNVKIEKEIAGLMLSAIISDSLLFKSPTCTDQDVAAAKELAEIAGVDAEEYGLNMLKAGADLSKKTVEELISLDAKEFTLGSKKVEIAQVNTVDIEDVKKRQAELEAVISKVVAEKNLDLFLLVITDILENDSLALAIGNEAAKVEKAFNVTLENNTALLKGVVSRKKQVVPVLTDAMA 2haw B 1.75 BS05 2PN B 1 D13 D75 H97 H98 D149 K205 R295 K296 D13 D75 H97 H98 D149 K205 R295 K296 3.6.1.1 0004427,0005737,0016462,0016787,0030145,0046872 Kd=12uM remove_due_to_license_issue P37487 17095506 2002 MEKILIFGHQNPDTDTICSAIAYADLKNKLGFNAEPVRLGQVNGETQYALDYFKQESPRLVETAANEVNGVILVDHNERQQSIKDIEEVQVLEVIDHHRIANFETAEPLYYRAEPVGCTATILNKMYKENNVKIEKEIAGLMLSAIISDSLLFKSPTCTDQDVAAAKELAEIAGVDAEEYGLNMLKAGADLSKKTVEELISLDAKEFTLGSKKVEIAQVNTVDIEDVKKRQAELEAVISKVVAEKNLDLFLLVITDILENDSLALAIGNEAAKVEKAFNVTLENNTALLKGVVSRKKQVVPVLTDAMA 2hb1 A 2.0 BS01 512 A 1 Y46 K120 F182 A217 I219 G220 R221 Q262 Y45 K119 F181 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=160uM remove_due_to_license_issue P18031 16806920 800 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2hb3 A 1.35 BS01 GRL B 1 D25 A28 D30 V82 I84 D25 A28 D30 V82 I84 D25 T26 G27 D25 T26 G27 3.4.23.4 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 16913714 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hb3 B 1.35 BS01 GRL B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.4.23.4 0004190,0006508,0042802 Ki=0.0045nM remove_due_to_license_issue Q7SSI0 16913714 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hb9 A 1.75 BS03 L13 A 1 Y33 W39 H116 H118 D120 F156 I162 H196 H263 Y10 W16 H83 H85 D87 F123 I127 H159 H224 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=15uM remove_due_to_license_issue P52700 17999929 500 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 2hb9 A 1.75 BS04 L13 A 2 P106 R107 K129 R130 T132 G133 P73 R74 K96 R97 T99 G100 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=15uM remove_due_to_license_issue P52700 17999929 501 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 2hd1 A 2.23 BS02 IBM A 1 I403 L420 Y424 Q453 F456 I223 L240 Y244 Q273 F276 3.1.4.35 0004114,0007165,0008081 ic50~500uM remove_due_to_license_issue IC50=>200000nM O76083 15210993 1 PTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQKK 2hd6 A 1.8 BS02 BOS A 1 H94 H119 L198 T199 T200 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=16nM remove_due_to_license_issue Ki=16nM P00918 16942027 266 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2hdd A 1.9 BS01 dna C 0 R5 T6 F8 Q44 N51 R1 T2 F4 Q40 N47 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 9309220 1 ~ 21 RTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFKNKRAKIKKS 2hdd A 1.9 BS02 dna D 0 Y25 R31 K50 R53 Y21 R27 K46 R49 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 9309220 22 ~ 42 RTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFKNKRAKIKKS 2hdd B 1.9 BS01 dna C 0 Y25 R31 K46 K50 R53 K57 Y24 R30 K45 K49 R52 K56 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 9309220 1 ~ 21 KRPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFKNKRAKIK 2hdd B 1.9 BS02 dna D 0 K2 R3 I47 N51 K1 R2 I46 N50 ? 0000981,0003677,0006355 remove_due_to_license_issue P02836 9309220 22 ~ 42 KRPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQIKIWFKNKRAKIK 2hdq A 2.1 BS01 C21 A 1 R148 Y150 K290 R145 Y147 K287 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=40mM remove_due_to_license_issue Ki=40000000nM P00811 17072304 501 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdq A 2.1 BS02 C21 A 2 P240 Q256 A307 R309 P330 P237 Q253 A304 R306 P327 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=40mM remove_due_to_license_issue Ki=40000000nM P00811 17072304 502 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdq A 2.1 BS03 C21 A 3 A141 W142 A143 A138 W139 A140 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=40mM remove_due_to_license_issue Ki=40000000nM P00811 17072304 503 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdq A 2.1 BS04 C21 A 4 V211 Y221 T319 G320 V208 Y218 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=40mM remove_due_to_license_issue Ki=40000000nM P00811 17072304 506 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdq A 2.1 BS05 C21 A 5 P38 A231 R232 Q235 P35 A228 R229 Q232 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=40mM remove_due_to_license_issue Ki=40000000nM P00811 17072304 509 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS01 4A3 A 1 V191 Y199 H210 V188 Y196 H207 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 501 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS02 4A3 A 2 Q120 S212 Y221 G320 Q117 S209 Y218 G311 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 503 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS03 4A3 A 3 K239 P240 L241 R309 K236 P237 L238 R300 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 506 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS04 4A3 A 4 A141 W142 A143 A138 W139 A140 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 508 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS05 4A3 A 5 V278 P280 W354 V275 P277 W345 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 509 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS06 4A3 A 6 I48 G206 I45 G203 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 510 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS07 4A3 A 7 V278 N279 V275 N276 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 511 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hdr A 2.2 BS08 4A3 A 8 V125 K126 P213 G214 A215 V122 K123 P210 G211 A212 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19mM remove_due_to_license_issue Ki=19000000nM P00811 17072304 513 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hds A 1.16 BS02 4MB A 1 R148 Y150 K290 L293 R145 Y147 K287 L290 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=10mM remove_due_to_license_issue Ki=10000000nM P00811 17072304 1601 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hds A 1.16 BS03 4MB A 2 T302 P303 T299 P300 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=10mM remove_due_to_license_issue Ki=10000000nM P00811 17072304 1602 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hds A 1.16 BS04 4MB A 3 L107 H108 W260 I301 T302 P304 L104 H105 W257 I298 T299 P301 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=10mM remove_due_to_license_issue Ki=10000000nM P00811 17072304 1603 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2hf8 A 2.1 BS04 GSP A 1 G43 G45 K46 T47 L48 R78 E120 N167 K168 D170 S199 L200 K201 G33 G35 K36 T37 L38 R68 E110 N157 K158 D160 S189 L190 K191 ? 0003924,0005525,0008270,0016151,0016787,0046872,0051604 Kd=3.4uM remove_due_to_license_issue Q57884 16807243 300 KDILKANKRLADKNRKLLNKHGVVAFDFMGAIGSGKTLLIEKLIDNLKDKYKIACIAGDVIAKFDAERMEKHGAKVVPLNTGKECHLDAHLVGHALEDLNLDEIDLLFIENVGNLICPADFDLGTHKRIVVISTTEGDDTIEKHPGIMKTADLIVINKIDLADAVGADIKKMENDAKRINPDAEVVLLSLKTMEGFDKVLEFIEKSVKEVK 2hf8 B 2.1 BS01 GSP A 1 K153 V175 K142 V164 ? 0003924,0005525,0008270,0016151,0016787,0046872,0051604 Kd=3.4uM remove_due_to_license_issue Q57884 16807243 300 DILKANKRLADKNRKLLNKHGVVAFDFMGAIGSGKTLLIEKLIDNLKDKYKIACIAGDVIAKFDAERMEKHGAKVVPLNTGKECHLDAHLVGHALEDLNLDEIDLLFIENVGNLICPADFDLGTHKRIVVISTTEGDDTIEKHPGIMKTADLIVINKIDLADAVGADIKKMENDAKRINPDAEVVLLSLKTMEGFDKVLEFIEKSVKEV 2hf8 B 2.1 BS05 GSP B 1 G43 G45 K46 T47 L48 R78 E120 N167 K168 D170 S199 L200 K201 G32 G34 K35 T36 L37 R67 E109 N156 K157 D159 S188 L189 K190 ? 0003924,0005525,0008270,0016151,0016787,0046872,0051604 Kd=3.4uM remove_due_to_license_issue Q57884 16807243 300 DILKANKRLADKNRKLLNKHGVVAFDFMGAIGSGKTLLIEKLIDNLKDKYKIACIAGDVIAKFDAERMEKHGAKVVPLNTGKECHLDAHLVGHALEDLNLDEIDLLFIENVGNLICPADFDLGTHKRIVVISTTEGDDTIEKHPGIMKTADLIVINKIDLADAVGADIKKMENDAKRINPDAEVVLLSLKTMEGFDKVLEFIEKSVKEV 2hfp A 2.0 BS02 NSI A 1 E259 K265 H266 I281 G284 C285 R288 L330 I341 S342 E54 K60 H61 I76 G79 C80 R83 L125 I136 S137 ? 0003677,0004879,0005634,0006355 ic50=3nM remove_due_to_license_issue IC50=3nM P37231 16919947 478 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2hfp A 2.0 BS03 NSI A 2 C285 Q286 S289 H323 Y327 F360 F363 M364 K367 H449 L452 L453 Y473 C80 Q81 S84 H118 Y122 F155 F158 M159 K162 H244 L247 L248 Y268 ? 0003677,0004879,0005634,0006355 ic50=3nM remove_due_to_license_issue IC50=3nM P37231 16919947 479 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2hgh A -1.00 BS01 rna B 0 Y105 K117 K118 H119 N120 Q121 K123 K144 F146 L148 S150 R151 K153 R154 H155 V158 Y162 T176 W177 T178 K182 Y2 K14 K15 H16 N17 Q18 K20 K41 F43 L45 S47 R48 K50 R51 H52 V55 Y59 T73 W74 T75 K79 ? remove_due_to_license_issue P03001 16405997 1 ~ 55 MYVCHFENCGKAFKKHNQLKVHQFSHTQQLPYECPHEGCDKRFSLPSRLKRHEKVHAGYPCKKDDSCSFVGKTWTLYLKHVAECHQD 2hh5 B 1.8 BS04 GNQ B 1 C25 K64 G68 G69 F70 A140 V162 N163 H164 G165 F211 C25 K64 G68 G69 F70 A140 V162 N163 H164 G165 F211 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 Ki=0.032uM remove_due_to_license_issue Ki=32nM P25774 16876402 501 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 2hh5 B 1.8 BS05 GNQ A 1 P143 F146 P143 F146 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 Ki=0.032uM remove_due_to_license_issue Ki=32nM P25774 16876402 401 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 2hha A 2.35 BS01 3TP A 1 E205 E206 Y547 Q553 K554 S630 Y662 Y666 E167 E168 Y509 Q515 K516 S592 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.122uM remove_due_to_license_issue IC50=122nM P27487 16919457 1000 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2hhn B 1.55 BS01 GNQ B 1 Q19 G20 C25 W26 G68 G69 F70 V162 N163 H164 W186 F211 Q19 G20 C25 W26 G68 G69 F70 V162 N163 H164 W186 F211 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 Ki=32nM remove_due_to_license_issue Ki=32nM P25774 16876402 901 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 2hhu A 1.8 BS01 dna B 0 T550 T552 T556 S557 A558 R578 K582 Y587 R615 Q624 N625 I626 P627 I628 R629 V828 H829 D830 T254 T256 T260 S261 A262 R282 K286 Y291 R319 Q328 N329 I330 P331 I332 R333 V532 H533 D534 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q5KWC1 17179038 19 ~ 29 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPDTKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNFGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hhu A 1.8 BS02 dna C 0 N527 N529 S530 S585 T586 L610 T611 Q612 T613 R615 S617 S618 T619 E620 N622 G711 Y714 S717 G720 L721 N724 R771 F786 R789 N793 Q797 N231 N233 S234 S289 T290 L314 T315 Q316 T317 R319 S321 S322 T323 E324 N326 G415 Y418 S421 G424 L425 N428 R475 F490 R493 N497 Q501 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q5KWC1 17179038 5 ~ 17 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPDTKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNFGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hiw A 2.2 BS01 7MP A 1 L266 Y271 V274 A287 K289 E304 M308 V317 I331 T333 M336 H379 L388 A398 D399 F400 L23 Y28 V31 A44 K46 E61 M65 V74 I88 T90 M93 H136 L145 A155 D156 F157 D381 A383 R385 N386 D399 P420 D138 A140 R142 N143 D156 P177 2.7.10.2 0004672,0004713,0005524,0006468 ic50=8nM remove_due_to_license_issue P00519 16873026 531 GAMDPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQE 2hiz A 2.5 BS01 LIJ A 1 D32 G34 S35 Y71 T72 Q73 F108 W115 I126 Y198 D228 G230 T231 T232 R235 D35 G37 S38 Y74 T75 Q76 F111 W118 I129 Y190 D220 G222 T223 T224 R227 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=112nM remove_due_to_license_issue P56817 17046251 801 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2hj4 B 1.8 BS01 PNZ D 1 F123 N124 G178 F51 N52 G106 M98 M26 1.4.9.2 0016491,0030058,0030059,0042597 remove_due_to_license_issue P84888 17636875 1201 REVLTGGHSVSAPQENRIYVMDSVFMHLTESRVHVYDYTNGKFLGMVPTAFNGHVQVSNDGKKIYTMTTYHERITRGKRSDVVEVWDADKLTFEKEISLPPKRVQGLNYDGLFRQTTDGKFIVLQNASPATSIGIVDVAKGDYVEDVTAAAGCWSVIPQPNRPRSFMTICGDGGLLTINLGEDGKVASQSRSKQMFSVKDDPIFIAPALDKDKAHFVSYYGNVYSADFSGDEVKVDGPWSLLNDEDKAKNWVPGGYNLVGLHRASGRMYVFMHPDGKEGTHKFPAAEIWVMDTKTKQRVARIPGRDALSMTIDQQRNLMLTLDGGNVNVYDISQPEPKLLRTIEGAAEASLQVQFHPV 2hj4 B 1.8 BS02 PNZ D 2 Y328 L380 A421 L423 Y256 L308 A349 L351 M98 M26 1.4.9.2 0016491,0030058,0030059,0042597 remove_due_to_license_issue P84888 17636875 1202 REVLTGGHSVSAPQENRIYVMDSVFMHLTESRVHVYDYTNGKFLGMVPTAFNGHVQVSNDGKKIYTMTTYHERITRGKRSDVVEVWDADKLTFEKEISLPPKRVQGLNYDGLFRQTTDGKFIVLQNASPATSIGIVDVAKGDYVEDVTAAAGCWSVIPQPNRPRSFMTICGDGGLLTINLGEDGKVASQSRSKQMFSVKDDPIFIAPALDKDKAHFVSYYGNVYSADFSGDEVKVDGPWSLLNDEDKAKNWVPGGYNLVGLHRASGRMYVFMHPDGKEGTHKFPAAEIWVMDTKTKQRVARIPGRDALSMTIDQQRNLMLTLDGGNVNVYDISQPEPKLLRTIEGAAEASLQVQFHPV 2hj4 D 1.8 BS01 PNZ D 1 D84 X109 N159 D14 X39 N89 W109 A134 F153 W39 A64 F83 1.4.9.2 0009308,0016491,0016638,0030059,0042597 Kd=4.29uM remove_due_to_license_issue P84887 17636875 1201 EVNSCDYWRHCAVDGFLCSCCGGTTTTCPPGSTPSPISWIGTCHNPHDGKDYLISYHDCCGKTACGRCQCNTQTRERPGYEFFLHNDVNWCMANENSTFHCTTSVLVGL 2hj4 D 1.8 BS02 PNZ D 2 D84 N141 D14 N71 W109 A134 F153 W39 A64 F83 1.4.9.2 0009308,0016491,0016638,0030059,0042597 Kd=4.29uM remove_due_to_license_issue P84887 17636875 1202 EVNSCDYWRHCAVDGFLCSCCGGTTTTCPPGSTPSPISWIGTCHNPHDGKDYLISYHDCCGKTACGRCQCNTQTRERPGYEFFLHNDVNWCMANENSTFHCTTSVLVGL 2hk5 A 2.0 BS01 1BM A 1 L251 A271 K273 E288 I314 T316 F318 M319 G322 A368 N369 L371 D382 L23 A43 K45 E60 I86 T88 F90 M91 G94 A140 N141 L143 D154 D364 R366 A368 N369 D382 F402 D136 R138 A140 N141 D154 F174 2.7.10.2 0004672,0004713,0005524,0006468 ic50=46nM remove_due_to_license_issue IC50=46nM P08631 16997556 499 AQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDF 2hl4 A 1.55 BS02 BO1 A 1 Q92 H94 H119 F131 L198 T199 T200 Q90 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=23nM remove_due_to_license_issue Ki=23nM P00918 17251017 264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2hm1 A 2.2 BS01 LIQ A 1 Q12 G13 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 Y198 D228 G230 T231 T232 R235 Q15 G16 L33 D35 G37 S38 Y74 T75 Q76 F111 W118 Y194 D224 G226 T227 T228 R231 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=2nM remove_due_to_license_issue P56817 17049233 801 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2hmu A 2.25 BS01 ATP A 1 R16 F17 D36 I37 K41 A57 I78 G79 R11 F12 D31 I32 K36 A52 I73 G74 ? 0006813 remove_due_to_license_issue O32080 16990138 601 NKQFAVIGLGRFGGSIVKELHRMGHEVLAVDINEEKVNAYASYATHAVIANATEENELLSLGIRNFEYVIVAIGANIQASTLTTLLLKELDIPNIWVKAQNYYHHKVLEKIGADRIIHPEKDMGVKIAQSLSDENVLNY 2hmu B 2.25 BS01 ATP B 1 R16 D36 I37 K41 A57 I78 G79 R10 D30 I31 K35 A51 I72 G73 ? 0006813 remove_due_to_license_issue O32080 16990138 602 KQFAVIGLGRFGGSIVKELHRMGHEVLAVDINEEKVNAYASYATHAVIANATEENELLSLGIRNFEYVIVAIGANIQASTLTTLLLKELDIPNIWVKAQNYYHHKVLEKIGADRIIHPEKDMGVKIAQSLSDENV 2hmv A 2.2 BS01 ADP A 1 G15 R16 D36 I37 K41 A57 I78 G79 G10 R11 D31 I32 K36 A52 I73 G74 ? 0006813 remove_due_to_license_issue O32080 16990138 601 NKQFAVIGLGRFGGSIVKELHRMGHEVLAVDINEEKVNAYASYATHAVIANATEENELLSLGIRNFEYVIVAIGANIQASTLTTLLLKELDIPNIWVKAQNYYHHKVLEKIGADRIIHPEKDMGVKIAQSLSDENVLNY 2hmv B 2.2 BS01 ADP B 1 G13 G15 D36 I37 K41 A57 I78 G7 G9 D30 I31 K35 A51 I72 ? 0006813 remove_due_to_license_issue O32080 16990138 602 KQFAVIGLGRFGGSIVKELHRMGHEVLAVDINEEKVNAYASYATHAVIANATEENELLSLGIRNFEYVIVAIGANIQASTLTTLLLKELDIPNIWVKAQNYYHHKVLEKIGADRIIHPEKDMGVKIAQSLSDENV 2hmw A 3.0 BS01 ATP A 1 R16 D36 I37 K41 A57 I78 G79 A80 R11 D31 I32 K36 A52 I73 G74 A75 ? 0006813 remove_due_to_license_issue O32080 16990138 601 NKQFAVIGLGRFGGSIVKELHRMGHEVLAVDINEEKVNAYASYATHAVIANATEENELLSLGIRNFEYVIVAIGANIQASTLTTLLLKELDIPNIWVKAQNYYHHKVLEKIGADRIIHPEKDMGVKIAQSLSDEN 2hmw B 3.0 BS01 ATP B 1 R16 D36 I37 N56 A57 I78 G79 A80 R9 D29 I30 N49 A50 I71 G72 A73 ? 0006813 remove_due_to_license_issue O32080 16990138 602 QFAVIGLGRFGGSIVKELHRMGHEVLAVDINEEKVNAYASYATHAVIANATEENELLSLGIRNFEYVIVAIGANIQASTLTTLLLKELDIPNIWVKAQNYYHHKVLEKIGADRIIHPEKDMGVKIAQSLSDENVLNY 2hnc A 1.55 BS02 1SA A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=60nM remove_due_to_license_issue Ki=60nM, IC50=2900nM P00918 17000110 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2hoc A 2.1 BS02 1CN A 1 H94 H119 F131 V135 L198 T199 T200 L204 H92 H117 F128 V132 L195 T196 T197 L201 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.3nM remove_due_to_license_issue Ki=0.3nM P00918 17000110 265 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2hoc A 2.1 BS03 1CN A 2 F20 P21 I22 V135 Q136 P202 L204 E205 F18 P19 I20 V132 Q133 P199 L201 E202 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.3nM remove_due_to_license_issue Ki=0.3nM P00918 17000110 266 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2hof A 2.4 BS01 dna C 0 F37 S38 H40 T41 Q90 I174 A175 K244 N245 R259 E262 K276 R282 Y283 S287 G288 H289 F18 S19 H21 T22 Q71 I155 A156 K212 N213 R227 E230 K244 R250 Y251 S255 G256 H257 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hof A 2.4 BS02 dna D 0 M44 S47 R50 R81 L83 A84 K86 T87 Q90 A131 K132 Q156 R159 R173 R241 V242 K244 L256 S257 R259 A260 R282 Y283 R292 W315 I320 Y324 M25 S28 R31 R62 L64 A65 K67 T68 Q71 A112 K113 Q137 R140 R154 R209 V210 K212 L224 S225 R227 A228 R250 Y251 R260 W283 I288 Y292 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hof B 2.4 BS01 dna C 0 K43 M44 S47 R50 R81 L83 A84 K86 T87 Q90 R118 K132 R159 R173 R241 V242 K244 S257 R259 A260 R282 W315 T316 N317 K24 M25 S28 R31 R62 L64 A65 K67 T68 Q71 R99 K113 R140 R154 R222 V223 K225 S238 R240 A241 R263 W296 T297 N298 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNAMVRLLED 2hof B 2.4 BS02 dna D 0 F37 S38 H40 T41 Q90 M97 R100 R101 R106 R121 I174 A175 A201 R243 N245 R259 E262 R282 Y283 S287 G288 H289 F18 S19 H21 T22 Q71 M78 R81 R82 R87 R102 I155 A156 A182 R224 N226 R240 E243 R263 Y264 S268 G269 H270 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNAMVRLLED 2hog A 1.9 BS01 710 A 1 Q13 L15 A36 K38 L84 E85 Y86 C87 G90 L137 S147 D148 Q12 L14 A35 K37 L76 E77 Y78 C79 G82 L129 S139 D140 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.3nM remove_due_to_license_issue O14757 16978863 324 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2hoi A 2.601 BS01 dna C 0 F37 S38 H40 T41 Q90 M97 I174 A175 R243 K244 N245 R259 E262 K276 R282 Y283 S287 G288 H289 F18 S19 H21 T22 Q71 M78 I155 A156 R224 K225 N226 R240 E243 K257 R263 Y264 S268 G269 H270 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 1 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi A 2.601 BS02 dna D 0 M44 S47 R50 R81 L83 A84 K86 T87 K132 Q156 R159 R173 T202 R241 V242 K244 L256 S257 R259 A260 R282 Y283 R292 W315 I320 Y324 M25 S28 R31 R62 L64 A65 K67 T68 K113 Q137 R140 R154 T183 R222 V223 K225 L237 S238 R240 A241 R263 Y264 R273 W296 I301 Y305 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi B 2.601 BS01 dna C 0 K43 M44 S47 R50 R81 L83 A84 K86 T87 Q90 R118 K122 K132 R159 R173 R241 V242 K244 S257 R259 R282 Y283 H289 R292 W315 T316 N317 I320 Y324 R326 K24 M25 S28 R31 R62 L64 A65 K67 T68 Q71 R99 K103 K113 R140 R154 R222 V223 K225 S238 R240 R263 Y264 H270 R273 W296 T297 N298 I301 Y305 R307 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 1 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi B 2.601 BS02 dna D 0 F37 S38 H40 T41 Q90 M97 R100 R101 R106 R118 R121 I174 A175 A201 R243 K244 R259 E262 K276 R282 Y283 S287 G288 F18 S19 H21 T22 Q71 M78 R81 R82 R87 R99 R102 I155 A156 A182 R224 K225 R240 E243 K257 R263 Y264 S268 G269 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi G 2.601 BS01 dna E 0 F37 S38 H40 T41 Q90 M97 R106 I174 A175 R243 N245 R259 E262 R282 Y283 S287 G288 H289 F18 S19 H21 T22 Q71 M78 R87 I155 A156 R224 N226 R240 E243 R263 Y264 S268 G269 H270 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi G 2.601 BS02 dna F 0 M44 S47 R50 R81 L83 A84 K86 T87 Q90 K132 Q156 R159 R173 T202 R241 V242 K244 L256 S257 R259 A260 R282 Y283 R292 W315 I320 Y324 M25 S28 R31 R62 L64 A65 K67 T68 Q71 K113 Q137 R140 R154 T183 R222 V223 K225 L237 S238 R240 A241 R263 Y264 R273 W296 I301 Y305 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi H 2.601 BS01 dna E 0 M44 S47 R81 L83 A84 K86 T87 Q90 K122 K132 R159 R173 R241 V242 K244 L256 S257 R259 A260 R282 Y283 H289 R292 W315 T316 N317 I320 Y324 R326 M25 S28 R62 L64 A65 K67 T68 Q71 K103 K113 R140 R154 R222 V223 K225 L237 S238 R240 A241 R263 Y264 H270 R273 W296 T297 N298 I301 Y305 R307 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hoi H 2.601 BS02 dna F 0 F37 S38 H40 T41 Q90 M97 R100 R101 R106 R118 R121 R173 I174 A175 A201 R243 N245 R259 E262 K276 R282 Y283 S287 G288 F18 S19 H21 T22 Q71 M78 R81 R82 R87 R99 R102 R154 I155 A156 A182 R224 N226 R240 E243 K257 R263 Y264 S268 G269 ? 0003677,0006310,0015074 remove_due_to_license_issue P06956 17573343 2 ~ 35 SDEVRKNLMDMFRDRQAFSEHTWKMLLSVCRSWAAWCKLNNRKWFPAEPEDVRDYLLYLQARGLAVKTIQQHLGQLNMLHRRSGLPRPSDSNAVSLVMRRIRKENVDAGERAKQALAFERTDFDQVRSLMENSDRCQDIRNLAFLGIAYNTLLRIAEIARIRVKDISRTDGGRMLIHIGRTATLVSTAGVEKALSLGVTKLVERWISVSGVADDPNNYLFCRVRKNGVAAPSATSQLSTRALEGIFEATHRLIYGAKDDSGQRYLAWSGHSARVGAARDMARAGVSIPEIMQAGGWTNVNIVMNYIRNLDSETGAMVRLLED 2hos A 1.9 BS01 dna C 0 R5 T6 F8 N51 R1 T2 F4 N47 ? 0003677 remove_due_to_license_issue P02836 17240973 1 ~ 21 RTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKST 2hos A 1.9 BS02 dna D 0 Y25 K50 R53 K57 Y21 K46 R49 K53 ? 0003677 remove_due_to_license_issue P02836 17240973 22 ~ 42 RTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKST 2hos B 1.9 BS01 dna C 0 Y25 R31 K46 K50 R53 K57 Y24 R30 K45 K49 R52 K56 ? 0003677 remove_due_to_license_issue P02836 17240973 1 ~ 21 KRPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKS 2hos B 1.9 BS02 dna D 0 R3 N51 R2 N50 ? 0003677 remove_due_to_license_issue P02836 17240973 22 ~ 42 KRPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKS 2hot A 2.19 BS01 dna C 0 R5 T6 F8 N51 K55 R1 T2 F4 N47 K51 ? 0003677 remove_due_to_license_issue P02836 17240973 1 ~ 21 RTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKST 2hot A 2.19 BS02 dna D 0 Y25 K50 R53 Y21 K46 R49 ? 0003677 remove_due_to_license_issue P02836 17240973 22 ~ 42 RTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKST 2hot B 2.19 BS01 dna C 0 Y25 K46 K50 R53 Y24 K45 K49 R52 ? 0003677 remove_due_to_license_issue P02836 17240973 1 ~ 21 KRPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKS 2hot B 2.19 BS02 dna D 0 K2 R3 N51 K1 R2 N50 ? 0003677 remove_due_to_license_issue P02836 17240973 22 ~ 42 KRPRTAFSSEQLARLKREFNENRYLTERRRQQLSSELGLNEAQVKGWFKNMRAKIKKS 2hpa A 2.9 BS01 PT3 A 1 R1011 H1012 R1015 I1018 R1079 H1257 D1258 R11 H12 R15 I18 R79 H257 D258 3.1.3.2,3.1.3.48,3.1.3.5 0003993,0004725,0004726,0005515,0005576,0005615,0005634,0005737,0005764,0005765,0005771,0005829,0005886,0006144,0006338,0006629,0006772,0008253,0009117,0012506,0016020,0016311,0016787,0016791,0030141,0030175,0030946,0031985,0033265,0035577,0042131,0042802,0042803,0045177,0046085,0051930,0052642,0060090,0060168,0070062,0106411,0140793 remove_due_to_license_issue P15309 9804805 1345 KELKFVTLVFRHGDRSPIDTFPTDPIKESSWPQGFGQLTQLGMEQHYELGEYIRKRYRKFLNESYKHEQVYIRSTDVDRTLMSAMTNLAALFPPEGVSIWNPILLWQPIPVHTVPLSEDQLLYLPFRNCPRFQELESETLKSEEFQKRLHPYKDFIATLGKLSGLHGQDLFGIWSKVYDPLYCESVHNFTLPSWATEDTMTKLRELSELSLLSLYGIHKQKEKSRLQGGVLVNEILNHMKRATQIPSYKKLIMYSAHDTTVSGLQMALDVYNGLLPPYASCHLTELYFEKGEYFVEMYYRNETQHEPYPLMLPGCSPSCPLERFAELVGPVIPQDWSTECMT 2hqu A 2.2 BS01 DUP A 1 R85 S86 G87 R59 S60 G61 A46 R85 G87 I94 D102 A20 R59 G61 I68 D76 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRRAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 2hqu A 2.2 BS02 DUP B 1 A98 G99 V100 I101 D102 Y105 G110 A72 G73 V74 I75 D76 Y79 G84 A46 R85 G87 I94 D102 A20 R59 G61 I68 D76 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRRAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 2hqu A 2.2 BS03 DUP C 1 R153 G157 F158 G159 S160 T161 R127 G131 F132 G133 S134 T135 A46 R85 G87 I94 D102 A20 R59 G61 I68 D76 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRRAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 2hqu B 2.2 BS01 DUP A 1 A98 G99 V100 I101 D102 Y105 G110 A75 G76 V77 I78 D79 Y82 G87 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 2hqu B 2.2 BS02 DUP B 1 R153 G157 F158 G159 S160 T161 R130 G134 F135 G136 S137 T138 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 2hqu B 2.2 BS03 DUP C 1 R85 S86 G87 Q131 R62 S63 G64 Q108 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 2hqu C 2.2 BS01 DUP B 1 R85 S86 G87 R62 S63 G64 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQF 2hqu C 2.2 BS02 DUP C 1 A98 G99 V100 I101 D102 Y105 G110 A75 G76 V77 I78 D79 Y82 G87 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 Kd=7.2uM remove_due_to_license_issue P33316 17880943 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQF 2hr1 A 1.96 BS01 dna C 0 Y44 I86 Q90 N123 K234 G236 Q237 G256 G257 S294 Q297 Y44 I86 Q90 N123 K234 G236 Q237 G256 G257 S294 Q297 C81 E119 R163 R165 C81 E119 R163 R165 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 16926025 402 ~ 413 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNFASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAITLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 2hr1 A 1.96 BS02 dna D 0 F79 C81 S85 I86 S87 G88 K89 R97 E119 V121 K162 R165 R228 Q237 R240 Y242 I249 T250 A253 Y254 G255 G256 N304 F79 C81 S85 I86 S87 G88 K89 R97 E119 V121 K162 R165 R228 Q237 R240 Y242 I249 T250 A253 Y254 G255 G256 N304 C81 E119 R163 R165 C81 E119 R163 R165 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 16926025 421 ~ 433 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNFASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAITLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 2hrm A 1.7 BS01 UC5 A 1 N84 L88 I89 D90 Y93 M98 N84 L88 I89 D90 Y93 M98 A29 R71 G73 I80 D90 A29 R71 G73 I80 D90 3.6.1.23 0000287,0004170,0005737,0005829,0006226,0009117,0016787,0032991,0042802,0046081,0046872,0070207 Kd=278.5uM remove_due_to_license_issue P06968 17932923 777 MMKKIDVKILDPRVGKEFPLPTYATSGSAGLDLRACLNDAVELAPGDTTLVPTGLAIHIADPSLAAMMLPRSGLGHKHGIVLGNLVGLIDSDYQGQLMISVWNRGQDSFTIQPGERIAQMIFVPVVQAEFNLVEDFD 2hs1 A 0.84 BS01 017 A 1 D25 G27 A28 D29 G48 I50 D25 G27 A28 D29 G48 I50 3.4.23.16 0004190,0006508,0042802 Ki=3.3nM remove_due_to_license_issue Q7SSI0 16962136 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hs1 B 0.84 BS01 017 A 1 D125 A128 D130 I132 P181 V182 D25 A28 D30 I32 P81 V82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=3.3nM remove_due_to_license_issue Q7SSI0 16962136 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hs1 B 0.84 BS02 017 B 1 P144 K145 K155 V156 R157 P44 K45 K55 V56 R57 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=3.3nM remove_due_to_license_issue Q7SSI0 16962136 203 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hs2 A 1.22 BS01 017 A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 3.4.23.16 0004190,0006508,0042802 Ki=4.9nM remove_due_to_license_issue Q7SSI0 16962136 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKLIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hs2 B 1.22 BS01 017 A 1 D125 G127 A128 D130 I150 P181 I184 D25 G27 A28 D30 I50 P81 I84 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=4.9nM remove_due_to_license_issue Q7SSI0 16962136 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKLIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2hs2 B 1.22 BS02 017 B 1 P144 K145 K155 V156 R157 P44 K45 K55 V56 R57 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=4.9nM remove_due_to_license_issue Q7SSI0 16962136 203 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKLIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2ht0 A 2.0 BS01 dna D 0 K45 R55 K57 P61 R63 R82 K88 K44 R54 K56 P60 R62 R81 K87 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 17097674 37 ~ 16 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 2ht0 A 2.0 BS02 dna E 0 G48 N51 K86 G47 N50 K85 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 17097674 15 ~ 29 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 2ht0 A 2.0 BS03 dna F 0 T4 K5 K57 R60 R63 N64 P65 I73 R76 T3 K4 K56 R59 R62 N63 P64 I72 R75 ? 0000976,0001216,0003677,0005737,0005829,0006310,0006351,0006355,0006417,0009295,0030527,0032993,0043565,0045893,1990177 remove_due_to_license_issue P0A6X7 17097674 30 ~ 49 ALTKAEMSEYLFDKLGLSKRDAKELVELFFEEIRRALENGEQVKLSGFGNFDLRDKNQRPGRNPKTGEDIPITARRVVTFRPGQKLKSRVENASPK 2ht0 B 2.0 BS01 dna C 0 R46 G47 S50 K81 K84 R46 G47 S50 K81 K84 ? 0003677,0005694,0005829,0006310,0006355,0006417,0030527 remove_due_to_license_issue Q14F22 17097674 50 ~ 38 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIEIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIY 2ht0 B 2.0 BS02 dna D 0 S4 K27 R62 N63 P64 L72 K75 S4 K27 R62 N63 P64 L72 K75 ? 0003677,0005694,0005829,0006310,0006355,0006417,0030527 remove_due_to_license_issue Q14F22 17097674 37 ~ 16 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIEIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIY 2ht0 B 2.0 BS03 dna F 0 E44 I45 R46 H54 R56 H79 E44 I45 R46 H54 R56 H79 ? 0003677,0005694,0005829,0006310,0006355,0006417,0030527 remove_due_to_license_issue Q14F22 17097674 30 ~ 49 MTKSELIERLATQQSHIPAKTVEDAVKEMLEHMASTLAQGERIEIRGFGSFSLHYRAPRTGRNPKTGDKVELEGKYVPHFKPGKELRDRANIY 2hu6 A 1.32 BS06 37A A 1 G179 I180 L181 H218 V235 F237 P238 T239 Y240 K241 G74 I75 L76 H113 V130 F132 P133 T134 Y135 K136 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=154uM remove_due_to_license_issue IC50=149000nM, Kd=154000nM P39900 16899369 400 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2hvc A 2.1 BS01 LGD A 1 L704 N705 G708 Q711 M742 M745 V746 M749 F764 M780 M787 L873 F876 T877 L36 N37 G40 Q43 M74 M77 V78 M81 F96 M112 M119 L205 F208 T209 ? remove_due_to_license_issue Ki=4.6nM, EC50=0.2nM P10275 17077481 2226 CQPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 2hvh A 2.492 BS01 dna B 0 T550 K551 T552 T556 A558 R578 K582 Y587 R615 Q624 N625 I626 P627 I628 R629 H829 D830 T254 K255 T256 T260 A262 R282 K286 Y291 R319 Q328 N329 I330 P331 I332 R333 H533 D534 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q45458 17179038 21 ~ 29 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvh A 2.492 BS02 dna C 0 N527 N529 S530 Q533 K582 T586 T611 Q612 T613 S617 S618 T619 E620 N622 Y714 I716 S717 G720 R771 F786 R789 Q797 N231 N233 S234 Q237 K286 T290 T315 Q316 T317 S321 S322 T323 E324 N326 Y418 I420 S421 G424 R475 F490 R493 Q501 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q45458 17179038 2 ~ 12 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvh D 2.492 BS01 dna E 0 T550 T552 T556 A558 R578 Q579 K582 Y587 R615 Q624 N625 P627 I628 R629 V828 H829 T254 T256 T260 A262 R282 Q283 K286 Y291 R319 Q328 N329 P331 I332 R333 V532 H533 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q45458 17179038 21 ~ 29 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvh D 2.492 BS02 dna F 0 N527 N529 S530 K582 T586 T611 Q612 T613 S617 S618 T619 E620 N622 G711 Y714 I716 S717 Y719 G720 R771 F786 R789 N793 Q797 N231 N233 S234 K286 T290 T315 Q316 T317 S321 S322 T323 E324 N326 G415 Y418 I420 S421 Y423 G424 R475 F490 R493 N497 Q501 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q45458 17179038 2 ~ 12 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvi A 1.98 BS01 dna B 0 T550 K551 T552 T556 S557 A558 R578 K582 Y587 R615 Q624 N625 I626 P627 I628 R629 H829 T254 K255 T256 T260 S261 A262 R282 K286 Y291 R319 Q328 N329 I330 P331 I332 R333 H533 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q5KWC1 17179038 21 ~ 29 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvi A 1.98 BS02 dna C 0 N527 N529 S530 S585 T586 T611 Q612 T613 S617 S618 T619 E620 N622 G711 Y714 I716 S717 Y719 G720 R771 F781 N782 F786 R789 N793 Q797 N231 N233 S234 S289 T290 T315 Q316 T317 S321 S322 T323 E324 N326 G415 Y418 I420 S421 Y423 G424 R475 F485 N486 F490 R493 N497 Q501 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q5KWC1 17179038 1 ~ 12 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvi D 1.98 BS01 dna E 0 T550 K551 T552 T556 S557 A558 R578 K582 Y587 R615 Q624 N625 I626 P627 I628 R629 V828 H829 T254 K255 T256 T260 S261 A262 R282 K286 Y291 R319 Q328 N329 I330 P331 I332 R333 V532 H533 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q5KWC1 17179038 21 ~ 29 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvi D 1.98 BS02 dna F 0 N527 N529 S530 K582 S585 T586 T611 Q612 T613 S617 S618 T619 E620 N622 G711 Y714 I716 S717 Y719 G720 R771 F786 R789 M790 N793 Q797 N231 N233 S234 K286 S289 T290 T315 Q316 T317 S321 S322 T323 E324 N326 G415 Y418 I420 S421 Y423 G424 R475 F490 R493 M494 N497 Q501 2.7.7.7 0003676,0003677,0003887,0006139,0006260,0006261,0008408 remove_due_to_license_issue Q5KWC1 17179038 1 ~ 12 KKMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNYGIVYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 2hvx A 2.6 BS01 DRX A 1 H57 Y94 T96 L99 D102 A190 F191 K192 S195 S214 Y215 G216 R217 H45 Y81 T83 L86 D89 A177 F178 K179 S182 S197 Y198 G199 R200 H57 D102 K192 G193 D194 S195 G196 H45 D89 K179 G180 D181 S182 G183 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 remove_due_to_license_issue Ki=36nM, IC50=29nM P23946 17361995 500 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPSQKNFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 2hw2 A 1.45 BS03 RFP A 1 F39 W59 G60 N86 V87 K90 K91 M126 G129 L130 L133 F34 W54 G55 N81 V82 K85 K86 M121 G124 L125 L128 2.4.2.30 0016740 Ki=1.07mM remove_due_to_license_issue A0QRS5 18349144 1200 PKPFEVHESGAYLHGTKAELKVGDRLVPGRESNFEAGRIMNHIYITQTLDAAVWGAELAAGEGRGRIFIVEPEGAIEDDPNVTDKKLPGNPTRSYRTREPVWIVGELTDWVGHPPEQLAAMRQGLEELRRKGLAVIYD 2hwh A 2.3 BS01 RNA A 1 L419 S476 Y477 I482 L497 W528 L414 S471 Y472 I477 L492 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=2uM remove_due_to_license_issue P26663 16934455 960 HHSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSL 2hwi A 2.0 BS01 VRX A 1 L419 R422 M423 H475 S476 Y477 I482 V485 A486 L497 W528 L414 R417 M418 H470 S471 Y472 I477 V480 A481 L492 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=3uM remove_due_to_license_issue P26663 16934455 600 HHSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSL 2hwo A 2.5 BS01 RBS A 1 V281 G344 C345 L393 D404 V26 G80 C81 L129 D140 D386 R388 A390 N391 D404 D122 R124 A126 N127 D140 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 17334377 1345 LAKDAWEIPRESLRLEVKLGGCFGEVWMGTWNGTTRVAIKTLKPFLQEAQVMKKLRHEKLVQLYAVVSPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2hwp A 2.48 BS01 DJK A 1 A293 K295 I336 C345 L393 D404 A35 K37 I66 C75 L123 D134 D386 R388 A390 N391 D404 F424 D116 R118 A120 N121 D134 F136 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>27000nM P00523 17334377 1345 AKDAWEIPRESLRVKLGQGCGEVWMGTWNGTTRVAIKTFLQAQVMKKLRHEKLVQLYAVVSEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2hxl A 1.8 BS01 422 A 1 T14 L15 A36 L84 C87 G90 L137 T13 L14 A35 L80 C83 G86 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=12nM remove_due_to_license_issue IC50=12nM O14757 16990002 324 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP 2hxm A 1.3 BS01 302 A 1 G143 Q144 D145 Y147 C157 F158 S169 N204 G246 S247 Y248 H268 S270 G62 Q63 D64 Y66 C76 F77 S88 N123 G165 S166 Y167 H187 S189 D145 Y147 F158 H268 D64 Y66 F77 H187 3.2.2.27 0004844,0006281,0006284,0016799 remove_due_to_license_issue P13051 17062624 401 MEFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPLSVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 2hxq A 2.0 BS01 373 A 1 Q13 L15 A36 L84 E85 Y86 C87 G90 L137 Q12 L14 A35 L80 E81 Y82 C83 G86 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=144nM remove_due_to_license_issue IC50=140nM O14757 16990002 324 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP 2hy0 A 1.7 BS01 306 A 1 Q13 L15 V23 A36 K38 E85 Y86 C87 G90 L137 D148 Q12 L14 V22 A35 K37 E77 Y78 C79 G82 L129 D140 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.65nM remove_due_to_license_issue IC50=0.650000nM, EC50=97nM O14757 16990002 324 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2hyy A 2.4 BS01 STI A 1 L248 Y253 A269 K271 E286 V289 M290 T315 F317 M318 I360 H361 L370 A380 D381 F382 L14 Y19 A35 K37 E51 V54 M55 T80 F82 M83 I125 H126 L135 A145 D146 F147 D363 A365 R367 N368 D381 P402 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0005524,0006468 ic50=170nM remove_due_to_license_issue IC50=38nM, Kd=44nM, Ki=13nM, EC50=7e+1nM P00519 17164530 600 WEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ 2hz0 A 2.1 BS01 GIN A 1 A269 K271 E286 M290 I313 T315 F317 H361 L370 A380 D381 F382 S385 A37 K39 E54 M58 I81 T83 F85 H129 L138 A148 D149 F150 S153 D363 A365 R367 N368 D381 P402 D131 A133 R135 N136 D149 P170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=330nM remove_due_to_license_issue P00519 17164530 600 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMF 2hz4 A 2.8 BS01 4ST A 1 W261 Y264 L266 K294 L302 W23 Y26 L28 K56 L64 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hz4 A 2.8 BS02 4ST C 1 Y342 F497 Q498 S500 Y104 F259 Q260 S262 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hzi A 1.7 BS01 JIN A 1 Y253 V256 A269 K271 T315 M318 Y320 G321 L370 A380 D381 F382 Y21 V24 A37 K39 T83 M86 Y88 G89 L138 A148 D149 F150 D363 A365 R367 N368 D381 P402 D131 A133 R135 N136 D149 P170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=70nM remove_due_to_license_issue P00519 17164530 600 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hzl A 1.4 BS02 PYR A 1 Y99 Y100 Q156 R177 W215 Y68 Y69 Q125 R146 W184 ? 0015849,0031317,0043177,0055085 Kd=270nM remove_due_to_license_issue Q3J1R2 17362499 601 VTWRLASSFPKSLDTIFGGAEVLSKMLSEATDGNFQIQVFSAGELVPGLQAADAVTEGTVECCHTVGYYYWGKDPTFALAAAVPFSLSARGINAWHYHGGGIDLYNEFLSQHNIVAFPGGNTGVQMGGWFRREINTVADMQGLKMRVGGFAGKVMERLGVVPQQIAGGDIYPALEKGTIDATEWVGPYDDEKLGFFKVAPYYYYPGWWEGGPTVHFMFNKSAYEGLTPTYQSLLRTACHAADANMLQLYDWKNPTAIKSLVAQGTQLRPFSPEILQACFEAANEVYAEMEASNPAFKKIWDSIKAFRSEHYTWAQIAEYNYDTFMMVQQNAGKL 2hzn A 2.7 BS01 KIN A 1 A269 E286 M290 T315 E316 F317 M318 L370 V379 A380 D381 S501 A42 E57 M61 T86 E87 F88 M89 L141 V150 A151 D152 S272 D363 A365 R367 N368 D381 P402 D134 A136 R138 N139 D152 P173 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 17164530 600 MDPSSPNYDKWEMERTDITMKHKLGGGEVYEGVWKKYSLTVAVKTLDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESS 2i03 B 2.4 BS01 AXD B 1 H126 E205 E206 Y547 S630 Y631 Y662 Y666 N710 V711 H88 E167 E168 Y509 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 17034148 1630 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2i0a A 1.8 BS01 MUI A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=0.004nM remove_due_to_license_issue O38723 17149864 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2i0a B 1.8 BS01 MUI A 1 R8 D25 A28 D30 P81 V82 R8 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38723 17149864 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2i0d A 1.95 BS01 MUT A 1 D25 G27 D29 G48 I50 D25 G27 D29 G48 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=0.0008nM remove_due_to_license_issue O38731 17149864 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2i0d B 1.95 BS01 MUT A 1 R8 D25 A28 D30 P81 V82 R8 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38731 17149864 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2i0e A 2.6 BS01 PDS A 1 L348 F353 V356 A369 T404 Y422 V423 D470 M473 A483 D484 L10 F15 V18 A31 T66 Y84 V85 D132 M135 A145 D146 D466 K468 D470 N471 D484 T504 D128 K130 D132 N133 D146 T166 2.7.11.13 0004672,0004674,0004697,0005524,0006468 remove_due_to_license_issue P05771 17115692 901 LTDFNFLMVLGKGSFGKVMLSERKGTDELYAVKILKKDVVIQDDDVECTMVEKRVLALPGKPPFLTQLHSCFQTMDRLYFVMEYVNGGDLMYHIQQVGRFKEPHAVFYAAEIAIGLFFLQSKGIIYRDLKLDNVMLDSEGHIKIADFGMCKENIWDGVTTKTFCGTPDYIAPEIIAYQPYGKSVDWWAFGVLLYEMLAGQAPFEGEDEDELFQSIMEHNVAYPKSMSKEAVAICKGLMTKHPGKRLGCGPEGERDIKEHAFFRYIDWEKLERKEIQPPYKPKACGRENFDRFFTRHPPVLTPPDQEVIRNIDQSEFEGFSFVNSEFLKP 2i0g A 2.5 BS01 I0G A 1 M295 E305 L339 H475 L476 M29 E39 L73 H202 L203 ? 0003677,0004879,0006355 Ki=0.19nM remove_due_to_license_issue Ki=0.19nM, EC50=0.66nM Q92731 17034120 1 DALSPEQLVLTLLEAEPPHVLISRPASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKVPVYDLLLEMLNAH 2i0h A 2.0 BS01 222 A 1 Y35 V38 A51 K53 L104 T106 L108 M109 G110 A111 D112 S154 Y32 V35 A48 K50 L101 T103 L105 M106 G107 A108 D109 S151 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=9nM remove_due_to_license_issue Q16539 16945533 400 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2i0h A 2.0 BS02 222 A 2 Y35 V38 A51 T106 M109 G110 D112 S154 Y32 V35 A48 T103 M106 G107 D109 S151 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=9nM remove_due_to_license_issue Q16539 16945533 3400 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2i0j A 2.9 BS01 I0G A 1 E353 L384 R394 F404 M421 I424 H524 E48 L79 R89 F99 M116 I119 H217 ? remove_due_to_license_issue Ki=2.7nM, EC50=19.4nM P03372 17034120 1 LALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSM 2i0v A 2.8 BS01 6C3 A 1 L588 A614 K616 T663 E664 Y665 C666 L785 F797 A800 L45 A71 K73 T120 E121 Y122 C123 L173 F185 A188 D778 A780 R782 N783 D796 N805 D166 A168 R170 N171 D184 N193 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=160nM P07333 17132624 1000 PKYQVRWKIIESYEGNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKRQLSSRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQAQE 2i0y A 1.9 BS01 5CN A 1 L588 V596 A614 K616 T663 Y665 C666 G669 L785 F797 A800 R801 L31 V39 A57 K59 T106 Y108 C109 G112 L159 F171 A174 R175 D778 A780 R782 N783 D796 N805 D152 A154 R156 N157 D170 N179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=24nM P07333 17132624 1000 VRWKIIESYESYTFIEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKRQLSSRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQAQE 2i19 A 2.28 BS03 1BY A 1 Y99 L100 D103 R112 T168 Q172 K212 K269 Y99 L100 D103 R112 T168 Q172 K212 K269 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 remove_due_to_license_issue Q86C09 17090032 3001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSLSPNNNGEEDDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 2i19 B 2.28 BS03 1BY B 1 Y99 D103 R112 Q172 K212 Y93 D97 R106 Q166 K206 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H92 D97 D101 R106 D169 K206 F245 D249 D250 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 remove_due_to_license_issue Q86C09 17090032 4001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSLSEDDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 2i1m A 1.8 BS01 5CN A 1 L588 G589 V596 V647 T663 Y665 C666 C667 G669 L785 F797 L40 G41 V48 V99 T115 Y117 C118 C119 G121 L175 F187 D778 A780 R782 N783 D796 N805 N814 D168 A170 R172 N173 D186 N195 N204 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=24nM P07333 17132624 1000 QVRWKIIESYNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKSRVLETDSTASTRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGNARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQAQEDRRER 2i1r A 2.2 BS01 VXR A 1 L419 R422 M423 S476 Y477 I482 W528 K533 L414 R417 M418 S471 Y472 I477 W523 K528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=9.7uM remove_due_to_license_issue P26663 17049849 600 HHSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSL 2i2b A 2.1 BS01 CC5 A 1 N122 E123 Y163 S166 N118 E119 Y159 S162 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 17686780 273 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIE 2i2b A 2.1 BS02 CC5 A 2 D45 F74 Y75 N122 T161 A162 D45 F74 Y75 N118 T157 A158 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 17686780 274 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIE 2i2c A 1.85 BS01 DTA A 1 D45 F74 Y75 N122 E123 T161 A162 Y163 S166 D45 F74 Y75 N122 E123 T161 A162 Y163 S166 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=0.02mM remove_due_to_license_issue Q8Y8D7 17686780 273 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIGKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 2i3i A 2.3 BS02 618 A 1 K121 V122 R123 G130 L131 Q132 S133 W134 D138 E143 W147 F148 K44 V45 R46 G53 L54 Q55 S56 W57 D61 E66 W70 F71 F81 F4 2.3.2.27 Ki=0.05uM remove_due_to_license_issue Q96CA5 17168540 501 GPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQDKVRCFFCYGGLQSWKRGDDPWTEHAKWFPGCQFLLRSKGQEYINNIH 2i3v A 2.4 BS02 GLU A 1 Y61 L90 T91 R96 G141 S142 T143 E193 Y59 L88 T89 R94 G139 S140 T141 E191 ? 0015276,0016020 remove_due_to_license_issue P19491 17018279 401 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGCNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 2i3z A 2.9 BS01 LIR A 1 E203 E204 F355 Y548 S631 Y632 Y663 Y667 E166 E167 F318 Y511 S594 Y595 Y626 Y630 Y548 S631 Y632 D709 H741 Y511 S594 Y595 D672 H704 3.4.14.5 0001618,0001662,0001666,0002020,0002337,0002709,0002717,0004177,0004252,0005102,0005518,0005576,0005886,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016324,0030027,0030139,0030163,0031258,0031295,0033632,0035641,0036343,0042110,0042277,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 remove_due_to_license_issue P14740 17010607 900 RRTYTLADYLKNTFRVKSYSLRWVSDSEYLYKQENNILLFNAEHGNSSIFLENSTFEIFGDSISDYSVSPDRLFVLLEYNYVKQWRHSYTASYSIYDLNKRQLITEEKIPNNTQWITWSQEGHKLAYVWKNDIYVKIEPHLPSHRITSTGKENVIFNGINDWVYEEEIFGAYSALWWSPNGTFLAYAQFNDTGVPLIEYSFYSDESLQYPKTVWIPYPKAGAVNPTVKFFIVNTDSLSSTTTTIPMQITAPASVTTGDHYLCDVAWVSEDRISLQWLRRIQNYSVMAICDYDKTTLVWNCPTTQEHIETSATGWCGRFRPAEPHFTSDGSSFYKIVSDKDGYKHICQFQKDRKPEQVCTFITKGAWEVISIEALTSDYLYYISNEYKEMPGGRNLYKIQLTDHTNKKCLSCDLNPERCQYYSVSLSKEAKYYQLGCRGPGLPLYTLHRSTDQKELRVLEDNSALDKMLQDVQMPSKKLDFIVLNETRFWYQMILPPHFDKSKKYPLLIDVYAGPCSQKADAAFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINKRLGTLEVEDQIEAARQFLKMGFVDSKRVAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDAGVDFQAMWYTDEDHGIASSTAHQHIYSHMSHFLQQCFSLR 2i40 A 2.8 BS01 BLZ A 1 I10 V18 A31 F80 F82 L83 H84 N132 L134 D145 I10 V18 A31 F77 F79 L80 H81 N129 L131 D142 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 16997559 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 2i4d A 1.5 BS01 QFI B 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q5RZ08 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGMTLNF 2i4d B 1.5 BS01 QFI B 1 D225 G227 A228 D229 D230 G248 G249 I250 F253 D25 G27 A28 D29 D30 G48 G49 I50 F53 D225 T226 G227 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=2.1pM remove_due_to_license_issue Q5RZ08 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGMTLNF 2i4j A 2.1 BS01 DRJ A 1 F226 C285 S289 A292 I296 H323 I326 M329 V339 I341 H449 L453 L469 Y473 F20 C79 S83 A86 I90 H117 I120 M123 V133 I135 H243 L247 L263 Y267 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Ki=88nM, Kd=270nM, EC50=73.3nM P37231 17403688 999 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2i4p A 2.1 BS01 DRH A 1 F226 F282 C285 Q286 R288 S289 I296 H323 I326 M329 L330 H449 Y473 F20 F76 C79 Q80 R82 S83 I90 H117 I120 M123 L124 H243 Y267 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Ki=971nM, Kd=1978nM, EC50=590nM P37231 17403688 999 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2i4u A 1.5 BS01 DJR A 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 3.4.23.16 0004190,0006508,0042802 Ki=2.7pM remove_due_to_license_issue Q7SSI0 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGMTLNF 2i4u B 1.5 BS01 DJR A 1 D225 G227 A228 D229 G248 I250 D25 G27 A28 D29 G48 I50 D225 T226 G227 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGMTLNF 2i4v A 1.5 BS01 DJR B 1 D25 A28 D30 I50 P81 V82 D25 A28 D30 I50 P81 V82 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q903J0 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLMTQIGMTLNF 2i4v B 1.5 BS01 DJR B 1 D225 G227 A228 D229 G248 I250 D25 G27 A28 D29 G48 I50 D225 T226 G227 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=6.3pM remove_due_to_license_issue Q903J0 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLMTQIGMTLNF 2i4w A 1.55 BS01 KGQ B 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 3.4.23.16 0004190,0006508 remove_due_to_license_issue O92139 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGMTLNF 2i4w B 1.55 BS01 KGQ B 1 D225 G227 A228 D229 G248 G249 I250 G252 F253 D25 G27 A28 D29 G48 G49 I50 G52 F53 D225 T226 G227 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=2.6pM remove_due_to_license_issue O92139 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGMTLNF 2i4x A 1.55 BS01 KGQ B 1 D25 G27 A28 D30 G49 P81 V82 D25 G27 A28 D30 G49 P81 V82 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q903J0 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLMTQIGMTLNF 2i4x B 1.55 BS01 KGQ B 1 D225 G227 A228 D229 G248 G249 I250 G252 F253 D25 G27 A28 D29 G48 G49 I50 G52 F53 D225 T226 G227 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=1.9pM remove_due_to_license_issue Q903J0 16979654 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLMTQIGMTLNF 2i4z A 2.25 BS01 DRH A 1 F282 C285 Q286 S289 A292 I296 I326 M329 L330 I341 M364 H449 L453 Y473 F76 C79 Q80 S83 A86 I90 I120 M123 L124 I135 M158 H243 L247 Y267 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Ki=971nM, Kd=1978nM, EC50=590nM P37231 17403688 999 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2i5f A 1.35 BS01 5IP A 1 K253 G255 H256 R257 R258 R264 Y277 K13 G15 H16 R17 R18 R24 Y37 ? ic50=2.2uM remove_due_to_license_issue P08567 18034889 550 FTGVIIKQGCLLKQGHRRKNWKVRKFILREDPAYLHYYDPAGAEDPLGAIHLRGCVVTSVESEENLFEIITADEVHYFLQAATPKERTEWIKAIQMASR 2i5j A 3.15 BS04 K05 A 1 V108 D186 L187 Y188 K223 L228 W229 V108 D186 L187 Y188 K223 L228 W229 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 17184135 4001 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 2i6a A 2.2 BS01 5I5 A 1 N14 D18 I39 G64 S65 C123 L134 F170 N12 D16 I37 G62 S63 C121 L132 F168 R132 G297 A298 G299 D300 R130 G295 A296 G297 D298 2.7.1.20 0003723,0004001,0004136,0005524,0005634,0005654,0005737,0005829,0005886,0006144,0006166,0006175,0006753,0009156,0016301,0032263,0034654,0044209,0046872,0106383 ic50=0.9nM remove_due_to_license_issue IC50=9.0nM P55263 17154503 500 SVRENILFGMGNPLLDISAVVDKDFLDKYSLKPNDQILAEDKHKELFDELVKKFKVEYHAGGSTQNSIKVAQWMIQQPHKAATFFGCIGIDKFGEILKRKAAEAHVDAHYYEQNEQPTGTCAACITGDNRSLIANLAAANCYKKEKHLDLEKNWMLVEKARVCYIAGFFLTVSPESVLKVAHHASENNRIFTLNLSAPFISQFYKESLMKVMPYVDILFGNETEAATFAREQGFETKDIKEIAKKTQALPKMNSKRQRIVIFTQGRDDTIMATESEVTAFAVLDQDQKEIIDTNGAGDAFVGGFLSQLVSDKPLTECIRAGHYAASIIIRRTGCTFPEKPDFH 2i6b A 2.3 BS01 89I A 1 N14 Q38 I39 L40 G64 S65 A136 L138 F170 F201 Y206 N13 Q37 I38 L39 G63 S64 A135 L137 F169 F200 Y205 R132 G297 A298 G299 D300 R131 G296 A297 G298 D299 2.7.1.20 0003723,0004001,0004136,0005524,0005634,0005654,0005737,0005829,0005886,0006144,0006166,0006175,0006753,0009156,0016301,0032263,0034654,0044209,0046872,0106383 ic50=68nM remove_due_to_license_issue IC50=68nM P55263 17154503 500 TSVRENILFGMGNPLLDISAVVDKDFLDKYSLKPNDQILAEDKHKELFDELVKKFKVEYHAGGSTQNSIKVAQWMIQQPHKAATFFGCIGIDKFGEILKRKAAEAHVDAHYYEQNEQPTGTCAACITGDNRSLIANLAAANCYKKEKHLDLEKNWMLVEKARVCYIAGFFLTVSPESVLKVAHHASENNRIFTLNLSAPFISQFYKESLMKVMPYVDILFGNETEAATFAREQGFETKDIKEIAKKTQALPKMNSKRQRIVIFTQGRDDTIMATESEVTAFAVLDQDQKEIIDTNGAGDAFVGGFLSQLVSDKPLTECIRAGHYAASII 2i72 A 2.2 BS01 VA1 A 1 S64 D123 Y150 N152 Y221 G317 A318 S61 D120 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 17956081 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2i7c A 1.71 BS01 AAT A 1 Q54 H64 G85 G86 D88 E108 I109 D139 A140 D157 S158 S159 D160 P164 A165 L168 Y225 Q53 H63 G84 G85 D87 E107 I108 D138 A139 D156 S157 S158 D159 P163 A164 L167 Y224 2.5.1.16 0003824 ic50=8.5uM remove_due_to_license_issue Q8II73 17822713 801 KKWFSEFSIMWPGQAFSLKIKKILYETKSKYQNVLVFESTTYGKVLVLDGVIQLTEKDEFAYHEMMTHVPMTVSKEPKNVLVVGGGDGGIIRELCKYKSVENIDICEIDETVIEVSKIYFKNISCGYEDKRVNVFIEDASKFLENVTNTYDVIIVDSSDPIGPAETLFNQNFYEKIYNALKPNGYCVAQCESLWIHVGTIKNMIGYAKKLFKKVEYANISIPTYPCGCIGILCCSKTDTGLTKPNKKLESKEFADLKYYNYENHSAAFKLPAFLLKEIENI 2i91 A 2.65 BS01 rna C 0 K172 Q173 K236 L259 K160 Q161 K219 L242 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 17041599 1 ~ 8 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNRGKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 2i91 A 2.65 BS02 rna D 0 K88 R120 T123 M166 K170 Y171 R174 R252 R255 T260 P277 L278 T279 A280 L282 R283 L285 G286 K287 K316 A317 R318 V326 A327 T330 G336 N337 R338 G339 L341 K84 R116 T119 M154 K158 Y159 R162 R235 R238 T243 P260 L261 T262 A263 L265 R266 L268 G269 K270 K299 A300 R301 V309 A310 T313 G319 N320 R321 G322 L324 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 17041599 2 ~ 15 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNRGKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 2i91 B 2.65 BS01 rna E 0 Q173 R174 K236 R237 L259 T260 Q162 R163 K225 R226 L248 T249 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 17041599 1 ~ 8 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNRGKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 2i91 B 2.65 BS02 rna F 0 K88 R120 T123 K170 Y171 R174 R252 R255 T260 K264 T279 A280 L282 R283 L285 G286 K287 K316 A317 R318 V326 A327 T330 G336 N337 R338 G339 L341 K84 R116 T119 K159 Y160 R163 R241 R244 T249 K253 T268 A269 L271 R272 L274 G275 K276 K305 A306 R307 V315 A316 T319 G325 N326 R327 G328 L330 ? 0003723,0005737,0030030,0034336,0046872,1990904 remove_due_to_license_issue P42700 17041599 1 ~ 15 MDQTQPLNEKQVPNSEGCYVWQVSDMNRLRRFLCFGSEGGTYYIEEKKLGQENAEALLRLIEDGKGCEVVQEIKTFSQEGRAAKQEPTLFALAVCSQCSDIKTKQAAFRAVPEVCRIPTHLFTFIQFKKDLKWGRALRKAVSDWYNTKDALNLAMAVTKYKQRNGWSHKDLLRLSHIKPANEGLTMVAKYVSKGWKEVQEAYKEKELSPETEKVLKYLEATERVKRTKDELEIIHLIDEYRLVREHLLTIHLKSKEIWKSLLQDMPLTALLRNLGKMTADSVLAPASSEVSSVCERLTNEKLLKKARIHPFHILVALETYKKGHGNRGKLRWIPDTSIVEALDNAFYKSFKLVEPTGKRFLLAIDVSASMNQRVLGSILNASVVAAAMCMLVARTEKDSHMVAFSDEMLPCPITVNMLLHEVVEKMSDITMGSTDCALPMLWAQKTNTAADIFIVFTDCETNVEDVHPATALKQYREKMGIPAKLIVCAMTSNGFSIADPDDRGMLDICGFDSGALDVIRNFTLDL 2i9k A 2.65 BS01 dna C 0 Y44 I86 Q90 N123 K234 G236 Q237 G256 G257 S294 Q297 Y44 I86 Q90 N123 K234 G236 Q237 G256 G257 S294 Q297 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 16919299 402 ~ 413 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNAASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAITLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 2i9k A 2.65 BS02 dna D 0 F79 C81 Q82 S85 I86 S87 G88 R97 E119 V121 K162 R165 R228 Q237 R240 Y242 I249 T250 S252 A253 Y254 G255 G256 N304 F79 C81 Q82 S85 I86 S87 G88 R97 E119 V121 K162 R165 R228 Q237 R240 Y242 I249 T250 S252 A253 Y254 G255 G256 N304 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 16919299 421 ~ 433 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNAASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAITLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 2ibs A 2.4 BS01 dna B 0 V21 N105 Y108 K116 K139 T167 L171 D173 F196 K199 K200 F268 R271 R323 H394 V1 N85 Y88 K96 K119 T147 L151 D153 F176 K179 K180 F248 R251 R303 H374 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 1 ~ 10 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibs A 2.4 BS02 dna C 0 G112 E113 K116 Y117 K126 K130 R271 S272 G295 R296 T336 K337 R353 E354 P393 G92 E93 K96 Y97 K106 K110 R251 S252 G275 R276 T316 K317 R333 E334 P373 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 11 ~ 20 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibs D 2.4 BS01 dna E 0 V21 N105 Y108 K139 T167 L171 D173 F196 K199 K200 F268 R271 H394 V1 N85 Y88 K119 T147 L151 D153 F176 K179 K180 F248 R251 H374 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 1 ~ 10 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibs D 2.4 BS02 dna F 0 G112 E113 K116 Y117 K126 K130 G138 R271 S272 K276 G295 R296 T336 K337 R353 E354 P393 G92 E93 K96 Y97 K106 K110 G118 R251 S252 K256 G275 R276 T316 K317 R333 E334 P373 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 11 ~ 20 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibt A 1.7 BS01 dna B 0 V21 N105 Y108 K139 T167 L171 E172 D173 F196 K199 K200 F268 R271 R323 H394 V1 N85 Y88 K119 T147 L151 E152 D153 F176 K179 K180 F248 R251 R303 H374 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 1 ~ 10 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibt A 1.7 BS02 dna C 0 G112 E113 K116 Y117 K126 K130 R271 S272 G295 R296 T336 K337 R353 E354 G92 E93 K96 Y97 K106 K110 R251 S252 G275 R276 T316 K317 R333 E334 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 11 ~ 20 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibt D 1.7 BS01 dna E 0 V21 N105 Y108 K139 T167 L171 E172 D173 F196 K199 K200 R267 F268 R271 H394 V1 N85 Y88 K119 T147 L151 E152 D153 F176 K179 K180 R247 F248 R251 H374 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 1 ~ 10 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ibt D 1.7 BS02 dna F 0 G112 E113 K116 Y117 K126 K130 G138 R271 S272 K276 G295 R296 T336 K337 R353 E354 G92 E93 K96 Y97 K106 K110 G118 R251 S252 K256 G275 R276 T316 K317 R333 E334 2.1.1.72 0003676,0003677,0006304,0008168,0009007,0009307,0032259 remove_due_to_license_issue P14385 17455934 11 ~ 20 VETPPEVVDFMVSLAEAPRGGRVLEPACAHGPFLRAFREAHGTAYRFVGVEIDPKALDLPPWAEGILADFLLWEPGEAFDLILGNPPYGIVGEASKYPIHVFKAVKDLYKKAFSTWKGKYNLYGAFLEKAVRLLKPGGVLVFVVPATWLVLEDFALLREFLAREGKTSVYYLGEVFPQKKVSAVVIRFQKSGKGLSLWDTQESESGFTPILWAEYPHWEGEIIRFETEETRKLEISGMPLGDLFHIRFAARSPEFKKHPAVRKEPGPGLVPVLTGRNLKPGWVDYEKNHSGLWMPKERAKELRDFYATPHLVVAHTKGTRVVAAWDERAYPWREEFHLLPKEGVRLDPSSLVQWLNSEAMQKHVRTLYRDFVPHLTLRMLERLPVRREYGFHT 2ica A 1.56 BS01 2IC A 1 V157 Y166 I235 I255 Y257 I259 K287 L302 I306 V30 Y39 I108 I128 Y130 I132 K160 L175 I179 ? ic50=20nM remove_due_to_license_issue IC50=20nM P20701 17125246 1 MNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKRKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKI 2idk A 2.55 BS01 C2F B 1 L207 M215 L203 M211 Y21 G137 H142 R175 Y194 Y20 G136 H141 R174 Y193 2.1.1.20 0005542,0005737,0005829,0005977,0006111,0006544,0006555,0006730,0008168,0008757,0016594,0017174,0032259,0034708,0042802,0046498,0046500,0051289,0098603,1901052,1904047 remove_due_to_license_issue P13255 17158459 1420 DSVYRTRSLGVAAEGIPDQYADGEAARVWQLYIGDTRSRTAEYKAWLLGLLRQHGCHRVLDVACGTGVDSIMLVEEGFSVTSVDASDKMLKYALKERWNRRKEPAFDKWVIEEANWLTLDKDVPAGDGFDAVICLGNSFAHLPDSKGDQSEHRLALKNIASMVRPGGLLVIDHRNYDYILSTGCAPPGKNIYYKSKDITTSVLTVNNKAHMVTLDYTVQFSKFRLSYYPHCLASFTELVQEAFGGRCQHSVLGDFKPYRPGQAYVPCYFIHVLKKTG 2idk B 2.55 BS01 C2F A 1 L207 M215 R239 L207 M215 R232 Y21 G137 H142 R175 Y194 Y21 G137 H142 R175 Y194 2.1.1.20 0005542,0005737,0005829,0005977,0006111,0006544,0006555,0006730,0008168,0008757,0016594,0017174,0032259,0034708,0042802,0046498,0046500,0051289,0098603,1901052,1904047 remove_due_to_license_issue P13255 17158459 1410 VDSVYRTRSLGVAAEGIPDQYADGEAARVWQLYIGDTRSRTAEYKAWLLGLLRQHGCHRVLDVACGTGVDSIMLVEEGFSVTSVDASDKMLKYALKERWNRRKEPAFDKWVIEEANWLTLDKDVPAGDGFDAVICLGNSFAHLPDSKGDQSEHRLALKNIASMVRPGGLLVIDHRNYDYILSTGCAPPGKNIYYKSDLTKDITTSVLTVNNKAHMVTLDYTVQVPGAFSKFRLSYYPHCLASFTELVQEAFGGRCQHSVLGDFKPYRPGQAYVPCYFIHVLKKTG 2idk B 2.55 BS02 C2F B 1 S3 Y5 S3 Y5 Y21 G137 H142 R175 Y194 Y21 G137 H142 R175 Y194 2.1.1.20 0005542,0005737,0005829,0005977,0006111,0006544,0006555,0006730,0008168,0008757,0016594,0017174,0032259,0034708,0042802,0046498,0046500,0051289,0098603,1901052,1904047 remove_due_to_license_issue P13255 17158459 1420 VDSVYRTRSLGVAAEGIPDQYADGEAARVWQLYIGDTRSRTAEYKAWLLGLLRQHGCHRVLDVACGTGVDSIMLVEEGFSVTSVDASDKMLKYALKERWNRRKEPAFDKWVIEEANWLTLDKDVPAGDGFDAVICLGNSFAHLPDSKGDQSEHRLALKNIASMVRPGGLLVIDHRNYDYILSTGCAPPGKNIYYKSDLTKDITTSVLTVNNKAHMVTLDYTVQVPGAFSKFRLSYYPHCLASFTELVQEAFGGRCQHSVLGDFKPYRPGQAYVPCYFIHVLKKTG 2idk C 2.55 BS01 C2F A 1 S3 Y5 S3 Y5 Y21 G137 H142 R175 Y194 Y21 G137 H142 R175 Y194 2.1.1.20 0005542,0005737,0005829,0005977,0006111,0006544,0006555,0006730,0008168,0008757,0016594,0017174,0032259,0034708,0042802,0046498,0046500,0051289,0098603,1901052,1904047 remove_due_to_license_issue P13255 17158459 1410 VDSVYRTRSLGVAAEGIPDQYADGEAARVWQLYIGDTRSRTAEYKAWLLGLLRQHGCHRVLDVACGTGVDSIMLVEEGFSVTSVDASDKMLKYALKERWNRRKEPAFDKWVIEEANWLTLDKDVPAGDGFDAVICLGNSFAHLPDSKGDQSEHRLALKNIASMVRPGGLLVIDHRNYDYILSTGCAPPGKNIYYKSDLTKDITTSVLTVNNKAHMVTLDYTVQFSKFRLSYYPHCLASFTELVQEAFGGRCQHSVLGDFKPYRPGQAYVPCYFIHVLKKTG 2idk C 2.55 BS02 C2F B 1 L207 M215 R239 L207 M215 R228 Y21 G137 H142 R175 Y194 Y21 G137 H142 R175 Y194 2.1.1.20 0005542,0005737,0005829,0005977,0006111,0006544,0006555,0006730,0008168,0008757,0016594,0017174,0032259,0034708,0042802,0046498,0046500,0051289,0098603,1901052,1904047 remove_due_to_license_issue P13255 17158459 1420 VDSVYRTRSLGVAAEGIPDQYADGEAARVWQLYIGDTRSRTAEYKAWLLGLLRQHGCHRVLDVACGTGVDSIMLVEEGFSVTSVDASDKMLKYALKERWNRRKEPAFDKWVIEEANWLTLDKDVPAGDGFDAVICLGNSFAHLPDSKGDQSEHRLALKNIASMVRPGGLLVIDHRNYDYILSTGCAPPGKNIYYKSDLTKDITTSVLTVNNKAHMVTLDYTVQFSKFRLSYYPHCLASFTELVQEAFGGRCQHSVLGDFKPYRPGQAYVPCYFIHVLKKTG 2idk D 2.55 BS01 C2F A 1 L207 H214 M215 L207 H214 M215 Y21 G137 H142 R175 Y194 Y21 G137 H142 R175 Y194 2.1.1.20 0005542,0005737,0005829,0005977,0006111,0006544,0006555,0006730,0008168,0008757,0016594,0017174,0032259,0034708,0042802,0046498,0046500,0051289,0098603,1901052,1904047 remove_due_to_license_issue P13255 17158459 1410 VDSVYRTRSLGVAAEGIPDQYADGEAARVWQLYIGDTRSRTAEYKAWLLGLLRQHGCHRVLDVACGTGVDSIMLVEEGFSVTSVDASDKMLKYALKERWNRRKEPAFDKWVIEEANWLTLDKDVPAGDGFDAVICLGNSFAHLPDSKGDQSEHRLALKNIASMVRPGGLLVIDHRNYDYILSTGCAPPGKNIYYKSDLTKDITTSVLTVNNKAHMVTLDYTVQVPGAPGFSKFRLSYYPHCLASFTELVQEAFGGRCQHSVLGDFKPYRPGQAYVPCYFIHVLKKTG 2idw A 1.1 BS01 017 B 1 D25 I47 G48 P81 I84 D25 I47 G48 P81 I84 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 15066436 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2idw B 1.1 BS01 017 B 1 D125 G127 A128 D129 D130 G148 I150 D25 G27 A28 D29 D30 G48 I50 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=1.3nM remove_due_to_license_issue Q7SSI0 15066436 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2ie4 C 2.6 BS03 OKA C 1 R89 H118 Y127 H191 W200 R214 L243 Y265 R84 H113 Y122 H186 W195 R209 L238 Y260 H167 H162 3.1.3.16 0000159,0000278,0000775,0000922,0001932,0004721,0004722,0004725,0005515,0005634,0005694,0005737,0005739,0005829,0005856,0005886,0006338,0006357,0006470,0007498,0008287,0010288,0010719,0015630,0016020,0016787,0017018,0033192,0035331,0035556,0035970,0040008,0043029,0045121,0045202,0045595,0046872,0046982,0048156,0050811,0051321,0051898,0070062,0070262,0071902,0090443,0140791,0180004,0180005,0180006,0180007,0180008,1900227,1904528,1904539,1990439,2000045 remove_due_to_license_issue IC50=7nM P67775 17055435 401 FTKELDQWIEQLNECKQLSESQVKSLCEKAKEILTKESNVQEVRCPVTVCGDVHGQFHDLMELFRIGGKSPDTNYLFMGDYVDRGYYSVETVTLLVALKVRYRERITILRGNHESRQITQVYGFYDECLRKYGNANVWKYFTDLFDYLPLTALVDGQIFCLHGGLSPSIDTLDHIRALDRLQEVPHEGPMCDLLWSDPDDRGGWGISPRGAGYTFGQDISETFNHANGLTLVSRAHQLVMEGYNWCHDRNVVTIFSAPNYCYRCGNQAAIMELDDTLKYSFLQFDPAP 2ieh A 2.7 BS02 MOY A 1 E116 G117 E118 R119 W127 A133 P137 L160 Y211 L214 E215 A218 R221 E102 G103 E104 R105 W113 A119 P123 L146 Y197 L200 E201 A204 R207 3.6.4.4 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=150nM P52732 17251189 602 KGKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 2ien A 1.3 BS01 017 B 1 D25 G27 A28 D30 V32 V82 I84 D25 G27 A28 D30 V32 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 15066436 402 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2ien B 1.3 BS01 017 B 1 D125 G127 A128 D129 G148 G149 I150 D25 G27 A28 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1nM remove_due_to_license_issue P03367 15066436 402 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2ieo A 1.53 BS01 017 A 1 D25 A28 D30 V32 V82 D25 A28 D30 V32 V82 3.4.23.16 0004190,0006508,0042802 Ki=3.2nM remove_due_to_license_issue Q7SSI0 15066436 402 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2ieo B 1.53 BS01 017 A 1 D125 G127 A128 D129 G148 G149 I150 D25 G27 A28 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 15066436 402 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2igv A 1.67 BS01 SER A 1 A108 N109 H133 A108 N109 H133 R62 F67 Q70 N109 F120 L129 H133 R62 F67 Q70 N109 F120 L129 H133 5.2.1.8 0000413,0003755,0005515,0005634,0005737,0005739,0006357,0006457,0016018,0140839,0140840 remove_due_to_license_issue P52011 17654646 201 MSRSKVFFDITIGGKASGRIVMELYDDVVPKTAGNFRALCTGENGIGKSGKPLHFKGSKFHRIIPNFMIQGGDFTRGNGTGGESIYGEKFPDENFKEKHTGPGVLSMANAGPNTNGSQFFLCTVKTEWLDGKHVVFGRVVEGLDVVKAVESNGSQSGKPVKDCMIADCGQLK 2igv A 1.67 BS02 PRO A 1 R62 Q70 F120 H133 R62 Q70 F120 H133 R62 F67 Q70 N109 F120 L129 H133 R62 F67 Q70 N109 F120 L129 H133 5.2.1.8 0000413,0003755,0005515,0005634,0005737,0005739,0006357,0006457,0016018,0140839,0140840 remove_due_to_license_issue P52011 17654646 202 MSRSKVFFDITIGGKASGRIVMELYDDVVPKTAGNFRALCTGENGIGKSGKPLHFKGSKFHRIIPNFMIQGGDFTRGNGTGGESIYGEKFPDENFKEKHTGPGVLSMANAGPNTNGSQFFLCTVKTEWLDGKHVVFGRVVEGLDVVKAVESNGSQSGKPVKDCMIADCGQLK 2igw A 1.78 BS02 PRO A 1 R62 Q70 F120 R62 Q70 F120 R62 F67 Q70 N109 F120 L129 H133 R62 F67 Q70 N109 F120 L129 H133 5.2.1.8 0000413,0003755,0005515,0005634,0005737,0005739,0006357,0006457,0016018,0140839,0140840 remove_due_to_license_issue P52011 17654646 202 MSRSKVFFDITIGGKASGRIVMELYDDVVPKTAGNFRALCTGENGIGKSGKPLHFKGSKFHRIIPNFMIQGGDFTRGNGTGGESIYGEKFPDENFKEKHTGPGVLSMANAGPNTNGSQFFLCTVKTEWLDGKHVVFGRVVEGLDVVKAVESNGSQSGKPVKDCMIADCGQLK 2igx A 1.7 BS01 A1T A 1 D34 G36 W41 Y77 F111 T114 Y115 S118 F120 I123 Y192 F294 D34 G36 W41 Y77 F111 T114 Y115 S118 F120 I123 Y192 F294 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue P46925 17091526 330 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 2igy A 2.6 BS01 A2T A 1 D34 G36 W41 Y77 F111 I123 Y192 G216 S218 D34 G36 W41 Y77 F111 I123 Y192 G216 S218 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue IC50=113nM P46925 17091526 330 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 2ihj A 2.0 BS01 CSF A 1 R63 D141 G142 S143 M144 G266 W270 K309 H311 S336 E338 S356 R39 D117 G118 S119 M120 G242 W246 K285 H287 S312 E314 S332 2.4.99.4 0016757 Ki=25.7uM remove_due_to_license_issue Q15KI8 17487984 1741 MKTITLYLDPASLPALNQLMDFTQNNEDKTHPRIFGLSRFKIPDNIITQYQNIHFVELKDNRPTEALFTILDQYPGNIELNIHLNIAHSVQLIRPILAYRFKHLDRVSIQQLNLYDDGSMEYVDLEKEENKDISAEIKQAEKQLSHYLLTGKIKFDNPTIARYVWQSAFPVKYHFLSTDYFEKAEFLQPLKEYLAENYQKMDWTAYQQLTPEQQAFYLTLVGFNDEVKQSLEVQQAKFIFTGTTTWEGNTDVREYYAQQQLNLLNHFTQAEGDLFIGDHYKIYFKGHPRGGEINDYILNNAKNITNIPANISFEVLMMTGLLPDKVGGVASSLYFSLPKEKISHIIFTSNNPYVKVMRRLGIIDESQVIFWDSLKQLG 2ihq A 2.0 BS01 LG7 A 1 L704 N705 L707 G708 Q711 M742 M745 V746 M749 F764 M780 M787 L873 F876 T877 M895 L34 N35 L37 G38 Q41 M72 M75 V76 M79 F94 M110 M117 L203 F206 T207 M225 ? Ki=3.2nM remove_due_to_license_issue P15207 17181141 90 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 2ihx A -1.00 BS01 rna B 0 R18 L20 C21 Y22 Y30 Q31 A32 Q33 R46 L49 C50 N51 M53 H55 A57 K58 Q59 C60 R61 K62 R4 L6 C7 Y8 Y16 Q17 A18 Q19 R32 L35 C36 N37 M39 H41 A43 K44 Q45 C46 R47 K48 3.4.23.- 0003676,0008270 remove_due_to_license_issue P03322 17070546 160 ~ 234 GRARGLCYTCGSPGHYQAQCPKKRKSGNSRERCQLCNGMGHNAKQCRKRD 2iit A 2.35 BS01 872 A 1 E205 E206 F357 S630 Y631 Y662 Y666 N710 V711 E167 E168 F319 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=2.6nM remove_due_to_license_issue IC50=2.6nM P27487 17055272 9001 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2iiv A 2.15 BS01 565 A 1 E205 E206 F357 Y547 S630 Y631 Y662 Y666 N710 V711 E167 E168 F319 Y509 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=6.6nM remove_due_to_license_issue IC50=6.6nM P27487 17055272 9001 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2iko A 1.9 BS01 7IG A 1 V31 D33 Y78 T80 P113 F114 L116 V122 D221 G223 V34 D36 Y81 T83 P116 F117 L119 V125 D224 G226 D33 S36 N38 W40 D221 A224 D36 S39 N41 W43 D224 A227 3.4.23.15 0004190,0006508 Kd=3571nM remove_due_to_license_issue IC50=4000nM P00797 17113558 601 LGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2iku A 2.6 BS01 LIY A 1 D33 Y78 T80 F114 F119 V122 D221 G223 D35 Y80 T82 F116 F121 V124 D223 G225 D33 S36 N38 W40 Y78 D221 A224 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=58nM P00797 17113558 336 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2il2 B 2.24 BS01 LIX B 1 T13 Q14 Y15 V31 D33 Y78 S79 T80 L116 V122 D221 G223 A224 S225 Y226 H296 M298 T16 Q17 Y18 V34 D36 Y81 S82 T83 L119 V125 D224 G226 A227 S228 Y229 H299 M301 D33 S36 N38 W40 Y78 D221 A224 D36 S39 N41 W43 Y81 D224 A227 3.4.23.15 0004190,0006508 Kd=79nM remove_due_to_license_issue IC50=27nM, Kd=79nM P00797 17113558 402 LGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2ilp A 1.9 BS02 GB5 A 1 I161 F194 H223 E224 H227 E262 Y366 F369 I163 F196 H223 E224 H227 E250 Y354 F357 H223 E224 H227 E262 R363 H223 E224 H227 E250 R351 3.4.24.69 0004222,0006508,0008270 ic50=15uM remove_due_to_license_issue P0DPI1 17524984 600 SSGLVPRGSHMQFVNKQFNYKDPVNGVDIAYIKIPQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEESLEVNPLLGAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFKEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGTTASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKNF 2ima A 1.94 BS02 GB4 A 1 I161 F163 F194 H223 E224 H227 E262 R363 Y366 F369 I162 F164 F195 H221 E222 H225 E248 R347 Y350 F353 H223 E224 H227 E262 R363 H221 E222 H225 E248 R347 3.4.24.69 0004222,0006508,0008270 Ki=300nM remove_due_to_license_issue Q84GJ4 17524984 600 SSGLVPRGSHMQFVNKQFNYKDPVNGVDIAYIKIPMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEESLENPLLGAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFKEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKN 2imb A 2.41 BS02 AHL A 1 F163 F194 H223 E224 H227 Y366 F161 F192 H212 E213 H216 Y341 H223 E224 H227 E262 R363 H212 E213 H216 E239 R338 3.4.24.69 0004222,0006508,0008270 remove_due_to_license_issue P0DPI1 17524984 600 SSGLVPRGSHMQFVNKQFNYKDPVNGVDIAYIKIPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEESLAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFKEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKN 2imd A 1.6 BS01 GSH A 1 S11 F13 G167 V168 W179 G180 N181 D182 S11 F13 G167 V168 W179 G180 N181 D182 5.99.1.4 0004364,0004602,0006749,0009056,0016491,0016853,0018845,0098869,1901170 Kd=14uM remove_due_to_license_issue Q51948 17508726 301 MIVDFYFDFLSPFSYLANQRLSKLAQDYGLTIRYNAIDLARVKIAIGNVGPSNRDLKVKLDYLKVDLQRWAQLYGIPLVFPANYNSRRMNIGFYYSGAEAQAAAYVNVVFNAVWGEGIAPDLESLPALVSEKLGWDRSAFEHFLSSNAATERYDEQTHAAIERKVFGVPTMFLGDEMWWGNDRLFMLESAMGRLCRQNADLSS 2in6 A 1.9 BS01 839 A 1 I305 A326 K328 V360 N376 E377 Y378 C379 G382 F433 D463 I15 A36 K38 V67 N83 E84 Y85 C86 G89 F140 D150 D426 K428 D133 K135 2.7.10.2 0004672,0005524,0006468 ic50=0.023uM remove_due_to_license_issue IC50=23nM P30291 17869387 901 MKSRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVL 2io6 A 2.2 BS01 330 A 1 I305 A326 K328 N376 E377 Y378 C379 G382 F433 D463 I15 A32 K34 N79 E80 Y81 C82 G85 F136 D146 D426 K428 D129 K131 2.7.10.2 0004672,0005524,0006468 ic50=0.03uM remove_due_to_license_issue IC50=30nM P30291 17869387 901 MKSRYTTEFHELEKIGSSVFKCVKRLDGCIYAIKRSKKPSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVL 2ioa A 2.8 BS03 GGA A 1 N241 R316 E330 N332 S335 A336 S337 D387 E391 E392 W442 A443 T446 R538 C539 R598 K607 N220 R295 E309 N311 S314 A315 S316 D366 E370 E371 W417 A418 T421 R509 C510 R569 K578 3.5.1.78,6.3.1.8 0005515,0005524,0005829,0006749,0008216,0008884,0008885,0016787,0016874,0046872 remove_due_to_license_issue P0AES0 17124497 6001 APFGTLLGYAPGGVAIYSSDYVFRSYIDDEYMGHKWQCVEFARRFLFLNYGVVFTDVGMAWEIFSLRFLREVVNDNILPLQAFPNGSPRAPVAGALLIWDKGGEFKDTGHVAIITQLHGNKVRIAEQNVIHSPLPQGQQWTRELEMVVENGCYTLKDTFDDTTILGWMIQTEDTEYSLPQPEIAGELLKISGARLENKGQFDGKWLDEKDPLQNAYVQANGQVINQDPYHYYTITESAEQELIKATNELHLMYLHATDKVLKDDNLLALFDIPKILWPRLRLSWQRRRHHMITGRMDFCMDERGLKVYEYNADSASCHTEAGLILERWAEQGYKGNGFNPAEGLINELAGAWKHSRARPFVHIMQDKDIEENYHAQFMEQALHQAGFETRILRGLDELGWQLIDGEGRLVNCVWKTWAWETAFDQIREVFAAVPIRTGHPQNEVRLIDVLLRPEVLVFEPLWTVIPGNKAILPILWSLFPHHRYLLDTDFTVNDELVKTGYAVKPIAGRCGSNIDLVSHHEEVLDKTSGKFAEQKNIYQQLWCLPKVDGKYIQVCTFTVGGNYGGTCLRGDESLVIKKESDIEPLIVVK 2iog A 1.6 BS01 IOG A 1 T347 D351 E353 W383 L387 L391 V418 I424 F425 G521 H524 L525 M528 C530 K531 T39 D43 E45 W75 L79 L83 V110 I116 F117 G213 H216 L217 M220 C222 K223 ? ic50=8nM remove_due_to_license_issue IC50=8nM P03372 17289385 600 SLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLHA 2iok A 2.4 BS01 IOK A 1 M343 A350 E353 L384 F404 L428 H524 L525 M31 A38 E41 L72 F92 L116 H212 L213 ? ic50=1nM remove_due_to_license_issue IC50=1nM P03372 17289385 600 LALSLTADQMVSALLDAEPPILYSEYEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKPLYDLLLEML 2ipo A 2.6 BS01 1IP A 1 S52 T53 R54 T55 R105 H134 R167 T168 R229 L267 S52 T53 R54 T55 R105 H134 R167 T168 R229 L267 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 remove_due_to_license_issue P0A786 18004787 401 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFETSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQETQGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPQYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 2iqg A 1.7 BS01 F2I A 1 Q12 G13 D32 G34 S35 Y71 T72 Q73 G74 F108 I110 W115 Y198 D228 G230 T232 Q15 G16 D35 G37 S38 Y74 T75 Q76 G77 F111 I113 W118 Y194 D224 G226 T228 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=5nM remove_due_to_license_issue IC50=5nM P56817 17300163 801 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2irf G 2.2 BS01 dna F 0 R7 M8 W58 T62 K64 N80 C83 A84 S87 L88 R3 M4 W54 T58 K60 N76 C79 A80 S83 L84 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1124 ~ 1136 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf H 2.2 BS01 dna A 0 W238 H240 A241 K275 K278 R282 W34 H36 A37 K71 K74 R78 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1001 ~ 1012 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf H 2.2 BS02 dna F 0 R207 M208 W258 T262 K264 N280 C283 A284 L288 R3 M4 W54 T58 K60 N76 C79 A80 L84 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1124 ~ 1136 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf I 2.2 BS01 dna A 0 W438 H440 A441 K475 K478 R482 R507 W34 H36 A37 K71 K74 R78 R103 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1001 ~ 1012 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf I 2.2 BS02 dna E 0 R407 M408 W458 T462 K464 N480 C483 A484 S487 R3 M4 W54 T58 K60 N76 C79 A80 S83 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1113 ~ 1124 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf I 2.2 BS03 dna F 0 H440 R443 H444 K500 K501 G502 H36 R39 H40 K96 K97 G98 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1124 ~ 1136 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf J 2.2 BS01 dna B 0 W638 H640 A641 K675 K678 R682 K700 R707 W34 H36 A37 K71 K74 R78 K96 R103 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1013 ~ 1024 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf J 2.2 BS02 dna E 0 R607 M608 W658 T662 K664 N680 C683 L688 R3 M4 W54 T58 K60 N76 C79 L84 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1113 ~ 1124 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf J 2.2 BS03 dna F 0 R643 K701 R39 K97 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1124 ~ 1136 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf K 2.2 BS01 dna B 0 W838 H840 A841 K875 K878 R882 W34 H36 A37 K71 K74 R78 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1013 ~ 1024 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf K 2.2 BS02 dna D 0 R805 R807 M808 W858 T862 K864 N880 C883 A884 S887 R1 R3 M4 W54 T58 K60 N76 C79 A80 S83 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1100 ~ 1112 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf K 2.2 BS03 dna E 0 R843 H844 K900 K901 G902 R39 H40 K96 K97 G98 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1113 ~ 1124 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf L 2.2 BS01 dna C 0 W2038 H2040 A2041 K2075 K2078 R2082 W34 H36 A37 K71 K74 R78 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1025 ~ 1036 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf L 2.2 BS02 dna D 0 R2007 M2008 W2058 T2062 K2064 N2080 C2083 R3 M4 W54 T58 K60 N76 C79 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1100 ~ 1112 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irf L 2.2 BS03 dna E 0 H2040 A2042 R2043 H36 A38 R39 ? 0000976,0003700,0006355 remove_due_to_license_issue P23906 10487755 1113 ~ 1124 RMRMRPWLEEQINSNTIPGLKWLNKEKKIFQIPWMHAARHGWDVEKDAPLFRNWAIHTGKHQPGIDKPDPKTWKANFRCAMNSLPDIEEVKDRSIKKGNNAFRVYRMLP 2irz A 1.8 BS01 I02 A 1 G11 Q12 G13 Y14 L30 D32 G34 Y71 Q73 D228 G230 T231 T232 N233 R235 A335 G17 Q18 G19 Y20 L36 D38 G40 Y77 Q79 D222 G224 T225 T226 N227 R229 A329 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=12nM remove_due_to_license_issue IC50=12nM P56817 17149856 386 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2is0 A 2.2 BS01 I03 A 1 G11 Q12 G13 Y14 L30 D32 S35 Y71 T72 Q73 D228 G230 T231 T232 N233 R235 A335 G17 Q18 G19 Y20 L36 D38 S41 Y77 T78 Q79 D222 G224 T225 T226 N227 R229 A329 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=200nM remove_due_to_license_issue P56817 17149856 386 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2iso A 2.1 BS01 dna T 0 H34 S229 K230 G231 T233 K234 R258 K280 R283 L287 T292 N294 E295 Y296 H25 S220 K221 G222 T224 K225 R249 K271 R274 L278 T283 N285 E286 Y287 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 17209556 1 ~ 16 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 2iso A 2.1 BS02 dna P 0 G105 G107 P108 S109 A110 M236 R254 D256 G96 G98 P99 S100 A101 M227 R245 D247 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 17209556 1 ~ 10 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 2iso A 2.1 BS03 dna D 0 K35 A38 Y39 P63 G64 V65 G66 K68 I69 K26 A29 Y30 P54 G55 V56 G57 K59 I60 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 17209556 1 ~ 5 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 2isp A 2.2 BS01 dna T 0 H34 S229 K230 G231 T233 K234 R258 K280 R283 T292 I293 N294 E295 Y296 H25 S220 K221 G222 T224 K225 R249 K271 R274 T283 I284 N285 E286 Y287 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 17209556 1 ~ 16 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 2isp A 2.2 BS02 dna P 0 G105 G107 P108 S109 A110 R254 D256 G96 G98 P99 S100 A101 R245 D247 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 17209556 1 ~ 10 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 2isp A 2.2 BS03 dna D 0 K35 A38 Y39 G64 G66 K68 I69 K26 A29 Y30 G55 G57 K59 I60 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 17209556 1 ~ 5 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGETKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 2isv A 2.3 BS02 PGH A 1 D83 H178 H210 G211 S213 N253 D255 S256 D82 H163 H186 G187 S189 N229 D231 S232 4.1.2.13 0004332,0005515,0005975,0006096,0008270,0016829,0016832,0046872 Ki=37nM remove_due_to_license_issue A8B2U2 17166851 325 PLCTLRQMLGEARKHKYGVGAFNVNNMEQIQGIMKAVVQLKSPVILQCSRGALKYSDMIYLKKLCEAALEKHPDIPICIHLDHGDTLESVKMAIDLGFSSVMIDASHHPFDENVRITKEVVAYAHARSVSVEAELGLTEPQDAKKFVELTGVDALAVAIGTSHGARLAIDRVKTISDLTGIPLVMHGSSSVPKDVKDMINKYGGKMPDAVGVPIESIVHAIGEGVCKINVDSDSRMAMTGAIRKVFVEHPEKFDPRDYLGPGRDAITEMLIPKIKAFGSAGHAGDYKVVSLEEAKAWY 2isv B 2.3 BS02 PGH B 1 D83 H178 G179 K182 H210 G211 S213 N253 D255 S256 D82 H168 G169 K172 H195 G196 S198 N238 D240 S241 4.1.2.13 0004332,0005515,0005975,0006096,0008270,0016829,0016832,0046872 Ki=37nM remove_due_to_license_issue A8B2U2 17166851 325 PLCTLRQMLGEARKHKYGVGAFNVNNMEQIQGIMKAVVQLKSPVILQCSRGALKYSDMIYLKKLCEAALEKHPDIPICIHLDHGDTLESVKMAIDLGFSSVMIDASHHPFDENVRITKEVVAYAHARSVSVEAELGQNTVQLTEPQDAKKFVELTGVDALAVAIGTSHGAYKFIRLAIDRVKTISDLTGIPLVMHGSSSVPKDVKDMINKYGGKMPDAVGVPIESIVHAIGEGVCKINVDSDSRMAMTGAIRKVFVEHPEKFDPRDYLGPGRDAITEMLIPKIKAFGSAGHAGDYKVVSLEEAKAWY 2isw A 1.75 BS02 PGH A 1 D83 H178 G179 K182 H210 G211 S213 N253 D255 S256 D82 H167 G168 K171 H195 G196 S198 N238 D240 S241 4.1.2.13 0004332,0005515,0005975,0006096,0008270,0016829,0016832,0046872 Ki=37nM remove_due_to_license_issue A8B2U2 17166851 325 PLCTLRQMLGEARKHKYGVGAFNVNNMEQIQGIMKAVVQLKSPVILQCSRGALKYSDMIYLKKLCEAALEKHPDIPICIHLDHGDTLESVKMAIDLGFSSVMIDASHHPFDENVRITKEVVAYAHARSVSVEAELGTLVQLTEPQDAKKFVELTGVDALAVAIGTSHGAYKFKSRLAIDRVKTISDLTGIPLVMHGSSSVPKDVKDMINKYGGKMPDAVGVPIESIVHAIGEGVCKINVDSDSRMAMTGAIRKVFVEHPEKFDPRDYLGPGRDAITEMLIPKIKAFGSAGHAGDYKVVSLEEAKAWY 2isz A 2.403 BS01 dna E 0 R27 A28 R29 R27 A28 R29 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz A 2.403 BS02 dna F 0 N2 T7 Q36 S37 P39 T40 Q43 R47 R50 N2 T7 Q36 S37 P39 T40 Q43 R47 R50 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz B 2.403 BS01 dna E 0 N2 T7 Q36 S37 P39 T40 Q43 R47 R50 R60 N2 T7 Q36 S37 P39 T40 Q43 R47 R50 R60 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz B 2.403 BS02 dna F 0 R27 A28 R29 P39 S42 R27 A28 R29 P39 S42 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz C 2.403 BS01 dna E 0 N2 T7 Q36 S37 P39 T40 R47 R50 N2 T7 Q36 S37 P39 T40 R47 R50 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz C 2.403 BS02 dna F 0 R27 A28 R29 S42 R60 R27 A28 R29 S42 R60 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz D 2.403 BS01 dna E 0 R27 A28 R29 P39 S42 R60 R27 A28 R29 P39 S42 R60 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2isz D 2.403 BS02 dna F 0 N2 T7 Q36 S37 P39 T40 R47 R50 N2 T7 Q36 S37 P39 T40 R47 R50 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 MNELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGV 2it0 A 2.6 BS01 dna E 0 R27 A28 R29 R60 R25 A26 R27 R58 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGVASENLYF 2it0 A 2.6 BS02 dna F 0 T7 Q36 S37 P39 T40 R47 R50 T5 Q34 S35 P37 T38 R45 R48 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGVASENLYF 2it0 B 2.6 BS01 dna E 0 T7 Q36 S37 P39 T40 Q43 R47 R50 T5 Q34 S35 P37 T38 Q41 R45 R48 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGVASENLYF 2it0 B 2.6 BS02 dna F 0 R27 A28 R29 P39 S42 R60 R25 A26 R27 P37 S40 R58 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELGVASENLYF 2it0 C 2.6 BS01 dna E 0 T7 Q36 S37 P39 T40 R47 R50 T5 Q34 S35 P37 T38 R45 R48 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELG 2it0 C 2.6 BS02 dna F 0 R27 A28 R29 R60 R25 A26 R27 R58 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELG 2it0 D 2.6 BS01 dna E 0 R27 A28 R29 S42 R60 R25 A26 R27 S40 R58 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELG 2it0 D 2.6 BS02 dna F 0 T7 Q36 S37 P39 T40 R47 R50 T5 Q34 S35 P37 T38 R45 R48 ? 0003677,0003700,0006355,0046914,0046983 remove_due_to_license_issue P9WMH1 17209554 1 ~ 33 ELVDTTEMYLRTIYDLEEEGVTPLRARIAERLDQSGPTVSQTVSRMERDGLLRVAGDRHLELTEKGRALAIAVMRKHRLAERLLVDVIGLPWEEVHAEACRWEHVMSEDVERRLVKVLNNPTTSPFGNPIPGLVELG 2it4 A 2.0 BS02 PPF A 1 H94 L198 H90 L194 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=24.1mM remove_due_to_license_issue P00915 17314045 500 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2ito A 3.25 BS01 IRE A 1 S719 A743 K745 M766 L788 T790 M793 G796 S24 A48 K50 M71 L93 T95 M98 G101 D837 A839 R841 N842 D855 D142 A144 R146 N147 D160 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 17349580 2020 GEAPNQALLRILKETEFKKIKVLSSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLMDEEDMDDVVDADEYLIP 2itp A 2.74 BS01 AEE A 1 L718 A743 K745 T790 Q791 M793 G796 E804 L844 L22 A47 K49 T94 Q95 M97 G100 E108 L148 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=5.3nM, IC50=2nM P00533 17349580 2019 EAPNQALLRILKETEFKKIKVLSSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDMDEEDMDDVVDADEYLI 2itt A 2.73 BS01 AEE A 1 L718 K745 M766 T790 Q791 M793 G796 E804 L844 L22 K49 M70 T94 Q95 M97 G100 E108 L148 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=5.3nM, IC50=2nM P00533 17349580 2020 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLMDEEDMDDVVDADEYLIP 2ity A 3.42 BS01 IRE A 1 L718 A743 L788 T790 L792 M793 G796 L844 L22 A47 L92 T94 L96 M97 G100 L148 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 17349580 2020 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLDEEDMDDVVDADEYLIP 2itz A 2.8 BS01 IRE A 1 A743 K745 L788 T790 L792 M793 D800 L844 D855 A47 K49 L92 T94 L96 M97 D104 L148 D159 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 17349580 2021 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPMDEEDMDDVVDADEYLIP 2iu0 B 2.53 BS01 203 B 1 K15 G36 G37 T38 K67 K12 G33 G34 T35 K64 K267 H268 N432 H593 K264 H265 N429 H590 2.1.2.3,3.5.4.10 0003824,0003937,0004643,0005737,0005829,0006164,0006189,0016740,0016787,0042803 remove_due_to_license_issue P31335 17324932 1595 RQQLALLSVSEKAGLVEFARSLNALGLGLIASGGTATALRDAGLPVRDVSDLTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMNKQDFSLVRVVVCNLYPFVKTVSSPGVTVPEAVEKIDIGGVALLRAAAKNHARVTVVCDPADYSSVAKEMAASKDKDTSVETRRHLALKAFTHTAQYDAAISDYFRKEYSKGVSQLPLRYGMNPHQSPAQLYTTRPKLPLTVVNGSPGFINLCDALNAWQLVKELKQALGIPAAASFKHVSPAGAAVGIPLSEEEAQVCMVHDLHKTLTPLASAYARSRGADRMSSFGDFIALSDICDVPTAKIISREVSDGVVAPGYEEEALKILSKKKNGGYCVLQMDPNYEPDDNEIRTLYGLQLMQKRNNAVIDRSLFKNIVTKNKTLPESAVRDLIVASIAVKYTQSNSVCYAKDGQVIGIGAGQQSRIHCTRLAGDKANSWWLRHHPRVLSMKFKAGVKRAEVSNAIDQYVTGTIGEDEDLVKWQAMFEEVPAQLTEAEKKQWIAKLTAVSLSSDAFFPFRDNVDRAKRIGVQFIVAPSGSAADEVVIEACNELGITLIHTNLRLFHH 2iuz A 1.95 BS01 D1H A 1 W52 F76 W137 T138 Y139 W384 W14 F38 W99 T100 Y101 W346 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 Ki=2.8uM remove_due_to_license_issue IC50=4800nM Q873X9 16844689 1440 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQT 2ivu A 2.5 BS01 ZD6 A 1 L730 V738 A756 K758 E775 V804 Y806 A807 K808 G810 L881 S891 L30 V38 A56 K58 E75 V104 Y106 A107 K108 G110 L158 S168 D850 D874 A876 R878 N879 D892 D127 D151 A153 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 Ki=375nM remove_due_to_license_issue Kd=14nM, IC50=4.00nM P07949 16928683 3015 GPLSLSVDAFKILDPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRRALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKR 2iw6 A 2.3 BS01 QQ2 A 1 I10 G11 V18 A31 L83 D86 L134 A144 I11 G12 V19 A32 L81 D84 L132 A142 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.14uM remove_due_to_license_issue IC50=2600nM P24941 16942020 1296 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKTFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPH 2iw8 A 2.3 BS01 4SP A 1 I10 E12 G13 A31 V64 F80 E81 V83 D84 Q85 D86 K89 L134 I11 E13 G14 A32 V65 F81 E82 V84 D85 Q86 D87 K90 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=103nM remove_due_to_license_issue IC50=6.0nM, Ki=6.0nM, Kd=1310nM P24941 16942020 1298 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEHVDQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 2iws A 2.7 BS01 NP4 A 1 N37 A41 D79 I82 M84 F124 T171 V213 N37 A41 D79 I82 M84 F121 T168 V210 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=5.0e+2nM P02829 17114002 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEV 2iwu A 2.8 BS01 NP5 A 1 N37 D79 M84 F124 T171 N37 D79 M84 F124 T171 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=3.5e+3nM P02829 17114002 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2iwx A 1.5 BS01 M1S A 1 N37 D40 D79 M84 N92 F124 T171 L173 N37 D40 D79 M84 N92 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.21uM remove_due_to_license_issue IC50=7.6e+2nM P02829 17114002 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2iyf A 1.7 BS01 ERY A 1 H19 W73 N80 F84 A182 S183 D329 H13 W67 N74 F78 A176 S177 D314 2.4.1.- 0008194,0016757,0016758,0017000,0046677 remove_due_to_license_issue Q53685 17376874 1400 AHIAMFSIAAHGHVNPSLEVIRELVARGHRVTYAIPPVFADKVAATGPRPVLYHSTLPGPDADPEAWGSTLLDNVEPFLNDAIQALPQLADAYADDIPDLVLHDITSYPARVLARRWGVPAVSLSPNLVAWKGYEEEVAEPMWREPRQTERGRAYYARFEAWLKENGITEHPDTFASHPPRSLVLIPKALQPHADRVDEDVYTFVGACQEGGWQRPAGAEKVVLVSLGSAFTQPAFYRECVRAFGNLPGWHLVLQIGTPAELGELPDNVEVHDWVPQLAILRQADLFVTHAGAGGSQEGLATATPMIAVPQAVDQFGNADMLQGLGVARKLATEEATADLLRETALALVDDPEVARRLRRIQAEMAQEGGTRRAADLIEAELPA 2izl B 1.48 BS01 IMI B 1 S27 Y43 S45 V47 W79 S88 T90 W108 S15 Y31 S33 V35 W67 S76 T78 W96 ? 0009374 Kd=1uM remove_due_to_license_issue P22629 9405158 300 AEAGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVK 2j27 A 1.15 BS01 PGA A 1 K13 H95 E167 I172 G212 S213 G234 G235 K12 H94 E166 I171 G211 S212 G233 G234 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=0.3mM remove_due_to_license_issue P04789 17176070 701 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEAVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 2j27 B 1.15 BS01 PGA B 1 K13 H95 E167 I172 G212 S213 G234 G235 K12 H94 E166 I171 G211 S212 G233 G234 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=0.3mM remove_due_to_license_issue P04789 17176070 702 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEAVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 2j2i B 1.9 BS01 LY4 B 1 L44 F49 V52 A65 L120 E121 R122 V126 D128 E171 L174 D186 L12 F17 V20 A33 L88 E89 R90 V94 D96 E139 L142 D154 N172 D186 L193 N140 D154 L161 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.2uM remove_due_to_license_issue Kd=270nM, IC50=200nM P11309 18077363 1307 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 2j2u A 1.9 BS01 GSQ A 1 E97 T98 Y99 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 E79 T80 Y81 D175 A176 Q178 V199 W201 G202 G204 C205 G212 I213 Y214 H57 D102 Q192 G193 D194 S195 G196 H42 D84 Q178 G179 D180 S181 G182 3.4.21.6 0004252,0006508 Ki=90nM remove_due_to_license_issue Ki=90nM P00742 16982192 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2j34 A 2.01 BS01 GS6 A 1 E97 T98 Y99 A190 Q192 V213 W215 G216 G219 G226 I227 Y228 E83 T84 Y85 A180 Q182 V203 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=15nM remove_due_to_license_issue Ki=15nM P00742 16982192 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2j3q A 2.8 BS01 TFL A 1 Y70 Y121 W279 F330 F331 A536 Y67 Y118 W276 F327 F328 A533 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 18512913 1538 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNATA 2j47 A 1.98 BS01 GDV A 1 G135 K166 D242 D243 Y282 W286 V314 W337 N339 D344 G122 K153 D229 D230 Y269 W273 V301 W324 N326 D331 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=3.9uM remove_due_to_license_issue Q89ZI2 17057847 1590 SLQPPPQQLIVQNKTIDYQLNGGEEANPHAVKVLKELLSGGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTD 2j4a A 2.2 BS01 OEF A 1 F272 I275 I276 R282 M310 M313 R316 R320 L330 S331 L346 H435 M442 F455 E460 F62 I65 I66 R72 M100 M103 R106 R110 L120 S121 L136 H225 M232 F245 E250 ? 0003677,0004879,0006355 remove_due_to_license_issue IC50=0.0251nM P10828 17154490 1461 KPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGQAPIVNAPEGGKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLSGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 2j4g A 2.25 BS01 NB1 A 1 G135 K166 D242 C278 Y282 T310 W337 N339 D344 G132 K163 D239 C275 Y279 T307 W334 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=0.25uM remove_due_to_license_issue Q89ZI2 17227027 1590 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTD 2j4i A 1.8 BS01 GSJ A 1 K96 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 K80 E81 T82 Y83 F160 D177 A178 Q180 V201 W203 G204 G206 C207 G214 I215 Y216 H57 D102 Q192 G193 D194 S195 G196 H42 D86 Q180 G181 D182 S183 G184 3.4.21.6 0004252,0006508 Ki=1nM remove_due_to_license_issue Ki=1nM P00742 16982190 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2j4k A 2.2 BS01 U5P A 1 G42 G43 D65 G68 I69 G112 Q114 Q117 T119 G42 G43 D65 G68 I69 G112 Q114 Q117 T119 2.7.4.22 0005524,0005737,0006221,0006225,0009041,0016301,0033862,0044210,0046940 Kd=14uM remove_due_to_license_issue Q97ZE2 17297917 227 MNIILKISGKFFDEDNVDNLIVLRQSIKELADNGFRVGIVTGGGSTARRYIKLAREIGIGEAYLDLLGIWASRLNAYLVMFSLQDLAYMHVPQSLEEFIQDWSHGKVVVTGGFQPGQSTAAVAALVAEASSSKTLVVATNVDGVYEKDPRIYADVKLIPHLTTQDLRKILLLDPLAIKIVERSKIRVIVMNYRKLNRIEVSSIIEPV 2j4k E 2.2 BS01 U5P E 1 G42 D65 G68 I69 G112 F113 Q114 Q117 S118 T119 G37 D60 G63 I64 G107 F108 Q109 Q112 S113 T114 2.7.4.22 0005524,0005737,0006221,0006225,0009041,0016301,0033862,0044210,0046940 Kd=14uM remove_due_to_license_issue Q97ZE2 17297917 227 MNIILKISGKFFDEDNVLRQSIKELADNGFRVGIVTGGGSTARRYIKLAREIGIGEAYLDLLGIWASRLNAYLVMFSLQDLAYMHVPQSLEEFIQDWSHGKVVVTGGFQPGQSTAAVAALVAEASSSKTLVVATNVDGVYEKDPRIYADVKLIPHLTTQDLRKILEGSQSVQAGTYELLDPLAIKIVERSKIRVIVMNYRKLNRIIDILKGEEVSSIIEPV 2j4z A 2.0 BS01 626 A 1 A160 Y212 A213 P214 G216 R220 E260 L263 A273 H280 A35 Y87 A88 P89 G91 R95 E135 L138 A148 H155 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=65nM remove_due_to_license_issue O14965 17125279 1389 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2j50 A 3.0 BS01 627 A 1 A160 K162 E211 Y212 A213 P214 L215 G216 T217 L263 A33 K35 E84 Y85 A86 P87 L88 G89 T90 L136 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 17125279 1390 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVTLCGTLDYLPPEMIEDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2j62 A 2.26 BS01 GSZ A 1 G187 K218 D297 D298 Y335 V370 W394 N396 D401 G148 K179 D258 D259 Y296 V331 W355 N357 D362 3.2.1.169 Ki=4.6pM remove_due_to_license_issue Q0TR53 17177381 1626 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYDRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2j62 B 2.26 BS01 GSZ B 1 G187 Y189 K218 D297 D298 Y335 V370 W394 N396 D401 G148 Y150 K179 D258 D259 Y296 V331 W355 N357 D362 3.2.1.169 Ki=4.6pM remove_due_to_license_issue Q0TR53 17177381 1627 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYDRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2j6m A 3.1 BS01 AEE A 1 A743 T790 M793 P794 G796 E804 L844 A47 T94 M97 P98 G100 E108 L148 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=5.3nM, IC50=2nM P00533 17349580 2021 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDEEDMDDVVDADEYLIPQ 2j75 A 1.85 BS01 NOY A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y290 E344 W391 E398 W399 F407 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N288 Y290 E344 3.2.1.21 0004553,0005975,0008422,0016798,0030245 remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j77 A 2.1 BS01 NOJ A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 Q18 H119 N163 E164 Y289 E342 W389 E396 W397 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N287 Y289 E342 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=12.9uM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j78 A 1.65 BS03 GOX A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y293 E348 W395 E402 W403 F411 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E348 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=384nM remove_due_to_license_issue Q08638 17279749 1451 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLED 2j79 A 1.94 BS01 GTL A 1 Q20 H121 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 E164 Y290 E343 W390 E397 W398 F406 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N288 Y290 E343 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=1.1uM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7b A 1.87 BS01 NTZ A 1 Q20 H121 N165 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y289 E343 W390 E397 W398 F406 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N287 Y289 E343 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=240nM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7d A 2.24 BS01 GI1 A 1 Q20 H121 E166 N222 Y295 W324 E351 W398 E405 W406 F414 Q18 H119 E164 N220 Y289 W316 E343 W390 E397 W398 F406 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N287 Y289 E343 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=74nM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7e A 2.19 BS01 GI2 A 1 Q20 H121 N165 E166 N222 Y295 E351 W398 E405 W406 F414 Q18 H119 N163 E164 N220 Y289 E342 W389 E396 W397 F405 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N287 Y289 E342 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=48nM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7f A 2.28 BS01 GI3 A 1 Q20 H121 E166 Y295 W324 E351 W398 E405 W406 F414 Q18 H119 E164 Y288 W314 E341 W388 E395 W396 F404 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N286 Y288 E341 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=445nM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASERAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7g A 1.91 BS01 GI4 A 1 Q20 H121 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 E164 Y290 E343 W390 E397 W398 F406 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N288 Y290 E343 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=100nM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7h A 1.95 BS01 AZF A 1 Q20 H121 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 E164 Y289 E344 W391 E398 W399 F407 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N287 Y289 E344 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=65nM remove_due_to_license_issue Q08638 17279749 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2j7w A 2.6 BS03 GTP A 1 S710 R729 R737 T794 S398 R417 R425 T482 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 remove_due_to_license_issue Q6YMS4 17301146 1886 MDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYESSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAASAKAAVEDEEFWKLVDRERELHKLGKCGSCVAIWYMWLGARYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 2j7x A 2.1 BS02 EST A 1 E260 L294 F311 H430 L431 E41 L75 F92 H205 L206 ? remove_due_to_license_issue EC50=0.14nM, IC50=1.7nM Q62986 1454 TLSPEQLVLTLLEAEPPNVLVSMPFTEASMMMSLTKLADKELVHMIGWAKKIPGFVELSLLDQVRLLESCWMEVLMVGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLAESSRKLTHLLNAVTDALVWVIAKSGISSQQQSVRLANLLMLLSHVRHISNKGMEHLLSMKCKNVVPVYDLLLEMLNAH 2j83 A 2.0 BS01 BAT A 1 S181 Q185 D186 I187 L188 G189 H228 E229 H232 H238 Y292 S119 Q123 D124 I125 L126 G127 H166 E167 H170 H176 Y230 3.4.24.- 0008237 ic50=61uM remove_due_to_license_issue Q8TL28 17097044 996 EIVKIPVVVHVVWNEEEENISDAQIQSQIDILNKDFRKLNSDVSQVPSVWSNLIADLGIEFFLATKDPNGNQTTGITRTQTSVTFFTTSDEVKFASSGGEDAWPADRYLNIWVCHVLKSEIGQDILGYAQFPGGPAETDGVVIVDAAFGTTGTALPPFDKGRTATHEIGHWLNLYHIWGDELRFEDPCSRSDEVDDTPNQADPNFGAPSYPHVSCSNGPNGDMFMNYMDYVDDKCMVMFTQGQATRVNACLDGPRSSFL 2j83 B 2.0 BS01 BAT B 1 Q185 D186 I187 L188 G189 H228 E229 H232 H238 Y292 Q123 D124 I125 L126 G127 H166 E167 H170 H176 Y230 3.4.24.- 0008237 ic50=61uM remove_due_to_license_issue Q8TL28 17097044 996 EIVKIPVVVHVVWNEEEENISDAQIQSQIDILNKDFRKLNSDVSQVPSVWSNLIADLGIEFFLATKDPNGNQTTGITRTQTSVTFFTTSDEVKFASSGGEDAWPADRYLNIWVCHVLKSEIGQDILGYAQFPGGPAETDGVVIVDAAFGTTGTALPPFDKGRTATHEIGHWLNLYHIWGDELRFEDPCSRSDEVDDTPNQADPNFGAPSYPHVSCSNGPNGDMFMNYMDYVDDKCMVMFTQGQATRVNACLDGPRSSFL 2j87 A 3.1 BS01 TTP A 1 M13 F14 S15 G16 K17 S18 D82 E83 F86 L109 F113 E158 I159 I160 G161 Y166 M10 F11 S12 G13 K14 S15 D64 E65 F68 L91 F95 E140 I141 I142 G143 Y148 2.7.1.21 0004797,0005524,0009157,0016301,0046104,0046872,0071897 remove_due_to_license_issue O57203 17062140 300 GHIQLIIGPMFSGKSTELIRRVRRYQIAQYKCVTIKYSNDNALEATKLCDVLQSITDFSVIGIDEGQFFPDIVEFCERMANEGKIVIVAALDGTFQRKPFNNILNLLILSEMVVKLTAVCMKCFKEASFSKRLGEETEIEIIGGNDMYQSVCRKCYVG 2j87 C 3.1 BS01 TTP C 1 M13 F14 S15 G16 K17 S18 D82 E83 F86 L109 F113 I157 E158 I159 I160 G161 Y166 M10 F11 S12 G13 K14 S15 D69 E70 F73 L96 F100 I144 E145 I146 I147 G148 Y153 2.7.1.21 0004797,0005524,0009157,0016301,0046104,0046872,0071897 remove_due_to_license_issue O57203 17062140 300 GHIQLIIGPMFSGKSTELIRRVRRYQIAQYKCVTIKYSNDDKNNFEALEATKLCDVLQSITDFSVIGIDEGQFFPDIVEFCERMANEGKIVIVAALDGTFQRKPFNNILNLLILSEMVVKLTAVCMKCFKEASFSKRLGEETEIEIIGGNDMYQSVCRKCYVG 2j94 A 2.1 BS01 G15 A 1 E97 T98 Y99 D189 A190 Q192 V213 W215 G216 G219 G226 I227 Y228 E83 T84 Y85 D179 A180 Q182 V203 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=534nM remove_due_to_license_issue P00742 17338508 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2j95 A 2.01 BS01 GSX A 1 E97 T98 Y99 F174 A190 Q192 W215 G216 G226 Y228 E83 T84 Y85 F162 A180 Q182 W205 G206 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=4nM remove_due_to_license_issue Ki=4nM P00742 17338508 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2j9a A 1.73 BS04 AHY D 1 K250 D255 M270 D273 D332 E334 L360 K250 D255 M270 D273 D332 E334 L360 K262 R336 K262 R336 3.4.11.1,3.4.11.5,3.4.13.23 0004177,0004180,0005737,0005739,0006508,0008233,0016805,0019538,0030145,0046872,0070006,0097718 remove_due_to_license_issue P00727 17157838 1 TKGLVLGIYSKEKEEDEPQFTSAGENFNKLVSGKLREILNISGPPLKAGKTRTFYGLHEDFPSVVVVGLGKKTAGIDEQENWHEGKENIRAAVAAGCRQIQDLEIPSVEVDPCGDAQAAAEGAVLGLYEYDDLKQKRKVVVSAKLHGSEDQEAWQRGVLFASGQNLARRLMETPANEMTPTKFAEIVEENLKSASIKTDVFIRPKSWIEEQEMGSFLSVAKGSEEPPVFLEIHYKGSPNASEPPLVFVGKGITFDSGGISIKAAANMDLMRADMGGAATICSAIVSAAKLDLPINIVGLAPLCENMPSGKANKPGDVVRARNGKTIQVDNTDAEGRLILADALCYAHTFNPKVIINAATLTGAMDIALGSGATGVFTNSSWLWNKLFEASIETGDRVWRMPLFEHYTRQVIDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHLDIAGVMTNKDEVPYLRKGMAGRPTRTLIEFLFRFSQE 2j9h A 2.4 BS01 GTX A 1 F9 R14 W39 K45 Q52 L53 Q65 S66 F8 R13 W38 K44 Q51 L52 Q64 S65 Y8 R14 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=410uM remove_due_to_license_issue P09211 18177897 300 PPYTVVYFPVRGRSAALRMLLADQGQSWKEEVVTVETWQEGSLKASALYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRAKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGSLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 2j9h B 2.4 BS01 GTX B 1 F9 R14 W39 K45 G51 Q52 L53 Q65 S66 F8 R13 W38 K44 G50 Q51 L52 Q64 S65 Y8 R14 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=410uM remove_due_to_license_issue P09211 18177897 300 PPYTVVYFPVRGRSAALRMLLADQGQSWKEEVVTVETWQEGSLKASALYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRAKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGSLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 2j9l A 2.3 BS01 ATP A 1 K587 L595 T596 Y617 S618 I722 T724 K726 D727 K10 L18 T19 Y40 S41 I145 T147 K149 D150 ? Kd=90uM remove_due_to_license_issue P51795 17195847 1752 HKTLAMDVMKPRRNDPLLTVLTQDSMTVEDVETIISETTYSGFPVVVSRESQRLVGFVLRRDLIISIENARKKQDGVVSTSIIYFTEHSPPLPPYTPPTLKLRNILDLSPFTVTDLTPMEIVVDIFRKLGLRQCLVTHNGRLLGIITKKDVLKHIAQMANFNEFLEV 2j9l C 2.3 BS01 ATP C 1 K587 L595 T596 Y617 S618 I722 T724 K726 D727 K10 L18 T19 Y40 S41 I145 T147 K149 D150 ? Kd=90uM remove_due_to_license_issue P51795 17195847 1755 HKTLAMDVMKPRRNDPLLTVLTQDSMTVEDVETIISETTYSGFPVVVSRESQRLVGFVLRRDLIISIENARKKQDGVVSTSIIYFTEHSPPLPPYTPPTLKLRNILDLSPFTVTDLTPMEIVVDIFRKLGLRQCLVTHNGRLLGIITKKDVLKHIAQMANQLFNEFLEVLFQ 2ja3 A 3.05 BS01 ADP A 1 K587 L595 T596 Y617 D727 K10 L18 T19 Y40 D150 ? remove_due_to_license_issue P51795 17195847 1752 HKTLAMDVMKPRRNDPLLTVLTQDSMTVEDVETIISETTYSGFPVVVSRESQRLVGFVLRRDLIISIENARKKQDGVVSTSIIYFTEHSPPLPPYTPPTLKLRNILDLSPFTVTDLTPMEIVVDIFRKLGLRQCLVTHNGRLLGIITKKDVLKHIAQMANFNEFLEV 2jaj A 2.0 BS01 D20 A 1 L29 D72 F75 D78 H172 K174 V267 D268 C273 L22 D63 F66 D69 H163 K165 V258 D259 C264 3.5.3.18 0000052,0003073,0003824,0005829,0006525,0006527,0007263,0008285,0016403,0016597,0016787,0043116,0045429,0045766,0046209,0046872,0070062,1900038 ic50<25uM remove_due_to_license_issue Ki=13000nM, IC50=29000nM O94760 17273169 500 AFGRATHAVVRALPESLGQHALRSGEEVDVARAERQHQLYVGVLGSKLGLQVVELPADESLPDCVFVEDVAVVCEETALITRPGAPSRRKEVDMMKEALEKLQLNIVEMKDENATLDGGDVLFTGREFFVGLSKRTNQRGAEILADTFKDYAVSTVPVADGLHLKSFCSMAGPNLIAIGSSESAQKALKIMQQMSDHRYDKLTVPDDIAANCIYLNIPNKGHVLLHRTPEEYPESAKVYEKLKDHMLIPVSMSELEKVDGLLTCCSVLINKK 2jal A 1.9 BS01 YLL A 1 Q20 H121 E166 E351 W398 E405 W406 F414 Q18 H119 E164 E342 W389 E396 W397 F405 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N286 Y288 E342 3.2.1.21 0004553,0005975,0008422,0016798,0030245 remove_due_to_license_issue Q08638 17252125 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASERAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2jb5 H 2.8 BS01 T5C H 1 Y32 A33 N35 Y99 M101 Y30 A31 N33 Y97 M99 remove_due_to_license_issue 18241888 1223 QLVQSGAEVKKPGSSVKVSCKASGGTFSNYAINWVRQAPGQGLEWMGNIEPYFGTANYAQKFQGRVTITADESTSTAYMELSSLRSEDTAVYYCARYFMSYKHLSDYWGQGTLVTVSSASTKGPSVFPLAPSSKSGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 2jb5 L 2.8 BS01 T5C H 1 Y34 Y51 G52 W93 L97 A212 P213 Y32 Y49 G50 W91 L95 A210 P211 ? 0002250,0003823,0005576,0005615,0005886,0016064,0019814,0070062,0071735,0072562 remove_due_to_license_issue P0DOY2 18241888 1223 ALTQPASVSGSPGQSITISCTGTSSDVGSNNYVSWYQQHPGKAPKLMIYGGSNRPSGVSNRFSGSKSGNTASLTISGLQAEDEADYYCRSWDSNLSYSVFGGGTKLTVLGQPKAAPSVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADSSPVKAGVETTTPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAP 2jb6 A 2.85 BS01 T5C B 1 Y34 Y51 G52 W93 Y32 Y49 G50 W91 ? 0002250,0003823,0005576,0005615,0005886,0016064,0019814,0070062,0071735,0072562 remove_due_to_license_issue P0DOY2 18241888 1222 ALTQPASVSGSPGQSITISCTGTSSDVGSNNYVSWYQQHPGKAPKLMIYGGSNRPSGVSNRFSGSKSGNTASLTISGLQAEDEADYYCRSWDSNLSYSVFGGGTKLTVLGQPKAAPSVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADSSPVKAGVETTTPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAP 2jb6 B 2.85 BS01 T5C B 1 Y32 A33 Y99 K104 Y25 A26 Y92 K97 remove_due_to_license_issue 18241888 1222 QLVQSGAEVKKPGSSVKVSCKASNYAINWVRQAPGQGLEWMGNIEPYFGTANYAQKFQGRVTITADESTSTAYMELSSLRSEDTAVYYCARYFMSYKHLSDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 2jbj A 2.19 BS04 G88 A 1 R210 N257 D387 E424 E425 D453 G518 Y552 H553 K699 Y700 R154 N201 D329 E366 E367 D395 G460 Y489 H490 K636 Y637 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=0.2nM remove_due_to_license_issue Ki=0.280000nM, IC50=300nM, Kd=0.5nM, EC50=0.620000nM Q04609 17372356 1768 NMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2jbk A 2.99 BS04 QUS A 1 R210 N257 E424 G427 L428 G518 Y552 K699 Y700 R154 N201 E366 G369 L370 G460 Y489 K636 Y637 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Q04609 17372356 1764 NMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2jbl L 2.4 BS04 SMA L 1 L189 H190 L193 E212 N213 F216 Y222 S223 G225 A226 I229 L189 H190 L193 E212 N213 F216 Y222 S223 G225 A226 I229 ? 0009772,0015979,0016020,0019684,0030077,0042314,0042717,0045156,0046872 remove_due_to_license_issue P06009 17337272 1277 ALLSFERKYRVRGGTLIGGDLFDFWVGPYFVGFFGVSAIFFIFLGVSLIGYAASQGPTWDPFAISINPPDLKYGLGAAPLLEGGFWQAITVCALGAFISWMLREVEISRKLGIGWHVPLAFCVPIFMFCVLQVFRPLLLGSWGHAFPYGILSHLDWVNNFGYQYLNWHYNPGHMSSVSFLFVNAMALGLHGGLILSVANPGDGDKVKTAEHENQYFRDVVGYSIGALSIHRLGLFLASNIFLTGAFGTIASGPFWTRGWPEWWGWWLDIPFWS 2jbo A 3.1 BS01 P4O A 1 L70 L72 K93 L141 D207 L27 L29 K50 L98 D164 D186 K188 E190 N191 D207 T226 D143 K145 E147 N148 D164 T175 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=8.5nM, EC50=49nM P49137 17449059 1348 PQFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTCYTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDK 2jbp A 3.31 BS01 P4O A 1 L70 L72 G73 K93 C140 L141 D142 L193 D207 L25 L27 G28 K48 C95 L96 D97 L146 D160 D186 K188 E190 N191 D207 D139 K141 E143 N144 D160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=8.5nM, EC50=49nM P49137 17449059 1351 FHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNSPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWE 2jbv A 1.86 BS01 FAO A 1 G22 S23 E44 A45 W71 A90 G95 C96 H99 N100 S101 I103 R231 A232 T269 G270 D273 V464 Y465 H466 D499 A500 N510 P511 N512 V515 G22 S23 E44 A45 W71 A90 G95 C96 H99 N100 S101 I103 R231 A232 T269 G270 D273 V464 Y465 H466 D499 A500 N510 P511 N512 V515 I333 P377 N378 V464 H466 V509 N510 I333 P377 N378 V464 H466 V509 N510 1.1.3.17 0000166,0016491,0016614,0019285,0033713,0050660 remove_due_to_license_issue Q7X2H8 18072756 1528 MHIDNIENLSDREFDYIVVGGGSAGAAVAARLSEDPAVSVALVEAGPDDRGVPEVLQLDRWMELLESGYDWDYPIEPQENGNSFMRHARAKVMGGCSSHNSCIAFWAPREDLDEWEAKYGATGWNAEAAWPLYKRLETNEDAGPDAPHHGDSGPVHLMNVPPKDPTGVALLDACEQAGIPRAKFNTGTTVVNGANFFQINRRADGTRSSSSVSYIHPIVEQENFTLLTGLRARQLVFDADRRCTGVDIVDSAFGHTHRLTARNEVVLSTGAIDTPKLLMLSGIGPAAHLAEHGIEVLVDSPGVGEHLQDHPEGVVQFEAKQPMVAESTQWWEIGIFTPTEDGLDRPDLMMHYGSVPFDMNTLRHGYPTTENGFSLTPNVTHARSRGTVRLRSRDFRDKPMVDPRYFTDPEGHDMRVMVAGIRKAREIAAQPAMAEWTGRELSPGVEAQTDEELQDYIRKTHNTVYHPVGTVRMGAVEDEMSPLDPELRVKGVTGLRVADASVMPEHVTVNPNITVMMIGERCADLIR 2jc0 A 2.2 BS01 699 A 1 R200 C366 S368 L384 G410 N411 Q446 Y448 G449 R195 C361 S363 L379 G405 N406 Q441 Y443 G444 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=20uM remove_due_to_license_issue P26663 17269759 1563 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSSWFVAGYSGGDIYH 2jc0 A 2.2 BS02 699 A 2 L419 R422 M423 L474 H475 S476 Y477 R501 W528 K533 L414 R417 M418 L469 H470 S471 Y472 R496 W523 K528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=20uM remove_due_to_license_issue P26663 17269759 1564 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSSWFVAGYSGGDIYH 2jdh A 1.1 BS01 FUC A 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 17623286 1115 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdh B 1.1 BS01 FUC E 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 17623286 2 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdk A 1.1 BS01 FUC A 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 17623286 1115 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdk B 1.1 BS01 FUC E 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 17623286 2 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdm B 1.7 BS03 MFU B 1 A22 S23 D96 D99 D101 D104 A22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=3.96uM remove_due_to_license_issue Q9HYN5 17540045 1117 ATQGVFTLPANTRFGVTAFANASGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdo A 1.8 BS02 I5S A 1 G159 K160 G161 G164 K165 V166 A179 K181 M229 A232 E279 N280 M282 D293 G14 K15 G16 G19 K20 V21 A34 K36 M84 A87 E134 N135 M137 D148 D275 K277 N280 D293 T313 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.23uM remove_due_to_license_issue IC50=260nM P31751 17275837 1480 KVTMNDFDYLKLLGKGTFGKVILVREKATGRYYAMKILRKEVIIAKDEVAHTVTESRVLQNTRHPFLTALKYAFQTHDRLCFVMEYANGGELFFHLSRERVFTEERARFYGAEIVSALEYLHSRDVVYRDIKLENLMLDKDGHIKITDFGLCKEGISDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHERLFELILMEEIRFPRTLSPEAKSLLAGLLKKDPKQRLGGGPSDAKEVMEHRFFLSINWQDVVQKKLLPPFKPQVTSEVDTRYFDDEFTAQSITMFEDFDYIADW 2jdp A 1.3 BS01 MFU A 1 S22 A23 D96 D99 D101 D104 S22 A23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=0.25uM remove_due_to_license_issue Q9HYN5 17540045 1115 ATQGVFTLPANTRFGVTAFANSAGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdp B 1.3 BS01 MFU B 1 S22 A23 D96 D99 D101 D104 S22 A23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=0.25uM remove_due_to_license_issue Q9HYN5 17540045 1115 ATQGVFTLPANTRFGVTAFANSAGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jds A 2.0 BS02 L20 A 1 G52 G55 R56 A70 K72 M120 E121 Y122 N171 L173 T183 D184 F327 G39 G42 R43 A57 K59 M107 E108 Y109 N158 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=6.3nM remove_due_to_license_issue IC50=6nM P00517 17275837 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2jdt A 2.15 BS02 I5S A 1 L49 G50 T51 G52 G55 R56 V57 A70 Y122 A123 E127 E170 N171 M173 T183 D184 F327 L35 G36 T37 G38 G41 R42 V43 A56 Y108 A109 E113 E156 N157 M159 T169 D170 F313 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue IC50=170nM P00517 17275837 1351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2jdu C 1.5 BS03 MFU C 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=0.19uM remove_due_to_license_issue Q9HYN5 17540045 1117 ATQGVFTLPANTRFGVTAFANSSNTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdu D 1.5 BS03 MFU D 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 Kd=0.19uM remove_due_to_license_issue Q9HYN5 17540045 1117 ATQGVFTLPANTRFGVTAFANSSNTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 2jdv A 2.08 BS02 L20 A 1 L49 G50 V57 A70 K72 M120 A123 E127 N171 M173 T183 D184 F327 L35 G36 V43 A56 K58 M106 A109 E113 N157 M159 T169 D170 F313 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue IC50=6nM P00517 17275837 1351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2jew A 1.4 BS03 720 A 1 E72 N144 R145 H196 Y198 D255 E270 E67 N139 R140 H192 Y194 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 Ki=206nM remove_due_to_license_issue Ki=206nM P09955 17990866 1310 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2jf4 A 2.2 BS01 VDM A 1 F153 Y157 W159 D160 N196 R205 R277 E279 G310 D312 W447 E511 Y512 F518 W520 F106 Y110 W112 D113 N149 R158 R230 E232 G263 D265 W400 E464 Y465 F471 W473 3.2.1.28 0004555,0005975,0005991,0005993,0006974,0016798,0030288,0042597,0071474 Kd=7nM remove_due_to_license_issue P13482 17455176 1548 PQPPDILLGPLFNDVQNAKLFPDQKTFADAVPNSDPLMILADYRMQQNQSGFDLRHFVNVNFTLPQSLREHIDGLWPVLTRSTENTEKWDSLLPLPEPYVVPGGRFREVYYWDSYFTMLGLAESGHWDKVADMVANFAHEIDTYGHIPNGNRSYYLSRSQPPFFALMVELLAQHEGDAALKQYLPQMQKEYAYWMDGVENLQAGQQEKRVVKLQDGTLLNRYWDDRDTPRPESWVEDIATAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDNPQQLNTLRTTSIVPVDLNSLMFKMEKILARASKAAGDNAMANQYETLANARQKGIEKYLWNDQQGWYADYDLKSHKVRNQLTAAALFPLYVNAAAKDRANKMATATKTHLLQPGGLNTTSVKSGQQWDAPNGWAPLQWVATEGLQNYGQKEVAMDISWHFLTNVQHTYDREKKLVEKYDVSTTGTGGGGGEYPLQDGFGWTNGVTLKMLDLICPKEQPCDNVPATRP 2jfh A 1.97 BS01 LK1 A 1 T36 R37 G73 H183 K348 A414 S415 L416 N421 F422 H439 T36 R37 G73 H183 K339 A405 S406 L407 N412 F413 H430 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 Ki=870uM remove_due_to_license_issue IC50=7.10e+5nM P14900 17507028 1441 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRCVSFGVNMGDYHLNETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2jfz A 1.86 BS01 003 A 1 V10 G11 F13 S152 H183 L186 Q248 W252 V10 G11 F13 S152 H183 L186 Q248 W252 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 Ki=5.8uM remove_due_to_license_issue Q9ZLT0 17568739 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLKL 2jg0 A 1.5 BS01 TTZ A 1 R152 F153 Y157 W159 D160 N196 Y202 R205 R277 E279 A307 G310 D312 W447 E511 Y512 F518 W520 R112 F113 Y117 W119 D120 N156 Y162 R165 R237 E239 A267 G270 D272 W407 E471 Y472 F478 W480 3.2.1.28 0004555,0005975,0005991,0005993,0006974,0016798,0030288,0042597,0071474 Kd=15nM remove_due_to_license_issue P13482 17455176 1548 PQPPDILLGPLFNDVQNAKLFPDQKTFADAVPNSDPLMILADYRMQQNQSGFDLRHFVNVNFTLPKYVPPEGQSLREHIDGLWPVLTRSTENTEKWDSLLPLPEPYVVPGGRFREVYYWDSYFTMLGLAESGHWDKVADMVANFAHEIDTYGHIPNGNRSYYLSRSQPPFFALMVELLAQHEGDAALKQYLPQMQKEYAYWMDGVENLQAGQQEKRVVKLQDGTLLNRYWDDRDTPRPESWVEDIATAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDNPQQLNTLRTTSIVPVDLNSLMFKMEKILARASKAAGDNAMANQYETLANARQKGIEKYLWNDQQGWYADYDLKSHKVRNQLTAAALFPLYVNAAAKDRANKMATATKTHLLQPGGLNTTSVKSGQQWDAPNGWAPLQWVATEGLQNYGQKEVAMDISWHFLTNVQHTYDREKKLVEKYDVSTTGTGGGGGEYPLQDGFGWTNGVTLKMLDLICPKEQPCDNVPATRP 2jg8 D 2.05 BS01 SEP D 1 Q160 R162 Q71 R73 ? Kd=37nM remove_due_to_license_issue P02745 18250442 1223 QPRPAFSAIRRNPPMGGNVVIFDTVITNQEEPYQNHSGRFVCTVPGYYYFTFQVLSQWEICLSIVSSSRGQVRRSLGFCDTTNKGLFQVVSGGMVLQLQQGDQVWVEKDPKKGHIYQGSEADSVFSGFLIFPS 2jgs A 1.9 BS01 BTN A 1 W28 F30 S31 S33 T35 W55 M76 S108 Y125 T127 W25 F27 S28 S30 T32 W49 M70 S87 Y104 T106 ? 0009374 Kd=0.000000064M remove_due_to_license_issue P02701 18381715 1001 ESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDKEVLKTMWLLRSSVNDIGDDWKATRVGIMIFTRCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYITAVT 2jgs B 1.9 BS01 BTN B 1 W28 F30 S31 S33 T35 W55 M76 S108 Y125 T127 W28 F30 S31 S33 T35 W55 M76 S94 Y111 T113 ? 0009374 Kd=0.000000064M remove_due_to_license_issue P02701 18381715 1001 GSKESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGIMIFTRLCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYITAVT 2jgs D 1.9 BS01 BTN D 1 W28 F30 S31 S33 T35 W55 M76 S108 Y125 T127 W25 F27 S28 S30 T32 W52 M73 S91 Y108 T110 ? 0009374 Kd=0.000000064M remove_due_to_license_issue P02701 18381715 1001 ESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGIMIFTRLCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYITAVT 2jh0 D 1.7 BS03 701 D 1 H57 Y60A W60D D189 A190 E192 V213 W215 G216 G219 C220 G226 F227 Y228 H43 Y47 W50 D192 A193 E195 V218 W220 G221 G223 C224 G231 F232 Y233 3.4.21.5 0004252,0005509,0006508,0007596 Ki=2nM remove_due_to_license_issue Ki=2nM P00734 17336062 1247 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2jh5 D 2.5 BS04 895 D 1 H57 Y60A W60D L99 D189 A190 C191 E192 V213 W215 G216 G219 C220 G226 F227 H43 Y47 W50 L96 D191 A192 C193 E194 V217 W219 G220 G222 C223 G230 F231 3.4.21.5 0004252,0005509,0006508,0007596 Ki=367nM remove_due_to_license_issue Ki=367nM P00734 17336062 1249 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2jh6 D 2.21 BS04 894 D 1 H57 Y60A W60D L99 D189 A190 E192 V213 W215 G216 G219 C220 G226 F227 H43 Y47 W50 L96 D192 A193 E195 V218 W220 G221 G223 C224 G231 F232 3.4.21.5 0004252,0005509,0006508,0007596 Ki=17nM remove_due_to_license_issue Ki=17nM P00734 17336062 1249 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2jiu A 3.05 BS01 AEE A 1 L718 A743 K745 L792 M793 P794 G796 D800 L844 L23 A48 K50 L97 M98 P99 G101 D105 L149 D837 A839 R841 N842 D855 G874 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=5.3nM, IC50=2nM P00533 18227510 2017 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPVVDADE 2jiw A 1.95 BS01 BEU A 1 K166 D242 D243 Y282 T310 W337 N339 V342 D344 Y345 K163 D239 D240 Y279 T307 W334 N336 V339 D341 Y342 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 17728868 1594 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPH 2jj3 A 2.28 BS01 JJ3 A 1 M295 L298 T299 A302 E305 L339 F356 H475 L476 V487 M29 L32 T33 A36 E39 L73 F90 H202 L203 V212 ? 0003677,0004879,0006355 Ki=0.28nM remove_due_to_license_issue Ki=0.28nM Q92731 17662603 1499 DALSPEQLVLTLLEAEPPHVLISRPASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKNVVPVYDLLLEMLNAH 2jjb A 1.9 BS01 3CU A 1 F153 W159 D160 G310 D312 W447 F518 W520 F113 W119 D120 G270 D272 W407 F476 W478 3.2.1.28 0004555,0005975,0005991,0005993,0006974,0016798,0030288,0042597,0071474 remove_due_to_license_issue P13482 19123216 1547 VTPQPPDILLGPLFNDVQNAKLFPDQKTFADAVPNSDPLMILADYRMQQNQFDLRHFVNVNFTLPKYVPPEGQSLREHIDGLWPVLTRSTENTEKWDSLLPLPEPYVVPGGRFREVYYWDSYFTMLGLAESGHWDKVADMVANFAHEIDTYGHIPNGNRSYYLSRSQPPFFALMVELLAQHEGDAALKQYLPQMQKEYAYWMDGVENLQAGQQEKRVVKLQDGTLLNRYWDDRDTPRPESWVEDIATAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDNPQQLNTLRTTSIVPVDLNSLMFKMEKILARASKAAGDNAMANQYETLANARQKGIEKYLWNDQQGWYADYDLKSHKVRNQLTAAALFPLYVNAAAKDRANKMATATKTHLLQPGGLNTTSVKSGQQWDAPNGWAPLQWVATEGLQNYGQKEVAMDISWHFLTNVQHTYDREKKLVEKYDVSTTGTGGGEYPLQDGFGWTNGVTLKMLDLICPKEQPCDNVPATR 2jjb A 1.9 BS02 GLC A 1 R152 Y157 N196 Y202 R205 R277 E279 D312 R112 Y117 N156 Y162 R165 R237 E239 D272 3.2.1.28 0004555,0005975,0005991,0005993,0006974,0016798,0030288,0042597,0071474 remove_due_to_license_issue P13482 19123216 1548 VTPQPPDILLGPLFNDVQNAKLFPDQKTFADAVPNSDPLMILADYRMQQNQFDLRHFVNVNFTLPKYVPPEGQSLREHIDGLWPVLTRSTENTEKWDSLLPLPEPYVVPGGRFREVYYWDSYFTMLGLAESGHWDKVADMVANFAHEIDTYGHIPNGNRSYYLSRSQPPFFALMVELLAQHEGDAALKQYLPQMQKEYAYWMDGVENLQAGQQEKRVVKLQDGTLLNRYWDDRDTPRPESWVEDIATAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDNPQQLNTLRTTSIVPVDLNSLMFKMEKILARASKAAGDNAMANQYETLANARQKGIEKYLWNDQQGWYADYDLKSHKVRNQLTAAALFPLYVNAAAKDRANKMATATKTHLLQPGGLNTTSVKSGQQWDAPNGWAPLQWVATEGLQNYGQKEVAMDISWHFLTNVQHTYDREKKLVEKYDVSTTGTGGGEYPLQDGFGWTNGVTLKMLDLICPKEQPCDNVPATR 2jjk A 2.0 BS01 R15 A 1 V17 M18 G21 G26 G28 L30 T31 V9 M10 G13 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=9nM remove_due_to_license_issue IC50=4nM P09467 18650089 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2jjk C 2.0 BS01 R15 A 1 V17 G21 R22 G26 T27 G28 L30 T31 M177 V9 G13 R14 G18 T19 G20 L22 T23 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=4nM P09467 18650089 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2jk7 A 2.82 BS01 BI6 A 1 K297 V298 G306 L307 T308 D309 W310 E314 W323 T345 K48 V49 G57 L58 T59 D60 W61 E65 W74 T96 2.3.2.27 remove_due_to_license_issue Ki=67nM P98170 18954041 1346 FPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLT 2jke A 1.7 BS01 NOJ A 1 W331 E391 W397 H437 E439 K467 V471 H507 E508 E526 E532 W292 E352 W358 H398 E400 K428 V432 H468 E469 E487 E493 3.2.1.3 0000272,0004339,0004558,0005509,0005886,0005983,0016798,0030246,0042597,0046872 Ki=59uM remove_due_to_license_issue G8JZS4 18848471 1727 QQKLTSPDNNLVMTFQVDSKGAPTYELTYKNKVVIKPSTLGLELKKEDSKTNLYDGFEVKDTQTATFDETWQPVWGEEKEIRNHYNELAVTLYQPMNDRSIVIRFRLFNDGLGFRYEFPQQKSLNYFVIKEEHSQFGMNGDHIAFWIPGDYDTQEYDYTISRLSEIRGLMKEAITPNSSQTPFSQTGVQTALMMKTDDGLYINLHEAALVDYSCMHLNLDDKNMVFESWLTPDAKGDKGYMQTPCNTPWRTIIVSDDARNILASRITLNLNEPCKIADAASWVKPVKYIGVWWDMITGKGSWAYTDELTSVKLGETDYSKTKPNGKHSANTANVKRYIDFAAAHGFDAVLVEGWNEGWEDWFGNSKDYVFDFVTPYPDFDVKEIHRYAARKGIKMMMHHETSASVRNYERHMDKAYQFMADNGYNSVKSGYVGNIIPRGEHHYGQWMNNHYLYAVKKAADYKIMVNAHEATRPTGICRTYPNLIGNESARGTEYESFGGNKVYHTTILPFTRLVGGPMDYTPGIFETHCNKMNPANNSQVRSTIARQLALYVTMYSPLQMAADIPENYERFMDAFQFIKDVALDWDETNYLEAEPGEYITIARKAKDTDDWYVGCTAGENGHTSKLVFDFLTPGKQYIATVYADAKDADWKENPQAYTIKKGILTNKSKLNLHAANGGGYAISIKEV 2jkh A 1.25 BS01 BI7 A 1 Y99 F174 D189 A190 C191 Q192 V213 W215 G216 G226 Y228 Y85 F162 D179 A180 C181 Q182 V203 W205 G206 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=9nM remove_due_to_license_issue P00742 19101972 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2jkk A 2.0 BS01 BI9 A 1 I428 A452 L501 C502 G505 N551 L553 D564 L567 I16 A40 L89 C90 G93 N139 L141 D152 L155 D546 A548 R550 N551 D564 D134 A136 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 ic50=6.24nM remove_due_to_license_issue Q00944 19030106 1686 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEK 2jkm A 2.31 BS01 BII A 1 I428 V436 A452 K454 L501 C502 G505 L553 I16 V24 A40 K42 L89 C90 G93 L141 D546 A548 R550 N551 D564 D134 A136 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 ic50=17.76nM remove_due_to_license_issue Q00944 19030106 1687 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ 2jko A 1.65 BS01 BIJ A 1 R426 I428 A452 C502 T503 G505 L553 G563 D564 L567 R12 I14 A38 C88 T89 G91 L139 G149 D150 L153 D546 A548 R550 N551 D564 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7.7nM remove_due_to_license_issue Q00944 19030106 1687 YEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ 2jkp A 1.99 BS01 CTS A 1 W331 W341 E391 W397 W400 H437 E439 K467 V471 H507 E508 E526 E532 W292 W302 E352 W358 W361 H398 E400 K428 V432 H468 E469 E487 E493 3.2.1.3 0000272,0004339,0004558,0005509,0005886,0005983,0016798,0030246,0042597,0046872 Ki=59uM remove_due_to_license_issue G8JZS4 18848471 1727 QQKLTSPDNNLVMTFQVDSKGAPTYELTYKNKVVIKPSTLGLELKKEDSKTNLYDGFEVKDTQTATFDETWQPVWGEEKEIRNHYNELAVTLYQPMNDRSIVIRFRLFNDGLGFRYEFPQQKSLNYFVIKEEHSQFGMNGDHIAFWIPGDYDTQEYDYTISRLSEIRGLMKEAITPNSSQTPFSQTGVQTALMMKTDDGLYINLHEAALVDYSCMHLNLDDKNMVFESWLTPDAKGDKGYMQTPCNTPWRTIIVSDDARNILASRITLNLNEPCKIADAASWVKPVKYIGVWWDMITGKGSWAYTDELTSVKLGETDYSKTKPNGKHSANTANVKRYIDFAAAHGFDAVLVEGWNEGWEDWFGNSKDYVFDFVTPYPDFDVKEIHRYAARKGIKMMMHHETSASVRNYERHMDKAYQFMADNGYNSVKSGYVGNIIPRGEHHYGQWMNNHYLYAVKKAADYKIMVNAHEATRPTGICRTYPNLIGNESARGTEYESFGGNKVYHTTILPFTRLVGGPMDYTPGIFETHCNKMNPANNSQVRSTIARQLALYVTMYSPLQMAADIPENYERFMDAFQFIKDVALDWDETNYLEAEPGEYITIARKAKDTDDWYVGCTAGENGHTSKLVFDFLTPGKQYIATVYADAKDADWKENPQAYTIKKGILTNKSKLNLHAANGGGYAISIKEV 2jkq A 2.6 BS01 VG8 A 1 I428 A452 L501 C502 T503 G505 E506 N551 L553 G563 D564 L567 I15 A39 L88 C89 T90 G92 E93 N138 L140 G150 D151 L154 D546 A548 R550 N551 D564 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q00944 19030106 1687 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ 2jld A 2.35 BS02 AG1 A 1 I62 G63 F67 V70 A83 K85 L132 D133 Y134 V135 P136 T138 Q185 L188 C199 D200 I28 G29 F33 V36 A49 K51 L97 D98 Y99 V100 P101 T103 Q150 L153 C164 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50<0.04nM remove_due_to_license_issue P49841 19035373 1385 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQ 2jle A 2.9 BS01 I15 A 1 P95 L100 K101 K103 Y181 Y188 F227 W229 L234 Y318 P95 L100 K101 K103 Y181 Y188 F227 W229 L234 Y318 3.1.26.13 0003676,0003677,0003964,0004190,0004519,0004523,0006278,0006310,0006508,0015074,0035613,0042802,0044826,0046718,0046872,0075713 remove_due_to_license_issue Q72547 19175319 1546 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGN 2jle B 2.9 BS01 I15 A 1 Q428 L429 Q414 L415 3.1.26.13 0003676,0003677,0003964,0004190,0004519,0004523,0006278,0006310,0006508,0015074,0035613,0042802,0044826,0046718,0046872,0075713 remove_due_to_license_issue Q72547 19175319 1546 SPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQL 2jnp A -1.00 BS05 NGH A 1 L164 A165 H166 H201 E202 H205 H211 L77 A78 H79 H114 E115 H118 H124 H201 E202 H205 H211 H114 E115 H118 H124 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=132nM, IC50=6500nM P08254 17710450 253 GIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGP 2jpp A -1.00 BS01 rna C 0 M1 L2 I3 L4 T5 M1 L2 I3 L4 T5 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 17704818 1 ~ 20 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQA 2jpp A -1.00 BS02 rna D 0 L23 G27 Q28 Q29 R31 A36 P37 V40 A41 V42 H43 R44 I47 R50 I51 L23 G27 Q28 Q29 R31 A36 P37 V40 A41 V42 H43 R44 I47 R50 I51 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 17704818 1 ~ 20 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQA 2jpp B -1.00 BS01 rna C 0 L23 G27 Q28 Q29 R31 A36 P37 K38 V40 A41 V42 H43 R44 I47 R50 I51 L23 G27 Q28 Q29 R31 A36 P37 K38 V40 A41 V42 H43 R44 I47 R50 I51 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 17704818 1 ~ 20 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQA 2jpp B -1.00 BS02 rna D 0 M1 L2 I3 L4 T5 M1 L2 I3 L4 T5 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 17704818 1 ~ 20 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQA 2jsd A -1.00 BS05 NGH A 1 T188 L189 A190 H226 E227 H230 H236 P246 Y248 T76 L77 A78 H114 E115 H118 H124 P134 Y136 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue O60882 17869250 277 GEPKWKKNTLTYRISKYTPSMSSVEVDKAVEMALQAWSSAVPLSFVRINSGEADIMISFENGDHGDSYPFDGPRGTLAHAFAPGEGLGGDTHFDNAEKWTMGTNGFNLFTVAAHEFGHALGLAHSTDPSALMYPTYKYKNPYGFHLPKDDVKGIQALYGP 2jst B -1.00 BS01 HLT A 1 W15 L18 W15 L18 remove_due_to_license_issue 18310239 101 MKKLREEAAKLFEEWKKLAEEAAKLLEGGGGGGGGELMKLCEEAAKKAEELFKLAEERLKKL 2jt5 A -1.00 BS05 JT5 A 1 N162 V163 L164 A165 L197 H201 E202 H205 H211 L218 Y220 P221 L222 Y223 N75 V76 L77 A78 L110 H114 E115 H118 H124 L131 Y133 P134 L135 Y136 H201 E202 H205 H211 H114 E115 H118 H124 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P08254 17710450 1 GIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGP 2jt6 A -1.00 BS05 JT6 A 1 H201 E202 H205 Y220 Y223 H114 E115 H118 Y133 Y136 H201 E202 H205 H211 H114 E115 H118 H124 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Kd=110nM, IC50=47nM P08254 17710450 1 GIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGP 2jxi A -1.00 BS01 dna C 0 R15 P29 H30 I33 R15 P29 H30 I33 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue Q88D80 18767154 1 ~ 14 MATTTLGVKLDDPTRERLKAAAQSIDRTPHWLIKQAIFNYLEKLE 2jxi A -1.00 BS02 dna D 0 T4 T5 L6 G7 T4 T5 L6 G7 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue Q88D80 18767154 15 ~ 28 MATTTLGVKLDDPTRERLKAAAQSIDRTPHWLIKQAIFNYLEKLE 2jxi B -1.00 BS01 dna C 0 T49 L51 G52 K64 T4 L6 G7 K19 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue Q88D80 18767154 1 ~ 14 MATTTLGVKLDDPTRERLKAAAQSIDRTPHWLIKQAIFNYLEKLE 2jxi B -1.00 BS02 dna D 0 R60 T73 P74 H75 R15 T28 P29 H30 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue Q88D80 18767154 15 ~ 28 MATTTLGVKLDDPTRERLKAAAQSIDRTPHWLIKQAIFNYLEKLE 2jxr A 2.4 BS02 2Z3 A 1 Q13 D32 G34 Y75 G76 T77 I120 D215 G217 T218 S219 Q14 D33 G35 Y76 G77 T78 I121 D218 G220 T221 S222 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D218 T221 3.4.23.25 0000324,0004190,0006508 Ki=90nM remove_due_to_license_issue P07267 9135120 327 GGHDVPLTNYLNAQYYTDITLGTPPQNFKVILDTGSSNLWVPSNECGSLACFLHSKYDHEASSSYKANGTEFAIQYGTGSLEGYISQDTLSIGDLTIPKQDFAEATSEPGLTFAFGKFDGILGLGYDTISVDKVVPPFYNAIQQDLLDEKRFAFYLGDTSKDTENGGEATFGGIDESKFKGDITWLPVRRKAYWEVKFEGIGLGDEYAELESHGAAIDTGTSLITLPSGLAEMINAEIGAKKGWTGQYTLDCNTRDNLPDLIFNFNGYNFTIGPYDYTLEVSGSCISAITPMDFPEPVGPLAIVGDAFLRKYYSIYDIGNNAVGLAKAI 2k0g A -1.00 BS01 CMP A 1 F296 G297 M299 A300 R307 S308 R348 F83 G84 M86 A87 R94 S95 R135 ? 0005221 remove_due_to_license_issue Q98GN8 19465888 370 GSQEVRRGDFVRNWQLVAAVPLFQKLGPAVLVEIVRALRARTVPAGAVICRIGEPGDRMFFVVEGSVSVATPNPVELGPGAFFGEMALISGEPRSATVSAATTVSLLSLHSADFQMLCSSSPEIAEIFRKTALERRGAAASA 2k0x A -1.00 BS01 PNS A 1 D41 S42 L43 D41 S42 L43 ? 0000035,0000036,0005829,0006633,0009245,0016020,0017000 remove_due_to_license_issue Q02054 18770515 87 MATLLTTDDLRRALVESAGETDGTDLSGDFLDLRFEDIGYDSLALMETAARLESRYGVSIPDDVAGRVDTPRELLDLINGALAEAA 2k2g A -1.00 BS03 DSV A 1 L181 L214 T215 H218 H222 H228 V235 M236 L83 L116 T117 H120 H124 H130 V137 M138 H218 E219 H222 H228 H120 E121 H124 H130 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 18425585 1 MFREMPGGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2k31 A -1.00 BS01 35G A 1 S176 F178 F195 D196 I211 I219 Y236 F241 N242 V245 T249 I275 S23 F25 F42 D43 I58 I66 Y83 F88 N89 V92 T96 I122 3.1.4.35 remove_due_to_license_issue Q8CG03 18534985 1 DVTALCHKIFLHIHGLISADRYSLFLVCEDSSKDKFLISRLFDVAEGSTLEEASNNCIRLEWNKGIVGHVAAFGEPLNIKDAYEDPRFNAEVDQITGYKTQSILCMPIKNHREEVVGVAQAINKKSGNGGTFTEKDEKDFAEYLAFCGE 2k4i A -1.00 BS01 PBU A 1 L21 R22 K27 H33 W36 S77 N80 T81 L20 R21 K26 H32 W35 S76 N79 T80 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0005198 remove_due_to_license_issue P04584 18657545 300 GARNSVLRGKKADELERIRLRPGGKKKYRLKHIVWAANKLDRFGLAESLLESKEGCQKILTVLDPMVPTGSENLKSLFNTVCVIWCIHAEEKVKDTEGAKQIVRRHLVAETGTAEKMPSTSRPTAPSSEKGGNY 2k62 A -1.00 BS01 ITL A 1 Y14 F17 L18 A22 L23 A31 I34 R55 D74 I111 F113 L118 R120 Y14 F17 L18 A22 L23 A31 I34 R55 D74 I111 F113 L118 R120 ? 0005504,0005634,0005737,0005829,0008289,0015908 remove_due_to_license_issue P80226 18939814 202 AFSGTWQVYAQENYEEFLKALALPEDLIKMARDIKPIVEIQQKGDDFVVTSKTPRQTVTNSFTLGKEADITTMDGKKLKCTVHLANGKLVTKSEKFSHEQEVKGNEMVETITFGGVTLIRRSKRV 2k7f A -1.00 BS01 dna B 0 Y385 R388 K436 T438 R452 S454 G455 Q456 S457 Y11 R14 K62 T64 R78 S80 G81 Q82 S83 ? remove_due_to_license_issue P35251 20081198 1 ~ 14 KRTNYQAYRSYLNREGPKALGSKEIPKGAENCLEGLIFVITGVLESIERDEAKSLIERYGGKVTGNVSKKTNYLVMGRDSGQSKSDKAAALGTKIIDEDGLLNLIRNLE 2k7f A -1.00 BS02 dna C 0 K375 Y379 R383 I414 T415 R423 G439 N440 K458 K1 Y5 R9 I40 T41 R49 G65 N66 K84 ? remove_due_to_license_issue P35251 20081198 19 ~ 28 KRTNYQAYRSYLNREGPKALGSKEIPKGAENCLEGLIFVITGVLESIERDEAKSLIERYGGKVTGNVSKKTNYLVMGRDSGQSKSDKAAALGTKIIDEDGLLNLIRNLE 2kae A -1.00 BS01 dna C 0 I123 R124 R129 I141 Y142 R144 K145 Y146 R150 Y158 K162 Q166 I13 R14 R19 I31 Y32 R34 K35 Y36 R40 Y48 K52 Q56 0006355,0008270,0043565 remove_due_to_license_issue 19095651 21 ~ 40 SFQCSNCSVTETIRWRNIRSKEGIQCNACFIYQRKYNKTRPVTAVNKYQKRKLKVQ 2kae A -1.00 BS02 dna B 0 R124 W125 R126 N127 I128 I141 R144 T153 A154 N156 K157 Y158 K160 R161 R14 W15 R16 N17 I18 I31 R34 T43 A44 N46 K47 Y48 K50 R51 0006355,0008270,0043565 remove_due_to_license_issue 19095651 1 ~ 20 SFQCSNCSVTETIRWRNIRSKEGIQCNACFIYQRKYNKTRPVTAVNKYQKRKLKVQ 2kaw A -1.00 BS01 SUZ A 1 F14 L15 G16 I17 S18 I19 V71 L74 R75 F14 L15 G16 I17 S18 I19 V71 L74 R75 ? 0016055 remove_due_to_license_issue P51141 19637179 91 NIITVTLNMERHHFLGISIVGQSNDRGDGGIYIGSIMKGGAVAADGRIEPGDMLLQVNDVNFENMSNDDAVRVLREIVSQTGPISLTVAK 2kce A 2.2 BS02 D16 A 1 H51 S54 I79 W80 W83 D169 G173 F176 Y209 H51 S54 I79 W80 W83 D169 G173 F176 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=0.67uM remove_due_to_license_issue IC50=2300nM P0A884 8939755 566 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 2kce B 2.2 BS03 D16 B 1 H51 S54 I79 W80 W83 D169 G173 F176 Y209 A263 H51 S54 I79 W80 W83 D169 G173 F176 Y209 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=0.67uM remove_due_to_license_issue IC50=2300nM P0A884 8939755 568 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 2kdh A -1.00 BS02 KDH A 1 F104 L121 F156 M157 V160 F15 L32 F67 M68 V71 ? 0005509 remove_due_to_license_issue P63316 19542563 1 MGKSEEELSDLFRMFDKNADGYIDLDELKIMLQATGETITEDDIEELMKDGDKNNDGRIDYDEFLEFMKGVE 2kdz A -1.00 BS01 dna B 0 K3 F4 T33 R34 N35 Q38 E41 R42 N88 N92 R93 M96 K3 F4 T33 R34 N35 Q38 E41 R42 N88 N92 R93 M96 ? remove_due_to_license_issue Q58HP2 19246540 1 ~ 16 KVKFTEEEDLKLQQLVMRYGAKDWIRISQLMITRNPRQCRERWNNYINPALRTDPWSPEEDMLLDQKYAEYGPKWNKISKFLKNRSDNNIRNRWMMIARHRAKHQKS 2kdz A -1.00 BS02 dna C 0 V2 K22 R37 Q38 R40 P73 W75 N76 D87 N88 R91 V2 K22 R37 Q38 R40 P73 W75 N76 D87 N88 R91 ? remove_due_to_license_issue Q58HP2 19246540 17 ~ 32 KVKFTEEEDLKLQQLVMRYGAKDWIRISQLMITRNPRQCRERWNNYINPALRTDPWSPEEDMLLDQKYAEYGPKWNKISKFLKNRSDNNIRNRWMMIARHRAKHQKS 2kei A -1.00 BS01 dna C 0 S16 Y17 Q18 R22 H29 V30 S31 K33 T34 L56 K59 S16 Y17 Q18 R22 H29 V30 S31 K33 T34 L56 K59 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kei A -1.00 BS02 dna D 0 T5 L6 Y7 Q18 S21 N25 Y47 P49 N50 A53 Q54 L56 A57 T5 L6 Y7 Q18 S21 N25 Y47 P49 N50 A53 Q54 L56 A57 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kei B -1.00 BS01 dna C 0 T5 L6 Y7 Y17 Q18 S21 N25 N50 A53 Q54 L56 A57 T5 L6 Y7 Y17 Q18 S21 N25 N50 A53 Q54 L56 A57 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kei B -1.00 BS02 dna D 0 S16 Q18 R22 H29 S31 T34 L56 S16 Q18 R22 H29 S31 T34 L56 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kej A -1.00 BS01 dna C 0 S16 Y17 Q18 R22 H29 V30 S31 T34 L56 Q60 S16 Y17 Q18 R22 H29 V30 S31 T34 L56 Q60 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kej A -1.00 BS02 dna D 0 T5 L6 Y7 Q18 S21 N25 Y47 N50 A53 Q54 L56 A57 K59 T5 L6 Y7 Q18 S21 N25 Y47 N50 A53 Q54 L56 A57 K59 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kej B -1.00 BS01 dna C 0 T5 L6 Y7 Y17 Q18 S21 A53 Q54 L56 A57 K59 T5 L6 Y7 Y17 Q18 S21 A53 Q54 L56 A57 K59 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kej B -1.00 BS02 dna D 0 S16 Q18 T19 R22 H29 V30 S31 T34 L56 S16 Q18 T19 R22 H29 V30 S31 T34 L56 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kek A -1.00 BS01 dna C 0 S16 Y17 Q18 R22 H29 S31 L56 A57 K59 S16 Y17 Q18 R22 H29 S31 L56 A57 K59 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kek A -1.00 BS02 dna D 0 T5 L6 Y7 Q18 S21 N25 Y47 P49 N50 A53 Q54 A57 G58 Q60 T5 L6 Y7 Q18 S21 N25 Y47 P49 N50 A53 Q54 A57 G58 Q60 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kek B -1.00 BS01 dna C 0 L6 Y7 Y17 R22 N25 K33 L56 A57 L6 Y7 Y17 R22 N25 K33 L56 A57 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kek B -1.00 BS02 dna D 0 S16 Q18 H29 S31 T34 L56 A57 S16 Q18 H29 S31 T34 L56 A57 ? 0003677,0006355 remove_due_to_license_issue P03023 19450607 -1 ~ 22 MKPVTLYDVAEYAGVSYQTVSRVVNQASHVSAKTREKVEAAMAELNYIPNRCAQQLAGKQSL 2kfx T -1.00 BS02 WW7 T 1 F27 I36 L41 M45 V72 F77 M80 M81 F27 I36 L41 M45 V72 F77 M80 M81 ? 0005509 remove_due_to_license_issue P63316 19419198 91 MDDIYKAAVEQLTEEQKNEFKAAFDIFVLGAEDGSISTKELGKVMRMLGQNPTPEELQEMIDEVDEDGSGTVDFDEFLVMMVRSMKDDS 2kfy A -1.00 BS01 rna B 0 K14 R16 G17 L18 W20 R52 S54 R75 R81 Y82 E84 V85 F86 K14 R16 G17 L18 W20 R52 S54 R75 R81 Y82 E84 V85 F86 ? 0003676,0003723 remove_due_to_license_issue P52597 20526337 1 ~ 6 MMLGPEGGEGFVVKLRGLPWSCSVEDVQNFLSDCTIHDGAAGVHFIYTREGRQSGEAFVELGSEDDVKMALKKDRESMGHRYIEVFKSHRTEMDWVLKHSGP 2kg0 A -1.00 BS01 rna B 0 R116 G117 L118 F120 K150 I151 H172 K173 R179 Y180 E182 F184 R14 G15 L16 F18 K48 I49 H70 K71 R77 Y78 E80 F82 ? 0003676,0003723 remove_due_to_license_issue P52597 20526337 1 ~ 6 NSADSANDGFVRLRGLPFGCTKEEIVQFFSGLEIVPNGITLPVDPEGKITGEAFVQFASQELAEKALGKHKERIGHRYIEVFKSSQEEVRSY 2kg1 A -1.00 BS01 rna B 0 R294 G295 P297 Y298 E330 D348 R349 R355 Y356 E358 L359 F360 R18 G19 P21 Y22 E54 D72 R73 R79 Y80 E82 L83 F84 ? 0003676,0003723 remove_due_to_license_issue P52597 20526337 1 ~ 6 GDSEFTVQSTTGHCVHMRGLPYKATENDIYNFFSPLNPVRVHIEIGPDGRVTGEADVEFATHEEAVAAMSKDRANMQHRYIELFLNSTTGASNGAYSSQVMQGMG 2kh9 A -1.00 BS01 rna B 0 T118 W120 T122 R148 L149 P150 R153 R158 Y162 K191 N194 T5 W7 T9 R35 L36 P37 R40 R45 Y49 K78 N81 ? 0003676,0003723 remove_due_to_license_issue P49960 20181740 49 ~ 54 MTECTLWMTNFPPSYTQRNIRDLLQDINVVALSIRLPSLRFNTSRRFAYIDVTSKEDARYCVEKLNGLKIEGYTLVTKVSNPLELE 2kkf A -1.00 BS01 dna B 0 K1147 R1150 S1152 R1154 N1183 K1186 Q1187 C1188 K1193 L1197 K1 R4 S6 R8 N37 K40 Q41 C42 K47 L51 2.1.1.-,2.1.1.364 0003677,0008270 remove_due_to_license_issue Q03164 20010842 101 ~ 112 KKGRRSRRCGQCPGCQVPEDCGVCTNCLDKPKFGGRNIKKQCCKMRKCQNLQWMPSK 2kkf A -1.00 BS02 dna C 0 K1147 K1148 R1150 R1151 T1171 I1184 K1185 K1186 K1203 K1 K2 R4 R5 T25 I38 K39 K40 K57 2.1.1.-,2.1.1.364 0003677,0008270 remove_due_to_license_issue Q03164 20010842 101 ~ 112 KKGRRSRRCGQCPGCQVPEDCGVCTNCLDKPKFGGRNIKKQCCKMRKCQNLQWMPSK 2kmk A -1.00 BS01 dna B 0 R13 T16 I23 H40 Q41 D44 I51 K65 Q69 K79 R13 T16 I23 H40 Q41 D44 I51 K65 Q69 K79 ? remove_due_to_license_issue Q07120 20153336 101 ~ 116 SFDCKICGKSFKRSSTLSTHLLIHSDTRPYPCQYCGKRFHQKSDMKKHTFIHTGEKPHKCQVCGKAFSQSSNLITHSRKHTG 2kmk A -1.00 BS02 dna C 0 R13 S15 S70 S71 I74 R13 S15 S70 S71 I74 ? remove_due_to_license_issue Q07120 20153336 201 ~ 216 SFDCKICGKSFKRSSTLSTHLLIHSDTRPYPCQYCGKRFHQKSDMKKHTFIHTGEKPHKCQVCGKAFSQSSNLITHSRKHTG 2kmx A -1.00 BS01 ATP A 1 E1081 H1086 L1088 I1182 G1183 E35 H40 L42 I136 G137 7.2.2.8 0000166 remove_due_to_license_issue Q04656 19917612 1232 SFTMHGTPVVNQVKVLTESNRISHHKILAIVGTAESNSEHPLGTAITKYCKQELDTETLGTCIDFQVVPGCGISCKVTNIEGLLHKNNWNIEDNNIKNASLVQIDASNEQSSTSSSMIIDAQISNALNAQQYKVLIGNREWMIRNGLVINNDVNDFMTEHERKGRTAVLVAVDDELCGLIAIADT 2ko0 A -1.00 BS01 dna B 0 M1 V2 Q3 Y14 F22 H23 K24 T28 K64 R65 L71 M1 V2 Q3 Y14 F22 H23 K24 T28 K64 R65 L71 ? 0043565 remove_due_to_license_issue Q9NVV9 20144952 1 ~ 16 MVQSCSAYGCKNRYDKDKPVSFHKFPLTRPSLCKEWEAAVRRKNFKPTKYSSICSEHFTPDSFKRESNNKLLKENAVPTIFLELVPR 2ko0 A -1.00 BS02 dna C 0 Q3 K11 F45 K46 P47 T48 Y50 S51 K70 Q3 K11 F45 K46 P47 T48 Y50 S51 K70 ? 0043565 remove_due_to_license_issue Q9NVV9 20144952 17 ~ 32 MVQSCSAYGCKNRYDKDKPVSFHKFPLTRPSLCKEWEAAVRRKNFKPTKYSSICSEHFTPDSFKRESNNKLLKENAVPTIFLELVPR 2ko7 A -1.00 BS01 JZF A 1 I67 W70 Y93 I67 W70 Y93 Y37 F47 D48 I67 Y93 F110 Y37 F47 D48 I67 Y93 F110 5.2.1.8 0003755,0006357,0006457,0046872,0140839,0140840 remove_due_to_license_issue Q63J95 21574961 130 GPGSMTVVTTESGLKYEDLTEGSGAEARAGQTVSVHYTGWLTDGQKFDSSKDRNDPFAFVLGGGMVIKGWDEGVQGMKVGGVRRLTIPPQLGYGARGAGGVIPPNATLVFEVELLDV 2kp8 A -1.00 BS01 XIG B 1 L56 L64 L56 L64 remove_due_to_license_issue 20004576 999 TSLIHSLIEESQNQQEKNEQELLELDGDGPQLLSGIVQQQNNLLRAIEAQQHLLQLTVWGIKQLQARILAVE 2kp8 B -1.00 BS01 XIG B 1 T101 S102 L103 V158 W159 K162 Q165 T1 S2 L3 V58 W59 K62 Q65 remove_due_to_license_issue 20004576 999 TSLIHSLIEESQNQQEKNEQELLELDGDGPQLLSGIVQQQNNLLRAIEAQQHLLQLTVWGIKQLQARILAVE 2kxn B -1.00 BS01 rna A 0 R111 F123 G124 S148 I149 V150 R159 F161 F163 Y165 R187 R188 R190 S194 I195 T196 K197 R198 P199 H200 R6 F18 G19 S43 I44 V45 R54 F56 F58 Y60 R82 R83 R85 S89 I90 T91 K92 R93 P94 H95 ? 0003676,0003723 remove_due_to_license_issue P62995 21399644 1 ~ 6 RHVGNRANPDPNCCLGVFGLSLYTTERDLREVFSKYGPIADVSIVYDQQSRRSRGFAFVYFENVDDAKEAKERANGMELDGRRIRVDFSITKRPH 2ky8 A -1.00 BS01 dna B 0 R24 R46 R22 R44 ? 0003677 remove_due_to_license_issue Q5EFL0 21531701 100 ~ 110 DKQGRTDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNAVDLSCFDFRTGKMM 2ky8 A -1.00 BS02 dna C 0 K32 R46 K30 R44 ? 0003677 remove_due_to_license_issue Q5EFL0 21531701 111 ~ 121 DKQGRTDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNAVDLSCFDFRTGKMM 2l1r A -1.00 BS03 SXK A 1 F27 L41 M60 M80 R83 C84 F27 L41 M60 M80 R83 C84 ? 0005509 remove_due_to_license_issue P63316 20801130 91 MDDIYKAAVEQLTEEQKNEFKAAFDIFVLGAEDGCISTKELGKVMRMLGQNPTPEELQEMIDEVDEDGSGTVDFDEFLVMMVRCMKDDS 2l2k B -1.00 BS01 rna A 0 P43 K46 N47 M50 E54 S70 H71 F75 R91 N92 K93 K94 K97 P1 K4 N5 M8 E12 S28 H29 F33 R49 N50 K51 K52 K55 3.5.4.37 remove_due_to_license_issue Q91ZS8 20946981 1 ~ 42 PSGKNPVMILNELRPGLKYDFLSESGESHAKSFVMSVVVDGQFFEGSGRNKKLAKARAAQSALATVFNLHL 2l3c A -1.00 BS01 rna B 0 K7 L10 M11 N14 E15 V31 H32 P34 T53 K54 K55 K58 K7 L10 M11 N14 E15 V31 H32 P34 T53 K54 K55 K58 3.5.4.37 remove_due_to_license_issue P51400 20946981 75 ~ 108 PGPVLPKNALMQLNEIKPGLQYMLLSQTGPVHAPLFVMSVEVNGQVFEGSGPTKKKAKLHAAEKALRSFVQFPN 2l41 A -1.00 BS01 rna B 0 R4 F6 N9 N34 K36 N37 F41 I68 E70 S72 R4 F6 N9 N34 K36 N37 F41 I68 E70 S72 ? 0003676,0003723 remove_due_to_license_issue P38996 21084293 78 ~ 81 PKSRLFIGNLPLKNVSKEDLFRIFSPYGHIMQINIKNAFGFIQFDNPQSVRDAIECESQEMNFGKKLILEVSSSNAR 2l4l A -1.00 BS01 dna B 0 F16 T24 R26 K33 C36 W37 Q45 M46 F6 T14 R16 K23 C26 W27 Q35 M36 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0008270 remove_due_to_license_issue P03366 21227929 123 ~ 126 KNVKCFNCGKEGHTARNCRAPRKKGCWKCGKEGHQMKDCTERQAN 2l65 A -1.00 BS01 MRP A 1 F65 M133 K135 G136 F65 M133 K135 G136 ? remove_due_to_license_issue Q8KNF0 17168523 627 NYDPFVRHSVTVKADRKTAFKTFLEGFPEWWPNNFRTTKVGAPLGVDKKGGRWYEIDEQGEEHTFGLIRKVDEPDTLVIGWRLNGFGRIDPDNSSEFTVTFVADGQKKTRVDVEHTHFDRMGTKHAKRVRNGMDKGWPTILQSFQDKIDEEGAKK 2l65 A -1.00 BS02 MTC A 1 F86 G87 F86 G87 ? remove_due_to_license_issue Q8KNF0 17168523 629 NYDPFVRHSVTVKADRKTAFKTFLEGFPEWWPNNFRTTKVGAPLGVDKKGGRWYEIDEQGEEHTFGLIRKVDEPDTLVIGWRLNGFGRIDPDNSSEFTVTFVADGQKKTRVDVEHTHFDRMGTKHAKRVRNGMDKGWPTILQSFQDKIDEEGAKK 2l84 A -1.00 BS01 J28 A 1 P1110 Q1113 L1120 Y1125 Y1167 R1173 P34 Q37 L44 Y49 Y91 R97 2.3.1.-,2.3.1.48 remove_due_to_license_issue IC50=5000nM, Kd=19600nM Q92793 21513889 201 GSHMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 2l8r A -1.00 BS01 APR A 1 D20 L21 F22 C33 I34 I44 P118 R119 I120 D125 Y150 L152 D18 L19 F20 C31 I32 I42 P116 R117 I118 D123 Y148 L150 3.2.2.-,3.5.1.- 0001883,0005515,0005634,0005654,0005694,0005730,0006974,0016787,0042278,0047407,0051725,0061463,0090734,0140291,0140293 remove_due_to_license_issue Q9Y530 21849506 186 SSLNEDPEGSRITYVKGDLFACPKTDSLAHCISEDCRMGAGIAVLFKKKFGGVQELLNQQKKSGEVAVLKRDGRYIYYLITKKRASHKPTYENLQKSLEAMKSHCLKNGVTDLSMPRIGCGLDRLQWENVSAMIEEVFEATDIKITVYTL 2l98 A -1.00 BS03 STL A 1 L117 L121 F153 F156 L28 L32 F64 F67 ? 0005509 remove_due_to_license_issue P63316 21226534 162 MGKSEEELSDLFRMFDKNADGYIDLDELKIMLQATGETITEDDIEELMKDGDKNNDGRIDYDEFLEFMKGVE 2lbs B -1.00 BS01 rna A 0 D367 M368 K371 Y375 S376 N419 I420 K421 D4 M5 K8 Y12 S13 N56 I57 K58 3.1.26.3 0003725,0006364 remove_due_to_license_issue Q02555 21742266 1 ~ 32 GSLDMNAKRQLYSLIGYASLRLHYVTVKKPTAVDPNSIVECRVGDGTVLGTGVGRNIKIAGIRAAENALRDKKMLDFYAKQRAAIPRSES 2lbv A -1.00 BS02 ACD A 1 W13 A37 I39 F41 V49 Y51 V85 Y92 I98 Y115 W13 A37 I39 F41 V49 Y51 V85 Y92 I98 Y115 ? 0005576,0036094,0042742,0045087,0050544,0070538,1903981 remove_due_to_license_issue Q9I9P7 21951132 300 MTVPDRSEIAGKWYVVALASNTEFFLREKDKMKMAMARISFLGEDELKVSYAVPKPNGCRKWETTFKKTSDDGEVYYSEEAKKKVEVLDTDYKSYAVIYATRVKDGRTLHMMRLYSRSPEVSPAATAIFRKLAGERNYTDEMVAMLPRQEECTVDEV 2ld5 A -1.00 BS01 dna B 0 K9 K10 R11 V12 K30 F31 Q56 R59 V60 K63 K3 K4 R5 V6 K24 F25 Q50 R53 V54 K57 ? 0000981,0003677,0006355 remove_due_to_license_issue Q62424 21829694 1 ~ 11 GRKKRVPYTKVQLKELEREYATNKFITKDKRRRISATTNLSERQVTIWFQNRRVKEKKVINKLKTTS 2ld5 A -1.00 BS02 dna C 0 R8 K10 R11 P13 Y14 Q50 I53 W54 N57 K61 K64 K68 R2 K4 R5 P7 Y8 Q44 I47 W48 N51 K55 K58 K62 ? 0000981,0003677,0006355 remove_due_to_license_issue Q62424 21829694 12 ~ 22 GRKKRVPYTKVQLKELEREYATNKFITKDKRRRISATTNLSERQVTIWFQNRRVKEKKVINKLKTTS 2leb A -1.00 BS01 rna B 0 M1 G4 R5 P6 K17 N20 D42 Y44 P46 R49 Y50 F57 F59 R61 A90 R91 G93 R94 P95 S98 H99 M1 G4 R5 P6 K17 N20 D42 Y44 P46 R49 Y50 F57 F59 R61 A90 R91 G93 R94 P95 S98 H99 ? 0003676,0003723 remove_due_to_license_issue Q01130 22002536 102 ~ 107 MSYGRPPPDVEGMTSLKVDNLTYRTSPDTLRRVFEKYGRVGDVYIPRDRYTKESRGFAFVRFHDKRDAEDAMDAMDGAVLDGRELRVQMARYGRPPDSHHS 2lec A -1.00 BS01 rna B 0 G4 R5 P6 K17 D42 Y44 P46 D48 R49 F57 F59 R61 R91 Y92 G93 R94 P95 S98 H99 G4 R5 P6 K17 D42 Y44 P46 D48 R49 F57 F59 R61 R91 Y92 G93 R94 P95 S98 H99 ? 0003676,0003723 remove_due_to_license_issue Q01130 22002536 102 ~ 107 MSYGRPPPDVEGMTSLKVDNLTYRTSPDTLRRVFEKYGRVGDVYIPRDRYTKESRGFAFVRFHDKRDAEDAMDAMDGAVLDGRELRVQMARYGRPPDSHHS 2lev A -1.00 BS01 dna B 0 R21 Q22 R24 R31 Q32 R34 ? remove_due_to_license_issue Q7DB51 22114557 1 ~ 15 SHHHHHHSMGNSSKGVYYRNEEGQTWSGVGRQPRWLKEALLNGMKKEDFLVKDTEEE 2lev A -1.00 BS02 dna C 0 Q14 W16 S17 G20 R21 P23 W25 Q24 W26 S27 G30 R31 P33 W35 ? remove_due_to_license_issue Q7DB51 22114557 16 ~ 30 SHHHHHHSMGNSSKGVYYRNEEGQTWSGVGRQPRWLKEALLNGMKKEDFLVKDTEEE 2lh8 A -1.00 BS01 VIB A 1 M48 M49 H50 D57 Y60 M14 M15 H16 D23 Y26 ? 0016020,0051260 remove_due_to_license_issue P04273 21848803 1 LGGYMLGSAMSRPMMHFGNDWEDRYYRENMNRYPNQVYYRPVDQYNNQNNFVHDCVNITIKQHTVTTTTKGENFTETDIKIMERVVEQMCTTQYQKESQAYYDG 2lha A -1.00 BS01 IHP A 1 Y311 I330 Y364 I367 G368 Y41 I60 Y94 I97 G98 ? 0016020 remove_due_to_license_issue P21579 22475172 1 EKLGDICFSLRYVPTAGKLTVVILEAKNLKKMDVGGLSDPYVKIHLMQNGKRLKKKKTTIKKNTLNPYYNESFSFEVPFEQIQKVQVVVTVLDYDKIGKNDAIGKVFVGYNSTGAELRHWSDMLANPRRPIAQWHTLQVEEEVDAMLAVKK 2li8 A -1.00 BS01 rna B 0 M129 K131 R132 R133 S134 D137 R138 Y140 H148 A149 K150 K159 K160 C161 H162 M170 V171 A172 M6 K8 R9 R10 S11 D14 R15 Y17 H25 A26 K27 K36 K37 C38 H39 M47 V48 A49 ? 0003676,0008270 remove_due_to_license_issue Q9H9Z2 22157959 1 ~ 7 PKGKSMQKRRSKGDRCYNCGGLDHHAKECKLPPQPKKCHFCQSISHMVASCPLKAQQGPSAQG 2liq A -1.00 BS01 MAG B 1 Y68 N102 Y103 Y68 N102 Y103 ? 0030246 remove_due_to_license_issue B3GA02 22615566 1 MGHHHHHHHHSGDSPAVTLSAGNYIIYNRVLSPRGEKLALTYPGRQRTPVTVSPLDGSSEQAWILRSYDSNSNTWTISPVGSPNSQIGWGAGNVPVVLPPNNYVWTLTLTSGGYNIQDGKRTVSWSLNNATAGEEVSIGADATFSGRWVIEKV 2liq A -1.00 BS02 FUC B 1 V104 G119 K120 V104 G119 K120 ? 0030246 remove_due_to_license_issue B3GA02 22615566 2 MGHHHHHHHHSGDSPAVTLSAGNYIIYNRVLSPRGEKLALTYPGRQRTPVTVSPLDGSSEQAWILRSYDSNSNTWTISPVGSPNSQIGWGAGNVPVVLPPNNYVWTLTLTSGGYNIQDGKRTVSWSLNNATAGEEVSIGADATFSGRWVIEKV 2lk1 A -1.00 BS01 AQN A 1 F15 R18 F22 D30 F15 R18 F22 D30 ? remove_due_to_license_issue P52756 22162216 32 KFEDWLCNKCCLNNFRKRLKCFRCGADKFD 2lkk A -1.00 BS01 OLA A 1 F15 M19 L28 K31 A54 S56 M74 F14 M18 L27 K30 A53 S55 M73 ? 0003682,0005324,0005504,0005515,0005543,0005634,0005654,0005737,0005782,0005829,0008289,0015908,0015909,0016209,0032000,0032052,0032991,0033552,0043066,0045179,0050892,0070062,0070301,0070538,0071456,0098869,1901363,2000117 remove_due_to_license_issue Kd=900nM P07148 22713574 128 SFSGKYQLQSQENFEAFMKAIGLPEELIQKGKDIKGVSEIVQNGKHFKFTITAGSKVIQNEFTVGEECELETMTGEKVKTVVQLEGDNKLVTTFKNIKSVTELNGDIITNTMTLGDIVFKRISKRI 2lkk A -1.00 BS02 OLA A 2 S39 F50 E72 F95 N111 M113 R122 S124 S38 F49 E71 F94 N110 M112 R121 S123 ? 0003682,0005324,0005504,0005515,0005543,0005634,0005654,0005737,0005782,0005829,0008289,0015908,0015909,0016209,0032000,0032052,0032991,0033552,0043066,0045179,0050892,0070062,0070301,0070538,0071456,0098869,1901363,2000117 remove_due_to_license_issue Kd=900nM P07148 22713574 129 SFSGKYQLQSQENFEAFMKAIGLPEELIQKGKDIKGVSEIVQNGKHFKFTITAGSKVIQNEFTVGEECELETMTGEKVKTVVQLEGDNKLVTTFKNIKSVTELNGDIITNTMTLGDIVFKRISKRI 2lko A -1.00 BS01 4IP A 1 V381 K383 L389 K390 K393 H419 V19 K21 L27 K28 K31 H57 ? 0007229 remove_due_to_license_issue Q96AC1 22030399 1228 GSHMGDITSIPELADYIKVFKPKKLTLKGYKQYWCTFKDTSISCYKSKEESSGTPAHQMNLRGCEVTPDVNISGQKFNIKLLIPVAEGMNEIWLRCDNEKQYAHWMAACRLASKGKTMADSSYNLEVQNILSFLKMQH 2lkx A -1.00 BS01 dna B 0 R3 R5 T6 K50 N51 R52 K55 R59 R5 R7 T8 K52 N53 R54 K57 R61 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99697 15895993 67 ~ 79 GSQRRQRTHFTSQQLQELEATFQRNRYPDMSTREEIAVWTNLTEARVRVWFKNRRAKWRKREEFIVTD 2lkx A -1.00 BS02 dna C 0 R2 R3 R5 Y25 M28 R31 K50 R53 R57 R4 R5 R7 Y27 M30 R33 K52 R55 R59 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99697 15895993 80 ~ 92 GSQRRQRTHFTSQQLQELEATFQRNRYPDMSTREEIAVWTNLTEARVRVWFKNRRAKWRKREEFIVTD 2ltt A -1.00 BS01 dna C 0 M1 L5 F7 A20 K21 W23 W32 N33 A35 E36 K38 D40 R42 T43 K50 M51 G52 K53 T56 S58 M1 L5 F7 A20 K21 W23 W32 N33 A35 E36 K38 D40 R42 T43 K50 M51 G52 K53 T56 S58 ? 0003677,0006355 remove_due_to_license_issue Q9CIP3 23303792 1 ~ 17 MADKLKFEIIEELIVLSENAKGWRKELNRVSWNDAEPKYDIRTWSPDHEKMGKGITLSEEEFGVLLKELGNKLE 2ltt B -1.00 BS01 dna C 0 M1 L5 F7 A20 K21 W23 W32 N33 A35 K38 D40 R42 T43 K50 M51 G52 K53 T56 S58 M1 L5 F7 A20 K21 W23 W32 N33 A35 K38 D40 R42 T43 K50 M51 G52 K53 T56 S58 ? 0003677,0006355 remove_due_to_license_issue Q9CIP3 23303792 1 ~ 17 MADKLKFEIIEELIVLSENAKGWRKELNRVSWNDAEPKYDIRTWSPDHEKMGKGITLSEEEFGVLLKELGNKLE 2lup B -1.00 BS01 rna A 0 K371 R372 Y375 S376 P393 A395 N419 K8 R9 Y12 S13 P30 A32 N56 3.1.26.3 0003725,0006364 remove_due_to_license_issue Q02555 21742266 1 ~ 32 GSLDMNAKRQLYSLIGYASLRLHYVTVKKPTAVDPNSIVECRVGDGTVLGTGVGRNIKIAGIRAAENALRDKKMLDFYAKQRAAIPRSES 2lwi A -1.00 BS02 KOB A 1 L56 A66 M67 Q70 Y71 L56 A66 M67 Q70 Y71 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01112 23630290 203 MTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPSIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHQYREQIKRVKDSDDVPMVLVGNKCDLAARTVESRQAQDLARSYGIPYIETSAKTRQGVEDAFYTLVREIRQH 2ly0 A -1.00 BS01 A2Y A 1 V27 A30 V9 A12 ? 0015078,0033644,0055036,1902600 remove_due_to_license_issue Q6XT21 23302696 100 SNDSSDPLVVAANIIGILHLILWILDRLFFK 2lyb A -1.00 BS01 8SP A 1 F44 L64 F43 L63 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0005198 remove_due_to_license_issue P12497 23401539 300 GARASVLSGGELDKWEKIRLRPGGKKQYKLKHIVWASRELERFAVNPGLLETSEGCRQILGQLQPSLQTGSEELRSLYNTIAVLYCVHQRIDVKDTKEALDKIEEEQNKSKKKAQQAAADTGNNSQVSQNY 2lzg A -1.00 BS01 13Q A 1 V14 T16 L54 G58 I61 Y67 V93 H96 V14 T16 L54 G58 I61 Y67 V93 H96 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue IC50=34nM Q00987 22991965 201 MCNTNMSVPTDGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVNQQESSDSGTSVSEN 2m3z A -1.00 BS03 1HF A 1 K3 N8 Q9 K14 C15 F16 I24 A25 K26 W37 M46 K3 N8 Q9 K14 C15 F16 I24 A25 K26 W37 M46 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0008270 remove_due_to_license_issue P12497 23485336 103 IQKGNFRNQRKTVKCFNCGKEGHIAKNCRAPRKKGCWKCGKEGHQMKDCTERQAN 2m3z A -1.00 BS04 1HF A 2 R32 K33 G35 C36 W37 Q45 M46 K47 R32 K33 G35 C36 W37 Q45 M46 K47 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0008270 remove_due_to_license_issue P12497 23485336 104 IQKGNFRNQRKTVKCFNCGKEGHIAKNCRAPRKKGCWKCGKEGHQMKDCTERQAN 2m8d B -1.00 BS01 rna A 0 P108 R109 Y112 P115 S116 R117 S133 W134 Q135 D136 K138 D139 Y149 A150 D151 Y153 R154 H183 E184 P3 R4 Y7 P10 S11 R12 S28 W29 Q30 D31 K33 D34 Y44 A45 D46 Y48 R49 H78 E79 ? 0003676,0003723 remove_due_to_license_issue Q07955 23836656 1 ~ 8 MAPRGRYGPPSRRSENRVVVSGLPPSGSWQDLKDHMREAGDVCYADVYRDGTGVVEFVRKEDMTYAVRKLDNTKFRSHEGETAYIRVKVDG 2mas A 2.3 BS02 PIR A 1 D14 N39 I81 M152 E166 F167 N168 D242 D13 N38 I80 M151 E165 F166 N167 D241 D10 D15 N39 I75 T126 F167 N168 H241 D242 D9 D14 N38 I74 T125 F166 N167 H240 D241 3.2.2.2,3.2.2.3 0005829,0006139,0006152,0008477,0009117,0016798,0016799,0045437,0046872,0047724 Kd=30nM remove_due_to_license_issue Q27546 9572842 400 AKKIILDCDPGLDDAVAILLAHGNPEIELLAITTVVGNQTLAKVTRNAQLVADIAGITGVPIAAGCDKPLVRKIMTAGHIHGESGMGTVAYPAEFKNKVDERHAVNLIIDLVMSHEPKTITLVPTGGLTNIAMAARLEPRIVDRVKEVVLMGGGYHEGNATSVAEFNIIIDPEAAHIVFNESWQVTMVGLDLTHQALATPPILQRVKEVDTNPARFMLEIMDYYTKIYQSNRYMAAAAVHDPCAVAYVIDPSVMTTERVPVDIELTGKLTLGMTVADFRNPRPEHCHTQVAVKLDFEKFWGLVLDALERIGDP 2mb0 B -1.00 BS01 rna A 0 K9 F11 L38 M40 R49 F51 F53 A78 I79 K80 T85 P87 F89 K9 F11 L38 M40 R49 F51 F53 A78 I79 K80 T85 P87 F89 ? 0003676,0003723 remove_due_to_license_issue P38159 24692659 96 ~ 101 MVEADRPGKLFIGGLNTETNEKALEAVFGKYGRIVEVLLMKDRETNKSRGFAFVTFESPADAKDAARDMNGKSLDGKAIKVEQATKPSFESGRRG 2mfc A -1.00 BS01 rna B 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 -3 ~ 19 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfc A -1.00 BS02 rna D 0 L23 G27 Q29 R31 A36 P37 K38 V40 V42 H43 R44 I47 R50 I51 L23 G27 Q29 R31 A36 P37 K38 V40 V42 H43 R44 I47 R50 I51 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 -3 ~ 19 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfc C -1.00 BS01 rna B 0 S26 G27 Q29 R31 A36 P37 K38 V40 V42 H43 R44 I47 R50 I51 T56 S26 G27 Q29 R31 A36 P37 K38 V40 V42 H43 R44 I47 R50 I51 T56 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 -3 ~ 19 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfc C -1.00 BS02 rna D 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 -3 ~ 19 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfe A -1.00 BS01 rna B 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 17 ~ 38 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfe A -1.00 BS02 rna D 0 L23 G27 Q28 Q29 R31 A36 P37 K38 V42 H43 R44 I47 R50 I51 P58 L23 G27 Q28 Q29 R31 A36 P37 K38 V42 H43 R44 I47 R50 I51 P58 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 17 ~ 38 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfe C -1.00 BS01 rna B 0 L23 G27 Q29 R31 A36 P37 K38 V42 H43 R44 I47 R50 I51 A57 P58 L23 G27 Q29 R31 A36 P37 K38 V42 H43 R44 I47 R50 I51 A57 P58 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 17 ~ 38 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfe C -1.00 BS02 rna D 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 17 ~ 38 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mff A -1.00 BS01 rna B 0 M1 L2 I3 L4 T5 K7 Q28 M1 L2 I3 L4 T5 K7 Q28 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 40 ~ 60 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mff A -1.00 BS02 rna D 0 T21 L23 S26 G27 Q28 Q29 R31 A36 P37 K38 V42 H43 R44 I47 T21 L23 S26 G27 Q28 Q29 R31 A36 P37 K38 V42 H43 R44 I47 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 40 ~ 60 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mff C -1.00 BS01 rna B 0 L23 V25 S26 G27 Q28 Q29 R31 A36 P37 K38 V42 H43 R44 I47 L23 V25 S26 G27 Q28 Q29 R31 A36 P37 K38 V42 H43 R44 I47 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 40 ~ 60 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mff C -1.00 BS02 rna D 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 40 ~ 60 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfg A -1.00 BS01 rna B 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 55 ~ 75 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfg A -1.00 BS02 rna D 0 L23 S26 G27 R31 A36 P37 K38 V40 A41 V42 H43 L23 S26 G27 R31 A36 P37 K38 V40 A41 V42 H43 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 55 ~ 75 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfg C -1.00 BS01 rna B 0 L23 G27 Q29 R31 A36 P37 K38 A41 V42 H43 R44 L23 G27 Q29 R31 A36 P37 K38 A41 V42 H43 R44 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 55 ~ 75 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfg C -1.00 BS02 rna D 0 M1 L2 I3 L4 T5 K7 M1 L2 I3 L4 T5 K7 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 55 ~ 75 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfh A -1.00 BS01 rna B 0 M1 L2 I3 L4 T5 M1 L2 I3 L4 T5 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 36 ~ 44 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfh A -1.00 BS02 rna D 0 L23 Q29 A36 P37 K38 V42 H43 R44 L23 Q29 A36 P37 K38 V42 H43 R44 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 36 ~ 44 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfh C -1.00 BS01 rna B 0 L23 R31 A36 P37 K38 A41 V42 H43 R44 L23 R31 A36 P37 K38 A41 V42 H43 R44 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 36 ~ 44 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mfh C -1.00 BS02 rna D 0 M1 L2 I3 L4 T5 M1 L2 I3 L4 T5 ? 0003723,0005737,0005829,0006109,0006402,0006417,0045947,0045948,0048027 remove_due_to_license_issue P0DPC3 24561806 36 ~ 44 MLILTRKVGESINIGDDITITILGVSGQQVRIGINAPKDVAVHREEIYQRIQAGLTAPD 2mjh A -1.00 BS01 rna B 0 N220 V222 G223 L226 G227 P228 R229 G230 A233 K234 K243 I244 M245 V246 R247 A260 R262 N266 W267 E307 G308 D310 K313 R314 L317 M318 L320 A321 Y327 R328 P329 M330 N26 V28 G29 L32 G33 P34 R35 G36 A39 K40 K49 I50 M51 V52 R53 A66 R68 N72 W73 E113 G114 D116 K119 R120 L123 M124 L126 A127 Y133 R134 P135 M136 ? 0003676,0003723 remove_due_to_license_issue Q17339 24838563 16 ~ 25 LPEPAGDMISITEKIYVPKNEYPDYNFVGRILGPRGMTAKQLEQDTGCKIMVRGKGSMRDKSKESAHRGKANWEHLEDDLHVLVQCEDTENRVHIKLQAALEQVKKLLIPAPEGTDELKRKQLMELAIINGTYRPMKSPNPA 2mji A -1.00 BS01 KTR A 1 Y14 F17 M21 K27 Y70 T76 F93 Y117 Y14 F17 M21 K27 Y70 T76 F93 Y117 ? 0005324,0005504,0005515,0005634,0005737,0005829,0005902,0006631,0008289,0015908,0015909,0036041,0045179,0050892,0098856 remove_due_to_license_issue Kd=5.67e+4nM, Ki=9.4e+3nM P12104 25144524 201 AFDSTWKVDRSENYDKFMEKMGVNIVKRKLAAHDNLKLTITQEGNKFTVKESSAFRNIEVVFELGVTFNYNLADGTELRGTWSLEGNKLIGKFKRTDNGNELNTVREIIGDELVQTYVYEGVEAKRIFKKD 2mki A -1.00 BS01 rna B 0 K66 F68 G71 P96 H97 Y110 F112 Y136 I144 K147 P148 Q150 R152 F176 R182 K215 G216 K251 V254 K14 F16 G19 P44 H45 Y58 F60 Y84 I92 K95 P96 Q98 R100 F124 R130 K163 G164 K199 V202 ? 0003676,0003723,0003730,0006417,0045182 remove_due_to_license_issue Q17RY0 24990967 1 ~ 5 SHQNGERVERYSRKVFVGGLPPDIDEDEITASFRRFGPLIVDWPHKAESKSYFPPKGYAFLLFQDESSVQALIDACIEEDGKLYLCVSSPTIKDKPVQIRPWNLSDSDFVMDGSQPLDPRKTIFVGGVPRPLRAVELAMIMDRLYGGVCYAGIDTDPELKYPKGAGRVAFSNQQSYIAAISARFVQLQHGEIDKRVEVKPYVL 2mkk A -1.00 BS01 rna B 0 F239 G242 P244 E265 P267 K279 Y281 Y283 Y313 K324 Q327 I329 F353 H358 G359 D385 K386 G392 S393 K422 D427 F22 G25 P27 E48 P50 K62 Y64 Y66 Y96 K107 Q110 I112 F136 H141 G142 D168 K169 G175 S176 K205 D210 ? 0003676,0003723,0003730,0006417,0045182 remove_due_to_license_issue Q9BZB8 24990967 1 ~ 5 MTWSGQLPPRNYKNPIYSCKVFLGGVPWDITEAGLVNTFRVFGSLSVEWPGKDGKHPRCPPKGYVYLVFELEKSVRSLLQACSHDPLSPDGLSEYYFKMSSRRMRCKEVQVIPWVLADSNFVRSPSQRLDPSRTVFVGALHGMLNAEALAAILNDLFGGVVYAGIDTDKHKYPIGSGRVTFNNQRSYLKAVSAAFVEIKTTKFTKKVQIDPYL 2mkn A -1.00 BS01 rna B 0 V198 K208 K211 Q212 K215 V18 K28 K31 Q32 K35 ? 0003676,0008270 remove_due_to_license_issue Q9UL40 24521053 1 ~ 19 IDPDKFCSLCHATFNDPVMAQQHYVGKKHRKQETKLKLMARYGR 2mkn A -1.00 BS02 rna C 0 D196 M199 Q202 H203 G206 K207 K208 D16 M19 Q22 H23 G26 K27 K28 ? 0003676,0008270 remove_due_to_license_issue Q9UL40 24521053 20 ~ 38 IDPDKFCSLCHATFNDPVMAQQHYVGKKHRKQETKLKLMARYGR 2mlm A -1.00 BS01 2W7 A 1 V108 E113 I124 C126 W136 R139 V108 E113 I124 C126 W136 R139 remove_due_to_license_issue 25282649 201 MQAKPQIPKDKSKVAGYIEIPDADIKEPVYPGPATPEQLNRGVSFAEENESLDDQNISIAGHTFIDRPNYQFTNLKAAKKGSMVYFKVGNETRKYKMTSIRDVKPTDVEVLDEQKGKDKQLTLITCDDYNEKTGVWEKRKIFVATEVK 2moe A -1.00 BS01 dna B 0 R97 K101 T102 L116 R20 K24 T25 L39 3.2.2.- 0003677 remove_due_to_license_issue O95243 25183517 201 ~ 210 GSTECRKSVPCGWERVVKQRLFGKTAGRFDVYFISPQGLKFRSKSSLANYLHKNGETSLKPEDFDFTVLSK 2mov A -1.00 BS01 IOR A 1 R78 C79 Q80 K90 N92 R78 C79 Q80 K90 N92 ? remove_due_to_license_issue Q15109 24824951 201 GSAQNITARIGEPLVLKCKGAPKKPPQRLEWKLNTGRTEAWKVLSPQGGGPWDSVARVLPNGSLFLPAVGIQDEGIFRCQAMNRNGKETKSNYRVRVYQIPGKPE 2mqv A -1.00 BS01 rna B 0 K8 Q9 Q12 R16 R17 R18 D22 R23 Q25 A27 Y28 K30 W35 A36 K41 K42 K8 Q9 Q12 R16 R17 R18 D22 R23 Q25 A27 Y28 K30 W35 A36 K41 K42 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0008270 remove_due_to_license_issue P03355 25209668 93 ~ 160 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSLL 2mru A -1.00 BS01 dna X 0 W9 N11 S12 W9 N11 S12 ? 0003677,0097351 remove_due_to_license_issue P0AE72 25564525 1 ~ 15 GIHSSVKRWGNSPAVRIPATLMQALNLNIDDEVKIDLVDGKLIIEPVRKE 2mru A -1.00 BS02 dna Y 0 S5 K7 R16 P18 A19 T20 S5 K7 R16 P18 A19 T20 ? 0003677,0097351 remove_due_to_license_issue P0AE72 25564525 1 ~ 15 GIHSSVKRWGNSPAVRIPATLMQALNLNIDDEVKIDLVDGKLIIEPVRKE 2mru B -1.00 BS01 dna X 0 K7 W9 R16 P18 A19 K7 W9 R16 P18 A19 ? 0003677,0097351 remove_due_to_license_issue P0AE72 25564525 1 ~ 15 GIHSSVKRWGNSPAVRIPATLMQALNLNIDDEVKIDLVDGKLIIEPVRKE 2mru B -1.00 BS02 dna Y 0 W9 N11 W9 N11 ? 0003677,0097351 remove_due_to_license_issue P0AE72 25564525 1 ~ 15 GIHSSVKRWGNSPAVRIPATLMQALNLNIDDEVKIDLVDGKLIIEPVRKE 2ms1 A -1.00 BS01 rna B 0 R17 R18 D22 R23 Q25 A27 Y28 K30 W35 A36 K41 K42 R17 R18 D22 R23 Q25 A27 Y28 K30 W35 A36 K41 K42 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0008270 remove_due_to_license_issue P03355 25209668 1 ~ 72 ATVVSGQKQDRQGGERRRSQLDRDQCAYCKEKGHWAKDCPKKPRGPRGPRPQTSL 2mtv A -1.00 BS01 rna B 0 K364 S365 N366 N370 S381 L383 P384 V385 R407 W431 P434 M437 M441 L442 K475 I476 G477 R478 D479 K18 S19 N20 N24 S35 L37 P38 V39 R61 W85 P88 M91 M95 L96 K129 I130 G131 R132 D133 ? 0003723 remove_due_to_license_issue Q9QY02 25389274 1 ~ 6 QTSKLKSVLQDARFFLIKSNNHENVSLAKAKGVWSTLPVNEKKLNLAFRSARSVILIFSVRESGKFQGFARLSSESHHGGSPIHWVLPAGMSAKMLGGVFKIDWICRRELPFTKSAHLTNPWNEHKPVKIGRDGQEIELECGTQLCLLFPPDESID 2mxf A -1.00 BS01 dna B 0 R80 T96 K97 N100 H101 K102 R2 T18 K19 N22 H23 K24 ? remove_due_to_license_issue Q9HW86 26068099 1 ~ 12 ARKVKQYKNPHTGEVIETKGGNHKTLKEWKAKWGPEAVESWATLLGH 2mxf A -1.00 BS02 dna C 0 A79 R80 K81 K83 Y85 G98 G99 N100 K105 K108 A1 R2 K3 K5 Y7 G20 G21 N22 K27 K30 ? remove_due_to_license_issue Q9HW86 26068099 13 ~ 24 ARKVKQYKNPHTGEVIETKGGNHKTLKEWKAKWGPEAVESWATLLGH 2mxy A -1.00 BS01 rna B 0 N4 V5 T6 N7 R17 F19 G21 N22 L26 V48 H49 K50 G51 F52 F54 D81 A85 P88 R92 K94 N3 V4 T5 N6 R16 F18 G20 N21 L25 V47 H48 K49 G50 F51 F53 D80 A84 P87 R91 K93 ? 0003676,0003723 remove_due_to_license_issue P07910 25216038 1 ~ 7 ASNVTNKTDPRSMNSRVFIGNLNTLVVKKSDVEAIFSKYGKIVGCSVHKGFAFVQYVNERNARAAVAGEDGRMIAGQVLDINLAAEPKVNRGKAGVKRSAAEMYG 2mz1 A -1.00 BS01 rna B 0 N4 V5 T6 N7 R17 F19 G21 N22 H49 G51 F52 F54 D81 A85 P88 R92 G93 K94 A95 G96 N3 V4 T5 N6 R16 F18 G20 N21 H48 G50 F51 F53 D80 A84 P87 R91 G92 K93 A94 G95 ? 0003676,0003723 remove_due_to_license_issue P07910 25216038 1 ~ 5 ASNVTNKTDPRSMNSRVFIGNLNTLVVKKSDVEAIFSKYGKIVGCSVHKGFAFVQYVNERNARAAVAGEDGRMIAGQVLDINLAAEPKVNRGKAGVKRSAAEMYG 2n06 A -1.00 BS01 44Z A 1 M53 L56 I60 Q71 H72 V92 L98 L102 M31 L34 I38 Q49 H50 V70 L76 L80 ? 0005634,0043066,0051726 remove_due_to_license_issue O15151 26812210 200 QINQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLAT 2n0u A -1.00 BS01 48M A 1 M53 G57 I60 Q71 H72 F90 V92 L98 M31 G35 I38 Q49 H50 F68 V70 L76 ? 0005634,0043066,0051726 remove_due_to_license_issue O15151 26812210 200 QINQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLAT 2n0w A -1.00 BS01 48L A 1 M53 G57 M61 Q71 H72 F90 V92 M31 G35 M39 Q49 H50 F68 V70 ? 0005634,0043066,0051726 remove_due_to_license_issue O15151 26812210 200 QINQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLAT 2n14 A -1.00 BS01 49H A 1 M53 L56 G57 I60 M61 Q71 H72 V92 M31 L34 G35 I38 M39 Q49 H50 V70 ? 0005634,0043066,0051726 remove_due_to_license_issue O15151 26812210 200 QINQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLAT 2n27 A -1.00 BS04 4DY A 1 L32 M76 M109 L32 M76 M109 V35 V35 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 remove_due_to_license_issue P0DP23 27339229 205 ADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAK 2n7b A -1.00 BS01 G6S B 1 R56 Y58 Q59 R56 Y58 Q59 ? remove_due_to_license_issue Q9NYZ4 27357658 2 MEGDRQYGDGYLLQVQELVTVQEGLSVHVPCSFSYPQDGWTDSDPVHGYWFRAGDRPYQDAPVATNNPDREVQAETQGRFQLLGDIWSNDCSLSIRDARKRDKGSYFFRLERGSMKWSYKSQLNYKTKQLSVFVTALTHGSLVPR 2n7b A -1.00 BS02 SIA B 1 Y7 Y11 Y58 R109 K116 W117 S118 Q122 Y7 Y11 Y58 R109 K116 W117 S118 Q122 ? remove_due_to_license_issue Q9NYZ4 27357658 3 MEGDRQYGDGYLLQVQELVTVQEGLSVHVPCSFSYPQDGWTDSDPVHGYWFRAGDRPYQDAPVATNNPDREVQAETQGRFQLLGDIWSNDCSLSIRDARKRDKGSYFFRLERGSMKWSYKSQLNYKTKQLSVFVTALTHGSLVPR 2n82 B -1.00 BS01 rna A 0 R118 H120 S122 N123 I124 P125 F126 I149 F150 N151 E152 R153 G154 S155 K156 G157 F158 F160 R184 N189 N190 A191 T192 A193 R194 V195 N198 K199 K200 N203 Y205 T206 R14 H16 S18 N19 I20 P21 F22 I45 F46 N47 E48 R49 G50 S51 K52 G53 F54 F56 R80 N85 N86 A87 T88 A89 R90 V91 N94 K95 K96 N99 Y101 T102 ? 0000381,0003676,0003723,0007399 remove_due_to_license_issue Q9NWB1 27001519 19 ~ 41 GSHMNTENKSQPKRLHVSNIPFRFRDPDLRQMFGQFGKILDVEIIFNERGSKGFGFVTFENSADADRAREKLHGTVVEGRKIEVNNATARVMTNKKTVNPYTNG 2n8a A -1.00 BS01 dna B 0 S16 R18 A19 S20 K22 R34 F44 V48 S120 R122 S123 R138 Q150 L151 I154 W157 S16 R18 A19 S20 K22 R34 F44 V48 S120 R122 S123 R138 Q150 L151 I154 W157 2.4.2.-,2.4.2.30 0003677,0008270 remove_due_to_license_issue P09874 26626479 1 ~ 45 MAESSDKLYRVEYAKSGRASCKKCSESIPKDSLRMAIMVQSPMFDGKVPHWYHFSCFWKVGHSIRHPDVEVDGFSELRWDDQQKVKKTAEAGGVTGKGQDGIGSKAEKTLGDFAAEYAKSNRSTCKGCMEKIEKGQVRLSKKMVDPEKPQLGMIDRWYHPGCFVKNREELGFRPEYSASQLKGFSLLATEDKEALKKQLPGVKSEGKRKGDEVD 2ndo A -1.00 BS01 SFQ A 1 H32 Q35 T168 M171 F174 H32 Q35 T168 M171 F174 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 remove_due_to_license_issue P0AEG4 27778134 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEKK 2nmx A 1.55 BS02 M25 A 1 H94 H119 L198 T199 H200 W209 H92 H117 L196 T197 H198 W207 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T197 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=2.7uM remove_due_to_license_issue P00915 17407288 311 PDWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2nmy A 1.1 BS01 ROC A 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2nmy B 1.1 BS01 ROC A 1 R108 D125 G127 G149 P181 I184 R8 D25 G27 G49 P81 I84 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2nmz A 0.97 BS01 ROC B 1 D25 G27 A28 D29 D30 G48 G49 I50 P81 D25 G27 A28 D29 D30 G48 G49 I50 P81 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2nmz B 0.97 BS01 ROC B 1 R108 D125 G127 G148 G149 I150 A182 R8 D25 G27 G48 G49 I50 A82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2nn1 A 1.65 BS02 M28 A 1 H94 H119 L198 T199 H200 W209 H92 H117 L196 T197 H198 W207 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T197 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=1.5uM remove_due_to_license_issue Ki=6690nM P00915 17407288 311 PDWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2nn7 A 1.85 BS02 M29 A 1 N69 Q92 H94 H119 L198 T199 H200 W209 N67 Q90 H92 H117 L196 T197 H198 W207 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T197 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=0.3uM remove_due_to_license_issue P00915 17407288 311 PDWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 2nnd A 1.6 BS01 PRZ A 1 L40 F94 Y124 L40 F84 Y114 ? 0036094 Kd=0.87uM remove_due_to_license_issue P02762 17991731 300 EEASSTGRNFNVEKINGEWHTIILASDKREKIEDNGNFRLFLEQIHVLEKSLVLKFHGSELSMVADKTEKAGEYSVTYDGFNTFTIPKTDYDNFLMAHLINEKDGETFQLMGLYGREPDLSSDIKERFAQLCEEHGILRENIIDLSNA 2nng A 1.2 BS02 ZYX A 1 H94 H119 L198 T199 T200 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=4.4uM remove_due_to_license_issue Ki=160nM, IC50=3100nM P00918 17407288 301 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2nnk A 1.25 BS01 ROC A 1 D25 G27 D29 D30 G48 G49 I50 P81 D25 G27 D29 D30 G48 G49 I50 P81 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2nnk B 1.25 BS01 ROC A 1 R108 D125 G127 G148 G149 I150 P181 R8 D25 G27 G48 G49 I50 P81 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2nno A 1.01 BS02 M28 A 1 H94 H119 L198 T199 T200 H93 H118 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.4uM remove_due_to_license_issue Ki=495nM P00918 17407288 301 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2nno A 1.01 BS03 M28 A 2 H4 W5 H15 W16 D19 H3 W4 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.4uM remove_due_to_license_issue Ki=495nM P00918 17407288 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2nnp A 1.2 BS01 ROC A 1 D25 G27 D29 D30 G48 I50 P81 D25 G27 D29 D30 G48 I50 P81 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2nnp B 1.2 BS01 ROC A 1 R108 D125 G127 G149 I150 V182 R8 D25 G27 G49 I50 V82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2nnq A 1.8 BS01 T4B A 1 F16 A33 A36 P38 S53 A75 D76 I104 R106 R126 Y128 F16 A33 A36 P38 S53 A75 D76 I104 R106 R126 Y128 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki<2nM remove_due_to_license_issue Kd=2050nM, Ki=220nM, IC50=221nM P15090 17502136 293 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 2nns A 1.03 BS02 M25 A 1 H94 H119 L198 T199 T200 H93 H118 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.9uM remove_due_to_license_issue P00918 17407288 301 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2nns A 1.03 BS03 M25 A 2 W5 N11 H15 W16 D19 W4 N10 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.9uM remove_due_to_license_issue P00918 17407288 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2nnv A 1.1 BS02 M29 A 1 H94 H96 H119 L198 T199 T200 H93 H95 H118 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.03uM remove_due_to_license_issue P00918 17407288 301 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2nnv A 1.1 BS03 M29 A 2 W5 H10 H15 W16 D19 W4 H9 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.03uM remove_due_to_license_issue P00918 17407288 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2no3 A 3.2 BS02 859 A 1 G33 V40 A53 M108 L110 M111 D112 L168 G26 V33 A46 M101 L103 M104 D105 L161 D151 K153 N156 D169 T188 D144 K146 N149 D162 T181 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=170nM P45983 17107797 901 NNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 2noe A 2.2 BS01 dna B 0 N149 R154 G202 Y203 R204 A288 N138 R143 G191 Y192 R193 A277 3.2.2.-,4.2.99.18 0000978,0003677,0003684,0003824,0004519,0005515,0005634,0005654,0005739,0005759,0005829,0006281,0006284,0006285,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045007,0045008,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O15527 17114185 3 ~ 15 SEFGHRTLASTPALWASIPCPRSELRLDLVLPSAQSFRWREQSPAHWSGVLADQVWTLTQTEEQLHCTVYRSQASRPTPDELEAVRKYFQLDVTLAQLYHHWGSVDSHFQEVAQKFQGVRLLRQDPIECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPSLQALAGPEVEAHLRKLGLGYRARYVSASARAILEEQGGLAWLQQLRESSYEEAHKALCILPGVGTQVADCICLMALDKPQAVPVDVHMWHIAQRDYSWHPTTSQAKGPSPQTNKELGNFFRSLWGPYAGWAQAVLFSADLRQ 2noe A 2.2 BS02 dna C 0 A42 S147 S148 N149 N150 N151 I152 P244 G245 G247 Q249 V250 P266 D268 V269 H270 Q315 F319 A34 S136 S137 N138 N139 N140 I141 P233 G234 G236 Q238 V239 P255 D257 V258 H259 Q304 F308 3.2.2.-,4.2.99.18 0000978,0003677,0003684,0003824,0004519,0005515,0005634,0005654,0005739,0005759,0005829,0006281,0006284,0006285,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045007,0045008,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O15527 17114185 19 ~ 31 SEFGHRTLASTPALWASIPCPRSELRLDLVLPSAQSFRWREQSPAHWSGVLADQVWTLTQTEEQLHCTVYRSQASRPTPDELEAVRKYFQLDVTLAQLYHHWGSVDSHFQEVAQKFQGVRLLRQDPIECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPSLQALAGPEVEAHLRKLGLGYRARYVSASARAILEEQGGLAWLQQLRESSYEEAHKALCILPGVGTQVADCICLMALDKPQAVPVDVHMWHIAQRDYSWHPTTSQAKGPSPQTNKELGNFFRSLWGPYAGWAQAVLFSADLRQ 2np2 A 3.02 BS01 dna C 0 E56 F57 R58 R68 K69 R71 N73 R75 P77 Q78 Y92 E51 F52 R53 R63 K64 R66 N68 R70 P72 Q73 Y87 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q57267 17244195 203 ~ 238 RPKVTKSDIVDQIALNIKNNNLKLEKKYIRLVIDAFFEELKSNLCSNNVIEFRSFGTFEVRKRKGRLNARNPQTGEYVKVLDHHVAYFRPGKDLKERVWGIK 2np2 A 3.02 BS02 dna D 0 T10 K11 R58 S59 R75 N76 P77 Q78 R94 K97 T5 K6 R53 S54 R70 N71 P72 Q73 R89 K92 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q57267 17244195 203 ~ 238 RPKVTKSDIVDQIALNIKNNNLKLEKKYIRLVIDAFFEELKSNLCSNNVIEFRSFGTFEVRKRKGRLNARNPQTGEYVKVLDHHVAYFRPGKDLKERVWGIK 2np2 B 3.02 BS01 dna C 0 K8 T10 K11 R58 S59 R75 N76 P77 Q78 K97 K3 T5 K6 R53 S54 R70 N71 P72 Q73 K92 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q57267 17244195 203 ~ 238 RPKVTKSDIVDQIALNIKNNNLKLEKKYIRLVIDAFFEELKSNLCSNNVIEFRSFGTFEVRKRKGRLNARNPQTGEYVKVLDHHVAYFRPGKDLKERVWGIK 2np2 B 3.02 BS02 dna D 0 F57 R58 R66 R68 R71 N73 R75 P77 Q78 F52 R53 R61 R63 R66 N68 R70 P72 Q73 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q57267 17244195 203 ~ 238 RPKVTKSDIVDQIALNIKNNNLKLEKKYIRLVIDAFFEELKSNLCSNNVIEFRSFGTFEVRKRKGRLNARNPQTGEYVKVLDHHVAYFRPGKDLKERVWGIK 2np8 A 2.25 BS01 CC3 A 1 L139 G142 K143 V147 A160 L194 A213 P214 G216 L263 L13 G16 K17 V21 A34 L68 A87 P88 G90 L137 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T160 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=42nM remove_due_to_license_issue IC50=42nM O14965 17157005 394 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2np9 A 2.45 BS01 YE1 A 1 L186 A188 E189 H222 Y225 A233 G234 I235 N236 K238 L251 R254 F292 I294 G295 G296 Q299 G327 F432 L176 A178 E179 H212 Y215 A223 G224 I225 N226 K228 L241 R244 F282 I284 G285 G286 Q289 G317 F422 I235 G296 Q299 A319 I225 G286 Q289 A309 1.13.11.80 0006635,0016491,0016702,0017000,0042802 Ki=2.7uM remove_due_to_license_issue Q8KLK7 17507985 999 TDGLWAALTEAAASVEKLLATLPEHGARSSAERAEIAAAHDAARALRVRFLDTHADAVYDRLTDHRRVHLRLAELVEAAATAFPGLVPTQQQLAVERSLPQAAKEGHEIDQGIFLRAVLRSPLAGPHLLDAMLRPTPRALELLPEFVRTGEVEMEAVHLERRDGVARLTMCRDDRLNAEDGQQVDDMETAVDLALLDPGVRVGLLRGGVMSHPRYRGKRVFSAGINLKYLSQGGISLVDFLMRRELGYIHKLVRGVLTNDDRPGWWHSPRIEKPWVAAVDGFAIGGGAQLLLVFDRVLASSDAYFSLPAAKEGIIPGAANLRLGRFAGPRVSRQVILEGRRIWAKEPEARLLVDEVVEPDELDAAIERSLTRLDGDAVLANRRMLNLADESPDGFRAYMAEFALMQALRLYGHDVIDKVGRFG 2nq6 A 1.5 BS04 HM4 A 1 P192 Y195 Y196 C203 H212 H310 W353 P103 Y106 Y107 C114 H123 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=1.5uM remove_due_to_license_issue EC50=>40000nM, IC50=400nM P53582 17114291 410 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 2nq7 A 1.6 BS03 HM5 A 1 P192 Y195 Y196 F198 C203 H212 H310 W353 P103 Y106 Y107 F109 C114 H123 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=2.9uM remove_due_to_license_issue IC50=2900nM P53582 17114291 410 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 2nq9 A 1.45 BS01 dna B 0 D229 R230 H231 D229 R230 H231 3.1.21.2 0003677,0003906,0004519,0005829,0006281,0006284,0008081,0008270,0008296,0008833,0016791,0046872 remove_due_to_license_issue P0A6C1 18408731 301 ~ 306 MKYIGAHVSAAGGLANAAIRAAEIDATAFALFTKNQRQWRAAPLTTQTIDEFKAACEKYHYTSAQILPHDSALINLGHPVTEALEKSRDAFIDEMQRCEQLGLSLLNFHPGSHLMQISEEDCLARIAESINIALDKTQGVTAVIENTAGQGSNLGFKFEHLAAIIDGVEDKSRVGVCIDTCHAFAAGYDLRTPAECEKTFADFARTVGFKYLRGMHLNDAKSTFGSRVDRHHSLGEGNIGHDAFRWIMQDDRFDGIPLILETINPDIWAEEIAWLKAQQ 2nq9 A 1.45 BS02 dna C 0 H7 S9 A10 A11 F32 N35 Q36 R37 H69 H109 E145 H182 H231 E261 H7 S9 A10 A11 F32 N35 Q36 R37 H69 H109 E145 H182 H231 E261 3.1.21.2 0003677,0003906,0004519,0005829,0006281,0006284,0008081,0008270,0008296,0008833,0016791,0046872 remove_due_to_license_issue P0A6C1 18408731 307 ~ 311 MKYIGAHVSAAGGLANAAIRAAEIDATAFALFTKNQRQWRAAPLTTQTIDEFKAACEKYHYTSAQILPHDSALINLGHPVTEALEKSRDAFIDEMQRCEQLGLSLLNFHPGSHLMQISEEDCLARIAESINIALDKTQGVTAVIENTAGQGSNLGFKFEHLAAIIDGVEDKSRVGVCIDTCHAFAAGYDLRTPAECEKTFADFARTVGFKYLRGMHLNDAKSTFGSRVDRHHSLGEGNIGHDAFRWIMQDDRFDGIPLILETINPDIWAEEIAWLKAQQ 2nq9 A 1.45 BS03 dna D 0 R37 Q38 W39 A72 L73 N75 Q150 G151 S152 R230 R37 Q38 W39 A72 L73 N75 Q150 G151 S152 R230 3.1.21.2 0003677,0003906,0004519,0005829,0006281,0006284,0008081,0008270,0008296,0008833,0016791,0046872 remove_due_to_license_issue P0A6C1 18408731 335 ~ 345 MKYIGAHVSAAGGLANAAIRAAEIDATAFALFTKNQRQWRAAPLTTQTIDEFKAACEKYHYTSAQILPHDSALINLGHPVTEALEKSRDAFIDEMQRCEQLGLSLLNFHPGSHLMQISEEDCLARIAESINIALDKTQGVTAVIENTAGQGSNLGFKFEHLAAIIDGVEDKSRVGVCIDTCHAFAAGYDLRTPAECEKTFADFARTVGFKYLRGMHLNDAKSTFGSRVDRHHSLGEGNIGHDAFRWIMQDDRFDGIPLILETINPDIWAEEIAWLKAQQ 2nqg A 2.04 BS03 NQG A 1 Q109 G113 C115 G208 S251 G271 H272 W298 Q77 G81 C83 G176 S219 G239 H240 W266 Q109 C115 H272 N296 W298 Q77 C83 H240 N264 W266 3.4.22.52 0004198,0006508 remove_due_to_license_issue P97571 17218315 501 NAIKYLGQDYENLRARCLQNGVLFQDDAFPPVSHSLGFKELGPNSSKTYGIKWKRPTELLSNPQFIVDGATRTDICQGALGDCWLLAAIASLTLNETILHRVVPYGQSFQEGYAGIFHFQLWQFGEWVDVVVDDLLPTKDGKLVFVHSAQGNEFWSALLEKAYAKVNGSYEALSGGCTSEAFEDFTGGVTEWYDLQKAPSDLYQIILKALERGSLLGCSINISDIRDLEAITFKNLVRGHAYSVTDAKQVTYQGQRVNLIRMRNPWGEVEWKGPWSDNSYEWNKVDPYEREQLRVKMEDGEFWMSFRDFIREFTKLEICNLT 2nqi A 2.04 BS03 NQI A 1 Q109 G113 C115 G207 G208 S251 G271 H272 A273 W298 Q77 G81 C83 G175 G176 S219 G239 H240 A241 W266 Q109 C115 H272 N296 W298 Q77 C83 H240 N264 W266 3.4.22.52 0004198,0006508 remove_due_to_license_issue P97571 17218315 501 NAIKYLGQDYENLRARCLQNGVLFQDDAFPPVSHSLGFKELGPNSSKTYGIKWKRPTELLSNPQFIVDGATRTDICQGALGDCWLLAAIASLTLNETILHRVVPYGQSFQEGYAGIFHFQLWQFGEWVDVVVDDLLPTKDGKLVFVHSAQGNEFWSALLEKAYAKVNGSYEALSGGCTSEAFEDFTGGVTEWYDLQKAPSDLYQIILKALERGSLLGCSINISDIRDLEAITFKNLVRGHAYSVTDAKQVTYQGQRVNLIRMRNPWGEVEWKGPWSDNSYEWNKVDPYEREQLRVKMEDGEFWMSFRDFIREFTKLEICNLT 2nqj A 2.45 BS01 dna C 0 H7 S9 A10 A11 G12 F32 N35 Q36 R37 Y72 H109 D229 R230 H231 Q261 H7 S9 A10 A11 G12 F32 N35 Q36 R37 Y72 H109 D229 R230 H231 Q261 3.1.21.2 0003677,0003906,0004519,0005829,0006281,0006284,0008081,0008270,0008296,0008833,0016791,0046872 remove_due_to_license_issue P0A6C1 18408731 301 ~ 315 MKYIGAHVSAAGGLANAAIRAAEIDATAFALFTKNQRQWRAAPLTTQTIDEFKAACEKYHYTSAQILPHDSYLINLGHPVTEALEKSRDAFIDEMQRCEQLGLSLLNFHPGSHLMQISEEDCLARIAESINIALDKTQGVTAVIENTAGQGSNLGFKFEHLAAIIDGVEDKSRVGVCIDTCHAFAAGYDLRTPAECEKTFADFARTVGFKYLRGMHLNDAKSTFGSRVDRHHSLGEGNIGHDAFRWIMQDDRFDGIPLILQTINPDIWAEEIAWLKAQQ 2nqj A 2.45 BS02 dna D 0 N35 R37 Q38 W39 L73 L114 Q150 G151 S152 V228 N35 R37 Q38 W39 L73 L114 Q150 G151 S152 V228 3.1.21.2 0003677,0003906,0004519,0005829,0006281,0006284,0008081,0008270,0008296,0008833,0016791,0046872 remove_due_to_license_issue P0A6C1 18408731 331 ~ 345 MKYIGAHVSAAGGLANAAIRAAEIDATAFALFTKNQRQWRAAPLTTQTIDEFKAACEKYHYTSAQILPHDSYLINLGHPVTEALEKSRDAFIDEMQRCEQLGLSLLNFHPGSHLMQISEEDCLARIAESINIALDKTQGVTAVIENTAGQGSNLGFKFEHLAAIIDGVEDKSRVGVCIDTCHAFAAGYDLRTPAECEKTFADFARTVGFKYLRGMHLNDAKSTFGSRVDRHHSLGEGNIGHDAFRWIMQDDRFDGIPLILQTINPDIWAEEIAWLKAQQ 2nr0 A 3.9 BS01 rna E 0 Q27 Q29 N30 Y140 V167 Q168 A238 T239 Q21 Q23 N24 Y134 V161 Q162 A232 T233 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 2 ~ 71 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 A 3.9 BS02 rna F 0 V46 R78 A82 G86 A89 V40 R72 A76 G80 A83 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 3 ~ 70 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 A 3.9 BS03 rna G 0 R110 F111 E158 S171 T173 R176 N197 R104 F105 E152 S165 T167 R170 N191 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 5 ~ 68 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 B 3.9 BS01 rna E 0 V46 N48 R78 A82 G86 V40 N42 R72 A76 G80 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 2 ~ 71 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 B 3.9 BS02 rna F 0 Y24 Q27 Q29 R58 A61 R110 F111 R126 Y140 V167 Q168 Q170 S171 R172 H201 H202 A238 T239 Y18 Q21 Q23 R52 A55 R104 F105 R120 Y134 V161 Q162 Q164 S165 R166 H195 H196 A232 T233 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 3 ~ 70 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 C 3.9 BS01 rna G 0 Y24 R28 Q29 N30 R58 D60 A61 R110 R126 Y140 V167 S171 R172 T173 H202 A238 T239 Y18 R22 Q23 N24 R52 D54 A55 R104 R120 Y134 V161 S165 R166 T167 H196 A232 T233 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 5 ~ 68 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 C 3.9 BS02 rna H 0 V46 N48 R78 A82 L85 A89 N90 V40 N42 R72 A76 L79 A83 N84 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 4 ~ 69 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 D 3.9 BS01 rna G 0 V46 N48 R78 A82 L85 G86 N90 V40 N42 R72 A76 L79 G80 N84 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 5 ~ 68 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nr0 D 3.9 BS02 rna H 0 Q29 N30 R126 Y140 V167 Q170 A238 T239 Q23 N24 R120 Y134 V161 Q164 A232 T233 5.4.99.12 0000049,0001522,0003723,0006396,0008033,0009451,0009982,0016853,0031119,0042803,0106029,0140098,0160147 remove_due_to_license_issue P07649 17466622 4 ~ 69 PPVYKIALGIEYDGSKYYGWQRQNEVRSVQEKLEKALSQVANEPITVFCAGRTDAGVHGTGQVVHFETTALRKDAAWTLGVNANLPGDIAVRWVKTVPDDFHARFSATARRYRYIIYNHRLRPAVLSKGVTHFYEPLDAERMHRAAQCLLGENDFTSFRAVQCQSRTPWRNVMHINVTRHGPYVVVDIKANAFVHHMVRNIVGSLMEVGAHNQPESWIAELLAAKDRTLAAATAKAEGLYLVAVDYPDRYDLPKPPMGPLFLAD 2nsj A 2.31 BS01 C2R A 1 G15 S16 S18 D19 S43 A44 Q45 R46 A70 G71 A74 H75 L76 G9 S10 S12 D13 S37 A38 Q39 R40 A64 G65 A68 H69 L70 5.4.99.18 0003824,0005829,0006164,0006189,0016853,0034023,0042802 Kd=16.3uM remove_due_to_license_issue P0AG18 17298082 242 PARVAIVMGSKSDWATMQFAAEIFEILNVPHHVEVVSAQRTPDKLFSFAESAEENGYQVIIAGAGGAAHLPGMIAAKTLVPVLGVPVQSAALSGVDSLYSIVQMPRGIPVGTLAIGKAGAANAALLAAQILATHDKELHQRLNDWRKAQTDEVLENPDPRGA 2nsl A 2.0 BS01 C2R A 1 S16 S18 D19 S43 A44 N45 R46 A70 G71 H75 S10 S12 D13 S37 A38 N39 R40 A64 G65 H69 5.4.99.18 0003824,0005829,0006164,0006189,0016853,0034023,0042802 Kd=20.9uM remove_due_to_license_issue P0AG18 17298082 300 PARVAIVMGSKSDWATMQFAAEIFEILNVPHHVEVVSANRTPDKLFSFAESAEENGYQVIIAGAGGAAHLPGMIAAKTLVPVLGVPVQSAALSGVDSLYSIVQMPRGIPVGTLAIGKAGAANAALLAAQILATHDKELHQRLNDWRKAQTDEVLENPDPRGA 2nsx B 2.11 BS01 IFM B 1 D127 W179 E235 Y313 E340 W381 D127 W179 E235 Y313 E340 W381 E235 E340 C342 N370 E235 E340 C342 N370 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 ic50=59nM remove_due_to_license_issue Ki=1.70nM, IC50=8.20nM P04062 17187079 506 ARPCIPKSFGYSSVVCVCNATYCDSFDPPTFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 2nt7 A 2.1 BS01 902 A 1 R24 A27 S28 D29 Y46 V49 K120 D181 F182 S216 A217 I219 G220 R221 G259 Q262 R23 A26 S27 D28 Y45 V48 K119 D180 F181 S215 A216 I218 G219 R220 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.3uM remove_due_to_license_issue P18031 17336064 800 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2nta A 2.1 BS01 521 A 1 Y46 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y45 D180 F181 C214 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=16uM remove_due_to_license_issue P18031 17336064 301 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLDMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2ntc A 2.4 BS01 dna W 0 N153 T155 R202 H203 R204 A207 N22 T24 R71 H72 R73 A76 ? 0003688,0006260 remove_due_to_license_issue Q98ZP7 17253903 1 ~ 21 VEDPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDFN 2ntc A 2.4 BS02 dna C 0 S147 H148 A149 F151 S152 N153 R154 N227 S16 H17 A18 F20 S21 N22 R23 N96 ? 0003688,0006260 remove_due_to_license_issue Q98ZP7 17253903 23 ~ 43 VEDPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDFN 2ntc B 2.4 BS01 dna W 0 S147 A149 F151 S152 N153 R154 N227 S15 A17 F19 S20 N21 R22 N95 ? 0003688,0006260 remove_due_to_license_issue Q98ZP7 17253903 1 ~ 21 EDPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDFN 2ntc B 2.4 BS02 dna C 0 N153 T155 R202 H203 R204 N210 N21 T23 R70 H71 R72 N78 ? 0003688,0006260 remove_due_to_license_issue Q98ZP7 17253903 23 ~ 43 EDPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDFN 2ntf H 3.18 BS01 OHM H 1 W33 H35 G95 S96 N100 N100A G100C W100D F100E W33 H35 G99 S100 N104 N105 G107 W108 F109 ? remove_due_to_license_issue Q99LC4 17400249 1001 QVQLQQSGSELVRPGASVKLSCKASGYTFTTYWIHWVKQRPGQGLEWIGTIYPGSDNTYYDEKFKNKATLTVDTSSSTAFMQLSSLTSEDSAVYFCTRGSLYYNNYGWFGYWGQGTLVTVSAAKTTPPSVYPLAPGSNAASQSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLTSSVTVPSSTWPSQTVTCNVAHPASSTKVDKKIVPR 2ntf L 3.18 BS01 OHM H 1 N34 W96 N36 W98 remove_due_to_license_issue 17400249 1001 QAVVTQESALTTSPGETVTLTCRSSTGAVTTRNYANWVQEKPDHFFTGLIGDTNNRAPGVPARFSGSLIGHKAALTITGAQTEDESVYFCALWYSNHWVFGGGTKLTVLGQPKSSPSVTLFPPSSEELETNKATLVCTITDFYPGVVTVDWKVDGTPVTQGMETTQPSKQSNNKYMASSYLTLTAGAWERHSSYSCQVTHEGHTVEKSLSR 2ntz A 3.35 BS01 dna E 0 D288 R292 D139 R143 ? remove_due_to_license_issue Q38420 17293348 24 ~ 39 QTALQHSIREIGLRLMRMKNDGMSQKDIAAKEGLSQAKVTRALQAASAPEELVALFPVQSELTFSDYKTLCAVGDEMGNLEFDQLIQNISPEINDILSIEEMAEDEVKNKILRLITKEASLLTDKKSVVTELWKFEDKDRFARKRVKGRAFSYEFNRLSKELQEELDRMIGHILRKSLDKKPK 2ntz A 3.35 BS02 dna U 0 R289 R306 R140 R157 ? remove_due_to_license_issue Q38420 17293348 2 ~ 17 QTALQHSIREIGLRLMRMKNDGMSQKDIAAKEGLSQAKVTRALQAASAPEELVALFPVQSELTFSDYKTLCAVGDEMGNLEFDQLIQNISPEINDILSIEEMAEDEVKNKILRLITKEASLLTDKKSVVTELWKFEDKDRFARKRVKGRAFSYEFNRLSKELQEELDRMIGHILRKSLDKKPK 2ntz B 3.35 BS01 dna Y 0 K287 D288 R292 K133 D134 R138 ? remove_due_to_license_issue Q38420 17293348 24 ~ 39 SIREIGLRLMRMKNDGMSQKDIAAKEGLSQAKVTRALQAASAPEELVALFPVQSELTFSDYKTLCAVGDEMGNKNLEFDQLIQNISPEINDILSIEEMAEDEVKNKILRLITKEASLLTDKSVVTELWKFEDKDRFARKRVKGRAFSYEFNRLSKELQEELDRMIGHILRKS 2ntz B 3.35 BS02 dna W 0 K287 D288 R306 S308 K309 K133 D134 R152 S154 K155 ? remove_due_to_license_issue Q38420 17293348 2 ~ 17 SIREIGLRLMRMKNDGMSQKDIAAKEGLSQAKVTRALQAASAPEELVALFPVQSELTFSDYKTLCAVGDEMGNKNLEFDQLIQNISPEINDILSIEEMAEDEVKNKILRLITKEASLLTDKSVVTELWKFEDKDRFARKRVKGRAFSYEFNRLSKELQEELDRMIGHILRKS 2nv7 A 2.1 BS02 555 A 1 M295 E305 L339 F356 I373 I376 H475 L476 M33 E43 L77 F94 I111 I114 H203 L204 ? 0003677,0004879,0006355 ic50=5nM remove_due_to_license_issue Q92731 17188490 501 LSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMDSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKCKNVVPVYDLLLEMLNAHVL 2nw4 A 3.0 BS01 8NH A 1 L701 L704 N705 L707 G708 M745 M749 F764 M780 T877 L31 L34 N35 L37 G38 M75 M79 F94 M110 T207 ? remove_due_to_license_issue P15207 17008401 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 2nwl A 2.96 BS01 ASP C 1 R276 S278 T314 T352 A353 G354 V355 G359 D394 R397 T398 N401 R262 S264 T300 T338 A339 G340 V341 G345 D380 R383 T384 N387 ? 0005283,0005886,0006865,0015108,0015183,0015293,0015501,0016020,0035725,0042802,0046872,0046942,0070207,0070778,0140009,1902476 remove_due_to_license_issue Kd=1.000000nM O59010 17230192 501 YPVLIKILIGLILGAIVGLILGHYGYAHAVHTYVKPFGDLFVRLLKMLVMPIVFASLVVGAASISPARLGRVGVKIVVYYLLTSAFAVTLGIIMARLFNPGAGIHLAVGGQQFPPLVHILLDIVPTNPFGALANGQVLPTIFFAIILGIAITYLMNSENEKVRKSAETLLDAINGLAEAMYKIVNGVMQYAPIGVFALIAYVMAEQGVHVVGELAKVTAAVYVGLTLQILLVYFVLLKIYGIDPISFIKHAKDAMLTAFVTRSSSGTLPVTMRVAKEMGISEGIYSFTLPLGATINMDGTALYQGVCTFFIANALGSHLTVGQQLTIVLTAVLASIGTAGVPGAGAIMLAMVLHSVGLPLTDPNVAAAYAMILGIDAILDMGRTMVNVTGDLTGTAIVAKTE 2nww A 3.2 BS01 TB1 A 1 S278 T314 A358 G359 D394 R397 T398 N401 S269 T305 A349 G350 D385 R388 T389 N392 ? 0005283,0005886,0006865,0015108,0015183,0015293,0015501,0016020,0035725,0042802,0046872,0046942,0070207,0070778,0140009,1902476 remove_due_to_license_issue Kd=100nM O59010 17230192 423 YPVLQKILIGLILGAIVGLILGHYGYAHAVHTYVKPFGDLFVRLLKMLVMPIVFASLVVGAASISPARLGRVGVKIVVYYLLTSAFAVTLGIIMARLFNPGAGIHLAVGGQQFQPHQAPPLVHILLDIVPTNPFGALANGQVLPTIFFAIILGIAITYLMNSENEKVRKSAETLLDAINGLAEAMYKIVNGVMQYAPIGVFALIAYVMAEQGVHVVGELAKVTAAVYVGLTLQILLVYFVLLKIYGIDPISFIKHAKDAMLTAFVTRSSSGTLPVTMRVAKEMGISEGIYSFTLPLGATINMDGTALYQGVCTFFIANALGSHLTVGQQLTIVLTAVLASIGTAGVPGAGAIMLAMVLHSVGLPLTDPNVAAAYAMILGIDAILDMGRTMVNVTGDLTGTAIVAKTE 2nyr A 2.06 BS02 SVR B 1 T69 F70 R71 A82 F101 Y102 R105 N141 I142 F223 Y255 M259 T34 F35 R36 A47 F66 Y67 R70 N106 I107 F188 Y220 M224 P68 T69 F70 R71 N141 D143 H158 P33 T34 F35 R36 N106 D108 H123 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue IC50=25000nM Q9NXA8 17355872 401 PSSSMADFRKFFAKAKHIVIISGAGVSAESGVPTFRGAGGYWRKWQAQDLATPLAFAHNPSRVWEFYHYRREVMGSKEPNAGHRAIAECETRLGKQGRRVVVITQNIDELHRKAGTKNLLEIHGSLFKTRCTSCGVVAENYKSPICPALSGKGAPEPGTQDASIPVEKLPRCEEAGCGGLLRPHVVWFGENLDPAILEEVDRELAHCDLCLVVGTSSVVYPAAMFAPQVAARGVPVAEFNTERFHFQGPCGTTLPEALA 2nyr B 2.06 BS01 SVR B 1 F70 R71 A86 Y102 R105 H158 V221 F223 G224 E225 N226 L232 V254 Y255 F35 R36 A51 Y67 R70 H123 V186 F188 G189 E190 N191 L197 V219 Y220 P68 T69 F70 R71 N141 D143 H158 P33 T34 F35 R36 N106 D108 H123 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue IC50=25000nM Q9NXA8 17355872 401 PSSSMADFRKFFAKAKHIVIISGAGVSAESGVPTFRGAGGYWRKWQAQDLATPLAFAHNPSRVWEFYHYRREVMGSKEPNAGHRAIAECETRLGKQGRRVVVITQNIDELHRKAGTKNLLEIHGSLFKTRCTSCGVVAENYKSPICPALSGKGAPEPGTQDASIPVEKLPRCEEAGCGGLLRPHVVWFGENLDPAILEEVDRELAHCDLCLVVGTSSVVYPAAMFAPQVAARGVPVAEFNTRFHFQGPCGTTLPEALA 2o0u A 2.1 BS01 C0M A 1 I70 A91 K93 M115 L144 M146 M149 A151 L206 I25 A46 K48 M70 L99 M101 M104 A106 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T176 2.7.11.24 0004672,0004707,0005524,0006468 ic50=3.2uM remove_due_to_license_issue IC50=3162.28nM P53779 17194588 2000 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYREHTIEEWKELIYKEVMN 2o1v A 2.45 BS01 ADP A 1 N107 A111 D149 M154 N162 G198 F199 N23 A27 D65 M70 N78 G83 F84 ? 0005524,0006457,0016887,0051082,0140662 Kd~5uM remove_due_to_license_issue IC50=11447nM, EC50=21000nM P41148 17936703 301 MMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKVWDWELMNDIKPIWQRPSKEVEDDEYKAFYKSFSKESDDPMAYIHFTAEGEVTFKSILFVPTSAPRYIKLYVRRVFITDDFHDMMPKYLNFVKGVVDSDDLPLNVSRETLQQHKLLKVIRKKLVRKTLDMIKKIADEKYNDTFWKEFGTNIKLGVIEDHSNRTRLAKLLRFQSSHHPSDITSLDQYVERMKEKQDKIYFMAGSSRKEAESSPFVERLLKKGYEVIYLTEPVDEYCIQALPEFDGKRFQNVAKEGVKFDESEKTKESREAIEKEFEPLLNWMKDKALKDKIEKAVVSQRLTESPCALVASQYGWSGNMERIMKAQAYQTGKDISTNYYASQKKTFEINPRHPLIKDMLRRVKEDEDDKTVSDLAVVLFETATLRSGYLLPDTKAYGDRIERMLRLSLNI 2o22 A -1.00 BS01 LIU A 1 A97 D100 F101 Y105 D108 F109 G142 V145 A146 F195 Y199 A57 D60 F61 Y65 D68 F69 G102 V105 A106 F155 Y159 ? 0042981 remove_due_to_license_issue P10415 17256834 1000 HAGRTGYDNREIVMKYIHYKLSQRGYEWDAGDDVEENRTEAPEGTESEVVHLTLRQAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGPSMR 2o2u A 2.45 BS01 738 A 1 A91 M146 M149 V196 L206 A44 M99 M102 V149 L159 D189 K191 N194 D207 T226 D142 K144 N147 D160 T166 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.4uM remove_due_to_license_issue IC50=398.11nM P53779 17194588 403 NQFYSVEVGDSTFTVLKRYQNLKPIGSGGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLAVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYHTIEEWKELIYKEVMN 2o3p A 2.24 BS01 QUE A 1 L44 F49 A65 K67 E121 R122 P123 V126 L174 I185 D186 L12 F17 A33 K35 E89 R90 P91 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=1.1uM remove_due_to_license_issue IC50=1100nM, Kd=25nM P11309 17218638 501 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2o3z A 2.25 BS03 AI7 A 1 I198 K202 G210 S211 I185 K189 G197 S198 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 Kd=2uM remove_due_to_license_issue O67648 17296300 301 GLEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFAFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQK 2o3z B 2.25 BS01 AI7 A 1 S211 L212 S198 L199 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 Kd=2uM remove_due_to_license_issue O67648 17296300 301 GLEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFAFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQK 2o3z B 2.25 BS05 AI7 B 1 I18 K202 G210 S211 V217 I17 K189 G197 S198 V204 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 Kd=2uM remove_due_to_license_issue O67648 17296300 301 GLEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFAFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQK 2o4h A 2.7 BS02 AS9 A 1 H21 E24 R63 N70 R71 H116 N117 I127 Y164 R168 E178 E285 Y288 H12 E15 R54 N61 R62 H107 N108 I118 Y155 R159 E169 E276 Y279 3.5.1.15 0005515,0005634,0005737,0005829,0006083,0006531,0016787,0016788,0016811,0019807,0022010,0042802,0046872,0048714 remove_due_to_license_issue P45381 18293939 501 HIQKVAIFGGTHGNELTGVFLVKHWLENGAEIQRTGLEVKPFITNPRAVKKCTRYIDCDLNRIFDLENLGKKMSEDLPYEVRRAQEINHLFGPKDSEDSYDIIFDLHNTTSNMGCTLILEDSRNNFLIQMFHYIKTSLAPLPCYVYLIEHPSLKYATTRSIAKYPVGIEVGPQPQGVLRADILDQMRKMIKHALDFIHHFNEGKEFPPCAIEVYKIIEKVDYPRDENGEIAAIIHPNLQDQDWKPLHPGDPMFLTLDGKTIPLGGDCTVYPVFVNEAAYYEKKEAFAKTTKLTLNAKSIRC 2o4j A 1.74 BS02 VD4 A 1 Y143 V230 S233 R270 S271 S274 W282 C284 H301 H393 Y21 V49 S52 R89 S90 S93 W101 C103 H120 H212 ? 0003677,0004879,0006355 Ki=0.08nM remove_due_to_license_issue P13053 17227670 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNE 2o4k A 1.6 BS01 DR7 A 1 R8 D25 G27 A28 D29 G48 G49 I50 V82 I84 R8 D25 G27 A28 D29 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=35pM remove_due_to_license_issue Q903J0 17360759 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4k B 1.6 BS01 DR7 A 1 D25 G27 A28 D29 G48 G49 I50 P81 I84 D25 G27 A28 D29 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17360759 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4l A 1.33 BS01 TPV A 1 D25 G27 A28 D29 D30 G48 V50 P81 D25 G27 A28 D29 D30 G48 V50 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=608pM remove_due_to_license_issue Q1G1C3 17360759 403 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4l B 1.33 BS01 TPV A 1 R8 D25 G27 G49 V50 V82 R8 D25 G27 G49 V50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17360759 403 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4n A 2.0 BS01 TPV A 1 D25 G27 A28 D29 D30 I32 G48 G49 I50 L82 D25 G27 A28 D29 D30 I32 G48 G49 I50 L82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Kd=15010pM remove_due_to_license_issue Q90SN9 17360759 300 PQITLWKRPLVTVKIGGQLKEALLDTGADDTIFEEMSLPGRWKPIMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPLNVIGRNLLTQIGCTLNF 2o4n B 2.0 BS01 TPV A 1 R8 D25 G27 G49 I50 L82 R8 D25 G27 G49 I50 L82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17360759 300 PQITLWKRPLVTVKIGGQLKEALLDTGADDTIFEEMSLPGRWKPIMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPLNVIGRNLLTQIGCTLNF 2o4p A 1.8 BS01 TPV A 1 R8 D25 A28 D29 D30 G48 G49 I50 V82 R8 D25 A28 D29 D30 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=19pM remove_due_to_license_issue Q5RZ08 17360759 300 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4p B 1.8 BS01 TPV A 1 R8 L23 D25 G27 G49 I50 V82 R8 L23 D25 G27 G49 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q5RZ08 17360759 300 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4r A 1.98 BS02 VD5 A 1 Y143 S233 R270 S271 S274 W282 C284 H301 H393 Y21 S52 R89 S90 S93 W101 C103 H120 H212 ? 0003677,0004879,0006355 Ki=0.4nM remove_due_to_license_issue P13053 17227670 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNE 2o4s A 1.54 BS01 AB1 A 1 D25 G27 A28 D29 G48 I84 D25 G27 A28 D29 G48 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=31pM remove_due_to_license_issue Q5RZ08 17360759 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4s B 1.54 BS01 AB1 A 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 V82 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17360759 400 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2o4z A 2.1 BS02 HSW A 1 H94 H96 L198 T199 T200 H91 H93 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=566nM remove_due_to_license_issue Ki=566nM P00918 17346964 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2o5d A 2.2 BS01 VR1 A 1 L419 R422 M423 H475 S476 Y477 I482 A486 L497 W528 K533 L414 R417 M418 H470 S471 Y472 I477 A481 L492 W523 K528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=7uM remove_due_to_license_issue P26663 17276060 600 HHSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSL 2o5k A 3.2 BS01 HBM A 1 I62 V70 A83 D133 Y134 V135 P136 R141 Q185 N186 L188 I28 V36 A49 D99 Y100 V101 P102 R107 Q151 N152 L154 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=15nM P49841 17764934 0 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 2o63 A 2.0 BS01 MYC A 1 L44 F49 A65 I104 E121 R122 L174 I185 D186 L12 F17 A33 I72 E89 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.78uM remove_due_to_license_issue IC50=780nM P11309 17218638 501 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2o64 A 2.44 BS01 MYU A 1 L44 A65 K67 E89 L120 E121 R122 V126 L174 I185 D186 L12 A33 K35 E57 L88 E89 R90 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.34uM remove_due_to_license_issue IC50=340nM P11309 17218638 501 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2o65 A 2.85 BS01 MYF A 1 L44 F49 V52 K67 L120 I185 D186 L12 F17 V20 K35 L88 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=650nM P11309 17218638 501 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2o6m A 2.3 BS01 dna C 0 A48 P49 G53 K56 N57 K65 T67 A47 P48 G52 K55 N56 K64 T66 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 17516660 401 ~ 421 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASQLCHNTRCHNPLHLCWESLDDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 2o6m A 2.3 BS02 dna D 0 N57 R61 Q63 R74 T95 A96 S97 Q98 N119 N123 N56 R60 Q62 R73 T94 A95 S96 Q97 N118 N122 N119 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 17516660 501 ~ 521 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASQLCHNTRCHNPLHLCWESLDDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 2o6m B 2.3 BS01 dna C 0 N257 R261 Q263 R274 T295 A296 Q298 N319 N323 N56 R60 Q62 R73 T94 A95 Q97 N118 N122 N319 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 17516660 401 ~ 421 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASQLCHNTRCHNPLHLCWESLDDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 2o6m B 2.3 BS02 dna D 0 A248 P249 V252 G253 K256 N257 T267 A47 P48 V51 G52 K55 N56 T66 N319 N118 3.1.-.- 0004519,0006314 remove_due_to_license_issue Q94702 17516660 501 ~ 521 ALTNAQILAVIDSWEETVGQFPVITHHVPLGGGLQGTLHCYEIPLAAPYGVGFAKNGPTRWQYKRTINQVVHRWGSHTVPFLLEPDNINGKTCTASQLCHNTRCHNPLHLCWESLDDNKGRNWCPGPNGGCVHAVVCLRQGPLYGPGATVAGPQQRGSHFVV 2o7e A 1.75 BS01 PMI A 1 Y60 X149 L153 N203 N333 F350 Y54 X143 L145 N195 N325 F342 Y60 G67 L90 N203 Y300 R303 F350 Q436 Y54 G61 L84 N195 Y292 R295 F342 Q428 4.3.1.23 0003824,0006572,0009698,0009699,0016829,0016841,0042802,0044550,0051289,0052883 remove_due_to_license_issue Q3IWB0 17185228 701 PKPAVELDRHIDLDQAHAVASGGARIVLAPPARDRCRASEARLGAVIREARHVYGLTTGFGPLANRLISGENVRTLQANLVHFLASGVGPVLDWTTARAMVLARLVSIAQGASGASEGTIARLIDLLNSELAPAVPSRGTVGGDLTPLAHMVLCLQGRGDFLDRDGTRLDGAEGLRRGRLQPLDLSHRDALALVNGTSAMTGIALVNAHACRHLGNWAVALTALLAECLRGRTEAWAAALSDLRPHPGQKDAAARLRARVDGSARVVRHVIAERRLDAGDIGTEPEAGQDAYSLRCAPQVLGAGFDTLAWHDRVLTIELNAVTDNPVFPPDGSVPALHGGNFMGQHVALTSDALATAVTVLAGLAERQIARLTDERLNRGLPPFLHRGPAGLNSGFMGAQVTATALLAEMRATGPASIHSISTNAANQDVVSLGTIAARLCREKIDRWAEILAILALCLAQAAELRCGSGLDGVSPAGKKLVQALREQFPPLETDRPLGQEIAALATHLLQQSPV 2o7e A 1.75 BS02 PMI D 1 Y300 R303 Y292 R295 Y60 G67 L90 N203 Y300 R303 F350 Q436 Y54 G61 L84 N195 Y292 R295 F342 Q428 4.3.1.23 0003824,0006572,0009698,0009699,0016829,0016841,0042802,0044550,0051289,0052883 remove_due_to_license_issue Q3IWB0 17185228 701 PKPAVELDRHIDLDQAHAVASGGARIVLAPPARDRCRASEARLGAVIREARHVYGLTTGFGPLANRLISGENVRTLQANLVHFLASGVGPVLDWTTARAMVLARLVSIAQGASGASEGTIARLIDLLNSELAPAVPSRGTVGGDLTPLAHMVLCLQGRGDFLDRDGTRLDGAEGLRRGRLQPLDLSHRDALALVNGTSAMTGIALVNAHACRHLGNWAVALTALLAECLRGRTEAWAAALSDLRPHPGQKDAAARLRARVDGSARVVRHVIAERRLDAGDIGTEPEAGQDAYSLRCAPQVLGAGFDTLAWHDRVLTIELNAVTDNPVFPPDGSVPALHGGNFMGQHVALTSDALATAVTVLAGLAERQIARLTDERLNRGLPPFLHRGPAGLNSGFMGAQVTATALLAEMRATGPASIHSISTNAANQDVVSLGTIAARLCREKIDRWAEILAILALCLAQAAELRCGSGLDGVSPAGKKLVQALREQFPPLETDRPLGQEIAALATHLLQQSPV 2o7e B 1.75 BS01 PMI B 1 Y60 X149 L153 N203 F350 Y54 X143 L145 N195 F342 Y60 G67 L90 N203 Y300 R303 F350 Q436 Y54 G61 L84 N195 Y292 R295 F342 Q428 4.3.1.23 0003824,0006572,0009698,0009699,0016829,0016841,0042802,0044550,0051289,0052883 remove_due_to_license_issue Q3IWB0 17185228 701 PKPAVELDRHIDLDQAHAVASGGARIVLAPPARDRCRASEARLGAVIREARHVYGLTTGFGPLANRLISGENVRTLQANLVHFLASGVGPVLDWTTARAMVLARLVSIAQGASGASEGTIARLIDLLNSELAPAVPSRGTVGGDLTPLAHMVLCLQGRGDFLDRDGTRLDGAEGLRRGRLQPLDLSHRDALALVNGTSAMTGIALVNAHACRHLGNWAVALTALLAECLRGRTEAWAAALSDLRPHPGQKDAAARLRARVDGSARVVRHVIAERRLDAGDIGTEPEAGQDAYSLRCAPQVLGAGFDTLAWHDRVLTIELNAVTDNPVFPPDGSVPALHGGNFMGQHVALTSDALATAVTVLAGLAERQIARLTDERLNRGLPPFLHRGPAGLNSGFMGAQVTATALLAEMRATGPASIHSISTNAANQDVVSLGTIAARLCREKIDRWAEILAILALCLAQAAELRCGSGLDGVSPAGKKLVQALREQFPPLETDRPLGQEIAALATHLLQQSPV 2o7e B 1.75 BS02 PMI C 1 Y300 R303 Y292 R295 Y60 G67 L90 N203 Y300 R303 F350 Q436 Y54 G61 L84 N195 Y292 R295 F342 Q428 4.3.1.23 0003824,0006572,0009698,0009699,0016829,0016841,0042802,0044550,0051289,0052883 remove_due_to_license_issue Q3IWB0 17185228 701 PKPAVELDRHIDLDQAHAVASGGARIVLAPPARDRCRASEARLGAVIREARHVYGLTTGFGPLANRLISGENVRTLQANLVHFLASGVGPVLDWTTARAMVLARLVSIAQGASGASEGTIARLIDLLNSELAPAVPSRGTVGGDLTPLAHMVLCLQGRGDFLDRDGTRLDGAEGLRRGRLQPLDLSHRDALALVNGTSAMTGIALVNAHACRHLGNWAVALTALLAECLRGRTEAWAAALSDLRPHPGQKDAAARLRARVDGSARVVRHVIAERRLDAGDIGTEPEAGQDAYSLRCAPQVLGAGFDTLAWHDRVLTIELNAVTDNPVFPPDGSVPALHGGNFMGQHVALTSDALATAVTVLAGLAERQIARLTDERLNRGLPPFLHRGPAGLNSGFMGAQVTATALLAEMRATGPASIHSISTNAANQDVVSLGTIAARLCREKIDRWAEILAILALCLAQAAELRCGSGLDGVSPAGKKLVQALREQFPPLETDRPLGQEIAALATHLLQQSPV 2o7e D 1.75 BS01 PMI A 1 Y300 R303 Y291 R294 Y60 G67 L90 N203 Y300 R303 F350 Q436 Y53 G60 L83 N194 Y291 R294 F341 Q427 4.3.1.23 0003824,0006572,0009698,0009699,0016829,0016841,0042802,0044550,0051289,0052883 remove_due_to_license_issue Q3IWB0 17185228 701 KPAVELDRHIDLDQAHAVASGGARIVLAPPARDRCRASEARLGAVIREARHVYGLTTGFGPLANRLISGENVRTLQANLVHFLASGVGPVLDWTTARAMVLARLVSIAQGASGASEGTIARLIDLLNSELAPAVPSRGTVGGDLTPLAHMVLCLQGRGDFLDRDGTRLDGAEGLRRGRLQPLDLSHRDALALVNGTSAMTGIALVNAHACRHLGNWAVALTALLAECLRGRTEAWAAALSDLRPHPGQKDAAARLRARVDGSARVVRHVIAERRLDAGDIGTEPEAGQDAYSLRCAPQVLGAGFDTLAWHDRVLTIELNAVTDNPVFPPDGSVPALHGGNFMGQHVALTSDALATAVTVLAGLAERQIARLTDERLNRGLPPFLHRGPAGLNSGFMGAQVTATALLAEMRATGPASIHSISTNAANQDVVSLGTIAARLCREKIDRWAEILAILALCLAQAAELRCGSGLDGVSPAGKKLVQALREQFPPLETDRPLGQEIAALATHLLQQSPV 2o7e D 1.75 BS02 PMI D 1 Y60 X149 L153 N203 N333 F350 Y53 X142 L144 N194 N324 F341 Y60 G67 L90 N203 Y300 R303 F350 Q436 Y53 G60 L83 N194 Y291 R294 F341 Q427 4.3.1.23 0003824,0006572,0009698,0009699,0016829,0016841,0042802,0044550,0051289,0052883 remove_due_to_license_issue Q3IWB0 17185228 701 KPAVELDRHIDLDQAHAVASGGARIVLAPPARDRCRASEARLGAVIREARHVYGLTTGFGPLANRLISGENVRTLQANLVHFLASGVGPVLDWTTARAMVLARLVSIAQGASGASEGTIARLIDLLNSELAPAVPSRGTVGGDLTPLAHMVLCLQGRGDFLDRDGTRLDGAEGLRRGRLQPLDLSHRDALALVNGTSAMTGIALVNAHACRHLGNWAVALTALLAECLRGRTEAWAAALSDLRPHPGQKDAAARLRARVDGSARVVRHVIAERRLDAGDIGTEPEAGQDAYSLRCAPQVLGAGFDTLAWHDRVLTIELNAVTDNPVFPPDGSVPALHGGNFMGQHVALTSDALATAVTVLAGLAERQIARLTDERLNRGLPPFLHRGPAGLNSGFMGAQVTATALLAEMRATGPASIHSISTNAANQDVVSLGTIAARLCREKIDRWAEILAILALCLAQAAELRCGSGLDGVSPAGKKLVQALREQFPPLETDRPLGQEIAALATHLLQQSPV 2o7n A 1.75 BS01 2O7 A 1 Y166 I235 Y257 L302 K305 I306 Y39 I108 Y130 L175 K178 I179 ? ic50=15nM remove_due_to_license_issue P20701 17291752 1 MNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKRKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIY 2o8h A 1.8 BS02 227 A 1 L625 F629 F686 M703 Q716 F719 L172 F176 F233 M250 Q263 F266 3.1.4.17 0004114,0007165,0008081 Ki=25nM remove_due_to_license_issue Ki=25nM Q9QYJ6 17228859 999 LPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIRGEE 2o8k A -1.00 BS01 dna B 0 S39 D40 R56 A60 R63 E64 S70 S26 D27 R43 A47 R50 E51 S57 ? 0001216,0016987 remove_due_to_license_issue O66858 17481658 101 ~ 114 HMLTQGELMKLIKEIVENEDKRKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERRI 2o8k A -1.00 BS02 dna C 0 H14 V54 A55 R57 T58 Y62 H1 V41 A42 R44 T45 Y49 ? 0001216,0016987 remove_due_to_license_issue O66858 17481658 115 ~ 128 HMLTQGELMKLIKEIVENEDKRKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERRI 2o9a A 1.8 BS01 PYR A 1 S65 G66 D118 C128 S145 S147 S65 G66 D118 C128 S145 S147 ? remove_due_to_license_issue P16528 17426033 905 GHMSRNLLAIVHPILRNLMEESGETVNMAVLDQSDHEAIIIDQVQCTHLMRMSAPIGGKLPMHASGAGKAFLAQLSEEQVTKLLHRKGLHAYTHATLVSPVHLKEDLAQTRKRGYSFDDEEHALGLRCLAACIFDEHREPFAAISISGPISRITDDRVTEFGAMVIKAAKEVTLAYGGMRGS 2o9a D 1.8 BS01 PYR D 1 S65 G66 D118 C128 S145 S147 S65 G66 D118 C128 S145 S147 ? remove_due_to_license_issue P16528 17426033 908 GHMSRNLLAIVHPILRNLMEESGETVNMAVLDQSDHEAIIIDQVQCTHLMRMSAPIGGKLPMHASGAGKAFLAQLSEEQVTKLLHRKGLHAYTHATLVSPVHLKEDLAQTRKRGYSFDDEEHALGLRCLAACIFDEHREPFAAISISGPISRITDDRVTEFGAMVIKAAKEVTLAYGGMR 2o9i A 2.8 BS02 444 A 1 L209 M243 M246 Q285 F288 W299 Y306 H407 L411 F420 L55 M89 M92 Q131 F134 W145 Y152 H253 L257 F266 ? 0003677,0004879,0006355 remove_due_to_license_issue EC50=36nM, IC50=40nM O75469 17215127 2 GLTEEQRMMIRELMDAQMKTFDTTFSHFKNFRLPGVLSREEAAKWSQVRKDLCSLKVSLQLRGEDGSVWNYKPPADSGGKEIFSLLPHMADMSTYMFKGIISFAKVISYFRDLPIEDQISLLKGAAFELSQLRFNTVFNAETGTWECGRLSYCLEDTAGGFQQLLLEPMLKFHYMLKKLQLHEEEYVLMQAISLFSPDRPGVLQHRVVDQLQEQFAITLKSYIECNRPQPAHRFLFLKIMAMLTELRSINAQHTQRLLRIQDIHPFATPLMQELFGITG 2o9j A 2.65 BS03 CZA A 1 L61 V62 N101 A102 L311 P312 L61 V62 N101 A102 L297 P298 D351 D703 D707 D337 D689 D693 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 17259168 1001 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 2o9l A -1.00 BS01 dna B 0 S26 D27 R43 R50 S57 R59 S26 D27 R43 R50 S57 R59 ? 0001216,0016987 remove_due_to_license_issue O66858 17481658 64 ~ 77 HMLTQGELMKLIKEIVENEDKRKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERRI 2o9l A -1.00 BS02 dna C 0 H1 V41 A42 R44 T45 Y49 H1 V41 A42 R44 T45 Y49 ? 0001216,0016987 remove_due_to_license_issue O66858 17481658 78 ~ 91 HMLTQGELMKLIKEIVENEDKRKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERRI 2oa0 A 3.4 BS01 CZA A 1 Q56 L61 V62 L98 N101 A102 E309 L311 P312 Q56 L61 V62 L98 N101 A102 E301 L303 P304 D351 D703 D707 D343 D695 D699 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 17259168 1001 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 2oag B 2.3 BS01 DLI B 1 E205 E206 V207 S209 F357 R358 S630 Y631 Y662 Y666 V711 H740 E167 E168 V169 S171 F319 R320 S592 Y593 Y624 Y628 V673 H702 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=3.4nM remove_due_to_license_issue Ki=3.4nM P27487 17276063 4000 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2oah A 1.8 BS01 QIN A 1 S10 Q12 G13 D32 Y71 T72 Q73 F108 D228 G230 T231 T232 N233 R235 S16 Q18 G19 D38 Y77 T78 Q79 F114 D221 G223 T224 T225 N226 R228 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=11nM remove_due_to_license_issue IC50=11nM P56817 17257835 902 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2oax A 2.29 BS01 SNL A 1 L766 L769 N770 L772 Q776 M807 L810 L814 F829 M845 L938 F941 C942 T945 F956 L26 L29 N30 L32 Q36 M67 L70 L74 F89 M105 L189 F192 C193 T196 F207 ? remove_due_to_license_issue IC50=11nM, Ki=2.323nM P08235 17569793 1001 PVMVLENIEPEIVYAGYDSDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMCLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFH 2oaz A 1.9 BS03 I96 A 1 F219 H231 D251 E364 H382 Y444 F96 H108 D128 E241 H259 Y321 D251 D262 H331 H339 E364 E459 D128 D139 H208 H216 E241 E336 3.4.11.18 0006508,0070006 Ki=2nM remove_due_to_license_issue P50579 17636946 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIIKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 2obf A 2.3 BS01 F83 A 1 Y35 N39 Y40 R44 V53 G54 L58 Y85 Y126 F182 E219 Y222 Y12 N16 Y17 R21 V30 G31 L35 Y62 Y103 F159 E196 Y199 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Ki=1.4nM remove_due_to_license_issue Ki=63nM P11086 17845018 2001 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWALRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2obj A 2.5 BS01 VRV A 1 G45 A65 K67 I104 L120 E121 L174 I185 D186 G13 A33 K35 I72 L88 E89 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.05uM remove_due_to_license_issue IC50=50nM P11309 17251021 400 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 2obo A 2.6 BS04 HUD A 1 H57 G137 S139 F154 R155 A156 A157 D168 H59 G139 S141 F156 R157 A158 A159 D170 H57 D81 G137 S139 H59 D83 G139 S141 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036,0097264 remove_due_to_license_issue Q91RS4 17444623 903 MGAPITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRSG 2oc0 A 2.3 BS04 HU1 A 1 H57 K136 G137 S139 F154 R155 A156 A157 C159 H57 K136 G137 S139 F154 R155 A156 A157 C159 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 17444623 999 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2oc1 A 2.7 BS04 HU2 A 1 Q41 T42 H57 R109 I132 K136 G137 S139 R155 A156 A157 D168 Q43 T44 H59 R111 I134 K138 G139 S141 R157 A158 A159 D170 H57 D81 G137 S139 H59 D83 G139 S141 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 17444623 999 MGAPITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2oc2 A 2.25 BS02 RX3 A 1 Q281 H353 A354 S355 A356 H383 E384 H387 F391 H410 E411 F457 K511 F512 H513 V518 Y520 Y523 Q242 H314 A315 S316 A317 H344 E345 H348 F352 H371 E372 F417 K471 F472 H473 V478 Y480 Y483 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H473 Y483 3.4.15.1 0006508,0008237,0008241,0016020 Ki=3nM remove_due_to_license_issue Ki=3nM P12821 17439247 680 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTP 2oc4 A 2.592 BS01 IMH A 1 A116 A117 G118 F200 E201 V217 M219 N243 D257 A116 A117 G118 F200 E201 V217 M219 N243 D257 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 D257 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 D257 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 17407325 300 MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANDEEVLAAGKQAAQKLEQFVSILMASIPLPD 2oc7 A 2.7 BS03 HU4 A 1 H57 L135 G137 S139 F154 R155 A156 A157 D168 H57 L135 G137 S139 F154 R155 A156 A157 D168 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 17444623 999 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2oc9 A 2.59 BS01 IMH A 1 A116 G118 F200 E201 V217 M219 N243 V260 A110 G112 F194 E195 V211 M213 N237 V254 S33 H86 Y88 E89 A116 M219 S220 N243 V245 G257 S33 H80 Y82 E83 A110 M213 S214 N237 V239 G251 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 17407325 300 MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANGEEVLAAGKQAAQKLEQFVSILMASIPL 2of2 A 2.0 BS01 547 A 1 L251 A271 Y318 M319 G322 N369 L371 L21 A41 Y88 M89 G92 N139 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.21uM remove_due_to_license_issue IC50=210nM P06239 17276681 201 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 2of4 A 2.7 BS01 979 A 1 L251 V259 A271 Y318 M319 G322 A368 L371 L21 V29 A41 Y88 M89 G92 A138 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=81nM P06239 17276681 101 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 2off A 2.2 BS01 OFF A 1 Q71 Q72 Y155 F196 T240 R242 R309 R310 Q60 Q61 Y144 F185 T229 R231 R292 R293 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=0.46uM remove_due_to_license_issue Ki=460nM P00489 17600143 930 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2ofu A 2.0 BS01 1N9 A 1 L251 V259 A271 K273 E288 T316 Y318 M319 G322 S323 L371 D382 L23 V31 A43 K45 E60 T88 Y90 M91 G94 S95 L143 D154 D364 R366 A368 N369 D382 A400 F402 D136 R138 A140 N141 D154 A172 F174 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.0006uM remove_due_to_license_issue IC50=0.6nM P06239 16884310 1 PQKPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 2ofv A 2.0 BS01 242 A 1 V259 A271 V272 K273 E288 L291 M292 I314 T316 Y318 M319 A381 D382 F383 V29 A41 V42 K43 E51 L54 M55 I77 T79 Y81 M82 A144 D145 F146 D364 R366 A368 N369 D382 D127 R129 A131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.2nM remove_due_to_license_issue IC50=0.2nM P06239 16970394 503 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLAIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFF 2og8 A 2.3 BS01 1N8 A 1 A271 K273 E288 M292 L300 T316 Y318 M319 L371 A381 D382 F383 A35 K37 E52 M56 L64 T80 Y82 M83 L135 A145 D146 F147 D364 R366 A368 N369 D382 D128 R130 A132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5nM remove_due_to_license_issue IC50=0.500000nM P06239 16970394 501 EWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFT 2ogm B 3.5 BS01 rna 0 0 G65 G110 G115 G139 S140 R144 G148 P189 G65 G110 G115 G139 S140 R144 G148 P189 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue Q9RXK2 17360517 1 ~ 2877 MKGILGTKIGMTQIWKNDRAIPVTVVLAGPCPIVQRKTAQTDGYEAVQIGYAPKAERKVNKPMQGHFAKAGVAPTRILREFRGFAPDGDSVNVDIFAEGEKIDATGTSKGKGTQGVMKRWNFAGGPASHGSKKWHRRPGSIGQRKTPGRVYKGKRMAGHMGMERVTVQNLEVVEIRAGENLILVKGAIPGANGGLVVLRSAAKAS 2ogn B 3.56 BS01 rna 0 0 M11 K61 G65 G110 Q114 G115 A123 G139 S140 G142 Q143 R144 G148 G153 P189 M11 K61 G65 G110 Q114 G115 A123 G139 S140 G142 Q143 R144 G148 G153 P189 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue Q9RXK2 17360517 1 ~ 2877 MKGILGTKIGMTQIWKNDRAIPVTVVLAGPCPIVQRKTAQTDGYEAVQIGYAPKAERKVNKPMQGHFAKAGVAPTRILREFRGFAPDGDSVNVDIFAEGEKIDATGTSKGKGTQGVMKRWNFAGGPASHGSKKWHRRPGSIGQRKTPGRVYKGKRMAGHMGMERVTVQNLEVVEIRAGENLILVKGAIPGANGGLVVLRSAAKAS 2ogo B 3.66 BS01 rna 0 0 G65 G110 S140 P189 G65 G110 S140 P189 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue Q9RXK2 17360517 2 ~ 2877 MKGILGTKIGMTQIWKNDRAIPVTVVLAGPCPIVQRKTAQTDGYEAVQIGYAPKAERKVNKPMQGHFAKAGVAPTRILREFRGFAPDGDSVNVDIFAEGEKIDATGTSKGKGTQGVMKRWNFAGGPASHGSKKWHRRPGSIGQRKTPGRVYKGKRMAGHMGMERVTVQNLEVVEIRAGENLILVKGAIPGANGGLVVLRSAAKAS 2ogy A 2.3 BS02 C2F A 1 E6 M11 F12 D75 N96 D160 G196 S198 Q202 R207 I227 E6 M11 F12 D75 N96 D160 G196 S198 Q202 R207 I227 2.1.1.258 0005509,0005515,0005829,0008168,0008705,0009086,0015977,0031419,0032259,0042558,0044237,0046653,0046872,0050667,0102036 Kd=33.2uM remove_due_to_license_issue Q46389 17172470 3000 MLIIGERINGMFGDIKRAIQERDPAPVQEWARRQEEGGARALDLNVGPAVQDKVSAMEWLVEVTQEVSNLTLCLDSTNIKAIEAGLKKCKNRAMINSTNAEREKVEKLFPLAVEHGAALIGLTMNKTGIPKDSDTRLAFAMELVAAADEFGLPMEDLYIDPLILPANVAQDHAPEVLKTLQQIKMLADPAPKTVLGLSAVSQNCQNRPLINRTFLAMAMACGLDAAIADACDEALIETAATAEILLNQTVYCDSFVKMFKTR 2ogz A 2.1 BS01 U1N A 1 E205 E206 Y547 S630 Y631 V656 Y662 Y666 V711 E167 E168 Y509 S592 Y593 V618 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=84nM remove_due_to_license_issue IC50=84nM P27487 17239592 767 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2oh0 E 2.2 BS02 2PY E 1 G55 A70 K72 E121 Y122 V123 N171 L173 T183 D184 G41 A56 K58 E107 Y108 V109 N157 L159 T169 D170 N171 D184 N157 D170 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=18nM remove_due_to_license_issue P00517 17258463 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2oh4 A 2.05 BS01 GIG A 1 V846 A864 E883 V897 F916 C917 G920 H1024 L1033 C1043 D1044 F1045 V33 A51 E70 V84 F103 C104 G107 H154 L163 C173 D174 F175 D1026 A1028 R1030 N1031 D1044 K1053 D1062 D156 A158 R160 N161 D174 K183 D192 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=3.5nM remove_due_to_license_issue P35968 17676829 303 HCERLPYDASKWEFPRDRLNLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQD 2ohk A 2.2 BS01 1SQ A 1 D32 Y71 D228 T231 D34 Y73 D220 T223 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=2000000nM P56817 17315856 390 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohl A 2.65 BS01 2AQ A 1 D32 G34 I118 D228 D34 G36 I120 D220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=800000nM, Kd=900000nM P56817 17315856 390 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohm A 2.7 BS01 8AP A 1 D32 G34 Y71 F108 I118 D228 T231 D34 G36 Y73 F110 I120 D220 T223 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=310000nM P56817 17315856 389 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohp A 2.25 BS01 6IP A 1 L30 D32 Y71 I118 D228 G230 L32 D34 Y73 I120 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=94uM remove_due_to_license_issue IC50=94000nM P56817 17315857 389 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohq A 2.1 BS01 7IP A 1 G11 G13 L30 D32 Y71 F108 I118 D228 S229 G230 G13 G15 L32 D34 Y73 F110 I120 D220 S221 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=25uM remove_due_to_license_issue IC50=25000nM P56817 17315857 404 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohr A 2.25 BS01 8IP A 1 G11 L30 D32 F108 D228 G230 T231 G13 L32 D34 F110 D220 G222 T223 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=100uM remove_due_to_license_issue IC50=100000nM P56817 17315857 504 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohs A 2.45 BS01 9IP A 1 G13 L30 D32 F108 D228 S229 G230 T231 G15 L32 D34 F110 D217 S218 G219 T220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=40uM remove_due_to_license_issue IC50=40000nM P56817 17315857 389 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2oht A 2.3 BS01 IP6 A 1 Q12 G13 L30 D32 Y71 F108 I110 W115 D228 G230 Q14 G15 L32 D34 Y73 F110 I112 W117 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=9.1uM remove_due_to_license_issue IC50=9100nM P56817 17315857 601 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohu A 2.35 BS01 IP7 A 1 Q12 D32 S35 V69 Y71 W76 F108 W115 R128 D228 G230 Q14 D34 S37 V71 Y73 W78 F110 W117 R130 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=4.2uM remove_due_to_license_issue IC50=4200nM P56817 17315857 390 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ohv A 2.5 BS01 NHL A 1 S11 D36 Y53 T75 T117 H185 S11 D36 Y48 T70 T112 H180 D10 S11 C73 E152 C183 H185 D10 S11 C68 E147 C178 H180 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0071555 Ki=16nM remove_due_to_license_issue Q9A1B7 17658548 400 MDTRPIGFLDSGVGGLTVVCELIRQLPHEKIVYIGDSARAPKKQIKEYTWELVNFLLTQNVKMIVFACNTATAVAWEEVKAALDIPVLGVVLPGASAAIKSTTKGQVGVIGTPMTVASDIYRKKIQLLAPSIQVRSLACPKFVPIVESNEMCSSIAKKIVYDSLAPLVGKIDTLVLGCTHYPLLRPIIQNVMGPSVKLIDSGAECVRDISVLLNYFDINGNYHQAVEHRFFTTANPEIFQEIASIWLKQKINVEHVTL 2oi0 A 2.0 BS02 283 A 1 T347 G349 L401 H405 E406 H409 A439 T132 G134 L186 H190 E191 H194 A224 3.4.24.86 0004222,0006508,0008237 Ki=28nM remove_due_to_license_issue P78536 17289381 1 ADPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYVGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERSNKVIEGR 2oi2 A 2.5 BS02 DP6 A 1 K13 H20 V22 S92 S132 D135 T175 G255 G256 K10 H17 V19 S85 S125 D128 T168 G248 G249 2.7.1.36 0004496,0005524,0005737,0005829,0006629,0008299,0016301,0019287,0046872 Kd=500nM remove_due_to_license_issue A0A0H2UNK6 17400916 300 KVGVGQAHSKIILIGEHAVVYGYPAISLPLLEVEVTCKVVPAESPWRLYEEDTLSMAVYASLEYLNITEACIRCEIDEKRGMGSSAAISIAAIRAVFDYYQADLPHDVLEILVNRAEMIAHMNPSGLDAKTCLSDQPIRFIKNVGFTELEMDLSAYLVIADTGVYGHTREAIQVVQNKGKDALPFLHALGELTQQAEIAISQKDAEGLGQILSQAHLHLKEIGVSSLEADSLVETALSHGALGAKMSGGGLGGCIIALVTNLTHAQELAERLEEKGAVQTWIESL 2oic A 2.4 BS01 STU A 1 M192 E194 G195 V200 A211 Y264 M265 G268 A315 N316 L318 M30 E32 G33 V38 A49 Y91 M92 G95 A142 N143 L145 D311 K313 A315 N316 D329 T351 D138 K140 A142 N143 D156 T172 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=4nM remove_due_to_license_issue Q9NWZ3 17312103 1 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARATVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 2oiq A 2.07 BS01 STI A 1 V281 A293 I294 K295 E310 M314 I336 T338 Y340 M341 V383 H384 A403 D404 F405 V26 A38 I39 K40 E55 M59 I81 T83 Y85 M86 V128 H129 A148 D149 F150 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F156 2.7.10.2 0004672,0004713,0005524,0006468 Kd=42uM remove_due_to_license_issue IC50=2784nM P00523 17355866 1001 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2oj9 A 2.0 BS01 BMI A 1 L975 G976 A1001 E1050 L1051 M1052 G1055 M1112 L22 G23 A48 E97 L98 M99 G102 M151 D1105 R1109 N1110 D1123 E1132 D144 R148 N149 D162 E171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.39uM remove_due_to_license_issue IC50=390nM P08069 17317169 301 ADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 2ojf E 2.1 BS02 4PY E 1 T51 G52 G55 R56 V57 A70 K72 E121 Y122 V123 L173 T183 D184 T37 G38 G41 R42 V43 A56 K58 E107 Y108 V109 L159 T169 D170 N171 D184 N157 D170 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=110nM remove_due_to_license_issue P00517 17258463 1000 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2ojg A 2.0 BS01 19A A 1 I29 G30 Y34 V37 K52 I82 Q103 L105 M106 K112 L154 C164 I13 G14 Y18 V21 K36 I66 Q87 L89 M90 K96 L138 C148 D147 K149 S151 N152 D165 T188 D131 K133 S135 N136 D149 T172 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Ki=2.3uM remove_due_to_license_issue Ki=2300nM P28482 17300186 360 FDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQPG 2oji A 2.6 BS01 33A A 1 G30 V37 K52 Q103 M106 L154 D165 G18 V25 K40 Q91 M94 L142 D153 D147 K149 S151 N152 D165 T188 D135 K137 S139 N140 D153 T176 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue Ki=85nM P28482 17300186 360 RGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 2ojj A 2.4 BS01 82A A 1 I29 G30 E31 G32 G35 V37 K52 I82 Q103 M106 N152 L154 D165 I17 G18 E19 G20 G23 V25 K40 I70 Q91 M94 N140 L142 D153 D147 K149 S151 N152 D165 T188 D135 K137 S139 N140 D153 T176 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Ki=0.002uM remove_due_to_license_issue Ki=2nM P28482 17300186 360 RGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 2ok1 A 2.4 BS01 33A A 1 P69 I70 A74 V78 A91 K93 M146 E147 M149 D150 L206 P24 I25 A27 V31 A44 K46 M99 E100 M102 D103 L159 D189 K191 N194 D207 T226 D142 K144 N147 D160 T166 2.7.11.24 0004672,0004707,0005524,0006468 Ki=0.55uM remove_due_to_license_issue Ki=550nM P53779 17300186 1 NQFYSVEVGDSTFTVLKRYQNLKPIGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLAVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPDEREHTIEEWKELIYKEVMN 2ole A 2.4 BS01 KR2 A 1 E205 E206 F357 S630 Y662 Y666 V711 H740 E167 E168 F319 S592 Y624 Y628 V673 H702 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=56.2nM remove_due_to_license_issue IC50=70nM P27487 17331715 1001 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2on3 A 3.0 BS01 XAP A 1 G237 F238 P275 G276 R277 Y389 G221 F222 P259 G260 R261 Y360 K69 H197 E274 K63 H181 E258 4.1.1.17 0001822,0003824,0004586,0005515,0005737,0005829,0006595,0006596,0008283,0008284,0009615,0016831,0033387,0042176,0042803 remove_due_to_license_issue P11926 17407445 601 EEFDCHFLDEGFTAKDILDQKINEVSSSDDKDAFYVADLGDILKKHLRWLKALPRVTPFYAVKCNDSKAIVKTLAATGTGFDCASKTEIQLVQSLGVPPERIIYANPCKQVSQIKYAANNGVQMMTFDSEVELMKVARAHPKAKLVLRIATVKFGATLRTSRLLLERAKELNIDVVGVSFHVGSGCTDPETFVQAISDARCVFDMGAEVGFSMYLLDIGGGFPGSEDVKLKFEEITGVINPALDKYFPSDSGVRIIAEPGRYYVASAFTLAVNIIAKKIVLEQTFMYYVNDGVYGSFNCILYDHAHVKPLLQKRPKPDEKYYSSSIWGPTCDGLDRIVERCDLPEMHVGDWMLFENMGAYTVAAASTFNGFQRPTIYYVMSGPAWQLMQQFQ 2on3 B 3.0 BS01 XAP B 1 H197 G236 G237 F238 P275 G276 R277 Y389 H181 G220 G221 F222 P259 G260 R261 Y360 K69 H197 E274 K63 H181 E258 4.1.1.17 0001822,0003824,0004586,0005515,0005737,0005829,0006595,0006596,0008283,0008284,0009615,0016831,0033387,0042176,0042803 remove_due_to_license_issue P11926 17407445 601 EEFDCHFLDEGFTAKDILDQKINEVSSSDDKDAFYVADLGDILKKHLRWLKALPRVTPFYAVKCNDSKAIVKTLAATGTGFDCASKTEIQLVQSLGVPPERIIYANPCKQVSQIKYAANNGVQMMTFDSEVELMKVARAHPKAKLVLRIATVKFGATLRTSRLLLERAKELNIDVVGVSFHVGSGCTDPETFVQAISDARCVFDMGAEVGFSMYLLDIGGGFPGSEDVKLKFEEITGVINPALDKYFPSDSGVRIIAEPGRYYVASAFTLAVNIIAKKIVLEQTFMYYVNDGVYGSFNCILYDHAHVKPLLQKRPKPDEKYYSSSIWGPTCDGLDRIVERCDLPEMHVGDWMLFENMGAYTVAAASTFNGFQRPTIYYVMSGPAWQLMQQFQ 2on6 A 2.503 BS01 IMH A 1 A116 A117 G118 F200 E201 V217 G218 M219 S220 N243 A112 A113 G114 F196 E197 V213 G214 M215 S216 N239 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 F257 S33 H60 H82 Y84 E85 A112 M215 S216 N239 V241 F253 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 Ki=172nM remove_due_to_license_issue P00491 17407325 300 MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANFEEVLAAGKQAAQKLEQFVSILMASIPLPD 2onb A 2.7 BS01 7PA A 1 R50 H196 R215 S216 R25 H150 R169 S170 E87 Y135 C195 R215 D218 E62 Y89 C149 R169 D172 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue Ki=2700nM P04818 17297914 319 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKME 2onc A 2.55 BS01 SY1 A 1 E205 E206 F357 Y547 S630 Y631 Y662 Y666 V711 E163 E164 F315 Y505 S588 Y589 Y620 Y624 V669 Y547 S630 Y631 D708 H740 Y505 S588 Y589 D666 H698 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=13nM P27487 17441705 800 AKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2onc A 2.55 BS02 SY1 A 2 E191 D192 F240 K250 R253 E149 D150 F198 K208 R211 Y547 S630 Y631 D708 H740 Y505 S588 Y589 D666 H698 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=13nM P27487 17441705 801 AKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2ony A 2.6 BS02 TMJ A 1 Y35 N39 Y40 R44 G54 K57 Y126 F182 E219 Y222 Y12 N16 Y17 R21 G31 K34 Y103 F159 E196 Y199 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 remove_due_to_license_issue Ki=210nM P11086 17845018 2001 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2onz A 2.8 BS02 TMJ A 1 Y35 N39 Y40 R44 V53 G54 Y85 Y126 F182 E219 Y222 Y12 N16 Y17 R21 V30 G31 Y62 Y103 F159 E196 Y199 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 remove_due_to_license_issue Ki=210nM P11086 17845018 2001 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWALRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2oo8 X 2.2 BS01 RAJ X 1 A853 E872 L876 I886 I902 Y904 A905 H962 A981 D982 F983 A13 E29 L33 I43 I55 Y57 A58 H115 A134 D135 F136 N969 D982 N122 D135 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1nM Q02763 17350837 1 GQVLKARIRMDAAIKRMKEKDDHRDFAGELEVLCKLGHHPNIINLLGACEHYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLMGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGID 2ooh B 1.85 BS01 OX3 B 1 P1 M2 K32 Y36 H62 S63 I64 M101 F113 P1 M2 K32 Y36 H62 S63 I64 M101 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=1.3uM remove_due_to_license_issue IC50=1300nM P14174 17526494 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 2ooh C 1.85 BS01 OX3 B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=1.3uM remove_due_to_license_issue IC50=1300nM P14174 17526494 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 2ooh C 1.85 BS02 OX3 C 1 P1 M2 K32 S63 I64 M101 V106 F113 P1 M2 K32 S63 I64 M101 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=1.3uM remove_due_to_license_issue IC50=1300nM P14174 17526494 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 2ooz A 1.8 BS01 OX5 A 1 P1 M2 Y36 H62 S63 V106 P1 M2 Y36 H62 S63 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM P14174 17526494 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 2ooz B 1.8 BS01 OX5 A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM P14174 17526494 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 2ooz B 1.8 BS02 OX5 B 1 P1 M2 Y36 H62 S63 I64 V106 P1 M2 Y36 H62 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=7uM remove_due_to_license_issue IC50=7000nM P14174 17526494 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 2op3 A 1.6 BS01 TF5 A 1 G23 C25 W26 N67 G68 G69 N163 H164 G165 G23 C25 W26 N67 G68 G69 N163 H164 G165 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue P25774 17469812 501 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 2op9 A 1.8 BS01 WR1 A 1 H41 M49 L141 N142 G143 S144 C145 M165 E166 R188 H42 M50 L142 N143 G144 S145 C146 M166 E167 R189 H41 G143 C145 H42 G144 C146 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=2200nM P0C6X7 17605471 601 ASGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCS 2op9 B 1.8 BS01 WR1 B 1 H41 M49 G143 S144 C145 M165 E166 D187 R188 H41 M48 G142 S143 C144 M163 E164 D185 R186 H41 G143 C145 H41 G142 C144 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=2200nM P0C6X7 17605471 602 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCS 2opb A 2.8 BS01 F21 A 1 Y35 N39 Y40 R44 V53 F182 E219 Y222 M258 D267 Y12 N16 Y17 R21 V30 F159 E196 Y199 M235 D244 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 remove_due_to_license_issue Ki=1200nM P11086 17845018 4001 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWALRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 2oph A 2.4 BS01 277 A 1 E205 E206 F357 R358 Y631 Y662 Y666 N710 E167 E168 F319 R320 Y593 Y624 Y628 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.016uM remove_due_to_license_issue IC50=16nM P27487 17350841 1001 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2opy A 2.8 BS02 CO9 A 1 L292 G306 L307 T308 E314 Q319 W323 L44 G58 L59 T60 E66 Q71 W75 2.3.2.27 remove_due_to_license_issue P98170 17336535 101 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 2oqi B 2.8 BS01 GGO B 1 E205 E206 R358 S630 Y631 Y662 Y666 V711 E167 E168 R320 S592 Y593 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue Ki=3.2nM P27487 17367123 901 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2oqv A 2.8 BS01 MA9 A 1 E205 E206 V207 S209 F357 R358 Y547 Y631 Y662 Y666 V711 E167 E168 V169 S171 F319 R320 Y509 Y593 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue Ki=4.0nM P27487 17367123 901 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 2or4 A 1.62 BS04 QUS A 1 R210 N257 E424 G427 L428 G518 Y552 K699 Y700 R152 N199 E366 G369 L370 G460 Y491 K638 Y639 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=9.5uM remove_due_to_license_issue Q04609 17567119 1801 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2ork B 1.89 BS04 IPD B 1 E321 N323 E329 N341 R343 E117 N119 E125 N137 R139 ? ic50=1.4mM remove_due_to_license_issue P35247 17417879 995 ASLRQQVEALQGQVQHLQAAFSQYKKVELFPNGQSVGEKIFKTAGFVKPFTEAQLLCTQAGGQLASPRSAAENAALQQLVVAKNEAAFLSMTDSKTEGKFTYPTGESLVYSNWAPGEPNDDGGSEDCVEIFTNGKWNDRACGEKRLVVCEF 2os9 A 1.7 BS04 INS A 1 E321 N323 E329 N341 R343 E117 N119 E125 N137 R139 ? remove_due_to_license_issue P35247 17417879 631 ASLRQQVEALQGQVQHLQAAFSQYKKVELFPNGQSVGEKIFKTAGFVKPFTEAQLLCTQAGGQLASPRSAAENAALQQLVVAKNEAAFLSMTDSKTEGKFTYPTGESLVYSNWAPGEPNDDGGSEDCVEIFTNGKWNDRACGEKRLVVCEF 2osc A 2.8 BS01 MUH A 1 E872 L876 L879 I902 Y904 A905 F960 H962 A981 D982 F983 E26 L30 L33 I52 Y54 A55 F110 H112 A131 D132 F133 D964 A966 R968 N969 D982 R999 D114 A116 R118 N119 D132 R138 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=17nM Q02763 17350837 50 QVLKARIMDAAIKRMKKDDHRDFAGELEVLCKLGHHPNIINLLGACEHYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLMGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGI 2osf A 1.6 BS02 TH0 A 1 H94 L197 T198 H91 L194 T195 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=148uM remove_due_to_license_issue P00918 18266323 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2osm A 1.6 BS02 HTS A 1 H94 V121 L197 T198 H92 V119 L195 T196 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.05uM remove_due_to_license_issue P00918 18266323 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2ot1 A 2.05 BS01 N3P A 1 R42 R303 Q306 R42 R303 Q306 D33 K146 E187 E189 K229 S300 Y363 D33 K146 E187 E189 K229 S300 Y349 4.1.2.13 0004332,0005515,0005737,0006096,0016829,0030335,0031430,0031674,0034316,0051289 Ki~0.1mM remove_due_to_license_issue P00883 17329259 3001 PHSHPALTPEQKKELSDIAHRIVAPGKGILAADESTGSIAKRLQSIGTENTEENRRFYRQLLLTADDRVNPCIGGVILFHETLYQKADDGRPFPQVIKSKGGVVGIKVDKGVVPLAGTNGETTTQGLDGLSERCAQYKKDGADFAKWRCVLKIGEHTPSALAIMENANVLARYASICQQNGIVPIVEPEILPDGDHDLKRCQYVTEKVLAAVYKALSDHHIYLEGTLLKPNMVTPGHACTQKYSHEEIAMATVTALRRTVPPAVTGVTFLSGGQSEEEASINLNAINKCPLLKPWALTFSYGRALQASALKAWGGKKENLKAAQEEYVKRALANSLACQGKYTPSNHAY 2otj 1 2.9 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 17321546 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 2otj 2 2.9 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R35 N36 H37 R40 H41 W42 R43 N45 T47 E49 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R32 N33 H34 R37 H38 W39 R40 N42 T44 E46 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 17321546 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 2otj 3 2.9 BS01 rna 0 0 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 S27 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 D66 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 S27 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 D66 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 17321546 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 2otj A 2.9 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 F201 G203 G204 G205 R206 Q207 H208 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 F201 G203 G204 G205 R206 Q207 H208 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 17321546 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 2otj B 2.9 BS01 rna 0 0 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 Q94 R95 P96 L97 E99 W101 R111 T112 L113 D114 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 S300 V301 P302 G303 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 Q94 R95 P96 L97 E99 W101 R111 T112 L113 D114 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 S300 V301 P302 G303 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 17321546 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 2otj C 2.9 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 P71 L73 D74 R76 A77 R78 V80 P81 Q82 V84 K85 R87 H90 P92 K93 E95 K96 L100 D101 N103 D104 K105 E106 R107 R127 V148 K149 T150 Q151 R168 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 P189 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 P71 L73 D74 R76 A77 R78 V80 P81 Q82 V84 K85 R87 H90 P92 K93 E95 K96 L100 D101 N103 D104 K105 E106 R107 R127 V148 K149 T150 Q151 R168 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 P189 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 17321546 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKLDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 2otj D 2.9 BS01 rna 0 0 K20 V22 H24 I27 T52 R56 E60 K72 Q97 D99 D100 T101 S105 F106 G107 D129 T131 N133 Y139 R156 K11 V13 H15 I18 T38 R42 E46 K58 Q83 D85 D86 T87 S91 F92 G93 D95 T97 N99 Y105 R122 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 17321546 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 2otj D 2.9 BS02 rna 9 0 E12 M13 Q47 M48 P49 V50 V73 T74 R76 P137 G138 R140 V141 R144 D145 R149 P152 H155 E3 M4 Q33 M34 P35 V36 V59 T60 R62 P103 G104 R106 V107 R110 D111 R115 P118 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 17321546 3001 ~ 3122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 2otj E 2.9 BS01 rna 0 0 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 G142 Q143 A146 R153 N155 K157 D158 R160 V161 F162 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 G142 Q143 A146 R153 N155 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 17321546 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 2otj F 2.9 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 17321546 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 2otj H 2.9 BS01 rna 0 0 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 K36 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M113 R114 A115 A116 F117 R151 R152 Y154 N155 K156 I157 T158 S160 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 K36 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M102 R103 A104 A105 F106 R140 R141 Y143 N144 K145 I146 T147 S149 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 17321546 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIDSSPAGNA 2otj I 2.9 BS01 rna 0 0 P74 T75 K80 T87 E91 P92 K112 D115 L116 L117 S118 Y119 N123 K126 E127 G130 T131 S134 L135 P4 T5 K10 T17 E21 P22 K42 D45 L46 L47 S48 Y49 N53 K56 E57 G60 T61 S64 L65 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 17321546 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 2otj J 2.9 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 G48 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 K80 T82 R84 G85 M86 P88 K90 K91 R95 E99 R102 V103 I127 K128 G140 I15 G17 R18 S21 L28 T44 G45 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 K77 T79 R81 G82 M83 P85 K87 K88 R92 E96 R99 V100 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 17321546 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 2otj K 2.9 BS01 rna 0 0 M1 A3 D7 T9 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 L44 T54 S56 R66 R77 K78 R81 R87 M1 A3 D7 T9 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 L44 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 17321546 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRLPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 2otj L 2.9 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G15 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 G34 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 T63 D65 R67 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G15 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 G34 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 T63 D65 R67 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 17321546 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 2otj M 2.9 BS01 rna 0 0 A1 S3 Y5 R9 E13 P15 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 H77 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 P110 N111 N116 G124 R125 K127 D135 N137 H138 P139 A140 D146 W149 D157 F160 R161 L163 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 S189 G191 G192 K193 A194 A1 S3 Y5 R9 E13 P15 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 H77 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 P110 N111 N116 G124 R125 K127 D135 N137 H138 P139 A140 D146 W149 D157 F160 R161 L163 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 S189 G191 G192 K193 A194 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 17321546 10 ~ 2914 ARSAYSYIRDAWENPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKA 2otj N 2.9 BS01 rna 0 0 P4 R5 Y6 K7 R13 A16 T18 H21 R25 L26 K28 S29 V101 L106 P109 F116 P130 N132 P4 R5 Y6 K7 R13 A16 T18 H21 R25 L26 K28 S29 V101 L106 P109 F116 P130 N132 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 17321546 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 2otj N 2.9 BS02 rna 9 0 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 17321546 3001 ~ 3122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 2otj O 2.9 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 V111 R112 V113 I114 R115 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 V111 R112 V113 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 17321546 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 2otj P 2.9 BS01 rna 0 0 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 17321546 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 2otj Q 2.9 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 17321546 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 2otj Q 2.9 BS02 rna 9 0 R19 P25 Q27 R19 P25 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 17321546 3001 ~ 3122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 2otj R 2.9 BS01 rna 0 0 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 V66 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 V66 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 17321546 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 2otj S 2.9 BS01 rna 0 0 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 R67 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 R67 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 17321546 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 2otj T 2.9 BS01 rna 0 0 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 D83 V87 R89 S94 N95 R97 D105 K107 R111 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 D83 V87 R89 S94 N95 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 17321546 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 2otj U 2.9 BS01 rna 0 0 S34 K35 N38 L42 R44 E50 W51 R56 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 17321546 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 2otj V 2.9 BS01 rna 0 0 T1 H4 E7 R9 Q34 P43 G44 K47 R50 K51 A54 R55 K57 T58 E62 T1 H4 E7 R9 Q34 P43 G44 K47 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 17321546 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 2otj W 2.9 BS01 rna 0 0 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 17321546 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 2otj W 2.9 BS02 rna 9 0 R8 H14 N49 D50 K129 H130 P131 K133 E134 R8 H14 N49 D50 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 17321546 3001 ~ 3122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 2otj X 2.9 BS01 rna 0 0 T11 P13 R15 R18 A19 P21 N22 H23 D27 K28 M30 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 S68 T5 P7 R9 R12 A13 P15 N16 H17 D21 K22 M24 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 17321546 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 2otj Y 2.9 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 N230 P231 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 N136 P137 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 17321546 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 2otj Z 2.9 BS01 rna 0 0 R10 G12 R13 G15 A16 R17 Y18 G19 R20 V21 R23 R46 R49 T52 Y59 R1 G3 R4 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 T43 Y50 ? 0003735,0005840,0006412 remove_due_to_license_issue P60619 17321546 10 ~ 2914 RSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 2ou7 A 2.4 BS03 ANP A 1 G62 A80 K82 C133 F183 D194 G196 L197 G26 A44 K46 C97 F147 D158 G160 L161 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=155uM remove_due_to_license_issue P53350 17461553 500 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 2ov4 A 2.5 BS01 AQP A 1 I8 Q9 S11 G17 N18 G21 V143 G144 D146 Q147 A181 I183 K192 M193 S194 K195 S196 I8 Q9 S11 G17 N18 G21 V143 G144 D146 Q147 A181 I183 K192 M193 S194 K195 S196 K111 K192 K195 K111 K192 K195 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0005829,0006412,0006418,0006436 Kd=18uM remove_due_to_license_issue P00953 17428498 400 MKTIFSGIQPSGVITIGNYIGALRQFVELQHEYNCYFCIVDQHAITVWQDPHELRQNIRRLAALYLAVGIDPTQATLFIQSEVPAHAQAAWMLQCIVYIGELERMTQFKEKSAGKEAVSAGLLTYPPLMAADILLYNTDIVPVGEDQKQHIELTRDLAERFNKRYGELFTIPEARIPKVGARIMSLVDPTKKMSKSDPNPKAYITLLDDAKTIEKKIKSAVTDSEGTIRYDKEAKPGISNLLNIYSTLSGQSIEELERQYEGKGYGVFKADLAQVVIETLRPIQERYHHWMESEELDRVLDEGAEKANRVASEMVRKMEQAMGLGRRR 2ovv A 2.0 BS02 PFH A 1 F629 L665 F686 Q716 G718 F719 V723 F176 L212 F233 Q263 G265 F266 V270 3.1.4.17 0004114,0007165,0008081 Ki=12nM remove_due_to_license_issue Ki=12nM Q9QYJ6 17228859 999 LPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 2ovx A 2.0 BS08 4MR A 1 L188 A189 H401 Q402 H405 H411 L418 Y420 P421 M422 Y423 L79 A80 H117 Q118 H121 H127 L134 Y136 P137 M138 Y139 H401 Q402 H405 H411 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P14780 17599356 501 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLY 2ovy A 1.8 BS02 PFJ A 1 F629 L665 F686 M703 Q716 G718 F719 A722 V723 F177 L213 F234 M251 Q264 G266 F267 A270 V271 3.1.4.17 0004114,0007165,0008081 Ki=4nM remove_due_to_license_issue Ki=4nM Q9QYJ6 17228859 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 2ovz A 2.0 BS08 5MR A 1 F110 G186 L187 L188 H190 V398 H401 Q402 H405 H411 L418 Y420 M422 Y423 F1 G77 L78 L79 H81 V114 H117 Q118 H121 H127 L134 Y136 M138 Y139 H401 Q402 H405 H411 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P14780 17599356 501 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLY 2ow0 A 2.0 BS07 6MR A 1 E111 L188 A189 H401 Q402 H405 H411 L418 Y420 P421 M422 Y423 E2 L79 A80 H117 Q118 H121 H127 L134 Y136 P137 M138 Y139 H401 Q402 H405 H411 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P14780 17599356 501 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLY 2ow1 A 2.2 BS07 7MR A 1 L188 A189 H401 Q402 H405 H411 L418 P421 M422 Y423 R424 L79 A80 H117 Q118 H121 H127 L134 P137 M138 Y139 R140 H401 Q402 H405 H411 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P14780 17599356 501 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLY 2ow2 A 2.9 BS06 8MR A 1 L188 A189 H401 Q402 H411 P421 Y423 L76 A77 H114 Q115 H124 P134 Y136 H401 Q402 H405 H411 H114 Q115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P14780 17599356 501 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLY 2ow3 A 2.8 BS01 BIM A 1 I62 F67 Y134 V135 P136 T138 Q185 L188 C199 D200 I28 F33 Y96 V97 P98 T100 Q147 L150 C161 D162 D181 K183 N186 D200 S219 D143 K145 N148 D162 S181 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=3.0nM P49841 17350261 387 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQ 2ow6 A 1.19 BS02 NK1 A 1 D92 W95 D204 R228 H471 D472 Y727 R876 D63 W66 D175 R199 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=2mM remove_due_to_license_issue Q24451 18076078 4001 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 2ow7 A 1.77 BS02 NK2 A 1 D92 W95 D204 F206 H471 D472 Y727 R876 D63 W66 D175 F177 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=14uM remove_due_to_license_issue Q24451 18076078 6001 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 2ow9 A 1.74 BS06 SP6 A 1 L197 H201 A217 L218 F220 I222 Y223 T224 Y225 T226 K228 H230 F231 M232 L115 H119 A135 L136 F138 I140 Y141 T142 Y143 T144 K146 H148 F149 M150 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=30nM remove_due_to_license_issue IC50=30nM, Ki=64nM P45452 17623656 501 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGD 2owb A 2.1 BS02 626 A 1 L59 G62 A65 K66 C67 A80 K82 E131 C133 R136 F183 L23 G26 A29 K30 C31 A44 K46 E95 C97 R100 F147 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=0.44uM remove_due_to_license_issue P53350 17461553 500 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAPS 2oxd A 2.3 BS01 K32 A 1 V53 I66 F113 V116 M163 I174 V47 I60 F107 V110 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue P28523 17768728 338 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 2oxn A 1.7 BS01 OAN A 1 I30 D62 R130 K160 H161 M204 M246 I30 D62 R130 K160 H161 M204 M246 3.2.1.52 0004553,0004563,0005737,0005975,0008360,0009252,0009254,0016231,0016798,0046677,0051301,0071555 Ki=0.036uM remove_due_to_license_issue Q9KU37 17439950 501 MGPLWLDVAGYELSAEDREILQHPTVGGVILFGRNYHDNQQLLALNKAIRQAAKRPILIGVDQEGGRVQRFREGFSRIPPAQYYARAENGVELAEQGGWLMAAELIAHDVDLSFAPVLDMGFACKAIGNRAFGEDVQTVLKHSSAFLRGMKAVGMATTGKHFPGHGAVIADSHLETPYDERETIAQDMAIFRAQIEAGVLDAMMPAHVVYPHYDAQPASGSSYWLKQVLREELGFKGIVFSDDLSMEGAAVMGGPVERSHQALVAGCDMILICNKREAAVEVLDNLPIMEVPQAEALLKKQQFSYSELKRLERWQQASANMQRLIEQFSEHHH 2oxx A 2.3 BS01 K22 A 1 V45 V53 I66 V116 M163 I174 V39 V47 I60 V110 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue P28523 17768728 501 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 2oxy A 1.812 BS01 K17 A 1 V53 I66 V95 F113 V116 M163 I174 V47 I60 V89 F107 V110 M157 I168 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue P28523 17768728 1001 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2oyk A 1.5 BS01 9MR A 1 K66 H135 D137 W178 E233 Y306 E351 W382 K24 H93 D95 W127 E182 Y255 E295 W326 3.2.1.123 0000272,0004553,0005975,0016042,0016798,0047876,1901136 Ki=5uM remove_due_to_license_issue O33853 17487923 600 PSYLKDDDGRSLILRGFNTASSAKSAPDGMPQFTEADLAREYADMGTNFVRFLISWRSVEPAPGVYDQQYLDRVEDRVGWYAERGYKVMLDMHQDVYSGAITPAIGNGAPAWATYMDGLPVEPQPRWELYYIQPGVMRAFDNFWNTTGKHPELVEHYAKAWRAVADRFADNDAVVAYDLMNEPFGGSLQGPAFEAGPLAAMYQRTTDAIRQVDQDTWVCVAPQAIGVNQGLPSGLTKIDDPRAGQQRIAYCPHLYPLPLHEGLARTLTDVTIDAWRANTAHTARVLGDVPIILGEFGLDTTLPGARDYIERVYGTAREMGAGVSYWSSDPGPWGPYLPDGTQTLLVDTLNKPYPRAVAGTPTEWSSTSDRLQLTIEPDAAITAPTEIYLPEAGFPGDVHVEGADVVGWDRQSRLLTVRTPADSGNVTVTVTPAA 2oyl A 1.8 BS01 IDC A 1 K66 H135 D137 W178 N232 E233 Y306 E351 W382 K24 H93 D95 W127 N181 E182 Y255 E295 W326 3.2.1.123 0000272,0004553,0005975,0016042,0016798,0047876,1901136 Ki=0.5uM remove_due_to_license_issue O33853 17487923 600 PSYLKDDDGRSLILRGFNTASSAKSAPDGMPQFTEADLAREYADMGTNFVRFLISWRSVEPAPGVYDQQYLDRVEDRVGWYAERGYKVMLDMHQDVYSGAITPAIGNGAPAWATYMDGLPVEPQPRWELYYIQPGVMRAFDNFWNTTGKHPELVEHYAKAWRAVADRFADNDAVVAYDLMNEPFGGSLQGPAFEAGPLAAMYQRTTDAIRQVDQDTWVCVAPQAIGVNQGLPSGLTKIDDPRAGQQRIAYCPHLYPLPLHEGLARTLTDVTIDAWRANTAHTARVLGDVPIILGEFGLDTTLPGARDYIERVYGTAREMGAGVSYWSSDPGPWGPYLPDGTQTLLVDTLNKPYPRAVAGTPTEWSSTSDRLQLTIEPDAAITAPTEIYLPEAGFPGDVHVEGADVVGWDRQSRLLTVRTPADSGNVTVTVTPAA 2oym A 1.86 BS01 MNI A 1 H135 D137 Y182 N232 E233 F235 Y306 E351 W382 H93 D95 Y130 N180 E181 F183 Y254 E295 W326 3.2.1.123 0000272,0004553,0005975,0016042,0016798,0047876,1901136 Ki=10uM remove_due_to_license_issue O33853 17487923 600 PSYLKDDDGRSLILRGFNTASSAKSAPDGMPQFTEADLAREYADMGTNFVRFLISWRSVEPAPGVYDQQYLDRVEDRVGWYAERGYKVMLDMHQDVYSGAITAIGNGAPAWATYMDGLPVEPQPRWELYYIQPGVMRAFDNFWNTTGKHPELVEHYAKAWRAVADRFADNDAVVAYDLMNEPFGGSLQGPAFEAGPLAAMYQRTTDAIRQVDQDTWVCVAPQAIGVNQGLPSGLTKIDDPRAGQQRIAYCPHLYPLPLDHEGLARTLTDVTIDAWRANTAHTARVLGDVPIILGEFGLDTTLPGARDYIERVYGTAREMGAGVSYWSSDPGPWGPYLPDGTQTLLVDTLNKPYPRAVAGTPTEWSSTSDRLQLTIEPDAAITAPTEIYLPEAGFPGDVHVEGADVVGWDRQSRLLTVRTPADSGNVTVTVTPAA 2oz2 A 1.95 BS01 D1R A 1 Q19 G23 C25 S64 G65 G66 L67 A138 A141 M145 D161 H162 W184 E208 Q19 G23 C25 S64 G65 G66 L67 A138 A141 M145 D161 H162 W184 E208 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 19620707 301 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 2oz2 C 1.95 BS01 D1R C 1 Q19 G23 C25 S64 G65 G66 L67 A138 M145 D161 H162 W184 Q19 G23 C25 S64 G65 G66 L67 A138 M145 D161 H162 W184 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 19620707 300 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 2oz5 A 2.0 BS01 7XY A 1 R59 E60 P81 H94 F98 Y125 E129 F133 C160 F161 A162 K164 D165 R166 R56 E57 P78 H90 F94 Y114 E118 F122 C149 F150 A151 K153 D154 R155 ? 0004438,0004721,0004722,0004725,0005576,0016311,0016791,0034594,0051701 Ki=0.33uM remove_due_to_license_issue IC50=440nM P96830 17437721 277 RELPGAWNFRDVADTATALRPGRLFRSSELSRLDDAGRATLRRLGITDVADLRSSREVARRGPGRVPDGIDVHLLPFPDLADDADDSAPHETAFKRLLTNGESSQSINDAATRYMTDEYRQFPTRNGAQRALHRVVTLLAAGRPVLTHCFAGKDRTGFVVALVLEAVGLDRDVIVADYLRSNDSVPQLRARISEMIQQRFDTELAPEVVTFTKARLSDGVLGVRAEYLAAARQTIDETYGSLGGYLRDAGISQATVNRMRGVLLG 2oz5 A 2.0 BS02 7XY A 2 E60 R63 F98 F161 M206 R210 F211 L227 E57 R60 F94 F150 M195 R199 F200 L216 ? 0004438,0004721,0004722,0004725,0005576,0016311,0016791,0034594,0051701 Ki=0.33uM remove_due_to_license_issue IC50=440nM P96830 17437721 278 RELPGAWNFRDVADTATALRPGRLFRSSELSRLDDAGRATLRRLGITDVADLRSSREVARRGPGRVPDGIDVHLLPFPDLADDADDSAPHETAFKRLLTNGESSQSINDAATRYMTDEYRQFPTRNGAQRALHRVVTLLAAGRPVLTHCFAGKDRTGFVVALVLEAVGLDRDVIVADYLRSNDSVPQLRARISEMIQQRFDTELAPEVVTFTKARLSDGVLGVRAEYLAAARQTIDETYGSLGGYLRDAGISQATVNRMRGVLLG 2oz6 A 2.8 BS01 CMP A 1 R59 E60 Q175 G178 R179 G182 C183 S184 R185 R52 E53 Q163 G166 R167 G170 C171 S172 R173 ? 0000976,0001216,0001217,0003677,0003700,0005829,0006351,0006355,0030552,0032993,0043565,0045892,0045893 Kd=1.0uM (21665969) remove_due_to_license_issue P55222 21665969 302 MKLKHLDKLLAHCHRRRYTAKSTIIYAGDRCETLFFIIKGSVTILIEDDDGREMIIGYLNSGDFFGELGLFEQERSAWVRAKVECEVAEISYAKFRELSQQDSEILYTLGSQMADRLRKTTRKVGDLAFLDVTGRVARTLLDLCQQPDAMTHPDGMQIKITRQEIGRIVGCSREMVGRVLKSLEEQGLVHVKGKTMVVFGT 2oz6 A 2.8 BS02 CMP A 2 I51 I63 F72 G73 E74 L75 R87 S88 A89 V91 R128 T132 I44 I56 F65 G66 E67 L68 R75 S76 A77 V79 R116 T120 ? 0000976,0001216,0001217,0003677,0003700,0005829,0006351,0006355,0030552,0032993,0043565,0045892,0045893 Kd=1.0uM (21665969) remove_due_to_license_issue P55222 21665969 301 MKLKHLDKLLAHCHRRRYTAKSTIIYAGDRCETLFFIIKGSVTILIEDDDGREMIIGYLNSGDFFGELGLFEQERSAWVRAKVECEVAEISYAKFRELSQQDSEILYTLGSQMADRLRKTTRKVGDLAFLDVTGRVARTLLDLCQQPDAMTHPDGMQIKITRQEIGRIVGCSREMVGRVLKSLEEQGLVHVKGKTMVVFGT 2oz7 A 1.8 BS01 CA4 A 1 L704 N705 L707 Q711 M742 F764 M780 F876 A877 L880 F891 L34 N35 L37 Q41 M72 F94 M110 F206 A207 L210 F221 ? remove_due_to_license_issue Ki=14nM, IC50=23nM P10275 17311914 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFAFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ozr A 2.3 BS06 GG1 A 1 L197 H201 L218 F220 I222 Y223 Y225 T226 K228 S229 F231 M232 L115 H119 L136 F138 I140 Y141 Y143 T144 K146 S147 F149 M150 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.67nM remove_due_to_license_issue IC50=0.670000nM P45452 17623656 2001 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGD 2ozr C 2.3 BS06 GG1 C 1 K119 F196 L197 H201 L218 F220 I222 Y223 Y225 T226 S229 F231 K37 F114 L115 H119 L136 F138 I140 Y141 Y143 T144 S147 F149 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.67nM remove_due_to_license_issue IC50=0.670000nM P45452 17623656 2003 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGD 2p09 A 1.65 BS02 ATP A 1 K34 R41 Y43 M45 F50 H62 G63 H64 K30 R37 Y39 M41 F46 H58 G59 H60 Kd=450nM remove_due_to_license_issue 17520026 500 DDDDKKTNWLKRIYRVRPCVKCKVAPRDWKVKNKHLRIYNMCKTCFNNSIDIGDDTYHGHVDWLMYADS 2p0d A 1.811 BS01 I3P A 1 R342 K343 W345 S397 S398 R23 K24 W26 S64 S65 ? remove_due_to_license_issue Q9BRR9 17339315 800 SHEVEKSGLLNMTKIAQGGRKLRKNWGPSWVVLTGNSLVFYREPRPESSVDLRGAALAHGRHLSSRRNVLHIRTIPGHEFLLQSDHETELRAWHRALRTVIERLVRW 2p0x A -1.00 BS02 ATP A 1 D17 R19 K21 R26 Y28 N29 M30 F35 H47 G48 H49 D17 R19 K21 R26 Y28 N29 M30 F35 H47 G48 H49 remove_due_to_license_issue 17583732 1318 GSFRVKPCVVCKVAPRDWRVKNRHLRIYNMCKTCFNNSIKSGDDTYHGHVDWLMYTDAKEFSST 2p15 A 1.94 BS02 EZT A 1 M343 L346 E353 L387 F404 V418 M421 I424 F425 H524 M36 L39 E46 L80 F97 V111 M114 I117 F118 H217 ? remove_due_to_license_issue P03372 17468738 600 SLALSLTADQMVSALLDAEPPILYSEYRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL 2p16 A 2.3 BS02 GG2 A 1 T98 E146 F174 A190 C191 Q192 S195 V213 W215 G216 C220 T84 E135 F162 A180 C181 Q182 S185 V203 W205 G206 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.08nM remove_due_to_license_issue Ki=0.08nM, IC50=210nM P00742 17914785 298 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2p1c A 2.45 BS04 GG3 A 1 Y99 D103 R112 T168 A169 Q172 K212 T213 Y216 D255 K269 Y89 D93 R102 T158 A159 Q162 K202 T203 Y206 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Ki=21nM remove_due_to_license_issue Q86C09 18442135 3001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 2p1c B 2.45 BS04 GG3 B 1 Y99 D103 R112 T168 Q172 K212 Y216 D255 K269 Y89 D93 R102 T158 Q162 K202 Y206 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Ki=21nM remove_due_to_license_issue Q86C09 18442135 8004 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 2p2a B 2.26 BS01 MP9 B 1 S11 Y13 Y58 P86 L87 T88 R93 G138 S139 T140 E190 T192 M193 Y217 S11 Y13 Y58 P86 L87 T88 R93 G138 S139 T140 E190 T192 M193 Y217 ? 0015276,0016020 Ki=0.75uM remove_due_to_license_issue P19491 17455929 802 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYEC 2p2h A 1.95 BS01 994 A 1 V848 A866 K868 E885 T916 F918 C919 G922 L1035 C1045 V30 A48 K50 E67 T98 F100 C101 G104 L167 C177 D1028 A1030 R1032 N1033 D1046 D160 A162 R164 N165 D178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=68nM remove_due_to_license_issue IC50=68nM P35968 17253678 501 EHAERLPYDASKWEFPRDRLKLGKPLGRQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHH 2p2i A 2.4 BS01 608 A 1 L840 A866 K868 E885 I892 V916 C919 C1024 H1026 L1035 C1045 D1046 F1047 L24 A47 K49 E62 I69 V93 C96 C151 H153 L162 C172 D173 F174 D1028 A1030 R1032 N1033 D1046 D155 A157 R159 N160 D173 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=38nM remove_due_to_license_issue IC50=38nM, Ki=10nM P35968 17253678 501 AERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDTCRTVAVKMLTHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLALPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 2p33 A 2.4 BS01 J07 A 1 V78 A91 M146 M149 A151 N152 L206 V34 A47 M102 M105 A107 N108 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 ic50=57nM remove_due_to_license_issue IC50=57nM P53779 17459703 507 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYREHTIEEWKELIYKEVMN 2p3a A 1.75 BS01 3TL A 1 D25 G27 D29 R45 M46 I47 G48 I50 P81 I84 D25 G27 D29 R45 M46 I47 G48 I50 P81 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=11nM remove_due_to_license_issue Q6BB74 17467738 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMALPGKWKPRMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANIIGRNLMTQIGCTLNF 2p3a B 1.75 BS01 3TL A 1 D25 G27 A28 D29 V32 I47 G48 G49 I50 P81 I84 D25 G27 A28 D29 V32 I47 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q6BB74 17467738 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMALPGKWKPRMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANIIGRNLMTQIGCTLNF 2p3b A 2.1 BS01 3TL A 1 D25 G27 A28 D29 G48 P81 D25 G27 A28 D29 G48 P81 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=3.3nM remove_due_to_license_issue Q9Q2G8 17467738 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2p3b B 2.1 BS01 3TL A 1 D25 G27 I47 G48 G49 I50 V82 D25 G27 I47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q9Q288 17467738 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2p3c A 2.1 BS01 3TL A 1 D25 G27 A28 D29 K45 I47 G48 P81 D25 G27 A28 D29 K45 I47 G48 P81 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=24nM remove_due_to_license_issue Q6Q004 17467738 201 PQITLWKRPLVTIKVGGQLKEALLDTGADDTVLEDIALPGKWKPKMIGGIGGFIKVKQYENVSLEICGHKAIGTVLVGPTPVNIIGRNMLTQIGCTLNF 2p3c B 2.1 BS01 3TL A 1 D25 G27 A28 D29 M46 I47 G48 G49 I50 V82 I84 D25 G27 A28 D29 M46 I47 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q6Q004 17467738 201 PQITLWKRPLVTIKVGGQLKEALLDTGADDTVLEDIALPGKWKPKMIGGIGGFIKVKQYENVSLEICGHKAIGTVLVGPTPVNIIGRNMLTQIGCTLNF 2p3d A 2.8 BS01 3TL A 1 D25 G27 A28 D29 I47 G48 G49 I50 F53 P81 I84 D25 G27 A28 D29 I47 G48 G49 I50 F53 P81 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q7SRY5 17467738 201 PQITLWKRPIVTIKVEGQLREALLDTGADDTVLEDINLSGKWKPKIIGGIRGFVKVKQYEDILIEICGHRAVGAVLVGPTPANIIGRNMLTQIGCTLNF 2p3d B 2.8 BS01 3TL A 1 D25 G27 A28 D29 I46 G48 G49 I50 P81 I84 D25 G27 A28 D29 I46 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q7SRY5 17467738 201 PQITLWKRPIVTIKVEGQLREALLDTGADDTVLEDINLSGKWKPKIIGGIRGFVKVKQYEDILIEICGHRAVGAVLVGPTPANIIGRNMLTQIGCTLNF 2p3g X 3.8 BS01 F10 X 1 L70 A91 K93 E139 C140 L141 T206 D207 L26 A47 K49 E95 C96 L97 T162 D163 N191 D207 N147 D163 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue EC50=372nM, IC50=8900nM P49137 17480064 401 QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSKYDKSCDMWSLGVIMYILLCGYPPFYSGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR 2p3i A 1.75 BS01 MNA A 1 R101 Y155 Y188 Y189 S190 R38 Y92 Y125 Y126 S127 ? 0019028,0019058 Kd=0.33mM remove_due_to_license_issue P12473 18974199 1000 VLDGPYQPTTFNPPVDYWMLLAPTAAGVVVEGTNNTDRWLATILVEPNVTSETRSYTLFGTQEQITIANASQTQWKFIDVVKTTQNGSYSQYGPLQSTPKLYAVMKHNGKIYTYNGETPNVTTKYYSTTNYDSVNMTAFCDFYIIPREEESTCTEYINNGL 2p3o A 2.756 BS02 GTA A 1 K14 L17 N18 F25 S150 S151 K8 L11 N12 F19 S144 S145 3.4.21.91,3.6.1.15,3.6.4.13 0003968,0004482,0004483,0005524,0008168,0032259 remove_due_to_license_issue Q9WLZ5 17686489 1012 ETLGEKWKSRLNALGKSEFQIYKKSGIQEVDRTLAKEGIKRGETDHHAVSRGSAKLRWFVERNLVTPEGKVVDLGCGRGGWSYYCGGLKNVREVKGLTKGGPGHEEPIPMSTYGWNLVRLQSGVDVFFIPPERCDTLLCDIGESSPNPTVEAGRTLRVLNLVENWLSNNTQFCVKVLNPYMSSVIEKMEALQRKHGGALVRNPLSRNSTHEMYWVSNASGNIVSSVNMISRMLINRFTMRHKKATYEPDVDLGSGTRN 2p4i A 2.5 BS01 MR9 A 1 V838 A853 E872 L879 I886 I902 Y904 A905 L971 I980 A981 D982 F983 V1 A11 E16 L23 I30 I42 Y44 A45 L111 I120 A121 D122 F123 D964 A966 R968 N969 D982 R999 D104 A106 R108 N109 D122 R134 2.7.10.1 0004672,0004713,0005524,0006468 ic50=10nM remove_due_to_license_issue IC50=10nM Q02763 17253678 301 VLKARIRMDAAIKRGELEVLCKLGHHPNIINLLGACEHYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLSRVKKTMGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGID 2p4j A 2.5 BS01 23I A 1 Q12 G13 D32 G34 P70 Y71 T72 Q73 I126 Y198 D228 S229 G230 T232 N233 R235 A335 Q16 G17 D36 G38 P74 Y75 T76 Q77 I130 Y202 D232 S233 G234 T236 N237 R239 A339 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=1.1nM remove_due_to_license_issue Ki=1.1nM P56817 17432843 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2p4s A 2.2 BS02 DIH A 1 Y173 A201 A202 G203 F285 E286 I302 G303 M304 N328 H342 Y84 A112 A113 G114 F196 E197 I213 G214 M215 N239 H253 S118 H149 H171 Y173 E174 A201 M304 S305 N328 C330 H342 S29 H60 H82 Y84 E85 A112 M215 S216 N239 C241 H253 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757 Ki=0.31nM remove_due_to_license_issue A4Q998 17918964 401 YTYDTLQEIATYLLERTELRPKVGIICGSGLGTLAEQLTDVDSFDYETIPHFPVSTVAGHVGRLVFGYLAGVPVMCMQGRFHHYEGYPLAKCAMPVRVMHLIGCTHLIATNAAGGANPKYRVGDIMLIKDHINLMGFAGNNPLQGPNDERFGPRFFGMANTYDPKLNQQAKVIARQIGIENELREGVYTCLGGPNFETVAEVKMLSMLGVDAIGMSTVHEIITARHCGMTCFAFSLITNMCTMSYEEEEEHCHDSIVGVGKNREKTLGEFVSRIVKHIHYEA 2p4s C 2.2 BS02 DIH C 1 Y173 A201 A202 G203 F285 E286 I302 M304 N328 H342 Y84 A112 A113 G114 F196 E197 I213 M215 N239 H253 S118 H149 H171 Y173 E174 A201 M304 S305 N328 C330 H342 S29 H60 H82 Y84 E85 A112 M215 S216 N239 C241 H253 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757 Ki=0.31nM remove_due_to_license_issue A4Q998 17918964 402 YTYDTLQEIATYLLERTELRPKVGIICGSGLGTLAEQLTDVDSFDYETIPHFPVSTVAGHVGRLVFGYLAGVPVMCMQGRFHHYEGYPLAKCAMPVRVMHLIGCTHLIATNAAGGANPKYRVGDIMLIKDHINLMGFAGNNPLQGPNDERFGPRFFGMANTYDPKLNQQAKVIARQIGIENELREGVYTCLGGPNFETVAEVKMLSMLGVDAIGMSTVHEIITARHCGMTCFAFSLITNMCTMSYEEEEEHCHDSIVGVGKNREKTLGEFVSRIVKHIHYEA 2p4y A 2.25 BS01 C03 A 1 F226 C285 R288 S289 A292 I296 M329 L330 I341 S342 L353 F363 M364 F22 C52 R55 S56 A59 I63 M96 L97 I108 S109 L120 F130 M131 ? 0003677,0004879,0005634,0006355 Ki=0.001uM remove_due_to_license_issue P37231 17940191 478 NPESADLRALAKHLYDSYIKSFPLTKAKARAILTKSPFVIYDMNSIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 2p53 A 2.1 BS02 NNG A 1 N61 E131 G141 T142 H143 H195 H216 N219 A220 H251 N273 F287 L306 G308 N61 E131 G141 T142 H143 H195 H216 N219 A220 H251 N273 F287 L306 G308 3.5.1.25 0006040,0006044,0006046,0008270,0008448,0016787,0016810,0019262,0032991,0042802,0046872,0051289 remove_due_to_license_issue P0AF18 17567048 411 MYALTQGRIFTGHEFLDDHAVVIADGLIKSVCPVAELPPEIEQRSLNGAILSPGFIDVQLNGCGGVQFNDTAEAVSVETLEIMQKANEKSGCTNYLPTLITTSDELMKQGVRVMREYLAKHPNQALGLHLEGPWLNLVKKGTHNPNFVRKPDAALVDFLCENADVITKVTLAPEMVPAEVISKLANAGIVVSAGHSNATLKEAKAGFRAGITFATHLYNAMPYITGREPGLAGAILDEADIYCGIIADGLHVDYANIRNAKRLKGDKLCLVTNATAPAGANIEQFIFAGKTIYYRNGLCVDENGTLSGSSLTMIEGVRNLVEHCGIALDEVLRMATLYPARAIGVEKRLGTLAAGKVANLTAFTPDFKITKTIVNGNEVVTQ 2p53 B 2.1 BS02 NNG B 1 N61 E131 G141 T142 H143 H195 H216 N219 A220 H251 N273 F287 L306 G308 N61 E131 G141 T142 H143 H195 H216 N219 A220 H251 N273 F287 L306 G308 3.5.1.25 0006040,0006044,0006046,0008270,0008448,0016787,0016810,0019262,0032991,0042802,0046872,0051289 remove_due_to_license_issue P0AF18 17567048 411 MYALTQGRIFTGHEFLDDHAVVIADGLIKSVCPVAELPPEIEQRSLNGAILSPGFIDVQLNGCGGVQFNDTAEAVSVETLEIMQKANEKSGCTNYLPTLITTSDELMKQGVRVMREYLAKHPNQALGLHLEGPWLNLVKKGTHNPNFVRKPDAALVDFLCENADVITKVTLAPEMVPAEVISKLANAGIVVSAGHSNATLKEAKAGFRAGITFATHLYNAMPYITGREPGLAGAILDEADIYCGIIADGLHVDYANIRNAKRLKGDKLCLVTNATAPAGANIEQFIFAGKTIYYRNGLCVDENGTLSGSSLTMIEGVRNLVEHCGIALDEVLRMATLYPARAIGVEKRLGTLAAGKVANLTAFTPDFKITKTIVNGNEVVTQ 2p59 B 2.9 BS03 GG4 B 1 Q1067 H1083 K1162 G1163 S1165 F1180 R1181 A1182 A1183 V1184 C1185 D1194 Q41 H57 K136 G137 S139 F154 R155 A156 A157 V158 C159 D168 H1083 D1107 G1163 S1165 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036,0097264 remove_due_to_license_issue Q91RS4 17482818 1208 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2p7a A 2.3 BS01 43M A 1 E275 L309 V313 Y326 F435 E42 L76 V80 Y93 F202 ? Kd=0.788uM remove_due_to_license_issue P62508 17964775 1 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEA 2p7c B -1.00 BS01 dna A 0 N25 T26 N27 Q45 L49 R50 H59 K61 V65 F66 N25 T26 N27 Q45 L49 R50 H59 K61 V65 F66 ? 0003677,0045892 remove_due_to_license_issue P06555 17576674 1 ~ 12 MKKIPQISDAELEVMKVIWKHSSINTNEVIKELSKTSTWSPKTIQTMLLRLIKKGALNHHKEGRVFVYTPNIDESDYIEVKS 2p7c B -1.00 BS02 dna C 0 P5 Q6 A10 E11 K42 T43 T46 M47 R50 L51 K54 K61 R64 P5 Q6 A10 E11 K42 T43 T46 M47 R50 L51 K54 K61 R64 ? 0003677,0045892 remove_due_to_license_issue P06555 17576674 13 ~ 24 MKKIPQISDAELEVMKVIWKHSSINTNEVIKELSKTSTWSPKTIQTMLLRLIKKGALNHHKEGRVFVYTPNIDESDYIEVKS 2p7g A 2.1 BS01 2OH A 1 E275 M306 L309 Y326 N346 I349 F435 E41 M72 L75 Y92 N112 I115 F201 ? Kd=0.297uM remove_due_to_license_issue IC50=13.1nM P62508 17964775 1 NKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEA 2p7z A 2.5 BS01 OHT A 1 C269 A272 D273 E275 L309 F435 I438 C35 A38 D39 E41 L75 F201 I204 ? Kd=0.262uM remove_due_to_license_issue IC50=1350nM, EC50=15nM P62508 17964775 201 NKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLE 2p83 A 2.5 BS01 MR0 A 1 G13 D32 G34 S35 Y71 T72 Q73 F108 W115 Y198 D228 G230 T232 R235 G16 D35 G37 S38 Y74 T75 Q76 F111 W118 Y190 D220 G222 T224 R227 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=11nM remove_due_to_license_issue IC50=11nM P56817 17434734 801 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2p8h A 1.8 BS01 MY9 A 1 G11 Q12 G13 Y14 L30 D32 G34 Y71 T72 Q73 F108 W115 Y198 D228 S229 G230 T232 N233 R235 A335 G17 Q18 G19 Y20 L36 D38 G40 Y77 T78 Q79 F114 W121 Y192 D222 S223 G224 T226 N227 R229 A329 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=71nM remove_due_to_license_issue P56817 17458843 386 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2p8n A 1.94 BS01 ADE A 1 Y80 V81 G121 Y123 I172 R180 Y75 V76 G116 Y118 I167 R175 V81 E177 R180 V76 E172 R175 3.2.2.22 0017148,0030598 Kd=0.7mM remove_due_to_license_issue P02879 17986339 271 YPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPP 2p8o C 1.5 BS02 BVA C 1 S190 C191 M192 G193 S195 W215 G216 S40 C41 M42 G43 S45 W65 G66 M192 G193 D194 S195 G196 M42 G43 D44 S45 G46 3.4.21.1 0004252,0006508 Ki=16uM remove_due_to_license_issue P00766 17469803 300 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 2p8s A 2.2 BS01 417 A 1 E205 E206 S209 Y547 S630 Y662 Y666 N710 V711 E167 E168 S171 Y509 S592 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=21nM remove_due_to_license_issue IC50=21nM P27487 17433672 1001 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2p93 A 1.9 BS01 ME1 A 1 E97 T98 Y99 A190 W215 G216 C220 G226 I227 Y228 E83 T84 Y85 A180 W205 G206 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=1.5nM remove_due_to_license_issue Ki=1.5nM P00742 17588746 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2p94 A 1.8 BS01 ME4 A 1 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G218 G226 Y228 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.67nM remove_due_to_license_issue Ki=0.67nM P00742 17588746 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2p95 A 2.2 BS01 ME5 A 1 E97 T98 Y99 F174 A190 Q192 V213 W215 G216 G218 C220 Y228 E83 T84 Y85 F162 A180 Q182 V203 W205 G206 G208 C209 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.43nM remove_due_to_license_issue Ki=0.43nM P00742 17588746 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2p98 A 1.7 BS02 YE7 A 1 Y62 Y65 D97 D108 F177 H178 W221 E235 Y61 Y64 D96 D107 F176 H177 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.64uM remove_due_to_license_issue IC50=2440nM P0AE18 17948983 266 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 2p99 A 1.8 BS02 YE6 A 1 Y62 Y65 H79 D97 D108 F177 H178 E204 W221 E235 Y61 Y64 H78 D96 D107 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=1.16uM remove_due_to_license_issue IC50=77100nM P0AE18 17948983 265 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISH 2p9a A 1.6 BS03 YE6 A 1 C59 Y62 H63 C70 H79 H178 W221 C58 Y61 H62 C69 H78 H177 W220 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=6.56uM remove_due_to_license_issue IC50=77100nM P0AE18 17948983 267 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 2pax A 2.4 BS01 4AN A 1 H862 G863 Y896 F897 A898 K903 S904 Y907 E988 H201 G202 Y235 F236 A237 K242 S243 Y246 E327 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 ic50=0.18uM remove_due_to_license_issue P26446 9521710 1 KSKLAKPIQDLIKMIFDVESMKKAMVEFEIDLQKMPLGKLSKRQIQSAYSILNEVQQAVSDGGSESQILDLSNRFYTLIPHDFGMKKPPLLSNLEYIQAKVQMLDNLLDIEVAYSLLRGGNEDGDKDPIDINYEKLRTDIKVVDKDSEEAKIIKQYVKNTHAATHNAYDLKVVEIFRIEREGESQRYKPFKQLHNRQLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQADPIGLILLGEVALGNMYELKNASHITKLPKGKHSVKGLGKTAPDPTATTTLDGVEVPLGNGISTGINDTCLLYNEYIVYDVAQVNLKYLLKLKFNYKT 2pbw A 2.5 BS01 DOQ A 1 E13 K60 Y61 P88 T90 R95 D139 G140 S141 T142 E190 E10 K57 Y58 P85 T87 R92 D136 G137 S138 T139 E187 ? 0015276,0016020 Ki=5.56nM remove_due_to_license_issue P22756 17581823 401 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWW 2pcp A 2.2 BS01 1PC B 1 Y32 F89 G91 Y96 Y37 F94 G96 Y101 remove_due_to_license_issue 9786848 227 DVLMTQTPLSLPVSLGDQASISCRSSQTIVHSNGNTYLEWYLQKPGQSPKLLIYKVTNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFQGTHAPYTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 2pcp B 2.2 BS01 1PC B 1 Y33 H35 S95 W97 D98 F100 Y33 H35 S99 W101 D102 F104 Kd=2nM remove_due_to_license_issue 9786848 227 EVQLQQSGPELVKPGASVKMSCKASGYTFTDYYIHWNKQSHGKSLEWIGYIYPNNGGNGYNHKFKGKATLTVDKSSSTAYMDVRTLTSEDSAVYYCGRSTWDDFDYWGQGTTLTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSPRPSETVTCNVAHPASSTKVDKKIV 2pe0 A 2.35 BS01 39Z A 1 L88 A109 S160 Y161 A162 G165 L212 L15 A36 S87 Y88 A89 G92 L139 D205 K207 E209 N210 D223 T245 D132 K134 E136 N137 D150 T162 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 17531483 501 PRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2pe1 A 2.14 BS01 517 A 1 L88 A109 K111 Y161 A162 G165 L212 T222 D223 L15 A36 K38 Y88 A89 G92 L139 T149 D150 D205 K207 E209 N210 D223 T245 D132 K134 E136 N137 D150 T162 2.7.11.1 0004672,0004674,0005524,0006468 ic50=6nM remove_due_to_license_issue O15530 17531483 501 PRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2pe2 A 2.13 BS01 464 A 1 L88 A109 K111 S160 Y161 A162 N164 G165 K169 Y170 K173 L212 T222 L15 A36 K38 S87 Y88 A89 N91 G92 K96 Y97 K100 L139 T149 D205 K207 E209 N210 D223 T245 D132 K134 E136 N137 D150 T162 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 17544272 501 PRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2pfy A 1.95 BS01 PCA A 1 R48 W120 Q123 R143 Y145 T165 T182 S183 R48 W120 Q123 R143 Y145 T165 T182 S183 ? 0055085 Kd=0.3uM remove_due_to_license_issue Q7VXB1 17499270 302 ATSWTMTAEQPDANYLTQNARQFADEVKAATAGALEIKVQSNSTLLKRPEVKRGVQQGVVQIGEVLVSALGNEDPLFEIDSVPFLASSFNESEKLWKATRPLLAQRLDKQGIVLVYGSPWPPQGIYTKKPVAALADLKGTRFRAYSASTSHMAALMGAVPTTVQTPEVPQAFSTGVIDAMLTSPATGVDSQAWDYVKYYYDAQAFIPQSFVIANKRAFQRLPAEVRQAVLDAGAKAEIRGWQTARAKTRELTDTLARNGMSVEPLPPQLAKELQAIGATMVSDWSKKAGADGQQLLDAYRK 2pg2 A 1.849 BS02 K01 A 1 E116 E118 R119 W127 A133 I136 P137 Y211 E101 E103 R104 W112 A118 I121 P122 Y196 ? 0003777,0005524,0007018,0008017 ic50=1.7uM remove_due_to_license_issue IC50=1700nM P52732 17498954 604 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2pg2 B 1.849 BS02 K01 B 1 E116 E118 R119 W127 A133 P137 Y211 E101 E103 R104 W112 A118 P122 Y196 ? 0003777,0005524,0007018,0008017 ic50=1.7uM remove_due_to_license_issue IC50=1700nM P52732 17498954 604 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2pgj A 1.71 BS01 N1C A 1 L124 W125 S126 R127 L145 E146 W189 T221 F222 E226 L80 W81 S82 R83 L101 E102 W145 T177 F178 E182 E146 T221 E226 E102 T177 E182 2.4.99.20,3.2.2.-,3.2.2.6 0061809 ic50=0.26mM remove_due_to_license_issue P28907 17591784 301 RWRQTWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFDTSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVEVHNLQPEKVQTLEAWVIHGGREDSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKNPEDSSC 2pgl A 1.76 BS01 N1C A 1 L124 W125 S126 R127 L145 E146 W189 S193 T221 F222 Q226 L80 W81 S82 R83 L101 E102 W145 S149 T177 F178 Q182 E146 T221 Q226 E102 T177 Q182 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue P28907 17591784 301 RWRQTWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFDTSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVQVHNLQPEKVQTLEAWVIHGGREDSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKNPEDSSC 2pgz A 1.76 BS01 COC A 1 Y93 W147 Y188 C190 C191 Y195 Y97 W151 Y192 C194 C195 Y199 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=1.8uM remove_due_to_license_issue Q8WSF8 17481657 401 DDDDKLHSQANLMRLKSDLFNRSYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2pgz B 1.76 BS01 COC A 1 Y55 Q57 I118 Y57 Q59 I120 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 17481657 401 DDDDKLHSQANLMRLKSDLFNYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRF 2ph6 A 2.0 BS01 712 A 1 G11 Q12 G13 L30 D32 G34 Y71 T72 Q73 D228 G230 T231 T232 N233 R235 A335 G15 Q16 G17 L34 D36 G38 Y75 T76 Q77 D219 G221 T222 T223 N224 R226 A321 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=27nM remove_due_to_license_issue IC50=163nM P56817 17482814 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2ph8 A 1.7 BS01 35A A 1 L30 D32 G34 Y71 T72 Q73 D228 G230 T231 T232 N233 R235 L34 D36 G38 Y75 T76 Q77 D218 G220 T221 T222 N223 R225 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=1800nM remove_due_to_license_issue P56817 17827011 388 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACFRTAAVEGPFVTLDMEDCGYN 2ph9 A 2.88 BS01 GNT A 1 W147 Y188 Y195 W151 Y192 Y199 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 17481657 301 DDDDKLHSQANLMRLKSDLFNRSYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2phb A 2.3 BS02 230 A 1 E97 T98 Y99 F174 A190 V213 W215 G216 G219 G226 Y228 E83 T84 Y85 F162 A180 V203 W205 G206 G208 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=0.32nM remove_due_to_license_issue IC50=0.57nM P00742 17683371 9001 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2pix A 2.4 BS02 FLF A 1 F673 N727 E829 L830 N833 Y834 E837 F3 N57 E159 L160 N163 Y164 E167 ? remove_due_to_license_issue IC50=>50000nM, EC50=67000nM P10275 17911242 2386 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 2piy A 1.43 BS02 528 A 1 H69 E72 R127 N144 R145 T164 H196 Y198 S207 I247 Y248 D255 E270 H64 E67 R122 N139 R140 T159 H192 Y194 S203 I243 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=20nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2piz A 1.6 BS02 606 A 1 E72 R127 S197 Y198 S207 I247 Y248 A250 D255 E270 E68 R123 S194 Y195 S204 I244 Y245 A247 D252 E267 H69 E72 R127 H196 E270 H65 E68 R123 H193 E267 3.4.17.2 0004181,0006508,0008270 ic50=170nM remove_due_to_license_issue P09955 18219114 401 TGHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj0 A 1.65 BS02 922 A 1 H69 E72 R127 N144 R145 T164 H196 S197 Y198 L203 S207 Y248 D255 E270 H64 E67 R122 N139 R140 T159 H192 S193 Y194 L199 S203 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=8.1nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj1 A 1.64 BS02 578 A 1 H69 R71 E72 R127 N144 R145 T164 H196 S197 Y198 L203 S207 I247 Y248 D255 E270 H64 R66 E67 R122 N139 R140 T159 H192 S193 Y194 L199 S203 I243 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=9.7nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj2 A 1.95 BS02 864 A 1 H69 R71 E72 R127 N144 R145 T164 H196 Y198 S207 I247 Y248 D255 E270 F279 H64 R66 E67 R122 N139 R140 T159 H192 Y194 S203 I243 Y244 D251 E266 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=12nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj3 A 1.64 BS02 86A A 1 H69 E72 R127 N144 R145 T164 H196 S197 Y198 L203 S207 Y248 D255 E270 H64 E67 R122 N139 R140 T159 H192 S193 Y194 L199 S203 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=6.6nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj4 A 2.0 BS02 414 A 1 H69 R71 E72 R127 N144 R145 T164 H196 Y198 S199 S207 Y248 A250 D255 E270 H64 R66 E67 R122 N139 R140 T159 H192 Y194 S195 S203 Y244 A246 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=13nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj5 A 1.65 BS02 11B A 1 H69 E72 R127 N144 R145 H196 Y198 L203 S207 I247 Y248 D255 E270 H64 E67 R122 N139 R140 H192 Y194 L199 S203 I243 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=15nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj6 A 1.6 BS02 059 A 1 H69 E72 R127 N144 R145 H196 S197 Y198 L203 S207 I247 Y248 D255 E270 H64 E67 R122 N139 R140 H192 S193 Y194 L199 S203 I243 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=49nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj7 A 1.77 BS02 235 A 1 H69 E72 R127 N144 R145 T164 H196 S197 Y198 S207 I247 Y248 D255 E270 H64 E67 R122 N139 R140 T159 H192 S193 Y194 S203 I243 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=17nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj8 A 1.7 BS02 17A A 1 H69 E72 R127 N144 R145 H196 Y198 S207 I247 Y248 D255 E270 F279 H64 E67 R122 N139 R140 H192 Y194 S203 I243 Y244 D251 E266 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=18nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pj9 A 1.56 BS02 281 A 1 H69 E72 R127 N144 R145 H196 Y198 L203 S207 Y248 D255 E270 H64 E67 R122 N139 R140 H192 Y194 L199 S203 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=12nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pja A 1.7 BS02 33Z A 1 H69 E72 R127 N144 R145 T164 H196 S197 Y198 S199 L203 S207 I247 Y248 A250 D255 E270 F279 H64 E67 R122 N139 R140 T159 H192 S193 Y194 S195 L199 S203 I243 Y244 A246 D251 E266 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=2.2nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pjb A 1.7 BS02 983 A 1 H69 E72 R127 N144 R145 G155 H196 Y198 S199 L203 S207 I247 A250 D255 E270 H64 E67 R122 N139 R140 G150 H192 Y194 S195 L199 S203 I243 A246 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=19nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pjc A 1.74 BS02 343 A 1 H69 E72 R127 N144 R145 T164 H196 S197 Y198 S199 L203 S207 I247 Y248 A250 D255 E270 F279 H64 E67 R122 N139 R140 T159 H192 S193 Y194 S195 L199 S203 I243 Y244 A246 D251 E266 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=1.9nM remove_due_to_license_issue P09955 18219114 401 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 2pjl A 2.3 BS01 047 A 1 V321 L324 F328 E331 F382 A396 L398 F495 V31 L34 F38 E41 F92 A106 L108 F196 ? ic50=190nM remove_due_to_license_issue IC50=190nM P11474 17556356 600 LEVLFQGPVNALVSHLLVVEPEKLYAMLPAVATLSDLFDREIVVTISWAKSIPGFSSLSLSDQMSVLQSVWMEVLVLGVAQRSLPLQDELAFAEDLVLDEEGARAAGLGELGAALLQLVRRLQALRLEREEYVLLKALALANSDSVHIEDAEAVEQLREALHEALLEYEAGRRRAGRLLLTLPLLRQTAGKVLAHFYGVKLEGKVPMHKLFLEMLEAM 2pjt A 2.8 BS06 347 A 1 L159 L160 A161 H197 E198 H201 H207 L214 P217 Y219 L81 L82 A83 H119 E120 H123 H129 L136 P139 Y141 H197 E198 H201 H207 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=860nM P45452 17606376 401 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTHFMLPDDDVQGIQSLYGP 2pk5 A 1.9 BS01 075 A 1 D25 G27 A28 D29 D30 V32 G48 P81 V82 I84 D25 G27 A28 D29 D30 V32 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=20pM remove_due_to_license_issue Q9J2P7 17581235 900 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pk5 B 1.9 BS01 075 A 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 D25 G27 A28 D29 D30 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q9J2P7 17581235 900 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pk6 A 1.45 BS01 O33 B 1 R8 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 V82 I84 R8 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q9Q2G8 17581235 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pk6 B 1.45 BS01 O33 B 1 D25 G27 A28 D29 G48 G49 I50 I84 D25 G27 A28 D29 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=13pM remove_due_to_license_issue Q9Q2G8 17581235 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pks C 2.5 BS02 G44 C 1 I209 D229 A230 S235 S256 W257 G258 I25 D45 A46 S51 S72 W73 G74 E232 G233 D234 S235 G236 E48 G49 D50 S51 G52 3.4.21.5 0004252,0006508 ic50=11uM remove_due_to_license_issue P00734 18019535 101 GQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 2pl0 A 2.8 BS01 STI A 1 A271 K273 E288 M292 V301 I314 T316 Y318 M319 I361 H362 A381 D382 F383 A41 K43 E58 M62 V71 I84 T86 Y88 M89 I131 H132 A151 D152 F153 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=40nM, IC50=320nM, Ki=6893nM P06239 17910071 200 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFF 2pll A 1.9 BS03 ABH A 1 D124 D128 S137 H141 G142 D183 D232 E277 D120 D124 S133 H137 G138 D179 D228 E273 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=5nM remove_due_to_license_issue P05089 17562323 555 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 2pmk A 1.6 BS01 128 A 1 Y477 G505 S506 G507 K508 S509 T510 K513 Y13 G41 S42 G43 K44 S45 T46 K49 ? 0005524,0016887 remove_due_to_license_issue P08716 18155559 301 HHDITFRNIRFRYKPDSPVILDNINLSIKQGEVIGIVGRSGSGKSTLTKLIQRFYIPENGQVLIDGHDLALADPNWLRRQVGVVLQDNVLLNRSIIDNISLANPGMSVEKVIYAAKLAGAHDFISELREGYNTIVGEQGAGLSGGQRQRIAIARALVNNPKILIFDEATSALDYESEHVIMRNMHKICKGRTVIIIAHRLSTVKNADRIIVMEKGKIVEQGKHKELLSEPESLYSYLYQLQSD 2pmn X 2.8 BS01 K51 X 1 L34 N35 K55 L101 Y117 Y119 M120 D123 L179 L39 N40 K60 L106 Y122 Y124 M125 D128 L184 N177 D190 N182 D195 2.7.12.2 0000165,0004672,0004674,0004676,0004677,0004679,0004694,0004708,0004711,0005524,0005634,0005737,0006338,0006468,0016301,0035175,0035401,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0044773,0072354,0072371,0072518,0106310,0140801,0140823,0140855,0140857,1990244 remove_due_to_license_issue Q7YTF7 18275814 344 GPLGSMKDILSNYSNLIYLNKYVKEKDKYINDYRIIRTLNQGKFNKIILCEKDNKFYALKKYEKSLLEKKRDFTKSNNDKISIKSKYDDFKNELQIITDIKNEYCLTCEGIITNYDEVYIIYEYMENDSILKFDEYFFVLDKNYTCFIPIQVIKCIIKSVLNSFSYIHNEKNICHRDVKPSNILMDKNGRVKLSDFGESEYMVDKKIKGSRGTYEFMPPEFFSNESSYNGAKVDIWSLGICLYVMFYNVVPFSLKISLVELFNNIRTKNIEYPLDRNHFLYPLTNFLSNEDIDFLKLFLRKNPAERITSEDALKHEWLADTNIEDLREFSKELYKKRKKL 2pnc A 2.4 BS04 CLU A 1 Y383 D385 M467 A470 D471 Y472 H521 Y299 D301 M373 A376 D377 Y378 H427 Y371 D385 Y470 H519 H521 H683 Y287 D301 Y376 H425 H427 H589 1.4.3.21 0005507,0005576,0005769,0005783,0005794,0005886,0008131,0009308,0016491,0016641,0046872,0048038,0052595 Ki=466uM remove_due_to_license_issue Q29437 17989349 808 QLFADLSREELTTVMSFLTQQLGPDLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGGQPQPNVTELVVGPLPQPSYMRDVTVERHGGPLPYYRRPVLLREYLDIDQMIFNRELPQAAGVLHHCCSYKQGGQKLLTMNSAPRGVQSGDRSTWFGIYYNITKGGPYLHPVGLELLVDHKALDPADWTVQKVFFQGRYYENLAQLEEQFEAGQVNVVVIPDRFSVQGNRVASSLWTFSFGLGAFSGPRVFDVRFQGERLAYEISLQEAGAVYGGNTPAAMLTRYMDSGFGMGYFATPLIRGVDCPYLATYMDWHFVVESQTPKTLHDAFCVFEQNKGLPLRRGGVAQTVLVFRSVSTMLNYDYVWDMVFYPNGAIEVKLHATGYISSAFLFGAARRYGNQVGEHTLGPVHTHSAHYKVDLDVGGLENWVWAEDMAFVPTAIPWSPEHQIQRLQVTRKQLETEEQAAFPLGGASPRYLYLASKQSNKWGHPRGYRIQTVSFAGGPMPQNSPMERAFSWGRYQLAITQRKETEPSSSSVFNQNDPWTPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDQEPSMD 2pog A 1.84 BS01 WST A 1 M343 E353 L384 L387 R394 F404 I424 H524 M30 E40 L71 L74 R81 F91 I111 H211 ? Ki=0.29nM remove_due_to_license_issue Ki=0.35nM P03372 17485205 201 LALSLTADQMVSALLDAEPPILYSEYASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKVPLYDLLLEMLDAHRLH 2poq X 2.59 BS01 ISD X 1 K1156 F1279 D1280 K155 F278 D279 1.1.1.179,1.3.1.20 0000166,0016491,0042843,0047115,0047837 remove_due_to_license_issue Q9TQS6 18453689 500 ALRWGIVSVGLISSDFTAVLQTLPRSEHQVVAVAARDLSRAKEFAQKHDIPKAYGSYEELAKDPNVEVAYVGTQHPQHKAAVMLCLAAGKAVLCEKPMGVNAAEVREMVTEARSRGLFLMEAIWTRFFPASEALRSVLAQGTLGDLRVARAEFGKNLTHVPRAVDWAQAGGALLDLGIYCVQFISMVFGGQKPEKISVMGRRHETGVDDTVTVLLQYPGEVHGSFTCSITAQLSNTASVSGTKGMAQLLNPCWCPTELVVKGEHKEFLLPPVPKNCNFDNGAGMSYEAKHVRECLRKGLKESPVIPLVESELLADILEEVRRAIGVTFPQD 2pou A 1.6 BS02 I7A A 1 H94 H96 H119 V121 F131 L141 V143 L198 T199 W209 H92 H94 H117 V119 F128 L138 V140 L195 T196 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=38nM remove_due_to_license_issue Ki=38nM, IC50=40nM P00918 17540563 1000 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2pov A 1.6 BS02 I7B A 1 H94 H119 V121 V143 L198 T199 W209 H92 H117 V119 V140 L195 T196 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=75nM remove_due_to_license_issue Ki=75nM, IC50=90nM P00918 17540563 1000 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2pow A 1.75 BS02 I7C A 1 Q92 H94 H119 F131 V143 L198 T199 Q89 H91 H116 F127 V139 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=63nM remove_due_to_license_issue Ki=63nM, IC50=340nM P00918 17540563 1000 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2pq9 A 1.6 BS01 GG9 A 1 K22 S23 R27 G96 T97 R124 S169 S170 Q171 S197 Y200 D313 N336 K340 R344 H385 R386 K411 K22 S23 R27 G96 T97 R124 S169 S170 Q171 S197 Y200 D313 N336 K340 R344 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 Ki=7.8nM remove_due_to_license_issue P0A6D3 17958399 501 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 2pqb A 1.8 BS01 GG9 A 1 K28 S29 R33 A100 T101 R128 S173 Q175 D326 K353 E354 R357 R405 K23 S24 R28 A95 T96 R123 S168 Q170 D321 K348 E349 R352 R400 K28 S29 D55 N98 R128 D326 E354 H404 R405 T431 K23 S24 D50 N93 R123 D321 E349 H399 R400 T426 2.5.1.19 0003824,0003866,0005737,0008652,0009073,0009423,0009635,0016740,0016765 Ki=63nM remove_due_to_license_issue Q9R4E4 17958399 501 SSRPATARKSSGLSGTVRIPGDKSISHRSFMFGGLASGETRITGLLEGEDVINTGKAMQAMGARIRKEGDTWIIDGVGNGGLLAPEAPLDFGNAATGCRLTMGLVGVYDFDSTFIGDASLTKRPMGRVLNPLREMGVQVKSEDGDRLPVTLRGPKTPTPITYRVPMASAQVKSAVLLAGLNTPGITTVIEPIMTRDHTEKMLQGFGANLTVETDADGVRTIRLEGRGKLTGQVIDVPGDPSSTAFPLVAALLVPGSDVTILNVLMNPTRTGLILTLQEMGADIEVINPRLAGGEDVADLRVRSSTLKGVTVPEDRAPSMIDEYPILAVAAAFAEGATVMNGLEELRVKESDRLSAVANGLKLNGVDCDEGETSLVVRGRPDGKGLGNASGAAVATHLDHRIAMSFLVMGLVSENPVTVDDATMIATSFPEFMDLMAGLGAKIELS 2pqc A 1.6 BS01 RC1 A 1 K28 S29 R33 T101 R128 S173 Q175 D326 K353 E354 R357 R405 K23 S24 R28 T96 R123 S168 Q170 D321 K348 E349 R352 R400 K28 S29 D55 N98 R128 D326 E354 H404 R405 T431 K23 S24 D50 N93 R123 D321 E349 H399 R400 T426 2.5.1.19 0003824,0003866,0005737,0008652,0009073,0009423,0009635,0016740,0016765 Ki=1800nM remove_due_to_license_issue Q9R4E4 17958399 601 SSRPATARKSSGLSGTVRIPGDKSISHRSFMFGGLASGETRITGLLEGEDVINTGKAMQAMGARIRKEGDTWIIDGVGNGGLLAPEAPLDFGNAATGCRLTMGLVGVYDFDSTFIGDASLTKRPMGRVLNPLREMGVQVKSEDGDRLPVTLRGPKTPTPITYRVPMASAQVKSAVLLAGLNTPGITTVIEPIMTRDHTEKMLQGFGANLTVETDADGVRTIRLEGRGKLTGQVIDVPGDPSSTAFPLVAALLVPGSDVTILNVLMNPTRTGLILTLQEMGADIEVINPRLAGGEDVADLRVRSSTLKGVTVPEDRAPSMIDEYPILAVAAAFAEGATVMNGLEELRVKESDRLSAVANGLKLNGVDCDEGETSLVVRGRPDGKGLGNASGAAVATHLDHRIAMSFLVMGLVSENPVTVDDATMIATSFPEFMDLMAGLGAKIELS 2pqj A 2.8 BS01 ADE A 1 Y94 L95 G128 V202 C206 R210 Y74 L75 G108 V152 C156 R160 3.2.2.22 0017148,0030598 remove_due_to_license_issue P25891 17855394 501 MKFTEIFPVEDANYPYSAFIASVRKDVIKHCTDHKGIFQPVLPPEKKVPELWLYTELKTRTSSITLAIRMDNLYLVGFRTPGGVWWEFGKDGDTHLLGDNPRWLGFGGRYQDLIGNKGLETVTMGRAEMTRAVNDLAKKKKADTKSKLVKLVVMVCEGLRFNTVSRTVDAGFNSQHGVTLTVTQGKQVQKWDRISKAAFEWADHPTAVIPDMQKLGIKDKNEAARIVALVKNQ 2pql A 2.2 BS01 TSS A 1 I21 R22 Y24 H35 I36 V39 Y94 F110 D111 E114 M135 I21 R22 Y24 H35 I36 V39 Y94 F110 D111 E114 M135 ? 0005549,0005576,0005615,0007608,0042311 Kd=53nM remove_due_to_license_issue Q7PNF2 17928288 145 ETVQDCENKLPPSLKSRLCEIRRYEIIEGPEMDKHIHCVMRALDFVYEDGRGDYHKLYDPLNIIELDKRHDVNLEKCIGECVQVPTSERAHVFYKCLLKSTTGRTFKKVFDLMELKKAGKVPQHQRYTAEFVQIMKDYDKALNC 2pqz A 1.55 BS01 G0G A 1 D25 G27 A28 D30 V32 G49 I50 I84 D25 G27 A28 D30 V32 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2.15uM remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pqz B 1.55 BS01 G0G A 1 D25 G27 G49 I50 P81 I84 D25 G27 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pre A 2.7 BS01 E64 A 1 Q19 G23 C25 H61 G65 N156 H157 Q19 G23 C25 H61 G65 N156 H157 Q19 C25 H157 N173 Q19 C25 H157 N173 3.4.22.- 0006508,0008234 remove_due_to_license_issue A8DS38 18167146 302 LPEQIDWRKKGAVTPVKNQGKCGSCWAFSTVSTVESINQIRTGNLISLSEQQLVDCNKKNHGCKGGAFVYAYQYIIDNGGIDTEANYPYKAVQGPCRAAKKVVRIDGYKGVPHCNENALKKAVASQPSVVAIDASSKQFQHYKSGIFSGPCGTKLNHGVVIVGYWKDYWIVRNSWGRYWGEQGYIRMKRVGGCGLCGIARLPYYPTKA 2pri A 2.3 BS01 D6G A 1 W67 Y75 R193 D227 R310 W55 Y63 R181 D215 R298 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=1.23mM remove_due_to_license_issue P00489 7500360 930 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 2prj A 2.3 BS01 NBG A 1 G135 L136 N284 H377 T378 N484 E672 G675 G123 L124 N272 H365 T366 N472 E660 G663 H377 K568 R569 K574 T676 K680 H365 K556 R557 K562 T664 K668 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=32uM remove_due_to_license_issue Ki=32000nM P00489 8580837 998 ISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 2psj A 1.8 BS01 CEI A 1 W156 D162 F180 K189 F261 H285 W152 D158 F176 K185 F257 H281 N53 D120 W121 E144 W156 G260 H285 N51 D118 W119 E142 W152 G256 H281 1.13.12.5 0003824,0004301,0004497,0008218,0016020,0016831,0050248 Ki~20nM remove_due_to_license_issue P27652 17980388 501 SKVYDPEQRKRMITGPQWWARCKQMNVLDSFINYYDSEKHAENAVIFLHGNATSSYLWRHVVPHIEPVARCIIPDLIGMGKSGKSGNGSYRLLDHYKYLTAWFELLNLPKKIIFVGHDWGAALAFHYAYEHQDRIKAIVHMESVVDVIESEWPDIEEDIALIKSEEGEKMVLENNFFVETVLPSKIMRKLEPEEFAAYLEPFKEKGEVRRPTLSWPREIPLVKGGKPDVVQIVRNYNAYLRASDDLPKLFIESDPGFFSNAIVEGAKKFPNTEFVKVKGLHFLQEDAPDEMGKYIKSFVERVLKNE 2psu A 1.93 BS01 MUU A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=24nM remove_due_to_license_issue O38723 17539822 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2psu B 1.93 BS01 MUU A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38723 17539822 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2psv A 1.75 BS01 MUV A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=58nM remove_due_to_license_issue O38707 17539822 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2psv B 1.75 BS01 MUV A 1 D25 G27 A28 I50 P81 V82 D25 G27 A28 I50 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38707 17539822 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pt9 A 2.2 BS01 S4M A 1 Q93 H103 G124 G125 D127 E147 I148 V152 D178 A179 D196 S198 P203 A204 Q53 H63 G84 G85 D87 E107 I108 V112 D138 A139 D156 S158 P163 A164 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 remove_due_to_license_issue Q8II73 17822713 501 KKWFSEFSIMWPGQAFSLKIKKILYETKSKYQNVLVFESTTYGKVLVLDGVIQLTEKDEFAYHEMMTHVPMTVSKEPKNVLVVGGGDGGIIRELCKYKSVENIDICEIDETVIEVSKIYFKNISCGYEDKRVNVFIEDASKFLENVTNTYDVIIVDSSDPIGPAETLFNQNFYEKIYNALKPNGYCVAQCESLWIHVGTIKNMIGYAKKLFKKVEYANISIPTYPCGCIGILCCSKTDTGLTKPNKKLESKEFADLKYYNYENHSAAFKLPAFLLKEIENI 2ptz A 1.65 BS03 PAH A 1 G38 A39 S40 Q164 E165 D243 D318 K343 R372 S373 K394 G40 A41 S42 Q166 E167 D245 D320 K345 R374 S375 K396 S40 H156 E165 E208 D243 E291 D318 K343 H371 K394 S42 H158 E167 E210 D245 E293 D320 K345 H373 K396 4.2.1.11 0000015,0000287,0004634,0005737,0005829,0006096,0016829,0046872,0097014 remove_due_to_license_issue Q38BV6 17822439 600 SHMTIQKVHGREVLDSRGNPTVEVEVTTEKGVFRSAVPSGASTGVYEACELRDGDKKRYVGKGCLQAVKNVNEVIGPALIGRDELKQEELDTLMLRLDGTPNKGKLGANAILGCSMAISKAAAAAKGVPLYRYLASLAGTKELRLPVPCFNVINGGKHAGNALPFQEFMIAPVKATSFSEALRMGSEVYHSLRGIIKKKYGQDAVNVGDEGGFAPPIKDINEPLPILMEAIEEAGHRGKFAICMDCAASETYDEKKQQYNLTFKSPEPTWVTAEQLRETYCKWAHDYPIVSIEDPYDQDDFAGFAGITEALKGKTQIVGDDLTVTNTERIKMAIEKKACNSLLLKINQIGTISEAIASSKLCMENGWSVMVSHRSGETEDTYIADLVVALGSGQIKTGAPCRGERTAKLNQLLRIEEELGAHAKFGFPGWS 2pu0 A 1.9 BS03 PAH A 1 G38 A39 S40 H156 Q164 E165 D243 D318 K343 R372 S373 K394 G40 A41 S42 H158 Q166 E167 D245 D320 K345 R374 S375 K396 S40 H156 E165 E208 D243 E291 D318 K343 H371 K394 S42 H158 E167 E210 D245 E293 D320 K345 H373 K396 4.2.1.11 0000015,0000287,0004634,0005737,0005829,0006096,0016829,0046872,0097014 remove_due_to_license_issue Q38BV6 17822439 600 SHMTIQKVHGREVLDSRGNPTVEVEVTTEKGVFRSAVPSGASTGVYEACELRDGDKKRYVGKGCLQAVKNVNEVIGPALIGRDELKQEELDTLMLRLDGTPNKGKLGANAILGCSMAISKAAAAAKGVPLYRYLASLAGTKELRLPVPCFNVINGGKHAGNALPFQEFMIAPVKATSFSEALRMGSEVYHSLRGIIKKKYGQDAVNVGDEGGFAPPIKDINEPLPILMEAIEEAGHRGKFAICMDCAASETYDEKKQQYNLTFKSPEPTWVTAEQLRETYCKWAHDYPIVSIEDPYDQDDFAGFAGITEALKGKTQIVGDDLTVTNTERIKMAIEKKACNSLLLKINQIGTISEAIASSKLCMENGWSVMVSHRSGETEDTYIADLVVALGSGQIKTGAPCRGERTAKLNQLLRIEEELGAHAKFGFPGWS 2pu1 A 1.8 BS03 FSG A 1 G38 A39 S40 Q164 E165 D243 D318 K343 R372 S373 K394 G40 A41 S42 Q166 E167 D245 D320 K345 R374 S375 K396 S40 H156 E165 E208 D243 E291 D318 K343 H371 K394 S42 H158 E167 E210 D245 E293 D320 K345 H373 K396 4.2.1.11 0000015,0000287,0004634,0005737,0005829,0006096,0016829,0046872,0097014 remove_due_to_license_issue Q9NDH8 17822439 600 SHMTIQKVHGREVLDSRGNPTVEVEVTTEKGVFRSAVPSGASTGVYEACELRDGDKKRYVGKGCLQAVKNVNEVIGPALIGRDELKQEELDTLMLRLDGTPNKGKLGANAILGCSMAISKAAAAAKGVPLYRYLASLAGTKELRLPVPCFNVINGGKHAGNALPFQEFMIAPVKATSFSEALRMGSEVYHSLRGIIKKKYGQDAVNVGDEGGFAPPIKDINEPLPILMEAIEEAGHRGKFAICMDCAASETYDEKKQQYNLTFKSPEPTWVTAEQLRETYCKWAHDYPIVSIEDPYDQDDFAGFAGITEALKGKTQIVGDDLTVTNTERIKMAIEKKACNSLLLKINQIGTISEAIASSKLCMENGWSVMVSHRSGETEDTYIADLVVALGSGQIKTGAPCRGERTAKLNQLLRIEEELGAHAKFGFPGWS 2pu2 A 1.86 BS01 DK2 A 1 S64 L119 Y150 Y221 G317 A318 T319 G320 S61 L116 Y147 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=37uM remove_due_to_license_issue P00811 18333608 702 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2pue A 2.7 BS01 dna B 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S12 T14 T15 R24 V26 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 9454587 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLEQNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 2puf A 3.0 BS01 dna B 0 S14 T16 T17 R26 A29 T32 L54 K55 S12 T14 T15 R24 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 9454587 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLEQNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 2pug A 2.7 BS01 dna B 0 S14 T16 T17 R26 V28 A29 T32 L54 K55 S12 T14 T15 R24 V26 A27 T30 L52 K53 ? 0000976,0001217,0002057,0003677,0003700,0005515,0005829,0006164,0006355,0042803,0045892,1900372 remove_due_to_license_issue P0ACP7 9454587 699 ~ 715 TIKDVAKRANVSTTTVSHVINKTRFVAEETRNAVWAAIKELHYSPSAVARSLKVNHTKSIGLLATSSEAAYFAEIIEAVEKNCFQKGYTLILGNAWNNLEKQRAYLSMMAQKRVDGLLVMCSEYPEPLLAMLEEYRHIPMVVMDWGEAKADFTDAVIDNAFEGGYMAGRYLIERGHREIGVIPGPLEQNTGAGRLAGFMKAMEEAMIKVPESWIVQGDFEPESGYRAMQQILSQPHRPTAVFCGGDIMAMGALCAADEMGLRVPQDVSLIGYDNVRNARYFTPALTTIHQPKDSLGETAFNMLLDRIVNKREEPQSIEVHPRLIERRSVADGPFRDYR 2pvh A 2.2 BS01 P19 A 1 V45 G46 V53 I66 V116 N118 M163 I174 V40 G41 V48 I61 V111 N113 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.26uM remove_due_to_license_issue Ki=260nM P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2pvj A 1.7 BS01 P44 A 1 I66 K68 F113 Y115 V116 N118 H160 M163 I174 I61 K63 F108 Y110 V111 N113 H155 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.005uM remove_due_to_license_issue P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAEN 2pvk A 1.9 BS01 P45 A 1 V45 I66 K68 F113 Y115 V116 D120 H160 M163 I174 V40 I61 K63 F108 Y110 V111 D115 H155 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.008uM remove_due_to_license_issue P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2pvl A 1.9 BS01 P55 A 1 R43 V45 V53 I66 F113 Y115 V116 N118 H160 M163 I174 R38 V40 V48 I61 F108 Y110 V111 N113 H155 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.024uM remove_due_to_license_issue P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2pvm A 2.0 BS01 P29 A 1 V45 V53 I66 Y115 V116 M163 I174 V40 V48 I61 Y110 V111 M158 I169 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.36uM remove_due_to_license_issue P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2pvn A 2.0 BS01 P63 A 1 V53 I66 K68 F113 Y115 V116 M163 I174 D175 V48 I61 K63 F108 Y110 V111 M158 I169 D170 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.00035uM remove_due_to_license_issue P28523 17540560 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2pvu A 1.79 BS01 LYS A 1 F31 W68 G86 I87 T88 R93 Q132 T135 T136 D175 F15 W52 G70 I71 T72 R77 Q116 T119 T120 D159 ? 0015276,0016020,0034220 Kd=0.49uM remove_due_to_license_issue D0VWX8 18022195 301 GATKKKVVVGTDAAFAPFEYMQKGKIVGFDVDLLDAVMKAAGLDYELKNIGWDPLFASLQSKEVDMGISGITITDERKQSYDFSDPYFEATQVILVKQGSPVKNALDLKGKTIGVQNATTGQEAAEKLFGKGPHIKKFETTVVAIMELLNGGVDAVITDNAVANEYVKNNPNKKLQVIEDPKNFASEYYGMIFPKNSELKAKVDEALKNVINSGKYTEIYKKWFGKEPKLDRLKQ 2pvv A 2.11 BS04 OSE A 1 F209 R210 E424 G427 L428 G518 Y552 K699 Y700 F155 R156 E370 G373 L374 G464 Y498 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=438uM remove_due_to_license_issue Q04609 17567119 1768 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2pvw A 1.71 BS04 G88 A 1 R210 N257 D387 E424 E425 G518 Y552 H553 K699 Y700 R155 N202 D332 E369 E370 G463 Y494 H495 K639 Y640 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.3nM remove_due_to_license_issue Ki=0.280000nM, IC50=300nM, Kd=0.5nM, EC50=0.620000nM Q04609 17567119 1768 HNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2pwc A 1.78 BS01 G3G A 1 D25 G27 A28 D30 G48 I50 V82 I84 D25 G27 A28 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.27uM remove_due_to_license_issue P03367 18348517 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pwc B 1.78 BS01 G3G A 1 L23 D25 A28 G49 I50 P81 I84 L23 D25 A28 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18348517 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pwd A 1.8 BS02 NOJ A 1 D61 Y64 H104 F164 D200 E254 H326 D327 R414 D61 Y64 H104 F164 D200 E254 H326 D327 R414 D99 R198 D200 E254 H326 D327 D99 R198 D200 E254 H326 D327 5.4.99.11 0004556,0005975,0009313,0016798,0016853,0046872 Ki=40uM remove_due_to_license_issue Q2PS28 17597061 8000 KPGAPWWKSAVFYQVYPRSFKDTNGDGIGDFKGLTEKLDYLKGLGIDAIWINPHYASPNTDNGYDISDYREVMKEYGTMEDFDRLMAELKKRGMRLMVDVVINHSSDQHEWFKSSRASKDNPYRDYYFWRDGKDGHEPNNYPSFFGGSAWEKDPVTGQYYLHYFGRQQPDLNWDTPKLREELYAMLRFWLDKGVSGMRFDTVATYSKTPGFPDLTPEQMKNFAEAYTQGPNLHRYLQEMHEKVFDHYDAVTAGEIFGAPLNQVPLFIDSRRKELDMAFTFDLIRYDRALDRWHTIPRTLADFRQTIDKVDAIAGEYGWNTFFLGNHDNPRAVSHFGDDRPQWREASAKALATVTLTQRGTPFIFQGDELGMTNYPFKTLQDFDDIEVKGFFQDYVETGKATAEELLTNVALTSRDNARTPFQWDDSANAGFTTGKPWLKVNPNYTEINAAREIGDPKSVYSFYRNLISIRHETPALSTGSYRDIDPSNADVYAYTRSQDGETYLVVVNFKAEPRSFTLPDGMHIAETLIESSSPAAPAAGAASLELQPWQSGIYKVK 2pwg A 2.2 BS02 CTS A 1 D61 Y64 H104 F164 D200 E254 D327 R414 D60 Y63 H103 F163 D199 E253 D326 R413 D99 R198 D200 E254 H326 D327 D98 R197 D199 E253 H325 D326 5.4.99.11 0004556,0005975,0009313,0016798,0016853,0046872 Ki=15uM remove_due_to_license_issue Q2PS28 17597061 8000 PGAPWWKSAVFYQVYPRSFKDTNGDGIGDFKGLTEKLDYLKGLGIDAIWINPHYASPNTDNGYDISDYREVMKEYGTMEDFDRLMAELKKRGMRLMVDVVINHSSDQHEWFKSSRASKDNPYRDYYFWRDGKDGHEPNNYPSFFGGSAWEKDPVTGQYYLHYFGRQQPDLNWDTPKLREELYAMLRFWLDKGVSGMRFDTVATYSKTPGFPDLTPEQMKNFAEAYTQGPNLHRYLQEMHEKVFDHYDAVTAGEIFGAPLNQVPLFIDSRRKELDMAFTFDLIRYDRALDRWHTIPRTLADFRQTIDKVDAIAGEYGWNTFFLGNHDNPRAVSHFGDDRPQWREASAKALATVTLTQRGTPFIFQGDELGMTNYPFKTLQDFDDIEVKGFFQDYVETGKATAEELLTNVALTSRDNARTPFQWDDSANAGFTTGKPWLKVNPNYTEINAAREIGDPKSVYSFYRNLISIRHETPALSTGSYRDIDPSNADVYAYTRSQDGETYLVVVNFKAEPRSFTLPDGMHIAETLIESSSPAAPAAGAASLELQPWQSGIYKVK 2pwr A 1.5 BS01 G4G B 1 D25 G27 A28 D30 V32 G48 I50 V82 I84 D25 G27 A28 D30 V32 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18348517 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pwr B 1.5 BS01 G4G B 1 L23 D25 A28 D29 D30 G48 G49 I50 P81 I84 L23 D25 A28 D29 D30 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.26uM remove_due_to_license_issue P03367 18348517 501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2py4 A 1.49 BS01 DUP A 1 N77 G80 T81 I82 D83 Y86 K91 N76 G79 T80 I81 D82 Y85 K90 A25 R64 G66 L73 D83 A24 R63 G65 L72 D82 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046080,0046081,0046872 Kd=0.2uM remove_due_to_license_issue P9WNS5 18519027 777 STTLAIVRLDPGLPLPSRAHDGDAGVDLYSAEDVELAPGRRALVRTGVAVAVPFGMVGLVHPRSGLATRVGLSIVNSPGTIDAGYRGEIKVALINLDPAAPIVVHRGDRIAQLLVQRVELVELVEVSSFDEAGLASTSRGDGGHGSSGGHASL 2pyi A 1.88 BS01 DL8 A 1 L136 N282 D283 N284 F286 H377 A383 V455 N484 E672 S674 G675 L127 N263 D264 N265 F267 H349 A355 V427 N456 E644 S646 G647 H377 K568 R569 K574 T676 K680 H349 K540 R541 K546 T648 K652 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=179uM remove_due_to_license_issue Ki=180000nM P00489 18041758 998 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 2pym A 1.9 BS01 1UN A 1 D25 G27 A28 D29 N30 I50 P81 I84 D25 G27 A28 D29 N30 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=150nM remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRDLLTQIGCTLNF 2pym B 1.9 BS01 1UN A 1 R8 L23 D25 G27 G49 I50 R8 L23 D25 G27 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRDLLTQIGCTLNF 2pyn A 1.85 BS01 1UN A 1 D25 G27 A28 D29 N30 I50 P81 I84 D25 G27 A28 D29 N30 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=27nM remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKVIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pyn B 1.85 BS01 1UN A 1 D25 G27 G49 I50 D25 G27 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKVIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2pyy A 2.1 BS01 GLU A 1 R10 V50 A68 S70 R75 T116 S119 T120 F155 D156 R7 V44 A62 S64 R69 T107 S110 T111 F146 D147 ? 0015276,0016020,0030313,0034220 Kd=0.000023M remove_due_to_license_issue D0VWX9 18164033 1620 PLLVATRVIPPFVLSNLSGFSIDLWRSIATQIGIESKLIEYSSVPELISAIKDNKVNLGIAAISITAEREQNFDFSLPIFASGLQIMVRNGDIRSIDDLPGKVVATTAGSTAATYLREHHISVLEVPKIEEAYKALQTKKADAVVFDAPVLLFYAANEGKGKVEIVGSILREESYGIILPNNSPYRKPINQALLNLKENGTYQSLYDKWFDP 2pze A 1.7 BS02 ATP A 1 W401 V440 T460 G461 G463 K464 T465 S466 Q493 W16 V23 T43 G44 G46 K47 T48 S49 Q76 5.6.1.6 0005524,0016887 Kd=0.84uM remove_due_to_license_issue P13569 20150177 1 SLTTTEVVMENVTAFWEEGGTPVLKDINFKIERGQLLAVAGSTGAGKTSLLMMIMGELEPSEGKIKHSGRISFCSQFSWIMPGTIKENIIFGVSYDEYRYRSVIKACQLEEDISKFAEKDNIVLGEGGITLSGGQRARISLARAVYKDADLYLLDSPFGYLDVLTEKEIFESCVCKLMANKTRILVTSKMEHLKKADKILILHEGSSYFYGTFSELQNLDFSSKLM 2pze A 1.7 BS03 ATP B 1 T547 S549 G550 G551 Q552 T130 S132 G133 G134 Q135 5.6.1.6 0005524,0016887 Kd=0.84uM remove_due_to_license_issue P13569 20150177 2 SLTTTEVVMENVTAFWEEGGTPVLKDINFKIERGQLLAVAGSTGAGKTSLLMMIMGELEPSEGKIKHSGRISFCSQFSWIMPGTIKENIIFGVSYDEYRYRSVIKACQLEEDISKFAEKDNIVLGEGGITLSGGQRARISLARAVYKDADLYLLDSPFGYLDVLTEKEIFESCVCKLMANKTRILVTSKMEHLKKADKILILHEGSSYFYGTFSELQNLDFSSKLM 2pzi A 2.4 BS01 AXX A 1 V235 I292 V161 I214 D276 K278 N281 D293 T309 D198 K200 N203 D215 T231 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004711,0005515,0005524,0005737,0005829,0005886,0006338,0006468,0006538,0006543,0030682,0035175,0035402,0035403,0035556,0035979,0042783,0042802,0043457,0044022,0044023,0044024,0044025,0046677,0052027,0052170,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=3uM remove_due_to_license_issue P9WI73 17616581 753 GSHMLGGGLVEIPRAPDIDPLEALMTNPVVPESKRFCWNCGRPVGRSGASEGWCPYCGSPYSFLPQLNPGDIVAGQYEVKGCIAHGGLGWIYLALDRNVNGRPVVLKGLVHSGDAEAQAMAMAERQFLAEVVHPSIVQIFNFVEHTDRHGDPVGYIVMEYVGGQSLKQKLPVAEAIAYLLEILPALSYLHSIGLVYNDLKPENIMLTEEQLKLIDLGAVSRINSFGYLYGTPGFQAPEIVRTGPTVATDIYTVGRTLAALTLDLPTRNGRYVDGLPEDDPVLKTYDSYGRLLRRAIDPDPRQRFTTAEEMSAQLTGVLREVVAQDTGVPRPGLSTIFSPSRSTFGVDLLVAHTDVYLDGQVHAEKLTANEIVTALSVPLVDPTDVAASVLQATVLSQPVQTLDSLRAARHGDFSESVELPLMEVRALLDLGDVAKATRKLDDLAERVGWRWRLVWYRAVAELLTGDYDSATKHFTEVLDTFPGELAPKLALAATAELAGNTDEHKFYQTVWSTNDGVISAAFGLARARSAEGDRVGAVRTLDEVPPTSRHFTTARLTSAVTLLVTEEQIRDAARRVEALPPTEPRVLQIRALVLGGALDWLKDNKASTNHILGFPFTSHGLRLGVEASLRSLARVAPTQRHRYTLVDMANKVRP 2pzy A 2.9 BS01 B18 A 1 L70 L72 G73 V78 M138 C140 L141 L193 T206 D207 L29 L31 G32 V37 M97 C99 L100 L149 T162 D163 D186 K188 E190 N191 D207 D142 K144 E146 N147 D163 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P49137 17576063 1 QFPQFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDK 2q11 A 2.4 BS01 XX4 A 1 D32 Y71 K75 W76 K107 F108 I118 D228 G230 T231 D35 Y74 K78 W79 K110 F111 I121 D231 G233 T234 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D231 T234 3.4.23.46 0004190,0006508,0016020 Ki=900nM remove_due_to_license_issue Ki=900nM P56817 17685503 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLQQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2q15 A 2.4 BS01 3MR A 1 L30 D32 V69 Y71 K75 I118 D228 R235 L30 D32 V69 Y71 K75 I118 D228 R235 D32 S35 N37 A39 Y71 D228 T231 D32 S35 N37 A39 Y71 D228 T231 3.4.23.46 0004190,0006508,0016020 Ki=11nM remove_due_to_license_issue Ki=8nM P56817 17685503 386 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLQQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2q1j A 1.9 BS02 FXI A 1 E97 T98 Y99 E147 F174 A190 Q192 V213 W215 G216 G219 C220 Y228 E83 T84 Y85 E135 F162 A180 Q182 V203 W205 G206 G208 C209 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=0.0008uM remove_due_to_license_issue P00742 16529937 801 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2q1l A 2.05 BS01 882 A 1 E559 C561 L562 S565 R568 K735 A751 N755 L853 A856 H861 E90 C92 L93 S96 R99 K266 A282 N286 L384 A387 H392 E559 K691 D767 E90 K222 D298 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=12.4nM remove_due_to_license_issue IC50=1.8nM P04035 17574412 876 AKFLSDAEIIQLVNAIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 2q1l A 2.05 BS02 882 A 2 R590 S684 D690 K692 R121 S215 D221 K223 E559 K691 D767 E90 K222 D298 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=12.4nM remove_due_to_license_issue IC50=1.8nM P04035 17574412 877 AKFLSDAEIIQLVNAIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 2q1l B 2.05 BS01 882 A 1 R590 S661 V683 S684 D690 K692 R130 S201 V223 S224 D230 K232 E559 K691 D767 E99 K231 D307 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue IC50=1.8nM P04035 17574412 876 AKFLSDAEIIQLVNAKHIPAYKLETLIHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 2q1l B 2.05 BS02 882 A 2 E559 C561 L562 S565 K735 H752 L853 A856 G860 E99 C101 L102 S105 K275 H292 L393 A396 G400 E559 K691 D767 E99 K231 D307 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue IC50=1.8nM P04035 17574412 877 AKFLSDAEIIQLVNAKHIPAYKLETLIHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 2q1q A 1.9 BS02 OSP A 1 Q92 H94 H119 L198 T199 T200 Q89 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7nM remove_due_to_license_issue Ki=9.0nM P00918 17588751 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2q2a A 1.79 BS01 ARG A 1 D28 F31 W68 S85 G86 I87 T88 R93 Q132 T135 T136 D175 D18 F21 W58 S75 G76 I77 T78 R83 Q122 T125 T126 D165 ? 0015276,0016020,0034220 Kd=0.039uM remove_due_to_license_issue D0VWX8 18022195 904 SSGGDGGATKKKVVVGTDAAFAPFEYMQKGKIVGFDVDLLDAVMKAAGLDYELKNIGWDPLFASLQSKEVDMGISGITITDERKQSYDFSDPYFEATQVILVKQGSPVKNALDLKGKTIGVQNATTGQEAAEKLFGKGPHIKKFETTVVAIMELLNGGVDAVITDNAVANEYVKNNPNKKLQVIEDPKNFASEYYGMIFPKNSELKAKVDEALKNVINSGKYTEIYKKWFGKEPKLDRLKQ 2q2c A 2.35 BS01 HIS A 1 F31 W68 S85 G86 I87 T88 R93 Q132 T135 T136 D175 F11 W48 S65 G66 I67 T68 R73 Q112 T115 T116 D155 ? 0015276,0016020,0034220 Kd=0.42uM remove_due_to_license_issue D0VWX8 18022195 504 KKVVVGTDAAFAPFEYMQKGKIVGFDVDLLDAVMKAAGLDYELKNIGWDPLFASLQSKEVDMGISGITITDERKQSYDFSDPYFEATQVILVKQGSPVKNALDLKGKTIGVQNATTGQEAAEKLFGKGPHIKKFETTVVAIMELLNGGVDAVITDNAVANEYVKNNPNKKLQVIEDPKNFASEYYGMIFPKNSELKAKVDEALKNVINSGKYTEIYKKWFGKEPKLDRLKQ 2q2k A 3.0 BS01 dna F 0 R29 G30 K32 T33 R37 R26 G27 K29 T30 R34 ? remove_due_to_license_issue O87365 18097417 12 ~ 31 KETKHLLKIKKEDYPQIFDFLENVPRGTKTAHIREALRRYIEEIG 2q2k B 3.0 BS01 dna F 0 L9 K11 L6 K8 ? remove_due_to_license_issue O87365 18097417 12 ~ 31 KETKHLLKIKKEDYPQIFDFLENVPRGTKTAHIREALRRYIEEI 2q2y A 2.5 BS02 MKR A 1 E116 E118 R119 A133 Y211 L214 E215 G217 E99 E101 R102 A116 Y194 L197 E198 G200 ? 0003777,0005524,0007018,0008017 ic50=1.6nM remove_due_to_license_issue IC50=1.6nM P52732 17766111 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2q2z A 3.0 BS02 MKK A 1 E116 E118 R119 A133 I136 P137 Y211 L214 E215 G217 E99 E101 R102 A116 I119 P120 Y194 L197 E198 G200 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue P52732 17766111 604 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2q38 A 1.95 BS02 LSA A 1 H94 H119 V121 L198 T199 T200 H91 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5950nM remove_due_to_license_issue Ki=5950nM P00918 17705204 503 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2q38 A 1.95 BS03 LSA A 2 G6 Y7 G8 F231 E239 G3 Y4 G5 F227 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5950nM remove_due_to_license_issue Ki=5950nM P00918 17705204 504 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 2q54 A 1.85 BS01 MU1 B 1 D25 G27 A28 D29 G48 G49 I50 P81 I84 D25 G27 A28 D29 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38710 17696512 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q54 B 1.85 BS01 MU1 B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=0.98nM remove_due_to_license_issue O38710 17696512 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q55 A 1.9 BS01 MU0 B 1 D25 G27 A28 D29 G48 G49 P81 I84 D25 G27 A28 D29 G48 G49 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38719 17696512 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q55 B 1.9 BS01 MU0 B 1 D25 A28 D30 I47 G48 G49 V82 D25 A28 D30 I47 G48 G49 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=2.04nM remove_due_to_license_issue O38719 17696512 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q5k A 1.95 BS01 AB1 A 1 D25 G27 A28 D29 G48 P81 I84 D25 G27 A28 D29 G48 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=0.005nM remove_due_to_license_issue O38710 17696512 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q5k B 1.95 BS01 AB1 A 1 D25 G27 A28 D29 D30 G48 G49 I50 P81 D25 G27 A28 D29 D30 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue O38710 17696512 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q63 A 2.2 BS01 1UN A 1 D25 G27 D29 N30 I50 P81 I84 D25 G27 D29 N30 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=66nM remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGRWKPKMIGGIGGFIAVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLMTQIGCTLNF 2q63 B 2.2 BS01 1UN A 1 D25 G27 G48 G49 I50 I84 D25 G27 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGRWKPKMIGGIGGFIAVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLMTQIGCTLNF 2q64 A 2.5 BS01 1UN B 1 D25 G27 N30 I50 P81 I84 D25 G27 N30 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q64 B 2.5 BS01 1UN B 1 L23 D25 G27 V32 G49 I50 I84 L23 D25 G27 V32 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=3nM remove_due_to_license_issue P03367 17977555 1001 PQITLWQRPLVTIKIGGQLKEALLDTGADNTVLEEMSLPGAWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2q6b A 2.0 BS01 HR2 A 1 R590 S661 V683 S684 D690 K692 R151 S222 V244 S245 D251 K253 E559 K691 D767 E120 K252 D328 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=0.3nM remove_due_to_license_issue P04035 17574411 3001 HEPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLVK 2q6b A 2.0 BS02 HR2 A 2 E559 C561 L562 S565 R568 K735 A751 L853 L862 E120 C122 L123 S126 R129 K296 A312 L414 L423 E559 K691 D767 E120 K252 D328 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=0.3nM remove_due_to_license_issue P04035 17574411 3002 HEPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLVK 2q6b B 2.0 BS01 HR2 A 1 E559 C561 L562 S565 R568 K735 A751 H752 L853 L862 E119 C121 L122 S125 R128 K295 A311 H312 L413 L422 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 17574411 3001 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLV 2q6b B 2.0 BS02 HR2 A 2 R590 S661 V683 S684 D690 K692 R150 S221 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 17574411 3002 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLV 2q6h A 1.85 BS04 CXX A 1 R30 Q34 F320 L400 D401 R28 Q32 F316 L396 D397 ? 0005886,0016020,0035725 ic50=250uM remove_due_to_license_issue O67854 17687333 801 VKREHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGTL 2q6h A 1.85 BS05 CXX A 2 R193 F194 I197 F350 R189 F190 I193 F346 ? 0005886,0016020,0035725 ic50=250uM remove_due_to_license_issue O67854 17687333 802 VKREHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGTL 2q70 A 1.95 BS01 DC8 A 1 E353 L384 L387 R394 F404 M421 I424 H524 E44 L75 L78 R85 F95 M112 I115 H215 ? Ki=8.3nM remove_due_to_license_issue Ki=8.3nM P03372 17614275 50 LALSLTADQMVSALLDAEPPILYSEYDPSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMVPLYDLLLEMLDAHRL 2q72 A 1.7 BS04 IXX A 1 R30 V33 Q34 A319 F320 D401 R27 V30 Q31 A314 F315 D396 ? 0005886,0016020,0035725 ic50=2090uM remove_due_to_license_issue O67854 17687333 801 KREHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGTL 2q72 A 1.7 BS05 IXX A 2 R193 F194 I197 F350 R188 F189 I192 F345 ? 0005886,0016020,0035725 ic50=2090uM remove_due_to_license_issue O67854 17687333 802 KREHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGTL 2q7m B 4.25 BS01 2CS A 2 V21 G24 F25 A27 H28 V21 G24 F25 A27 H28 ? 0002540,0002675,0004051,0004364,0004464,0004602,0005515,0005634,0005635,0005783,0005789,0006691,0008047,0016020,0019370,0019372,0019899,0031965,0042802,0044877,0050544,0070207,0071277,0098869 remove_due_to_license_issue IC50=2nM P20292 17600184 503 MDQETVGNVVLLAIVTLISVVQNGFFAHKVEHESRTQNGRSFQRTGTLAFERVYTANQNCVDAYPTFLAVLWSAGLLCSQVPAAFAGLMYLFVRQKYFVGYLGERTQSTPGYIFGKRIILFLFLMSVAGIFNYYLIFFFGSDFENYIA 2q7m B 4.25 BS02 2CS C 1 D62 A63 K116 I119 L120 F123 D62 A63 K116 I119 L120 F123 ? 0002540,0002675,0004051,0004364,0004464,0004602,0005515,0005634,0005635,0005783,0005789,0006691,0008047,0016020,0019370,0019372,0019899,0031965,0042802,0044877,0050544,0070207,0071277,0098869 remove_due_to_license_issue IC50=2nM P20292 17600184 501 MDQETVGNVVLLAIVTLISVVQNGFFAHKVEHESRTQNGRSFQRTGTLAFERVYTANQNCVDAYPTFLAVLWSAGLLCSQVPAAFAGLMYLFVRQKYFVGYLGERTQSTPGYIFGKRIILFLFLMSVAGIFNYYLIFFFGSDFENYIA 2q7m C 4.25 BS01 2CS A 1 D62 A63 I119 L120 D62 A63 I119 L120 ? 0002540,0002675,0004051,0004364,0004464,0004602,0005515,0005634,0005635,0005783,0005789,0006691,0008047,0016020,0019370,0019372,0019899,0031965,0042802,0044877,0050544,0070207,0071277,0098869 remove_due_to_license_issue IC50=2nM P20292 17600184 502 MDQETVGNVVLLAIVTLISVVQNGFFAHKVEHESRTQNGRSFQRTGTLAFERVYTANQNCVDAYPTFLAVLWSAGLLCSQVPAAFAGLMYLFVRQKYFVGYLGERTQSTPGYIFGKRIILFLFLMSVAGIFNYYLIFFFGSDFENYIAT 2q7m C 4.25 BS02 2CS C 1 V21 N23 G24 F25 A27 V21 N23 G24 F25 A27 ? 0002540,0002675,0004051,0004364,0004464,0004602,0005515,0005634,0005635,0005783,0005789,0006691,0008047,0016020,0019370,0019372,0019899,0031965,0042802,0044877,0050544,0070207,0071277,0098869 remove_due_to_license_issue IC50=2nM P20292 17600184 501 MDQETVGNVVLLAIVTLISVVQNGFFAHKVEHESRTQNGRSFQRTGTLAFERVYTANQNCVDAYPTFLAVLWSAGLLCSQVPAAFAGLMYLFVRQKYFVGYLGERTQSTPGYIFGKRIILFLFLMSVAGIFNYYLIFFFGSDFENYIAT 2q7o E 2.9 BS01 IMH E 1 A116 A117 G118 F200 E201 V217 M219 T242 N243 A116 A117 G118 F200 E201 V217 M219 T242 N243 S33 H64 H86 Y88 E89 A116 M219 S220 N243 H257 S33 H64 H86 Y88 E89 A116 M219 S220 N243 H257 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 18154341 291 MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPL 2q7y A 1.95 BS01 IGC A 1 Y73 F77 D80 L84 W133 W142 D153 T156 Y67 F71 D74 L78 W127 W136 D147 T150 ? remove_due_to_license_issue P11609 18295796 601 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 2q80 A 2.7 BS03 GRG A 1 L31 S32 D64 R73 Q126 K151 T152 L155 F156 A159 K202 L26 S27 D59 R68 Q121 K146 T147 L150 F151 A154 K191 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 remove_due_to_license_issue O95749 16698791 500 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHPDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRDDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 2q80 B 2.7 BS03 GRG B 1 L31 T53 D64 R73 Q126 K151 L155 A159 K212 L26 T48 D59 R68 Q121 K146 L150 A154 K201 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 remove_due_to_license_issue O95749 16698791 500 ETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHPDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRDDYANLHSKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMF 2q88 A 1.9 BS01 4CS A 1 E21 F24 Y60 G78 L79 F80 R85 G132 T133 E134 P172 E22 F25 Y61 G79 L80 F81 R86 G133 T134 E135 P173 ? 0033294,0051470 Kd=1.6uM remove_due_to_license_issue Q92WC8 17996893 501 RDENKLEELKEQGFARIAIANEPPFTAVGADGKVSGAAPDVAREIFKRLGVADVVASISEYGAMIPGLQAGRHDAITAGLFMKPERCAAVAYSQPILCDAEAFALKKGNPLGLKSYKDIADNPDAKIGAPGGGTEEKLALEAGVPRDRVIVVPDGQSGLKMLQDGRIDVYSLPVLSINDLVSKANDPNVEVLAPVEGAPVYCDGAAFRKGDEALRDAFDVELAKLKESGEFAKIIEPYGFSAKAAMSTTREKLCAAK 2q89 A 2.3 BS01 6CS A 1 E21 F24 Y60 G78 L79 F80 R85 G132 T133 E134 P172 E22 F25 Y61 G79 L80 F81 R86 G133 T134 E135 P173 ? 0033294,0051470 Kd=0.5uM remove_due_to_license_issue Q92WC8 17996893 501 RDENKLEELKEQGFARIAIANEPPFTAVGADGKVSGAAPDVAREIFKRLGVADVVASISEYGAMIPGLQAGRHDAITAGLFMKPERCAAVAYSQPILCDAEAFALKKGNPLGLKSYKDIADNPDAKIGAPGGGTEEKLALEAGVPRDRVIVVPDGQSGLKMLQDGRIDVYSLPVLSINDLVSKANDPNVEVLAPVEGAPVYCDGAAFRKGDEALRDAFDVELAKLKESGEFAKIIEPYGFSAKAAMSTTREKLCAAK 2q8g A 1.9 BS01 AZX A 1 Q61 F62 F65 T74 S75 F78 L79 L194 Q197 Q21 F22 F25 T34 S35 F38 L39 L152 Q155 H275 E279 K282 N283 H223 E227 K230 N231 2.7.11.2 0004672,0004740,0005515,0005524,0005739,0005759,0006006,0008283,0008631,0010510,0010906,0016301,0045254,0097411 ic50=0.087uM remove_due_to_license_issue IC50=41nM Q15118 17683942 438 GVPGQVDFYARFSPSPLSMKQFLDFGSVNACEKTSFMFLRQELPVRLANIMKEISLLPDNLLRTPSVQLVQSWYIQSLQELLDFKDKSAEDAKAIYDFTDTVIRIRNRHNDVIPTMAQGVIEYKESFDPVTSQNVQYFLDRFYMSRISIRMLLNQHSLLFGKHIGSINPNCNVLEVIKDGYENARRLCDLYYINSPELELEELNAKSPGQPIQVVYVPSHLYHMVFELFKNAMRATMEHHANRGVYPPIQVHVTLGNEDLTVKMSDRGGGVPLRKIDRLFNYMYSTAPRPRVETSRAVPLAGFGYGLPISRLYAQYFQGDLKLYSLEGYGTDAVIYIKALSTDSIERLPVYNKAAWKHYNTNDDWCVP 2q8h A 2.0 BS01 TF4 A 1 Y114 R188 I191 Y71 R143 I146 H275 E279 K282 N283 H219 E223 K226 N227 2.7.11.2 0004672,0004740,0005515,0005524,0005739,0005759,0006006,0008283,0008631,0010510,0010906,0016301,0045254,0097411 Ki=1mM remove_due_to_license_issue IC50=5100000nM Q15118 17683942 438 GVPGQVDFYARFSPSPLSMKQFLDFGSCEKTSFMFLRQELPVRLANIMKEISLLPDNLLRTPSVQLVQSWYIQSLQELLDFKDKSAEDAKAIYDFTDTVIRIRNRHNDVIPTMAQGVIEYKESFDPVTSQNVQYFLDRFYMSRISIRMLLNQHSLLFGHIGSINPNCNVLEVIKDGYENARRLCDLYYINSPELELEELNAKSPGQPIQVVYVPSHLYHMVFELFKNAMRATMEHHANRGVYPPIQVHVTLGNEDLTVKMSDRGGGVPLRKIDRLFNYMYSTAPRPRVETSRAVPLAGFGYGLPISRLYAQYFQGDLKLYSLEGYGTDAVIYIKALSTDSIERLPVYNKAAWKHYNTNADDWCVP 2q8i A 2.6 BS01 RDC A 1 N251 A255 D287 V292 L300 L328 T352 N237 A241 D273 V278 L286 L296 T320 H243 E247 K250 N251 H229 E233 K236 N237 2.7.11.2 0004672,0004674,0004740,0005515,0005524,0005730,0005739,0005759,0010510,0010906,0016301,0018105,0035357,0071333,0071398,0097411,2000377 remove_due_to_license_issue Q15120 17683942 408 PKQIERYSRFSPSPLSIKQFLDFGRDNACEKTSYMFLRKELPVRLANTMREVNLLPDNLLNRPSVGLVQSWYMQSFLELLEYENKSPEDPQVLDNFLQVLIKVRNRHNDVVPTMAQGVIEYKEKFGFDPFISTNIQYFLDRFYTNRISFRMLINQHTLLFGTNPVHPKHIGSIDPTCNVADVVKDAYETAKMLCEQYYLVAPELEVEEFNAKAPDKPIQVVYVPSHLFHMLFELFKNSMRATVELYEDRKEGYPAVKTLVTLGKEDLSIKISDLGGGVPLRKIDRLFNYMYSGYGLPISRLYARYFQGDLKLYSMEGVGTDAVIYLKALSSESFERLPVFNKSAWRHYKTTPEADDWSNPSSEPRDASK 2q8m A 2.05 BS05 AMP A 1 I8 Q12 F15 A18 T19 G20 E21 L22 K104 Y105 I8 Q12 F15 A18 T19 G20 E21 L22 K82 Y83 E89 E90 D110 L112 D113 E275 E67 E68 D88 L90 D91 E253 3.1.3.11 0000166,0000287,0005737,0005829,0005975,0006000,0006002,0006094,0016787,0016791,0030388,0032991,0042132,0042578,0042802,0046872 Ki=94uM remove_due_to_license_issue P0A993 17567577 341 MKTLGEFIVEKQHEFSHATGELTALLSAIKLGAKIIHRDINKAGLFANEKLKAALKARDIVAGIASEEEDEIVVFEGCEHAKYVVLMDPLDGSSNIDVNVSVGTIFSIYRRVTPVGTPVTEEDFLQPGNKQVAAGYVVYGSSTMLVYTTGCGVHAFTYDPSLGVFCLCQERMRFPEKGKTYSINEGNYIKFPNGVKKYIKFCQEEDKSTNRPYTSRYIGSLVADFHRNLLKGGIYLYPSTASHPDGKLRLLYECNPMAFLAEQAGGKASDGKERILDIIPETLHQRRSFFVGNDHMVEDVERFIREFPDA 2q8s A 2.3 BS01 L92 A 1 F282 G284 C285 Q286 S289 H323 Y327 M348 L353 M364 H449 Y473 F61 G63 C64 Q65 S68 H102 Y106 M127 L132 M143 H228 Y252 ? 0003677,0004879,0005634,0006355 ic50=0.185uM remove_due_to_license_issue EC50=140nM, IC50=185nM P37231 18394907 1001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 2q8z A 1.8 BS01 NUP A 1 D23 K102 N104 D136 K138 T194 T195 P264 Q269 N291 G293 R294 D30 K109 N111 D143 K145 T201 T202 P271 Q276 N298 G300 R301 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=2.1uM remove_due_to_license_issue Q8IJH3 18189347 401 GLVPRGSMGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNMES 2q8z A 1.8 BS02 NUP B 1 D141 I142 T145 D148 I149 T152 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=2.1uM remove_due_to_license_issue Q8IJH3 18189347 401 GLVPRGSMGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNMES 2q8z B 1.8 BS01 NUP A 1 D141 I142 T145 D141 I142 T145 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=2.1uM remove_due_to_license_issue Q8IJH3 18189347 401 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNM 2q8z B 1.8 BS02 NUP B 1 D23 K102 N104 D136 K138 T194 T195 P264 Q269 N291 G293 R294 D23 K102 N104 D136 K138 T194 T195 P264 Q269 N291 G293 R294 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=2.1uM remove_due_to_license_issue Q8IJH3 18189347 401 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNM 2q92 A 1.9 BS03 B23 A 1 C59 Y62 Y65 C70 D97 D108 H171 F177 H178 E204 W221 E235 C58 Y61 Y64 C69 D96 D107 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=1.1uM remove_due_to_license_issue IC50=1080nM P0AE18 18093325 400 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 2q93 A 1.6 BS03 B21 A 1 Y62 Y65 H79 D97 D108 H171 H178 E204 E235 Y61 Y64 H78 D96 D107 H170 H177 E203 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.56uM remove_due_to_license_issue IC50=>200000nM P0AE18 18093325 400 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2q94 A 1.63 BS03 A04 A 1 C59 Y62 Y65 H79 D97 D108 H171 H178 E204 W221 E235 C58 Y61 Y64 H78 D96 D107 H170 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=0.37uM remove_due_to_license_issue IC50=197000nM P0AE18 18093325 400 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 2q95 A 1.7 BS03 A05 A 1 Y62 H63 H79 D97 D108 H171 H178 E204 W221 E235 Y61 H62 H78 D96 D107 H170 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=1.6uM remove_due_to_license_issue IC50=48600nM P0AE18 18093325 400 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2q96 A 1.6 BS03 A18 A 1 C59 Y62 Y65 H79 D97 D108 H171 H178 E204 W221 E235 C58 Y61 Y64 H78 D96 D107 H170 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=1.2uM remove_due_to_license_issue IC50=158000nM P0AE18 18093325 400 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2q9m A 2.05 BS01 LK7 A 1 S64 N152 G317 S318 S63 N151 G316 S317 S64 K67 Y112 V121 Y150 G156 E272 K315 S318 S63 K66 Y111 V120 Y149 G155 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P05364 17665896 0 PVSEKQLAEVVANTITPLMKAQSVPGMAVAVIYQGKPHYYTFGKADIAANKPVTPQTLFELGSISKTFTGVLGGDAIARGEISLDDAVTRYWPQLTGKQWQGIRMLDLATYTAGGLPLQVPDEVTDNASLLRFYQNWQPQWKPGTTRLYANASIGLFGALAVKPSGMPYEQAMTTRVLKPLKLDHTWINVPKAEEAHYAWGYRDGKAVRVSPGMLDAQAYGVKTNVQDMANWVMANMAPENVADASLKQGIALAQSRYWRIGSMYQGLGWEMLNWPVEANTVVEGSDSKVALAPLPVAEVNPPAPPVKASWVHKTGSTGGFGSYVAFIPEKQIGIVMLANTSYPNPARVEAAYHILEAL 2q9n A 2.2 BS01 LK5 A 1 S64 L119 Q120 Y150 N152 R204 Y221 G317 S318 T319 G320 S63 L118 Q119 Y149 N151 R203 Y220 G316 S317 T318 G319 S64 K67 Y112 V121 Y150 G156 E272 K315 S318 S63 K66 Y111 V120 Y149 G155 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P05364 17665896 0 PVSEKQLAEVVANTITPLMKAQSVPGMAVAVIYQGKPHYYTFGKADIAANKPVTPQTLFELGSISKTFTGVLGGDAIARGEISLDDAVTRYWPQLTGKQWQGIRMLDLATYTAGGLPLQVPDEVTDNASLLRFYQNWQPQWKPGTTRLYANASIGLFGALAVKPSGMPYEQAMTTRVLKPLKLDHTWINVPKAEEAHYAWGYRDGKAVRVSPGMLDAQAYGVKTNVQDMANWVMANMAPENVADASLKQGIALAQSRYWRIGSMYQGLGWEMLNWPVEANTVVEGSDSKVALAPLPVAEVNPPAPPVKASWVHKTGSTGGFGSYVAFIPEKQIGIVMLANTSYPNPARVEAAYHILEAL 2q9y B 2.85 BS03 BTM B 1 L97 R182 G186 L187 M221 Y295 W298 L95 R180 G184 L185 M219 Y293 W296 Y93 T96 L97 D100 R182 K232 R304 Y305 Y91 T94 L95 D98 R180 K230 R302 Y303 4.2.3.6 0016106,0016829,0016838,0045482,0046872 remove_due_to_license_issue P13513 17678871 704 NFPTEYFLNTTVRLLEYIRYRDSNYTREERIENLHYAYNKAAHHFAQPRQQQLLKVDPKRLQASLQTIVGMVVYSWAKVSKECMADLSIHYTYTLVLDDSKDDPYPTMVNYFDDLQAGREQAHPWWALVNEHFPNVLRHFGPFCSLNLIRSTLDFFEGCWIEQYNFGGFPGSHDYPQFLRRMNGLGHCVGASLWPKEQFNERSLFLEITSAIAQMENWMVWVNDLMSFYKEFDDERDQISLVKNYVVSDEISLHEALEKLTQDTLHSSKQMVAVFSDKDPQVMDTIECFMHGYVTWHLCDRRYRLSEIYEKVKEEKTEDAQKFCKFYEQAANVGAVSPSEWAYPPVAQLANV 2qa8 A 1.85 BS02 GEN A 1 M343 L346 A350 E353 L387 M421 H524 L525 M33 L36 A40 E43 L77 M111 H206 L207 ? remove_due_to_license_issue IC50=395nM, EC50=240nM, Ki=370nM P03372 18344977 600 SLALSLTADQMVSALLDAEPPILYSEFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 2qbp A 2.5 BS01 527 A 1 R24 S28 D29 Y46 V49 K120 F182 S216 I219 R221 G259 Q262 R23 S27 D28 Y45 V48 K119 F181 S215 I218 R220 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.004uM remove_due_to_license_issue Ki=4nM P18031 17705360 800 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2qbq A 2.1 BS01 4B3 A 1 R24 Y46 V49 K120 F182 I219 R221 M258 Q262 R23 Y45 V48 K119 F181 I218 R220 M257 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.036uM remove_due_to_license_issue Ki=36nM P18031 17705360 800 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2qbr A 2.3 BS01 910 A 1 Y46 D48 K120 F182 A217 I219 R221 G259 Q262 Y45 D47 K119 F181 A216 I218 R220 G258 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.47uM remove_due_to_license_issue Ki=470nM P18031 17705360 800 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 2qbs A 2.1 BS01 024 A 1 Y46 V49 K120 F182 I219 R221 Q262 Y45 V48 K119 F181 I218 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=0.21uM remove_due_to_license_issue Ki=210nM P18031 17705360 800 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2qbu A 2.1 BS01 SAH B 1 L102 G103 D104 I107 Y108 T132 S133 M175 K176 N202 C203 Y220 L221 A222 T223 L102 G103 D104 I107 Y108 T132 S133 M175 K176 N202 C203 Y220 L221 A222 T223 ? 0008168,0008757,0009236,0030788,0032259 remove_due_to_license_issue O27402 17567575 501 MHGKLIGVGVGPGDSELLTLRAVNVLRSVPVICAPRSSSERESIALSIVEDILTERRDGCRILDPVFPMTDDRDELESHWDSAARMVAAELEDGRDVAFITLGDPSIYSTFSYLQQRIEDMGFKTEMVPGVTSFTACAATAGRTLVEGDEILLVVPRVDDRFERVLRDVDACVIMKTSRHGRRAMEVVESDPRGKDVVSVANCSMDDEVVERGFASGGGYLATTLVRF 2qbu B 2.1 BS01 SAH B 2 P12 L102 G103 D104 I107 Y108 T132 S133 M175 K176 C203 Y220 L221 A222 T223 P12 L102 G103 D104 I107 Y108 T132 S133 M175 K176 C203 Y220 L221 A222 T223 ? 0008168,0008757,0009236,0030788,0032259 Kd=0.645uM remove_due_to_license_issue O27402 17567575 502 MHGKLIGVGVGPGDSELLTLRAVNVLRSVPVICAPRSSSERESIALSIVEDILTERRDGCRILDPVFPMTDDRDELESHWDSAARMVAAELEDGRDVAFITLGDPSIYSTFSYLQQRIEDMGFKTEMVPGVTSFTACAATAGRTLVEGDEILLVVPRVDDRFERVLRDVDACVIMKTSRHGRRAMEVVESDPRGKDVVSVANCSMDDEVVERGFASGGGYLATTLVRF 2qc6 A 1.85 BS01 G12 A 1 V53 I66 K68 F113 V116 M163 I174 D175 V47 I60 K62 F107 V110 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=0.1uM remove_due_to_license_issue P28523 18251491 1 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 2qcd A 2.03 BS01 U5P A 1 S257 D259 K281 H283 K314 M371 S372 P417 Q430 Y432 G450 R451 S36 D38 K60 H62 K93 M150 S151 P196 Q209 Y211 G229 R230 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 1 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcd A 2.03 BS02 U5P B 1 D317 I318 T321 D96 I97 T100 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 2 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcd B 2.03 BS01 U5P A 1 D317 I318 T321 D96 I97 T100 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 1 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcd B 2.03 BS02 U5P B 1 S257 D259 H283 K314 M371 S372 P417 Q430 Y432 G450 R451 S36 D38 H62 K93 M150 S151 P196 Q209 Y211 G229 R230 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 2 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcf A 1.22 BS01 5FU A 1 S257 D259 K281 H283 N312 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 N90 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue Ki=98000nM P11172 18184586 501 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcg A 1.75 BS01 5BU A 1 S257 D259 K281 H283 D312 M371 S372 P417 Q430 Y432 G450 R451 S36 D38 K60 H62 D91 M150 S151 P196 Q209 Y211 G229 R230 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 1 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcg A 1.75 BS02 5BU B 1 D317 I318 T321 D96 I97 T100 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 2 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcg B 1.75 BS01 5BU A 1 D317 T321 D96 T100 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 1 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qcg B 1.75 BS02 5BU B 1 S257 D259 K281 H283 D312 K314 I368 M371 S372 P417 Q430 Y432 G450 R451 S36 D38 K60 H62 D91 K93 I147 M150 S151 P196 Q209 Y211 G229 R230 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 2 AMELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qch A 1.95 BS02 5IU A 1 D259 K314 I368 M371 S372 P417 Q430 Y432 G450 R451 D36 K91 I145 M148 S149 P194 Q207 Y209 G227 R228 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 1 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 2qch A 1.95 BS04 5IU B 1 D317 I318 T321 D94 I95 T98 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 3 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 2qch B 1.95 BS01 5IU A 1 D317 I318 T321 D94 I95 T98 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 1 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 2qch B 1.95 BS04 5IU B 1 D259 K281 K314 I368 M371 P417 Q430 Y432 V449 G450 R451 D36 K58 K91 I145 M148 P194 Q207 Y209 V226 G227 R228 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 3 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 2qci A 1.2 BS01 065 B 1 D25 A28 N30 P81 D25 A28 N30 P81 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADNTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2qci B 1.2 BS01 065 B 1 D125 G127 D129 N130 G148 G149 I150 D25 G27 D29 N30 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.6nM remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADNTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2qcm A 1.67 BS01 JW5 A 1 S257 D259 H283 N312 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 H61 N90 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 18184586 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 2qd6 A 1.28 BS01 065 B 1 D25 A28 D30 P81 D25 A28 D30 P81 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2qd6 B 1.28 BS01 065 B 1 D125 G127 D129 D130 G148 G149 V150 D25 G27 D29 D30 G48 G49 V50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2.1nM remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2qd7 A 1.11 BS01 065 B 1 D25 A28 D30 P81 I84 D25 A28 D30 P81 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2qd7 B 1.11 BS01 065 B 1 D125 G127 A128 D129 D130 G148 I150 D25 G27 A28 D29 D30 G48 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.8nM remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 2qd8 A 1.35 BS01 065 B 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2qd8 B 1.35 BS01 065 B 1 D125 G127 D129 G148 G149 I150 D25 G27 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.85nM remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 2qd9 A 1.7 BS01 LGF A 1 V30 A51 K53 L104 T106 M109 G110 A111 A157 L167 V26 A45 K47 L98 T100 M103 G104 A105 A148 L158 D150 K152 N155 D168 D141 K143 N146 D159 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=13nM remove_due_to_license_issue IC50=13nM Q16539 17664068 361 RPTFYRQELNKTIWEVPERYQNLSPVGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2qdt A 2.0 BS03 I38 A 1 D88 H160 S187 P189 D87 H159 S186 P188 H84 H86 D88 H89 H160 Y191 H225 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=6.5uM remove_due_to_license_issue P52700 18563261 501 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 2qe2 A 2.9 BS01 452 A 1 P197 R200 C366 R386 G410 N411 M414 Y415 Q446 Y448 P161 R164 C328 R348 G372 N373 M376 Y377 Q408 Y410 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q99AU2 17402724 579 LLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAFGYGAKDVRNLSSKAVNHIHSVWKDLLEDPIDTTIMAKNEVFCVQPEGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASLSGWFVAGYSGGDIYH 2qe4 A 2.4 BS01 JJ3 A 1 T347 A350 E353 W383 M421 I424 H524 L525 T37 A40 E43 W73 M111 I114 H203 L204 ? Ki=11nM remove_due_to_license_issue Ki=11nM P03372 17662603 601 LALSLTADQMVSALLDAEPPILYSEPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSM 2qe5 A 2.6 BS01 617 A 1 P197 R200 C366 L384 G410 N411 M414 Y415 Q446 I447 Y448 P197 R200 C366 L384 G410 N411 M414 Y415 Q446 I447 Y448 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q99AU2 17402724 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASLSGWFVAGYSGGDIYH 2qf6 A 3.1 BS01 A56 A 1 A55 M98 N106 L107 F138 T184 A39 M82 N90 L91 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Ki=3.2e+2nM, Kd=<1.0e+4nM P07900 17630989 256 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2qfo A 1.68 BS01 A13 A 1 A55 G97 M98 A39 G81 M82 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=20uM remove_due_to_license_issue Ki=1.8e+4nM, Kd=2.0e+4nM P07900 17630989 900 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2qft A 1.55 BS01 GPJ A 1 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 remove_due_to_license_issue P0A6D3 17855366 801 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRSLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 2qfu A 1.6 BS01 GPJ A 1 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 remove_due_to_license_issue P0A6D3 17855366 801 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGTAMRLLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 2qg0 A 1.85 BS01 A94 A 1 N51 D54 A55 I96 G97 M98 N106 G135 V136 F138 N35 D38 A39 I80 G81 M82 N90 G119 V120 F122 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=1.9uM remove_due_to_license_issue P07900 17630989 2001 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2qg0 B 1.85 BS01 A94 B 1 N51 D54 A55 K58 I96 M98 N106 G135 V136 F138 Y139 N35 D38 A39 K42 I80 M82 N90 G119 V120 F122 Y123 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=1.9uM remove_due_to_license_issue P07900 17630989 2002 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2qg2 A 1.8 BS01 A91 A 1 A55 G97 L103 L107 F138 W162 A39 G81 L87 L91 F122 W146 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=4uM remove_due_to_license_issue P07900 17630989 300 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2qh6 A 2.7 BS02 ODE A 1 M343 T347 E353 F404 M421 F425 G521 H524 L525 M38 T42 E48 F99 M116 F120 G206 H209 L210 ? remove_due_to_license_issue P03372 18344977 700 NSLALSLTADQMVSALLDAEPPILYSEYDRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVPLSDLLLEMLDAHR 2qhc A 2.802 BS01 AB1 B 1 D25 A28 D30 G49 I50 D25 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q9J2P7 18560011 9001 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMAGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qhc B 2.802 BS01 AB1 B 1 D25 G27 A28 D29 G48 G49 D25 G27 A28 D29 G48 G49 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q9J2P7 18560011 9001 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMAGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qhd A 1.95 BS01 DAO A 1 G30 C45 H48 G29 C44 H47 F28 G30 G32 H48 S49 Y52 Y73 D99 F27 G29 G31 H47 S48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0042130,0047498,0050482 remove_due_to_license_issue P48650 18586854 501 SVVELGKMIIQETGKSPFPSYTSYGCFCGGGERGPPLDATDRCCLAHSCCYDTLPDCSPKTDRYKYKRENGEIICENSTSCKKRICECDKAVAVCLRKNLNTYNKKYTYYPNFWCKGDIEKC 2qhd B 1.95 BS01 DAO B 1 G30 C45 H48 S49 G29 C44 H47 S48 F28 G30 G32 H48 S49 Y52 Y73 D99 F27 G29 G31 H47 S48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0042130,0047498,0050482 remove_due_to_license_issue P48650 18586854 502 SVVELGKMIIQETGKSPFPSYTSYGCFCGGGERGPPLDATDRCCLAHSCCYDTLPDCSPKTDRYKYKRENGEIICENSTSCKKRICECDKAVAVCLRKNLNTYNKKYTYYPNFWCKGDIEKC 2qhm A 2.0 BS01 7CS A 1 L15 V23 A36 E85 C87 E134 N135 L137 S147 L14 V18 A31 E73 C75 E122 N123 L125 S135 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=660nM remove_due_to_license_issue O14757 17804227 500 AVPFVEDWDLVQTLGGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2qhn A 1.7 BS01 582 A 1 L15 G16 A36 E85 Y86 C87 G90 L137 L14 G15 A31 E73 Y74 C75 G78 L125 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=980nM remove_due_to_license_issue O14757 17804227 500 AVPFVEDWDLVQTLGGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2qhy A 1.85 BS01 MZ1 A 1 D25 G27 A28 D29 G48 G49 I50 V82 I84 D25 G27 A28 D29 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=33nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qhy B 1.85 BS01 MZ1 A 1 D25 A28 D30 G48 P81 V82 I84 D25 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qhz A 1.85 BS01 MZ2 A 1 D25 G27 A28 D30 G48 I50 P81 V82 D25 G27 A28 D30 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=53nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qhz B 1.85 BS01 MZ2 A 1 D25 A28 D30 G48 P81 V82 I84 D25 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi0 A 2.1 BS01 MZ3 B 1 D25 G27 A28 D30 G48 I50 V82 I84 D25 G27 A28 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi0 B 2.1 BS01 MZ3 B 1 D25 A28 D30 I47 G49 I50 P81 V82 I84 D25 A28 D30 I47 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=42nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi1 A 2.0 BS01 MZ4 A 1 D25 G27 A28 D30 G48 G49 I50 P81 V82 I84 D25 G27 A28 D30 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=50nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi1 B 2.0 BS01 MZ4 A 1 D25 A28 D30 I47 G49 I50 V82 D25 A28 D30 I47 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi3 A 1.95 BS01 MZ5 B 1 D25 G27 A28 G48 D25 G27 A28 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi3 B 1.95 BS01 MZ5 B 1 D25 A28 D30 G48 D25 A28 D30 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.063nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi4 A 1.8 BS01 MZ6 A 1 D25 G27 D29 D30 I50 V82 D25 G27 D29 D30 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.036nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi4 B 1.8 BS01 MZ6 A 1 D25 A28 D30 I50 P81 V82 D25 A28 D30 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi5 A 1.85 BS01 MZ7 B 1 D25 G27 A28 D29 G48 G49 I50 P81 V82 D25 G27 A28 D29 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi5 B 1.85 BS01 MZ7 B 1 D25 G27 A28 D30 G48 I50 P81 V82 D25 G27 A28 D30 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.014nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi6 A 1.85 BS01 MZ8 A 1 D25 G27 D29 D30 I50 D25 G27 D29 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.027nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi6 B 1.85 BS01 MZ8 A 1 D25 A28 D30 G48 I50 P81 V82 D25 A28 D30 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi7 A 1.85 BS01 MZ9 B 1 D25 G27 D29 G48 G49 I50 V82 D25 G27 D29 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qi7 B 1.85 BS01 MZ9 B 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.062nM remove_due_to_license_issue P03369 18412349 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qiq A 1.9 BS01 CYV A 1 T26 H41 F140 L141 N142 C145 H163 H164 M165 E166 P168 D187 Q189 T190 Q192 T26 H41 F140 L141 N142 C145 H163 H164 M165 E166 P168 D187 Q189 T190 Q192 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=80uM remove_due_to_license_issue IC50=80000nM P0C6X7 17855091 302 AGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCS 2qju A 2.9 BS02 DSM A 1 R30 Q34 A319 F320 D401 R26 Q30 A313 F314 D395 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 17690258 801 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 2qk5 A 2.2 BS01 CS5 A 1 G72 L91 D93 G95 S96 Y132 T133 Q134 F169 Y259 D289 G291 T293 G20 L39 D41 G43 S44 Y80 T81 Q82 F117 Y207 D237 G239 T241 D93 S96 N98 A100 Y132 D289 T292 D41 S44 N46 A48 Y80 D237 T240 3.4.23.46 0004190,0006508,0016020 ic50=8nM remove_due_to_license_issue IC50=20nM P56817 18023580 1 AAGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2qk8 A 2.4 BS01 MTX A 1 M6 V7 A8 E28 L29 V32 I51 R53 L55 R58 F96 M6 V7 A8 E28 L29 V32 I51 R53 L55 R58 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 ic50~20nM remove_due_to_license_issue IC50=15nM Q81R22 17696333 200 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQ 2ql2 A 2.5 BS01 dna E 0 R550 E551 R554 R8 E9 R12 ? 0046983 remove_due_to_license_issue P15806 18069799 1 ~ 16 RRMANNARERVRVRDINEAFRELGRMCQLHLKAQTKLLILQQAVQVILGLEQQVRE 2ql2 A 2.5 BS02 dna F 0 R544 N548 E551 R552 N559 T580 K581 R2 N6 E9 R10 N17 T35 K36 ? 0046983 remove_due_to_license_issue P15806 18069799 20 ~ 35 RRMANNARERVRVRDINEAFRELGRMCQLHLKAQTKLLILQQAVQVILGLEQQVRE 2ql2 B 2.5 BS01 dna E 0 N107 R111 S138 K139 N7 R11 S38 K39 ? 0046983 remove_due_to_license_issue Q60867 18069799 1 ~ 16 SRRMKANARERNRMHGLNAALDNLRKVVPCYSKTQKLSKIETLRLAKNYIWALSEILRS 2ql2 B 2.5 BS02 dna F 0 E110 R113 E10 R13 ? 0046983 remove_due_to_license_issue Q60867 18069799 20 ~ 35 SRRMKANARERNRMHGLNAALDNLRKVVPCYSKTQKLSKIETLRLAKNYIWALSEILRS 2ql2 C 2.5 BS01 dna G 0 R550 R554 R8 R12 ? 0046983 remove_due_to_license_issue P15806 18069799 1 ~ 16 RRMANNARERVRVRDINEAFRELGRMCQLHLKSDQTKLLILQQAVQVILGLEQQVRER 2ql2 C 2.5 BS02 dna H 0 N548 T580 K581 N6 T36 K37 ? 0046983 remove_due_to_license_issue P15806 18069799 20 ~ 35 RRMANNARERVRVRDINEAFRELGRMCQLHLKSDQTKLLILQQAVQVILGLEQQVRER 2ql2 D 2.5 BS01 dna G 0 N107 E110 R111 K139 N6 E9 R10 K38 ? 0046983 remove_due_to_license_issue Q60867 18069799 1 ~ 16 RRMKANARERNRMHGLNAALDNLRKVVPCYSKTQKLSKIETLRLAKNYIWALSEILR 2ql2 D 2.5 BS02 dna H 0 E110 R113 E9 R12 ? 0046983 remove_due_to_license_issue Q60867 18069799 20 ~ 35 RRMKANARERNRMHGLNAALDNLRKVVPCYSKTQKLSKIETLRLAKNYIWALSEILR 2qlm A 2.1 BS01 F68 A 1 G135 L136 N282 D283 H377 N484 E672 S674 G675 G124 L125 N265 D266 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=2300nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qln A 2.15 BS01 F59 A 1 E88 G135 L136 N282 D283 R292 H341 H377 E385 N484 E672 S674 G675 E77 G124 L125 N265 D266 R275 H315 H351 E359 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=3700nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qlq A 2.33 BS01 SR2 A 1 V281 A293 K295 T338 M341 C345 D348 L393 D404 V26 A38 K40 T69 M72 C76 D79 L124 D135 D386 R388 A390 N391 D404 D117 R119 A121 N122 D135 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>27000nM P00523 18316192 1345 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLAQVMKKLRHEKLVQLYAVVSEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2qlq A 2.33 BS02 SR2 A 2 C483 P484 E486 C487 E489 C195 P196 E198 C199 E201 D386 R388 A390 N391 D404 D117 R119 A121 N122 D135 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>27000nM P00523 18316192 1483 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLAQVMKKLRHEKLVQLYAVVSEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2qm7 A 1.85 BS01 GDP A 1 G65 V66 G67 K68 S69 T70 N201 K202 D204 S241 L243 G61 V62 G63 K64 S65 T66 N188 K189 D191 S228 L230 ? 0003924,0005525,0005737 remove_due_to_license_issue Q8RPA0 17728257 601 LPDMDTLRERLLAGDRAALARAITLAESRRADHRAAVRDLIDAVLPQTGRAIRVGITGVPGVGKSTTIDALGSLLTAAGHKVAVLAVDPSSTRTRMARLAIDRNAFIRPSPSSGTLGGVAAKTRETMLLCEAAGFDVILVETVGVGQSETAVADLTDFFLVLMLPGAGDELQGIKKGIFELADMIAVNKADDGDGERRASAAASEYRAALHILTPPSATWTPPVVTISGLHGKGLDSLWSRIEDHRSKLTATGEIAGKRREQDVKWMWALVHERLHQRLVGSAEVRQATAEAERAVAGGEHSPAAGADAIATLI 2qm9 A 2.31 BS01 TDZ A 1 P38 S53 S55 F57 K58 T60 D76 R126 Y128 P46 S61 S63 F65 K66 T68 D84 R134 Y136 ? 0005324,0005634,0005654,0005737,0008289,0009617,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0071285,0071356,0120162 Kd=17nM remove_due_to_license_issue P04117 17761196 201 SSSKVYKMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDLVTIRSESTFKNTEISFKLGVEFDEITADDRKVKSIITLDGGALVQVQKWDGKSTTIKRKRDGDKLVVECVMKGVTSTRVYERA 2qm9 B 2.31 BS01 TDZ B 1 Y19 P38 S53 S55 K58 T60 A75 R78 I104 R126 Y128 Y20 P39 S54 S56 K59 T61 A76 R79 I105 R127 Y129 ? 0005324,0005634,0005654,0005737,0008289,0009617,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0071285,0071356,0120162 Kd=17nM remove_due_to_license_issue P04117 17761196 202 MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDLVTIRSESTFKNTEISFKLGVEFDEITADDRKVKSIITLDGGALVQVQKWDGKSTTIKRKRDGDKLVVECVMKGVTSTRVYERA 2qmd A 1.65 BS01 CS7 A 1 G72 D93 G95 S96 P131 Y132 T133 Q134 G135 F169 Y259 D289 G291 T293 G15 D36 G38 S39 P74 Y75 T76 Q77 G78 F112 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=5nM remove_due_to_license_issue IC50=150nM P56817 18023580 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2qmf A 1.75 BS01 CS9 A 1 G72 Q73 D93 G95 S96 Y132 T133 Q134 G135 F169 I171 R189 Y259 D289 G291 T293 G15 Q16 D36 G38 S39 Y75 T76 Q77 G78 F112 I114 R132 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=3nM remove_due_to_license_issue IC50=165nM P56817 18023580 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2qmg A 1.89 BS01 SC6 A 1 G72 L91 D93 G95 Y132 T133 Q134 F169 I171 R189 D289 G291 T292 T293 R296 G15 L34 D36 G38 Y75 T76 Q77 F112 I114 R132 D232 G234 T235 T236 R239 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=0.7nM remove_due_to_license_issue P56817 17980584 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2qn1 A 2.401 BS01 0AS A 1 I68 Q71 Q72 R310 I57 Q60 Q61 R293 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue IC50=17000nM P00489 18517260 930 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qn2 A 2.698 BS01 0MA A 1 Q71 Q72 F196 R309 R310 Q60 Q61 F185 R292 R293 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 18517260 930 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qn3 A 1.96 BS01 F55 A 1 G135 L136 N282 D283 H377 N484 E672 A673 S674 G675 G124 L125 N268 D269 H354 N461 E649 A650 S651 G652 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=4400nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qnb A 1.8 BS01 BZD A 1 G135 L136 D283 H377 N484 E672 A673 S674 G675 G124 L125 D266 H351 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=4600nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 2qnb A 1.8 BS02 BZD A 2 R60 W189 E190 K191 P229 R49 W178 E179 K180 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=4600nM P00489 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 2qnn A 1.48 BS01 QN1 B 1 D25 G27 A28 D30 G48 I50 V82 I84 D25 G27 A28 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qnn B 1.48 BS01 QN1 B 1 R8 L23 D25 A28 D29 D30 G48 G49 I50 P81 R8 L23 D25 A28 D29 D30 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.07uM remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qnp A 1.41 BS01 QN2 A 1 D25 G27 A28 D30 I50 V82 I84 D25 G27 A28 D30 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.39uM remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qnp B 1.41 BS01 QN2 A 1 L23 D25 G27 G48 G49 I50 P81 I84 L23 D25 G27 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qnq A 2.3 BS01 QN3 A 1 D25 G27 A28 D30 G48 I50 V82 I84 D25 G27 A28 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.77uM remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qnq B 2.3 BS01 QN3 A 1 D25 A28 G48 G49 I50 P81 I84 D25 A28 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18348517 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2qnx A 2.7 BS01 UDT A 1 C112 H244 N274 C122 H258 N289 2.3.1.301 0000062,0004315,0005515,0005737,0006633,0008610,0016746,0030497,0033818,0035336,0061990 remove_due_to_license_issue P9WNG3 18420147 860 MTEIATTSGARSVGLLSVGAYRPERVVTNDEICQHIDSSDEWIYTRTGIKTRRFAADDESAASMATEACRRALSNAGLSAADIDGVIVTTNTHFLQTPPAAPMVAASLGAKGILGFDLSAGCAGFGYALGAAADMIRGGGAATMLVVGTEKLSPTIDMYDRGNCFIFADGAAAVVVGETPFQGIGPTVAGSDGEQADAIRQDIDWITFAQNPSGPRPFVRLEGPAVFRWAAFKMGDVGRRAMDAAGVRPDQIDVFVPHQANSRINELLVKNLQLRPDAVVANDIEHTGNTSAASIPLAMAELLTTGAAKPGDLALLIGYGAGLSYAAQVVRMPK 2qnx B 2.7 BS01 UDT B 1 I189 L207 H244 A246 N274 I197 L219 H256 A258 N287 2.3.1.301 0000062,0004315,0005515,0005737,0006633,0008610,0016746,0030497,0033818,0035336,0061990 remove_due_to_license_issue P9WNG3 18420147 860 MTEIATTSGARSVGLLSVGAYRPERVVTNDEICIDSSDEWIYTRTGIKTRRFAADDESAASMATEACRRALSNAGLSAADIDGVIVTTNTHFLQTPPAAPMVAASLGAKGILGFDLSAGCAGFGYALGAAADMIRGGGAATMLVVGTEKLSPTIDMYDRGNCFIFADGAAAVVVGETPFQGIGPTVAGSDGEQADAIRQDIDWITFAQNPSGPRPFVRLEGPAVFRWAAFKMGDVGRRAMDAAGVRPDQIDVFVPHQANSRINELLVKNLQLRPDAVVANDIEHTGNTSAASIPLAMAELLTTGAAKPGDLALLIGYGAGLSYAAQVVRMPK 2qnz A 2.3 BS01 DFD A 1 C112 L142 T145 Q191 P203 F204 V205 S276 G305 A306 C118 L148 T151 Q197 P213 F214 V215 S287 G316 A317 2.3.1.301 0000062,0004315,0005515,0005737,0006633,0008610,0016746,0030497,0033818,0035336,0061990 remove_due_to_license_issue P9WNG3 18420147 760 MTEIATTSGARSVGLLSVGAYRPERVVTNDEICQSDEWIYTRTGIKTRRFAADDESAASMATEACRRALSNAGLSAADIDGVIVTTNTHFLQTPPAAPMVAASLGAKGILGFDLSAGCAGFGYALGAAADMIRGGGAATMLVVGTEKLSPTIDMYDRGNCFIFADGAAAVVVGETPFQGIGPTVAGSDGEQADAIRQDIDWITFAQNPSGPRPFVRLEGPAVFRWAAFKMGDVGRRAMDAAGVRPDQIDVFVPHQANSRINELLVKNLQLRPDAVVANDIEHTGNTSAASIPLAMAELLTTGAAKPGDLALLIGYGAGLSYAAQVVRMPK 2qnz B 2.3 BS01 DFD B 1 C112 T145 I189 Q191 V205 S276 A306 C117 T150 I194 Q196 V214 S286 A316 2.3.1.301 0000062,0004315,0005515,0005737,0006633,0008610,0016746,0030497,0033818,0035336,0061990 remove_due_to_license_issue P9WNG3 18420147 760 MTEIATTSGARSVGLLSVGAYRPERVVTNDEICSDEWIYTRTGIKTRRFAADDESAASMATEACRRALSNAGLSAADIDGVIVTTNTHFLQTPPAAPMVAASLGAKGILGFDLSAGCAGFGYALGAAADMIRGGGAATMLVVGTEKLSPTIDMYDRGNCFIFADGAAAVVVGETPFQGIGPTVAGSDGEQADAIRQDIDWITFAQNPSGPRPFVRLEGPAVFRWAAFKMGDVGRRAMDAAGVRPDQIDVFVPHQANSRINELLVKNLQLRPDAVVANDIEHTGNTSAASIPLAMAELLTTGAAKPGDLALLIGYGAGLSYAAQVVRMPK 2qo1 A 2.6 BS01 VZZ A 1 W32 V212 A246 W42 V226 A260 2.3.1.301 0000062,0004315,0005515,0005737,0006633,0008610,0016746,0030497,0033818,0035336,0061990 remove_due_to_license_issue P9WNG3 18420147 760 MTEIATTSGARSVGLLSVGAYRPERVVTNDEICQHIDSSDEWIYTRTGIKTRRFAADDESAASMATEACRRALSNAGLSAADIDGVIVTTNTHFLQTPPAAPMVAASLGAKGILGFDLSAGCAGFGYALGAAADMIRGGGAATMLVVGTEKLSPTIDMYDRGNCFIFADGAAAVVVGETPFQGIGPTVAGSDGEQADAIRQDIDWITFAQNPSGPRPFVRLEGPAVFRWAAFKMGDVGRRAMDAAGVRPDQIDVFVPHQANSRINELLVKNLQLRPDAVVANDIEHTGNTSAASIPLAMAELLTTGAAKPGDLALLIGYGAGLSYAAQVVRMPK 2qo8 A 1.4 BS02 3CC A 1 H94 H119 V121 F131 L198 T199 H93 H118 V120 F129 L196 T197 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.4nM remove_due_to_license_issue Ki=0.9nM P00918 18161740 800 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2qoa A 1.6 BS02 MAJ A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=52nM remove_due_to_license_issue Ki=52nM P00918 18161740 800 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2qoa A 1.6 BS03 MAJ A 2 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=52nM remove_due_to_license_issue Ki=52nM P00918 18161740 801 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2qoe A 2.3 BS01 448 A 1 E205 E206 F357 S630 Y631 Y662 Y666 N710 V711 E167 E168 F319 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=25nM remove_due_to_license_issue IC50=25nM P27487 17827003 1282 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2qoh A 1.95 BS01 P3Y A 1 G249 Y253 V256 A269 V299 T315 M318 G321 N322 L370 G22 Y26 V29 A42 V69 T85 M88 G91 N92 L140 D363 A365 R367 N368 D381 P402 D133 A135 R137 N138 D151 P172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 17718712 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESS 2qp6 A 1.45 BS02 MB1 A 1 H64 H94 H119 L198 T199 T200 H62 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=208nM remove_due_to_license_issue P00918 18481843 800 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2qp8 A 1.5 BS01 SC7 A 1 G72 D93 G95 Y132 T133 Q134 F169 Y259 D289 G291 T293 G15 D36 G38 Y75 T76 Q77 F112 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=8nM remove_due_to_license_issue IC50=106nM P56817 18023580 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 2qpj A 2.05 BS02 I20 A 1 F106 N542 A543 F544 Y545 S547 V580 H583 E584 H587 E646 W693 H711 R717 F53 N489 A490 F491 Y492 S494 V527 H530 E531 H534 E593 W640 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 remove_due_to_license_issue P08473 17704566 755 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 2qpu A 1.7 BS04 QPU A 1 Y380 H395 D398 Y380 H395 D398 D180 E205 D291 D180 E205 D291 3.2.1.1 0004556,0005509,0005576,0005975,0005983,0016798,0043169,0046872 remove_due_to_license_issue P00693 17803687 3000 HQVLFQGFNWESWKQSGGWYNMMMGKVDDIAAAGVTHVWLPPPSHSVSNEGYMPGRLYDIDASKYGNAAELKSLIGALHGKGVQAIADIVINHRCADYKDSRGIYCIFEGGTSDGRLDWGPHMICRDDTKYSDGTANLDTGADFAAAPDIDHLNDRVQRELKEWLLWLKSDLGFDAWRLDFARGYSPEMAKVYIDGTSPSLAVAEVWDNMATGGDGKPNYDQDAHRQNLVNWVDKVGGAASAGMVFDFTTKGILNAAVEGELWRLIDPQGKAPGVMGWWPAKAVTFVDNHDTGSTQAMWPFPSDKVMQGYAYILTHPGIPCIFYDHFFNWGFKDQIAALVAIRKRNGITATSALKILMHEGDAYVAEIDGKVVVKIGPRYDVGAVIPAGFVTSAHGNDYAVWEK 2qpu A 1.7 BS05 QPU A 2 Q227 D234 W278 W279 Q227 D234 W278 W279 D180 E205 D291 D180 E205 D291 3.2.1.1 0004556,0005509,0005576,0005975,0005983,0016798,0043169,0046872 remove_due_to_license_issue P00693 17803687 4000 HQVLFQGFNWESWKQSGGWYNMMMGKVDDIAAAGVTHVWLPPPSHSVSNEGYMPGRLYDIDASKYGNAAELKSLIGALHGKGVQAIADIVINHRCADYKDSRGIYCIFEGGTSDGRLDWGPHMICRDDTKYSDGTANLDTGADFAAAPDIDHLNDRVQRELKEWLLWLKSDLGFDAWRLDFARGYSPEMAKVYIDGTSPSLAVAEVWDNMATGGDGKPNYDQDAHRQNLVNWVDKVGGAASAGMVFDFTTKGILNAAVEGELWRLIDPQGKAPGVMGWWPAKAVTFVDNHDTGSTQAMWPFPSDKVMQGYAYILTHPGIPCIFYDHFFNWGFKDQIAALVAIRKRNGITATSALKILMHEGDAYVAEIDGKVVVKIGPRYDVGAVIPAGFVTSAHGNDYAVWEK 2qq7 A 2.38 BS01 SR2 A 1 A293 K295 E310 M338 M341 G344 C345 L347 D348 L393 D404 A36 K38 E42 M70 M73 G76 C77 L79 D80 L125 D136 D386 R388 A390 N391 D404 D118 R120 A122 N123 D136 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>27000nM P00523 18316192 1345 KDAWEIPRESLRLEVKLGQGFGEVWMGTWNGTTRVAIKTLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 2qrg A 1.85 BS01 M07 A 1 L136 N284 H341 H377 N484 E672 S674 G675 L125 N267 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=6.6uM remove_due_to_license_issue Ki=6600nM P00489 19781947 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qrh A 1.83 BS01 M08 A 1 L136 N284 H341 H377 N484 E672 S674 G675 L125 N267 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=19.6uM remove_due_to_license_issue Ki=19600nM P00489 19781947 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qrk A 1.75 BS01 AMP A 1 L202 G203 R204 C205 D227 I228 T231 I250 L200 G201 R202 C203 D225 I226 T229 I248 1.5.1.7 0003729,0004753,0004754,0005515,0005737,0005777,0006553,0009085,0016491,0016558,0019878 Ki=55uM remove_due_to_license_issue P38998 17939687 500 AVTLHLRAETKPLEARAALTPTTVKKLIAKGFKIYVEDSPQSTFNINEYRQAGAIIVPAGSWKTAPRDRIIIGLKEMPETDTFPLVHEHIQFAHCYKDQAGWQNVLMRFIKGHGTLYDLEFLENDQGRRVAAFGFYAGFAGAALGVRDWAFKQTHSDDEDLPAVSPYPNEKALVKDVTKDYKEALATGARKPTVLIIGALGRCGSGAIDLLHKVGIPDANILKWDIKETSRGGPFDEIPQADIFINCIYLSKPIAPFTNMEKLNNPNRRLRTVVDVSADTTNPHNPIPIYTVATVFNKPTVLVPTTAGPKLSVISIDHLPSLLPREASEFFSHDLLPSLELLPQRKTAPVWVRAKKLFDRHCARV 2qrm A 1.9 BS01 M09 A 1 L136 N284 H341 H377 N484 E672 S674 G675 L125 N267 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=92.5uM remove_due_to_license_issue P00489 19781947 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 2qrp A 1.86 BS01 S06 A 1 L136 N282 N284 F285 H341 H377 A383 V455 N484 E672 S674 G675 L127 N267 N269 F270 H317 H353 A359 V431 N460 E648 S650 G651 H377 K568 R569 K574 T676 K680 H353 K544 R545 K550 T652 K656 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=0.63uM remove_due_to_license_issue P00489 19781947 998 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 2qrq A 1.8 BS01 S13 A 1 G135 L136 D283 H341 H377 N484 E672 S674 G675 G126 L127 D265 H314 H350 N457 E645 S647 G648 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=7.9uM remove_due_to_license_issue P00489 19781947 998 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 2qry A 2.25 BS01 TPS A 1 Y27 D59 G60 S161 T162 P163 W197 Y215 S218 E245 N279 M281 Y9 D41 G42 S143 T144 P145 W179 Y197 S200 E227 N261 M263 ? 0015888,0016020,0030288,0030975,0030976,0042597,0055052,0055085,0071934 Kd=2.3nM remove_due_to_license_issue Kd=2.3nM P31550 18177053 400 KPVLTVYTYDSFAADWGPGPVVKKAFEADCNCELKLVALEDGVSLLNRLRMEGKNSKADVVLGLDNNLLDAASKTGLFAKSGVAADAVNVPGGWNNDTFVPFDYGYFAFVYDKNKLKNPPQSLKELVESDQNWRVIYQDPRTSTPGLGLLLWMQKVYGDDAPQAWQKLAKKTVTVTKGWSEAYGLFLKGESDLVLSYTTSPAYHILEEKKDNYAAANFSEGHYLQVEVAARTAASKQPELAQKFLQFMVSPAFQNAIPTGNWMYPVANVTLPAGFEKLTKPATTLEFTPAEVAAQRQAWISEWQRAVS 2qt9 A 2.1 BS01 524 A 1 R125 E205 E206 F357 R358 Y547 S630 Y631 Y662 Y666 N710 V711 R87 E167 E168 F319 R320 Y509 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.0023uM remove_due_to_license_issue IC50=2.3nM P27487 17851076 1522 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2qtb A 2.25 BS01 474 A 1 R125 E205 E206 F357 R358 Y547 S630 Y631 Y662 Y666 N710 V711 R87 E167 E168 F319 R320 Y509 S592 Y593 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=4.8nM remove_due_to_license_issue IC50=4.8nM P27487 17851076 1521 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2qtg A 1.84 BS01 MTH A 1 M35 T116 C117 G118 L181 K199 D200 M201 E202 D225 M14 T95 C96 G97 L160 K178 D179 M180 E181 D204 3.2.2.16 0000003,0003824,0005829,0005886,0008930,0009086,0009116,0010087,0016787,0019509 Ki=8.3uM remove_due_to_license_issue Q9T0I8 18342331 268 ILRPISSVVFVIAMQAEALPLVNKFGLSETTDSPLGKGLPWVLYHGVHKDLRINVVCPGRDAALGIDSVGTVPASLITFASIQALKPDIIINAGTCGGFKVKGANIGDVFLVSDVVFHDRRIPIPMFDLYGVGLRQAFSTPNLLKELNLKIGRLSTGDSLDMSTQDETLIIANDATLKDMEGAAVAYVADLLKIPVVFLKAVTDLVDGDKPTAEEFLQNLTVVTAALEGTATKVINFINGRNLSDL 2qtg B 1.84 BS01 MTH B 1 V90 T116 C117 G118 L181 K199 D200 M201 E202 D225 F237 V68 T94 C95 G96 L159 K177 D178 M179 E180 D203 F215 3.2.2.16 0000003,0003824,0005829,0005886,0008930,0009086,0009116,0010087,0016787,0019509 Ki=8.3uM remove_due_to_license_issue Q9T0I8 18342331 269 LRPISSVVFVIAMQAEALPLVNKFGLSETTDSPLGKGLPWVLYHGVHKDLRINVVCPGRDAALGIDSVGTVPASLITFASIQALKPDIIINAGTCGGFKVKGANIGDVFLVSDVVFHDRRIPIPMFDLYGVGLRQAFSTPNLLKELNLKIGRLSTGDSLDMSTQDETLIIANDATLKDMEGAAVAYVADLLKIPVVFLKAVTDLVDGDKPTAEEFLQNLTVVTAALEGTATKVINFINGRNLSDL 2qtn B 2.4 BS01 NCN B 1 G8 G9 Y84 T85 W116 G8 G9 Y84 T85 W116 0003824,0009058,0009435,0016779 remove_due_to_license_issue 18977360 191 MRKIGIIGGTFDPPHYGHLLIANEVYHALNLEEVWFLPNQIPPHKQGRDITSVESRLQMLELATEAEEHFSICLEELSRKGPSYTYDTMLQLTKKYPDVQFHFIIGGDMVEYLPKWYNIEALLDLVTFVGVARPGYKLRTPYPITTVEIPEFAVSSSLLRERYKEKKTCKYLLPEKVQVYIERNGLYES 2qtt B 1.93 BS01 FMC B 1 T116 C117 G118 L181 K199 D200 M201 E202 D225 F237 T94 C95 G96 L159 K177 D178 M179 E180 D203 F215 3.2.2.16 0000003,0003824,0005829,0005886,0008930,0009086,0009116,0010087,0016787,0019509 Ki=48uM remove_due_to_license_issue Q9T0I8 18342331 269 LRPISSVVFVIAMQAEALPLVNKFGLSETTDSPLGKGLPWVLYHGVHKDLRINVVCPGRDAALGIDSVGTVPASLITFASIQALKPDIIINAGTCGGFKVKGANIGDVFLVSDVVFHDRRIPIPMFDLYGVGLRQAFSTPNLLKELNLKIGRLSTGDSLDMSTQDETLIIANDATLKDMEGAAVAYVADLLKIPVVFLKAVTDLVDGDKPTAEEFLQNLTVVTAALEGTATKVINFINGRNLSDL 2qtu A 2.53 BS01 3AS A 1 L298 T299 E305 M336 L339 I373 I376 F377 H475 L476 L32 T33 E39 M70 L73 I107 I110 F111 H202 L203 ? 0003677,0004879,0006355 remove_due_to_license_issue Ki=0.53nM Q92731 17804226 1 DALSPEQLVLTLLEAEPPHVLISRPASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKVYDLLLEMLNAH 2qu2 A 2.6 BS01 251 A 1 D94 G96 S97 W138 F170 W177 I180 R190 D290 D35 G37 S38 W79 F111 W118 I121 R131 D225 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D225 T228 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=3700nM P56817 17761418 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHDEFRTAAVEGPFVDCG 2qu3 A 2.0 BS01 462 A 1 Q74 G75 L92 D94 G96 Y133 W138 F170 W177 D290 Q14 G15 L32 D34 G36 Y73 W78 F110 W117 D224 D94 S97 N99 A101 Y133 D290 T293 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.59uM remove_due_to_license_issue IC50=590nM P56817 17761418 1 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCG 2qu5 A 2.95 BS01 276 A 1 L840 V848 A866 K868 E885 L889 T916 E917 F918 C919 G922 L1019 L1035 C1045 D1046 F1047 L25 V33 A51 K53 E70 L74 T101 E102 F103 C104 G107 L154 L170 C180 D181 F182 D1028 A1030 R1032 N1033 D1046 D1064 D163 A165 R167 N168 D181 D186 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue Ki=9nM P35968 17696416 501 HAERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLADARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQ 2qu6 A 2.1 BS01 857 A 1 V848 A866 E885 T916 E917 F918 C919 I1025 L1035 C1045 D1046 F1047 V27 A43 E59 T90 E91 F92 C93 I149 L159 C169 D170 F171 D1028 A1030 R1032 N1033 D1046 D152 A154 R156 N157 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 Ki=3nM remove_due_to_license_issue IC50=4.6nM, Ki=2.8nM P35968 17696416 501 AERLPYDASKWEFPRDRLKLGKPLGQVIEADAFGIDKTCRTVAVKMLKTHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 2qv7 A 2.3 BS02 ADP A 1 N10 T12 T41 E42 I44 G67 G69 T70 E73 G93 T94 N14 T16 T45 E46 I48 G71 G73 T74 E77 G97 T98 2.7.1.107 0004143,0005524,0005886,0008654,0016301,0016310,0042802,0046872 remove_due_to_license_issue Q6GFF9 18611377 500 GSHMMRKRARIIYNPTSGKEQFKRELPDALIKLEKAGYETSAYATEKIGDATLEAERAMHENYDVLIAAGGDGTLNEVVNGIAEKPNRPKLGVIPMGTVNDFGRALHIPNDIMGALDVIIEGHSTKVDIGKMNNRYFINLAAGGQLTQGPFAYYIKGFEMLPQMKAVDLRIEYDGNVFQGEALLFFLGLTNSMAGFEKLVPDAKLDDGYFTLIIVEKSNLAELGHIMTLASRGEHTKHPKVIYEKAKAINISSFTDLQLNVDGEYGGKLPANFLNLERHIDVFAPNDIVNEELINNDHVDDNL 2qve A 2.0 BS01 247 A 1 Y63 G70 H93 X152 L156 N205 F356 Q442 Y52 G59 H82 X141 L143 N192 F343 Q429 Y63 G70 H93 N205 Y308 R311 F356 Q442 Y52 G59 H82 N192 Y295 R298 F343 Q429 4.3.1.23,5.4.3.6 0003824,0009403,0016829,0016841,0016853,0017000,0050368,0052883 remove_due_to_license_issue Q8GMG0 18078753 991 PVSVDGETLTVEAVRRVAEERATVDVPAESIAKAQKSREIFEGIAEQNIPIYGVTTGYGEMIYMQVDKSKEVELQTNLVRSHSAGVGPLFAEDEARAIVAARLNTLAKGHSAVRPIILERLAQYLNEGITPAIPEIGSLGGDLAPLSHVASTLIGEGYVLRDGRPVETAQVLAERGIEPLELRFKEGLALINGTSGMTGLGSLVVGRALEQAQQAEIVTALLIEAVRGSTSPFLAEGHDIARPHEGQIDTAANMRALMRGSGLTVEHADLRRELQKDKEAGKDVQRSEIYLQKAYSLRAIPQVVGAVRDTLYHARHKLRIELNSANDNPLFFEGKEIFHGANFHGQPIAFAMDFVTIALTQLGVLAERQINRVLNRHLSYGLPEFLVSGDPGLHSGFAGAQYPATALVAENRTIGPASTQSVPSNGDNQDVVSMGLISARNARRVLSNNNKILAVEYLAAAQAVDISGRFDGLSPAAKATYEAVRRLVPTLGVDRYMADDIELVADALSRGEFLRAIARETDIQLR 2qve A 2.0 BS02 247 B 1 Y308 R311 Y295 R298 Y63 G70 H93 N205 Y308 R311 F356 Q442 Y52 G59 H82 N192 Y295 R298 F343 Q429 4.3.1.23,5.4.3.6 0003824,0009403,0016829,0016841,0016853,0017000,0050368,0052883 remove_due_to_license_issue Q8GMG0 18078753 992 PVSVDGETLTVEAVRRVAEERATVDVPAESIAKAQKSREIFEGIAEQNIPIYGVTTGYGEMIYMQVDKSKEVELQTNLVRSHSAGVGPLFAEDEARAIVAARLNTLAKGHSAVRPIILERLAQYLNEGITPAIPEIGSLGGDLAPLSHVASTLIGEGYVLRDGRPVETAQVLAERGIEPLELRFKEGLALINGTSGMTGLGSLVVGRALEQAQQAEIVTALLIEAVRGSTSPFLAEGHDIARPHEGQIDTAANMRALMRGSGLTVEHADLRRELQKDKEAGKDVQRSEIYLQKAYSLRAIPQVVGAVRDTLYHARHKLRIELNSANDNPLFFEGKEIFHGANFHGQPIAFAMDFVTIALTQLGVLAERQINRVLNRHLSYGLPEFLVSGDPGLHSGFAGAQYPATALVAENRTIGPASTQSVPSNGDNQDVVSMGLISARNARRVLSNNNKILAVEYLAAAQAVDISGRFDGLSPAAKATYEAVRRLVPTLGVDRYMADDIELVADALSRGEFLRAIARETDIQLR 2qve B 2.0 BS01 247 A 1 Y308 R311 Y295 R298 Y63 G70 H93 N205 Y308 R311 F356 Q442 Y52 G59 H82 N192 Y295 R298 F343 Q429 4.3.1.23,5.4.3.6 0003824,0009403,0016829,0016841,0016853,0017000,0050368,0052883 remove_due_to_license_issue Q8GMG0 18078753 991 PVSVDGETLTVEAVRRVAEERATVDVPAESIAKAQKSREIFEGIAEQNIPIYGVTTGYGEMIYMQVDKSKEVELQTNLVRSHSAGVGPLFAEDEARAIVAARLNTLAKGHSAVRPIILERLAQYLNEGITPAIPEIGSLGGDLAPLSHVASTLIGEGYVLRDGRPVETAQVLAERGIEPLELRFKEGLALINGTSGMTGLGSLVVGRALEQAQQAEIVTALLIEAVRGSTSPFLAEGHDIARPHEGQIDTAANMRALMRGSGLTVEHADLRRELQKDKEAGKDVQRSEIYLQKAYSLRAIPQVVGAVRDTLYHARHKLRIELNSANDNPLFFEGKEIFHGANFHGQPIAFAMDFVTIALTQLGVLAERQINRVLNRHLSYGLPEFLVSGDPGLHSGFAGAQYPATALVAENRTIGPASTQSVPSNGDNQDVVSMGLISARNARRVLSNNNKILAVEYLAAAQAVDISGRFDGLSPAAKATYEAVRRLVPTLGVDRYMADDIELVADALSRGEFLRAIARETDIQLR 2qve B 2.0 BS02 247 B 1 Y63 G70 H93 X152 L156 N205 F356 Q442 Y52 G59 H82 X141 L143 N192 F343 Q429 Y63 G70 H93 N205 Y308 R311 F356 Q442 Y52 G59 H82 N192 Y295 R298 F343 Q429 4.3.1.23,5.4.3.6 0003824,0009403,0016829,0016841,0016853,0017000,0050368,0052883 remove_due_to_license_issue Q8GMG0 18078753 992 PVSVDGETLTVEAVRRVAEERATVDVPAESIAKAQKSREIFEGIAEQNIPIYGVTTGYGEMIYMQVDKSKEVELQTNLVRSHSAGVGPLFAEDEARAIVAARLNTLAKGHSAVRPIILERLAQYLNEGITPAIPEIGSLGGDLAPLSHVASTLIGEGYVLRDGRPVETAQVLAERGIEPLELRFKEGLALINGTSGMTGLGSLVVGRALEQAQQAEIVTALLIEAVRGSTSPFLAEGHDIARPHEGQIDTAANMRALMRGSGLTVEHADLRRELQKDKEAGKDVQRSEIYLQKAYSLRAIPQVVGAVRDTLYHARHKLRIELNSANDNPLFFEGKEIFHGANFHGQPIAFAMDFVTIALTQLGVLAERQINRVLNRHLSYGLPEFLVSGDPGLHSGFAGAQYPATALVAENRTIGPASTQSVPSNGDNQDVVSMGLISARNARRVLSNNNKILAVEYLAAAQAVDISGRFDGLSPAAKATYEAVRRLVPTLGVDRYMADDIELVADALSRGEFLRAIARETDIQLR 2qw1 A 1.7 BS01 3MG A 1 H152 W183 N211 D236 H151 W182 N210 D235 ? 0005509,0006935,0015757,0015765,0016020,0030246,0030288,0042597,0046872,0055052,0055085 Ki=125uM remove_due_to_license_issue P0AEE5 19348466 310 DTRIGVTIYKYDDNFMSVVRKAIEQDAKAAPDVQLLMNDSQNDQSKQNDQIDVLLAKGVKALAINLVDPAAAGTVIEKARGQNVPVVFFNKEPSRKALDSYDKAYYVGTDSKESGIIQGDLIAKHWAANQGWDLNKDGQIQFVLLKGEPGHPDAEARTTYVIKELNDKGIKTEQLQLDTAMWDTAQAKDKMDAWLSGPNANKIEVVIANNDAMAMGAVEALKAHNKSSIPVFGVDALPEALALVKSGALAGTVLNDANNQAKATFDLAKNLADGKGAADGTNWKIDNKVVRVPYVGVDKDNLAEF 2qwb A 2.0 BS01 SIA A 1 R118 E119 D151 A246 E276 K292 R371 Y406 R37 E38 D70 A166 E196 K212 R290 Y324 D151 E277 K292 R371 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=1820uM remove_due_to_license_issue P03472 9655825 800 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCKDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 2qwb A 2.0 BS02 SIA A 2 S367 S370 S372 N400 D402 W403 K432 S286 S289 S291 N318 D320 W321 K352 D151 E277 K292 R371 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=1820uM remove_due_to_license_issue P03472 9655825 801 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCKDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 2qwc A 1.6 BS02 DAN A 1 R118 E119 D151 R152 W178 A246 E276 K292 R371 Y406 R37 E38 D70 R71 W98 A166 E196 K212 R290 Y324 D151 E277 K292 R371 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=280uM remove_due_to_license_issue IC50=13000nM P03472 9655825 800 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCKDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 2qwd A 2.0 BS02 4AM A 1 R118 E119 D151 R152 W178 A246 E276 K292 R371 Y406 R37 E38 D70 R71 W98 A166 E196 K212 R290 Y324 D151 E277 K292 R371 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=14uM remove_due_to_license_issue P03472 9655825 800 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCKDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 2qwf A 1.9 BS02 G20 A 1 R118 E119 D151 R152 W178 I222 E227 E277 R371 Y406 R37 E38 D70 R71 W98 I142 E147 E197 R290 Y324 D151 E277 K292 R371 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=2.16uM remove_due_to_license_issue P03472 9655825 800 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCKDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 2qwg A 1.8 BS02 G28 A 1 R118 E119 D151 R152 W178 E276 E277 R371 Y406 R37 E38 D70 R71 W98 E196 E197 R290 Y324 D151 E277 K292 R371 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=230uM remove_due_to_license_issue P03472 9655825 800 RDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCKDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 2qx0 A 1.8 BS04 PH2 A 1 T43 K44 P45 L46 F54 N56 D96 F124 T43 K44 P45 L46 F54 N56 D96 F124 R83 R93 D96 D98 R83 R93 D96 D98 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=0.78uM remove_due_to_license_issue A0A5P8YCA3 18007032 181 MIRVYIALGSNLAMPLQQVSAAREALAHLPRSRLVACSPLYRTKPLGPQDQPDFLNAVVALDTSLPPEQLLDHTQAIERNQGRVRKEQRWGPRTLDLDIMLYGDQVIKTDRLTIPHYGLKAREFMLYPLADIAPDLIFPDGESLSECLKRVDKNGLVLW 2qx0 B 1.8 BS04 PH2 B 1 T43 K44 P45 L46 F54 N56 F124 T43 K44 P45 L46 F54 N56 F124 R83 R93 D96 D98 R83 R93 D96 D98 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=0.78uM remove_due_to_license_issue A0A5P8YCA3 18007032 182 MIRVYIALGSNLAMPLQQVSAAREALAHLPRSRLVACSPLYRTKPLGPQDQPDFLNAVVALDTSLPPEQLLDHTQAIERNQGRVRKEQRWGPRTLDLDIMLYGDQVIKTDRLTIPHYGLKAREFMLYPLADIAPDLIFPDGESLSECLKRVDKNGLVLW 2qyk A 2.1 BS01 NPV A 1 Y371 H372 N533 I548 F552 M569 S580 Q581 F584 Y83 H84 N245 I260 F264 M281 S292 Q293 F296 3.1.4.53 0004114,0007165,0008081 ic50=3.3uM remove_due_to_license_issue IC50=3300nM, EC50=20nM P27815 17727341 3 MNIPRFGVKTDQEELLAQELENLNKWGLNIFCVSDYAGGRSLTCIMYMIFQERDLLKKFRIPVDTMVTYMLTLEDHYHADVAYHNSLHAADVLQSTHVLLATPALDAVFTDLEILAALFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEDNCDIFQNLSKRQRQSLRKMVIDMVLATDMSKHMTLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLRNMVHCADLSNPTKPLELYRQWTDRIMAEFFQQGDRERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVHPDAQEILDTLEDNRDWYYSAI 2qyl A 1.95 BS03 NPV A 1 Y233 M347 N395 I410 F414 Q443 F446 Y83 M197 N245 I260 F264 Q293 F296 3.1.4.53 0004114,0007165,0008081 ic50=0.65uM remove_due_to_license_issue IC50=650nM Q07343 17727341 1 MSISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 2qyn A 1.57 BS01 NPV A 1 Y159 M273 N321 I336 F340 M357 Q369 F372 Y74 M188 N236 I251 F255 M272 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=0.57uM remove_due_to_license_issue IC50=1nM Q08499 17727341 1 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 2qzk A 1.8 BS01 I21 A 1 G11 Q12 G13 L30 D32 G34 Y71 T72 Q73 W115 D228 S229 G230 T231 T232 N233 G14 Q15 G16 L33 D35 G37 Y74 T75 Q76 W118 D219 S220 G221 T222 T223 N224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=27nM remove_due_to_license_issue P56817 17827011 400 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2qzl A 1.8 BS01 IXS A 1 G11 Q12 G13 Y14 L30 D32 G34 Y71 T72 Q73 F108 W115 D228 G230 T231 T232 N233 R235 A335 G16 Q17 G18 Y19 L35 D37 G39 Y76 T77 Q78 F113 W120 D222 G224 T225 T226 N227 R229 A325 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=8nM remove_due_to_license_issue IC50=8nM P56817 16690314 449 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2qzr A 1.95 BS02 S79 A 1 D102 Y106 D156 I201 G229 G230 A232 M260 G261 D92 Y96 D133 I178 G206 G207 A209 M237 G238 D102 D280 C318 C320 C323 H349 D92 D257 C295 C297 C300 H326 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=55nM remove_due_to_license_issue P28720 17902085 500 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSEEGVTFKMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 2r0u A 1.9 BS01 M54 A 1 L15 V23 A36 K38 L84 E85 Y86 C87 S88 G90 E134 L137 D148 L14 V19 A32 K34 L73 E74 Y75 C76 S77 G79 E123 L126 D137 D130 K132 E134 N135 D148 T170 D119 K121 E123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1nM O14757 17900896 324 AVPFVEDWDLVQTLGEGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2r1x A 1.6 BS01 KDA C 1 S91 R95 S97 R101 ? 0046872 remove_due_to_license_issue Q52L64 18272175 1 DIVMSQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTITSVQAEDLAVYYCKQSYNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 2r1x B 1.6 BS01 KDA C 1 Y33 R52 E100A Y33 R52 E107 ? 0002250,0005576,0019814,0046872 remove_due_to_license_issue A2NU21 18272175 1 EVKLVESGGGLVQSGGSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKANGYTTEYSPSVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDHDGYYERFSYWGQGTLVTVSAAKTTPPSVYPLAPGSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVP 2r1y A 1.6 BS01 KDO C 1 S91 R95 S97 R101 ? 0046872 remove_due_to_license_issue Q52L64 18272175 2 DIVMSQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTITSVQAEDLAVYYCKQSYNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 2r1y B 1.6 BS02 KDO C 1 Y33 R52 E100A Y33 R52 E107 ? 0002250,0005576,0019814,0046872 remove_due_to_license_issue A2NU21 18272175 2 EVKLVESGGGLVQSGGSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKANGYTTEYSPSVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDHDGYYERFSYWGQGTLVTVSAAKTTPPSVYPLAPNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 2r2l B 2.23 BS03 PB9 B 1 L96 S99 W102 W106 H149 D297 D359 Y361 H362 L74 S77 W80 W84 H127 D275 D337 Y339 H340 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H226 R269 K272 D275 C277 Y278 D330 D337 H340 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=0.58nM remove_due_to_license_issue Q02293 17606674 425 LYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 2r2m B 2.1 BS03 I50 B 1 H79 Y83 W86 E130 D229 A230 C231 S235 S256 W257 G258 H43 Y47 W50 E94 D191 A192 C193 S197 S218 W219 G220 H79 D135 E232 G233 D234 S235 G236 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 Ki=47.1nM remove_due_to_license_issue P00734 17889527 5000 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 2r2w U 2.01 BS01 4PG U 1 H57 H99 D189 S190 Q192 S195 W215 G216 G219 G226 H46 H94 D192 S193 Q195 S198 W218 G219 G221 G229 3.4.21.73 0004252,0006508 Ki=34uM remove_due_to_license_issue P00749 17905583 300 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2r38 A 1.81 BS01 G4G B 1 D25 G27 A28 D29 D30 V32 G48 I50 V82 D25 G27 A28 D29 D30 V32 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 2r38 B 1.81 BS01 G4G B 1 R8 L23 D25 A28 D30 G48 I50 P81 R8 L23 D25 A28 D30 G48 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.036uM remove_due_to_license_issue P04587 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 2r3f A 1.5 BS01 SC8 A 1 I10 G11 E12 V18 A31 K33 L83 H84 K89 Q131 L134 I10 G11 E12 V18 A31 K33 L75 H76 K81 Q123 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=500nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3g A 1.55 BS01 SC9 A 1 I10 G11 E12 G13 A31 K33 L83 H84 D86 L134 I10 G11 E12 G13 A31 K33 L72 H73 D75 L123 D127 K129 Q131 N132 D145 T158 T165 D116 K118 Q120 N121 D134 T147 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=800nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3h A 1.5 BS01 SCE A 1 I10 A31 F82 L83 H84 L134 I10 A31 F73 L74 H75 L125 D127 K129 Q131 N132 D145 T158 T165 D118 K120 Q122 N123 D136 T149 T156 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=20000nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3i A 1.28 BS01 SCF A 1 I10 A31 K33 L83 H84 Q131 N132 L134 I10 A31 K33 L75 H76 Q123 N124 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1000nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3j A 1.65 BS01 SCJ A 1 I10 A31 F80 F82 L83 H84 L134 I10 A31 F72 F74 L75 H76 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=10nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAREVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3k A 1.7 BS01 SCQ A 1 I10 A31 F80 L83 H84 Q131 L134 I10 A31 F72 L75 H76 Q123 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=100nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3l A 1.65 BS01 SCW A 1 I10 A31 F80 L83 H84 L134 I10 A31 F73 L76 H77 L127 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T143 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=100nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLATLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3m A 1.7 BS01 SCX A 1 I10 A31 F80 L83 H84 Q85 K89 Q131 N132 L134 I10 A31 F72 L75 H76 Q77 K81 Q123 N124 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=10nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAREVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3n A 1.63 BS01 SCZ A 1 I10 G11 E12 V18 A31 F80 F82 L83 H84 Q85 Q131 L134 I10 G11 E12 V18 A31 F72 F74 L75 H76 Q77 Q123 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T143 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=70nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3o A 1.8 BS01 2SC A 1 I10 G11 A31 K33 F82 L83 H84 Q85 Q131 L134 I10 G11 A31 K33 F74 L75 H76 Q77 Q123 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=600nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3p A 1.66 BS01 3SC A 1 I10 A31 F80 L83 H84 Q131 N132 L134 D145 I10 A31 F72 L75 H76 Q123 N124 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=900nM remove_due_to_license_issue P24941 17937404 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r3t A 1.8 BS01 G4G B 1 D25 G27 A28 D29 D30 V32 G48 V50 V82 I84 D25 G27 A28 D29 D30 V32 G48 V50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2r3t B 1.8 BS01 G4G B 1 L23 D25 G27 D30 V32 I47 G48 G49 V50 I84 L23 D25 G27 D30 V32 I47 G48 G49 V50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.4uM remove_due_to_license_issue P04587 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2r3w A 1.92 BS01 G3G A 1 D25 G27 A28 D30 V32 G48 I50 V82 D25 G27 A28 D30 V32 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.128uM remove_due_to_license_issue P04587 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 2r3w B 1.92 BS01 G3G A 1 L23 D25 A28 G48 I50 P81 V82 L23 D25 A28 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 2r43 A 1.58 BS01 G3G B 1 D25 G27 D30 V32 G48 G49 V50 I84 D25 G27 D30 V32 G48 G49 V50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2r43 B 1.58 BS01 G3G B 1 L23 D25 A28 G48 G49 V50 P81 I84 L23 D25 A28 G48 G49 V50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1uM remove_due_to_license_issue P03367 18692068 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2r4b A 2.4 BS01 GW7 A 1 A749 K751 M772 V781 L783 L794 T796 M799 C803 L850 T860 D861 F862 A56 K58 M73 V82 L84 L95 T97 M100 C104 L151 T161 D162 F163 D843 A845 R847 N848 D861 G880 D144 A146 R148 N149 D162 G181 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q15303 18287036 1 LVEPLTPSGTAPNQAQLRILKETELKRVKVLGSGAFGTVYKGIWVPEGETVKIPVAIKILNANVEFMDEALIMASMDHPHLVRLLGVCLSPTIQLVTQLMPHGCLLEYVHEHKDNIGSQLLLNWCVQIAKGMMYLEERRLVHRDLAARNVLVKSPNHVKITDFGLARLLEGDEKEYNADGGKMPIKWMALECIHYRKFTHQSDVWSYGVTIWELMTFGGKPYDGIPTREIPDLLEKGERLPQPPICTIDVYMVMVKCWMIDADSRPKFKELAAEFSRMARDPQRYLVIQGDD 2r4f A 1.7 BS01 RIE A 1 R590 S661 V683 S684 D690 K692 R150 S221 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=1.5nM remove_due_to_license_issue P04035 18072721 876 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 2r4f A 1.7 BS02 RIE B 1 E559 C561 L562 A564 S565 R568 K735 A751 L853 A856 E119 C121 L122 A124 S125 R128 K295 A311 L413 A416 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=1.5nM remove_due_to_license_issue P04035 18072721 876 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 2r4f B 1.7 BS01 RIE A 1 E559 C561 L562 A564 S565 K735 A751 N755 L853 A856 E104 C106 L107 A109 S110 K280 A296 N300 L398 A401 E559 K691 D767 E104 K236 D312 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=1.5nM remove_due_to_license_issue P04035 18072721 876 EPRPNEECLQILAKFLSDAEIIQLVNAKLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 2r4f B 1.7 BS02 RIE B 1 R590 S661 S684 D690 K692 R135 S206 S229 D235 K237 E559 K691 D767 E104 K236 D312 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=1.5nM remove_due_to_license_issue P04035 18072721 876 EPRPNEECLQILAKFLSDAEIIQLVNAKLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 2r58 A 2.0 BS01 MLY A 1 D324 N327 W351 F355 D151 N154 W178 F182 ? 0005634,0006355 remove_due_to_license_issue Q9VHA0 17932512 436 AFDWDAYLEETGSEAAPAKCFKQAQNPPNNDFKIGMKLEALDPRNVTSTCIATVVGVLGSRLRLRLDGSDSQNDFWRLVDSTEIHAIGHCEKNGGMLQPPLGFCMNASSWPGYLCKILNNAMVAPEEIFQPEPPEPEENLFKVGQKLEAVDKKNPQLICCATVDAIKDDQIHVTFDGWRGAFDYWCNYRSRDIFPAGWCARSCHPMQPPGHK 2r59 A 1.89 BS02 PH0 A 1 Q136 Y267 G268 G269 E271 H295 E296 H299 E318 Y378 S379 S380 Y383 R563 K565 Q136 Y267 G268 G269 E271 H295 E296 H299 E318 Y378 S379 S380 Y383 R563 K565 E271 H295 E296 H299 E318 D375 Y383 E271 H295 E296 H299 E318 D375 Y383 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 Ki=6.5nM remove_due_to_license_issue P09960 18804029 706 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 2r5a A 2.3 BS01 MLZ A 1 D324 C332 F348 W351 D151 C159 F175 W178 ? 0005634,0006355 Kd=2500uM remove_due_to_license_issue Q9VHA0 17932512 436 AFDWDAYLEETGSEAAPAKCFKQAQNPPNNDFKIGMKLEALDPRNVTSTCIATVVGVLGSRLRLRLDGSDSQNDFWRLVDSTEIHAIGHCEKNGGMLQPPLGFCMNASSWPGYLCKILNNAMVAPEEIFQPEPPEPEENLFKVGQKLEAVDKKNPQLICCATVDAIKDDQIHVTFDGWRGAFDYWCNYRSRDIFPAGWCARSCHPMQPPGHK 2r5p A 2.3 BS01 MK1 B 1 R8 D25 G27 G48 G49 I50 V82 I84 R8 D25 G27 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue O12158 18092815 902 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5p B 2.3 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 I84 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.3nM remove_due_to_license_issue O12158 18092815 902 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5q A 2.3 BS01 1UN B 1 D25 G27 G49 D25 G27 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue O12158 18092815 900 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5q B 2.3 BS01 1UN B 1 D25 G27 D29 D30 G48 G49 P81 I84 D25 G27 D29 D30 G48 G49 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2.7nM remove_due_to_license_issue O12158 18092815 900 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5y A 2.6 BS01 dna C 0 R105 T106 Y108 R143 Q144 I147 N151 R17 T18 Y20 R55 Q56 I59 N63 ? 0000981,0003677,0003700,0005634,0006355 remove_due_to_license_issue P09077 17981120 1 ~ 20 GKKNPPQIYPWMKRVQRTSYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEHK 2r5y A 2.6 BS02 dna D 0 V88 R105 Y125 R128 R131 Q150 R153 M154 K157 V15 R17 Y37 R40 R43 Q62 R65 M66 K69 ? 0000981,0003677,0003700,0005634,0006355 remove_due_to_license_issue P09077 17981120 21 ~ 40 GKKNPPQIYPWMKRVQRTSYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEHK 2r5y B 2.6 BS01 dna C 0 R205 F208 Q244 N247 N251 R255 R1 F4 Q43 N46 N50 R54 ? 0000981,0003677,0006355 remove_due_to_license_issue P40427 17981120 1 ~ 20 RRNFSKQASEILNEYFYSHLSNPYPSEEAKEELARKCGITVSQVSNWFGNKRIRYKKNI 2r5y B 2.6 BS02 dna D 0 R205 R206 Y225 R253 I254 K257 R1 R2 Y24 R52 I53 K56 ? 0000981,0003677,0006355 remove_due_to_license_issue P40427 17981120 21 ~ 40 RRNFSKQASEILNEYFYSHLSNPYPSEEAKEELARKCGITVSQVSNWFGNKRIRYKKNI 2r5z A 2.6 BS01 dna C 0 H89 R105 T106 Y108 Q144 I147 N151 K155 H15 R19 T20 Y22 Q58 I61 N65 K69 ? 0000981,0003677,0003700,0005634,0006355 remove_due_to_license_issue P09077 17981120 1 ~ 20 KKNPPQIYPWMKRVHLRQRTSYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEHK 2r5z A 2.6 BS02 dna D 0 V88 H89 R103 R105 Y125 R131 Q150 R153 M154 K157 V14 H15 R17 R19 Y39 R45 Q64 R67 M68 K71 ? 0000981,0003677,0003700,0005634,0006355 remove_due_to_license_issue P09077 17981120 21 ~ 40 KKNPPQIYPWMKRVHLRQRTSYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEHK 2r5z B 2.6 BS01 dna C 0 F208 Q244 N247 W248 N251 R255 F4 Q43 N46 W47 N50 R54 ? 0000981,0003677,0006355 remove_due_to_license_issue P40427 17981120 1 ~ 20 RRNFSKQASEILNEYFYSHLSNPYPSEEAKEELARKCGITVSQVSNWFGNKRIRYKKNI 2r5z B 2.6 BS02 dna D 0 R205 R206 N207 Y225 R253 I254 K257 R1 R2 N3 Y24 R52 I53 K56 ? 0000981,0003677,0006355 remove_due_to_license_issue P40427 17981120 21 ~ 40 RRNFSKQASEILNEYFYSHLSNPYPSEEAKEELARKCGITVSQVSNWFGNKRIRYKKNI 2r64 A 2.3 BS01 740 A 1 E8 I10 V18 A31 F80 E81 F82 L83 H84 Q85 L134 D145 E8 I10 V18 A31 F72 E73 F74 L75 H76 Q77 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.03uM remove_due_to_license_issue IC50=30nM P24941 18353638 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2r6f A 3.2 BS01 ADP A 1 H12 N13 G34 S35 G36 K37 S38 S39 Y816 Q821 H12 N13 G34 S35 G36 K37 S38 S39 Y766 Q771 ? 0003677,0003824,0004518,0005524,0005737,0006281,0006289,0008270,0009380,0009381,0009432,0016887,0046872 remove_due_to_license_issue Q5KVB6 18158267 1000 MDKIIVKGARAHNLKNIDVEIPRGKLVVLTGLSGSGKSSLAFDTIYAEGQRRYVESLSAYARQFLGQMEKPDVDAIEGLSPAISIDQKTTSRNPRSTVGTVTEIYDYLRLLFARIGRPICPTHGIEIQSQTIEQMVDRLLSYPERTKMQILAPIDVVVDRIIIKDGIAARLADSLETALKLADGKVVVDVIGEGELLFSEKHACPYCGFSIGELEPRLFSFNSPFGACPDCDGLGAKLEVDLDLVIPNDELTLKEHAIAPWEPYYPQLLEAVCRHYGIPMDVPVKDLPKEQLDKILYGSGGEPIYFRYTNDFGQVREQYIAFEGVIPNVERRYRETSSDYIREQMEKYMAEQPCPTCQGYRLKKESLAVLVGGKHIGEVTAMSVTEALAFFDGLELTEKEAQIARLILREIRDRLGFLQNVGLDYLTLSRSAGTLSGGEAQRIRLATQIGSRLTGVLYVLDEPSIGLHQRDNDRLIATLKSMRDLGNTLIVVEHDEDTMLAADYLIDIGPGAGIHGGEVVAAGTPEEVMNDPNSLTGQYLSGKKFIPIPAERRRPDGRWLEVVGAREHNLKNVSVKIPLGTFVAVTGVSGSGKSTLVNEVLYKALAQKLHRAKAKPGEHRDIRGLEHLDKVIDIDQSPIGRTPRSNPATYTGVFDDIRDVFASTNEAKVRGYKKGRFSFNVKGGRCEACHGDGIIKIEMHFLPDVYVPCEVCHGKRYNRETLEVTYKGKNIAEVLDMTVEDALDFFASIPKIKRKLETLYDVGLGYMKLGQPATTLSGGEAQRVKLAAELHRRSNGRTLYILDEPTTGLHVDDIARLLDVLHRLVDNGDTVLVIEHNLDVIKTADYIIDLGPEGGDRGGQIVAVGTPEEVAEVKESHTGRYLKPILERDRARMQARYEA 2r6f A 3.2 BS02 ADP A 2 R480 H618 N619 G640 S641 G642 K643 S644 T645 R430 H568 N569 G590 S591 G592 K593 S594 T595 ? 0003677,0003824,0004518,0005524,0005737,0006281,0006289,0008270,0009380,0009381,0009432,0016887,0046872 remove_due_to_license_issue Q5KVB6 18158267 1001 MDKIIVKGARAHNLKNIDVEIPRGKLVVLTGLSGSGKSSLAFDTIYAEGQRRYVESLSAYARQFLGQMEKPDVDAIEGLSPAISIDQKTTSRNPRSTVGTVTEIYDYLRLLFARIGRPICPTHGIEIQSQTIEQMVDRLLSYPERTKMQILAPIDVVVDRIIIKDGIAARLADSLETALKLADGKVVVDVIGEGELLFSEKHACPYCGFSIGELEPRLFSFNSPFGACPDCDGLGAKLEVDLDLVIPNDELTLKEHAIAPWEPYYPQLLEAVCRHYGIPMDVPVKDLPKEQLDKILYGSGGEPIYFRYTNDFGQVREQYIAFEGVIPNVERRYRETSSDYIREQMEKYMAEQPCPTCQGYRLKKESLAVLVGGKHIGEVTAMSVTEALAFFDGLELTEKEAQIARLILREIRDRLGFLQNVGLDYLTLSRSAGTLSGGEAQRIRLATQIGSRLTGVLYVLDEPSIGLHQRDNDRLIATLKSMRDLGNTLIVVEHDEDTMLAADYLIDIGPGAGIHGGEVVAAGTPEEVMNDPNSLTGQYLSGKKFIPIPAERRRPDGRWLEVVGAREHNLKNVSVKIPLGTFVAVTGVSGSGKSTLVNEVLYKALAQKLHRAKAKPGEHRDIRGLEHLDKVIDIDQSPIGRTPRSNPATYTGVFDDIRDVFASTNEAKVRGYKKGRFSFNVKGGRCEACHGDGIIKIEMHFLPDVYVPCEVCHGKRYNRETLEVTYKGKNIAEVLDMTVEDALDFFASIPKIKRKLETLYDVGLGYMKLGQPATTLSGGEAQRVKLAAELHRRSNGRTLYILDEPTTGLHVDDIARLLDVLHRLVDNGDTVLVIEHNLDVIKTADYIIDLGPEGGDRGGQIVAVGTPEEVAEVKESHTGRYLKPILERDRARMQARYEA 2r6n A 1.95 BS01 CKE A 1 G23 C25 G64 G65 G66 Y67 N161 G24 C26 G65 G66 G67 Y68 N162 Q19 C25 H162 N182 Q20 C26 H163 N183 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 17911019 300 RAPDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 2r6w A 2.0 BS01 LLB A 1 T347 A350 D351 E353 W383 L387 I424 H524 L525 L536 T34 A37 D38 E40 W70 L74 I111 H211 L212 L216 ? Ki=0.44nM remove_due_to_license_issue P03372 18474858 1 LALSLTADQMVSALLDAEPPILYSEYASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYVPLYDLLLEMLDAHRL 2r6y A 2.0 BS01 LLC A 1 T347 A350 D351 E353 W383 L387 F404 M421 I424 H524 L525 T35 A38 D39 E41 W71 L75 F92 M109 I112 H212 L213 ? Ki=0.32nM remove_due_to_license_issue IC50=120nM P03372 18474858 1 LALSLTADQMVSALLDAEPPILYSEYDPSMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMVPLYDLLLEMLDAHRL 2r75 1 1.402 BS01 01G 1 1 G16 G17 G18 N21 A67 A69 G100 G103 G104 T105 G106 E135 F179 D183 G9 G10 G11 N14 A60 A62 G93 G96 G97 T98 G99 E128 F172 D176 ? 0000917,0003924,0005525,0005737,0032153,0043093,0051258,0051301,0090529 Kd=714nM remove_due_to_license_issue O66809 18291323 614 CKIKVIGVGGGGSNAVNRMYEDGIEGVELYAINTDVQHLSTLKVPNKIQIGEKVTRGLGAGAKPEVGEEAALEDIDKIKEILRDTDMVFISAGLGGGTGTGAAPVIAKTAKEMGILTVAVATLPFRFEGPRKMEKALKGLEKLKESSDAYIVIHNDKIKELSNRTLTIKDAFKEVDSVLSKAVRGITSIVVTPAVINVDFADVRTTLEEGGLSIIGMGEGRGDEKADIAVEKAVTSPLLEGNTIEGARRLLVTIWTSEDIPYDIVDEVMERIHSKVHPEAEIIFGAVLEPQEQDFIRVAIVATDFPEEKFQVGEKEVKFKVIK 2r7b A 2.7 BS02 253 A 1 V96 A109 S160 Y161 A162 L212 T222 V22 A35 S86 Y87 A88 L138 T148 D205 K207 E209 N210 D223 T245 D131 K133 E135 N136 D149 T160 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=60nM O15530 17941624 701 RKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2r8q A 1.5 BS02 IBM A 1 N838 F890 N242 F294 3.1.4.- 0004114,0007165,0008081 ic50=580uM remove_due_to_license_issue IC50=580000nM Q6S996 17944832 3 VIAVTPEEREAVMSIDFGGAYDFTSPGFNLFEVREKYSEPMDAAAGVVYNLLWNSGLPEKFGCREQTLLNFILQCRRRYRRVPYHNFYHVVDVCQTLHTYLYTGKASELLTELECYVLLVTALVHDLDHMGVNNSFYLKTDSPLGILSSASGNNSVLEVHHCSLAIEILSDPAADVFEGLSGQDVAYAYRALIDCVLATDMAKHADALSRFTELATSGFEKDNDTHRRLVMETLIKAGDVSNVTKPFETSRMWAMAVTEEFYRQGDMEKEKGVEVLPMFDRSKNNELARGQIGFIDFVAGKFFRDIVGNLFHGMQWCVDTVNSNRAKWQEILDGR 2r8s H 1.95 BS01 rna R 0 G26 F27 N28 Y30 S52 S54 Y57 R98 R99 A100 G102 M103 S104 T105 Y106 G107 D109 G26 F27 N28 Y30 S52 S54 Y57 R98 R99 A100 G102 M103 S104 T105 Y106 G107 D109 remove_due_to_license_issue 18162543 102 ~ 261 EVQLVESGGGLVQPGGSLRLSCAASGFNLYSSSIHWVRQAPGKGLEWVAYISSSYGYTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRAAGMSTYGFDYWGQGTLVTVSSASTKGPSVFPLAPSGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 2r8s L 1.95 BS01 rna R 0 S30 L46 Y49 S50 S56 G57 V58 P59 S60 R66 Y92 S30 L46 Y49 S50 S56 G57 V58 P59 S60 R66 Y92 remove_due_to_license_issue 18162543 102 ~ 261 DIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSYSSPITFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 2r9m A 1.97 BS01 Y11 A 1 G23 C25 K64 G68 G69 F70 M71 V162 N163 G23 C25 K64 G68 G69 F70 M71 V162 N163 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue IC50=1.5nM P25774 281 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 2r9s A 2.4 BS01 255 A 1 I70 G71 N89 A91 M146 L148 M149 D150 A151 N152 V196 L206 I25 G26 N44 A46 M101 L103 M104 D105 A106 N107 V151 L161 D189 K191 N194 D207 D144 K146 N149 D162 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.15uM remove_due_to_license_issue IC50=150nM P53779 17911023 502 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDKQLDEREHTIEEWKELIYKEVMNS 2r9w A 1.8 BS01 23C A 1 S64 L119 Q120 N152 Y221 A318 T319 G320 S61 L116 Q117 N149 Y218 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=8uM remove_due_to_license_issue Ki=5000nM P00811 18333608 365 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2r9x A 1.9 BS01 WH6 A 1 S64 Q120 Y221 G317 A318 T319 G320 S61 Q117 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=14uM remove_due_to_license_issue P00811 18333608 365 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2ra0 A 2.3 BS01 JNJ A 1 E97 T98 Y99 E146 D189 A190 C191 Q192 W215 G216 C220 E83 T84 Y85 E135 D179 A180 C181 Q182 W205 G206 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=15.9nM remove_due_to_license_issue Ki=15.9nM P00742 18159923 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2ra6 A 1.5 BS02 ETY A 1 L61 G63 L78 T79 A80 F112 F114 F129 L36 G38 L53 T54 A55 F87 F89 F104 ? 0005576,0005615,0036094 remove_due_to_license_issue Q29147 17685895 604 RHWHTVVLASSDRSLIEEEGPFRNFIQNITVESGNLNGFFLTRKNGQCIPLYLTAFKTEEARQFKLNYYGTNDVYYESSKPNEYAKFIFYNYHDGKVNVVANLFGRTPNLSNEIKKRFEEDFMNRGFRRENILDISEVDHC 2rbf A 2.25 BS01 dna C 0 T5 T28 P29 H30 W31 T3 T26 P27 H28 W29 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue P09546 18586269 3 ~ 21 TTTMGVKLDDATRERIKSAATRIDRTPHWLIKQAIFSYLEQLEN 2rbf A 2.25 BS02 dna D 0 T4 T5 M6 G7 K9 T2 T3 M4 G5 K7 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue P09546 18586269 1 ~ 19 TTTMGVKLDDATRERIKSAATRIDRTPHWLIKQAIFSYLEQLEN 2rbf B 2.25 BS01 dna C 0 G7 K9 G4 K6 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue P09546 18586269 3 ~ 21 TTMGVKLDDATRERIKSAATRIDRTPHWLIKQAIFSYLEQLENSD 2rbf B 2.25 BS02 dna D 0 T28 P29 H30 T25 P26 H27 1.2.1.88,1.5.5.2 0006355 remove_due_to_license_issue P09546 18586269 1 ~ 19 TTMGVKLDDATRERIKSAATRIDRTPHWLIKQAIFSYLEQLENSD 2rc8 A 1.45 BS01 DSN A 1 Y97 S123 F124 S125 R130 S179 S180 M223 D224 Y94 S120 F121 S122 R127 S176 S177 M220 D221 ? 0015276,0016020 remove_due_to_license_issue Q9R1M7 18636091 901 KLHLRVVTLIEHPFVFTREVDDEGLCPAGQLCLDPMTNDSSMLDRLFSSLHSSNDTVPIKFKKCCYGYCIDLLEQLAEDMNFDFDLYIVGDGKYGAWKNGHWTGLVGDLLSGTANMAVTSFSINTARSQVIDFTSPFFSTSLGILVRTRGTELSGIHDPKLHHPSQGFRFGTVRESSAEDYVRQSFPEMHEYMRRYNVPATPDGVQYLKNDPEKLDAFIMDKALLDYEVSIDADCKLLTVGKPFAIEGYGIGLPPNSPLTSNISELISQYKSHGFMDVLHDKWY 2rc9 A 1.96 BS01 1AC A 1 Y97 S123 F124 S125 R130 S179 S180 M223 D224 Y94 S120 F121 S122 R127 S176 S177 M220 D221 ? 0015276,0016020 remove_due_to_license_issue Q9R1M7 18636091 1001 KLHLRVVTLIEHPFVFTREVDDEGLCPAGQLCLDPMTNDSSMLDRLFSSLHSSNDTVPIKFKKCCYGYCIDLLEQLAEDMNFDFDLYIVGDGKYGAWKNGHWTGLVGDLLSGTANMAVTSFSINTARSQVIDFTSPFFSTSLGILVRTRGTELSGIHDPKLHHPSQGFRFGTVRESSAEDYVRQSFPEMHEYMRRYNVPATPDGVQYLKNDPEKLDAFIMDKALLDYEVSIDADCKLLTVGKPFAIEGYGIGLPPNSPLTSNISELISQYKSHGFMDVLHDKWYKVV 2rcb A 1.62 BS01 DSN A 1 Y95 S121 F122 S123 R128 S177 S178 D222 Y92 S118 F119 S120 R125 S174 S175 D219 ? 0015276,0016020 remove_due_to_license_issue Q8VHN2 18636091 901 RPKLRVVTLVEHPFVFTRESDEDGQCPAGQLCLDPGTNDSARLDALFAALVNGSVPRTLRRCCYGYCIDLLERLAEDLAFDFELYIVGDGKYGALRDGRWTGLVGDLLAGRAHMAVTSFSINSARSQVVDFTSPFFSTSLGIMVRTRGTELSGIHDPKLHHPSQGFRFGTVWESSAEAYIKASFPEMHAHMRRHSAPTTPHGVAMLTSDPPKLNAFIMDKSLLDYEVSIDADCKLLTVGKPFAIEGYGIGLPQNSPLTSNLSEFISRYKSSGFIDLLHDKWY 2rcn A 2.25 BS02 GDP A 1 N168 K169 D171 L172 S199 S200 H201 G225 V226 G227 K228 S229 S230 N114 K115 D117 L118 S145 S146 H147 G171 V172 G173 K174 S175 S176 3.6.1.- 0003924,0005525,0005737,0016787,0019843,0042254,0042274,0046872 Kd=1uM remove_due_to_license_issue Q8ZKB0 18007041 600 LFGEPAEGIVISRFGMHADVESADGEVHRCNIRRTIRSLVTGDRVVWRPGKVKGIVEAVHERTSVLTRPVKPIAANIDQIVIVSAILPELSLNIIDRYLVGCETLQVEPLIVLNKIDLLDDEGMDFVNEQMDIYRNIGYRVLMVSSHTQDGLKPLEEALTGRISIFAGQSGVGKSSLLNALLGLQNEILTNTAARLYHFPHGGDVIDSPGVREFGLWHLEPEQITQGFVEFHDYLGHCKYRDCKHDADPGCAIREAVENGAIAETRFENYHRILESMA 2rcw A 2.8 BS01 AAI A 1 V101 H201 G202 Y228 Y235 F236 S243 Y246 E327 V101 H201 G202 Y228 Y235 F236 S243 Y246 E327 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Ki=8nM, EC50=3nM P09874 400 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 2rcx A 2.0 BS01 SM4 A 1 S64 L119 Y150 N152 Y221 G317 A318 T319 G320 N343 S61 L116 Y147 N149 Y218 G314 A315 T316 G317 N340 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 17997318 964 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 2rd6 A 2.3 BS01 78P A 1 H201 G202 Y235 F236 K242 S243 Y246 E327 H201 G202 Y235 F236 K242 S243 Y246 E327 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=1.5nM, Ki=5nM, EC50=5.9nM, Kd=1.7nM P09874 900 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 2reg A 1.9 BS01 CHT A 1 W43 W90 Y119 N156 D157 W205 W15 W62 Y91 N128 D129 W177 ? 0015871,0022857,0033265,0042597,0043190,0055085 Kd=2.3uM remove_due_to_license_issue Q92N37 18779321 1 EPESCGTVRFSDVGWTDITATTATATTILEALGYETDVKVLSVPVTYTSLKNKDIDVFLGNWMPTMEADIAPYREDKSVETVRENLAGAKYTLATNAKGAELGIKDFKDIAAHKDELDGKIYGIEPGNDGNRLIIDMVEKGTFDLKGFEVVESSEQGMLAQVARAEKSGDPIVFLGWEPHPMNANFKLTYLSGGDDVFGPNYGGATVHTNVRAGYTTECPNVDKLLQNLSFSLQMENEIMGKILNDGEDPEKAAAAWLKDNPQSIEPWLSGVATKDGGDGLAAVKAALGL 2rf2 A 2.4 BS01 MRX A 1 L100 K101 V106 V179 Y181 L234 H235 Y318 L97 K98 V103 V176 Y178 L231 H232 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=3.6nM remove_due_to_license_issue P04585 18083561 561 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 2rfh A 1.7 BS02 23N A 1 H69 R127 N144 R145 H196 I243 A250 E270 H69 R127 N144 R145 H196 I243 A250 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=0.15uM remove_due_to_license_issue P00730 18289863 1309 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 2rfn A 2.5 BS01 AM7 A 1 I1084 F1089 V1092 A1108 K1110 F1124 E1127 G1128 M1131 L1140 L1142 V1155 L1157 Y1159 M1160 K1161 G1163 M1211 I28 F29 V32 A48 K50 F64 E67 G68 M71 L80 L82 V95 L97 Y99 M100 K101 G103 M151 D1204 A1206 R1208 N1209 D1222 D144 A146 R148 N149 D162 2.7.10.1 0004672,0004713,0005524,0006468 ic50=5nM remove_due_to_license_issue IC50=8.9nM, Ki=8.9nM P08581 18055465 1 ALNPELVQAVQHVVIGPSSLIVHFNEVIFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 2rg5 A 2.4 BS01 279 A 1 A51 K53 E71 L75 T106 L108 M109 A111 L167 D168 A44 K46 E64 L68 T99 L101 M102 A104 L160 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=3.1nM remove_due_to_license_issue IC50=3.1nM, EC50=61nM Q16539 18072718 501 ERPTFYRQELNKTIWEVPERYQNLSPVYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 2rg6 A 1.72 BS01 287 A 1 A51 K53 E71 L75 T106 L108 M109 A111 L167 D168 A44 K46 E64 L68 T99 L101 M102 A104 L160 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=2.2nM remove_due_to_license_issue IC50=2.2nM, EC50=10nM Q16539 18072718 501 ERPTFYRQELNKTIWEVPERYQNLSPVGGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2rg6 A 1.72 BS02 287 A 2 L195 N196 A255 Y258 L178 N179 A238 Y241 D150 K152 N155 D168 T185 D143 K145 N148 D161 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=2.2nM remove_due_to_license_issue IC50=2.2nM, EC50=10nM Q16539 18072718 502 ERPTFYRQELNKTIWEVPERYQNLSPVGGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2rgp A 2.0 BS01 HYZ A 1 L718 A743 K745 C775 R776 L788 T790 M793 L844 T854 D855 F856 L17 A38 K40 C65 R66 L78 T80 M83 L134 T144 D145 F146 D837 A839 R841 N842 D855 D127 A129 R131 N132 D145 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.03uM remove_due_to_license_issue P00533 18653333 1 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPVKIPVAIKELRKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMNFYRALMDVVDADEY 2ri9 A 1.95 BS02 LDY F 1 F1468 E1472 T1501 E1502 F433 E437 T466 E467 E1122 R1126 D1267 E1409 E87 R91 D232 E374 3.2.1.113 0004571,0005509,0005576,0005783,0005975,0006486,0016020,0016798,0036503,0046872 remove_due_to_license_issue P31723 18323617 2 SNQAKADAVKEAFQHAWNGYMKYAFPHDELTPVSNGHADSRNGWGASAVDALSTAVIMGKADVVNAILEHVADIDFSKTSDTVSLFETTIRYLAGMLSGYDLLQGPAKNLVDNQDLIDGLLDQSRNLADVLKFAFDTPSGVPYNNINITSHGNDGATTNGLAVTGTLVLEWTRLSDLTGDEEYAKLSQKAESYLLKPQPSSSEPFPGLVGSSININDGQFADSRVSWNGGDDSFYEYLIKMYVYDPKRFETYKDRWVLAAESTIKHLKSHPKSRPDLTFLSSYSNRNYDLSSQHLTCFDGGSFLLGGTVLDRQDFIDFGLELVDGCEATYNSTLTKIGPDSWGWDPKKVPSDQKEFYEKAGFYISSGSYVLRPEVIESFYYAHRVTGKEIYRDWVWNAFVAINSTCRTDSGFAAVSDVNKANGGSKYDNQESFLFAEVMKYSYLAHSEDAAWQVQKGGKNTFVYNTEAHPISVAR 2ria A 1.8 BS04 289 A 1 E321 N323 E329 N341 R343 E112 N114 E120 N132 R134 ? ic50=2.7mM remove_due_to_license_issue P35247 18092821 356 QVEALQGQVQHLQAAFSQYKKVELFPNGQSVGEKIFKTAGFVKPFTEAQLLCTQAGGQLASPRSAAENAALQQLVVAKNEAAFLSMTDSKTEGKFTYPTGESLVYSNWAPGEPNDDGGSEDCVEIFTNGKWNDRACGEKRLVVCEF 2rib A 1.8 BS04 GMH A 1 E321 N323 D325 E329 N341 E116 N118 D120 E124 N136 ? remove_due_to_license_issue P35247 18092821 356 SLRQQVEALQGQVQHLQAAFSQYKKVELFPNGQSVGEKIFKTAGFVKPFTEAQLLCTQAGGQLASPRSAAENAALQQLVVAKNEAAFLSMTDSKTEGKFTYPTGESLVYSNWAPGEPNDDGGSEDCVEIFTNGKWNDRACGEKRLVVCEF 2rin A 1.8 BS01 ACH A 1 W43 D45 W90 Y119 I152 N156 D157 W205 W13 D15 W60 Y89 I122 N126 D127 W175 ? 0015871,0022857,0033265,0042597,0043190,0055085 Kd=100uM remove_due_to_license_issue Q92N37 18779321 1 ESCGTVRFSDVGWTDITATTATATTILEALGYETDVKVLSVPVTYTSLKNKDIDVFLGNWMPTMEADIAPYREDKSVETVRENLAGAKYTLATNAKGAELGIKDFKDIAAHKDELDGKIYGIEPGNDGNRLIIDMVEKGTFDLKGFEVVESSEQGMLAQVARAEKSGDPIVFLGWEPHPMNANFKLTYLSGGDDVFGPNYGGATVHTNVRAGYTTECPNVDKLLQNLSFSLQMENEIMGKILNDGEDPEKAAAAWLKDNPQSIEPWLSGVATKDGGDGLAAVKAALGL 2rio A 2.4 BS02 ADP A 1 Y25 G26 V32 A43 K45 E89 C91 N94 L147 D171 Y18 G19 V25 A36 K38 E82 C84 N87 L128 D152 D140 K142 N145 D171 T195 D121 K123 N126 D152 T162 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue P32361 18191223 1101 NFEQSLKNLVVSEKILGYGSSGTVVFQGSFQGRPVAVKRMLIDFCDIALMEIKLLTESDDHPNVIRYYCSETTDRFLYIALELCNLNLQDLVESKYNPISLLRQIASGVAHLHSLKIIHRDLKPQNILVSTSSRFTADQQTGAENLRILISDFGLCKKLDSTSGWRAPELLEESNNLQTKRRLTRSIDIFSMGCVFYYILSKGKHPFGDKYSRESNIIRGIFSLDEMKCLHDRSLIAEATDLISQMIDHDPLKRPTAMKVLRHPLFWPKSKKLEFLLKVSDRLEIENRDPPSALLMKFDAGSDFVIPSGDWTVKFDKTFMDRKYHSSKLMDLLRALRNKYHHFMDLPEDIAELMGPVPDGFYDYFTKRFPNLLIGVYMIVKENLSDDQILREFLYS 2rip A 2.9 BS01 34Q A 1 E205 E206 S209 F357 S630 Y662 Y666 N710 V711 E168 E169 S172 F320 S593 Y625 Y629 N673 V674 Y547 S630 Y631 D708 H740 Y510 S593 Y594 D671 H703 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=65nM P27487 17977724 800 DSRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 2rjp A 2.8 BS05 886 A 1 T329 L330 G331 M332 F357 H361 Q362 H365 H371 V390 P393 V394 M395 V398 P403 T112 L113 G114 M115 F140 H144 Q145 H148 H154 V173 P176 V177 M178 V181 P186 3.4.24.82 0004222,0006508,0008237 remove_due_to_license_issue IC50=100nM O75173 18042673 510 ASLSRFVETLVVADDKMAAFHGAGLKRYLLTVMAAAAKAFKHPSIRNPVSLVVTRLVILEGPQVGPSAAQTLRSFCAWQRGLNTPEDSDPDHFDTAILFTRQDLCGVSTCDTLGMADVGTVCDPARSCAIVEDDGLQSAFTAAHQLGHVFNMLHDNSKPCISLNGPLSTSRHVMAPVMAHVDPEEPWSPCSARFITDFLDNGYGHCLLDKPEAPLHLPVTFPGKDYDADRQCQLTFGPDSRHCPQLPPPCAALWCSGHLNGHAMCQTKHSPWADGTPCGPAQACMGGRCLH 2rjr A 2.1 BS01 295 A 1 Y63 G70 H93 X152 L156 N205 F356 Q442 Y52 G59 H82 X141 L143 N192 F343 Q429 Y63 G70 H93 N205 Y308 R311 F356 Q442 Y52 G59 H82 N192 Y295 R298 F343 Q429 4.3.1.23,5.4.3.6 0003824,0009403,0016829,0016841,0016853,0017000,0050368,0052883 remove_due_to_license_issue Q8GMG0 18078753 1001 PVSVDGETLTVEAVRRVAEERATVDVPAESIAKAQKSREIFEGIAEQNIPIYGVTTGYGEMIYMQVDKSKEVELQTNLVRSHSAGVGPLFAEDEARAIVAARLNTLAKGHSAVRPIILERLAQYLNEGITPAIPEIGSLGGDLAPLSHVASTLIGEGYVLRDGRPVETAQVLAERGIEPLELRFKEGLALINGTSGMTGLGSLVVGRALEQAQQAEIVTALLIEAVRGSTSPFLAEGHDIARPHEGQIDTAANMRALMRGSGLTVEHADLRRELQKDKEAGKDVQRSEIYLQKAYSLRAIPQVVGAVRDTLYHARHKLRIELNSANDNPLFFEGKEIFHGANFHGQPIAFAMDFVTIALTQLGVLAERQINRVLNRHLSYGLPEFLVSGDPGLHSGFAGAQYPATALVAENRTIGPASTQSVPSNGDNQDVVSMGLISARNARRVLSNNNKILAVEYLAAAQAVDISGRFDGLSPAAKATYEAVRRLVPTLGVDRYMADDIELVADALSRGEFLRAIARETDIQLR 2rk8 A 2.0 BS02 PPF A 1 R87 K244 H264 S286 D311 R405 R87 K244 H264 S286 D311 R405 R87 Y235 K244 H264 S286 C288 D311 R405 R87 Y235 K244 H264 S286 C288 D311 R405 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 Ki=230uM remove_due_to_license_issue P07379 18197707 3969 MPPQLHNGLDFSAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEATAAAEHKGKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 2rka A 1.95 BS01 PGA A 1 R87 G237 K244 F333 R405 R84 G234 K241 F330 R402 R87 Y235 K244 H264 S286 C288 D311 R405 R84 Y232 K241 H261 S283 C285 D308 R402 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 Ki=1mM remove_due_to_license_issue P07379 18197707 623 QLHNGLDFSAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEAKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 2rkd A 1.9 BS03 3PP A 1 R87 G237 K244 R405 R85 G235 K242 R403 R87 Y235 K244 H264 S286 C288 D311 R405 R85 Y233 K242 H262 S284 C286 D309 R403 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 Ki=1.9mM remove_due_to_license_issue P07379 18197707 703 PQLHNGLDFSAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEAGKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 2rke A 1.8 BS03 SAT A 1 R87 Y235 G237 R84 Y232 G234 R87 Y235 K244 H264 S286 C288 D311 R405 R84 Y232 K241 H261 S283 C285 D308 R402 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 Ki=82.5uM remove_due_to_license_issue P07379 18197707 704 QLHNGLDFSAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEAGKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 2rkf A 1.8 BS01 AB1 A 1 D25 G27 A28 D29 D30 I32 I50 P81 D25 G27 A28 D29 D30 I32 I50 P81 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.83nM remove_due_to_license_issue Q90JJ9 18400858 501 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 2rkf B 1.8 BS01 AB1 A 1 D25 G27 A28 D29 I32 G48 G49 A82 I84 D25 G27 A28 D29 I32 G48 G49 A82 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90JJ9 18400858 501 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 2rkg A 1.8 BS01 AB1 B 1 D25 G27 A28 D29 G49 G50 I85 D25 G27 A28 D29 G49 G50 I85 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue A0F6C5 18400858 501 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 2rkg B 1.8 BS01 AB1 B 1 D25 G27 A28 D29 D30 G50 I51 P82 D25 G27 A28 D29 D30 G50 I51 P82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=8.2nM remove_due_to_license_issue A0F6C5 18400858 501 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 2rkm A 1.8 BS01 LYS A 1 E32 V34 Y109 W416 C417 D419 E32 V34 Y109 W416 C417 D419 ? 0015031,0015833,0030288,0042597,0043190,0055085,1904680 remove_due_to_license_issue P06202 9245406 2001 ADVPAGVQLADKQTLVRNNGSEVQSLDPHKIEGVPESNVSRDLFEGLLISDVEGHPSPGVAEKWENKDFKVWTFHLRENAKWSDGTPVTAHDFVYSWQRLADPNTASPYASYLQYGHIANIDDIIAGKKPATDLGVKALDDHTFEVTLSEPVPYFYKLLVHPSVSPVPKSAVEKFGDKWTQPANIVTNGAYKLKNWVVNERIVLERNPQYWDNAKTVINQVTYLPISSEVTDVNRYRSGEIDMTYNNMPIELFQKLKKEIPNEVRVDPYLCTYYYEINNQKAPFNDVRVRTALKLALDRDIIVNKVKNQGDLPAYSYTPPYTDGAKLVEPEWFKWSQQKRNEEAKKLLAEAGFTADKPLTFDLLYNTSDLHKKLAIAVASIWKKNLGVNVNLENQEWKTFLDTRHQGTFDVARAGWCADYNEPTSFLNTMLSDSSNNTAHYKSPAFDKLIADTLKVADDTQRSELYAKAEQQLDKDSAIVPVYYYVNARLVKPWVGGYTGKDPLDNIYVKNLYIIKH 2rkm A 1.8 BS02 LYS A 2 E32 G33 V34 W397 W416 T438 E32 G33 V34 W397 W416 T438 ? 0015031,0015833,0030288,0042597,0043190,0055085,1904680 remove_due_to_license_issue P06202 9245406 2002 ADVPAGVQLADKQTLVRNNGSEVQSLDPHKIEGVPESNVSRDLFEGLLISDVEGHPSPGVAEKWENKDFKVWTFHLRENAKWSDGTPVTAHDFVYSWQRLADPNTASPYASYLQYGHIANIDDIIAGKKPATDLGVKALDDHTFEVTLSEPVPYFYKLLVHPSVSPVPKSAVEKFGDKWTQPANIVTNGAYKLKNWVVNERIVLERNPQYWDNAKTVINQVTYLPISSEVTDVNRYRSGEIDMTYNNMPIELFQKLKKEIPNEVRVDPYLCTYYYEINNQKAPFNDVRVRTALKLALDRDIIVNKVKNQGDLPAYSYTPPYTDGAKLVEPEWFKWSQQKRNEEAKKLLAEAGFTADKPLTFDLLYNTSDLHKKLAIAVASIWKKNLGVNVNLENQEWKTFLDTRHQGTFDVARAGWCADYNEPTSFLNTMLSDSSNNTAHYKSPAFDKLIADTLKVADDTQRSELYAKAEQQLDKDSAIVPVYYYVNARLVKPWVGGYTGKDPLDNIYVKNLYIIKH 2rkn A 1.6 BS03 LP3 A 1 N13 K16 F40 L43 F55 P75 N13 K16 F40 L43 F55 P75 ? 0005504,0005515,0005783,0006869,0006952,0008270,0008289,0009506,0009627,0009862,0046872,0048046,0070161,0099503 Kd=0.06uM remove_due_to_license_issue Q8W453 18552128 101 AIDLCGMSQDELNECKPAVSKENPTSPSQPCCTALQHADFACLCGYKNSPWLGSFGVDPELASALPKQCGLANAPTC 2rkn A 1.6 BS04 LP3 A 2 Q9 K47 W51 P59 A62 S63 C77 Q9 K47 W51 P59 A62 S63 C77 ? 0005504,0005515,0005783,0006869,0006952,0008270,0008289,0009506,0009627,0009862,0046872,0048046,0070161,0099503 Kd=0.06uM remove_due_to_license_issue Q8W453 18552128 102 AIDLCGMSQDELNECKPAVSKENPTSPSQPCCTALQHADFACLCGYKNSPWLGSFGVDPELASALPKQCGLANAPTC 2rku A 1.95 BS02 R78 A 1 R57 L59 C67 A80 V114 E131 C133 R136 F183 R21 L23 C31 A44 V78 E95 C97 R100 F147 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=8nM remove_due_to_license_issue IC50=0.830000nM, Kd=0.190000nM, Ki=<1nM P53350 18005335 500 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAPS 2rl5 A 2.65 BS01 2RL A 1 L840 V848 A866 E885 L889 T916 F918 C919 L1019 L1035 C1045 D1046 F1047 L26 V31 A49 E68 L72 T99 F101 C102 L152 L168 C178 D179 F180 D1028 A1030 R1032 N1033 D1046 D1064 D161 A163 R165 N166 D179 D183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=0.5nM P35968 18311900 501 EHAERLPYDASKWEFPRDRLKLGKPLGRGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHH 2rok A -1.00 BS01 7MG A 1 W449 K450 W468 D470 W27 K28 W46 D48 3.1.13.4 0003676,0003723,0004535,0005634,0005737,0006402,0046872 remove_due_to_license_issue Q8VDG3 18641416 523 GSSGSSGGPDLQPKRDHVLHVTFPKEWKTSDLYQLFSAFGNIQISWIDDTSAFVSLSQPEQVQIAVNTSKYAESYRIQTYAEYVGKKQKGKQVKSGPSSG 2rok A -1.00 BS02 GDP A 1 K447 D471 K25 D49 3.1.13.4 0003676,0003723,0004535,0005634,0005737,0006402,0046872 remove_due_to_license_issue Q8VDG3 18641416 524 GSSGSSGGPDLQPKRDHVLHVTFPKEWKTSDLYQLFSAFGNIQISWIDDTSAFVSLSQPEQVQIAVNTSKYAESYRIQTYAEYVGKKQKGKQVKSGPSSG 2rox A 2.0 BS01 T44 A 1 A108 A109 L110 A99 A100 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=10500nM P02766 15299640 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNPKE 2rox B 2.0 BS01 T44 B 1 A108 A109 L110 T119 A99 A100 L101 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=10500nM P02766 15299640 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 2rqc A -1.00 BS01 rna B 0 Q394 F404 Y406 Q410 S429 A430 K431 F433 I434 K436 K442 F446 S448 K473 K477 R478 Q19 F29 Y31 Q35 S54 A55 K56 F58 I59 K61 K67 F71 S73 K98 K102 R103 ? 0003676,0003723 remove_due_to_license_issue Q92879 19553194 491 ~ 496 GSSGSSGLTQQSIGAAGSQKEGPEGANLFIYHLPQEFGDQDLLQMFMPFGNVVSAKVFIDKQTNLSKCFGFVSYDNPVSAQAAIQSMNGFQIGMKRLKVQLKRSKNDSKSGPSSG 2rra A -1.00 BS01 rna B 0 R111 F123 G124 G160 F161 F163 Y165 R187 R188 R190 D192 S194 I195 T196 K197 R198 R9 F21 G22 G58 F59 F61 Y63 R85 R86 R88 D90 S92 I93 T94 K95 R96 ? 0003676,0003723 remove_due_to_license_issue P62995 20926394 1 ~ 6 GSSGSSGNRANPDPNCCLGVFGLSLYTTERDLREVFSKYGPIADVSIVYDQQSRRSRGFAFVYFENVDDAKEAKERANGMELDGRRIRVDFSITKRPHT 2ru3 A -1.00 BS01 rna B 0 K36 F38 G40 G41 L42 P43 Y44 I67 D69 R70 R76 Y78 F80 R103 N106 N108 A110 G113 A114 K115 R117 K18 F20 G22 G23 L24 P25 Y26 I49 D51 R52 R58 Y60 F62 R85 N88 N90 A92 G95 A96 K97 R99 ? 0003676,0003723 remove_due_to_license_issue O45189 25132178 7 ~ 12 GSTNAEPVVGSRDTMFTKIFVGGLPYHTSDKTLHEYFEQFGDIEEAVVITDRNTQKSRGYGFVTMKDRASAERACKDPNPIIDGRKANVNLAYLGAKPRTNVQ 2sim A 1.6 BS01 DAN A 1 R37 I38 D62 M99 D100 W128 R246 R309 Y342 R36 I37 D61 M98 D99 W127 R245 R308 Y341 S61 D62 E231 Y342 S60 D61 E230 Y341 3.2.1.18 0004308,0005737,0006689,0009313,0016020,0016798,0043231 Ki=0.38mM remove_due_to_license_issue P29768 8656428 800 TVEKSVVFKAEGEHFTDQKGNTIVGSGSGGTTKYFRIPAMCTTSKGTIVVFADARHNTASDQSFIDTAAARSTDGGKTWNKKIAIYNDRVNSKLSRVMDPTCIVANIQGRETILVMVGKWNNNDKTWGAYRDKAPDTDWDLVLYKSTDDGVTFSKVETNIHDIVTKNGTISAMLGGVGSGLQLNDGKLVFPVQMVRTKNITTVLNTSFIYSTDGITWSLPSGYCEGFGSENNIIEFNASLVNNIRNSGLRRSFETKDFGKTWTEFPPMDKKVDNRNHGVQGSTITIPSGNKLVAAHSSAQNKNNDYTRSDISLYAHNLYSGEVKLIDDFYPKVGNASGAGYSCLSYRKNVDKETLYVVYEANGSIEFQDLSRHLPVIKSYN 2ssp E 2.25 BS01 dna A 0 D145 S169 G246 S247 H268 S270 P271 S273 R276 D64 S88 G165 S166 H187 S189 P190 S192 R195 3.2.2.27 0004844,0006281,0006284,0016799 remove_due_to_license_issue P13051 9724657 1 ~ 10 MEFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPASVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 2ssp E 2.25 BS02 dna B 0 P271 Y275 P190 Y194 3.2.2.27 0004844,0006281,0006284,0016799 remove_due_to_license_issue P13051 9724657 21 ~ 31 MEFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPASVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 2std A 2.1 BS01 CRP A 1 W26 Y50 V75 L76 F158 W18 Y42 V67 L68 F150 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Kd=0.14nM remove_due_to_license_issue Ki=30nM P56221 9665698 175 DEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFG 2tmn E 1.6 BS06 0FA E 1 N112 A113 E143 H146 E166 R203 H231 N112 A113 E143 H146 E166 R203 H231 3.4.24.27 0004222,0006508 Ki=1.3uM remove_due_to_license_issue Ki=21300nM, Kd=1288nM P00800 3709536 322 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 2toh A 2.3 BS02 HBI A 1 V291 L294 L295 X300 P327 E332 Y371 V129 L132 L133 X138 P165 E170 Y209 H331 H336 E376 S395 H169 H174 E214 S233 1.14.16.2 0004497,0005506,0009072,0016714 Ki=70uM remove_due_to_license_issue P04177 9753429 500 REDKVPWFPRKVSELDKCHHLVTPDLDLDHPGFSDQVYRQRRKLIAEIAFQYKHGEPIPHVEYTAEEIATWKEVYVTLKGLYATHACREHLEGFQLLERYCGYREDSIPQLEDVSRFLKERTGFQLRPVAGLLSARDYLASLAFRVFQCTQYIRHASSPMHSPEPDCCHELLGHVPMLADRTFAQFSQDIGLASLGASDEEIEKLSTVYWFTVEFGLCKQNGELKAYGAGLLSSYGELLHSLSEEPEVRAFDPDTAAVQPYQDQTYQPVYFVSESFNDAKDKLRNYASRIQRPFSVKFDPYTLAIDVLDSPHTIQRSLEGVQDELHTLAHALSAIS 2tpi Z 2.1 BS01 ILE Z 1 I138 G142 N143 T144 K156 D189 D194 I115 G119 N120 T121 K133 D168 D173 G193 S195 G196 G172 S174 G175 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 1016 GYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2tpi Z 2.1 BS02 VAL Z 1 G19 T144 K188 D189 G1 T121 K167 D168 G193 S195 G196 G172 S174 G175 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 1017 GYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2tsr A 2.6 BS02 D16 A 1 R72 I102 D212 G216 F219 Y252 R52 I82 D192 G196 F199 Y232 E81 W103 Y129 C189 R209 D212 E61 W83 Y109 C169 R189 D192 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0097421,1901363,1990825 remove_due_to_license_issue P45352 9894005 309 QHGELQYLRQVEHIMRCGFKKEDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVRIWDANGSRDFLDSLGFSARQEGDLGPVYGFQWRHFGADYKDMDSDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPKDLPLMALPPCHALCQFYVVNGELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLQPGDFVHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVETIDDFKVEDFQIEGYNPHPTI 2tsr B 2.6 BS02 D16 B 1 R101 I102 W103 D212 G216 F219 Y252 R81 I82 W83 D192 G196 F199 Y232 E81 W103 Y129 C189 R209 D212 E61 W83 Y109 C169 R189 D192 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0097421,1901363,1990825 remove_due_to_license_issue P45352 9894005 409 QHGELQYLRQVEHIMRCGFKKEDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVRIWDANGSRDFLDSLGFSARQEGDLGPVYGFQWRHFGADYKDMDSDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPKDLPLMALPPCHALCQFYVVNGELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLQPGDFVHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVETIDDFKVEDFQIEGYNPHPTI 2upj A 3.0 BS01 U02 A 1 D25 A28 D29 D30 G48 G49 I50 D25 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 7658450 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2upj B 3.0 BS01 U02 A 1 D25 A28 D29 D30 G49 P81 V82 D25 A28 D29 D30 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 7658450 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2usn A 2.2 BS06 IN8 A 1 F86 Y155 H166 A167 Y168 A169 E202 H205 H211 F4 Y73 H84 A85 Y86 A87 E120 H123 H129 H201 E202 H205 H211 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 Ki=0.31uM remove_due_to_license_issue P08254 9792098 300 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYG 2uue A 2.06 BS01 MTZ A 1 I10 A31 K33 F80 E81 F82 L83 H84 Q85 D86 K89 L134 I10 A31 K33 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 17051658 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2uuo A 2.5 BS01 LK3 A 1 G12 R37 G73 H183 K348 A414 S415 L416 N421 F422 G12 R37 G73 H183 K339 A405 S406 L407 N412 F413 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=170uM remove_due_to_license_issue IC50=170000nM P14900 19007109 1441 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPRCVSFGVNMGDYHLNHETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGS 2uup A 1.88 BS01 LK4 A 1 D35 T36 R37 G73 H183 K348 A414 S415 L416 N421 F422 H439 D35 T36 R37 G73 H183 K348 A414 S415 L416 N421 F422 H439 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=105uM remove_due_to_license_issue IC50=105000nM P14900 19007109 1440 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRGADERCVSFGVNMGDYHLNHQQGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2uvm A 1.94 BS01 GVF A 1 K14 G16 E17 Y18 R23 R25 N53 F55 R86 E115 K14 G16 E17 Y18 R23 R25 N53 F55 R86 E115 2.7.11.1 remove_due_to_license_issue Ki=80nM P31749 17432822 1116 MSDVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDVDQREAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKQEE 2uw0 A 2.0 BS02 GVK A 1 G50 T51 G52 G55 R56 V57 A70 E121 Y122 A123 E127 E170 N171 M173 T183 D184 F327 G37 T38 G39 G42 R43 V44 A57 E108 Y109 A110 E114 E157 N158 M160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 17451235 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uw3 A 2.19 BS02 GVG A 1 L49 V57 A70 M120 Y122 M173 T183 L36 V44 A57 M107 Y109 M160 T170 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=80uM remove_due_to_license_issue P00517 17451234 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uw4 A 2.0 BS02 L15 A 1 V57 A70 E121 Y122 A123 E170 M173 T183 V43 A56 E107 Y108 A109 E156 M159 T169 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=5.2uM remove_due_to_license_issue P00517 17451234 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uw5 A 2.14 BS02 GVN A 1 G50 T51 V57 A70 E121 Y122 E170 N171 M173 T183 D184 G36 T37 V43 A56 E107 Y108 E156 N157 M159 T169 D170 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=34nM remove_due_to_license_issue P00517 17451234 1351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uw6 A 2.23 BS02 GVO A 1 G50 T51 V57 A70 Y122 E127 E170 M173 T183 D184 Y330 G37 T38 V44 A57 Y109 E114 E157 M160 T170 D171 Y317 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=0.28uM remove_due_to_license_issue P00517 17451234 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uw7 A 2.1 BS02 GVP A 1 G50 G52 G55 R56 V57 A70 E121 E127 E170 M173 T183 D184 G37 G39 G42 R43 V44 A57 E108 E114 E157 M160 T170 D171 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=18nM remove_due_to_license_issue P00517 17451234 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uw8 A 2.0 BS02 GVQ A 1 G50 T51 G55 R56 V57 E170 G37 T38 G42 R43 V44 E157 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=77uM remove_due_to_license_issue P00517 17451234 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2uwd A 1.9 BS03 2GG A 1 N51 S52 A55 D93 I96 G97 M98 D102 L107 G108 F138 T184 V186 N36 S37 A40 D78 I81 G82 M83 D87 L92 G93 F123 T169 V171 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=4.5nM remove_due_to_license_issue P07900 17431102 1228 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2uwl A 1.9 BS01 895 A 1 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=4nM remove_due_to_license_issue Ki=4nM P00742 17420122 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2uwm A 2.31 BS01 rna C 0 A596 R599 S605 R606 K607 L610 R624 D627 R629 A156 R159 S165 R166 K167 L170 R184 D187 R189 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q2RFK4 17502103 13 ~ 35 QAWWQAVTRALEEFHSRYPLRPGLAREELRSRYFSRLPARVYQALLEEWSREGRLQLAANTVALAGFTPSFSETQKKLLKDLEDKYRVSRWQPPSFKEVAGSFNLDPSELEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRRVGDKRVVVG 2uwm A 2.31 BS02 rna D 0 R457 Y458 R461 N500 E551 E552 H555 V558 R559 Q618 R17 Y18 R21 N60 E111 E112 H115 V118 R119 Q178 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q2RFK4 17502103 13 ~ 35 QAWWQAVTRALEEFHSRYPLRPGLAREELRSRYFSRLPARVYQALLEEWSREGRLQLAANTVALAGFTPSFSETQKKLLKDLEDKYRVSRWQPPSFKEVAGSFNLDPSELEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRRVGDKRVVVG 2uwm B 2.31 BS01 rna C 0 R457 Y458 R461 E552 H555 Q618 R27 Y28 R31 E122 H125 Q188 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q2RFK4 17502103 13 ~ 35 DLYAISTERYQAWWQAVTRALEEFHSRYPLRPGLAREELRSRYFSRLPARVYQALLEEWSREGRLQLAANTVALAGFTPSFSETQKKLLKDLEDKYRVSRWQPPSFKEVAGSFNLDPSELEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRRVGDKRVVVG 2uwm B 2.31 BS02 rna D 0 R599 S605 R606 K607 L610 R624 R629 R169 S175 R176 K177 L180 R194 R199 ? 0001514,0003723,0003746,0005525,0005737 remove_due_to_license_issue Q2RFK4 17502103 13 ~ 35 DLYAISTERYQAWWQAVTRALEEFHSRYPLRPGLAREELRSRYFSRLPARVYQALLEEWSREGRLQLAANTVALAGFTPSFSETQKKLLKDLEDKYRVSRWQPPSFKEVAGSFNLDPSELEELLHYLVREGVLVKINDEFYWHRQALGEAREVIKNLASTGPFGLAEARDALGSSRKYVLPLLEYLDQVKFTRRVGDKRVVVG 2uwo A 1.75 BS01 701 A 1 E97 T98 Y99 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 E81 T82 Y83 D177 A178 Q180 V201 W203 G204 G206 C207 G214 I215 Y216 H57 D102 Q192 G193 D194 S195 G196 H42 D86 Q180 G181 D182 S183 G184 3.4.21.6 0004252,0006508 Ki=2nM remove_due_to_license_issue Ki=2nM P00742 17420122 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2uwp A 1.75 BS01 894 A 1 E97 T98 Y99 F174 A190 Q192 V213 W215 G216 G226 I227 Y228 E83 T84 Y85 F162 A180 Q182 V203 W205 G206 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=154nM remove_due_to_license_issue Ki=154nM P00742 17420122 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2uxi A 2.5 BS01 G50 A 1 A74 S77 E78 C137 A70 S73 E74 C133 ? 0000976,0001217,0003677,0003700,0006355,0032993,0045892 Kd=0.05uM remove_due_to_license_issue Q9AIU0 17466326 1211 TKEEAQETRAQIIEAAERAFYKRGVARTTLADIAELAGVTRGAIYWHFNNKAELVQALLDSLHETHDHLARASESEDEVDPLGCMRKLLLQVFNELVLDARTRRINEILHHKCEFTDDMCEIRQQRQSAVLDCHKGITLALANAVRRGQLPGELDAERAAVAMFAYVDGLIRRWLLLPDSVDLLGDVEKWVDTGLDMLRLSPALRK 2uxi B 2.5 BS01 G50 B 1 L66 R130 D172 L61 R125 D167 ? 0000976,0001217,0003677,0003700,0006355,0032993,0045892 Kd=0.05uM remove_due_to_license_issue Q9AIU0 17466326 1211 KEEAQETRAQIIEAAERAFYKRGVARTTLADIAELAGVTRGAIYWHFNNKAELVQALLDSLHETHDHLARASESEDEVDPLGCMRKLLLQVFNELVLDARTRRINEILHHKCEFTDDMCEIRQQRQSAVLDCHKGITLALANAVRRGQLPGELDAERAAVAMFAYVDGLIRRWLLLPDSVDLLGDVEKWVDTGLDMLRLSPALRK 2uxi B 2.5 BS02 G50 B 2 A74 S77 E78 M89 I141 F168 V171 I175 A69 S72 E73 M84 I136 F163 V166 I170 ? 0000976,0001217,0003677,0003700,0006355,0032993,0045892 Kd=0.05uM remove_due_to_license_issue Q9AIU0 17466326 1212 KEEAQETRAQIIEAAERAFYKRGVARTTLADIAELAGVTRGAIYWHFNNKAELVQALLDSLHETHDHLARASESEDEVDPLGCMRKLLLQVFNELVLDARTRRINEILHHKCEFTDDMCEIRQQRQSAVLDCHKGITLALANAVRRGQLPGELDAERAAVAMFAYVDGLIRRWLLLPDSVDLLGDVEKWVDTGLDMLRLSPALRK 2uxu A 2.3 BS01 NAR A 1 L93 N110 I141 M167 I175 L89 N106 I137 M163 I171 ? 0000976,0001217,0003677,0003700,0006355,0032993,0045892 Kd=18uM remove_due_to_license_issue Q9AIU0 17466326 1211 TKEEAQETRAQIIEAAERAFYKRGVARTTLADIAELAGVTRGAIYWHFNNKAELVQALLDSLHETHDHLARASESEDEVDPLGCMRKLLLQVFNELVLDARTRRINEILHHKCEFTDDMCEIRQQRQSAVLDCHKGITLALANAVRRGQLPGELDAERAAVAMFAYVDGLIRRWLLLPDSVDLLGDVEKWVDTGLDMLRLSPALRK 2uxx A 2.74 BS01 FAJ A 1 G285 G287 S289 E308 A309 R310 G315 R316 G330 A331 M332 V333 T335 V590 L625 P626 W751 W756 S760 Y761 G800 E801 T810 V811 G115 G117 S119 E138 A139 R140 G145 R146 G160 A161 M162 V163 T165 V420 L455 P456 W581 W586 S590 Y591 G630 E631 T640 V641 T335 D553 K661 T165 D383 K491 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 17569509 900 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYT 2uxz A 1.75 BS01 HI1 A 1 R8 L23 D25 G27 A28 D29 G48 G49 I50 V82 R8 L23 D25 G27 A28 D29 G48 G49 I50 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.3nM remove_due_to_license_issue P03366 18215014 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2uxz B 1.75 BS01 HI1 A 1 D125 G127 A128 D129 D130 G148 I150 P181 V182 D25 G27 A28 D29 D30 G48 I50 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 18215014 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2uy0 A 1.76 BS01 HV1 B 1 R8 D25 G27 D29 I47 G48 G49 I50 P81 V82 R8 D25 G27 D29 I47 G48 G49 I50 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 18215014 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2uy0 B 1.76 BS01 HV1 B 1 R108 L123 D125 G127 A128 D129 D130 V132 G148 I150 P181 V182 R8 L23 D25 G27 A28 D29 D30 V32 G48 I50 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=120nM remove_due_to_license_issue P03366 18215014 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2uy3 A 1.9 BS01 H33 A 1 Y32 F60 A110 D155 E157 Q212 Y214 W285 Y7 F35 A85 D130 E132 Q187 Y189 W260 3.2.1.14 0004553,0005975 Ki=600uM remove_due_to_license_issue Ki=340000nM P29029 17524989 1311 NTNIAVYWGQNSAGTQESLATYCESSDADIFLLSFLNQFPTLGLNFANACSDTFSDGLLHCTQIAEDIETCQSLGKKVLLSLGGASGSYLFSDDSQAETFAQTLWDTFGEGTGASERPFDSAVVDGFDFDIENNNEVGYSALATKLRTLFAEGTKQYYLSAAPQCPYPDASVGDLLENADIDFAFIQFYNNYCSVSGQFNWDTWLTYAQTVSPNKNIKLFLGLPGSASAAGSGYISDTSLLESTIADIASSSSFGGIALWDASQAFSNELNGEPYVEILKNLLTS 2uy4 A 1.75 BS01 AZM A 1 F60 A110 D155 Q212 Y214 W285 L307 S310 F34 A84 D129 Q186 Y188 W259 L280 S283 3.2.1.14 0004553,0005975 Ki=21uM remove_due_to_license_issue Ki=21000nM P29029 17524989 1311 TNIAVYWGQNSAGTQESLATYCESSDADIFLLSFLNQFPTLGLNFANACSDTFSDGLLHCTQIAEDIETCQSLGKKVLLSLGGASGSYLFSDDSQAETFAQTLWDTFGEGTGASERPFDSAVVDGFDFDIENNNEVGYSALATKLRTLFAEGTKQYYLSAAPQCPYPDASVGDLLENADIDFAFIQFYNNYCSVSGQFNWDTWLTYAQTVSPNKNIKLFLGLPGSASAAGSGYISDTSLLESTIADIASSSSFGGIALWDASQAFSNELGEPYVEILKNLLTS 2uy5 A 1.6 BS01 H35 A 1 Y32 D155 E157 F210 Q212 Y214 A283 W285 Y7 D130 E132 F185 Q187 Y189 A258 W260 3.2.1.14 0004553,0005975 Ki=3.2uM remove_due_to_license_issue Ki=3200nM P29029 17524989 1313 NTNIAVYWGQNSAGTQESLATYCESSDADIFLLSFLNQFPTLGLNFANACSDTFSDGLLHCTQIAEDIETCQSLGKKVLLSLGGASGSYLFSDDSQAETFAQTLWDTFGEGTGASERPFDSAVVDGFDFDIENNNEVGYSALATKLRTLFAEGTKQYYLSAAPQCPYPDASVGDLLENADIDFAFIQFYNNYCSVSGQFNWDTWLTYAQTVSPNKNIKLFLGLPGSASAAGSGYISDTSLLESTIADIASSSSFGGIALWDASQAFSNELEPYVEILKNLLTSAS 2uyi A 2.1 BS02 K02 A 1 E116 E118 R119 W127 A133 I136 P137 Y211 L214 E215 G217 R221 F239 E101 E103 R104 W112 A118 I121 P122 Y196 L199 E200 G202 R206 F224 ? 0003777,0005524,0007018,0008017 ic50=0.48uM remove_due_to_license_issue IC50=480nM P52732 17498954 604 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2uym A 2.11 BS02 K03 A 1 E116 E118 R119 W127 A133 I136 P137 Y211 L214 E215 G217 R221 F239 E101 E103 R104 W112 A118 I121 P122 Y196 L199 E200 G202 R206 F224 ? 0003777,0005524,0007018,0008017 ic50=3.1uM remove_due_to_license_issue IC50=3100nM P52732 17498954 604 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 2uyn A 1.6 BS01 2KT A 1 F84 R105 S106 C107 F83 R104 S105 C106 3.5.4.- 0005829,0006566,0016787,0019239,0042802,0070689 remove_due_to_license_issue P0AGL2 17506874 1129 KKIIETQRAPGAIGPYVQGVDLGSMVFTSGQIPVCPQTGEIPADVQDQARLSLENVKAIVVAAGLSVGDIIKMTVFITDLNDFATINEVYKQFFDEHQATYPTRSCVQVARLPKDVKLEIEAIAVRS 2uyn B 1.6 BS01 2KT A 1 Y17 E120 Y16 E119 3.5.4.- 0005829,0006566,0016787,0019239,0042802,0070689 remove_due_to_license_issue P0AGL2 17506874 1129 KKIIETQRAPGAIGPYVQGVDLGSMVFTSGQIPVCPQTGEIPADVQDQARLSLENVKAIVVAAGLSVGDIIKMTVFITDLNDFATINEVYKQFFDEHQATYPTRSCVQVARLPKDVKLEIEAIAVRS 2uyn B 1.6 BS02 2KT B 1 F84 R105 S106 C107 F83 R104 S105 C106 3.5.4.- 0005829,0006566,0016787,0019239,0042802,0070689 remove_due_to_license_issue P0AGL2 17506874 1129 KKIIETQRAPGAIGPYVQGVDLGSMVFTSGQIPVCPQTGEIPADVQDQARLSLENVKAIVVAAGLSVGDIIKMTVFITDLNDFATINEVYKQFFDEHQATYPTRSCVQVARLPKDVKLEIEAIAVRS 2uyq A 1.8 BS01 SAM A 1 A110 D132 D161 L162 R163 A85 D107 D136 L137 R138 2.1.1.- 0008168,0032259 Kd=2.1uM remove_due_to_license_issue Q9CCZ4 17660248 1311 VGTTAVMVAAARAAETDRPDALIRDPYAKLLVTNTGAGALWEAMDAEAAAMVEHMRSYQAVRTNFFDTYFNNAVIDGIRQFVILASGLDSRAYRLDWPTGTTVYEIDQPKVLAYKSTTLAEHGVTPTADRREVPIDLRQDWPPALRSAGFDPSARTAWLAEGLLMYLPATAQDGLFTEIGGLSAVGSRIAVETSPLHGDEWREQMQLRFRRVSDALIYHDENRAVVADWLNRHGWRATAQSAPDEMRRVGRWGDGVPMADDKDAFAEFVTAHRL 2uyw A 1.7 BS01 BTN A 1 L16 S18 Y35 T37 V39 S40 L41 W69 F71 S72 S74 T76 W78 W96 L13 S15 Y32 T34 V36 S37 L38 W66 F68 S69 S71 T73 W75 W93 ? 0009374 remove_due_to_license_issue A7YYL1 19788720 1123 QKCNLQGQWRNKLGSNLIIESVSQNGEFTGTYFTSVSLTNSTIRISPLTGYQKLTEKPTFGFTVHWAFSDSITVWTGQCFLNEKGEEILHTMWLLRSSQEKEQDNWTGTRVGANTFTRL 2uyw D 1.7 BS01 BTN D 1 L16 S18 Y35 T37 V39 S40 L41 W69 F71 S72 S74 T76 W78 W96 L12 S14 Y31 T33 V35 S36 L37 W65 F67 S68 S70 T72 W74 W92 ? 0009374 remove_due_to_license_issue A7YYL1 19788720 1124 KCNLQGQWRNKLGSNLIIESVSQNGEFTGTYFTSVSLTNSTIRISPLTGYQKLTEKPTFGFTVHWAFSDSITVWTGQCFLNEKGEEILHTMWLLRSSQEKEQDNWTGTRVGANTFTRLS 2uz9 A 2.3 BS02 XAN A 1 H84 L99 L103 R213 F214 H240 E243 D330 H77 L92 L96 R206 F207 H233 E236 D323 3.5.4.3 0000255,0005829,0006139,0006147,0006161,0007399,0008270,0008892,0016787,0016810,0043605,0046038,0046055,0046098,0046872 remove_due_to_license_issue Q9Y2T3 1453 PLAHIFRGTFVHSTWTCPMEVLRDHLLGVSDSGKIVFLEEASQQEKLAKEWCFKPCEIRELSHHEFFMPGLVDTHIHASQYSFAGSSIDLPLLEWLTKYTFPAEHRFQNIDFAEEVYTRVVRRTLKNGTTTACYFATIHTDSSLLLADITDKFGQRAFVGKVCMDLNDTFPEYKETTEESIKETERFVSEMLQKNYSRVKPIVTPRFSLSCSETLMGELGNIAKTRDLHIQSHISENRDEVEAVKNLYPSYKNYTSVYDKNNLLTNKTVMAHGCYLSAEELNVFHERGASIAHCPNSNLSLSSGFLNVLEVLKHEVKIGLGTDVAGGYSYSMLDAIRRAVMVSNILLINKVNEKSLTLKEVFRLATLGGSQALGLDGEIGNFEVGKEFDAILINPKASDSPIDLFYGDFFGDISEAVIQKFLYLGDDRNIEEVYVGGKQVVPFS 2uzb A 2.7 BS01 C75 A 1 I10 A31 K33 F80 D86 K89 L134 D145 I10 A31 K33 F80 D86 K89 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=120nM P24941 17570665 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2uzd A 2.72 BS01 C85 A 1 I10 F80 L83 Q85 D86 K89 L134 D145 I10 F80 L83 Q85 D86 K89 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=180nM P24941 17570665 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2uze A 2.4 BS01 C95 A 1 I10 A31 K33 F80 L83 H84 Q85 L134 D145 I10 A31 K33 F80 L83 H84 Q85 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=47uM remove_due_to_license_issue IC50=47000nM P24941 17570665 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2uzj A 1.55 BS01 E64 A 1 Q17 C47 D130 G136 S137 Q187 G194 H195 Q17 C47 D130 G136 S137 Q187 G194 H195 C47 H195 W212 C47 H195 W212 3.4.22.10 0006508,0008234 remove_due_to_license_issue P0C0J0 19712682 1254 QPVVKSLLDSKGIHYNQGNPYNLLTPVIEKVKPGEQSFVGQHAATGCVATATAQIMKYHNYPNKGLKDYTYTLSSNNPYFNHPKNLFAAISTRQYNWNNILPTYSGRESNVQKMAISELMADVGISVDMDYGPSSGSAGSSRVQRALKENFGYNQSVHQINRSDFSKQDWEAQIDKELSQNQPVYYQGVGKVGGHAFVIDGADGRNFYHVNWGWGGVSDGFFRLDALNPSALGAGGFNGYQSAVVGIKP 2uzl A 2.4 BS01 C94 A 1 I10 A31 K33 F80 F82 L83 H84 Q85 D86 L134 D145 I10 A31 K33 F80 F82 L83 H84 Q85 D86 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.61uM remove_due_to_license_issue IC50=610nM P24941 17570665 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2uzn A 2.3 BS01 C96 A 1 A31 F80 L83 H84 D86 K89 L134 D145 A31 F71 L74 H75 D77 K80 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.03uM remove_due_to_license_issue IC50=30nM P24941 17570665 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2uzo A 2.3 BS01 C62 A 1 I10 A31 K33 F80 L83 H84 Q85 D86 K89 L134 D145 I10 A31 K33 F74 L77 H78 Q79 D80 K83 L128 D139 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=27uM remove_due_to_license_issue IC50=27000nM P24941 17570665 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2uzv A 2.5 BS02 SS5 A 1 T51 G52 A70 K72 V104 M120 E121 Y122 V123 N171 L173 T183 D184 F327 T37 G38 A56 K58 V90 M106 E107 Y108 V109 N157 L159 T169 D170 F313 N171 D184 N157 D170 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50>3uM remove_due_to_license_issue IC50=>3000nM P00517 17523610 1351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2v00 A 1.55 BS01 V15 A 1 D33 D35 Y79 D81 F116 D219 G221 D33 D35 Y79 D81 F116 D219 G221 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Kd=0.22mM remove_due_to_license_issue Kd=220000nM P11838 17985861 1336 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 2v0c A 1.85 BS05 ANZ A 1 F246 T247 T248 R249 V328 L329 Y332 I337 M338 H343 D344 F243 T244 T245 R246 V325 L326 Y329 I334 M335 H340 D341 F41 H49 H52 D80 C159 C162 F501 H541 F551 V637 K640 F38 H46 H49 D77 C156 C159 F498 H538 F548 V634 K637 6.1.1.4 0000166,0002161,0004812,0004823,0005524,0005737,0005829,0006412,0006418,0006429,0046872,0106074 remove_due_to_license_issue Q7SIE4 17588934 1817 MEKYNPHAIEAKWQRFWEEKGFMKAKDLPGKQYVLVMFPYPSGDLHMGHLKNYTMGDVLARFRRMQGYEVLHPMGWDAFGLPAENAALKFGVHPKDWTYANIRQAKESLRLMGILYDWDREVTTCEPEYYRWNQWIFLKMWEKGLAYRAKGLVNWCPKCQTVLANEQVVEGRCWRHEDTPVEKRELEQWYLRITAYAERLLKDLEGLNWPEKVKAMQRAWIGRSEGAEILFPVEGKEVRIPVFTTRPDTLFGATFLVLAPEHPLTLELAAPEKREEVLAYVEAAKRKTEIERQAEGREKTGVFLGAYALNPATGERIPIWTADYVLFGYGTGAIMAVPAHDQRDYEFARKFGLPIKKVIERPGEPLPEPLERAYEEPGIMVNSGPFDGTESEEGKRKVIAWLEEKGLGKGRVTYRLRDWLISRQRYWGTPIPMVHCEACGVVPVPEEELPVLLPDLKDVEDIRPKGKSPLEAHPEFYETTCPKCGGPAKRDTDTMDTFFDSSWYYLRYTDPHNDRLPFDPEKANAWMPVDQYIGGVEHAVLHLLYSRFFTKFLHDLGMVKVEEPFQGLFTQGMVLAWTDFGPVEVEGSVVRLPEPTRIRLEIPESALSLEDVRKMGAELRPHEDGTLHLWKPAVMSKSKGNGVMVGPFVKEQGADIARITILFAAPPENEMVWTEEGVQGAWRFLNRIYRRVAEDREALLETSGVFQAEALEGKDRELYGKLHETLKKVTEDLEALRFNTAIAALMEFLNALYEYRKDRPVTPVYRTAIRYYLQMLFPFAPHLAEELWHWFWPDSLFEAGWPELDEKALE 2v0n A 2.71 BS03 C2E A 1 R359 D362 D383 I387 R390 R358 D361 D382 I386 R389 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 remove_due_to_license_issue B8GZM2 17697997 503 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAHHHHHH 2v0n A 2.71 BS04 C2E A 2 N357 R359 R390 N356 R358 R389 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 remove_due_to_license_issue B8GZM2 17697997 505 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAHHHHHH 2v0n A 2.71 BS08 C2E B 2 R313 L316 R312 L315 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 remove_due_to_license_issue B8GZM2 17697997 505 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAHHHHHH 2v0n B 2.71 BS01 C2E A 2 R313 L316 R312 L315 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 remove_due_to_license_issue B8GZM2 17697997 505 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAH 2v0n B 2.71 BS04 C2E B 1 R359 D362 D383 I387 R390 R358 D361 D382 I386 R389 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 remove_due_to_license_issue B8GZM2 17697997 503 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAH 2v0n B 2.71 BS05 C2E B 2 N357 R359 R390 N356 R358 R389 2.7.7.65 0000160,0005525,0005737,0005886,0016740,0030154,0043709,0046872,0052621,1902201 remove_due_to_license_issue B8GZM2 17697997 505 SARILVVDDIEANVRLLEAKLTAEYYEVSTAMDGPTALAMAARDLPDIILLDVMMPGMDGFTVCRKLKDDPTTRHIPVVLITALDGRGDRIQGLESGASDFLTKPIDDVMLFARVRSLTRFKLVIDELRQREASGRRMGVIAGAAARLDGLGGRVLIVDDNERQAQRVAAELGVEHRPVIESDPEKAKISAGGPVDLVIVNAAAKNFDGLRFTAALRSEERTRQLPVLAMVDPDDRGRMVKALEIGVNDILSRPIDPQELSARVKTQIQRKRYTDYLRNNLDHSLELAVTDQLTGLHNRRYMTGQLDSLVKRATLGGDPVSALLIDIDFFKKINDTFGHDIGDEVLREFALRLASNVRAIDLPCRYGGEEFVVIMPDTALADALRIAERIRMHVSGSPFTVAHGREMLNVTISIGVSATAGEGDTPEALLKRADEGVYQAKASGRNAVVGKAAH 2v0z C 2.2 BS01 C41 C 1 T12 Q13 Y14 V30 D32 G34 R74 Y75 F117 V120 D215 G217 A218 S219 T18 Q19 Y20 V36 D38 G40 R82 Y83 F124 V127 D224 G226 A227 S228 3.4.23.15 0004190,0006508 ic50=0.0006uM remove_due_to_license_issue IC50=0.6nM P00797 10903938 1328 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2v10 C 3.1 BS01 C61 C 1 Q19 Y20 V36 D38 G40 R82 Y83 S84 P118 F124 V127 G228 Q16 Y17 V33 D35 G37 R79 Y80 S81 P115 F121 V124 G221 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=1nM P00797 10903938 1341 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2v11 C 3.1 BS01 C80 C 1 T18 Q19 Y20 V36 D38 S41 Y83 P118 A122 F124 D226 T227 G228 A229 S230 T15 Q16 Y17 V33 D35 S38 Y80 P115 A119 F121 D219 T220 G221 A222 S223 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=3nM P00797 10903938 1341 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2v12 C 3.2 BS01 C39 C 1 T18 Y20 D38 G40 S41 Y83 T85 A122 F124 D226 G228 A229 T15 Y17 D35 G37 S38 Y80 T82 A119 F121 D219 G221 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.9nM P00797 10903938 350 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2v13 A 2.8 BS01 C40 A 1 Q19 Y20 D38 G40 R82 Y83 T85 P118 F124 D226 G228 Q15 Y16 D34 G36 R78 Y79 T81 P114 F120 D215 G217 D38 S41 N43 W45 Y83 D226 A229 D34 S37 N39 W41 Y79 D215 A218 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=22nM P00797 10903938 1341 NTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2v16 C 2.8 BS01 C47 C 1 T12 Q13 D32 G34 S35 R74 Y75 S76 P111 A115 F117 D215 G217 A218 S219 T15 Q16 D35 G37 S38 R79 Y80 S81 P115 A119 F121 D219 G221 A222 S223 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.8nM P00797 10903938 1327 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 2v22 B 2.6 BS01 C35 B 1 M210 I213 W217 E224 R250 L253 Q254 I281 T282 M36 I39 W43 E50 R76 L79 Q80 I107 T108 ? 0016538,0044772 remove_due_to_license_issue P20248 17051658 1433 VPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAILVDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQLVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRMEHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAMFLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPESLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYKNSKYHGVSLLNPPETLNL 2v25 A 1.49 BS01 ASP A 1 K19 R67 T82 T84 R89 A131 T132 Y156 D174 I177 K17 R65 T80 T82 R87 A129 T130 Y154 D172 I175 ? remove_due_to_license_issue Q0P9X8 17631313 1234 GKLESIKSKGQLIVGVKNDVPHYALLDQATGEIKGFEVDVAKLLAKSILGDDKKIKLVAVNAKTRGPLLDNGSVDAVIATFTITPERKRIYNFSEPYYQDAIGLLVLKEKKYKSLADMKGANIGVAQAATTKKAIGEAAKKIGIDVKFSEFPDYPSIKAALDAKRVDAFSVDKSILLGYVDDKSEILPDSFEPQSYGIVTKKDDPAFAKYVDDFVKEHKNEIDALAKKWGL 2v2c A 1.89 BS01 PGA A 1 K13 H95 E167 I172 G212 S213 G234 G235 K12 H94 E166 I171 G211 S212 G233 G234 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=0.39mM remove_due_to_license_issue P04789 18219118 1254 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVLTPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 2v2h A 1.18 BS01 PGA A 1 N11 K13 H95 E167 I172 G173 G212 S213 G234 G235 N10 K12 H86 E158 I163 G164 G203 S204 G225 G226 N11 K13 H95 E97 E167 G173 S213 N10 K12 H86 E88 E158 G164 S204 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=0.17mM remove_due_to_license_issue P04789 18219118 1251 SKPQPIAAANWKSGSPDSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAGNADALASLKDFGVNWIVLGHSERRWYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVLTPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 2v2q A 2.3 BS02 NVG A 1 Y24 H25 K145 S170 T171 Y175 Y25 H26 K146 S171 T172 Y176 K9 D130 K10 D131 2.7.1.148 0005524,0008299,0016114,0016301,0019288,0050515 Ki=71.2uM remove_due_to_license_issue O67060 18033714 1274 HMIKVLSPAKINLGLWVLGRLPSGYHEILTLYQEIPFYDEIYIREGVLRVETNIGIPQEENLVYKGLREFERITGIEINYSIFIQKNIPPGAGLGGGSSNLAVVLKKVNELLGSPLSEEELRELVGSISADAPFFLLGKSAIGRGKGEVLEPVETEISGKITLVIPQVSSSTGRVYSSLREEHFVTPEYAEEKIQRIISGEVEEIENVLGDIARELYPEINEVYRFVEYLGFKPFVSGSGSTVYFFGGASEELKKAAKMRGWKVVELEL 2v2v A 2.4 BS04 V12 A 1 Y24 H25 K145 S170 T171 Y175 Y26 H27 K147 S172 T173 Y177 K9 D130 K11 D132 2.7.1.148 0005524,0008299,0016114,0016301,0019288,0050515 Ki=85.8uM remove_due_to_license_issue O67060 18033714 1277 SHMIKVLSPAKINLGLWVLGRLPSGYHEILTLYQEIPFYDEIYIREGVLRVETNIGIPQEENLVYKGLREFERITGIEINYSIFIQKNIPPGAGLGGGSSNLAVVLKKVNELLGSPLSEEELRELVGSISADAPFFLLGKSAIGRGKGEVLEPVETEISGKITLVIPQVSSSTGRVYSSLREEHFVTPEYAEEKIQRIISGEVEEIENVLGDIARELYPEINEVYRFVEYLGFKPFVSGSGSTVYFFGGASEELKKAAKMRGWKVVELEL 2v3d A 1.96 BS01 NBV A 1 D127 F128 W179 N234 E235 F246 Y313 E340 W381 N396 D125 F126 W177 N232 E233 F244 Y311 E338 W379 N394 E235 E340 C342 N370 E233 E338 C340 N368 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 Ki=116uM remove_due_to_license_issue IC50=400000nM, Ki=116000nM P04062 17666401 1503 EFARPCIPKSFGYSSVVCVCNATYCDSFDPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 2v3e A 2.0 BS01 NND A 1 D127 F128 W179 N234 E235 F246 Y313 E340 W381 N396 D128 F129 W180 N235 E236 F247 Y314 E341 W382 N397 E235 E340 C342 N370 E236 E341 C343 N371 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 Ki=0.3uM remove_due_to_license_issue Ki=300nM, IC50=300nM P04062 17666401 1502 EFARPCIPKSFGYSSVVCVCNATYCDSFDPPTPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 2v3u A 1.74 BS01 DSN A 1 Y58 A85 T87 R92 Y105 S137 A138 V139 W193 D194 Y58 A85 T87 R92 Y105 S137 A138 V139 W188 D189 ? 0015276,0016020 Kd=1mM remove_due_to_license_issue Q63226 17715062 1262 GGVVLRVVTVLEEPFVMVSENVLGKPKKYQGFSIDVLDALSNYLGFNYEIYVAPDHKYGSPQEDGTWNGLVGELVFKRADIGISALTITPDRENVVDFTTRYMDYSVGVLLRRGTSIQSLQDLSKQTDIPYGTVLDSAVYQHVRMKGLNPFERDSMYSQMWRMINRNNVLESQAGIQKVKYGNYAFVWDAAVLEYVAINDPDCSFYTVGADRGYGIALQHGSPYRDVFSQRILELQQSGDMDILKHKWWPKNG 2v54 A 2.4 BS01 TYD A 1 D13 K17 F38 L53 F68 R72 R93 S97 G98 Y101 Y144 D13 K17 F38 L53 F68 R72 R93 S97 G98 Y101 Y144 2.7.4.9 0004550,0004798,0005524,0006227,0006233,0006235,0009165,0016301,0046940 remove_due_to_license_issue P68693 18971333 1205 MSRGALIVFEGLDKSGKTTQCMNIMESIPANTIKYLNFPQRSTVTGKMIDDYLTRKKTYNDHIVNLLFCANRWEFASFIQEQLEQGITLIVDRYAFSGVAYAAAKGASMTLSKSYESGLPKPDLVIFLESGSKEINRNVGEEIYEDVTFQQKVLQEYKKMIEEGDIHWQIISSEFEEDVKKELIKNIVIEAIHTVTGPVGQLWM 2v57 A 1.9 BS01 PRL A 1 H67 S70 N71 Y106 D125 W152 H56 S59 N60 Y95 D114 W136 ? 0000976,0003677,0003700,0006355 Kd=79nM remove_due_to_license_issue Q58L87 19820093 1188 ERTRRAILDAAMLVLADHPTAALGDIAAAAGVGRSTVHRYYPERTDLLRALARHVHDLSNAAIERADPTSGPVDAALRRVVESQLDLGPIVLFVYYEPSILADPELAAYFDIGDEAIVEVLNRASYPPGWARRVFWALMQAGYEAAKDGMPRHQIVDAIMTSLTSGIITLP 2v58 A 2.1 BS01 LZJ A 1 I157 K159 E201 Y203 L204 H209 Q233 H236 L278 I437 I157 K159 E201 Y203 L204 H209 Q233 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 Kd=0.82nM remove_due_to_license_issue IC50=<1nM P24182 19164768 1448 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2v59 A 2.4 BS01 LZK A 1 K159 Y203 L204 H209 Q233 H236 L278 I437 K159 Y203 L204 H209 Q233 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 Kd=6.53nM remove_due_to_license_issue P24182 19164768 1446 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLG 2v5a A 2.31 BS01 LZL A 1 I157 K159 M169 E201 Y203 L204 Q233 H236 L278 I437 I157 K159 M169 E201 Y203 L204 Q233 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=150nM remove_due_to_license_issue P24182 19164768 1447 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2v5x A 2.25 BS02 V5X A 1 D101 H142 H143 F152 D178 H180 F208 P209 M274 Y306 D88 H129 H130 F139 D165 H167 F195 P196 M261 Y293 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 Kd=220nM remove_due_to_license_issue Q9BY41 17721440 1380 LVPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHV 2v5x A 2.25 BS03 V5X B 1 K33 P35 Y306 K20 P22 Y293 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 Kd=220nM remove_due_to_license_issue Q9BY41 17721440 1380 LVPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHV 2v6e A 3.2 BS01 dna C 0 N67 S71 R74 R212 Q216 W219 M276 I277 K300 R302 N357 A361 T362 N365 K369 V378 Y379 K380 K485 T487 N488 S489 R492 T498 R499 G520 Q521 N64 S68 R71 R209 Q213 W216 M273 I274 K297 R299 N354 A358 T359 N362 K366 V375 Y376 K377 K482 T484 N485 S486 R489 T495 R496 G517 Q518 3.1.22.- remove_due_to_license_issue Q6UAV6 17889664 1 ~ 25 VKIGELINSLVSEVEAIDASDRPQGDKTKKIKAAALKYKNALFNDKRKFRGKGLEKRISANTFNSYMSRARKRFDDRLHHNFEKNVIKLSEKYPLYSEELSSWLSMPAASIRQHMSRLQAKLKEIMPLAEDLSNIKIGTKNSEAKINKLANKYPEWQFAISDLNSEDWKDKRDYLYKLFQQGSSLLEDLNNLKVNHEVLYHLQLSSAERTSIQQRWANVLSEKKRNVVVIDYPRYMQAIYDIINKPIVSFDLTTRRGMAPLAFALAALSGRRMIEIMLQGEFSVAGKYTVTFLGQAKKRSEDKGISRKIYTLCDATLFVSLVNELRSCPAAADFDEVIKGYGENDTRSENGRINAILATAFNPWVKTFLGDDRRVYKDSRAIYARIAYEMFFRVDPRWKNVDEDVFFMEILGHDDENTQLHYKQFKLANFSRTWRPNVGEENARLAALQKLDSMMPDFARGDAGVRIHETVKQLVEQDPSIKITNSTLRPFNFSTRLIPRYLEFAADALGQFVGENGQWQLKDEAPAIVLP 2v6e A 3.2 BS02 dna D 0 G7 E8 L9 I61 S62 N64 T65 Y69 W219 K226 T257 R258 R259 K300 Y344 R350 A358 T362 K380 H424 Y425 G4 E5 L6 I58 S59 N61 T62 Y66 W216 K223 T254 R255 R256 K297 Y341 R347 A355 T359 K377 H421 Y422 3.1.22.- remove_due_to_license_issue Q6UAV6 17889664 26 ~ 44 VKIGELINSLVSEVEAIDASDRPQGDKTKKIKAAALKYKNALFNDKRKFRGKGLEKRISANTFNSYMSRARKRFDDRLHHNFEKNVIKLSEKYPLYSEELSSWLSMPAASIRQHMSRLQAKLKEIMPLAEDLSNIKIGTKNSEAKINKLANKYPEWQFAISDLNSEDWKDKRDYLYKLFQQGSSLLEDLNNLKVNHEVLYHLQLSSAERTSIQQRWANVLSEKKRNVVVIDYPRYMQAIYDIINKPIVSFDLTTRRGMAPLAFALAALSGRRMIEIMLQGEFSVAGKYTVTFLGQAKKRSEDKGISRKIYTLCDATLFVSLVNELRSCPAAADFDEVIKGYGENDTRSENGRINAILATAFNPWVKTFLGDDRRVYKDSRAIYARIAYEMFFRVDPRWKNVDEDVFFMEILGHDDENTQLHYKQFKLANFSRTWRPNVGEENARLAALQKLDSMMPDFARGDAGVRIHETVKQLVEQDPSIKITNSTLRPFNFSTRLIPRYLEFAADALGQFVGENGQWQLKDEAPAIVLP 2v6e A 3.2 BS03 dna E 0 R275 K300 K301 R302 D417 T421 R272 K297 K298 R299 D414 T418 3.1.22.- remove_due_to_license_issue Q6UAV6 17889664 1 ~ 25 VKIGELINSLVSEVEAIDASDRPQGDKTKKIKAAALKYKNALFNDKRKFRGKGLEKRISANTFNSYMSRARKRFDDRLHHNFEKNVIKLSEKYPLYSEELSSWLSMPAASIRQHMSRLQAKLKEIMPLAEDLSNIKIGTKNSEAKINKLANKYPEWQFAISDLNSEDWKDKRDYLYKLFQQGSSLLEDLNNLKVNHEVLYHLQLSSAERTSIQQRWANVLSEKKRNVVVIDYPRYMQAIYDIINKPIVSFDLTTRRGMAPLAFALAALSGRRMIEIMLQGEFSVAGKYTVTFLGQAKKRSEDKGISRKIYTLCDATLFVSLVNELRSCPAAADFDEVIKGYGENDTRSENGRINAILATAFNPWVKTFLGDDRRVYKDSRAIYARIAYEMFFRVDPRWKNVDEDVFFMEILGHDDENTQLHYKQFKLANFSRTWRPNVGEENARLAALQKLDSMMPDFARGDAGVRIHETVKQLVEQDPSIKITNSTLRPFNFSTRLIPRYLEFAADALGQFVGENGQWQLKDEAPAIVLP 2v6e B 3.2 BS01 dna C 0 R275 K300 K301 R302 D417 T421 P534 R272 K297 K298 R299 D414 T418 P531 3.1.22.- remove_due_to_license_issue Q6UAV6 17889664 1 ~ 25 VKIGELINSLVSEVEAIDASDRPQGDKTKKIKAAALKYKNALFNDKRKFRGKGLEKRISANTFNSYMSRARKRFDDRLHHNFEKNVIKLSEKYPLYSEELSSWLSMPAASIRQHMSRLQAKLKEIMPLAEDLSNIKIGTKNSEAKINKLANKYPEWQFAISDLNSEDWKDKRDYLYKLFQQGSSLLEDLNNLKVNHEVLYHLQLSSAERTSIQQRWANVLSEKKRNVVVIDYPRYMQAIYDIINKPIVSFDLTTRRGMAPLAFALAALSGRRMIEIMLQGEFSVAGKYTVTFLGQAKKRSEDKGISRKIYTLCDATLFVSLVNELRSCPAAADFDEVIKGYGENDTRSENGRINAILATAFNPWVKTFLGDDRRVYKDSRAIYARIAYEMFFRVDPRWKNVDEDVFFMEILGHDDENTQLHYKQFKLANFSRTWRPNVGEENARLAALQKLDSMMPDFARGDAGVRIHETVKQLVEQDPSIKITNSTLRPFNFSTRLIPRYLEFAADALGQFVGENGQWQLKDEAPAIVLP 2v6e B 3.2 BS02 dna E 0 N67 S71 R74 R212 Q216 W219 M276 I277 K300 R302 N357 A361 T362 N365 K369 V378 Y379 K380 K485 T487 N488 S489 R492 T498 R499 G520 Q521 N64 S68 R71 R209 Q213 W216 M273 I274 K297 R299 N354 A358 T359 N362 K366 V375 Y376 K377 K482 T484 N485 S486 R489 T495 R496 G517 Q518 3.1.22.- remove_due_to_license_issue Q6UAV6 17889664 1 ~ 25 VKIGELINSLVSEVEAIDASDRPQGDKTKKIKAAALKYKNALFNDKRKFRGKGLEKRISANTFNSYMSRARKRFDDRLHHNFEKNVIKLSEKYPLYSEELSSWLSMPAASIRQHMSRLQAKLKEIMPLAEDLSNIKIGTKNSEAKINKLANKYPEWQFAISDLNSEDWKDKRDYLYKLFQQGSSLLEDLNNLKVNHEVLYHLQLSSAERTSIQQRWANVLSEKKRNVVVIDYPRYMQAIYDIINKPIVSFDLTTRRGMAPLAFALAALSGRRMIEIMLQGEFSVAGKYTVTFLGQAKKRSEDKGISRKIYTLCDATLFVSLVNELRSCPAAADFDEVIKGYGENDTRSENGRINAILATAFNPWVKTFLGDDRRVYKDSRAIYARIAYEMFFRVDPRWKNVDEDVFFMEILGHDDENTQLHYKQFKLANFSRTWRPNVGEENARLAALQKLDSMMPDFARGDAGVRIHETVKQLVEQDPSIKITNSTLRPFNFSTRLIPRYLEFAADALGQFVGENGQWQLKDEAPAIVLP 2v6e B 3.2 BS03 dna F 0 G7 E8 L9 I61 S62 N64 T65 Y69 W219 K226 T257 R258 R259 K300 Y344 R350 A358 T362 K380 H424 Y425 G4 E5 L6 I58 S59 N61 T62 Y66 W216 K223 T254 R255 R256 K297 Y341 R347 A355 T359 K377 H421 Y422 3.1.22.- remove_due_to_license_issue Q6UAV6 17889664 26 ~ 44 VKIGELINSLVSEVEAIDASDRPQGDKTKKIKAAALKYKNALFNDKRKFRGKGLEKRISANTFNSYMSRARKRFDDRLHHNFEKNVIKLSEKYPLYSEELSSWLSMPAASIRQHMSRLQAKLKEIMPLAEDLSNIKIGTKNSEAKINKLANKYPEWQFAISDLNSEDWKDKRDYLYKLFQQGSSLLEDLNNLKVNHEVLYHLQLSSAERTSIQQRWANVLSEKKRNVVVIDYPRYMQAIYDIINKPIVSFDLTTRRGMAPLAFALAALSGRRMIEIMLQGEFSVAGKYTVTFLGQAKKRSEDKGISRKIYTLCDATLFVSLVNELRSCPAAADFDEVIKGYGENDTRSENGRINAILATAFNPWVKTFLGDDRRVYKDSRAIYARIAYEMFFRVDPRWKNVDEDVFFMEILGHDDENTQLHYKQFKLANFSRTWRPNVGEENARLAALQKLDSMMPDFARGDAGVRIHETVKQLVEQDPSIKITNSTLRPFNFSTRLIPRYLEFAADALGQFVGENGQWQLKDEAPAIVLP 2v6n A 1.98 BS01 XP1 A 1 P39 H41 M49 C145 H164 M165 D187 R188 P39 H41 M49 C145 H164 M165 D187 R188 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=1380nM P0C6X7 18559270 2307 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 2v77 A 1.603 BS01 PAY A 1 H69 E72 R127 N144 R145 H196 Y198 M203 I247 Y248 T268 E270 F279 H69 E72 R127 N144 R145 H196 Y198 M203 I247 Y248 T268 E270 F279 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=8.7uM remove_due_to_license_issue P15085 18566513 400 ARSTDTFNYATYHTLEEIYDFLDLLVAENPHLVSKIQIGNTYEGRPIYVLKFSTGGSKRPAIWIDTGIHSREWVTQASGVWFAKKITQDYGQDAAFTAILDTLDIFLEIVTNPDGFAFTHSTNRMWRKTRSHTAGSLCIGVDPNRNWDAGFGLSGASSNPCSETYHGKFANSEVEVKSIVDFVKDHGNIKAFISIHSYSQLLMYPYGYKTEPVPDQDELDQLSKAAVTALASLYGTKFNYGSIIKAIYQASGSTIDWTYSQGIKYSFTFELRDTGRYGFLLPASQIIPTAKETWLALLTIMEHTLNHP 2v7a A 2.5 BS01 627 A 1 L248 A269 K271 E316 F317 M318 T319 G321 N368 L370 L16 A37 K39 E84 F85 M86 T87 G89 N136 L138 D363 A365 R367 N368 D381 P402 D131 A133 R135 N136 D149 P170 2.7.10.2 0004672,0004713,0005524,0006468 Kd=0.005uM remove_due_to_license_issue P00519 17804707 1504 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSI 2v95 A 1.93 BS01 HCY A 1 P14 R252 D256 F357 K359 W362 P8 R242 D246 F325 K327 W330 ? 0004867,0005496,0005576,0005615,0008150,0008211 remove_due_to_license_issue P31211 17644521 1375 NSHRGLAPTNVDFAFNLYQRLVALNPDKNTLISPVSISMALAMVSLGSTQSLQSLGFNLTETSEAEIHQSFQYLNYLLKQSDTGLEMNMGNAMFLLQKLKLKDSFLADVKQYYESEALAIDFEDWTKASQQINQHVKDKTQGKIEHVFSDSPASFILVNYIFLRGIWELPFSPENTREEDFYVNETSTVKVPMMVQSGSIGYFRDSVFPCQLIQMDYVGNGTAFFILPDQGQMDTVIAALSRDTIDRWGKLMTPRQVNLYIPKFSMSDTYDLKDVLEDLNIKDLLTNLTLTMVHKAMLQLDEGNVLLRSEPLDIKFNKPFILLLFDKFTWSSLMMSQVVNPA 2v96 A 2.4 BS01 CFQ A 1 Y70 Y121 W279 I287 F288 F290 F331 Y334 G335 Y67 Y118 W276 I284 F285 F287 F328 Y331 G332 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=29uM remove_due_to_license_issue P04058 18007027 1536 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 2v96 A 2.4 BS02 CFQ A 2 W84 G117 E199 S200 F330 F331 Y334 H440 W81 G114 E196 S197 F327 F328 Y331 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=29uM remove_due_to_license_issue P04058 18007027 1537 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 2va5 A 2.75 BS01 C8C A 1 L30 D32 I118 D228 G230 L32 D34 I120 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=130000nM P56817 17985862 1389 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2va6 A 2.5 BS01 H24 A 1 S10 G11 G13 D32 Y71 F108 D228 S229 G230 S12 G13 G15 D34 Y73 F110 D219 S220 G221 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.67uM remove_due_to_license_issue IC50=91000nM P56817 17985862 1504 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2va7 A 2.2 BS01 C27 A 1 S10 G11 G13 D32 Y71 F108 W115 D228 S229 G230 T232 S12 G13 G15 D34 Y73 F110 W117 D217 S218 G219 T221 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=0.2uM remove_due_to_license_issue IC50=200nM P56817 17985862 1505 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vaq A 3.01 BS01 VAW A 1 W149 Y151 V208 F226 M276 H277 H307 E309 L323 F324 W121 Y123 V180 F198 M248 H249 H279 E281 L295 F296 E309 E281 4.3.3.2 0005773,0009058,0009820,0012505,0016787,0016844 remove_due_to_license_issue P68175 18081287 1334 PILKEILIEAPSYAPNSFTFDSTNKGFYTSVQDGRVIKYEGPNSGFVDFAYASPYWNKAFCENSTDAEKRPLCGRTYDISYNLQNNQLYIVDCYYHLSVVGSEGGHATQLATSVDGVPFKWLYAVTVDQRTGIVYFTDVSTLYDDRGVQQIMDTSDKTGRLIKYDPSTKETTLLLKELHVPGGAEVSADSSFVLVAEFLSHQIVKYWLEGPKKGTAEVLVKIPNPGNIKRNADGHFWVSSSEELDGNMHGRVDPKGIKFDEFGNILEVIPLPPPFAGEHFEQIQEHDGLLYIGTLFHGSVGILVY 2vb8 A 1.52 BS01 TLM A 1 C163 F229 M269 V270 A271 P272 H298 T300 H333 F390 G391 F392 G394 C162 F228 M268 V269 A270 P271 H297 T299 H332 F389 G390 F391 G393 C163 H298 E309 K328 H333 F390 F392 C162 H297 E308 K327 H332 F389 F391 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 remove_due_to_license_issue IC50=12000nM P0A953 18084068 1405 KRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2vb8 B 1.52 BS01 TLM B 1 C163 F229 A271 P272 H298 T300 F390 G391 F392 G394 C162 F228 A270 P271 H297 T299 F389 G390 F391 G393 C163 H298 E309 K328 H333 F390 F392 C162 H297 E308 K327 H332 F389 F391 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 remove_due_to_license_issue IC50=12000nM P0A953 18084068 1405 KRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2vba A 1.36 BS01 P4T A 1 A162 C163 F201 M204 F229 L335 F392 A162 C163 F201 M204 F229 L335 F392 C163 H298 E309 K328 H333 F390 F392 C163 H298 E309 K328 H333 F390 F392 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 Kd=25uM remove_due_to_license_issue P0A953 18084068 1405 MKRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2vba B 1.36 BS01 P4T A 1 V134 M138 V134 M138 C163 H298 E309 K328 H333 F390 F392 C163 H298 E309 K328 H333 F390 F392 2.3.1.41 0004315,0005737,0005829,0006633,0016746,0016747,0044281,1903966 remove_due_to_license_issue P0A953 18084068 1405 MKRAVITGLGIVSSIGNNQQEVLASLREGRSGITFSQELKDSGMRSHVWGNVKLDTTGLIDRKVVRFMSDASIYAFLSMEQAIADAGLSPEAYQNNPRVGLIAGSGGGSPRFQVFGADAMRGPRGLKAVGPYVVTKAMASGVSACLATPFKIHGVNYSISSACATSAHCIGNAVEQIQLGKQDIVFAGGGEELCWEMACEFDAMGALSTKYNDTPEKASRTYDAHRDGFVIAGGGGMVVVEELEHALARGAHIYAEIVGYGATSDGADMVAPSGEGAVRCMKMAMHGVDTPIDYLNSHGTSTPVGDVKELAAIREVFGDKSPAISATKAMTGHSLGAAGVQEAIYSLLMLEHGFIAPSINIEELDEQAAGLNIVTETTDRELTTVMSNSFGFGGTNATLVMRKL 2vc7 A 2.05 BS03 HT5 A 1 H24 Y97 H170 R223 L226 F229 C258 I261 W263 H24 Y97 H170 R223 L226 F229 C258 I261 W263 H22 H24 K137 H170 H199 D202 R223 D256 H22 H24 K137 H170 H199 D202 R223 D256 3.1.8.1 0004063,0008270,0009056,0016787,0016788,0046872 Ki=432.7uM remove_due_to_license_issue Q97VT7 18486146 1335 MRIPLVGKDSIESKDIGFTLIHEHLRVFSEAVRQQWPHLYNEDEEFRNAVNEVKRAMQFGVKTIVDPTVMGLGRDIRFMEKVVKATGINLVAGTGIYIYIDLPFYFLNRSIDEIADLFIHDIKEGIQGTLNKAGFVKIAADEPGITKDVEKVIRAAAIANKETKVPIITHSNAHNNTGLEQQRILTEEGVDPGKILIGHLGDTDNIDYIKKIADKGSFIGLDRYGLDLFLPVDKRNETTLRLIKDGYSDKIMISHDYCCTIDWGTAKPEYKPKLAPRWSITLIFEDTIPFLKRNGVNEEVIATIFKENPKKFFS 2vc7 B 2.05 BS03 HT5 B 1 H24 Y97 H170 L226 F229 C258 I261 W263 T265 K271 H24 Y97 H170 L226 F229 C258 I261 W263 T265 K271 H22 H24 K137 H170 H199 D202 R223 D256 H22 H24 K137 H170 H199 D202 R223 D256 3.1.8.1 0004063,0008270,0009056,0016787,0016788,0046872 Ki=432.7uM remove_due_to_license_issue Q97VT7 18486146 1328 MRIPLVGKDSIESKDIGFTLIHEHLRVFSEAVRQQWPHLYNEDEEFRNAVNEVKRAMQFGVKTIVDPTVMGLGRDIRFMEKVVKATGINLVAGTGIYIYIDLPFYFLNRSIDEIADLFIHDIKEGIQGTLNKAGFVKIAADEPGITKDVEKVIRAAAIANKETKVPIITHSNAHNNTGLEQQRILTEEGVDPGKILIGHLGDTDNIDYIKKIADKGSFIGLDRYGLDLFLPVDKRNETTLRLIKDGYSDKIMISHDYCCTIDWGTAKPEYKPKLAPRWSITLIFEDTIPFLKRNGVNEEVIATIFKENPKKFFS 2vc9 A 2.36 BS01 NOK A 1 C301 Y305 W366 H482 E483 W517 E601 Y825 D908 C276 Y280 W341 H457 E458 W492 E576 Y800 D883 3.2.1.50 Kd=3.6nM remove_due_to_license_issue A0A0H2YU91 18443291 1909 GVEITEGVTVTAKGNTEGNTADLAIDGDLSTYWESSNDYKWIEVDLGGIYELSKIEIFNKDEAVYKYNIYASEDGENFNKIAYKNNDNVSDSNGNMHTIDNVRAGKIRIDVVQNSNSDRVNIAEINVFGKNTGESLPEVKKIATSNFSETPWATEYEKFNSDSAYANEKTLNEIKNLVGRVIGREFKDKFIFEIRDQLNGNDVFEVSDSGDGKVLIKGNNGVSLASGFNYYLKNYCNVSYNPIMGSNLKMPETMPSVGERVVIDTPYEHRYALNFCTYSYTMSFWDWDQYEEFLDWCAMNGVNLVLDIIGQEEVLRRTLNEFGYSDEEVKEFISGPAYFAWFYMQNMTGFGGPLPNDWFEQRAELGRKMHDRMQSFGINPVLQGYSGMVPRDFKEKNQEAQTISQGGWCGFDRPDMLKTYVNEGEADYFQKVADVFYEKQKEVFGDVTNFYGVDPFHEGGNTGDLDNGKIYEIIQNKMIEHDNDAVWVIQNWQGNPSNNKLEGLTKKDQAMVLDLFSEVSPDWNRLEERDLPWIWNMLHNFGGRMGMDAAPEKLATEIPKALANSEHMVGIGITPEAINTNPLAYELLFDMAWTRDQINFRTWTEDYIERRYGKTNKEILEAWNIILDTAYKKRNDYYQGAAESIINARPGFGIKSASTWGHSKIVYDKSEFEKAIEIFAKNYDEFKDSDAFLYDFADILKQLLANSAQEYYEVMCNAYNNGNGEKFKFVSGKFLELIKLQERVLSTRPEFLIGNWIEDARTMLKDSDDWTKDLFEFNARALVTTWGSRNNADGGGLKDYSNRQWSGLTEDYYYARWEKWINGLQAELDGGAKAPNIDWFKMEYDWVNKKSDTDKLYPTEASNENLGELAKIAMESYSVTNMD 2vcb A 2.2 BS01 OAN A 1 C301 Y305 W366 M369 H482 E483 W517 F566 E601 Q664 W685 Y825 K909 C275 Y279 W340 M343 H456 E457 W491 F540 E575 Q638 W659 Y799 K882 3.2.1.50 remove_due_to_license_issue A0A0H2YU91 18443291 1911 GVEITEGVTVTAKGNTEGNTADLAIDGDLSTYWESSNDYKWIEVDLGGIYELSKIEIFNKDEAVYKYNIYASEDGENFNKIAYKNNDNVSDSNGNMHTIDNVRAGKIRIDVVQNSNSDRVNIAEINVFGKNTGESLPEKKIATSNFSETPWATEYEKFNSDSAYANEKTLNEIKNLVGRVIGREFKDKFIFEIRDQLNGNDVFEVSDSGDGKVLIKGNNGVSLASGFNYYLKNYCNVSYNPIMGSNLKMPETMPSVGERVVIDTPYEHRYALNFCTYSYTMSFWDWDQYEEFLDWCAMNGVNLVLDIIGQEEVLRRTLNEFGYSDEEVKEFISGPAYFAWFYMQNMTGFGGPLPNDWFEQRAELGRKMHDRMQSFGINPVLQGYSGMVPRDFKEKNQEAQTISQGGWCGFDRPDMLKTYVNEGEADYFQKVADVFYEKQKEVFGDVTNFYGVDPFHEGGNTGDLDNGKIYEIIQNKMIEHDNDAVWVIQNWQGNPSNNKLEGLTKKDQAMVLDLFSEVSPDWNRLEERDLPWIWNMLHNFGGRMGMDAAPEKLATEIPKALANSEHMVGIGITPEAINTNPLAYELLFDMAWTRDQINFRTWTEDYIERRYGKTNKEILEAWNIILDTAYKKRNDYYQGAAESIINARPGFGIKSASTWGHSKIVYDKSEFEKAIEIFAKNYDEFKDSDAFLYDFADILKQLLANSAQEYYEVMCNAYNNGNGEKFKFVSGKFLELIKLQERVLSTRPEFLIGNWIEDARTMLKDSDDWTKDLFEFNARALVTTWGSRNNADGGGLKDYSNRQWSGLTEDYYYARWEKWINGLQAELDGAKAPNIDWFKMEYDWVNKKSDTDKLYPTEASNENLGELAKIAMESYSVTNMDK 2vcg A 1.9 BS02 S17 A 1 L27 I106 H148 H149 F158 D186 H188 F214 Y318 L21 I100 H142 H143 F152 D180 H182 F208 Y312 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 18054239 1378 HAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADI 2vcg A 1.9 BS03 S17 D 1 Y344 E346 F347 Y338 E340 F341 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 18054239 1381 HAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADI 2vcg D 1.9 BS01 S17 A 1 E346 F347 E346 F347 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 18054239 1378 MHHHHHHAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 2vcg D 1.9 BS04 S17 D 1 L27 I106 H148 H149 F158 D186 H188 F214 Y318 L27 I106 H148 H149 F158 D186 H188 F214 Y318 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 18054239 1381 MHHHHHHAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 2vci A 2.0 BS01 2GJ A 1 N51 A55 K58 D93 I96 G97 M98 L107 T109 F138 T184 E223 N36 A40 K43 D78 I81 G82 M83 L92 T94 F123 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.021uM remove_due_to_license_issue IC50=61nM, EC50=7nM, Ki=9nM P07900 18020435 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2vcj A 2.5 BS01 2EQ A 1 N51 A55 D93 I96 G97 M98 D102 L107 T184 E223 N36 A40 D78 I81 G82 M83 D87 L92 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.021uM remove_due_to_license_issue IC50=<10000nM P07900 18020435 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2vcq B 1.95 BS02 D25 B 1 M11 G13 R14 M99 W104 M10 G12 R13 M98 W103 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50=0.92uM remove_due_to_license_issue IC50=920nM O60760 18341273 1201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2vcw B 1.95 BS02 ZZA B 1 G13 R14 M99 W104 G12 R13 M98 W103 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50=890uM remove_due_to_license_issue Kd=140000nM, IC50=890000nM O60760 18341273 1201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2vcx B 2.1 BS02 D26 B 1 M11 G13 R14 M99 W104 Y152 M10 G12 R13 M98 W103 Y151 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50=0.021uM remove_due_to_license_issue Kd=51nM, IC50=21nM, EC50=110nM O60760 18341273 1201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2vd0 B 2.2 BS01 D27 B 1 M11 G13 R14 M99 W104 A105 Y152 L199 M10 G12 R13 M98 W103 A104 Y151 L198 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50=11.6uM remove_due_to_license_issue IC50=11600nM O60760 18341273 1200 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2vd1 B 2.25 BS01 D28 B 1 M11 G13 R14 Q36 M99 W104 Y152 L199 M10 G12 R13 Q35 M98 W103 Y151 L198 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50=0.138uM remove_due_to_license_issue IC50=94600nM O60760 18341273 1200 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2vd4 A 1.9 BS01 P21 A 1 Y139 M221 V223 E224 Q231 L235 Y136 M218 V220 E221 Q228 L232 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=18uM remove_due_to_license_issue P43889 18218712 1454 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 2vd7 A 2.25 BS02 PD2 A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 H276 Y127 Y172 F180 H183 E185 K201 W203 K236 H271 G170 Y177 H188 E190 H276 S288 G165 Y172 H183 E185 H271 S283 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=4200nM O75164 18942826 1356 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 2ves A 1.9 BS02 GVR A 1 L18 M62 E77 H78 T190 F191 G192 I197 G209 A214 H237 D241 H264 L18 M62 E77 H78 T190 F191 G192 I197 G209 A214 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue P47205 18287278 1296 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPI 2ves C 1.9 BS03 GVR C 1 L18 M62 E77 H78 T190 F191 G192 I197 G209 N213 A214 H237 D241 H264 L18 M62 E77 H78 T190 F191 G192 I197 G209 N213 A214 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue P47205 18287278 1301 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 2veu A 2.4 BS01 IZ1 A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 D298 Y44 R45 D46 D179 F180 C213 S214 A215 I217 G218 R219 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=100nM remove_due_to_license_issue P18031 18037290 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2vev A 1.8 BS01 IZ2 A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 L299 Y45 R46 D47 D180 F181 C214 S215 A216 I218 G219 R220 Q261 L298 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=300nM remove_due_to_license_issue P18031 18037290 1300 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 2vew A 2.0 BS01 IZ3 A 1 Y46 D48 V49 D181 F182 C215 S216 A217 I219 G220 R221 D298 Y44 D46 V47 D179 F180 C213 S214 A215 I217 G218 R219 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=64nM remove_due_to_license_issue P18031 18037290 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2vex A 2.2 BS01 IZ4 A 1 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 L299 Y44 D46 D179 F180 C213 S214 A215 I217 G218 R219 L297 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=130nM remove_due_to_license_issue P18031 18037290 1300 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 2vey A 2.2 BS01 IZ5 A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 M258 G259 Q262 L299 Y44 R45 D46 D179 F180 C213 S214 A215 I217 G218 R219 M256 G257 Q260 L297 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=43nM remove_due_to_license_issue P18031 18037290 1300 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 2vf6 A 2.1 BS01 M0N A 1 F99 L100 D103 R112 T167 Q171 K200 T201 Y204 D243 K257 F86 L87 D90 R99 T154 Q158 K187 T188 Y191 D230 K244 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F85 D90 D94 R99 D161 K187 F226 D230 D231 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=3nM P14324 1351 VYAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 2vfk A 1.5 BS01 AMP A 1 T134 F179 R219 H224 T226 T47 F92 R132 H137 T139 Kd=194uM remove_due_to_license_issue 18082768 1293 YQPNYFLSIPITNKKITAGIKVLQNSILRQDNRLTKAMVGDGSFHITLLVMQLLNEDEVNIGTDALLELKPFVEEILEGKHLTLPFHGIGTFQGQVGFVKLADGDHVSALLEIAETAKRTFQEKGILAGESRTFKPHLTFMKLSKAPMLWKKGVRKIEPGLYEQFIDHRFGEEILYQIDLCSMLKKKQSNGYYHCESSIVIGEKD 2vfz A 2.4 BS01 UPF A 1 F134 V136 Y139 I198 S199 R202 D225 V226 D227 H280 A281 A282 D316 E317 K359 F53 V55 Y58 I117 S118 R121 D144 V145 D146 H199 A200 A201 D235 E236 K278 W314 W233 2.4.1.87 0005975,0016020,0016758 Ki=245uM remove_due_to_license_issue P14769 17493636 1360 KLKLSDWFNPFKRPEVVTMTKWKAPVVWEGTYNRAVLDNYYAKQKITVGLTVFAVGRYIEHYLEEFLTSANKHFMVGHPVIFYIMVDDVSRMPLIELGPLRSFKVFKIKPEKRWQDISMMRMKTIGEHIVAHIQHEVDFLFCMDVDQVFQDKFGVETLGESVAQLQAWWYKADPNDFTYERRKESAAYIPFGEGDFYYHAAIFGGTPTQVLNITQECFKGILKDKKNDIEAQWHDESHLNKYFLLNKPTKILSPEYCWDYHIGLPADIKLVKMSWQTK 2vgc C 1.8 BS02 V35 C 1 S195 S214 W215 G216 S217 S45 S64 W65 G66 S67 M192 G193 D194 S195 G196 M42 G43 D44 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 9425066 358 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 2vgo A 1.7 BS01 AD5 A 1 G100 V107 A120 L154 L170 E171 F172 A173 G176 E177 L223 G14 V21 A34 L68 L84 E85 F86 A87 G90 E91 L137 D216 K218 E220 N221 D234 T252 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 ic50=500nM remove_due_to_license_issue Q6DE08 18483302 1357 KFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY 2vgp A 1.7 BS01 AD6 A 1 L99 F172 A173 G176 L223 L12 F82 A83 G86 L133 D216 K218 E220 N221 D234 T252 D126 K128 E130 N131 D144 T162 2.7.11.1 0004672,0005524,0006468 ic50=577nM remove_due_to_license_issue Q6DE08 18307303 1357 FTIDDFDIGRPLGKGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQ 2vh0 A 1.7 BS03 GSI A 1 K96 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G226 I227 Y228 K82 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki<1nM remove_due_to_license_issue P00742 18053714 1247 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2vh6 A 1.95 BS01 GSV A 1 E97 T98 Y99 F174 D189 A190 C191 Q192 V213 W215 G216 G219 G226 I227 Y228 E81 T82 Y83 F160 D177 A178 C179 Q180 V201 W203 G204 G206 G214 I215 Y216 H57 D102 Q192 G193 D194 S195 G196 H42 D86 Q180 G181 D182 S183 G184 3.4.21.6 0004252,0006508 Ki=0.2nM remove_due_to_license_issue P00742 18054228 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2vhj A 1.8 BS01 ADP A 1 N133 S134 G135 K136 T137 P138 N234 S292 N133 S134 G135 K136 T137 P138 N223 S281 ? 0005524,0019072,0046872 remove_due_to_license_issue Q94M05 18057007 1301 MIHLYDAKSFAKLRAAQYAAFHTDAPGSWFDHTSGVLESVEDGTPVLAIGVESGDAIVFDKNAQRIVAYKEKSVKAEDGSVSVVQVENGFMKQGHRGWLVDLTGELVGCSPVVAEFGGHRYASGMVIVTGKGNSGKTPLVHALGEALGGKDKYATVRFGEPLSGYNTDFNVFVDDIARAMLQHRVIVIDSLKNVIISRGAFDLLSDIGAMAASRGCVVIASLNPTSNDDKIVELVKEASRANSTSLVISTDVDGEWQVLTRTGEGLQRLTHTLQTSYGEHSVLTIHTS 2vhj A 1.8 BS02 ADP B 1 G276 L277 Q278 R279 G265 L266 Q267 R268 ? 0005524,0019072,0046872 remove_due_to_license_issue Q94M05 18057007 1301 MIHLYDAKSFAKLRAAQYAAFHTDAPGSWFDHTSGVLESVEDGTPVLAIGVESGDAIVFDKNAQRIVAYKEKSVKAEDGSVSVVQVENGFMKQGHRGWLVDLTGELVGCSPVVAEFGGHRYASGMVIVTGKGNSGKTPLVHALGEALGGKDKYATVRFGEPLSGYNTDFNVFVDDIARAMLQHRVIVIDSLKNVIISRGAFDLLSDIGAMAASRGCVVIASLNPTSNDDKIVELVKEASRANSTSLVISTDVDGEWQVLTRTGEGLQRLTHTLQTSYGEHSVLTIHTS 2vhq A 2.15 BS01 ATP A 1 G135 K136 T137 P138 N234 Y288 S292 G135 K136 T137 P138 N223 Y277 S281 ? 0005524,0019072,0046872 remove_due_to_license_issue Q94M05 18057007 1327 MIHLYDAKSFAKLRAAQYAAFHTDAPGSWFDHTSGVLESVEDGTPVLAIGVESGDAIVFDKNAQRIVAYKEKSVKAEDGSVSVVQVENGFMKQGHRGWLVDLTGELVGCSPVVAEFGGHRYASGMVIVTGKGNSGKTPLVHALGEALGGKDKYATVRFGEPLSGYNTDFNVFVDDIARAMLQHRVIVIDSLKNVIISRGAFDLLSDIGAMAASRGCVVIASLNPTSNDDKIVELVKEASRANSTSLVISTDVDGEWQVLTRTGEGLQRLTHTLQTSYGEHSVLTIHTSQTVIKNDELESVLR 2vhq A 2.15 BS02 ATP B 1 G276 L277 Q278 R279 G265 L266 Q267 R268 ? 0005524,0019072,0046872 remove_due_to_license_issue Q94M05 18057007 1327 MIHLYDAKSFAKLRAAQYAAFHTDAPGSWFDHTSGVLESVEDGTPVLAIGVESGDAIVFDKNAQRIVAYKEKSVKAEDGSVSVVQVENGFMKQGHRGWLVDLTGELVGCSPVVAEFGGHRYASGMVIVTGKGNSGKTPLVHALGEALGGKDKYATVRFGEPLSGYNTDFNVFVDDIARAMLQHRVIVIDSLKNVIISRGAFDLLSDIGAMAASRGCVVIASLNPTSNDDKIVELVKEASRANSTSLVISTDVDGEWQVLTRTGEGLQRLTHTLQTSYGEHSVLTIHTSQTVIKNDELESVLR 2vi5 A 2.3 BS01 Y19 A 1 W27 G58 A59 I60 E61 V81 V82 I83 W17 G48 A49 I50 E51 V71 V72 I73 H89 H79 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ki=110uM remove_due_to_license_issue P9WHE9 18331058 201 PSLDASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2vi5 A 2.3 BS02 Y19 E 1 A113 N114 A103 N104 H89 H79 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ki=110uM remove_due_to_license_issue P9WHE9 18331058 201 PSLDASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2vi5 B 2.3 BS01 Y19 A 1 A113 N114 A142 A100 N101 A129 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ki=110uM remove_due_to_license_issue P9WHE9 18331058 201 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2vi5 B 2.3 BS02 Y19 B 1 W27 G58 A59 I60 E61 V81 V82 I83 W14 G45 A46 I47 E48 V68 V69 I70 H89 H76 2.5.1.78 0000906,0005737,0005829,0009231,0009349,0016740 Ki=110uM remove_due_to_license_issue P9WHE9 18331058 201 DASGVRLAIVASSWHGKICDALLDGARKVAAGCGLDDPTVVRVLGAIEIPVVAQELARNHDAVVALGVVIRGQTPHFDYVCDAVTQGLTRVSLDSSTPIANGVLTTNTEEQALDRAGLPTSAEDKGAQATVAALATALTLRELRAHS 2vie A 1.9 BS01 VG0 A 1 G74 L91 D93 G95 Y132 T133 Q134 F169 W176 Y259 D289 G291 T292 T293 N294 N446 G13 L30 D32 G34 Y71 T72 Q73 F108 W115 Y186 D216 G218 T219 T220 N221 N373 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D216 T219 3.4.23.46 0004190,0006508,0016020 ic50=33nM remove_due_to_license_issue IC50=210nM P56817 18166458 1448 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vin A 1.9 BS01 505 A 1 D189 S190 C191 Q192 S195 W215 G216 G219 D192 S193 C194 Q195 S198 W218 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50>1mM remove_due_to_license_issue IC50=>1000000nM P00749 18163548 1247 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2vio A 1.8 BS01 L1O A 1 H57 D189 S190 C191 Q192 W215 G216 G219 C220 H46 D192 S193 C194 Q195 W218 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=40uM remove_due_to_license_issue IC50=40000nM P00749 18163548 1246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2vip A 1.72 BS01 L1R A 1 H57 C58 D189 S190 C191 Q192 S195 S214 W215 G216 G219 C220 H46 C47 D192 S193 C194 Q195 S198 S217 W218 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=5.2uM remove_due_to_license_issue IC50=5200nM P00749 18163548 1247 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2viq A 2.0 BS01 D55 A 1 H57 H99 D189 S190 C191 Q192 S195 G216 G219 H46 H94 D192 S193 C194 Q195 S198 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=1.3uM remove_due_to_license_issue IC50=1300nM P00749 18163548 1246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2viv A 1.72 BS01 VG2 A 1 H57 H99 D189 S190 C191 Q192 S195 G216 G219 C220 H46 H94 D192 S193 C194 Q195 S198 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=520nM remove_due_to_license_issue IC50=520nM P00749 18163548 1247 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2viw A 2.05 BS01 D56 A 1 H57 H99 D189 S190 Q192 S195 W215 G216 G219 H46 H94 D192 S193 Q195 S198 W218 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=72nM remove_due_to_license_issue IC50=72nM P00749 18163548 1246 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 2viy A 1.82 BS01 VG3 A 1 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 R189 D289 G291 T292 T293 N294 R296 N446 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 R128 D215 G217 T218 T219 N220 R222 N372 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D215 T218 3.4.23.46 0004190,0006508,0016020 ic50=1.8uM remove_due_to_license_issue P56817 18171614 1448 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2viz A 1.6 BS01 VG4 A 1 G74 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 D289 G291 T292 T293 N294 N446 G13 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 D213 G215 T216 T217 N218 N370 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D213 T216 3.4.23.46 0004190,0006508,0016020 ic50=605nM remove_due_to_license_issue P56817 18171614 1448 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vj1 B 2.25 BS01 XP1 B 1 N142 G143 C145 E166 N141 G142 C144 E165 H41 G143 C145 H40 G142 C144 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=1380nM P0C6X7 18559270 1304 GFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCS 2vj6 A 1.8 BS01 VG5 A 1 G72 G74 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 D289 G291 T292 T293 N294 R296 N446 G11 G13 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 D213 G215 T216 T217 N218 R220 N370 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D213 T216 3.4.23.46 0004190,0006508,0016020 ic50=13nM remove_due_to_license_issue IC50=310nM P56817 18166458 1447 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vj7 A 1.6 BS01 VG6 A 1 G74 D93 G95 S96 Y132 T133 Q134 F169 W176 I179 Y259 D289 G291 T292 T293 N294 N446 G13 D32 G34 S35 Y71 T72 Q73 F108 W115 I118 Y183 D213 G215 T216 T217 N218 N370 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D213 T216 3.4.23.46 0004190,0006508,0016020 ic50=40nM remove_due_to_license_issue IC50=200nM P56817 18166458 1448 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vj8 A 1.8 BS02 HA2 A 1 Q134 Q136 A137 Y267 G268 G269 E271 H295 E296 F314 E318 P374 Y378 Y383 R563 K565 Q134 Q136 A137 Y267 G268 G269 E271 H295 E296 F314 E318 P374 Y378 Y383 R563 K565 E271 H295 E296 H299 E318 D375 Y383 E271 H295 E296 H299 E318 D375 Y383 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 Ki=0.002uM remove_due_to_license_issue P09960 12207002 1616 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 2vj9 A 1.6 BS01 VG7 A 1 G74 L91 D93 G95 Y132 T133 Q134 F169 W176 Y259 D289 G291 T292 T293 N294 T450 G13 L30 D32 G34 Y71 T72 Q73 F108 W115 Y183 D213 G215 T216 T217 N218 T374 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D213 T216 3.4.23.46 0004190,0006508,0016020 ic50=180nM remove_due_to_license_issue IC50=180nM P56817 18166458 1452 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQT 2vjx A 1.85 BS01 IFL A 1 W198 D199 W200 W395 N461 W533 Y537 E555 W645 W656 W171 D172 W173 W367 N433 W505 Y509 E527 W617 W628 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=11uM remove_due_to_license_issue Ki=1.1e+4nM Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKKGEELPVNIKHIRETYK 2vk2 A 1.2 BS01 GZL A 1 E13 S14 R17 D90 R91 R146 F170 N199 D227 L247 E12 S13 R16 D89 R90 R145 F169 N198 D226 L246 ? 0005534,0015757,0030246,0030288,0042597,0055052,0055085,0140271 Kd=0.13uM remove_due_to_license_issue P39325 19744923 1298 PLTVGFSQVGSESGWRAAETNVAKSEAEKRGITLKIADGQQKQENQIKAVRSFVAQGVDAIFIAPVVATGWEPVLKEAKDAEIPVFLLDRSIDVKDKSLYMTTVTADNILEGKLIGDWLVKEVNGKPCNVVELQGTVGASVAIDRKKGFAEAIKNAPNIKIIRSQSGDFTRSKGKEVMESFIKAENNGKNICMVYAHNDDMVIGAIQAIKEAGLKPGKDILTGSIDGVPDIYKAMMDGEANASVELTPNMAGPAFDALEKYKKDGTMPEKLTLTKSTLYLPDTAKEELEKKKNMGY 2vk6 A 1.5 BS02 DAN A 1 R1266 I1267 I1327 D1328 F1353 Y1485 Q1493 R1555 R1615 Y1655 R24 I25 I85 D86 F111 Y243 Q251 R313 R373 Y413 A1290 D1291 E1539 Y1655 A48 D49 E297 Y413 3.2.1.18 0004308 remove_due_to_license_issue Q59310 18218621 2692 VEGAVKTEPVDLFHPGFLNSSNYRIPALFKTKEGTLIASIDARRHGGADAPNNDIDTAVRRSEDGGKTWDEGQIIMDYPDKSSVIDTTLIQDDETGRIFLLVTHFPSKYGFWNAGLGSGFKNIDGKEYLCLYDSSGKEFTVRENVVYDKDSNKTEYTTNALGDLFKNGTKIDNINSSTAPLKAKGTSYINLVYSDDDGKTWSEPQNINFQVKKDWMKFLGIAPGRGIQIKNGEHKGRIVVPVYYTNEKGKQSSAVIYSDDSGKNWTIGESPNDNRKLENGKIINSKTLSDDAPQLTECQVVEMPNGQLKLFMRNLSGYLNIATSFDGGATWDETVEKDTNVLEPYCQLSVINYSQKVDGKDAVIFSNPNARSRSNGTVRIGLINQVGTYENGEPKYEFDWKYNKLVKPGYYAYSCLTELSNGNIGLLYEGTPSEEMSYIEMNLKYLES 2vkm A 2.05 BS01 BSD A 1 Q12 G13 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 I118 D228 G230 T231 T232 N233 R235 Q16 G17 L34 D36 G38 S39 Y75 T76 Q77 F112 W119 I122 D232 G234 T235 T236 N237 R239 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=1.8nM remove_due_to_license_issue IC50=1nM, Ki=1.8nM P56817 18180160 1386 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vl4 A 1.9 BS01 MNM A 1 W198 D199 W200 W395 N461 E462 W533 Y537 E555 W645 W656 W171 D172 W173 W368 N434 E435 W506 Y510 E528 W618 W629 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=975nM remove_due_to_license_issue Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGDRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKKEELPVNIKHIRETYK 2vl8 A 2.31 BS01 UDP A 1 I101 W102 I103 L265 S269 D286 V287 I101 W102 I103 L265 S269 D286 V287 2.4.1.-,3.4.22.- 0016757 remove_due_to_license_issue Q46342 18505687 1543 MNLVNKAQLQKMAYVKFRIQEDEYVAILNALEEYHNMSESSVVEKYLKLKDINNLTDNYLNTYKKSGRNKALKKFKEYLTMEVLELKNNSLTPVEKNLHFIWIGGQINDTAINYINQWKDVNSDYTVKVFYDSNAFLINTLKKTIVESATNNTLESFRENLNDPEFDYNKFYRKRMEIIYDKQKHFIDYYKSQIEENPEFIIDNIIKTYLSNEYSKDLEALNKYIEESLNKITANNGNDIRNLEKFADEDLVRLYNQELVERWNLAAASDILRISMLKEDGGVYLDVDMLPGIQPDLFKSINKPDSITNTSWEMIKLEAIMKYKEYIPGYTSKNFDMLDEEVQRSFESALSSKSDKSEIFLPLDDIKVSPLEVKIAFANNSVINQALISLKDSYCSDLVINQIKNRYKILNDNLNPSINEGTDFNTTMKIFSDKLASISNEDNMMFMIKITNYLKVGFAPDVRSTINLSGPGVYTGAYQDLLMFKDNSTNIHLLEPELRNFEFPKTKISQLTEQEITSLWSARAKSQFEEYKKGYFEGA 2vla A 1.3 BS01 dna L 0 R15 K63 N67 T70 E71 K75 M119 D120 K121 K124 K201 E202 S204 Y205 R15 K63 N67 T70 E71 K75 M119 D120 K121 K124 K201 E202 S204 Y205 3.1.21.4 remove_due_to_license_issue A3FMN7 18433771 101 ~ 112 MNYNPEEQFRCTIIRGKAKNMLDNLLPAYANIIDDICPCDKASFVKDFNNRLIEILGEETTKKTLDNHRTEIAGKLFGMFYEDDEVIFPSGRTNKYIEDSDQPAFFKDICFKFQFPNGMDKLDKVIEKVGAKIQIRQFPYILQVLLTADNNNIQLSKDDIAYYVLNSLQVLQGKIKPIEVIEKIIEDRSNDITKKVRHPGKETSYSMQHIREQLNYLELANLIRIDGNLVKLNYREAENINYIAQFWGNKPEFNAYKYDFTSEDDKKSFFKDWQQYYSNV 2vla A 1.3 BS02 dna M 0 R15 G16 K17 K19 N20 T61 K63 T64 N67 H68 K121 L122 Q208 R211 R15 G16 K17 K19 N20 T61 K63 T64 N67 H68 K121 L122 Q208 R211 3.1.21.4 remove_due_to_license_issue A3FMN7 18433771 201 ~ 212 MNYNPEEQFRCTIIRGKAKNMLDNLLPAYANIIDDICPCDKASFVKDFNNRLIEILGEETTKKTLDNHRTEIAGKLFGMFYEDDEVIFPSGRTNKYIEDSDQPAFFKDICFKFQFPNGMDKLDKVIEKVGAKIQIRQFPYILQVLLTADNNNIQLSKDDIAYYVLNSLQVLQGKIKPIEVIEKIIEDRSNDITKKVRHPGKETSYSMQHIREQLNYLELANLIRIDGNLVKLNYREAENINYIAQFWGNKPEFNAYKYDFTSEDDKKSFFKDWQQYYSNV 2vle A 2.4 BS01 DZN A 1 M124 F170 M174 W177 F292 F296 C301 C302 D457 V458 F459 M118 F164 M168 W171 F286 F290 C295 C296 D451 V452 F453 N169 K192 E268 C302 E399 E476 N163 K186 E262 C296 E393 E470 1.2.1.3 0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627 remove_due_to_license_issue IC50=80nM P05091 18613661 1501 AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS 2vle B 2.4 BS01 DZN B 1 M124 F170 L173 M174 W177 F292 F296 C301 D457 V458 F459 M118 F164 L167 M168 W171 F286 F290 C295 D451 V452 F453 N169 K192 E268 C302 E399 E476 N163 K186 E262 C296 E393 E470 1.2.1.3 0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627 remove_due_to_license_issue IC50=80nM P05091 18613661 1501 AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS 2vmc A 1.9 BS02 NGA A 1 Q216 R218 W238 Q211 R213 W233 ? 0005737,0005829,0007010,0007155,0009617,0009986,0016936,0030246,0030247,0031012,0031160,0031982,0045335,0046871,0046872,0070492,0098609,0098636,0140582 remove_due_to_license_issue P42530 18384150 505 GSVSCLANALLNLRSSTDYNADHGVKNSILNFSNSKDASRFDGSESWSSSVLDKNQFIVAGSDSVKHFVAISTQGRGDHDQWVTSYKLRYTLDNVNWVEYNNGEIINANKDRNSIVTINFNPPIKARSIAIHPQTYNNHISLRWELYALPVKSYSNPSVQVGEVSIGDRSLNSGTGSRTIVRHVKFPVEFLSVPIVSIGCKKVDAHTDNGQMRWEGKSENITTKGFDLTFITWGNNAVYDLTFDYVAVEFNN 2vmd A 1.9 BS02 MBG A 1 Q216 R218 W238 Q211 R213 W233 ? 0005737,0005829,0007010,0007155,0009617,0009986,0016936,0030246,0030247,0031012,0031160,0031982,0045335,0046871,0046872,0070492,0098609,0098636,0140582 Kd=0.95mM remove_due_to_license_issue P42530 18384150 501 GSVSCLANALLNLRSSTDYNADHGVKNSILNFSNSKDASRFDGSESWSSSVLDKNQFIVAGSDSVKHFVAISTQGRGDHDQWVTSYKLRYTLDNVNWVEYNNGEIINANKDRNSIVTINFNPPIKARSIAIHPQTYNNHISLRWELYALPVKSYSNPSVQVGEVSIGDRSLNSGTGSRTIVRHVKFPVEFLSVPIVSIGCKKVDAHTDNGQMRWEGKSENITTKGFDLTFITWGNNAVYDLTFDYVAVEFNN 2vmf A 2.1 BS01 MVL A 1 W198 D199 W200 W395 N461 E462 W533 Y537 E555 W645 W656 W171 D172 W173 W367 N433 E434 W505 Y509 E527 W617 W628 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=1400nM remove_due_to_license_issue Ki=1400nM Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKKGELPVNIKHIRETYK 2vnm A 1.79 BS01 CM8 A 1 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 Y259 D289 G291 T292 T293 N294 R296 N446 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 Y187 D217 G219 T220 T221 N222 R224 N374 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=3nM remove_due_to_license_issue IC50=3nM P56817 18457381 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vnm A 1.79 BS02 CM8 A 2 L145 T155 Q204 L84 T94 Q143 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=3nM remove_due_to_license_issue IC50=3nM P56817 18457381 2001 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vnn A 1.87 BS01 CM7 A 1 G72 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 Y259 D289 G291 T292 T293 N294 R296 N446 G11 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 Y187 D217 G219 T220 T221 N222 R224 N374 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=2nM remove_due_to_license_issue IC50=2nM P56817 18457381 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2vnp A 2.19 BS03 DED A 1 K21 R51 C67 G68 H69 R83 E114 E116 W161 K18 R48 C64 G65 H66 R80 E111 E113 W158 H25 H32 C67 H69 E87 Y104 E114 E116 W161 H22 H29 C64 H66 E84 Y101 E111 E113 W158 5.3.3.2 0000287,0003824,0004452,0005737,0006974,0008270,0008299,0016853,0046872,0050992 Ki=0.12nM remove_due_to_license_issue Q46822 18391416 1182 EHVILLNAQGVPTGTLEKYAAHTADTRLHLAFSSWLFNAKGQLLVTRRALSKKAWPGVWTNSVCGHPQLGESNEDAVIRRCRYELGVEITPPESIYPDFRYRATDPSGIVENEVCPVFAARTTSALQINDDEVMDYQWCDLADVLHGIDATPWAFSPWMVMQATNREARKRLSAFT 2vnt A 2.2 BS01 QGG A 1 D201 S202 Q204 S207 V225 W227 G228 R229 G230 C231 D201 S202 Q204 S207 V225 W227 G228 R229 G230 C231 H55 D106 Q204 G205 D206 S207 G208 H55 D106 Q204 G205 D206 S207 G208 3.4.21.73 0004252,0006508 Ki=9.9nM remove_due_to_license_issue Ki=9.9nM P00749 17447747 1258 KFQCGQKTLIIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLMSPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEE 2vo4 A 1.75 BS02 4NM A 1 W11 R20 Y32 K197 S198 P200 W11 R20 Y32 K197 S198 P200 2.5.1.18 0004364,0005737,0005829,0006749,0016740 remove_due_to_license_issue O49235 19014949 1221 MQDEVVLLDFWPSPFGMRVRIALAEKGIKYEYKEEDLRNKSPLLLQMNPVHKKIPVLIHNGKPICESLIAVQYIEEVWNDRNPLLPSDPYQRAQTRFWADYVDKKIYDLGRKIWTSKGEEKEAAKKEFIEALKLLEEQLGDKTYFGGDNLGFVDIALVPFYTWFKAYETFGTLNIESECPKFIAWAKRCLQKESVAKSLPDQQKVYEFIMDLRKKLGIE 2vo5 A 2.3 BS01 VBZ A 1 W198 D199 W200 W395 N461 E462 W470 W533 Y537 E555 W645 W656 W171 D172 W173 W368 N434 E435 W443 W506 Y510 E528 W618 W629 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=13uM remove_due_to_license_issue Ki=1.3e+4nM Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGDRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKLPVNIKHIRETYK 2vo7 A 1.98 BS02 M05 A 1 V15 F18 L152 E155 K292 I303 Y306 Q307 V2 F5 L139 E142 K279 I290 Y293 Q294 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=168nM remove_due_to_license_issue P00517 18345609 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2vo7 A 1.98 BS03 M05 A 2 T51 A70 M120 E121 Y122 V123 E127 L173 T183 D184 F327 T38 A57 M107 E108 Y109 V110 E114 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=168nM remove_due_to_license_issue P00517 18345609 1352 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 2vot A 1.95 BS01 NHV A 1 W198 D199 W200 W395 N461 E462 W470 W533 Y537 E555 W645 W656 W171 D172 W173 W368 N434 E435 W443 W506 Y510 E528 W618 W629 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=72nM remove_due_to_license_issue Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGDRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKKGEELPVNIKHIRETYK 2vpl A 2.3 BS01 rna B 0 H3 G4 R6 Y7 A35 K36 F37 T40 E42 H44 K46 D166 T168 H172 P174 S211 Y213 T217 M218 G219 S221 H3 G4 R6 Y7 A35 K36 F37 T40 E42 H44 K46 D75 T77 H81 P83 S120 Y122 T126 M127 G128 S130 ? remove_due_to_license_issue P27150 18778715 2 ~ 49 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 2vpl C 2.3 BS01 rna D 0 H3 G4 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 D166 T168 H172 P174 S211 Y213 T217 M218 G219 S221 H3 G4 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 D75 T77 H81 P83 S120 Y122 T126 M127 G128 S130 ? remove_due_to_license_issue P27150 18778715 2 ~ 49 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 2vpn A 1.55 BS01 4CS A 1 E8 E9 F66 R144 W167 N184 P185 W188 F209 E8 E9 F62 R140 W163 N180 P181 W184 F205 ? 0042597,0055085 Kd=0.19uM remove_due_to_license_issue E1VBK1 18702523 1311 DNWRYAHEEYEGDVQDVFAQAFKGYVEDNSDHTVQVYRFGELDIMEQTQNGILQFVNQSPGFTGSLIPSAQIFFIPYLMPTDMDTVLEFFDESKAINEMFPKLYAEHGLELLKMYPEGEMVVTADEPITSPEDFDNKKIRTMTNPLLAETYKAFGATPTPLPWGEVYGGLQTGIIDGQENPIFWIESGGLYEVSPNLTFTSHGWFTTAMMANQDFYEGLSEEDQQLVQDAADAAYDHTIEHIKGLSEESLEKIKAASDEVTVTRLNDEQIQAFKERAPQVEEKFIEMTGEQGQELLDQFKADLKAV 2vpo A 1.8 BS01 6CS A 1 E8 E9 F66 R144 N184 P185 W188 F209 E8 E9 F62 R140 N180 P181 W184 F205 ? 0042597,0055085 Kd=3.8uM remove_due_to_license_issue E1VBK1 18702523 1312 DNWRYAHEEYEGDVQDVFAQAFKGYVEDNSDHTVQVYRFGELDIMEQTQNGILQFVNQSPGFTGSLIPSAQIFFIPYLMPTDMDTVLEFFDESKAINEMFPKLYAEHGLELLKMYPEGEMVVTADEPITSPEDFDNKKIRTMTNPLLAETYKAFGATPTPLPWGEVYGGLQTGIIDGQENPIFWIESGGLYEVSPNLTFTSHGWFTTAMMANQDFYEGLSEEDQQLVQDAADAAYDHTIEHIKGLSEESLEKIKAASDEVTVTRLNDEQIQAFKERAPQVEEKFIEMTGEQGQELLDQFKADLKAVQ 2vpp A 2.2 BS01 GEO A 1 I29 E52 W57 Y70 F80 Q81 R105 A110 F114 E172 I12 E35 W40 Y53 F63 Q64 R88 A93 F97 E155 E52 R105 E35 R88 2.7.1.145 0004136,0004137,0004138,0004797,0004849,0005524,0005737,0005739,0006139,0006170,0006222,0009157,0009224,0016301,0019136,0043174,0043771,0071897,1901293 remove_due_to_license_issue Q9XZT6 19285960 1210 TQPFTVLIEGNIGSGKTTYLNHFEKYKNDICLLTEPVEKWRNVNGVNLLELMYKDPKKWAMPFQSYVTLTMLQSHTAPTNKKLKIMERSIFSARYCFVENMRRNGSLEQGMYNTLEEWYKFIEESIHVQADLIIYLRTSPEVAYERIRQRARSEESCVPLKYLQELHELHEDWLIHQRRPKVLVLDADL 2vqj A 2.1 BS01 TFG A 1 P156 H159 G167 F168 D196 H198 F227 G330 P151 H154 G162 F163 D191 H193 F222 G325 3.5.1.98 remove_due_to_license_issue P56524 18614528 1414 PRFTTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPLNRQKLDSKKLLGSLASVFVRLPCGGVGVDSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELDPLPEKVLQQRPNANAVRSMEKVMEIHSKYWRCLQRTTSTAGRSLIEAQTCENE 2vqm A 1.8 BS01 HA3 A 1 P156 G167 F168 H198 F227 P140 G151 F152 H182 F211 3.5.1.98 ic50=978nM remove_due_to_license_issue P56524 18614528 1410 PRFTTGLVYDTLMLKHQCTCGHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPLNRQKKLLGSLASVFVRLPCGGVGVDSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELDPLPEKVLQQRPNANAVRSMEKVMEIHSKYWRCLQRTTSTAGRSLIEAQTCENE 2vqt A 2.1 BS01 15A A 1 W198 D199 W200 W395 N461 E462 W533 Y537 E555 W645 W656 W171 D172 W173 W367 N433 E434 W505 Y509 E527 W617 W628 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=1uM remove_due_to_license_issue Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKKGEELPVNIKHIRETYK 2vr0 C 2.8 BS05 HQO C 1 F42 N67 K82 A85 G86 D89 F28 N53 K68 A71 G72 D75 1.10.2.- 0005886,0009055,0009061,0016020,0019333,0020037,0046872 remove_due_to_license_issue Q72EF4 18597779 1005 LVLGGATLGVVALATVAFGMKYTDQRPFCTSCHIMNPVGVTHKLSGHANISCNDCHAPHNLLAKLPFKAIAGARDVYMNTLGHPGDLILAGMETKEVVNANCKACHTMTNVEVASMEAKKYCTDCHRNVQHMRMKPISTREVAD 2vr4 A 1.8 BS01 17B A 1 W198 D199 W200 W395 N461 E462 W533 Y537 E555 W645 W656 W171 D172 W173 W368 N434 E435 W506 Y510 E528 W618 W629 3.2.1.25 0004553,0004567,0005576,0005975,0006516,0016798 Ki=2.1uM remove_due_to_license_issue Q8AAK6 18408714 1865 NDTSEVMLLDTGWEFSQSGTEKWMPATVPGTVHQDLISHELLPNPFYGMNEKKIQWVENEDWEYRTSFIVSEEQLNRDGIQLIFEGLDTYADVYLNGSLLLKADNMFVGYTLPVKSVLRKGENHLYIYFHSPIRQTLPQYASNGFNYPADNDHHEKHLSVFSRKAPYSYGWDWGIRMVTSGVWRPVTLRFYDIATISDYYVRQLSLTDENARLSNELIVNQIVPQKIPAEVRVNVSLNGTTVTEVKQQVTLQPGINHITLPAEVTNPVRWMPNGWGTPTLYDFSAQIACGDRIVAEQSHRIGLRTIRVVNEKDKDGESFYFEVNGIPMFAKGANYIPQDALLPNVTTERYQTLFRDMKEANMNMVRIWGGGTYENNLFYDLADENGILVWQDFMFACTPYPSDPTFLKRVEAEAVYNIRRLRNHASLAMWCGNNEILEALKYWGFEKKFTPEVYQGLMHGYDKLFRELLPSTVKEFDSDRFYVHSSPYLANWGRPESWGTGDSHNWGVWYGKKPFESLDTDLPRFMSEFGFQSFPEMKTIAAFAAPEDYQIESEVMNAHQKSSIGNSLIRTYMERDYIIPESFEDFVYVGLVLQGQGMRHGLEAHRRNRPYCMGTLYWQLNDSWPVVSWSSIDYYGNWKALHYQAKRAFAPVLINPIQQNDSLSVYLISDRLDTMEQMTLEMKVVDFDGKTLGKKIQVHSLEVPANTSKCVYRAKLDGWLTPEDCRRSFLKLILKDKSGHQVAESVHFFRKTKDLQLPPTSVSYQMKQTDGKCELTLFSSMLAKDIFIETPLQGARYSDNFFDLLPGERKKVIITSPRIKKGELPVNIKHIRETYK 2vrj A 1.9 BS01 NCW A 1 Q20 H121 E166 H180 Y295 E351 W398 E405 W406 A407 E408 Q18 H119 E164 H178 Y290 E344 W391 E398 W399 A400 E401 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N288 Y290 E344 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=0.5uM remove_due_to_license_issue Q08638 18833549 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2vrx A 1.86 BS01 447 A 1 L99 V107 K122 E141 Q145 L154 L168 L170 F172 A173 P174 G176 L223 L13 V21 K36 E55 Q59 L68 L82 L84 F86 A87 P88 G90 L137 D216 K218 E220 N221 D234 T252 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=45nM Q6DE08 18559266 1356 KFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY 2vt3 A 2.0 BS01 ATP A 1 V93 G94 D118 I119 K123 L136 V153 P154 V75 G76 D94 I95 K99 L112 V129 P130 ? 0003677,0003700,0005737,0006355,0045892,0051775 remove_due_to_license_issue O05521 18485070 302 ATAKRLPLYYRFLKNLHASGKQRVSSAELSDAVKVDSATIRRDFSYFGALGYNVDYLLSFFRKTLDQDDVILIGVGNLGTAFLHYNTKISMAFDINESKIGTEVGGVPVYNLDDLEQHVKDESVAILTVPAVAAQSITDRLVALGIKGILNFTPARLNVPEHIRIHHIDLAVELQSLVYFLKHYS 2vt3 B 2.0 BS01 ATP B 1 G92 V93 G94 N95 D118 I119 K123 P154 G86 V87 G88 N89 D112 I113 K117 P148 ? 0003677,0003700,0005737,0006355,0045892,0051775 remove_due_to_license_issue O05521 18485070 302 KIPQATAKRLPLYYRFLKNLHASGKQRVSSAELSDAVKVDSATIRRDFSYFGALGKKGYGYNVDYLLSFFRKTLDQDEMTDVILIGVGNLGTAFLHYNFTKNNNTKISMAFDINESKIGTEVGGVPVYNLDDLEQHVKDESVAILTVPAVAAQSITDRLVALGIKGILNFTPARLNVPEHIRIHHIDLAVELQSLVYFLKHYSVLEEI 2vta A 2.0 BS01 LZ1 A 1 A31 F82 L83 L134 A31 F73 L74 L125 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=185uM remove_due_to_license_issue IC50=185000nM P24941 18656911 1301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtd A 1.94 BS01 LKM A 1 D35 T36 R37 F161 H183 K348 A414 S415 L416 N421 F422 H439 D35 T36 R37 F161 H183 K343 A409 S410 L411 N416 F417 H434 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=85uM remove_due_to_license_issue Kd=7000nM, IC50=85000nM P14900 19007109 1441 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRERCVSFGVNMGDYHLNHGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2vte A 2.2 BS01 IK4 A 1 D35 T36 R37 G73 H183 K348 A414 S415 N421 F422 S438 D35 T36 R37 G73 H183 K343 A409 S410 N416 F417 S433 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=122uM remove_due_to_license_issue IC50=122000nM P14900 19007109 1440 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRERCVSFGVNMGDYHLNHQETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGS 2vth A 1.9 BS01 LZ2 A 1 I10 A31 E81 F82 L83 L134 I10 A31 E72 F73 L74 L125 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=120uM remove_due_to_license_issue IC50=120000nM P24941 18656911 1300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vti A 2.0 BS01 LZ3 A 1 I10 A31 F80 E81 L83 H84 Q85 D86 K89 L134 I10 A31 F72 E73 L75 H76 Q77 D78 K81 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T147 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.66uM remove_due_to_license_issue IC50=660nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtj A 2.2 BS01 LZ4 A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 I10 A31 F71 F73 L74 H75 Q76 D77 K80 L125 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T143 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1.9uM remove_due_to_license_issue IC50=9100nM P24941 18656911 1300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtl A 2.0 BS01 LZ5 A 1 A31 E81 F82 L83 H84 L134 A31 E73 F74 L75 H76 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=97uM remove_due_to_license_issue IC50=97000nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtm A 2.25 BS01 LZM A 1 A31 K33 F80 E81 L83 L134 A31 K33 F72 E73 L75 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50~1mM remove_due_to_license_issue P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtn A 2.2 BS01 LZ7 A 1 A31 F80 E81 F82 L83 H84 L134 D145 A31 F72 E73 F74 L75 H76 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T141 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.85uM remove_due_to_license_issue IC50=850nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vto A 2.19 BS01 LZ8 A 1 V18 A31 E81 F82 L83 H84 D86 L134 D145 V18 A31 E74 F75 L76 H77 D79 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.14uM remove_due_to_license_issue IC50=140nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtp A 2.15 BS01 LZ9 A 1 I10 V18 A31 E81 F82 L83 H84 D86 L134 A144 D145 I10 V18 A31 E73 F74 L75 H76 D78 L126 A136 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T148 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.003uM remove_due_to_license_issue IC50=3.0nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtq A 1.9 BS01 LZA A 1 V18 A31 E81 F82 L83 H84 Q85 L134 D145 V18 A31 E72 F73 L74 H75 Q76 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T141 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.14uM remove_due_to_license_issue IC50=140nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtr A 1.89 BS01 LZB A 1 A31 V64 F80 F82 L83 H84 L134 A31 V56 F72 F74 L75 H76 L126 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=1.5uM remove_due_to_license_issue IC50=1500nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vts A 1.9 BS01 LZC A 1 I10 A31 K33 F80 F82 L83 H84 Q85 N132 L134 D145 I10 A31 K33 F72 F74 L75 H76 Q77 N124 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.03uM remove_due_to_license_issue IC50=30nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vtt A 1.68 BS01 LZD A 1 I10 V18 A31 K33 E81 L83 H84 D86 L134 D145 I10 V18 A31 K33 E70 L72 H73 D75 L123 D134 D127 K129 Q131 N132 D145 T165 D116 K118 Q120 N121 D134 T139 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.044uM remove_due_to_license_issue IC50=44nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vu3 A 1.85 BS01 LZE A 1 I10 V18 A31 K33 F80 E81 F82 L83 H84 L134 D145 I10 V18 A31 K33 F71 E72 F73 L74 H75 L125 D136 D127 K129 Q131 N132 D145 T158 T165 D118 K120 Q122 N123 D136 T145 T152 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.047uM remove_due_to_license_issue IC50=47nM, Ki=510nM, Kd=30nM P24941 18656911 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vuk B 1.5 BS01 P83 B 1 L145 V147 T150 P151 C220 E221 P222 P223 D228 T230 L51 V53 T56 P57 C126 E127 P128 P129 D134 T136 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=125uM remove_due_to_license_issue Kd=140000nM P04637 18650397 1291 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 2vur A 2.2 BS01 YX1 A 1 G187 D297 V331 Y335 V370 W394 D401 G147 D257 V291 Y295 V330 W354 D361 3.2.1.169 ic50=30uM remove_due_to_license_issue Q0TR53 18721751 1626 VLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYNRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2vv9 A 1.9 BS01 IM9 A 1 I10 V18 A31 K33 L83 K89 L134 D145 I10 V18 A31 K33 L77 K83 L128 D139 D127 K129 Q131 N132 D145 T165 D121 K123 Q125 N126 D139 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.017uM remove_due_to_license_issue IC50=17nM P24941 18617397 1300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2vvc A 1.95 BS01 LZF A 1 T98 Y99 E147 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 T84 Y85 E135 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=3nM P00742 19200624 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2vvn A 1.85 BS01 NHT A 1 G135 K166 D242 D243 C278 Y282 W337 N339 D344 G132 K163 D239 D240 C275 Y279 W334 N336 D341 3.2.1.169 remove_due_to_license_issue Q89ZI2 18587388 1718 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMLPLQVKANRVLISPVEIELDAIYPGENIQINFRLSAGLQKAPVKFVRFQFVLTIEK 2vvo A 1.85 BS01 A6P A 1 D11 H12 G69 G70 S71 G74 E75 R113 D9 H10 G67 G68 S69 G72 E73 R111 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 ic50=6.3mM remove_due_to_license_issue P9WKD7 18640127 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVP 2vvo A 1.85 BS02 A6P B 1 H102 N103 R137 R141 H100 N101 R135 R139 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 ic50=6.3mM remove_due_to_license_issue P9WKD7 18640127 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVP 2vvo B 1.85 BS01 A6P A 1 H102 N103 R137 R141 H100 N101 R135 R139 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 ic50=6.3mM remove_due_to_license_issue P9WKD7 18640127 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVP 2vvo B 1.85 BS02 A6P B 1 D11 H12 Y46 G69 G70 S71 G74 E75 R113 D9 H10 Y44 G67 G68 S69 G72 E73 R111 D11 G69 S71 H102 H138 D9 G67 S69 H100 H136 5.3.1.6 0004751,0005515,0005576,0005975,0006098,0009052,0016853,0016861,0019316 ic50=6.3mM remove_due_to_license_issue P9WKD7 18640127 200 GMRVYLGADHAGYELKQRIIEHLKQTGHEPIDCGALRYDADDDYPAFCIAAATRTVADPGSLGIVLGGSGNGEQIAANKVPGARCALAWSVQTAALAREHNNAQLIGIGGRMHTVAEALAIVDAFVTTPWSKAQRHQRRIDILAEYERTHEAPPVP 2vvs A 2.24 BS01 OAN A 1 G135 K166 D242 D243 Y282 W286 V314 W337 N339 D344 H433 G123 K154 D230 D231 Y270 W274 V302 W325 N327 D332 H421 3.2.1.169 Ki=46nM remove_due_to_license_issue Q89ZI2 18842583 900 LQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMP 2vvt A 1.65 BS01 I24 A 1 V14 V152 E153 N155 H187 L190 I250 W254 V20 V158 E159 N161 H193 L196 I251 W255 D11 S12 C74 E153 C185 H187 D17 S18 C80 E159 C191 H193 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 ic50=5.8uM remove_due_to_license_issue IC50=5800nM Q836J0 18614367 1269 VPRGSHMSNQEAIGLIDSGVGGLTVLKEALKQLPNERLIYLGDTARCPYGPRPAEQVVQFTWEMADFLLKKRIKMLVIACNTATAVALEEIKAALPIPVVGVILPGARAAVKVTKNNKIGVIGTLGTIKSASYEIAIKSKAPAIEVTSLACPKFVPIVESNQYRSSVAKKIVAETLQALQLKGLDTLILGCTHYPLLRPVIQNVMGSHVTLIDSGAETVGEVSMLLDYFDIAHTPPHEFYTTGSAKMFEEIASSWLGIENLKAQQIHLG 2vvu A 2.3 BS01 H22 A 1 E97 T98 Y99 F174 D189 A190 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=8nM P00742 19200624 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2vvv A 1.73 BS01 H21 A 1 E97 T98 Y99 F174 D189 A190 C191 Q192 V213 W215 G216 G218 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 C181 Q182 V203 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=6nM P00742 19200624 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2vw1 A 2.39 BS01 DAN A 1 R245 D270 I326 D327 N352 T539 R557 R619 Y653 W674 R207 D232 I288 D289 N314 T501 R519 R581 Y615 W636 D270 E541 Y653 D232 E503 Y615 3.2.1.18 0004308,0005975 Ki=0.3mM remove_due_to_license_issue Q54727 18835278 1000 ISPIFQGGSYQLNNKSIDISSLLLDKLSGESQTVVMKFKADKPNSLQALFGLSNSKAGFKNNYFSIFMRDSGEIGVEIRDAQKGINYLFSRPASLWGKHKGQAVENTLVFVSDSKDKTYTMYVNGIEVFSETVDTFLPISNINGIDKATLGAVNREGKEHYLAKGSIDEISLFNKAISDQEVSTIPLSNPFQLIFQSGDSTQANYFRIPTLYTLSSGRVLSSIDARYGGTHDSKSKINIATSYSDDNGKTWSEPIFAMKFNDYEEQLVYWPRDNKLKNSQISGSASFIDSSIVEDKKSGKTILLADVMPAGIGNNNANKADSGFKEINGHYYLKLKKNGDNDFRYTVRENGVVYNETTNKPTNYTINDKYEVLEGGKSLTVEQYSVDFDSGSLRERHNGKQVPMNVFYKDSLFKVTPTNYIAMTTSQNRGESWEQFKLLPPFLGEKHNGTYLCPGQGLALKSSNRLIFATYTSGELTYLISDDSGQTWKKSSASIPFKNATAEAQMVELRDGVIRTFFRTTTGKIAYMTSRDSGETWSKVSYIDGIQQTSYGTQVSAIKYSQLIDGKEAVILSTPNSRSGRKGGQLVVGLVNKEDDSIDWKYHYDIDLPSYGYAYSAITELPNHHIGVLFEKYDSWSRNELHLSNVVQYIDLEINDLT 2vw2 A 1.7 BS01 NHE A 1 R245 D270 D327 N352 Y489 R557 R619 Y653 W674 R207 D232 D289 N314 Y451 R519 R581 Y615 W636 D270 E541 Y653 D232 E503 Y615 3.2.1.18 0004308,0005975 remove_due_to_license_issue Q54727 18835278 1000 ISPIFQGGSYQLNNKSIDISSLLLDKLSGESQTVVMKFKADKPNSLQALFGLSNSKAGFKNNYFSIFMRDSGEIGVEIRDAQKGINYLFSRPASLWGKHKGQAVENTLVFVSDSKDKTYTMYVNGIEVFSETVDTFLPISNINGIDKATLGAVNREGKEHYLAKGSIDEISLFNKAISDQEVSTIPLSNPFQLIFQSGDSTQANYFRIPTLYTLSSGRVLSSIDARYGGTHDSKSKINIATSYSDDNGKTWSEPIFAMKFNDYEEQLVYWPRDNKLKNSQISGSASFIDSSIVEDKKSGKTILLADVMPAGIGNNNANKADSGFKEINGHYYLKLKKNGDNDFRYTVRENGVVYNETTNKPTNYTINDKYEVLEGGKSLTVEQYSVDFDSGSLRERHNGKQVPMNVFYKDSLFKVTPTNYIAMTTSQNRGESWEQFKLLPPFLGEKHNGTYLCPGQGLALKSSNRLIFATYTSGELTYLISDDSGQTWKKSSASIPFKNATAEAQMVELRDGVIRTFFRTTTGKIAYMTSRDSGETWSKVSYIDGIQQTSYGTQVSAIKYSQLIDGKEAVILSTPNSRSGRKGGQLVVGLVNKEDDSIDWKYHYDIDLPSYGYAYSAITELPNHHIGVLFEKYDSWSRNELHLSNVVQYIDLEINDLT 2vw2 A 1.7 BS02 NHE A 2 K334 K499 E658 K296 K461 E620 D270 E541 Y653 D232 E503 Y615 3.2.1.18 0004308,0005975 remove_due_to_license_issue Q54727 18835278 1001 ISPIFQGGSYQLNNKSIDISSLLLDKLSGESQTVVMKFKADKPNSLQALFGLSNSKAGFKNNYFSIFMRDSGEIGVEIRDAQKGINYLFSRPASLWGKHKGQAVENTLVFVSDSKDKTYTMYVNGIEVFSETVDTFLPISNINGIDKATLGAVNREGKEHYLAKGSIDEISLFNKAISDQEVSTIPLSNPFQLIFQSGDSTQANYFRIPTLYTLSSGRVLSSIDARYGGTHDSKSKINIATSYSDDNGKTWSEPIFAMKFNDYEEQLVYWPRDNKLKNSQISGSASFIDSSIVEDKKSGKTILLADVMPAGIGNNNANKADSGFKEINGHYYLKLKKNGDNDFRYTVRENGVVYNETTNKPTNYTINDKYEVLEGGKSLTVEQYSVDFDSGSLRERHNGKQVPMNVFYKDSLFKVTPTNYIAMTTSQNRGESWEQFKLLPPFLGEKHNGTYLCPGQGLALKSSNRLIFATYTSGELTYLISDDSGQTWKKSSASIPFKNATAEAQMVELRDGVIRTFFRTTTGKIAYMTSRDSGETWSKVSYIDGIQQTSYGTQVSAIKYSQLIDGKEAVILSTPNSRSGRKGGQLVVGLVNKEDDSIDWKYHYDIDLPSYGYAYSAITELPNHHIGVLFEKYDSWSRNELHLSNVVQYIDLEINDLT 2vw5 A 1.9 BS01 BC6 A 1 N37 D40 A41 K44 D79 N92 K98 G121 V122 F124 N37 D40 A41 K44 D79 N92 K98 G121 V122 F124 ? 0005524,0006457,0016887,0051082,0140662 Kd=3nM remove_due_to_license_issue P02829 18800759 500 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2vwc A 2.4 BS01 BC2 A 1 N37 D40 A41 K44 M84 N92 L93 K98 G121 V122 F124 E214 N36 D39 A40 K43 M83 N91 L92 K97 G120 V121 F123 E213 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.24uM remove_due_to_license_issue P02829 18357975 1215 ASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2vwj A 2.78 BS01 dna B 0 D6 Y7 Y37 V93 Y112 D113 I114 P115 F116 K240 Q242 R265 P271 Y273 R612 R613 T667 R668 Y673 K674 R709 I710 G711 N735 D6 Y7 Y37 V93 Y112 D113 I114 P115 F116 K240 Q242 R265 P271 Y273 R612 R613 T667 R668 Y673 K674 R709 I710 G711 N735 2.7.7.7 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0034061,0071897 remove_due_to_license_issue P56689 18614176 0 ~ 25 MILDTDYITEDGKPVIRIFKKENGEFKIDYDRNFEPYIYALLKDDSAIEDVKKITAERHGTTVRVVRAEKVKKKFLGRPIEVWKLYFTHPQDVPAIRDKIKEHPAVVDIYEYDIPFAKRYLIDKGLIPMEGDEELKMLAFDIETLYHEGEKFAEGPILMISYADEEGARVITWRNIDLPYVDVVSTEKEMIKRFLKVVKEKDPDVLITYNGDNFAFAYLKKRSEKLGVKFILGREGSEPKIQRMGDRFAVEVKGRIHFDLYPVIRRTINLPTYTLEAVYEAIFGQPKEKVYAEEIAQAWETGEGLERVARYSMEDAKVTYELGKEFFPMEAQLSRLVGQSLWDVSRSSTGNLVEWFLLRKAYERNELAPNKPDERELARRRESYAGGYVKEPERGLWENIVYLDFRSLYPSIIITHNVSPDTLNREGCEEYDVAPQVGHKFCKDFPGFIPSLLGDLLEERQKVKKKMKATIDPIEKKLLDYRQRAIKILANSFYGYYGYAKARWYCKECAESVTAWGRQYIETTIREIEEKFGFKVLYADTDGFFATIPGADAETVKKKAKEFLDYINAKLPGLLELEYEGFYKRGFFVTKKKYAVIDEEDKITTRGLEIVRRDWSEIAKETQARVLEAILKHGDVEEAVRIVKEVTEKLSKYEVPPEKLVIYEQITRDLKDYKATGPHVAVAKRLAARGIKIRPGTVISYIVLKGSGRIGDRAIPFDEFDPAKHKYDAEYYIENQVLPAVERILRAFGYRKEDLRY 2vwl A 1.8 BS01 LZH A 1 E97 T98 Y99 F174 D189 A190 C191 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 C181 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=95nM P00742 19200624 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2vwm A 1.96 BS01 LZI A 1 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 E217 G218 C220 G226 I227 Y228 T83 Y84 F161 D178 A179 Q181 V202 W204 G205 E206 G207 C208 G215 I216 Y217 H57 D102 Q192 G193 D194 S195 G196 H42 D87 Q181 G182 D183 S184 G185 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=93nM P00742 19200624 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2vwn A 1.61 BS01 H25 A 1 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=10nM P00742 19200624 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2vwo A 1.6 BS01 LZG A 1 E97 T98 Y99 F174 D189 A190 C191 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 C181 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=31nM P00742 19200624 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2vwu A 2.0 BS01 7X1 A 1 I621 A645 K647 E664 I691 T693 M696 E697 G699 L747 S757 I13 A37 K39 E52 I79 T81 M84 E85 G87 L135 S145 D740 A742 R744 N745 D758 P783 D128 A130 R132 N133 D146 P149 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.35uM remove_due_to_license_issue IC50=350nM P54760 18434142 1888 EIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIV 2vwv A 1.9 BS01 7X3 A 1 I621 V629 A645 T693 M696 G699 L747 I16 V24 A40 T84 M87 G90 L138 D740 A742 R744 N745 D758 K781 P783 D131 A133 R135 N136 D149 K151 P153 2.7.10.1 0004672,0004713,0005524,0006468 ic50=16uM remove_due_to_license_issue IC50=16000nM P54760 18434142 1888 FAKEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLK 2vww A 1.9 BS01 7X2 A 1 I621 A645 K647 E664 I677 I691 T693 M696 G699 A700 L747 S757 I13 A37 K39 E52 I65 I79 T81 M84 G87 A88 L135 S145 D740 A742 R744 N745 D758 P783 D128 A130 R132 N133 D146 P149 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.24uM remove_due_to_license_issue IC50=240nM P54760 18434142 1888 EIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIV 2vwx A 1.65 BS01 7X4 A 1 I621 A645 K647 E664 I691 T693 F695 M696 E697 N698 G699 L747 S757 I14 A38 K40 E57 I84 T86 F88 M89 E90 N91 G92 L140 S150 D740 A742 R744 N745 D758 K781 P783 D133 A135 R137 N138 D151 K167 P169 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.04uM remove_due_to_license_issue IC50=40nM P54760 18851911 1889 KEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLEENSSDGGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2vwy A 1.65 BS01 7X5 A 1 I621 A645 K647 E664 I691 T693 M696 G699 L747 S757 I14 A38 K40 E57 I84 T86 M89 G92 L140 S150 D740 A742 R744 N745 D758 K781 P783 D133 A135 R137 N138 D151 K167 P169 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.09uM remove_due_to_license_issue IC50=90nM P54760 18851911 1889 KEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLEENSSDGGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2vwz A 1.65 BS01 7X6 A 1 I621 A645 K647 E664 I691 T693 M696 G699 L747 I14 A38 K40 E57 I84 T86 M89 G92 L140 D740 A742 R744 N745 D758 K781 P783 D133 A135 R137 N138 D151 K167 P169 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.794uM remove_due_to_license_issue IC50=741nM P54760 18851911 1889 KEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLEENSSDGGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2vx0 A 2.1 BS01 7X7 A 1 I621 A645 K647 E664 I691 T693 M696 E697 G699 L747 S757 I14 A38 K40 E57 I84 T86 M89 E90 G92 L140 S150 D740 A742 R744 N745 D758 K781 P783 D133 A135 R137 N138 D151 K166 P168 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.58uM remove_due_to_license_issue IC50=580nM P54760 18434142 1889 KEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLEENSSDGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2vx1 A 1.65 BS01 7X8 A 1 I621 A645 K647 E664 I691 T693 M696 G699 L747 S757 I14 A38 K40 E57 I84 T86 M89 G92 L140 S150 D740 A742 R744 N745 D758 K781 P783 D133 A135 R137 N138 D151 K167 P169 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.22uM remove_due_to_license_issue IC50=900nM P54760 18851911 1889 KEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLEENSSDGGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2vx9 A 1.65 BS01 RBF A 1 V35 W36 V34 W35 ? 0005737,0005829 remove_due_to_license_issue B0R5M0 19224924 1064 VFKKVLLTGTSEESFTAAADDAIDRAEDTLDNVVWAEVVDQGVAIGAVEERTYQTEVQVAFEL 2vxa A 2.6 BS01 RBF A 1 Y6 W39 Y4 W37 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa A 2.6 BS02 RBF L 1 R46 H48 Q58 R44 H46 Q56 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa C 2.6 BS01 RBF C 1 Y6 W39 Y4 W37 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa C 2.6 BS02 RBF F 1 R46 H48 Q58 R44 H46 Q56 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa E 2.6 BS01 RBF A 1 R46 H48 Q58 R44 H46 Q56 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa E 2.6 BS02 RBF E 1 Y6 W39 Y4 W37 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa F 2.6 BS01 RBF F 1 Y6 W39 Y4 W37 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxa F 2.6 BS02 RBF G 1 R46 H48 Q58 R44 H46 Q56 ? 0000166 remove_due_to_license_issue A1WUH0 19224924 200 DHVYKIVELTGSSPNGIEEAVNNAIARAGETLRHLRWFEVVDTRGHIEGGRVNHWQVTVKVGFTLE 2vxn A 0.82 BS01 PGH A 1 K13 H95 E167 I172 G173 G212 S213 L232 G234 G235 K12 H94 E166 I171 G172 G211 S212 L231 G233 G234 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 remove_due_to_license_issue P48499 20235230 1251 AKPQPIAAANWKCNGTTASIEKLVQVFNEHTISHDVQCVVAPTFVHIPLVQAKLRNPKYVISAQNAIAKSGAFTGEVSMPILKDIGVHWVILGHSERRTYYGETDEIVAQKVSEACKQGFMVIACIGETLQQREANQTAKVVLSQTSAIAAKLTKDAWNQVVLAYEPVWAIGTGKVATPEQAQEVHLLLRKWVSENIGTDVAAKLRILYGGSVNAANAATLYAKPDINGFLVGGASLKPEFRDIIDATR 2vy1 A 2.104 BS01 dna W 0 R237 T290 N291 R295 K307 Y377 T380 A398 A399 R1 T54 N55 R59 K71 Y141 T144 A162 A163 ? 0003677,0006355 remove_due_to_license_issue Q00958 18784751 1 ~ 20 REHPFIVTEPGEVARGKKNGLDYLFHLYEQCREFLLQVQTIAKDRGEKCPTKVTNQVFRYAKKSGASYINKPKMRHYVHCYALHCLDEEASNALRRAFKERGENVGSWRQACYKPLVNIACRHGWDIDAVFNAHPRLSIWYVPTKLRQLCHLERNNAVAAAAA 2vye A 4.1 BS01 dna C 0 Q326 R330 R332 Q318 R322 R324 3.6.4.12 0003677,0003678,0003689,0004386,0005524,0005829,0006260,0006268,0006269,0006338,0009378,0016787,0016853,0016887,0036121,0061749,0061775,0140584,0140588,0140665,0140849,1990077,1990518 remove_due_to_license_issue Q5KU75 19074952 2001 ~ 2009 IPPQSIEAEQAVLGAVFLDPTALTLASERLIPEDFYRAAHQKIFHAMLRVADKGEPVDLVTVTAELAALEQLEEVGGVSYLSELADSVPTAANVEYYARIVEEKSLLRRLIRTATSIAQDGYTREDEIDVLLDEAERKIMEVSQRKHSGAFKNIKDVLVQTYDNIEMLHNRNGDITGIPTGFTELDRMTSGFQRSDLIIVAARPSVGKTAFALNIAQNVATKTNENVAIFSLEMSAQQLVMRMLCAEGNINAQNLRTGKLTPEDWGKLTMAMGSLSNAGIYIDDTPSIRVSDIRAKCRRLKQESGLGMVVIDYLQLIQGSGRNRENRQQEVSEISRSLKALARELEVPVIALSQLSRSVEQRQDPMMSDLRESGSIEQDADIVAFLYRDDNKDSENKNIIEIIIAKQRNGVQLAFIKEYNKFVN 2vye B 4.1 BS01 dna C 0 R1045 Q1079 R1117 R1120 R1145 K1146 E1149 R1330 R1332 R1344 T1426 R39 Q73 R111 R114 R139 K140 E143 R311 R313 R325 T380 3.6.4.12 0003677,0003678,0003689,0004386,0005524,0005829,0006260,0006268,0006269,0006338,0009378,0016787,0016853,0016887,0036121,0061749,0061775,0140584,0140588,0140665,0140849,1990077,1990518 remove_due_to_license_issue Q5KU75 19074952 2001 ~ 2009 ERIPPQSIEAEQAVLGAVFLDPTALTLASERLIPEDFYRAAHQKIFHAMLRVADKGEPVDLVTVTAELAALEQLEEVGGVSYLSELADSVPTAANVEYYARIVEEKSLLRRLIRTATSIAQDGYTREDEIDVLLDEAERKIMEVSQRKHSGAFKDVLVQTYDNIEMLHNRNGDITGIPTGFTELDRMTSGFQRSDLIIVAARPSVGKTAFALNIAQNVATKTNENVAIFSLEMSAQQLVMRMLCAEGNLTPEDWGKLTMAMGSLSNAGIYIDDTPSIRVSDIRAKCRRLKQESGLGMVVIDYLQLIQGSGRNRENRQQEVSEISRSLKALARELEVPVIALSQLSRSVEQRQDKRDLRESGSIEQDADIVAFIIAKQRGT 2vyt A 1.9 BS01 MLZ A 1 D182 N185 F206 W209 F213 D153 N156 F177 W180 F184 ? 0005634,0006355 Kd=1.84mM remove_due_to_license_issue Q9UQR0 18706910 1244 RDDFHWEEYLKETGSISAPSECFRQSQIPPVNDFKVGMKLEARDPRNATSVCIATVIGITGARLRLRLDGSDNRNDFWRLVDSPDIQPVGTCEKEGDLLQPPLGYQMNTSSWPMFLLETLNGSEMASATLFKKEPPKPPLNNFKVGMKLEAIDKKNPYLICPATIGDVKGDEVHITFDGWSGAFDYWCKYDSRDIFPAGWCRLTGDVLQPPGTS 2vzr A 1.95 BS02 GCU A 1 H22 N32 N35 R67 W90 N121 H20 N30 N33 R65 W88 N119 3.2.1.165 0030246 Ka=19000M^-1 remove_due_to_license_issue Q56F26 19218457 1129 PVDYQAEDATIVQGAVESNHAGYTGTGFVNYDNVAGSSVEWTVTVPSAGTYDVVVRYANGTTTSRPLDFSVNGSISASGVAFGSTGTWPAWTTKTVRVTLAAGVNKIKAVATTANGGPNVDKITL 2w05 A 1.9 BS01 FRT A 1 I10 V18 A31 V64 E81 L83 H84 Q85 D86 K89 L134 I10 V18 A31 V55 E72 L74 H75 Q76 D77 K80 L125 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T143 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.001uM remove_due_to_license_issue IC50=1nM P24941 18815031 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2w06 A 2.04 BS01 FRV A 1 I10 V18 A31 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 V18 A31 F73 F75 L76 H77 Q78 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 18815031 1300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2w08 A 1.7 BS03 TPO A 1 N59 Y74 E136 Q148 N59 Y74 E136 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=380uM remove_due_to_license_issue P02743 19372378 500 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w0d A 2.0 BS06 CGS A 1 I180 L181 A182 H218 H222 H228 P238 Y240 I75 L76 A77 H113 H117 H123 P133 Y135 H218 A219 H222 H228 H113 A114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM remove_due_to_license_issue P39900 19239231 1273 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2w0d A 2.0 BS07 CGS C 1 G179 I180 G74 I75 H218 A219 H222 H228 H113 A114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM remove_due_to_license_issue P39900 19239231 1273 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2w0j A 2.05 BS01 ZAT A 1 L226 I251 E273 L301 M304 G307 L354 T367 D368 L17 I39 E46 L74 M77 G80 L127 T140 D141 D347 K349 N352 D368 T387 D120 K122 N125 D141 T158 2.7.11.1 0004672,0005524,0006468 ic50=240nM remove_due_to_license_issue O96017 19177354 1511 SVYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENETALPQ 2w0s A 2.918 BS03 BVP A 1 D13 L53 N65 F68 R72 R93 G98 Y101 A102 Y144 D12 L52 N64 F67 R71 R92 G97 Y100 A101 Y143 2.7.4.9 0004550,0004798,0005524,0006227,0006233,0006235,0009165,0016301,0046940 remove_due_to_license_issue P68693 18971333 1207 SRGALIVFEGLDKSGKTTQCMNIMESIPANTIKYLNFPQRSTVTGKMIDDYLTRKKTYNDHIVNLLFCANRWEFASFIQEQLEQGITLIVDRYAFSGVAYAAAKGASMTLSKSYESGLPKPDLVIFLESGSKEINRNVGEEIYEDVTFQQKVLQEYKKMIEEGDIHWQIISSEFEEDVKKELIKNIVIEAIHTVTGPVGQLWM 2w0x A 2.12 BS02 PD2 A 1 Y145 T196 H199 N205 F207 K214 H279 I281 N294 W296 Y138 T189 H192 N198 F200 K207 H272 I274 N287 W289 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=625uM remove_due_to_license_issue IC50=8600nM Q9NWT6 20822901 1351 AVASGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2w12 A 1.46 BS02 WR2 A 1 N106 T107 I108 G109 R110 H142 E143 H146 H152 S168 V169 L170 N106 T107 I108 G109 R110 H142 E143 H146 H152 S168 V169 L170 3.4.24.- 0004222,0006508,0008237 remove_due_to_license_issue P83512 19485419 1204 ERFSPRYIELAVVADHGIFTKYNSNLNTIRTRVHEMLNTVNGFYRSVDVHAPLANLEVWSKQDLIKVQKDSSKTLKSFGEWRERDLLPRISHDHAQLLTAVVFDGNTIGRAYTGGMCDPRHSVGVVRDHSKNNLWVAVTMAHELGHNLGIHHDTGSCSCGAKSCIMASVLSKVLSYEFSDCSQNQYETYLTNHNPQCILNKP 2w17 A 2.15 BS01 I19 A 1 I10 V18 A31 K33 V64 F80 L83 H84 Q85 D86 L134 D145 I10 V17 A30 K32 V58 F73 L76 H77 Q78 D79 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.002uM remove_due_to_license_issue IC50=2nM P24941 18996007 1300 MENFQKVEKIGETYGVVYKARNKLTGEVVALKKIRLDVPSTAIREISLLKELNHPNIVKLLDVIHTEKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2w1c A 3.24 BS01 L0C A 1 R137 V147 L194 Y212 A213 P214 G216 L263 K389 R11 V21 L68 Y86 A87 P88 G90 L137 K263 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 19143567 1391 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2w1d A 2.97 BS01 L0D A 1 A160 Y212 A213 G216 L263 K389 A34 Y86 A87 G90 L137 K251 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=910nM O14965 19143567 1391 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVGTLDYLPPEMIEGRMHDKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2w1e A 2.93 BS01 L0E A 1 L139 G140 V147 A160 Y212 A213 G216 T217 R220 L263 K389 L13 G14 V21 A34 Y86 A87 G90 T91 R94 L137 K252 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 19143567 1390 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2w1f A 2.85 BS01 L0F A 1 R137 K141 V147 Y212 A213 G216 L263 S387 K389 R11 K15 V21 Y86 A87 G90 L137 S251 K253 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=5.9nM O14965 19143567 1390 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2w1g A 2.71 BS01 L0G A 1 R137 L139 V147 L194 A213 P214 G216 L263 K389 R11 L13 V21 L68 A87 P88 G90 L137 K254 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 19143567 1390 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2w1h A 2.15 BS01 L0F A 1 I10 A31 E81 F82 L83 H84 Q85 L134 D145 I10 A31 E77 F78 L79 H80 Q81 L130 D141 D127 K129 Q131 N132 D145 T165 D123 K125 Q127 N128 D141 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.052uM remove_due_to_license_issue IC50=52nM P24941 19143567 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2w1i A 2.6 BS01 L0I A 1 L855 G856 V863 A880 E930 Y931 L932 G935 L983 L13 G14 V21 A38 E84 Y85 L86 G89 L137 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue O60674 19143567 2133 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG 2w26 A 2.08 BS01 RIV A 1 E97 T98 Y99 F174 A190 V213 W215 G216 E217 G219 G226 I227 Y228 E83 T84 Y85 F162 A180 V203 W205 G206 E207 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.4nM remove_due_to_license_issue IC50=700nM, Ki=0.400000nM P00742 16161994 1001 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2w2i A 2.1 BS01 PD2 A 1 Y133 F186 H189 E191 K207 W209 K242 H277 Y121 F174 H177 E179 K195 W197 K226 H261 G171 Y178 H189 E191 H277 A289 G159 Y166 H177 E179 H261 A273 1.14.11.66 remove_due_to_license_issue IC50=1400nM, Ki=914000nM B2RXH2 21914792 602 HTIMTFYPTMEEFADFNTYVAYMESQGAHQAGLAKVIPPKEWKARQMYDDIEDILIATPLQQVTSGQGGVFTQYHKKKKAMRVGQYRRLANSKKYQTPPHQNFADLEQRYWKSHPGNPPIYGADISGSLFEESTKQWNLGHLGTILDLLEQECGVVIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHFGEPKTWYVVPPEHGQHLERLARELFPDISAFLRHKVALISPTVLKENGIPFNCMTQEAGEFMVTFPYGYHAGFNHGFNCAEAINFATPRWIDYGKMAVTFSMDPFVRIVQPESY 2w3i A 1.9 BS02 L1C A 1 E97 T98 Y99 E147 F174 A190 Q192 V213 W215 G216 G219 G226 Y228 E83 T84 Y85 E135 F162 A180 Q182 V203 W205 G206 G208 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=0.1nM remove_due_to_license_issue IC50=0.1nM P00742 19231206 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2w3k A 2.05 BS01 L1D A 1 E97 T98 Y99 R143 E147 F174 A190 V213 W215 G216 G219 G226 Y228 E83 T84 Y85 R132 E135 F162 A180 V203 W205 G206 G208 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=0.08nM remove_due_to_license_issue IC50=0.08nM P00742 19231206 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2w3l A 2.1 BS01 DRO A 1 F63 Y67 D70 M74 V92 E95 L96 A108 F112 F39 Y43 D46 M50 V68 E71 L72 A84 F88 ? 0042981 remove_due_to_license_issue IC50=30nM P10415 19027294 1166 YDNREIVMKYIHYKLSQRGYEWDASEVVHKTLREAGDDFSRRYRRDFAEMSSGLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGPSM 2w42 A 1.9 BS01 dna P 0 Y118 Y123 Y124 K127 Q137 F138 M139 R140 I143 Y152 N155 L156 Q159 K163 N378 R380 R385 L427 Y108 Y113 Y114 K117 Q127 F128 M129 R130 I133 Y142 N145 L146 Q149 K153 N351 R353 R358 L395 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 19187762 1 ~ 6 LTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDILSNRNLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGYEGTKVKLSSKRYLLTLLQMVTPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPIRSLQTNPWFL 2w42 A 1.9 BS02 dna Q 0 T26 G27 I30 R147 N148 T150 F151 D154 R383 T16 G17 I20 R137 N138 T140 F141 D144 R356 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 19187762 9 ~ 14 LTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDILSNRNLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGYEGTKVKLSSKRYLLTLLQMVTPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPIRSLQTNPWFL 2w42 B 1.9 BS01 dna R 0 T120 Y123 K127 Q137 F138 M139 R140 I143 Y152 L156 Q159 K163 R380 L427 T110 Y113 K117 Q127 F128 M129 R130 I133 Y138 L142 Q145 K149 R348 L389 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 19187762 1 ~ 6 LTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDINLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGYEGTKVKLSSKRYLLTLLQVTPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPISLQTNPWFL 2w42 B 1.9 BS02 dna S 0 I30 T150 F151 D154 I20 T136 F137 D140 ? 0003676,0003677,0003723,0046872 remove_due_to_license_issue O28951 19187762 11 ~ 14 LTYRIGNGASVPISNTGELIKGLRNYGPYEVPSLKYNQIALIHNNQFSSLINQLKSQISSKIDEVWHIHNINISEFIYDSPHFDSIKSQVDNAIDTGVDGIMLVLPEYNTPLYYKLKSYLINSIPSQFMRYDINLTFYVDNLLVQFVSKLGGKPWILNVDPEKGSDIIIGTGATRIDNVNLFCFAMVFKKDGTMLWNEISPIVTSSEYLTYLKSTIKKVVYGFKKSNPDWDVEKLTLHVSGKRPKMKDGETKILKETVEELKKQEMVSRDVKYAILHLNETHPFWVMGYEGTKVKLSSKRYLLTLLQVTPIKPLSVEIVSDNWTSEEYYHNVHEILDEIYYLSKMNWRGFRSRNLPVTVNYPKLVAGIIANVNRYGGYPISLQTNPWFL 2w4i A 1.87 BS02 VGA B 1 P38 T41 S143 V146 P147 E150 E151 P38 T41 S143 V146 P147 E150 E151 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 remove_due_to_license_issue IC50=500nM Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLKL 2w4i B 1.87 BS02 VGA B 1 P38 T41 V146 P147 E150 E151 P38 T41 V146 P147 E150 E151 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 ic50=0.5uM remove_due_to_license_issue IC50=500nM Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK 2w4x A 2.42 BS01 STZ A 1 G135 D242 Y282 V314 W337 D344 Y345 G125 D232 Y272 V304 W327 D334 Y335 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Kd=14uM remove_due_to_license_issue Q89ZI2 19217614 1591 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTD 2w54 B 3.3 BS02 HHR B 1 E232 P306 R310 F344 F459 T460 L461 A529 E730 E231 P305 R309 F343 F442 T443 L444 A512 E713 Q197 E232 R310 H314 R342 G729 E730 Q196 E231 R309 H313 R341 G712 E713 1.1.1.204 0005506,0016491,0030151,0046872 remove_due_to_license_issue O54051 19109249 1780 SVGKPLPHDSARAHVTGQARYLDDLPCPANTLHLAFGLSTEASAAITGLDLEPVRESPGVIAVFTAADLPHDNDASPAPSPEPVLATGEVHFVGQPIFLVAATSHRAARIAARKARITYAPRPAILTLDQALAADSRFEGGPVIWARGDVETALAGAAHLAEGCFEIGGQEHFYLEGQAALALPAEGGVVIHCSSQHPSEIQHKVAHALGLAFHDVRVEMRRMGGGFGGKESQGNHLAIACAVAARATGRPCKMRYDRDDDMVITGKRHDFRIRYRIGADASGKLLGADFVHLARCGWSADLSLPVCDRAMLHADGSYFVPALRIESHRLRTNTQSNTAFRGFGGPQGALGMERAIEHLARGMGRDPAELRALNFYDPPEKKTQTTHYGQEVADCVLGELVTRLQKSANFTTRRAEIAAWNSTNRTLARGIALSPVKFGISFTLTHLNQAGALVQIYTDGSVALNHGGTEMGQGLHAKMVQVAAAVLGIDPVQVRITATDTSKVPNTSATAASSGADMNGMAVKDACETLRGRLAGFVAAREGCAARDVIFDAGQVQASGKSWRFAEIVAAAYMARISLSATGFYATPKLSWDRLRGQGRPFLYFAYGAAITEVVIDRLTGENRILRTDILHDAGASLNPALDIGQIEGAYVQGAGWLTTEELVWDHCGRLMTHAPSTYKIPAFSDRPRIFNVALWDQPNREETIFRSKAVGEPPFLLGISAFLALHDACAACGPHWPDLQAPATPEAVLAAVRRAEGRA 2w5g A 1.7 BS01 ATP A 1 Q11 H12 N67 Q69 N71 A109 H119 Q11 H12 N67 Q69 N71 A109 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=0.86uM remove_due_to_license_issue P61823 19191310 1125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 2w5i A 2.4 BS01 ATP A 1 H12 K41 C65 N67 Q69 N71 A109 E111 V118 H119 H11 K40 C64 N66 Q68 N70 A108 E110 V117 H118 H12 K41 H119 F120 D121 H11 K40 H118 F119 D120 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=0.86uM remove_due_to_license_issue P61823 19191310 1125 ETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 2w66 A 2.27 BS01 HQ6 A 1 G135 Y137 K166 D242 D243 Y282 V314 W337 N339 D344 N372 G132 Y134 K163 D239 D240 Y279 V311 W334 N336 D341 N369 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=89uM remove_due_to_license_issue Q89ZI2 19331390 1716 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMLPLQVKANRVLISPVEIELDAIYPGENIQINFRLSAGLQKAPVKFVRFFVLTIEK 2w67 A 2.25 BS01 F34 A 1 K166 D242 D243 Y282 V314 W337 N339 D344 K160 D236 D237 Y276 V308 W331 N333 D338 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=11uM remove_due_to_license_issue Q89ZI2 19331390 1716 LQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMNLPLQVKANRVLISPVEIELDAIYPGENIQINFGLQKAPVKFVRFQFVLTIEK 2w68 A 2.5 BS01 SIA D 1 R74 R118 Q188 G196 S198 R53 R97 Q167 G175 S177 3.2.1.18 0033691 remove_due_to_license_issue P0C6E9 19124471 3 AAMALFDYNATGDTEFDSPAKQGWMQDNTNNGSGVLTNADGMPAWLVQGIGGRAQWTYSLSTNQHAQASSFGWRMTTEMKVLSGGMITNYYANGTQRVLPIISLDSSGNLVVEFEGQTGRTVLATGTAATEYHKFELVFLPGSNPSASFYFDGKLIRDNIQPTASKQNMIVWGNGSSNTDGVAAYRDIKFEIQGD 2w6c X 2.69 BS01 BM4 X 1 W84 G118 Y121 S200 F330 Y334 H440 W81 G115 Y118 S197 F327 Y331 H437 G118 G119 S200 A201 H440 G115 G116 S197 A198 H437 3.1.1.7 0001507,0003990,0004104 remove_due_to_license_issue P04058 19326912 601 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 2w6m A 2.0 BS01 OA1 A 1 I157 K159 M169 E201 K202 Y203 H236 L278 I437 I157 K159 M169 E201 K202 Y203 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=21.5uM remove_due_to_license_issue IC50=21500nM P24182 19413326 1447 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w6n A 1.87 BS01 OA2 A 1 I157 K159 M169 E201 K202 Y203 L278 I157 K159 M169 E201 K202 Y203 L278 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=0.125uM remove_due_to_license_issue IC50=125nM P24182 19413326 1446 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLG 2w6o A 2.5 BS01 OA3 A 1 K159 K202 Y203 L204 L278 I437 K159 K202 Y203 L204 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=60.8uM remove_due_to_license_issue IC50=60800nM P24182 19413326 1446 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLG 2w6p A 1.85 BS01 OA4 A 1 K159 Y203 L204 Q233 H236 L278 I437 K159 Y203 L204 Q233 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=0.333uM remove_due_to_license_issue IC50=333nM P24182 19413326 1447 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w6q A 2.05 BS01 OA5 A 1 I157 K159 E201 K202 Y203 L204 H236 L278 I157 K159 E201 K202 Y203 L204 H236 L278 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=25.4uM remove_due_to_license_issue IC50=25400nM P24182 19413326 1447 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w6z A 1.9 BS01 L21 A 1 K159 Y203 L204 L278 K159 Y203 L204 L278 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=1500uM remove_due_to_license_issue IC50=1500000nM P24182 19413326 1447 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w70 A 1.77 BS01 L22 A 1 I157 K159 G166 M169 E201 Y203 L204 L278 I157 K159 G166 M169 E201 Y203 L204 L278 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=12uM remove_due_to_license_issue IC50=12000nM P24182 19413326 1447 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w71 A 1.99 BS01 L23 A 1 K159 Y203 L204 H209 Q233 H236 L278 I437 K159 Y203 L204 H209 Q233 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=0.334uM remove_due_to_license_issue IC50=334nM P24182 19413326 1448 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w7n A 1.85 BS01 dna E 0 E18 V19 G20 Q22 T47 A50 Q53 R57 E17 V18 G19 Q21 T46 A49 Q52 R56 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KKRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKK 2w7n A 1.85 BS02 dna F 0 Q37 A38 R48 S52 Q53 Q36 A37 R47 S51 Q52 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KKRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKK 2w7n A 1.85 BS03 dna G 0 Q37 A38 R48 S52 Q53 Q36 A37 R47 S51 Q52 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KKRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKK 2w7n A 1.85 BS04 dna H 0 E18 G20 Q22 T23 L46 T47 A50 Q53 R57 E17 G19 Q21 T22 L45 T46 A49 Q52 R56 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KKRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKK 2w7n B 1.85 BS01 dna E 0 P36 Q37 A38 R48 G49 S52 Q53 P34 Q35 A36 R46 G47 S50 Q51 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKKKQ 2w7n B 1.85 BS02 dna F 0 E18 V19 G20 T23 T47 A50 Q53 R57 E16 V17 G18 T21 T45 A48 Q51 R55 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKKKQ 2w7n B 1.85 BS03 dna G 0 E18 G20 T47 A50 Q53 R57 E16 G18 T45 A48 Q51 R55 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKKKQ 2w7n B 1.85 BS04 dna H 0 Q37 A38 R48 S52 Q53 Q35 A36 R46 S50 Q51 ? 0003677,0005515 remove_due_to_license_issue P03052 19190096 1 ~ 18 KRLTESQFQEAIQGLEVGQQTIEIARGVLVDGKPQATFATSLGLTRGAVSQAVHRVWAAFEDKNLPEGYARVTAVLPEHQAYIVRKWEADAKKKQ 2w7x A 2.07 BS01 D1A A 1 L226 K249 I251 E273 L301 M304 E305 G307 L354 T367 D368 L17 K39 I41 E48 L76 M79 E80 G82 L129 T142 D143 D347 K349 N352 D368 T387 D122 K124 N127 D143 T162 2.7.11.1 0004672,0005524,0006468 ic50=24nM remove_due_to_license_issue O96017 19741151 601 SVYPKALRDEYIMSKTLGSGAGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2w7y A 2.35 BS01 GAL C 1 Y46 A104 Q153 F155 W280 Y9 A67 Q116 F118 W243 remove_due_to_license_issue 19285508 1 EVLEFYHGYHHSEDEWPVAKTMRDLYDKFAEEHSGVEFKPTPVNGDLKDIMNNKVASGEFPDVIDLAGNAVSLAAIEQKLVLDLKPYIDSNKLEKNVGLNYKQNQKDGKIYTVHEQLFTMGLWYNKDIFAKAGAKTPDQWNTWDDFTQAMASIRKQDGVYAFGAGEPSIRLFNTVLGTTENGRKLLDKPLTKEGIESKEFADALKMVMKEIQANGSKNAGGDANAYSKDFQEGKSAVFFNGVWASGEMSKNPSLAPGIYPAGVAISSSGGGITISSKMSEAKQKLALEFLKYMTSDDVQKVIFEKVGANPSNENVNVKELSEKSSEATTKILGQAITQVKNAKAVVPTVSDVWGGDVHTAIINALTESAAENVDVDQKVKSTQDVLKSL 2w7y A 2.35 BS02 FUC C 1 G45 Y46 H48 A104 G8 Y9 H11 A67 remove_due_to_license_issue 19285508 2 EVLEFYHGYHHSEDEWPVAKTMRDLYDKFAEEHSGVEFKPTPVNGDLKDIMNNKVASGEFPDVIDLAGNAVSLAAIEQKLVLDLKPYIDSNKLEKNVGLNYKQNQKDGKIYTVHEQLFTMGLWYNKDIFAKAGAKTPDQWNTWDDFTQAMASIRKQDGVYAFGAGEPSIRLFNTVLGTTENGRKLLDKPLTKEGIESKEFADALKMVMKEIQANGSKNAGGDANAYSKDFQEGKSAVFFNGVWASGEMSKNPSLAPGIYPAGVAISSSGGGITISSKMSEAKQKLALEFLKYMTSDDVQKVIFEKVGANPSNENVNVKELSEKSSEATTKILGQAITQVKNAKAVVPTVSDVWGGDVHTAIINALTESAAENVDVDQKVKSTQDVLKSL 2w87 A 1.6 BS03 GCU A 1 H30 N40 N43 R75 W99 N130 H22 N32 N35 R67 W91 N122 3.2.1.- 0030246 remove_due_to_license_issue Q51815 19218457 1150 ALLLQEAQAGFCRVDGTIDNNHTGFTGSGFANTNNAQGAAVVWAIDATSSGRRTLTIRYANGGTANRNGSLVINGGSNGNYTVSLPTTGAWTTWQTATIDVDLVQGNNIVQLSATTAEGLPNIDSLSVVGGTVRAGNCG 2w8f A 2.7 BS01 BS1 A 1 Y91 W145 Y193 Y91 W145 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 19331415 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2w8f B 2.7 BS01 BS1 A 1 Q55 M114 I116 Q55 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 19331415 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2w8g A 2.6 BS01 BS2 A 1 Y91 W145 Y186 C188 C189 Y193 Y91 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 19331415 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2w8g A 2.6 BS02 BS2 E 1 Y53 M114 I116 Y53 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 19331415 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2w8g B 2.6 BS01 BS2 A 1 M114 I116 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 19331415 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2w8j A 1.5 BS01 PLS A 1 G134 Y135 H159 D231 A233 H234 T262 S264 K265 R378 I419 G113 Y114 H138 D210 A212 H213 T241 S243 K244 R357 I398 Y73 H159 E202 S206 D231 H234 K265 Y52 H138 E181 S185 D210 H213 K244 2.3.1.50 0005737,0006629,0006665,0009058,0016020,0016740,0016746,0030170 remove_due_to_license_issue Q93UV0 19376777 1420 RDLLSKFDGLIAERQKLLDSGVTDPFAIVMEQVKSPTEAVIRGKDTILLGTYNYMGMTFDPDVIAAGKEALEKFGSGTNGSRMLNGTFHDHMEVEQALRDFYGTTGAIVFSTGYMANLGIISTLAGKGEYVILDADSHASIYDGCQQGNAEIVRFRHNSVEDLDKRLGRLPKEPAKLVVLEGVYSMLGDIAPLKEMVAVAKKHGAMVLVDEAHSMGFFGPNGRGVYEAQGLEGQIDFVVGTFSKSVGTVGGFVVSNHPKFEAVRLACRPYIFTASLPPSVVATATTSIRKLMTAHEKRERLWSNARALHGGLKAMGFRLGTETCDSAIVAVMLEDQEQAAMMWQALLDGGLYVNMARPPATPAGTFLLRCSICAEHTPAQIQTVLGMFQAAGRAVGVI 2w8k A 3.1 BS01 dna P 0 D105 E106 P184 G185 I186 G187 I189 T190 V296 S297 R298 G299 T301 I341 D106 E107 P185 G186 I187 G188 I190 T191 V297 S298 R299 G300 T302 I342 2.7.7.7 0000287,0003677,0003684,0003887,0005737,0006260,0006261,0006281,0006974,0034061,0042276,0046872 remove_due_to_license_issue Q97W02 19059910 1 ~ 14 HMIVLFVDFDYFYAQVEEVLNPSLKGKPVVVCVFSGRFEDSGAVATANYEARKFGVKAGIPIVEAKKILPNAVYLPMRKEVYQQVSSRIMNLLREYSEKIEIASIDEAYLDISDKVRDYREAYNLGLEIKNKILEKEKITVTVGISKNKVFAKIAADMAKPNGIKVIDDEEVKRLIRELDIADVPGIGNITAEKLKKLGINKLVDTLSIEFDKLKGMIGEAKAKYLISLARDEYNEPIRTRVRKSIGRIVTMKRNSRNLEEIKPYLFRAIEESYYKLDKRIPKAIHVVAVTEDLDIVSRGRTFPHGISKETAYSESVKLLQKILEEDERKIRRIGVRFSKFI 2w8k A 3.1 BS02 dna T 0 V32 G41 G58 G218 A220 R242 K243 S244 I245 G246 R247 I248 T250 R331 R332 R336 V33 G42 G59 G219 A221 R243 K244 S245 I246 G247 R248 I249 T251 R332 R333 R337 2.7.7.7 0000287,0003677,0003684,0003887,0005737,0006260,0006261,0006281,0006974,0034061,0042276,0046872 remove_due_to_license_issue Q97W02 19059910 3 ~ 18 HMIVLFVDFDYFYAQVEEVLNPSLKGKPVVVCVFSGRFEDSGAVATANYEARKFGVKAGIPIVEAKKILPNAVYLPMRKEVYQQVSSRIMNLLREYSEKIEIASIDEAYLDISDKVRDYREAYNLGLEIKNKILEKEKITVTVGISKNKVFAKIAADMAKPNGIKVIDDEEVKRLIRELDIADVPGIGNITAEKLKKLGINKLVDTLSIEFDKLKGMIGEAKAKYLISLARDEYNEPIRTRVRKSIGRIVTMKRNSRNLEEIKPYLFRAIEESYYKLDKRIPKAIHVVAVTEDLDIVSRGRTFPHGISKETAYSESVKLLQKILEEDERKIRRIGVRFSKFI 2w8l A 3.0 BS01 dna P 0 S103 E106 K152 P184 G185 G187 I189 T190 R240 V296 S297 R298 T301 I341 S104 E107 K153 P185 G186 G188 I190 T191 R241 V297 S298 R299 T302 I342 2.7.7.7 0000287,0003677,0003684,0003887,0005737,0006260,0006261,0006281,0006974,0034061,0042276,0046872 remove_due_to_license_issue Q97W02 19059910 1 ~ 14 HMIVLFVDFDYFYAQVEEVLNPSLKGKPVVVCVFSGRFEDSGAVATANYEARKFGVKAGIPIVEAKKILPNAVYLPMRKEVYQQVSSRIMNLLREYSEKIEIASIDEAYLDISDKVRDYREAYNLGLEIKNKILEKEKITVTVGISKNKVFAKIAADMAKPNGIKVIDDEEVKRLIRELDIADVPGIGNITAEKLKKLGINKLVDTLSIEFDKLKGMIGEAKAKYLISLARDEYNEPIRTRVRKSIGRIVTMKRNSRNLEEIKPYLFRAIEESYYKLDKRIPKAIHVVAVTEDLDIVSRGRTFPHGISKETAYSESVKLLQKILEEDERKIRRIGVRFSKFI 2w8l A 3.0 BS02 dna T 0 V32 S34 G41 A42 E219 A220 R242 K243 S244 I245 R247 I248 T250 R331 R332 R336 V33 S35 G42 A43 E220 A221 R243 K244 S245 I246 R248 I249 T251 R332 R333 R337 2.7.7.7 0000287,0003677,0003684,0003887,0005737,0006260,0006261,0006281,0006974,0034061,0042276,0046872 remove_due_to_license_issue Q97W02 19059910 3 ~ 18 HMIVLFVDFDYFYAQVEEVLNPSLKGKPVVVCVFSGRFEDSGAVATANYEARKFGVKAGIPIVEAKKILPNAVYLPMRKEVYQQVSSRIMNLLREYSEKIEIASIDEAYLDISDKVRDYREAYNLGLEIKNKILEKEKITVTVGISKNKVFAKIAADMAKPNGIKVIDDEEVKRLIRELDIADVPGIGNITAEKLKKLGINKLVDTLSIEFDKLKGMIGEAKAKYLISLARDEYNEPIRTRVRKSIGRIVTMKRNSRNLEEIKPYLFRAIEESYYKLDKRIPKAIHVVAVTEDLDIVSRGRTFPHGISKETAYSESVKLLQKILEEDERKIRRIGVRFSKFI 2w8w A 2.14 BS01 PLS A 1 G134 Y135 H159 D231 H234 T262 S264 K265 I419 G112 Y113 H137 D209 H212 T240 S242 K243 I397 Y73 H159 E202 S206 D231 H234 K265 Y51 H137 E180 S184 D209 H212 K243 2.3.1.50 0005737,0006629,0006665,0009058,0016020,0016740,0016746,0030170 remove_due_to_license_issue Q93UV0 19376777 1420 DLLSKFDGLIAERQKLLDSGVTDPFAIVMEQVKSPTEAVIRGKDTILLGTYNYMGMTFDPDVIAAGKEALEKFGSGTYGSRMLNGTFHDHMEVEQALRDFYGTTGAIVFSTGYMANLGIISTLAGKGEYVILDADSHASIYDGCQQGNAEIVRFRHNSVEDLDKRLGRLPKEPAKLVVLEGVYSMLGDIAPLKEMVAVAKKHGAMVLVDEAHSMGFFGPNGRGVYEAQGLEGQIDFVVGTFSKSVGTVGGFVVSNHPKFEAVRLACRPYIFTASLPPSVVATATTSIRKLMTAHEKRERLWSNARALHGGLKAMGFRLGTETCDSAIVAVMLEDQEQAAMMWQALLDGGLYVNMARPPATPAGTFLLRCSICAEHTPAQIQTVLGMFQAAGRAVGVI 2w8y A 1.8 BS01 486 A 1 L715 L718 N719 L721 G722 E723 Q725 W755 M756 M759 F794 L797 Y890 C891 M909 L33 L36 N37 L39 G40 E41 Q43 W73 M74 M77 F112 L115 Y208 C209 M227 ? remove_due_to_license_issue IC50=0.300000nM, Ki=1.1nM, EC50=>10000nM P06401 19372222 1000 LIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 2w92 A 1.65 BS01 NGT A 1 W264 F333 N335 Y373 F412 E441 F471 W92 F161 N163 Y201 F240 E269 F299 ? 0005737,0033925 Kd=28uM remove_due_to_license_issue Q93HW0 19181667 1809 TLKPKEIKFNSWEELLKWEPGAREDDAINRGSVVLASRRTGHLVNEKASKEAKVQALSNTNSKAKDHASVGGEEFKAYAFDYWQYLDSMVFWEGLVPTPDVIDAGHRNGVPVYGTLFFNWSNSIADQERFAEALKQDADGSFPIARKLVDMAKYYGYDGYFINQETTGDLVKPLGEKMRQFMLYSKEYAAKVNHPIKYSWYDAMTYNYGRYHQDGLGEYNYQFMQPEGDKVPADNFFANFNWDKAKNDYTIATANWIGRNPYDVFAGLELQQGGSYKTKVKWNDILDENGKLRLSLGLFAPDTITSLGKTGEDYHKNEDIFFTGYQGDPTGQKPGDKDWYGIANLVADRTPAVGNTFTTSFNTGHGKKWFVDGKVSKDSEWNYRSVSGVLPTWRWWQTSTGEKLRAEYDFTDAYNGGNSLKFSGDVAGKTDQDVRLYSTKLEVTEKTKLRVAHKGGKGSKVYMAFSTTPDYKFDDADAWKELTLSDNWTNEEFDLSSLAGKTIYAVKLFFEHEGAVKDYQFNLGQLTISDNHQEPQSPTSFSVVKQSLKNAQEAEAVVQFKGNKDADFYEVYEKDGDSWKLLTGSSSTTIYLPKVSRSASAQGTTQELKVVAVGKNGVRSEAATTTFDWGMTVKD 2w9h A 1.48 BS01 TOP A 1 L5 V6 A7 L20 D27 V31 S49 F92 L5 V6 A7 L20 D27 V31 S49 F92 L5 L20 W22 D27 L28 V31 L54 V89 T111 L5 L20 W22 D27 L28 V31 L54 V89 T111 1.5.1.3 0004146,0005829,0006730,0016491,0046452,0046654,0046655,0050661 Kd=430nM remove_due_to_license_issue Ki=3.4nM, IC50=14.4nM P0A017 19280600 1160 TLSILVAHDLQRVIGFENQLPWHLPNDLKHVKKLSTGHTLVMGRKTFESIGKPLPNRRNVVLTSDTSFNVEGVDVIHSIEDIYQLPGHVFIFGGQTLFEEMIDKVDDMYITVIEGKFRGDTFFPPYTFEDWEVASSVEGKLDEKNTIPHTFLHLIRK 2wa3 A 2.5 BS02 A29 A 1 Y145 L188 T196 H199 D201 N205 F207 H279 I281 N294 W296 Y131 L174 T182 H185 D187 N191 F193 H265 I267 N280 W282 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=1mM remove_due_to_license_issue Q9NWT6 20822901 400 EPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2wa4 A 2.5 BS02 069 A 1 Y145 T196 H199 F207 H279 I281 N294 Y131 T182 H185 F193 H265 I267 N280 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=18uM remove_due_to_license_issue Q9NWT6 20822901 400 EPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2wa4 A 2.5 BS03 069 A 2 H199 D201 H279 H185 D187 H265 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=18uM remove_due_to_license_issue Q9NWT6 20822901 401 EPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2waj A 2.4 BS01 SNB A 1 A91 K93 I124 L144 M146 M149 L206 A44 K46 I77 L97 M99 M102 L159 D189 K191 N194 D207 T226 D142 K144 N147 D160 T176 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.398uM remove_due_to_license_issue IC50=398.11nM P53779 19303774 1401 NQFYSVEVGDSTFTVLKRYQNLKPIGSGGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTSFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQDKQLDEREHTIEEWKELIYKEVMN 2wap A 2.8 BS01 PIX A 1 F192 S193 I238 G239 S241 Y335 L372 F381 F432 T488 V491 M495 W531 F160 S161 I206 G207 S209 Y303 L340 F349 F400 T456 V459 M463 W499 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 19389627 1574 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMT 2wb5 A 2.31 BS01 VGB A 1 G187 K218 D297 D298 Y335 V370 W394 D401 Y402 G148 K179 D258 D259 Y296 V331 W355 D362 Y363 3.2.1.169 remove_due_to_license_issue Q0TR53 19275764 1628 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYDRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVALNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2wbb A 2.22 BS01 RO3 A 1 M18 G21 R22 G26 G28 L30 T31 M10 G13 R14 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.92uM remove_due_to_license_issue P09467 19969452 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2wbb C 2.22 BS01 RO3 C 1 M18 G21 R22 A24 G26 G28 L30 T31 M10 G13 R14 A16 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.92uM remove_due_to_license_issue P09467 19969452 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2wbd A 2.4 BS01 RO5 A 1 V17 M18 G21 R22 G26 G28 L30 T31 V9 M10 G13 R14 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.23uM remove_due_to_license_issue IC50=100nM P09467 19969452 1337 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2wbd C 2.4 BS01 RO5 C 1 V17 M18 G21 R22 G26 G28 L30 T31 M177 V9 M10 G13 R14 G18 G20 L22 T23 M159 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.23uM remove_due_to_license_issue IC50=100nM P09467 19969452 1337 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2wbg A 1.85 BS01 LGS A 1 Q20 H121 N165 E166 Y295 H298 W324 E351 W398 E405 W406 Q18 H119 N163 E164 Y293 H296 W322 E349 W396 E403 W404 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E349 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Ki=35.2uM remove_due_to_license_issue Q08638 19532990 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2wc3 A 2.0 BS01 AM3 A 1 Q20 H121 N165 E166 Y295 H298 W324 E351 W398 E405 W406 F414 Q19 H120 N164 E165 Y294 H297 W321 E348 W395 E402 W403 F411 R77 H121 E166 V169 N293 Y295 E351 R76 H120 E165 V168 N292 Y294 E348 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Ki=0.83uM remove_due_to_license_issue Q08638 19532990 1446 NVKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2wc4 A 1.7 BS01 AMF A 1 Q20 H121 N165 E166 Y295 W324 E351 W398 E405 W406 F414 Q18 H119 N163 E164 Y293 W322 E349 W396 E403 W404 F412 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E349 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=5.1uM remove_due_to_license_issue Q08638 19532990 1446 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 2wca A 2.3 BS01 NP6 A 1 G135 Y282 W286 T310 V314 W337 N339 D344 Y345 H433 G124 Y271 W275 T299 V303 W326 N328 D333 Y334 H422 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 19499593 900 LQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTD 2wcg A 2.3 BS01 MT5 A 1 D127 F128 N234 E235 Y313 E340 W381 D122 F123 N229 E230 Y308 E335 W376 E235 E340 C342 N370 E230 E335 C337 N365 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 Ki=0.42uM remove_due_to_license_issue P04062 19437524 1509 ARPCIPKSFGYSSVVCVCNATYCDSFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQL 2wcx A 2.0 BS03 VGC A 1 V37 L392 A393 A395 A396 H428 L492 V494 P495 R503 V23 L373 A374 A376 A377 H409 L473 V475 P476 R484 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.025uM remove_due_to_license_issue P26663 19672916 1534 SMSYTWTGALITPCAAEESKLMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVK 2wd1 A 2.0 BS01 ZZY A 1 I1084 V1092 A1108 L1157 Y1159 M1160 M1211 A1221 D1222 Y1230 I30 V38 A54 L100 Y102 M103 M154 A164 D165 Y173 D1204 A1206 R1208 N1209 D1222 A1243 D147 A149 R151 N152 D165 A186 2.7.10.1 0004672,0004713,0005524,0006468 ic50=82nM remove_due_to_license_issue IC50=82nM P08581 19369077 2347 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 2wd3 A 1.8 BS01 MS4 A 1 L60 N67 E69 Q92 H94 H119 F130 L197 T198 W208 L57 N64 E66 Q89 H91 H116 F127 L194 T195 W205 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=86nM remove_due_to_license_issue IC50=86nM P00918 20148564 1261 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2wd3 A 1.8 BS02 MS4 A 2 D72 I91 Q92 W123 D129 F130 G131 D69 I88 Q89 W120 D126 F127 G128 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=86nM remove_due_to_license_issue IC50=86nM P00918 20148564 1262 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2wd7 A 1.9 BS02 VGD A 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0000166,0016491,0047040 Ki=10.6uM remove_due_to_license_issue Ki=10600nM O76290 19527033 1269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 2we3 A 2.0 BS01 DUT A 1 G73 I75 D76 Y79 R84 R171 S172 G173 G70 I72 D73 Y76 R81 R155 S156 G157 3.6.1.23 0004170,0009117,0016787,0046080,0046872 remove_due_to_license_issue P03195 19586911 1257 MEACPHIRYAFQNDKLLLQQGRLTLVNKTTILLRPMKTTTVDLGLYARPPEGHGLMLWGSTSRPVTSHVGIIDPGYTGELRLILQNQRRYNSTLRPSELKIHLAAFRYATPQPGDVGLDVSLPKDLALFPHQTVSVTLTVPPPSIPHHRPTIFGRSGLAMQGILVKPCRWRRGGVDVSLTNFSDQTVFLNKYRRFCQLVYLHKHHLTSFYSPHSDAGVLGPRSLFRWASCTFEEVPSLAM 2web A 1.5 BS01 PP4 A 1 D33 G35 Y75 G76 D77 F112 D115 D213 G215 T216 D33 G35 Y75 G76 D77 F112 D115 D213 G215 T216 D33 S36 D38 W40 Y75 D213 T216 D33 S36 D38 W40 Y75 D213 T216 3.4.23.20 0004190,0005576,0006508 Ki=7.6uM remove_due_to_license_issue P00798 326 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 2wec A 1.5 BS01 PP5 A 1 G76 D77 T216 T217 L218 G76 D77 T216 T217 L218 D33 S36 D38 W40 Y75 D213 T216 D33 S36 D38 W40 Y75 D213 T216 3.4.23.20 0004190,0005576,0006508 Ki=110uM remove_due_to_license_issue P00798 326 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 2wed A 1.5 BS01 PP6 A 1 D33 G35 Y75 G76 D77 D213 G215 T216 I297 D33 G35 Y75 G76 D77 D213 G215 T216 I297 D33 S36 D38 W40 Y75 D213 T216 D33 S36 D38 W40 Y75 D213 T216 3.4.23.20 0004190,0005576,0006508 Ki=0.8uM remove_due_to_license_issue P00798 327 AASGVATNTPTANDEEYITPVTIGGTTLNLNFDTGSADLWVFSTELPASQQSGHSVYNPSATGKELSGYTWSISYGDGSSASGNVFTDSVTVGGVTAHGQAVQAAQQISAQFQQDTNNDGLLGLAFSSINTVQPQSQTTFFDTVKSSLAQPLFAVALKHQQPGVYDFGFIDSSKYTGSLTYTGVDNSQGFWSFNVDSYTAGSQSGDGFSGIADTGTTLLLLDDSVVSQYYSQVSGAQQDSNAGGYVFDCSTNLPDFSVSISGYTATVPGSLINYGPSGDGSTCLGGIQSNSGIGFSIFGDIFLKSQYVVFDSDGPQLGFAPQA 2weg A 1.1 BS02 FBV A 1 H94 H119 L198 T199 T200 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=314nM remove_due_to_license_issue P00918 19882701 1263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2weh A 2.09 BS02 FB1 A 1 H94 H96 H119 L198 T199 T200 H92 H94 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1125nM remove_due_to_license_issue P00918 19882701 1263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2wei A 1.65 BS01 VGG A 1 L82 A103 K105 M136 I150 Y155 L205 I218 L22 A43 K45 M76 I90 Y95 L145 I158 D198 K200 E202 N203 D219 T238 D138 K140 E142 N143 D159 T178 2.7.1.17 0004672,0005524,0006468 ic50=3.4nM remove_due_to_license_issue A3FQ16 21962082 600 SGRENLYFQGTFAERYNIVCMLGKGSFGEVLKCKDRITQQEYAVKVINKASAKNKDTSTILREVELLKKLDHPNIMKLFEILEDSSSFYIVGELYTGGELFDEIIKRKRFSEHDAARIIKQVFSGITYMHKHNIVHRDLKPENILLESKEKDCDIKIIDFGLSTCFQQNTKMKDRIGTAYYIAPEVLRGTYDEKCDVWSAGVILYILLSGTPPFYGKNEYDILKRVETGKYAFDLPQWRTISDDAKDLIRKMLTFHPSLRITATQCLEHPWIQKYSSE 2wej A 1.45 BS02 FB2 A 1 H94 H119 L198 T199 T200 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=839nM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 19882701 1263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2weo A 1.4 BS02 FBW A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=118nM remove_due_to_license_issue P00918 19882701 1263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2weq A 2.2 BS01 GDM A 1 N37 D40 A41 K44 E88 N92 L93 K98 G121 V122 F124 N36 D39 A40 K43 E87 N91 L92 K97 G120 V121 F123 ? 0005524,0006457,0016887,0051082,0140662 Kd=1.27uM remove_due_to_license_issue P02829 19236053 1215 ASETFEFQAEITQLMSLIINTVYSNKEIFLREIVSNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2wer A 1.6 BS01 RDC A 1 N37 D40 A41 K44 D79 M84 F124 L173 N37 D40 A41 K44 D79 M84 F124 L173 ? 0005524,0006457,0016887,0051082,0140662 Kd=90nM remove_due_to_license_issue IC50=2e+2nM P02829 19236053 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLREIVSNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2wev A 2.3 BS01 CK7 A 1 I10 A31 F80 L83 H84 L134 D145 I10 A31 F80 L83 H84 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=10.0nM, Ki=2nM P24941 19472269 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 2wey A 2.8 BS01 EV1 A 1 Y524 H525 L635 I692 F696 G725 F729 Y78 H79 L189 I246 F250 G279 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=36nM Q9Y233 19622871 1771 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 2wez A 1.7 BS01 ZYE A 1 Q73 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 D289 G291 T292 T293 N294 N446 Q12 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 D215 G217 T218 T219 N220 N372 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D215 T218 3.4.23.46 0004190,0006508,0016020 ic50=0.023uM remove_due_to_license_issue P56817 19428244 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2wf0 A 1.6 BS01 ZY0 A 1 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 D289 G291 T292 T293 N294 N446 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 D215 G217 T218 T219 N220 N372 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D215 T218 3.4.23.46 0004190,0006508,0016020 ic50=0.21uM remove_due_to_license_issue IC50=210nM P56817 19428244 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2wf1 A 1.6 BS01 ZY1 A 1 G72 Q73 D93 G95 Y132 T133 Q134 F169 W176 D289 G291 T292 T293 N294 R296 N446 G11 Q12 D32 G34 Y71 T72 Q73 F108 W115 D217 G219 T220 T221 N222 R224 N374 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=0.002uM remove_due_to_license_issue IC50=2nM P56817 19477642 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2wf2 A 1.8 BS01 ZY2 A 1 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 I179 D289 G291 T292 T293 N294 N446 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 I118 D217 G219 T220 T221 N222 N374 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=0.026uM remove_due_to_license_issue P56817 19477642 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2wf3 A 2.08 BS01 ZY3 A 1 G72 Q73 L91 D93 G95 Y132 T133 Q134 F169 D289 G291 T292 T293 N294 R296 N446 G11 Q12 L30 D32 G34 Y71 T72 Q73 F108 D217 G219 T220 T221 N222 R224 N374 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=0.019uM remove_due_to_license_issue P56817 19477642 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2wf4 A 1.8 BS01 ZY4 A 1 G72 Q73 L91 D93 G95 Y132 T133 Q134 F169 Y259 I287 D289 G291 T292 T293 N294 N446 G11 Q12 L30 D32 G34 Y71 T72 Q73 F108 Y185 I213 D215 G217 T218 T219 N220 N372 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D215 T218 3.4.23.46 0004190,0006508,0016020 ic50=13nM remove_due_to_license_issue P56817 19406640 2000 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2wf5 A 1.3 BS01 BG6 A 1 D10 H20 G46 V47 R49 A115 S116 D10 H20 G46 V47 R49 A115 S116 D8 L9 D10 T16 K45 S114 A115 K145 E169 D170 D8 L9 D10 T16 K45 S114 A115 K145 E169 D170 5.4.2.6 0000287,0003824,0005737,0005975,0008801,0016853,0046872 remove_due_to_license_issue P71447 20164409 1831 MFKAVLFDLDGVITDTAEYHFRAWKALAEEIGINGVDRQFNEQLKGVSREDSLQKILDLADKKVSAEEFKELAKRKNDNYVKMIQDVSPADVYPGILQLLKDLRSNKIKIALASASKNGPFLLERMNLTGYFDAIADPAEVAASKPAPDIFIAAAHAVGVAPSESIGLEDSQAGIQAIKDSGALPIGVGRPEDLGDDIVIVPDTSHYTLEFLKEVWLQ 2wfg A 2.2 BS01 ZZB A 1 A315 T316 L317 R318 T321 L404 K407 V412 D418 S419 K483 Y487 A37 T38 L39 R40 T43 L126 K129 V134 D140 S141 K205 Y209 0000166,0002161,0004823,0005524,0006418,0006429 ic50=38uM remove_due_to_license_issue 19426743 1529 GYVGIKIRLTDVAPQAQELFKKESLDVKENKVYLVAATLRPETMYGQTCCFVSPKIDYGVFDAGNGDYFITTERAFKNMSFQNLTPKRGYYKPLFTINGKTLIGSRIDAPYAVNKNLRVLPMETVLATKGTGVVTCVPSDSPDDFVTTRDLANKPEYYGIEKDWVQTDIVPIVHTEKYGDKCAEFLVNDLKIQSPKDSVQLANAKELAYKEGFYNGTMLIGKYKGDKVEDAKPKVKQDLIDEGLAFVYNE 2wgi A 2.85 BS01 PNM A 1 S67 S115 L155 T206 F208 R250 S47 S95 L125 T176 F178 R220 S67 K70 S115 F120 A154 F208 S47 K50 S95 F100 A124 F178 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0042597,0046677,0071555 remove_due_to_license_issue P14489 19860471 700 SITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNDLARASKEYLPASTFKIPNAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLTLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNALEGQLRISAVNQVEFLESLYLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKETEVYFFAFNMDIDNESKLPLRKSIPTKIMESEGII 2wgj A 2.0 BS01 VGH A 1 V1092 A1108 Y1159 M1160 G1163 M1211 A1221 D1222 Y1230 F1344 V41 A53 Y104 M105 G108 M156 A166 D167 Y175 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.002uM remove_due_to_license_issue IC50=8nM, Kd=2.0nM, Ki=2nM P08581 21812414 2346 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 2wgs A 2.55 BS01 1AZ A 1 Y129 G131 E133 N229 F232 H278 S280 W282 K361 R364 Y122 G124 E126 N222 F225 H271 S273 W275 K354 R357 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E126 E128 E212 E220 H269 R340 E359 R361 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 remove_due_to_license_issue P9WN39 19695264 501 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 2who A 2.0 BS03 VGI A 1 R422 M423 R501 W528 R422 M423 R501 W528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.02uM remove_due_to_license_issue IC50=20nM, EC50=7100nM P26663 19877603 1534 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVK 2whp A 2.2 BS01 HI6 A 1 Y124 X203 E285 W286 F297 S298 Y337 Y341 Y124 X203 E278 W279 F290 S291 Y330 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd~100uM remove_due_to_license_issue P21836 19536291 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 2wi1 A 2.3 BS02 ZZ2 A 1 N51 M98 N36 M83 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50>4000uM remove_due_to_license_issue P07900 19610616 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wi2 A 2.09 BS01 ZZ3 A 1 A55 M98 T184 A40 M83 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=350uM remove_due_to_license_issue P07900 19610616 1226 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wi3 A 1.9 BS02 ZZ3 A 1 N51 D93 M98 L107 N36 D78 M83 L92 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=350uM remove_due_to_license_issue P07900 19610616 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wi4 A 2.4 BS01 ZZ4 A 1 N51 A55 D93 M98 D102 L107 F138 T184 E223 N36 A40 D78 M83 D87 L92 F123 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=1.56uM remove_due_to_license_issue P07900 19610616 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wi5 A 2.1 BS01 ZZ5 A 1 N51 I96 G97 M98 L107 T109 G135 V136 F138 Y139 T184 E223 N36 I81 G82 M83 L92 T94 G120 V121 F123 Y124 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.9uM remove_due_to_license_issue P07900 19610616 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wi6 A 2.18 BS01 ZZ6 A 1 A55 I96 G97 M98 D102 N106 L107 F138 Y139 E223 A40 I81 G82 M83 D87 N91 L92 F123 Y124 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.23uM remove_due_to_license_issue P07900 19610616 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wi7 A 2.5 BS01 2KL A 1 N51 A55 I96 G97 M98 D102 G135 F138 E223 N36 A40 I81 G82 M83 D87 G120 F123 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.058uM remove_due_to_license_issue P07900 19610616 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2wib A 2.56 BS01 GDP A 1 N13 G15 K16 T17 T18 N120 M121 D123 I124 V149 T151 N13 G15 K16 T17 T18 N120 M121 D123 I124 V149 T151 ? 0005525 remove_due_to_license_issue A6TF32 20123128 1262 MQKLTVGLIGNPNSGKTTLFNQLTGARQRVGNWAGVTVERKEGIFATTDHQVTLVDLPGTYSLTTISSQTSLDEQIACHYILSGDADMLINVVDASNLERNLYLTLQLLELGIPCVVALNMLDIAEKQQVRIDIDALAARLGCPVIPLVSTRGRGIEALKIALDRHQANSDLELVHYPQPLLREADLLAQQMSAQIPPRQRRWLGLQMLEGDIYSRAYAGDAADKLDIALANLSDEIDDPALHIADARYQTIAAICDAVSN 2wib A 2.56 BS02 GDP B 1 D123 T151 D123 T151 ? 0005525 remove_due_to_license_issue A6TF32 20123128 1263 MQKLTVGLIGNPNSGKTTLFNQLTGARQRVGNWAGVTVERKEGIFATTDHQVTLVDLPGTYSLTTISSQTSLDEQIACHYILSGDADMLINVVDASNLERNLYLTLQLLELGIPCVVALNMLDIAEKQQVRIDIDALAARLGCPVIPLVSTRGRGIEALKIALDRHQANSDLELVHYPQPLLREADLLAQQMSAQIPPRQRRWLGLQMLEGDIYSRAYAGDAADKLDIALANLSDEIDDPALHIADARYQTIAAICDAVSN 2wic A 2.05 BS01 GNP A 1 N13 S14 G15 K16 T17 T18 N120 M121 D123 V149 T151 N13 S14 G15 K16 T17 T18 N104 M105 D107 V133 T135 ? 0005525 remove_due_to_license_issue A6TF32 20123128 1265 MQKLTVGLIGNPNSGKTTLFNQLTGARQKEGIFATTDHQVTLVDLPGTYSLTTISSDEQIACHYILSGDADMLINVVDASNLERNLYLTLQLLELGIPCVVALNMLDIAEKQQVRIDIDALAARLGCPVIPLVSTRGRGIEALKIALDRHQANSDLELVHYPQPLLREADLLAQQMSAQIPPRQRRWLGLQMLEGDIYSRAYAGDAADKLDIALANLSDEIDDPALHIADARYQTIAAICDAVSNTLT 2wig A 2.15 BS03 TC3 A 1 G116 G117 S198 A199 W231 L286 F398 H438 G114 G115 S196 A197 W229 L284 F396 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 19368529 601 DIIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWTDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPV 2wih A 2.5 BS01 P48 A 1 I10 Y15 V18 A31 K33 F80 L83 H84 L134 D145 I14 Y19 V22 A35 K37 F84 L87 H88 L138 D149 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.045uM remove_due_to_license_issue IC50=45nM P24941 19603809 1299 PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2wij A 2.1 BS03 TN7 A 1 G116 G117 S198 A199 W231 H438 G114 G115 S196 A197 W229 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 19368529 601 DIIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 2wik A 2.1 BS03 TC5 A 1 G116 G117 S198 A199 W231 L286 V288 G114 G115 S196 A197 W229 L284 V286 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 19368529 601 DIIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 2wj1 A 1.84 BS01 S99 A 1 S190 M191 F192 S217 T236 D237 I238 G239 S241 C269 T488 S157 M158 F159 S184 T203 D204 I205 G206 S208 C236 T455 K142 S217 S218 T236 I238 G239 G240 S241 F244 K109 S184 S185 T203 I205 G206 G207 S208 F211 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 19722626 1577 RQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQK 2wj2 A 2.55 BS01 OL1 A 1 M191 F192 S217 T236 D237 I238 G239 S241 C269 L278 T488 M159 F160 S185 T204 D205 I206 G207 S209 C237 L246 T456 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 19722626 1579 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQP 2wjg A 2.2 BS01 GDP A 1 N13 V14 G15 K16 S17 T18 N116 K117 D119 S145 A147 N17 V18 G19 K20 S21 T22 N120 K121 D123 S149 A151 ? 0005525 remove_due_to_license_issue Q57986 19615379 200 GGSHMKSYEIALIGNPNVGKSTIFNALTGENVYIGNWPGVTVEKKEGEFEYNGEKFKVVDLPGVYSLTANSIDEIIARDYIINEKPDLVVNIVDATALERNLYLTLQLMEMGANLLLALNKMDLAKSLGIEIDVDKLEKILGVKVVPLSAAKKMGIEELKKAISIAVKDK 2wji A 1.903 BS01 GNP A 1 P12 N13 G15 K16 S17 T18 N116 K117 D119 S145 A147 P12 N13 G15 K16 S17 T18 N111 K112 D114 S140 A142 ? 0005525 remove_due_to_license_issue Q57986 19615379 1166 MKSYEIALIGNPNVGKSTIFNALTGENVYIGTVEKKEGEFEYNGEKFKVVDLPGVYSLTANSIDEIIARDYIINEKPDLVVNIVDATALERNLYLTLQLMEMGANLLLALNKMDLAKSLGIEIDVDKLEKILGVKVVPLSAAKKMGIEELKKAISIAVKD 2wk2 A 2.05 BS01 SN5 B 1 W275 T276 E473 I476 W252 T253 E450 I453 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAGV 2wk2 A 2.05 BS02 SN5 C 1 D391 F392 Y418 D368 F369 Y395 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAGV 2wk2 A 2.05 BS03 SN5 C 2 W275 E315 D391 R446 W252 E292 D368 R423 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 2 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAGV 2wk2 A 2.05 BS04 NGT A 1 Y163 F191 W275 E315 M388 Y390 D391 W539 Y140 F168 W252 E292 M365 Y367 D368 W516 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1565 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAGV 2wk6 A 2.5 BS01 IUR A 1 H116 T118 L148 Y199 R202 I214 S217 I218 K221 H82 T84 L114 Y165 R168 I180 S183 I184 K187 D114 K115 H116 S117 T154 D195 R202 S217 K221 K222 D80 K81 H82 S83 T120 D161 R168 S183 K187 K188 2.4.2.4 0000002,0001525,0004645,0005515,0005829,0006206,0006213,0006935,0007165,0008083,0009032,0016154,0016757,0016763,0030154,0031641,0042803,0046074,0051969,1905333 Ki=0.48mM remove_due_to_license_issue P19971 19555658 1482 QLPELIRMKRDGGRLSEADIRGFVAAVVNGSAQGAQIGAMLMAIRLRGMDLEETSVLTQALAQSGQQLEWPEAWRQQLVDKHSTGGVGDKVSLVLAPALAACGCKVPMISGRGLGHTGGTLDKLESIPGFNVIQSPEQMQVLLDQAGCCIVGQSEQLVPADGILYAARDVTATVDSLPLITASILSKKLVEGLSALVVDVKFGGAAVFPNQEQARELAKTLVGVGASLGLRVAAALTAMDKPLGRCVGHALEVEEALLCMDGAGPPDLRDLVTTLGGALLWLSGHAGTQAQGAARVAAALDDGSALGRFERMLAAQGVDPGLARALCSGSPAERRQLLPRAREQEELLAPADGTVELVRALPLALVLHELGAGRSRAGEPLRLGVGAELLVDVGQRLRRGTPWLRVHRDGPALSGPQSRALQEALVLSDRAPFAAPSPFAELVLPP 2wks A 2.95 BS01 CB6 A 1 L11 Y22 N76 G78 A79 H82 H102 L103 T104 R113 L11 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue Q48255 19911771 1154 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQE 2wks B 2.95 BS01 CB6 A 1 D89 L93 D89 L93 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue Q48255 19911771 1154 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQE 2wks B 2.95 BS02 CB6 B 1 L11 Y22 N76 G78 A79 H82 H102 L103 T104 R113 L11 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue Q48255 19911771 1154 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQE 2wky A 2.2 BS01 IBC A 1 E13 Y61 L89 T90 R95 G140 S141 T142 E190 S193 E10 Y58 L86 T87 R92 G137 S138 T139 E187 S190 ? 0015276,0016020 Ki=2.57nM remove_due_to_license_issue P22756 19588945 1260 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 2wkz A 1.7 BS01 5AH B 1 R8 D25 G27 A28 D29 V32 G48 G49 I50 P81 V82 I84 R8 D25 G27 A28 D29 V32 G48 G49 I50 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 19961222 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2wkz B 1.7 BS01 5AH B 1 D125 G127 A128 D129 G148 G149 I150 F153 V182 I184 D25 G27 A28 D29 G48 G49 I50 F53 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.7nM remove_due_to_license_issue P12499 19961222 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2wl0 A 1.9 BS01 5AH A 1 R8 D25 G27 A28 D29 D30 V32 G48 I50 P81 T82 R8 D25 G27 A28 D29 D30 V32 G48 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=16nM remove_due_to_license_issue P12499 19961222 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 2wl0 B 1.9 BS01 5AH A 1 L123 D125 G127 A128 D129 G148 G149 I150 P181 T182 L23 D25 G27 A28 D29 G48 G49 I50 P81 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 19961222 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 2wly A 2.4 BS01 SN5 A 1 F191 W275 T276 E473 I476 F168 W252 T253 E450 I453 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1571 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAGV 2wly A 2.4 BS02 NGT A 1 Y163 W275 E315 M388 Y390 D391 W539 Y140 W252 E292 M365 Y367 D368 W516 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1572 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAGV 2wlz A 1.82 BS01 NGT A 1 Y163 F191 W275 E315 M388 Y390 D391 W539 Y140 F168 W252 E292 M365 Y367 D368 W516 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1569 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAG 2wm0 A 1.9 BS01 NGT A 1 Y163 F191 W275 E315 M388 Y390 D391 W539 Y140 F168 W252 E292 M365 Y367 D368 W516 D311 D313 E315 Y390 D288 D290 E292 Y367 3.2.1.14 0000272,0004553,0004568,0005975,0006032,0008061,0008843,0016798 remove_due_to_license_issue P07254 20209544 1564 AAPGKPTIAWGNTKFAIVEVDQAATAYNNLVKVKNAADVSVSWNLWNGDTGTTAKILLNGKEAWSGPSTGSSGTANFKVNKGGRYQMQVALCNADGCTASDATEIVVADTDGSHLAPLKEPLLEKNKPYKQNSGKVVGSYFVEWGVYGRNFTVDKIPAQNLTHLLYGFIPICGGNGINDSLKEIEGSFQALQRSCQGREDFKVSIHDPFAALQKAQKGVTAWDDPYKGNFGQLMALKQAHPDLKILPSIGGWTLSDPFFFMGDKVKRDRFVGSVKEFLQTWKFFDGVDIDWEFPGGKGANPNLGSPQDGETYVLLMKELRAMLDQLSAETGRKYELTSAISAGKDKIDKVAYNVAQNSMDHIFLMSYDFYGAFDLKNLGHQTALNAPAWKPDTAYTTVNGVNALLTQGVKPGKIVVGTAMYGRGWTGVNGYQNNIPFTGTATGPVKGTWENGIVDYRQIASQFMSGEWQYTYDATAEAPYVFKPSTGDLITFDDARSVQAKGKYVLDKQLGGLFSWEIDADNGDILNSMNASLGNSAG 2wmr A 2.43 BS01 ZYR A 1 L15 A36 E85 Y86 C87 L137 L9 A30 E69 Y70 C71 L121 D130 K132 E134 N135 D148 T170 D114 K116 E118 N119 D132 T154 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=52uM remove_due_to_license_issue IC50=52000nM O14757 19572549 1271 EDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2wmu A 2.6 BS01 ZYU A 1 L15 G16 A36 Y86 C87 L137 L7 G8 A23 Y62 C63 L113 D130 K132 E134 N135 D148 T170 D106 K108 E110 N111 D124 T146 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=42000nM O14757 19572549 1271 WDLVQTLGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2wmv A 2.009 BS01 ZYV A 1 L15 A36 Y86 C87 E91 L137 L9 A25 Y67 C68 E72 L118 D130 K132 E134 N135 D148 T170 D111 K113 E115 N116 D129 T151 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=9.2uM remove_due_to_license_issue IC50=9200nM O14757 19572549 1271 EDWDLVQTLGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2wmw A 2.43 BS01 ZYW A 1 V23 A36 Y86 C87 L137 V11 A24 Y64 C65 L115 D130 K132 E134 N135 D148 T170 D108 K110 E112 N113 D126 T148 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.39uM remove_due_to_license_issue IC50=390nM O14757 19572549 1270 EDWDLVQTLGVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2wmx A 2.45 BS01 ZY6 A 1 V23 C87 E91 L137 V12 C66 E70 L116 D130 K132 E134 N135 D148 T170 D109 K111 E113 N114 D127 T149 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.86uM remove_due_to_license_issue IC50=890nM O14757 19572549 1270 EDWDLVQTLGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2wn9 A 1.75 BS01 ZY5 A 1 Y93 W147 Y94 W148 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=3nM remove_due_to_license_issue Q8WSF8 19696737 301 LHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wn9 A 1.75 BS02 ZY5 B 1 T36 M116 I118 D164 S167 T37 M117 I119 D165 S168 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=3nM remove_due_to_license_issue Q8WSF8 19696737 301 LHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wn9 E 1.75 BS01 ZY5 A 1 T36 I118 D164 S167 T43 I125 D171 S174 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=3nM remove_due_to_license_issue Q8WSF8 19696737 301 DYKDDDDKLHSQANLMRLKSDLFNRSYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2wn9 E 1.75 BS02 ZY5 E 1 Y93 W147 Y188 C190 Y195 Y100 W154 Y195 C197 Y202 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=3nM remove_due_to_license_issue Q8WSF8 19696737 301 DYKDDDDKLHSQANLMRLKSDLFNRSYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2wnc A 2.2 BS01 TKT A 1 Y93 W147 Y188 C190 Y195 Y98 W152 Y193 C195 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=479nM remove_due_to_license_issue Q8WSF8 19696737 300 DDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAG 2wnc A 2.2 BS02 TKT B 1 Q57 M116 I118 Q62 M121 I123 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=479nM remove_due_to_license_issue Q8WSF8 19696737 300 DDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAG 2wnc E 2.2 BS01 TKT A 1 Y55 Q57 I118 Y60 Q62 I123 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=479nM remove_due_to_license_issue Q8WSF8 19696737 300 DDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnc E 2.2 BS02 TKT E 1 Y93 W147 C190 C191 Y195 Y98 W152 C195 C196 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=479nM remove_due_to_license_issue Q8WSF8 19696737 300 DDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnj A 1.8 BS01 ZY7 A 1 Y93 W147 Y188 C190 Y94 W148 Y189 C191 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=330nM remove_due_to_license_issue Q8WSF8 19696737 301 LHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnj A 1.8 BS02 ZY7 B 1 Y55 Q57 V108 I118 Y56 Q58 V109 I119 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=330nM remove_due_to_license_issue Q8WSF8 19696737 301 LHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnj E 1.8 BS01 ZY7 A 1 T36 I118 S167 T45 I127 S176 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=330nM remove_due_to_license_issue Q8WSF8 19696737 301 DYKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnj E 1.8 BS02 ZY7 E 1 Y93 W147 Y188 Y195 Y102 W156 Y197 Y204 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=330nM remove_due_to_license_issue Q8WSF8 19696737 301 DYKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnl F 2.7 BS01 AN5 F 1 Y93 W147 Y96 W150 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 19696737 300 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wnl J 2.7 BS01 AN5 F 1 Y55 S167 Y58 S170 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 19696737 300 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2wo8 A 2.0 BS04 077 A 1 A182 H218 E219 H222 H228 V235 T239 Y240 A78 H114 E115 H118 H124 V131 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.52uM remove_due_to_license_issue IC50=520nM P39900 19703773 1271 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGDPKE 2wo9 A 1.7 BS04 068 A 1 I180 L181 A182 H218 E219 H222 H228 V235 T239 Y240 F248 I75 L76 A77 H113 E114 H117 H123 V130 T134 Y135 F143 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=0.062uM remove_due_to_license_issue IC50=62nM P39900 19703773 1271 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGDPKE 2woa A 2.3 BS04 576 A 1 L181 A182 L214 H218 E219 H228 V235 F237 T239 Y240 K241 L77 A78 L110 H114 E115 H124 V131 F133 T135 Y136 K137 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=1.15uM remove_due_to_license_issue P39900 19703773 1273 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGDPKE 2won A 2.8 BS01 ZZE A 1 L100 K103 V106 V108 Y188 G190 F227 W229 L234 H235 P236 Y318 L100 K103 V106 V108 Y188 G190 F227 W229 L234 H235 P236 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 20660667 1558 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 2woq A 1.75 BS01 AYC A 1 D131 S175 Y202 K205 Y211 F214 K260 Y283 V285 S286 Y324 D126 S170 Y197 K200 Y206 F209 K255 Y278 V280 S281 Y319 K205 K260 K200 K255 4.2.1.24 0004655,0005829,0006779,0006782,0006783,0008270,0016829,0033014,0046872 remove_due_to_license_issue Q59643 19822707 1333 ANRAYPYTRLRRNRRDDFSRRLVRENVLTVDDLILPVFVLDGVNQRESIPSMPGVERLSIDQLLIEAEEWVALGIPALALFPVTPVEKKSLDAAEAYNPEGIAQRATRALRERFPELGIITDVALDPFTTHGQDGILDDDGYVLNDVSIDVLVRQALSHAEAGAQVVAPSDMMDGRIGAIREALESAGHTNVRIMAYSAKYASAYYGPFRDAVGSASNLGKGNKATYQMDPANSDEALHEVAADLAEGADMVMVKPGMPYLDIVRRVKDEFRAPTFVYQVSGEYAMHMGAIQNGWLAESVILESLTAFKRAGADGILTYFAKQAAEQL 2wor A 1.7 BS02 2AN A 1 G11 M12 D14 M15 K18 G11 M12 D14 M15 K18 ? 0000302,0001525,0005509,0005515,0005576,0005615,0005634,0005737,0005783,0005829,0005925,0008270,0008544,0010820,0030216,0032496,0035578,0046872,0046914,0048306,0050786,0061844,0062023,0070374,0071624,0090026,0140486 Kd=125uM remove_due_to_license_issue P31151 19810752 1098 SNTQAERSIIGMIDMFHKYTRRDDKIDKPSLLTMMKENFPNFLSACDKKGTNYLADVFEKKDKNEDKKIDFSEFLSLLGDIATDYHKQSHGAAPCS 2wos A 1.7 BS02 6AN A 1 R7 S8 G11 M12 R7 S8 G11 M12 ? 0000302,0001525,0005509,0005515,0005576,0005615,0005634,0005737,0005783,0005829,0005925,0008270,0008544,0010820,0030216,0032496,0035578,0046872,0046914,0048306,0050786,0061844,0062023,0070374,0071624,0090026,0140486 remove_due_to_license_issue P31151 19810752 1098 SNTQAERSIIGMIDMFHKYTRRDDKIDKPSLLTMMKENFPNFLSACDKKGTNYLADVFEKKDKNEDKKIDFSEFLSLLGDIATDYHKQSHGAAPCS 2wot A 1.85 BS01 ZZG A 1 I211 A230 K232 L260 L278 S280 Y282 H283 G286 L340 A350 D351 I14 A33 K35 L63 L81 S83 Y85 H86 G89 L143 A153 D154 D333 K335 N338 D351 T375 D136 K138 N141 D154 T178 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=44nM remove_due_to_license_issue IC50=44nM, EC50=55nM P36897 19736928 1500 GGTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG 2wou A 2.3 BS01 ZZF A 1 I211 A230 L260 L278 S280 D281 Y282 H283 G286 D290 L340 I14 A33 L63 L81 S83 D84 Y85 H86 G89 D93 L143 D333 K335 N338 D351 T375 D136 K138 N141 D154 T178 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=72nM remove_due_to_license_issue EC50=22nM, IC50=72nM P36897 19736928 1500 GGTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLS 2wpa A 2.51 BS01 889 A 1 I10 Y15 A31 K33 F80 L83 Q85 N132 L134 D145 I14 Y19 A35 K37 F84 L87 Q89 N136 L138 D149 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 20153204 1301 PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2wpb A 2.05 BS01 ZZI A 1 G189 Y190 D191 N192 S208 G194 Y195 D196 N197 S213 S47 Y110 Y137 L142 K165 I206 S52 Y115 Y142 L147 K170 I211 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262,0042802,0044010 Ki=1.3mM remove_due_to_license_issue P0A6L4 20826162 1298 HHHHHHATNLRGVMAALLTPFDQQQALDKASLRRLVQFNIQQGIDGLYVGGSTGEAFVQSLSEREQVLEIVAEEAKGKIKLIAHVGCVSTAESQQLAASAKRYGFDAVSAVTPFYYPFSFEEHCDHYRAIIDSADGLPMVVYNIPALSGVKLTLDQINTLVTLPGVGALKQTSGDLYQMEQIRREHPDLVLYNGYDNIFASGLLAGADGGIGSTYNIMGWRYQGIVKALKEGDIQTAQKLQTECNKVIDLLIKTGVFRGLKTVLHYMDVVSVPLCRKPFGPVDEKYLPELKALAQQLMQERG 2wpb C 2.05 BS01 ZZI C 1 G189 Y190 D191 G207 S208 G188 Y189 D190 G206 S207 S47 Y110 Y137 L142 K165 I206 S46 Y109 Y136 L141 K164 I205 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262,0042802,0044010 Ki=1.3mM remove_due_to_license_issue P0A6L4 20826162 1297 ATNLRGVMAALLTPFDQQQALDKASLRRLVQFNIQQGIDGLYVGGSTGEAFVQSLSEREQVLEIVAEEAKGKIKLIAHVGCVSTAESQQLAASAKRYGFDAVSAVTPFYYPFSFEEHCDHYRAIIDSADGLPMVVYNIPALSGVKLTLDQINTLVTLPGVGALKQTSGDLYQMEQIRREHPDLVLYNGYDNIFASGLLAGADGGIGSTYNIMGWRYQGIVKALKEGDIQTAQKLQTECNKVIDLLIKTGVFRGLKTVLHYMDVVSVPLCRKPFGPVDEKYLPELKALAQQLMQER 2wpb D 2.05 BS01 ZZI D 1 G189 Y190 D191 G207 S208 I243 G188 Y189 D190 G206 S207 I242 S47 Y110 Y137 L142 K165 I206 S46 Y109 Y136 L141 K164 I205 4.1.3.3 0005737,0005829,0005975,0008747,0016829,0019262,0042802,0044010 Ki=1.3mM remove_due_to_license_issue P0A6L4 20826162 1297 ATNLRGVMAALLTPFDQQQALDKASLRRLVQFNIQQGIDGLYVGGSTGEAFVQSLSEREQVLEIVAEEAKGKIKLIAHVGCVSTAESQQLAASAKRYGFDAVSAVTPFYYPFSFEEHCDHYRAIIDSADGLPMVVYNIPALSGVKLTLDQINTLVTLPGVGALKQTSGDLYQMEQIRREHPDLVLYNGYDNIFASGLLAGADGGIGSTYNIMGWRYQGIVKALKEGDIQTAQKLQTECNKVIDLLIKTGVFRGLKTVLHYMDVVSVPLCRKPFGPVDEKYLPELKALAQQLMQER 2wq4 A 1.42 BS01 SFU A 1 Y48 T83 G84 R85 Y48 T83 G84 R85 ? remove_due_to_license_issue B4EH86 20152153 200 PLLSASIVSAPVVTSETYVDIPGLYLDVAKAGIRDGKLQVILNVPTPYATGNNFPGIYFAIATNQGVVADGCFTYSSKVPESTGRMPFTLVATIDVGSGVTFVKGQWKSVRGSAMHIDSYASLSAIWGTAAPSS 2wq4 A 1.42 BS02 SFU B 1 T74 R111 T74 R111 ? remove_due_to_license_issue B4EH86 20152153 200 PLLSASIVSAPVVTSETYVDIPGLYLDVAKAGIRDGKLQVILNVPTPYATGNNFPGIYFAIATNQGVVADGCFTYSSKVPESTGRMPFTLVATIDVGSGVTFVKGQWKSVRGSAMHIDSYASLSAIWGTAAPSS 2wq4 C 1.42 BS01 SFU A 1 T74 R111 T74 R111 ? remove_due_to_license_issue B4EH86 20152153 200 PLLSASIVSAPVVTSETYVDIPGLYLDVAKAGIRDGKLQVILNVPTPYATGNNFPGIYFAIATNQGVVADGCFTYSSKVPESTGRMPFTLVATIDVGSGVTFVKGQWKSVRGSAMHIDSYASLSAIWGTAA 2wq4 C 1.42 BS02 SFU C 1 Y48 T83 R85 Y48 T83 R85 ? remove_due_to_license_issue B4EH86 20152153 200 PLLSASIVSAPVVTSETYVDIPGLYLDVAKAGIRDGKLQVILNVPTPYATGNNFPGIYFAIATNQGVVADGCFTYSSKVPESTGRMPFTLVATIDVGSGVTFVKGQWKSVRGSAMHIDSYASLSAIWGTAA 2wq5 A 1.65 BS01 MIY A 1 L2 W18 A22 G29 R30 F63 F64 L2 W18 A22 G29 R30 F63 F64 Y27 G29 G31 H47 D48 Y51 Y67 D93 Y27 G29 G31 H47 D48 Y51 Y67 D93 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0046872,0047498,0047499,0050482 Kd=180uM remove_due_to_license_issue P15445 20211188 1120 NLYQFKNMIKCTVPSRSWWDFADYGCYCGRGGSGTPVDDLDRCCQVHDNCYNEAEKISKCWPFFKTYSYKCSQGTLTCKGGNNACAASVCDCDRLAAICFAGAPYNDNNYNIDLKARCQ 2wqb A 2.95 BS01 QQ1 A 1 A853 K855 I902 E903 Y904 A905 N969 F983 A36 K38 I72 E73 Y74 A75 N139 F153 N964 A966 R968 N969 D982 Y992 R999 N134 A136 R138 N139 D152 Y162 R168 2.7.10.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=540nM Q02763 19854647 2121 YPVLDWNDIKFQDVIGEGGQVLKARIKKDGLRMDAAIKRMKELEVLCKLGHHPNIINLLGACEHRGYLYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRNLAARNILVGENYVAKIADFGLSRGQEVYVKKTGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGIDCSA 2wqp A 1.75 BS01 WQP A 1 E25 K53 Q55 N74 T110 F112 K129 S132 S154 Y186 S213 H215 D247 E24 K52 Q54 N73 T109 F111 K128 S131 S153 Y185 S212 H214 D246 ? 0016051,0046872,0047444,0070085 Ki=3.1uM remove_due_to_license_issue Q7DDU0 19719325 1350 QNNNEFKIGNRSVGYNHEPLIICEIGINHEGSLKTAFEMVDAAYNAGAEVVKHQTHIVEDEMSDEAKQVIPGNADVSIYEIMERCALNEEDEIKLKEYVESKGMIFISTLFSRAAALRLQRMDIPAYKIGSGECNNYPLIKLVASFGKPIILSTGMNSIESIKKSVEIIREAGVPYALLHCTNIYPTPYEDVRLGGMNDLSEAFPDAIIGLSDHTLDNYACLGAVALGGSILERHFTDRMDRPGPDIVCSMNPDTFKELKQGAHALKLARGGKKDTIIAGEKPTKDFAFASVVADKDIKKGELLSGDNLWVKRPGNGDFSVNEYETLFGKVAACNIRKGAQIKKTDIE 2wr8 A 1.77 BS01 SAH A 1 F181 N183 Y212 S226 E231 M236 F183 N185 Y214 S228 E233 M238 3.13.2.3 0016787 Ki=3.6uM remove_due_to_license_issue O58212 19739191 1257 GSHMITLTTDFGLKGPYVGEMKVAMLRINPNAKIVDVTHSVTRHSILEGSFVMEQVVKYSPKGTVHVGVIDPGVGERRAIVIEGDQYLVVPDNGLATLPLKHIKVKSVYEIIPDKIRKFTGWEISSTFHGRDIFGPAGALIEKGIHPEEFGREIPVDSIVKLNVEPRKEGDVWILKVIYIDDFGNVILNLENYEKPRTVELLDFNLRLPYLETYGLVEKGEMLALPGSHDYLEIAVNMGSAAERLNVKVGDELRVRLL 2wsx A 3.5 BS01 NM2 A 1 W142 W323 Y327 M331 W135 W316 Y320 M324 ? 0005886,0009437,0015226,0015297,0015879,0016020,0022857,0044667,0071705,1900749,1900751,1902270,1902603 remove_due_to_license_issue P31553 20829798 1504 TGIEPKVFFPPLIIVGILCWLTVRDLDAANVVINAVFSYVTNVWGWAFEWYMVVMLFGWFWLVFGPYAKKRLGEEPPEFSTASWIFMMFASCTSAAVLFWGSIEIYYYISTPPFGLEPNSTGAKELGLAYSLFHWGPLPWATYSFLSVAFAYFFFVRKMEVIRPSSTLVPLVGEKHAKGLFGTIVDNFYLVALIFAMGTSLGLATPLVTECMQWLFGIPHTLQLDAIIITCWIILNAICVACGLQKAVRIASDVRSYLSFLMLGWVFIVSGASFIMNYFTDSVGMLLMYLPRMLFYTDPIAKGGFPQGWTVFYWAWWVIYAIQMSIFLARISRGRTVRELCFGMVLGLTASTWILWTVLGSNTLLLIDKNILNIPNLIEQYGVARAIIETWAALPLSTATMWGFFILCFIATVTLVNACSYTLAMSTCREVRDGEDPPLLVRIGWSILVGIIGIVLLALGGLKPIQTAIIAGGCPLFFVNIMVTLSFIKDAKQNWK 2wsx A 3.5 BS02 NM2 A 2 G311 G315 Q473 G304 G308 Q466 ? 0005886,0009437,0015226,0015297,0015879,0016020,0022857,0044667,0071705,1900749,1900751,1902270,1902603 remove_due_to_license_issue P31553 20829798 1505 TGIEPKVFFPPLIIVGILCWLTVRDLDAANVVINAVFSYVTNVWGWAFEWYMVVMLFGWFWLVFGPYAKKRLGEEPPEFSTASWIFMMFASCTSAAVLFWGSIEIYYYISTPPFGLEPNSTGAKELGLAYSLFHWGPLPWATYSFLSVAFAYFFFVRKMEVIRPSSTLVPLVGEKHAKGLFGTIVDNFYLVALIFAMGTSLGLATPLVTECMQWLFGIPHTLQLDAIIITCWIILNAICVACGLQKAVRIASDVRSYLSFLMLGWVFIVSGASFIMNYFTDSVGMLLMYLPRMLFYTDPIAKGGFPQGWTVFYWAWWVIYAIQMSIFLARISRGRTVRELCFGMVLGLTASTWILWTVLGSNTLLLIDKNILNIPNLIEQYGVARAIIETWAALPLSTATMWGFFILCFIATVTLVNACSYTLAMSTCREVRDGEDPPLLVRIGWSILVGIIGIVLLALGGLKPIQTAIIAGGCPLFFVNIMVTLSFIKDAKQNWK 2wtc A 3.0 BS01 VGM A 1 L226 K249 L301 L303 M304 G307 L354 T367 D368 L16 K35 L75 L77 M78 G81 L128 T141 D142 D347 K349 N352 D368 T387 D121 K123 N126 D142 T159 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=310nM O96017 20022510 1513 VYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 2wtd A 2.75 BS01 ZZK A 1 L226 K249 L301 L303 M304 L354 T367 D368 L17 K36 L76 L78 M79 L129 T142 D143 D347 K349 N352 D368 T387 D122 K124 N127 D143 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue EC50=10000nM O96017 20022510 1513 SVYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 2wti A 2.5 BS01 WTI A 1 L226 A247 K249 L301 L303 M304 E305 L354 T367 D368 L17 A34 K36 L76 L78 M79 E80 L129 T142 D143 D347 K349 N352 D368 T387 D122 K124 N127 D143 T161 2.7.11.1 0004672,0005524,0006468 ic50=0.092uM remove_due_to_license_issue EC50=5000nM O96017 20022510 1513 SVYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 2wtj A 2.1 BS01 WTJ A 1 A247 L303 M304 E305 G307 L354 D368 A35 L79 M80 E81 G83 L130 D144 D347 K349 N352 D368 T387 D123 K125 N128 D144 T162 2.7.11.1 0004672,0005524,0006468 ic50=0.7uM remove_due_to_license_issue IC50=700nM O96017 20022510 1513 MSVYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 2wtv A 2.4 BS01 ZZL A 1 L139 G140 V147 K162 L194 Y212 A213 G216 L263 A273 D274 G276 V279 L15 G16 V23 K38 L70 Y88 A89 G92 L139 A149 D150 G152 V155 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Ki=1.8nM remove_due_to_license_issue IC50=34nM, Kd=6.5nM O14965 20067443 1390 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPRGEVYKELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2wtw A 3.302 BS01 ZZL A 1 R137 G140 V147 K162 L194 L210 Y212 A213 G216 L263 A273 D274 R10 G13 V20 K35 L67 L83 Y85 A86 G89 L136 A146 D147 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T159 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=34nM, Kd=6.5nM O14965 20067443 1390 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPRGEVYKELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2wtx C 2.2 BS02 VDO C 1 D130 H154 I225 R262 R300 D361 G362 M363 N364 D119 H143 I214 R246 R284 D345 G346 M347 N348 H154 D361 H143 D345 2.4.1.15 0003824,0003825,0005992,0006950,0006970,0006974,0016757,0016758,0070415 Ki=1.3mM remove_due_to_license_issue P31677 20077550 1458 SRLVVVSNRIAPGLAVGILGALKAAGGLWFGWSGETGNQPLKKVKKGNITWASFNLSEQDLDEYYNQFSNAVLWPAFHYRLDLVQFQRPAWDGYLRVNALLADKLLPLLQDDDIIWIHDYHLLPFAHELRKRGVNNRIGFFLHIPFPTPEIFNALPTYDTLLEQLCDYDLLGFQTENDRLAFLDCLSNLTRVTTRSAKSHTAWGKAFRTEVYPIGIEPKEIAKQAAGPAQLKAELKNVQNIFSVERLDYSKGLPERFLAYEALLEKYPQHHGKIRYTQIAPTSRGDVQAYQDIRHQLENEAGRINGKYGQLGWTPLYYLNQHFDRKLLMKIFRYSDVGLVTPLRDGMNLVAKEYVAAQDPANPGVLVLSQFAGAANELTSALIVNPYDRDEVAAALDRALTMSLAERISRHAEMLDVIVKNDINHWQECFISDLKQIVPR 2wu6 A 1.92 BS01 DKI A 1 L162 V170 A184 V220 F236 L239 G240 K241 L290 D320 L29 V37 A51 V87 F103 L106 G107 K108 L157 D187 D283 K285 N288 D320 T337 D150 K152 N155 D187 T204 2.7.12.1 0004672,0005524,0006468 ic50=29.2nM remove_due_to_license_issue IC50=29nM P49761 21276940 1484 RSVEDDKEGHLVCRIGDWLQERYEIVGNLGEGTFGKVVECLDHARGKSQVALKIIRNVGKYREAARLEINVLKKIKEKDKENKFLCVLMSDWFNFHGHMCIAFELLGKNTFEFLKENNFQPYPLPHVRHMAYQLCHALRFLHENQLTHTDLKPENILFVNSEFETLYNEHKSCEEKSVKNTSIRVADFGSATFDHEHHTTIVATRHYRPPEVILELGWAQPCDVWSIGCILFEYYRGFTLFQTHENREHLVMMEKILGPIPSHMIHRTRKQKYFYKGGLVWDENSSDGRYVKENCKPLKSYMLQDSLEHVQLFDLMRRMLEFDPAQRITLAEALLHPFFAGLTPEERSFH 2wu7 A 2.25 BS01 V25 A 1 L162 G163 E164 V170 A184 K186 L239 E287 L290 L28 G29 E30 V36 A50 K52 L105 E153 L156 D283 K285 N288 D320 T337 D149 K151 N154 D186 T203 2.7.12.1 0004672,0005524,0006468 ic50=530nM remove_due_to_license_issue P49761 21276940 1483 SVEDDKEGHLVCRIGDWLQERYEIVGNLGEGTFGKVVECLDHARGKSQVALKIIRNVGKYREAARLEINVLKKIKEKDKENKFLCVLMSDWFNFHGHMCIAFELLGKNTFEFLKENNFQPYPLPHVRHMAYQLCHALRFLHENQLTHTDLKPENILFVNSEFETLYNEHKSCEEKSVKNTSIRVADFGSATFDHEHHTTIVATRHYRPPEVILELGWAQPCDVWSIGCILFEYYRGFTLFQTHENREHLVMMEKILGPIPSHMIHRTRKQKYFYKGGLVWDENSSDGRYVKENCKPLKSYMLQDSLEHVQLFDLMRRMLEFDPAQRITLAEALLHPFFAGLTPEERSF 2wuf B 1.9 BS01 KEM B 1 G44 G45 G46 A114 L115 L158 F212 H269 W270 G38 G39 G40 A108 L109 L152 F206 H263 W264 G45 G46 G48 N113 A114 L115 R192 D241 H269 W270 G39 G40 G42 N107 A108 L109 R186 D235 H263 W264 3.7.1.17,3.7.1.8 0005515,0005886,0006694,0009274,0016042,0016787,0018774,0034820,0051701,0102296 Kd=51uM remove_due_to_license_issue P9WNH5 19875455 1289 LTFESTSRFAEVDVDGPLKLHYHEAGVGNDQTVVLLHGGGPGAASWTNFSRNIAVLARHFHVLAVDQPGYGHSDKRAEHGQFNRYAAMALKGLFDQLGLGRVPLVGNALGGGTAVRFALDYPARAGRLVLMGPGGLSINLFAPDPTEGVKRLSKFSVAPTRENLEAFLRVMVYDKNLITPELVDQRFALASTPESLTATRAMGKSFAGADFEAGMMWREVYRLRQPVLLIWGREDRVNPLDGALVALKTIPRAQLHVFGQCGHWVQVEKFDEFNKLTIEFLG 2wuu A 1.42 BS01 NHW A 1 H12 A13 F14 W15 Y80 V81 I166 N167 L169 C170 V171 R176 E177 R179 L180 A181 P182 I185 T189 V192 W198 A200 Y202 T203 A204 L208 Y404 H2 A3 F4 W5 Y70 V71 I153 N154 L156 C157 V158 R163 E164 R166 L167 A168 P169 I172 T176 V179 W185 A187 Y189 T190 A191 L195 Y385 N167 F168 L169 T203 L421 N154 F155 L156 T190 L402 2.3.1.97 0004379,0005737,0006499,0016746 ic50=68.7nM remove_due_to_license_issue D0AB09 20036251 1422 AHAFWSTQPVPQTEDETEKIVFAGPMDEPKTVADIPEEPYPIASTFEWWTPNMEAADDIHAIYELLRDNYVESMFRFNYSEEFLQWALCPPSYIPDWHVAVRRKADKKLLAFIAGVPVTLRMGTPKYMKVKAQEKGQEEEAAKYDAPRHICEINFLCVHKQLREKRLAPILIKEVTRRVNRTNVWQAVYTAGVLLPTPYASGQYFHRSLNPEKLVEIRFSGIPAQYQKFQNPMAMLKRNYQLPNAPKNSGLREMKPSDVPQVRRILMNYLDNFDVGPVFSDAEISHYLLPRDGVVFTYVVENDKKVTDFFSFYRIPSTVIILNAAYVHYYAATSMPLHQLILDLLIVAHSRGFDVCNMVEILDNRSFVEQLKFGAGDGHLRYYFYNWAYPKIKPSQVALVML 2wva V 2.2 BS01 TPU V 1 G413 H414 I415 G439 G441 S442 N467 G469 Y470 T471 I472 E473 G412 H413 I414 G438 G440 S441 N466 G468 Y469 T470 I471 E472 L116 G117 T388 G413 D440 N467 G469 I472 E473 L115 G116 T387 G412 D439 N466 G468 I471 E472 4.1.1.1 0000287,0000949,0003824,0004737,0005829,0016831,0019752,0030976,0046872 remove_due_to_license_issue P06672 20099870 600 SYTVGTYLAERLVQIGLKHHFAVAGDYNLVLLDNLLLNKNMEQVYCCNELNCGFSAEGYARAKGAAAAVVTYSVGALSAFDAIGGAYAENLPVILISGAPNNNDHAAGHVLHHALGKTDYHYQLEMAKNITAAAEAIYTPEEAPAKIDHVIKTALREKKPVYLEIACNIASMPCAAPGPASALFNDEASDEASLNAAVEETLKFIANRDKVAVLVGSKLRAAGAEEAAVKFADALGGAVATMAAAKSFFPEENPHYIGTSWGEVSYPGVEKTMKEADAVIALAPVFNDYSTTGWTDIPDPKKLVLAEPRSVVVNGIRFPSVHLKDYLTRLAQKVSKKTGALDFFKSLNAGELKKAAPADPSAPLVNAEIARQVEALLTPNTTVIAETGDSWFNAQRMKLPNGARVEYEMQWGHIGWSVPAAFGYAVGAPERRNILMVGDGSFQLTAQEVAQMVRLKLPVIIFLINNYGYTIEVMIHDGPYNNIKNWDYAGLMEVFNGNGGYDSGAGKGLKAKTGGELAEAIKVALANTDGPTLIECFIGREDCTEELVKWGKRVAAANSRKPVNK 2wva V 2.2 BS04 TPU Z 1 A25 E50 V75 H114 A24 E49 V74 H113 L116 G117 T388 G413 D440 N467 G469 I472 E473 L115 G116 T387 G412 D439 N466 G468 I471 E472 4.1.1.1 0000287,0000949,0003824,0004737,0005829,0016831,0019752,0030976,0046872 remove_due_to_license_issue P06672 20099870 600 SYTVGTYLAERLVQIGLKHHFAVAGDYNLVLLDNLLLNKNMEQVYCCNELNCGFSAEGYARAKGAAAAVVTYSVGALSAFDAIGGAYAENLPVILISGAPNNNDHAAGHVLHHALGKTDYHYQLEMAKNITAAAEAIYTPEEAPAKIDHVIKTALREKKPVYLEIACNIASMPCAAPGPASALFNDEASDEASLNAAVEETLKFIANRDKVAVLVGSKLRAAGAEEAAVKFADALGGAVATMAAAKSFFPEENPHYIGTSWGEVSYPGVEKTMKEADAVIALAPVFNDYSTTGWTDIPDPKKLVLAEPRSVVVNGIRFPSVHLKDYLTRLAQKVSKKTGALDFFKSLNAGELKKAAPADPSAPLVNAEIARQVEALLTPNTTVIAETGDSWFNAQRMKLPNGARVEYEMQWGHIGWSVPAAFGYAVGAPERRNILMVGDGSFQLTAQEVAQMVRLKLPVIIFLINNYGYTIEVMIHDGPYNNIKNWDYAGLMEVFNGNGGYDSGAGKGLKAKTGGELAEAIKVALANTDGPTLIECFIGREDCTEELVKWGKRVAAANSRKPVNK 2wva Z 2.2 BS01 TPU V 1 A25 E50 V75 H114 A24 E49 V74 H113 L116 G117 T388 G413 D440 N467 G469 I472 E473 L115 G116 T387 G412 D439 N466 G468 I471 E472 4.1.1.1 0000287,0000949,0003824,0004737,0005829,0016831,0019752,0030976,0046872 remove_due_to_license_issue P06672 20099870 600 SYTVGTYLAERLVQIGLKHHFAVAGDYNLVLLDNLLLNKNMEQVYCCNELNCGFSAEGYARAKGAAAAVVTYSVGALSAFDAIGGAYAENLPVILISGAPNNNDHAAGHVLHHALGKTDYHYQLEMAKNITAAAEAIYTPEEAPAKIDHVIKTALREKKPVYLEIACNIASMPCAAPGPASALFNDEASDEASLNAAVEETLKFIANRDKVAVLVGSKLRAAGAEEAAVKFADALGGAVATMAAAKSFFPEENPHYIGTSWGEVSYPGVEKTMKEADAVIALAPVFNDYSTTGWTDIPDPKKLVLAEPRSVVVNGIRFPSVHLKDYLTRLAQKVSKKTGALDFFKSLNAGELKKAAPADPSAPLVNAEIARQVEALLTPNTTVIAETGDSWFNAQRMKLPNGARVEYEMQWGHIGWSVPAAFGYAVGAPERRNILMVGDGSFQLTAQEVAQMVRLKLPVIIFLINNYGYTIEVMIHDGPYNNIKNWDYAGLMEVFNGNGGYDSGAGKGLKAKTGGELAEAIKVALANTDGPTLIECFIGREDCTEELVKWGKRVAAANSRKPVNK 2wva Z 2.2 BS04 TPU Z 1 G389 D390 G413 H414 I415 G439 G441 S442 G469 Y470 T471 I472 E473 G388 D389 G412 H413 I414 G438 G440 S441 G468 Y469 T470 I471 E472 L116 G117 T388 G413 D440 N467 G469 I472 E473 L115 G116 T387 G412 D439 N466 G468 I471 E472 4.1.1.1 0000287,0000949,0003824,0004737,0005829,0016831,0019752,0030976,0046872 remove_due_to_license_issue P06672 20099870 600 SYTVGTYLAERLVQIGLKHHFAVAGDYNLVLLDNLLLNKNMEQVYCCNELNCGFSAEGYARAKGAAAAVVTYSVGALSAFDAIGGAYAENLPVILISGAPNNNDHAAGHVLHHALGKTDYHYQLEMAKNITAAAEAIYTPEEAPAKIDHVIKTALREKKPVYLEIACNIASMPCAAPGPASALFNDEASDEASLNAAVEETLKFIANRDKVAVLVGSKLRAAGAEEAAVKFADALGGAVATMAAAKSFFPEENPHYIGTSWGEVSYPGVEKTMKEADAVIALAPVFNDYSTTGWTDIPDPKKLVLAEPRSVVVNGIRFPSVHLKDYLTRLAQKVSKKTGALDFFKSLNAGELKKAAPADPSAPLVNAEIARQVEALLTPNTTVIAETGDSWFNAQRMKLPNGARVEYEMQWGHIGWSVPAAFGYAVGAPERRNILMVGDGSFQLTAQEVAQMVRLKLPVIIFLINNYGYTIEVMIHDGPYNNIKNWDYAGLMEVFNGNGGYDSGAGKGLKAKTGGELAEAIKVALANTDGPTLIECFIGREDCTEELVKWGKRVAAANSRKPVNK 2wvt A 1.8 BS01 FHN A 1 H66 E87 W88 H135 H136 D229 E288 W316 H32 E53 W54 H101 H102 D195 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Kd=755nM remove_due_to_license_issue Q8A3I4 20092273 1473 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAA 2wvz A 2.4 BS02 KIF A 1 S86 W88 W347 D348 W385 C393 M394 E533 D644 S67 W69 W328 D329 W366 C374 M375 E514 D625 ? 0000224,0005829,0005975,0006516,0030246,0046872 Ki=96uM remove_due_to_license_issue Q8A0N1 20081828 801 KDWTQYVNPLMGSQSTFELSTGNTYPAIARPWGMNFWTPQTGKMGDGWQYTYTANKIRGFKQTHQPSPWINDYGQFSIMPIVGQPVFDEEKRASWFAHKGEVATPYYYKVYLAEHDIVTEMTPTERAVLFRFTFPENDHSYVVVDAFDKGSYIKIIPEENKIIGYTTRNSGGVPENFKNYFIIEFDKPFTYKATVENGNLQENVAEQTTDHAGAIIGFKTRKGEQVNARIASSFISFEQAAANMNELGKDNIEQLAQKGKDAWNQVLGKIEVEGGNLDQYRTFYSCLYRSLLFPRKFYELDANGQPIHYSPYNGQVLPGYMFTDTGFWDTFRCLFPLLNLMYPSVNKEMQEGLINTYLESGFFPEWASPGHRGCMVGNNSASILVDAYMKGVKVDDIKTLYEGLIHGTENVHPEVSSTGRLGYEYYNKLGYVPYDVKINENAARTLEYAYDDWCIYRLAKELKRPKKEISLFAKRAMNYKNLFDKESKLMRGRNEDGTFQSPFSPLKWGDAFTEGNSWHYTWSVFHDPQGLIDLMGGKEMFVTMMDSVFAVPPIFDDSYYGQVIHEIREMTVMNMGNYAHGNQPIQHMIYLYDYAGQPWKAQYWLRQVMDRMYTPGPDGYCGDEDNGQTSAWYVFSALGFYPVCPGTDEYVMGTPLFKKATLHFENGNSLVIDAPNNSTENFYIDSMSFNGADHTKNYLRHEDLFKGGTIKVDMSNRPNLNRGTKEEDMPYSFSKELE 2ww0 A 2.8 BS02 SWA A 1 W347 D348 W385 M394 E533 N601 D644 W328 D329 W366 M375 E514 N582 D625 ? 0000224,0005829,0005975,0006516,0030246,0046872 remove_due_to_license_issue Q8A0N1 20081828 801 KDWTQYVNPLMGSQSTFELSTGNTYPAIARPWGMNFWTPQTGKMGDGWQYTYTANKIRGFKQTHQPSPWINDYGQFSIMPIVGQPVFDEEKRASWFAHKGEVATPYYYKVYLAEHDIVTEMTPTERAVLFRFTFPENDHSYVVVDAFDKGSYIKIIPEENKIIGYTTRNSGGVPENFKNYFIIEFDKPFTYKATVENGNLQENVAEQTTDHAGAIIGFKTRKGEQVNARIASSFISFEQAAANMNELGKDNIEQLAQKGKDAWNQVLGKIEVEGGNLDQYRTFYSCLYRSLLFPRKFYELDANGQPIHYSPYNGQVLPGYMFTDTGFWDTFRCLFPLLNLMYPSVNKEMQEGLINTYLESGFFPEWASPGHRGCMVGNNSASILVDAYMKGVKVDDIKTLYEGLIHGTENVHPEVSSTGRLGYEYYNKLGYVPYDVKINENAARTLEYAYDDWCIYRLAKELKRPKKEISLFAKRAMNYKNLFDKESKLMRGRNEDGTFQSPFSPLKWGDAFTEGNSWHYTWSVFHDPQGLIDLMGGKEMFVTMMDSVFAVPPIFDDSYYGQVIHEIREMTVMNMGNYAHGNQPIQHMIYLYDYAGQPWKAQYWLRQVMDRMYTPGPDGYCGDEDNGQTSAWYVFSALGFYPVCPGTDEYVMGTPLFKKATLHFENGNSLVIDAPNNSTENFYIDSMSFNGADHTKNYLRHEDLFKGGTIKVDMSNRPNLNRGTKEEDMPYSFSKE 2ww2 B 1.9 BS01 SWA B 1 W94 W353 D354 W391 M400 E537 D648 W73 W332 D333 W370 M379 E516 D627 ? 0000224,0005829,0005975,0006516,0030246 Ki=14uM remove_due_to_license_issue Q8A5N9 20081828 900 SKKTVEFVDYVNPLMGTESTFAFSHGNTYPAVAVPWGMNFWSPQTGENGSGWMYTYTDSLMRGFRQTHQPSPWINDYGTFSIMPLAGELKMSHKERLVPFSHQQEKATPYNYSVTFNNGLQTSLSATSRGAVFEVSFPEKEDQYVVVDAYNGGSSITIEPEKRLVKGATRYNNGGVPDNFANYFMMEFSHPVIEYGTYNGDTLLHHQTDVAADYTCAYLKFDVPAGEKLTIRTASSFISPEQAAINFNREVADADVQLISGKAREQWNNYLGRVEAEGGTDEQLRTFYSCLYRTLLFPREFYEFDSQGNPVYYSPYDGNVHDGYMYTDNGFWDTFRAVHPLFTLLYPEVSERVTQSIINAYNESGFMPEWASPGHRGCMIGNNSVSLLVDAWMKGIQTVDAEKALEAMIHQTQARHAEIASVGRDGFEYYDKLGYVPYPEVPEATAKTLEYAYADWCIARFAESLGKQDIADQYYQKAPNYRNLYYPEHGFMWTKDAKGNWRDRFDATEWGGPFTEGSSWHWTWSVFHDPEGLSELMGGHEPMIARLDSMFVAPNTYNYGTYGFVIHEIAEMVALNMGQYAHGNQPVQHAIYLYDYIGQPWKTQYHLRNVMDKLYNSGSKGYCGDEDNGQTSAWYVFSAMGFYPVCPGMPEYAIGSPLFKKVTLHLPEGKNFVVSAADNAADRPYIRKALLNGQEFTRNYLTHDELKQGGELNLSMDSVPNQQRGTQPADFPYSYSK 2wwj A 2.6 BS02 Y28 A 1 I71 N86 Y132 Y177 F185 H188 E190 S196 N198 K206 W208 K241 H276 I64 N79 Y125 Y170 F178 H181 E183 S189 N191 K199 W201 K234 H269 G170 Y177 H188 E190 H276 S288 G163 Y170 H181 E183 H269 S281 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=33000nM O75164 20088513 1354 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEF 2wxd M 1.6 BS01 E18 M 1 Q187 S190 R259 Y330 F331 W457 E464 F473 Q185 S188 R257 Y328 F329 W455 E462 F471 3.2.1.147 0004553,0005773,0005975,0008422,0016798,0019137,0046872 ic50=3.3uM remove_due_to_license_issue P29736 20124710 1501 EITCQENLPFTCGNTDALNSSSFSSDFIFGVASSAYQIEGTIGRGLNIWDGFTHRYPNKSGPDHGNGDTTCDSFSYWQKDIDVLDELNATGYRFSIAWSRIIPRGKRSRGVNEKGIDYYHGLISGLIKKGITPFVTLFHWDLPQTLQDEYEGFLDPQIIDDFKDYADLCFEEFGDSVKYWLTINQLYSVPTRGYGSALDAPGRCSPTVDPSCYAGNSSTEPYIVAHHQLLAHAKVVDLYRKNYTHQGGKIGPTMITRWFLPYNDTDRHSIAATERMKEFFLGWFMGPLTNGTYPQIMIDTVGERLPSFSPEESNLVKGSYDFLGLNYYFTQYAQPSPNPVNSTNHTAMMDAGAKLTYINASGHYIGPLFEKDKADSTDNIYYYPKGIYSVMDYFKNKYYNPLIYVTENGISTPGDENRNQSMLDYTRIDYLCSHLCFLNKVIKEKDVNVKGYLAWALGDNYEFNKGFTVRFGLSYIDWNNVTDRDLKKSGQWYQSFISP 2wxf A 1.9 BS01 039 A 1 F751 M752 P758 L759 W760 I777 Y813 E826 V828 D832 T833 N836 M900 I910 F555 M556 P562 L563 W564 I581 Y617 E630 V632 D636 T637 N640 M704 I714 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=180nM remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxg A 2.0 BS01 ZZN A 1 F751 M752 P758 W760 I777 K779 D787 Y813 I825 V828 D832 T833 M900 I910 D911 F564 M565 P571 W573 I590 K592 D600 Y626 I638 V641 D645 T646 M713 I723 D724 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=0.7nM remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVELLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELEEELREILERSGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFKNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxh A 1.9 BS01 ZZO A 1 F751 M752 P758 W760 I777 K779 D787 Y813 I825 V828 D832 T833 M900 I910 D911 F555 M556 P562 W564 I581 K583 D591 Y617 I629 V632 D636 T637 M704 I714 D715 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxi A 2.8 BS01 S30 A 1 M752 P758 L759 W760 I777 D787 Y813 I825 E826 V827 V828 D832 T833 M900 I910 D911 M549 P555 L556 W557 I574 D584 Y610 I622 E623 V624 V625 D629 T630 M697 I707 D708 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxj A 2.6 BS01 RW3 A 1 M752 W760 I777 D787 Y813 I825 V828 D832 M900 I910 M556 W564 I581 D591 Y617 I629 V632 D636 M704 I714 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxk A 2.9 BS01 RW4 A 1 F751 M752 P758 W760 K779 Y813 V827 V828 I910 D911 F564 M565 P571 W573 K592 Y626 V640 V641 I723 D724 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVELLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELEEELREILERSGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFKNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxl A 1.99 BS01 ZS4 A 1 M752 I777 K779 D787 Y813 I825 E826 V828 T833 I910 D911 M557 I582 K584 D592 Y618 I630 E631 V633 T638 I715 D716 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=4.6nM remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELQLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxm A 2.8 BS01 ZZM A 1 W760 I777 K779 I825 V828 M900 I910 D911 W564 I581 K583 I629 V632 M704 I714 D715 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxn A 2.6 BS01 DLN A 1 W760 D787 Y813 I825 V828 M900 D911 W564 D591 Y617 I629 V632 M704 D715 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxo A 2.49 BS01 ZZP A 1 M752 S754 W760 I777 K779 Y813 E826 V828 M900 I910 D911 M556 S558 W564 I581 K583 Y617 E630 V632 M704 I714 D715 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=90nM remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxp A 2.3 BS01 GD9 A 1 M752 D753 K779 D787 Y813 I825 E826 V828 M900 I910 D911 M556 D557 K583 D591 Y617 I629 E630 V632 M704 I714 D715 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=3nM remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxq A 2.7 BS01 ZZQ A 1 M752 D753 W760 E826 V827 V828 M900 I910 M556 D557 W564 E630 V631 V632 M704 I714 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 20081827 1500 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2wxv C 2.6 BS01 WXV C 1 I10 Y15 A31 K33 F80 L83 Q85 D86 K89 L134 D145 I11 Y16 A32 K34 F81 L84 Q86 D87 K90 L135 D146 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 20141146 1299 DMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2wyf A 2.4 BS01 MBG I 1 H50 Q53 H50 Q53 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Kd=70000nM Q05097 20410292 1 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 2wyf A 2.4 BS02 GLA I 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 20410292 2 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 2wyg A 1.88 BS01 461 A 1 E97 Y99 F174 D189 A190 Q192 V213 W215 G216 G226 I227 Y228 E77 Y79 F156 D173 A174 Q176 V197 W199 G200 G210 I211 Y212 H57 D102 Q192 G193 D194 S195 G196 H42 D82 Q176 G177 D178 S179 G180 3.4.21.6 0004252,0006508 Ki=2nM remove_due_to_license_issue Ki=2nM P00742 20006499 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2wyj A 2.38 BS01 898 A 1 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G219 G226 I227 Y228 T81 Y82 F159 D176 A177 Q179 V200 W202 G203 G205 G213 I214 Y215 H57 D102 Q192 G193 D194 S195 G196 H42 D85 Q179 G180 D181 S182 G183 3.4.21.6 0004252,0006508 Ki=1nM remove_due_to_license_issue Ki=0.8nM P00742 20006499 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2wyn B 2.1 BS01 LG9 B 1 F153 W159 D160 G310 D312 W447 Y512 F518 W520 F118 W124 D125 G275 D277 W412 Y469 F475 W477 3.2.1.28 0004555,0005975,0005991,0005993,0006974,0016798,0030288,0042597,0071474 remove_due_to_license_issue P13482 20461849 1547 ETPVTPQPPDILLGPLFNDVQNAKLFPDQKTFADAVPNSDPLMILADYRMQQNQSGFDLRHFVNVNFTLPKYVPPEGQSLREHIDGLWPVLTRSTENTEKWDSLLPLPEPYVVPGGRFREVYYWDSYFTMLGLAESGHWDKVADMVANFAHEIDTYGHIPNGNRSYYLSRSQPPFFALMVELLAQHEGDAALKQYLPQMQKEYAYWMDGVENLQAGQQEKRVVKLQDGTLLNRYWDDRDTPRPESWVEDIATAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDNPQQLNTLRTTSIVPVDLNSLMFKMEKILARASKAAGDNAMANQYETLANARQKGIEKYLWNDQQGWYADYDLKSHKVRNQLTAAALFPLYVNAAAKDRANKMATATKTHLLQPGGLNTTSVKSGQQWDAPNGWAPLQWVATEGLQNYGQKEVAMDISWHFLTNVQHTYDREKKLVEKYDVSTTYPLQDGFGWTNGVTLKMLDLICPKEQPCDNVPATR 2wyn B 2.1 BS02 GLC B 1 R152 Y157 N196 Y202 R205 E279 R117 Y122 N161 Y167 R170 E244 3.2.1.28 0004555,0005975,0005991,0005993,0006974,0016798,0030288,0042597,0071474 remove_due_to_license_issue P13482 20461849 1548 ETPVTPQPPDILLGPLFNDVQNAKLFPDQKTFADAVPNSDPLMILADYRMQQNQSGFDLRHFVNVNFTLPKYVPPEGQSLREHIDGLWPVLTRSTENTEKWDSLLPLPEPYVVPGGRFREVYYWDSYFTMLGLAESGHWDKVADMVANFAHEIDTYGHIPNGNRSYYLSRSQPPFFALMVELLAQHEGDAALKQYLPQMQKEYAYWMDGVENLQAGQQEKRVVKLQDGTLLNRYWDDRDTPRPESWVEDIATAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDNPQQLNTLRTTSIVPVDLNSLMFKMEKILARASKAAGDNAMANQYETLANARQKGIEKYLWNDQQGWYADYDLKSHKVRNQLTAAALFPLYVNAAAKDRANKMATATKTHLLQPGGLNTTSVKSGQQWDAPNGWAPLQWVATEGLQNYGQKEVAMDISWHFLTNVQHTYDREKKLVEKYDVSTTYPLQDGFGWTNGVTLKMLDLICPKEQPCDNVPATR 2wzf A 2.1 BS01 UDP A 1 I138 W139 F140 P225 A226 S229 D246 N514 G517 L518 S519 W520 I130 W131 F132 P217 A218 S221 D238 N506 G509 L510 S511 W512 ? 0000166,0046872 remove_due_to_license_issue Q5ZVS2 20030628 1525 LSKLRMRFFSALNHTSEIDLQVLFNDLKSILTLDSIEHLKEGSVAYAIIQELLKQDDAQNKIQSFLHGAIKNVIHPGVIKGLTPDEINWNVAKAYPKYYEHEEFPDVTFGGFKVRDSNEFKFKTNIQTSIWFSIKPDLFMPSKQQEALKRRREQYPGCEIRLIYSSSLLNAEANRQMKAFARKQNISLIDIDSVKTDSPLYPLLKAELAHLGKGGNPAAASDLCRWIPELFNEGFYVDIDLPVDSSKIVEGHQITGGVPIMLNMGSIISEPIAPHHRRQEAVCMNTDIIAYSNDKRTQKMMDTVARYLKNIYDDPYTALKDTPLAQTAFFNKCQEERKSIFDLRKGLQDAFRSDSLLQLYDFLGADKFKEVFKLKEAQSKYINEHISEFSEKDLLLNLISDKPSEISQHTLDFVKAKAMYIDIAKEHYSAFYKPLVEEISGPGAIYNALGGAGSFTTTHRRLTGPMLPTTPPRVLQVFCDAHDKGPFVSDNIARWQTNVRDLGVLNREGLSWLPS 2wzm A 1.64 BS01 NA7 A 1 Y195 G196 P197 L198 G199 V200 G201 L204 A221 I236 R238 S239 R244 N248 R274 Y186 G187 P188 L189 G190 V191 G192 L195 A212 I227 R229 S230 R235 N239 R265 D53 Y58 K83 H116 D44 Y49 K74 H107 1.1.1.- 0004033,0016491,0016616,0044281 remove_due_to_license_issue A0QV09 20188740 1284 AIPTVTLNDDNTLPVVGIGVGELSDSEAERSVSAALEAGYRLIDTAAAYGNEAAVGRAIAASGIPRDEIYVTTKLATPDQGFTSSQAAARASLERLGLDYVDLYLIHWPGGDTSKYVDSWGGLMKVKEDGIARSIGVCNFGAEDLETIVSLTYFTPAVNQIELHPLLNQAALREVNAGYNIVTEAYGPLGVGRLLDHPAVTAIAEAHGRTAAQVLLRWSIQLGNVVISRSANPERIASNLDVFGFELTADEMETLNGLDDGTRFRPDPATYTGS 2wzs A 2.25 BS02 MVL A 1 S86 W88 W347 D348 W385 C393 M394 E533 D644 S67 W69 W328 D329 W366 C374 M375 E514 D625 ? 0000224,0005829,0005975,0006516,0030246,0046872 Ki=140uM remove_due_to_license_issue Q8A0N1 20081828 801 KDWTQYVNPLMGSQSTFELSTGNTYPAIARPWGMNFWTPQTGKMGDGWQYTYTANKIRGFKQTHQPSPWINDYGQFSIMPIVGQPVFDEEKRASWFAHKGEVATPYYYKVYLAEHDIVTEMTPTERAVLFRFTFPENDHSYVVVDAFDKGSYIKIIPEENKIIGYTTRNSGGVPENFKNYFIIEFDKPFTYKATVENGNLQENVAEQTTDHAGAIIGFKTRKGEQVNARIASSFISFEQAAANMNELGKDNIEQLAQKGKDAWNQVLGKIEVEGGNLDQYRTFYSCLYRSLLFPRKFYELDANGQPIHYSPYNGQVLPGYMFTDTGFWDTFRCLFPLLNLMYPSVNKEMQEGLINTYLESGFFPEWASPGHRGCMVGNNSASILVDAYMKGVKVDDIKTLYEGLIHGTENVHPEVSSTGRLGYEYYNKLGYVPYDVKINENAARTLEYAYDDWCIYRLAKELKRPKKEISLFAKRAMNYKNLFDKESKLMRGRNEDGTFQSPFSPLKWGDAFTEGNSWHYTWSVFHDPQGLIDLMGGKEMFVTMMDSVFAVPPIFDDSYYGQVIHEIREMTVMNMGNYAHGNQPIQHMIYLYDYAGQPWKAQYWLRQVMDRMYTPGPDGYCGDEDNGQTSAWYVFSALGFYPVCPGTDEYVMGTPLFKKATLHFENGNSLVIDAPNNSTENFYIDSMSFNGADHTKNYLRHEDLFKGGTIKVDMSNRPNLNRGTKEEDMPYSFSKE 2wzx A 1.4 BS01 ZX0 A 1 S90 Q146 Y177 N179 Y249 T343 G344 S345 S63 Q119 Y150 N152 Y222 T316 G317 S318 S90 K93 Y177 E299 K342 S345 S63 K66 Y150 E272 K315 S318 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 20044254 600 EAPADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLEQ 2wzy F 2.51 BS01 SQX F 1 Y93 K143 W147 V148 Y188 Y195 Y94 K144 W148 V149 Y189 Y196 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 20224036 301 LHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2wzy F 2.51 BS02 SQX G 1 Y55 I118 S167 Y56 I119 S168 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 20224036 301 LHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2wzy J 2.51 BS01 SQX F 1 Y55 I118 S167 Y59 I122 S171 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 20224036 301 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wzy J 2.51 BS02 SQX J 1 Y93 K143 W147 V148 Y188 C190 Y195 Y97 K147 W151 V152 Y192 C194 Y199 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 20224036 301 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2wzz A 1.57 BS01 ZX1 A 1 S90 Q146 Y177 N179 T343 G344 S345 S62 Q118 Y149 N151 T315 G316 S317 S90 K93 Y177 E299 K342 S345 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 20044254 600 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLE 2x00 A 2.4 BS01 GYN A 1 Y93 K143 W147 Y188 C190 Y195 Y101 K151 W155 Y196 C198 Y203 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.0047nM remove_due_to_license_issue Q8WSF8 20224036 301 YKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2x00 A 2.4 BS02 GYN B 1 Y55 I118 Y63 I126 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.0047nM remove_due_to_license_issue Q8WSF8 20224036 301 YKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2x00 E 2.4 BS01 GYN A 1 Y55 I118 Y59 I122 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.0047nM remove_due_to_license_issue Q8WSF8 20224036 301 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2x00 E 2.4 BS02 GYN E 1 Y93 K143 W147 Y188 C190 Y195 Y97 K147 W151 Y192 C194 Y199 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=0.0047nM remove_due_to_license_issue Q8WSF8 20224036 301 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 2x09 A 2.4 BS01 X09 A 1 D203 W204 E394 C419 D469 M512 Y516 E541 W642 W653 D155 W156 E346 C371 D421 M464 Y468 E493 W594 W605 3.2.1.165 0004553,0005975,0030246 Ki=175uM remove_due_to_license_issue Q56F26 19795054 1900 GNATPIPGYVIQSSAQVSDDSAVSKPGFPTSGWYPVSSRSTVYAGLLQNGKYADPFYSTNMQNVPAAQFSVPWWYRTDLNVDDTSSRTYLDFSGVLSKADVWVNGTKVATKDQVNGAYTRHDLDITAQVHTGVNSVAFKVYPNDPNRDLSMGWIDWAQTPPDQNMGIVRDVLVRRSGAVALRSAHVIQKLNSALDHADLTVKADVRNDSANAVQTTVAGTVAGKPISQTVSLAAKERKTVTFPLVGLDRPNVWWPAGMGGQHRYDLDLTASVGGTPSDAAKSKFGVRDVKATLNSSGGRQYSVNGKPLLIRGGGYTPDLFLRWNETAAADKLKYVLNLGLNTVRLEGHIEPDEFFDIADDLGVLTMPGWECCDKWEGQVNGEEKGEPWVESDYPIAKASMFSEAERLRDHPSVISFHIGSDFAPDRRIEQGYLDAMKAADFLLPVIPAASARPSPITGASGMKMNGPYDYVPPVYWYDKSQKDRGGAWSFNSETSAGVDIPTMDTLKRMMSASELDTMWKNPSAKQYHRSSSDTFGNLKLFGDALTKRYGASANLNDFVRKAQLSQYENVRAEFESHSRNYTDSTNPSTGLIYWMLNSPWTSLHWQLFDAYMDQNGAYYGAKKANEPLHIQYSHDNRSVVVINQTSNAVSGLTATTKLYNLDGTEKYSNTKTGLSVGALGAKATAVTVPAVSGLSTTYLAKNVLTDSSGKEVSRNVYWLSTKADTLNWGGSDWYYTPQSAFADLSGLNNLGQSAVGATANSVAGADGTTTTTVTLKNTSGGRLPAFYVDSKVVDSAGKPVLPVEWNDNAVSLWPGETTTLTAKYRTADLKGSKPSVRISGWNTGTQTVPA 2x0y A 2.25 BS01 X0T A 1 G187 D297 V331 Y335 W394 N396 D401 G147 D257 V291 Y295 W354 N356 D361 3.2.1.169 Ki=25uM remove_due_to_license_issue Q0TR53 20026047 1625 VLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYNRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2x0y B 2.25 BS01 X0T B 1 G187 K218 D297 V331 Y335 W394 N396 D401 G148 K179 D258 V292 Y296 W355 N357 D362 3.2.1.169 Ki=25uM remove_due_to_license_issue Q0TR53 20026047 1625 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITVPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYNRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2x24 A 2.4 BS01 X24 A 1 R483 F485 L554 E555 E557 G558 E561 I562 R457 F459 L528 E529 E531 G532 E535 I536 0003989,0016874 remove_due_to_license_issue 21515056 1715 LQAKRFQAQSLGTTYVYDFPEMFRQALFKMWPSPDKYPKDILTYTELVLDPQGQLVEMNRLPGGNEVGMVAFKMTLKTLEYPEGRDIILISNDITFRIGSFGPGEDLLYLRASELARAEGIPRVYLAANSGARIGLAEEIKHMFQVAWVDPEDPHKGIKYLYLTPQDYTRISSLNSVHCKHVEEDGESRYVITDIIGKEEGLGVENLRGSGMIAGETSQDYDEIVTISMVSCRALGIGAYLVRLGQRVIQVENSHIILTGATALNKVLGRDVYTSNNQLGGVQIMHHNGVSHVTVPDDFEGVCTILEWLSYMPKDNRSPVPVVTPKDPIDREIEFQPSRGPYDPRWLLAGRPHPTLKGSWQSGFFDQGSFKEIMVPWAQTVVTGRARLGGIPVGVIAAETRTVELVVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRKYRQPVLIYIPPYAEVRGGSWAVMDTSINPLCIEMYADRESRASVLEPEGTVEIKYQKKDLVKTIRRLDPISKQLKAREDLLLPMYHQVALHFADLHDTAGRMLEKGVIYDILEWKTARSFLYWRLRRLLLESQVKQVQSMLRRWFVETEGAVKAYLWDNNQTVVQWLEAHG 2x24 A 2.4 BS02 X24 B 1 T285 A289 L290 K292 V293 L294 T259 A263 L264 K266 V267 L268 0003989,0016874 remove_due_to_license_issue 21515056 1714 LQAKRFQAQSLGTTYVYDFPEMFRQALFKMWPSPDKYPKDILTYTELVLDPQGQLVEMNRLPGGNEVGMVAFKMTLKTLEYPEGRDIILISNDITFRIGSFGPGEDLLYLRASELARAEGIPRVYLAANSGARIGLAEEIKHMFQVAWVDPEDPHKGIKYLYLTPQDYTRISSLNSVHCKHVEEDGESRYVITDIIGKEEGLGVENLRGSGMIAGETSQDYDEIVTISMVSCRALGIGAYLVRLGQRVIQVENSHIILTGATALNKVLGRDVYTSNNQLGGVQIMHHNGVSHVTVPDDFEGVCTILEWLSYMPKDNRSPVPVVTPKDPIDREIEFQPSRGPYDPRWLLAGRPHPTLKGSWQSGFFDQGSFKEIMVPWAQTVVTGRARLGGIPVGVIAAETRTVELVVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRKYRQPVLIYIPPYAEVRGGSWAVMDTSINPLCIEMYADRESRASVLEPEGTVEIKYQKKDLVKTIRRLDPISKQLKAREDLLLPMYHQVALHFADLHDTAGRMLEKGVIYDILEWKTARSFLYWRLRRLLLESQVKQVQSMLRRWFVETEGAVKAYLWDNNQTVVQWLEAHG 2x24 B 2.4 BS01 X24 B 1 R483 F485 S486 G487 L554 E555 E557 G558 R458 F460 S461 G462 L529 E530 E532 G533 0003989,0016874 remove_due_to_license_issue 21515056 1714 LLQAKRFQAQSLGTTYVYDFPEMFRQALFKMWPSPDKYPKDILTYTELVLDPQGQLVEMNRLPGGNEVGMVAFKMTLKTLEYPEGRDIILISNDITFRIGSFGPGEDLLYLRASELARAEGIPRVYLAANSGARIGLAEEIKHMFQVAWVDPEDPHKGIKYLYLTPQDYTRISSLNSVHCKHVEEDGESRYVITDIIGKEEGLGVENLRGSGMIAGETSQDYDEIVTISMVSCRALGIGAYLVRLGQRVIQVENSHIILTGATALNKVLGRDVYTSNNQLGGVQIMHHNGVSHVTVPDDFEGVCTILEWLSYMPKDNRSPVPVVTPKDPIDREIEFQPSRGPYDPRWLLAGRPHPTLKGSWQSGFFDQGSFKEIMVPWAQTVVTGRARLGGIPVGVIAAETRTVELVVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRKYRQPVLIYIPPYAEVRGGSWAVMDTSINPLCIEMYADRESRASVLEPEGTVEIKYQKKDLVKTIRRLDPISKQLKAREDLLLPMYHQVALHFADLHDTAGRMLEKGVIYDILEWKTARSFLYWRLRRLLLESQVKQEVLRACPELSHMHVQSMLRRWFVETEGAVKAYLWDNNQTVVQWLEAH 2x2k A 2.6 BS01 X2K A 1 L730 V738 A756 Y806 A807 G810 L881 D892 L28 V36 A54 Y104 A105 G108 L158 D169 D850 D874 A876 R878 N879 D892 D127 D151 A153 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=300nM P07949 20117004 2017 GPLSLSVDAFKIPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVRALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKRR 2x2l A 2.0 BS01 X2L A 1 L730 V738 A756 Y806 A807 G810 L881 D892 L29 V37 A55 Y105 A106 G109 L159 D170 D850 D874 A876 R878 N879 D892 D128 D152 A154 R156 N157 D170 2.7.10.1 0004672,0004713,0005524,0006468 ic50=5.3uM remove_due_to_license_issue IC50=5300nM P07949 20117004 2015 GPLSLSVDAFKILPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVRALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMV 2x2m A 2.5 BS01 X2M A 1 L730 A756 K758 E805 Y806 A807 G810 L881 S891 L30 A54 K56 E103 Y104 A105 G108 L155 S165 D850 D874 A876 R878 N879 D892 D124 D148 A150 R152 N153 D166 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.17uM remove_due_to_license_issue IC50=170nM P07949 20117004 2016 GPLSLSVDAFKILDPKWEFPRKNLVLGKTLGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKRR 2x2r A 2.2 BS02 X2O A 1 E116 G117 E118 R119 P137 L214 R221 E100 G101 E102 R103 P121 L198 R205 ? 0003777,0005524,0007018,0008017 Ki=76.2nM remove_due_to_license_issue P52732 21344920 1367 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEV 2x38 A 2.2 BS01 IC8 A 1 M752 P758 W760 I777 E826 V828 D832 T833 M900 I910 M556 P562 W564 I581 E630 V632 D636 T637 M704 I714 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=130nM remove_due_to_license_issue O35904 20081827 2028 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 2x39 A 1.93 BS02 X39 A 1 G161 G164 V166 A179 K181 M229 E230 A232 E236 M282 D293 F439 G16 G19 V21 A34 K36 M84 E85 A87 E91 M137 D148 F294 D275 K277 N280 D293 T313 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 ic50=2.2nM remove_due_to_license_issue IC50=2.2nM P31751 20151677 1480 KVTMNDFDYLKLLGKGTFGKVILVREKATGRYYAMKILRKEVIIAKDEVAHTVTESRVLQNTRHPFLTALKYAFQTHDRLCFVMEYANGGELFFHLSRERVFTEERARFYGAEIVSALEYLHSRDVVYRDIKLENLMLDKDGHIKITDFGLCKEGISDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHERLFELILMEEIRFPRTLSPEAKSLLAGLLKKDPKQRLGGGPSDAKEVMEHRFFLSINWQDVVQKKLLPPFKPQVTSEVDTRYFDDEFTAQSITQEMFEDFDYIADW 2x52 A 1.7 BS01 GYT A 1 S62 Y64 H66 E72 Y73 S62 Y64 H66 E72 Y73 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1172 ERCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 A 1.7 BS02 GYT A 2 S19 Y23 D29 Y30 S19 Y23 D29 Y30 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1173 ERCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 A 1.7 BS03 GYT B 1 D86 S105 W107 Y109 S114 E115 F116 D86 S105 W107 Y109 S114 E115 F116 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1172 ERCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 A 1.7 BS04 GYT B 2 D129 S148 W150 S152 P157 Y159 D129 S148 W150 S152 P157 Y159 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1173 ERCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 B 1.7 BS01 GYT A 1 D86 S105 W107 Y109 S114 E115 F116 D85 S104 W106 Y108 S113 E114 F115 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1172 RCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 B 1.7 BS02 GYT A 2 D129 S148 W150 S152 P157 Y159 D128 S147 W149 S151 P156 Y158 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1173 RCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 B 1.7 BS03 GYT B 1 S62 Y64 H66 A71 E72 Y73 S61 Y63 H65 A70 E71 Y72 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1172 RCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x52 B 1.7 BS04 GYT B 2 S19 Y21 Y23 G28 D29 Y30 S18 Y20 Y22 G27 D28 Y29 ? 0008061,0030246 remove_due_to_license_issue P10969 20527753 1173 RCGEQGSGMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGKTCPNNHCCSQYGHCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGYCGLGSEFCGEGCQNGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 2x5o A 1.46 BS01 VSV A 1 D35 T36 R37 S71 P72 G73 F161 H183 K348 A414 S415 L416 N421 F422 D35 T36 R37 S71 P72 G73 F161 H183 K348 A414 S415 L416 N421 F422 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=85uM remove_due_to_license_issue P14900 20804196 500 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRGADERCVSFGVNMGDYHLNHQQGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2x6d A 2.796 BS01 X6D A 1 L139 G140 K141 G145 N146 A160 Y212 A213 G216 R220 L14 G15 K16 G20 N21 A35 Y83 A84 G87 R91 D256 K258 E260 N261 D274 T292 D127 K129 E131 N132 D145 T159 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=12nM O14965 20565112 1391 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2x6e A 3.35 BS01 YM4 A 1 L139 G140 K141 G142 N146 V147 A160 Y212 A213 P214 G216 R220 L14 G15 K16 G17 N21 V22 A35 Y87 A88 P89 G91 R95 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=15nM O14965 20565112 1389 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHTLDYLPPEMIEHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2x6f A 3.3 BS01 3MA A 1 I696 Y746 V747 S749 I822 I291 Y341 V342 S344 I417 2.7.1.137 0016301,0016303,0046854 remove_due_to_license_issue Q9W1M7 20339072 1949 ASIRDQLHTIVYRYPPTYVLSSEEQDLVWKFRFYLSSHKKALTKFLKCINWKLEDEVTQALWMLANWAPMDVEDALELLSPTFTHPQVRKYAVSRLAQAPDEDLLLYLLQLVQALKYEDPRHIVHLHGCIFPNLCTFLIQRACTNATLANYFYWYLSIEVEEQDERAHDMYAMVLKMFLKVLENGNFNLRGIFYNLRKQRRFIDELVKLVKLVAKEPGNRNKKTEKFQKLLAEQDMFKVNFTNFEPIPFPLDPEIYITKIVPMRTSLFKSALMPAKLTFVTSIAHHEYAAIFKHGDDLRQDQLILQMITLMDKLLRRENLDLKLTPYKVLATSSKHGFLQYVDSCTVAEVLAREGNIHNFFRKHHPCDNGPYGISAEVMDTYIKSCAGYCVITYLLGVGDRHLDNLLLTTNGKLFHIDFGYILGRDPKPMPPPMKLSKEMVEAMGGISSEHHHEFRKQCYTAYLHLRRHANVMLNLFSLMVDATVPDIALEPDKAVKKVEENLQLGLTDEEAVQHLQSLLDVSITAVMPALVEQIHRFTQYWR 2x6i A 3.4 BS01 090 A 1 K674 I696 K698 D706 Y732 Y746 V747 S749 L812 I822 D823 K272 I294 K296 D304 Y330 Y344 V345 S347 L410 I420 D421 2.7.1.137 0016301,0016303,0046854 remove_due_to_license_issue Q9W1M7 20339072 1949 ASIRDQLHTIVYRYPPTYVLSSEEQDLVWKFRFYLSSHKKALTKFLKCINWKLEDEVTQALWMLANWAPMDVEDALELLSPTFTHPQVRKYAVSRLAQAPDEDLLLYLLQLVQALKYEDPRHIVHLHGCIFPANLCTFLIQRACTNATLANYFYWYLSIEVEERKQDERAHDMYAMVLKMFLKVLENGNFNLRGIFYNLRKQRRFIDELVKLVKLVAKEPGNRNKKTEKFQKLLAEQDMFKVNFTNFEPIPFPLDPEIYITKIVPMRTSLFKSALMPAKLTFVTSIAHHEYAAIFKHGDDLRQDQLILQMITLMDKLLRRENLDLKLTPYKVLATSSKHGFLQYVDSCTVAEVLAREGNIHNFFRKHHPCDNGPYGISAEVMDTYIKSCAGYCVITYLLGVGDRHLDNLLLTTNGKLFHIDFGYILGRDPKPMPPPMKLSKEMVEAMGGISSEHHHEFRKQCYTAYLHLRRHANVMLNLFSLMVDATVPDIALEPDKAVKKVEENLQLGLTDEEAVQHLQSLLDVSITAVMPALVEQIHRFTQYWR 2x6j A 3.5 BS01 093 A 1 I696 K698 L744 Y746 V747 S749 I822 D823 I293 K295 L341 Y343 V344 S346 I419 D420 2.7.1.137 0016301,0016303,0046854 remove_due_to_license_issue Q9W1M7 20339072 1949 ASIRDQLHTIVYRYPPTYVLSSEEQDLVWKFRFYLSSHKKALTKFLKCINWKLEDEVTQALWMLANWAPMDVEDALELLSPTFTHPQVRKYAVSRLAQAPDEDLLLYLLQLVQALKYEDPRHIVHLHGCIFPANLCTFLIQRACTNATLANYFYWYLSIEVEEKQDERAHDMYAMVLKMFLKVLENGNFNLRGIFYNLRKQRRFIDELVKLVKLVAKEPGNRNKKTEKFQKLLAEQDMFKVNFTNFEPIPFPLDPEIYITKIVPMRTSLFKSALMPAKLTFVTSIAHHEYAAIFKHGDDLRQDQLILQMITLMDKLLRRENLDLKLTPYKVLATSSKHGFLQYVDSCTVAEVLAREGNIHNFFRKHHPCDNGPYGISAEVMDTYIKSCAGYCVITYLLGVGDRHLDNLLLTTNGKLFHIDFGYILGRDPKPMPPPMKLSKEMVEAMGGISSEHHHEFRKQCYTAYLHLRRHANVMLNLFSLMVDATVPDIALEPDKAVKKVEENLQLGLTDEEAVQHLQSLLDVSITAVMPALVEQIHRFTQYWR 2x6k A 3.5 BS01 X6K A 1 K674 I696 K698 D706 L744 V747 I822 D823 K276 I298 K300 D308 L346 V349 I424 D425 2.7.1.137 0016301,0016303,0046854 remove_due_to_license_issue Q9W1M7 20339072 1951 ASIRDQLHTIVYRYPPTYVLSSEEQDLVWKFRFYLSSHKKALTKFLKCINWKLEDEVTQALWMLANWAPMDVEDALELLSPTFTHPQVRKYAVSRLAQAPDEDLLLYLLQLVQALKYEDPRHIVHLHGCIFPANLCTFLIQRACTNATLANYFYWYLSIEVEEVESVRKQDERAHDMYAMVLKMFLKVLENGNFNLRGIFYNLRKQRRFIDELVKLVKLVAKEPGNRNKKTEKFQKLLAEQDMFKVNFTNFEPIPFPLDPEIYITKIVPMRTSLFKSALMPAKLTFVTSIAHHEYAAIFKHGDDLRQDQLILQMITLMDKLLRRENLDLKLTPYKVLATSSKHGFLQYVDSCTVAEVLAREGNIHNFFRKHHPCDNGPYGISAEVMDTYIKSCAGYCVITYLLGVGDRHLDNLLLTTNGKLFHIDFGYILGRDPKPMPPPMKLSKEMVEAMGGISSEHHHEFRKQCYTAYLHLRRHANVMLNLFSLMVDATVPDIALEPDKAVKKVEENLQLGLTDEEAVQHLQSLLDVSITAVMPALVEQIHRFTQYWR 2x6v A 2.2 BS01 dna C 0 S175 T215 P231 F232 K234 G235 S123 T154 P170 F171 K173 G174 ? 0000978,0003700,0005634,0006355,0045893 remove_due_to_license_issue Q99593 20450920 1 ~ 11 GIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADTAFCTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFRG 2x6v A 2.2 BS02 dna D 0 R81 R82 K159 Y217 T223 K226 I227 N230 F232 F236 R29 R30 K107 Y156 T162 K165 I166 N169 F171 F175 ? 0000978,0003700,0005634,0006355,0045893 remove_due_to_license_issue Q99593 20450920 12 ~ 22 GIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADTAFCTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFRG 2x7c A 1.9 BS02 KZ9 A 1 E116 E118 R119 D130 A133 I136 P137 Y211 E99 E101 R102 D113 A116 I119 P120 Y194 ? 0003777,0005524,0007018,0008017 ic50=2uM remove_due_to_license_issue IC50=2000nM P52732 20597485 1365 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 2x7d A 2.3 BS03 EGB A 1 E116 E118 R119 W127 D130 A133 I136 P137 Y211 A218 E100 E102 R103 W111 D114 A117 I120 P121 Y195 A202 ? 0003777,0005524,0007018,0008017 ic50=200nM remove_due_to_license_issue P52732 20597485 1369 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 2x7o A 3.7 BS01 ZOP A 1 I211 G212 V219 K232 L260 L278 S280 H283 H285 G286 R294 L340 I41 G42 V49 K62 L90 L108 S110 H113 H115 G116 R124 L170 D333 K335 N338 D351 T375 D163 K165 N168 D181 T205 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue EC50=105nM, IC50=34nM P36897 20919678 600 ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG 2x7s A 1.64 BS01 WZC A 1 H94 H119 L197 T198 T199 H90 H115 L193 T194 T195 H64 H94 H96 E106 H119 T198 H61 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1660nM remove_due_to_license_issue IC50=526nM, Ki=10330nM P00918 20297840 1263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2x7s A 1.64 BS02 WZC A 2 N67 I91 Q92 D129 F130 G131 N64 I87 Q88 D125 F126 G127 H64 H94 H96 E106 H119 T198 H61 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1660nM remove_due_to_license_issue IC50=526nM, Ki=10330nM P00918 20297840 1264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2x7t A 1.89 BS01 WZB A 1 H94 H119 F130 L197 T198 T199 P201 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=232nM remove_due_to_license_issue Ki=232nM, IC50=290nM P00918 20297840 1261 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2x7u A 2.12 BS03 WZA A 1 Q92 H94 H119 V121 F130 V134 L197 T198 T199 P200 P201 Q89 H91 H116 V118 F127 V131 L194 T195 T196 P197 P198 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5340nM remove_due_to_license_issue P00918 20297840 1263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 2x81 A 2.91 BS01 ZZL A 1 R137 L139 G140 V147 A160 L210 Y212 A213 G216 N261 L263 A273 R11 L13 G14 V18 A31 L81 Y83 A84 G87 N132 L134 A144 D256 K258 E260 N261 T292 D127 K129 E131 N132 T146 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=34nM, Kd=6.5nM O14965 20426425 1389 QWALEDFEIGRPLGFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2x8d A 1.9 BS01 X8D A 1 L15 A36 E85 C87 L137 S280 L14 A35 E84 C86 L136 S279 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.8uM remove_due_to_license_issue IC50=800nM O14757 20673630 1282 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2x8e A 2.5 BS01 X8E A 1 L15 V23 Y86 C87 G90 L137 L7 V15 Y75 C76 G79 L126 D130 K132 E134 N135 D148 T170 D119 K121 E123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.014uM remove_due_to_license_issue IC50=14nM O14757 20673630 1271 WDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2x8i A 1.92 BS01 X8I A 1 L15 G16 E17 A36 E85 Y86 E91 E134 L137 L14 G15 E16 A35 E77 Y78 E83 E126 L129 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.19uM remove_due_to_license_issue O14757 20673630 1270 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2x8z A 1.98 BS01 X8Z A 1 Q265 H337 H367 E368 F441 K495 H497 Y504 Y507 Q249 H321 H351 E352 F425 K479 H481 Y488 Y491 H337 A338 H367 E368 H371 E395 H497 Y507 H321 A322 H351 E352 H355 E379 H481 Y491 3.4.15.1 0006508,0008237,0008241,0016020 Ki=11nM remove_due_to_license_issue Q10714 20488190 1615 ALVKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 2x91 A 1.98 BS01 LPR A 1 Q265 H337 A338 H367 E368 E395 K495 H497 V502 Y504 Y507 Q246 H318 A319 H348 E349 E376 K476 H478 V483 Y485 Y488 H337 A338 H367 E368 H371 E395 H497 Y507 H318 A319 H348 E349 H352 E376 H478 Y488 3.4.15.1 0006508,0008237,0008241,0016020 Ki=180nM remove_due_to_license_issue Q10714 20488190 1615 KEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 2x95 A 1.96 BS02 X95 A 1 Q265 H337 A338 T364 H367 E368 H371 E395 D399 K495 H497 V502 Y504 Y507 F511 Q249 H321 A322 T348 H351 E352 H355 E379 D383 K479 H481 V486 Y488 Y491 F495 H337 A338 H367 E368 H371 E395 H497 Y507 H321 A322 H351 E352 H355 E379 H481 Y491 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Q10714 20488190 1623 ALVKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 2x96 A 1.85 BS01 RX3 A 1 Q266 H337 A338 S339 A340 H367 E368 H371 F375 H394 E395 D399 F441 K495 H497 V502 Y504 Y507 Q250 H321 A322 S323 A324 H351 E352 H355 F359 H378 E379 D383 F425 K479 H481 V486 Y488 Y491 H337 A338 H367 E368 H371 E395 H497 Y507 H321 A322 H351 E352 H355 E379 H481 Y491 3.4.15.1 0006508,0008237,0008241,0016020 Ki=94uM remove_due_to_license_issue Q10714 20488190 1615 ALVKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 2x97 A 1.85 BS01 RX4 A 1 Q265 H337 A338 S339 A340 H367 E368 H371 F375 E395 F441 K495 Y496 H497 V502 Y504 Y507 Q249 H321 A322 S323 A324 H351 E352 H355 F359 E379 F425 K479 Y480 H481 V486 Y488 Y491 H337 A338 H367 E368 H371 E395 H497 Y507 H321 A322 H351 E352 H355 E379 H481 Y491 3.4.15.1 0006508,0008237,0008241,0016020 Ki=2200nM remove_due_to_license_issue Q10714 20488190 1615 ALVKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 2x9e A 3.1 BS01 SVE A 1 K529 I531 S537 V539 Q541 K553 C604 G605 N606 I607 S611 N652 L654 D664 Q794 K15 I17 S23 V25 Q27 K39 C90 G91 N92 I93 S97 N138 L140 D150 Q253 D647 K649 N652 D664 T686 D133 K135 N138 D150 T157 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=182nM P33981 21159646 1796 NECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 2x9f A 1.75 BS01 X9F A 1 I621 A645 K647 E664 T693 F695 M696 E697 G699 L747 S757 D758 I14 A38 K40 E54 T83 F85 M86 E87 G89 L137 S147 D148 D740 A742 R744 N745 D758 K781 P783 D130 A132 R134 N135 D148 K158 P160 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.061uM remove_due_to_license_issue IC50=61nM P54760 20850301 1889 KEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLGGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2xa4 A 2.04 BS01 AZ5 A 1 L855 V863 A880 M929 Y931 L932 G935 N981 L983 G993 L13 V19 A36 M81 Y83 L84 G87 N133 L135 G145 D976 A978 R980 N981 D994 S1016 D128 A130 R132 N133 D146 S164 2.7.10.2 0004672,0004713,0005524,0006468 ic50<0.003uM remove_due_to_license_issue IC50=58nM O60674 21138246 2131 QFEERHLKFLQQLGKFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQAHAERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 2xab A 1.9 BS01 VHD A 1 N51 A55 D93 I96 G97 M98 L107 F138 T184 N36 A40 D78 I81 G82 M83 L92 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.54nM remove_due_to_license_issue P07900 20662534 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xae A 2.6 BS01 2XA A 1 E116 G117 E118 R119 A133 P137 Y211 L214 E215 E100 G101 E102 R103 A117 P121 Y195 L198 E199 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=200nM, IC50=53.3nM P52732 21344920 1365 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKEEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 2xb7 A 2.5 BS01 GUI A 1 L1122 H1124 V1130 A1148 K1150 M1199 G1202 E1210 L1256 L28 H30 V36 A47 K49 M98 G101 E109 L155 D1249 A1251 R1253 N1254 D1270 D148 A150 R152 N153 D169 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.65nM remove_due_to_license_issue Q9UM73 20695522 1501 NYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMAAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 2xb8 A 2.4 BS01 XNW A 1 N12 L13 Y24 N75 G77 G78 H81 H101 I102 S103 V105 R112 N10 L11 Y22 N73 G75 G76 H79 H99 I100 S101 V103 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=26nM remove_due_to_license_issue P9WPX7 20815012 1144 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 2xb9 A 2.75 BS01 XNW A 1 N10 Y22 N76 A79 H82 H102 L103 T104 R113 N10 Y22 N76 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue Q48255 20815012 201 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKNN 2xba A 1.95 BS01 571 A 1 A1148 K1150 L1196 E1197 L1198 M1199 A1200 G1202 R1253 L1256 Y1401 A40 K42 L88 E89 L90 M91 A92 G94 R145 L148 Y283 D1249 A1251 R1253 N1254 D1270 D141 A143 R145 N146 D162 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=23.68nM remove_due_to_license_issue Q9UM73 20695522 1501 NYCFAGKTSSISDLKEVPRKNITLIRGLVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 2xbj A 2.3 BS01 XBJ A 1 L226 A247 I286 L301 M304 G307 E308 E351 L354 L16 A36 I62 L77 M80 G83 E84 E127 L130 D347 K349 N352 D368 T387 D123 K125 N128 D144 T161 2.7.11.1 0004672,0005524,0006468 ic50=0.003uM remove_due_to_license_issue IC50=30nM O96017 21186793 1513 VYPKALRDEYIMSKTLGSGAGEVKLAFERKTCKKVAIKIISKALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 2xbp A 1.2 BS01 ATP A 1 G27 M28 T29 V64 R101 R103 G27 M28 T29 V64 R101 R103 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 Kd=9.6uM remove_due_to_license_issue P0A3F4 20399792 1114 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGRQKGQTERYRGSEYTVEFLQKLKLEIVVEDAQVDTVIDKIVAAARTGENGDGKIFVSPVDQTIRIRTGEKNADAIS 2xbv A 1.66 BS01 XBV A 1 E97 T98 Y99 R143 E147 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 R132 E135 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Kd=3.7nM remove_due_to_license_issue Kd=3.7nM P00742 20650636 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2xbw A 1.72 BS01 455 A 1 E97 T98 Y99 K148 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 K136 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.01uM remove_due_to_license_issue Ki=10nM P00742 20650636 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2xbx A 1.85 BS01 RR8 A 1 E97 T98 Y99 E147 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 E83 T84 Y85 E135 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.015uM remove_due_to_license_issue Ki=15nM P00742 20650636 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2xc0 A 2.05 BS01 8NC A 1 E97 T98 Y99 E147 F174 A190 V213 S214 W215 G216 G218 C220 G226 Y228 E83 T84 Y85 E135 F162 A180 V203 S204 W205 G206 G208 C209 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.192uM remove_due_to_license_issue Ki=192nM P00742 20650636 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2xc4 A 1.67 BS02 IVK A 1 E97 T98 Y99 F174 D189 A190 V213 W215 G216 G218 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 V203 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.009uM remove_due_to_license_issue Ki=9nM P00742 20650636 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2xc7 A -1.00 BS01 rna P 0 E21 P22 K23 L55 F56 I57 M58 N59 R62 T65 G67 G68 L71 K75 F89 E21 P22 K23 L55 F56 I57 M58 N59 R62 T65 G67 G68 L71 K75 F89 ? 0006408 remove_due_to_license_issue Q9H814 20430857 600 ~ 603 GAMAEDSQEKVADEISFRLQEPKKDLIARVVRIIGNKKAIELLMETAEVEQNGGLFIMNGSRRRTPGGVFLNLLKNTPSISEEQIKDIFYIENQKEYENKKAAR 2xcg A 1.9 BS03 XCG A 1 L88 P102 F168 I199 I316 Y326 L86 P100 F166 I197 I314 Y324 G62 R197 K296 G60 R195 K294 1.4.3.21,1.4.3.4 0005515,0005739,0005740,0005741,0008131,0009055,0009410,0009636,0010044,0010269,0014063,0016491,0019607,0021762,0030425,0032496,0042420,0042802,0043025,0045471,0045964,0048545,0050660,0050665,0051412,0052595,0097621 Kd=9nM remove_due_to_license_issue P27338 20855894 602 NKCDVVVVGGGISGMAAAKLLHDSGLNVVVLEARDRVGGRTYTLRNQKVKYVDLGGSYVGPTQNRILRLAKELGLETYKVNEVERLIHHVKGKSYPFRGPFPPVWNPITYLDHNNFWRTMDDMGREIPSDAPWKAPLAEEWDNMTMKELLDKLCWTESAKQLATLFVNLCVTAETHEVSALWFLWYVKQCGGTTRIISTTNGGQERKFVGGSGQVSERIMDLLGDRVKLERPVIYIDQTRENVLVETLNHEMYEAKYVISAIPPTLGMKIHFNPPLPMMRNQMITRVPLGSVIKCIVYYKEPFWRKKDYCGTMIIDGEEAPVAYTLDDTKPEGNYAAIMGFILAHKARKLARLTKEERLKKLCELYAKVLGSLEALEPVHYEEKNWCEEQYSGGCYTTYFPPGILTQYGRVLRQPVDRIYFAGTETATHWSGYMEGAVEAGERAAREILHAMGKIPEDEIWQSEPESVDVPAQPITTTFLERHLPSVPGLLRLIGLTTI 2xch A 2.0 BS01 CKG A 1 L88 V96 A109 K111 L159 Y161 A162 G165 E166 E209 L212 T222 L16 V24 A37 K39 L87 Y89 A90 G93 E94 E137 L140 T150 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T165 2.7.11.1 0004672,0004674,0005524,0006468 ic50=374nM remove_due_to_license_issue O15530 20621725 1360 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSNSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2xck A 2.3 BS01 MH4 A 1 L88 S94 A109 K111 L159 A162 G165 L212 T222 D223 L13 S19 A34 K36 L84 A87 G90 L137 T147 D148 D205 K207 E209 N210 D223 T245 D130 K132 E134 N135 D148 T162 2.7.11.1 0004672,0004674,0005524,0006468 ic50=713nM remove_due_to_license_issue O15530 20621725 1360 KKRPEDFKFGKILGEGSFSTTVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSNSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2xcn A 3.02 BS03 C8D A 1 H57 R123 G137 S139 F154 R155 A156 A157 D168 H57 R123 G137 S139 F154 R155 A156 A157 D168 H57 D81 G137 S139 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036,0097264 remove_due_to_license_issue Q91RS4 20493689 1181 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMR 2xcs B 2.1 BS05 RXV F 1 D1083 M1121 D264 M302 5.6.2.2 0003677,0003918,0005524,0006259,0006265 remove_due_to_license_issue P66937,Q99XG5 20686482 1021 KLADCSSKSPEECEIFLVEGDSAGGSTKSGRDSRTQAILPLRGKILNVEKARLDRILNNNEIRQMITAFGTGIGGDFDLAKARYHKIVIMTDADVDGAHIRTLLLTFFYRFMRPLIEAGYVYIAQPPTGYKGLGEMNADQLWETTMNPEHRALLQVKLEDAIEADQTFEMLMGDVVENRRQFIEDNAVYANERNITSEMRESFLDYAMSVIVARALPDVRDGLKPVHRRILYGLNEQGMTPDKSYKKSARIVGDVMGKYHPHGDSSIYEAMVRMAQDFSYRYPLVDGQGNFGSMDGDGAAAMRFTEARMTKITLELLRDINKDTIDFIDNYDGNEREPSVLPARFPNLLANGASGIAVGMATNIPPHNLTELINGVLSLSKNPDISIAELMEDIEGPDFPTAGLILGKSGIRRAYETGRGSIQMRSRAVIEERGGGRQRIVVTEIPFQVNKARMIEKIAELVRDKKIDGITDLRDETSLRTGVRVVIDVRKDANASVILNNLYKQTPLQTSFGVNMIALVNGRPKLINLKEALVHYLEHQKTVVRRRTQYNLRKAKDRAHILEGLRIALDHIDEIISTIRESDTDKVAMESLQQRFKLSEKQAQAILDMRLRRLTGLERDKIEAEYNELLNYISELETILADEEVLLQLVRDELTEIRDRFGDDRRTEIQLG 2xcs D 2.1 BS04 RXV F 1 D1083 M1121 D263 M301 5.6.2.2 0003677,0003918,0005524,0006259,0006265 remove_due_to_license_issue P66937,Q99XG5 20686482 1021 KLADCSSKSPEECEIFLVEGDSAGGSTKSGRDSRTQAILPLRGKILNVEKARLDRILNNNEIRQMITAFGTGIGGDFDLAKARYHKIVIMTDADVDGAHIRTLLLTFFYRFMRPLIEAGYVYIAQPPTGYKGLGEMNADQLWETTMNPEHRALLQVKLEDAIEADQTFEMLMGDVVENRRQFIEDNAVYNERNITSEMRESFLDYAMSVIVARALPDVRDGLKPVHRRILYGLNEQGMTPDKSYKKSARIVGDVMGKYHPHGDSSIYEAMVRMAQDFSYRYPLVDGQGNFGSMDGDGAAAMRFTEARMTKITLELLRDINKDTIDFIDNYDGNEREPSVLPARFPNLLANGASGIAVGMATNIPPHNLTELINGVLSLSKNPDISIAELMEDIEGPDFPTAGLILGKSGIRRAYETGRGSIQMRSRAVIEERGGGRQRIVVTEIPFQVNKARMIEKIAELVRDKKIDGITDLRDETSLRTGVRVVIDVRKDANASVILNNLYKQTPLQTSFGVNMIALVNGRPKLINLKEALVHYLEHQKTVVRRRTQYNLRKAKDRAHILEGLRIALDHIDEIISTIRESDTDKVAMESLQQRFKLSEKQAQAILDMRLRRLTGLERDKIEAEYNELLNYISELETILADEEVLLQLVRDELTEIRDRFGDDRRTEIQL 2xct B 3.35 BS04 CPF G 1 R458 S1084 R42 S262 5.6.2.2 0003677,0003918,0005524,0006259,0006265 remove_due_to_license_issue P66937,Q99XG5 20686482 1020 KLADCSSKSPEECEIFLVEGDSAGGSTKSGRDSRTQAILPLRGKILNVEKARLDRILNNNEIRQMITAFGTGIGGDFDLAKARYHKIVIMTDADVDGAHIRTLLLTFFYRFMRPLIEAGYVYIAQPPTGYKGLGEMNADQLWETTMNPEHRALLQVKLEDAIEADQTFEMLMGDVVENRRQFIEDNANERNITSEMRESFLDYAMSVIVARALPDVRDGLKPVHRRILYGLNEQGMTPDKSYKKSARIVGDVMGKYHPHGDSSIYEAMVRMAQDFSYRYPLVDGQGNFGSMDGDGAAAMRFTEARMTKITLELLRDINKDTIDFIDNYDGNEREPSVLPARFPNLLANGASGIAVGMATNIPPHNLTELINGVLSLSKNPDISIAELMEDIEGPDFPTAGLILGKSGIRRAYETGRGSIQMRSRAVIEERGGGRQRIVVTEIPFQVNKARMIEKIAELVRDKKIDGITDLRDETSLRTGVRVVIDVRKDANASVILNNLYKQTPLQTSFGVNMIALVNGRPKLINLKEALVHYLEHQKTVVRRRTQYNLRKAKDRAHILEGLRIALDHIDEIISTIRESDTDKVAMESLQQRFKLSEKQAQAILDMRLRRLTGLERDKIEAEYNELLNYISELETILADEEVLLQLVRDELTEIRDRFGDDRRTEIQLG 2xct D 3.35 BS04 CPF H 1 R458 S1084 R42 S262 5.6.2.2 0003677,0003918,0005524,0006259,0006265 remove_due_to_license_issue P66937,Q99XG5 20686482 1020 KLADCSSKSPEECEIFLVEGDSAGGSTKSGRDSRTQAILPLRGKILNVEKARLDRILNNNEIRQMITAFGTGIGGDFDLAKARYHKIVIMTDADVDGAHIRTLLLTFFYRFMRPLIEAGYVYIAQPPTKGLGEMNADQLWETTMNPEHRALLQVKLEDAIEADQTFEMLMGDVVENRRQFIEDNAVYNERNITSEMRESFLDYAMSVIVARALPDVRDGLKPVHRRILYGLNEQGMTPDKSYKKSARIVGDVMGKYHPHGDSSIYEAMVRMAQDFSYRYPLVDGQGNFGSMDGDGAAAMRFTEARMTKITLELLRDINKDTIDFIDNYDGNEREPSVLPARFPNLLANGASGIAVGMATNIPPHNLTELINGVLSLSKNPDISIAELMEDIEGPDFPTAGLILGKSGIRRAYETGRGSIQMRSRAVIEERGGGRQRIVVTEIPFQVNKARMIEKIAELVRDKKIDGITDLRDETSLRTGVRVVIDVRKDANASVILNNLYKQTPLQTSFGVNMIALVNGRPKLINLKEALVHYLEHQKTVVRRRTQYNLRKAKDRAHILEGLRIALDHIDEIISTIRESDTDKVAMESLQQRFKLSEKQAQAILDMRLRRLTGLERDKIEAEYNELLNYISELETILADEEVLLQLVRDELTEIRDRFGDDRRTEIQLG 2xd6 A 2.2 BS01 XD6 A 1 N37 A41 K44 D79 I82 M84 F124 T171 L173 N37 A41 K44 D79 I82 M84 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 ic50=0.65uM remove_due_to_license_issue P02829 20661961 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2xd9 A 1.95 BS01 XD9 A 1 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=0.35uM remove_due_to_license_issue Q48255 21275050 200 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQE 2xd9 B 1.95 BS01 XD9 B 1 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=0.35uM remove_due_to_license_issue Q48255 21275050 200 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQ 2xda A 1.85 BS01 JPS A 1 N10 L11 M13 Y22 N76 A79 H82 H102 L103 T104 R113 N10 L11 M13 Y22 N76 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=0.6uM remove_due_to_license_issue Q48255 21275050 1151 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKA 2xde A 1.4 BS01 1B0 A 1 N53 L56 N57 M66 Q67 K70 T107 Y130 N53 L56 N57 M66 Q67 K70 T97 Y120 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0016032 Kd=3.42uM remove_due_to_license_issue P12497 21170360 1148 PIVQNLQGQMVHQAISPRTLNAWVKVVEEKAFSPEVIPMFSALSEGATPQDLNTMLNTVGGHQAAMQMLKETINEEAAEWDRLHPVGEPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYS 2xdk A 1.97 BS01 XDK A 1 A55 M98 N106 T184 A45 M88 N96 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=250uM remove_due_to_license_issue P07900 20718493 1226 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 2xdl A 1.98 BS01 2DL A 1 N51 A55 D93 M98 L107 F138 T184 E223 N35 A39 D77 M82 L91 F122 T168 E207 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=790uM remove_due_to_license_issue P07900 20718493 1225 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xdm B 2.4 BS01 BO8 B 1 S49 W139 D142 Y147 S298 N300 L349 G412 T413 M414 S415 S49 W139 D142 Y147 S298 N300 L349 G412 T413 M414 S415 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue P39045 20608745 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAP 2xdx A 2.42 BS01 WOE A 1 N51 A55 G97 M98 N106 L107 F138 T184 E223 N41 A45 G87 M88 N96 L97 F128 T174 E213 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.35uM remove_due_to_license_issue Ki=1200nM P07900 20718493 1224 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xe0 A 2.31 BS01 dna C 0 G19 D20 S22 Q26 Y44 T46 Q47 K48 Q75 N136 D137 S138 R141 K142 G18 D19 S21 Q25 Y43 T45 Q46 K47 Q74 N135 D136 S137 R140 K141 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQINPNASSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIAPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKASPAAFLEVCTWVDQIAALNDSATRKTTSETVAAVLD 2xe0 A 2.31 BS02 dna D 0 S32 S33 K34 R38 R40 Y66 R68 E80 I81 K116 S31 S32 K33 R37 R39 Y65 R67 E79 I80 K115 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNKEFLLYLAGFVDGDGSIIAQINPNASSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIAPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKASPAAFLEVCTWVDQIAALNDSATRKTTSETVAAVLD 2xe0 B 2.31 BS01 dna C 0 R30 S32 N33 K34 Q38 Y66 Y68 I81 K116 K139 R29 S31 N32 K33 Q37 Y65 Y67 I80 K115 K138 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPRASNKFAHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLAIIEQLPSAKASPDAFLEVCTWVDQIAALNDSKTRATTSATVRAALD 2xe0 B 2.31 BS02 dna D 0 G19 D20 S22 I24 Q26 K28 R30 T46 Q47 K48 R51 R77 N136 D137 S138 A142 G18 D19 S21 I23 Q25 K27 R29 T45 Q46 K47 R50 R76 N135 D136 S137 A141 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNKEFLLYLAGFVDGDGSIIAQIKPRASNKFAHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLAIIEQLPSAKASPDAFLEVCTWVDQIAALNDSKTRATTSATVRAALD 2xef A 1.59 BS01 AR8 A 1 K207 R210 N257 E424 L428 R463 D465 R511 S513 K514 G516 G518 N519 R534 R536 W541 E542 Y552 H553 N698 K699 Y700 A701 G702 K153 R156 N203 E370 L374 R409 D411 R457 S459 K460 G462 G464 N465 R480 R482 W487 E488 Y498 H499 N642 K643 Y644 A645 G646 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=0.145nM remove_due_to_license_issue Q04609 20726553 1770 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVQPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2xeg A 1.59 BS04 CI9 A 1 K207 R210 N257 E424 R463 R511 S513 G518 N519 R534 R536 W541 E542 Y552 H553 N698 K699 Y700 K153 R156 N203 E370 R409 R457 S459 G464 N465 R480 R482 W487 E488 Y498 H499 N642 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=0.02nM remove_due_to_license_issue Q04609 20726553 1768 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVQPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2xei A 1.69 BS04 ARK A 1 R210 E424 R463 S501 R511 S513 G518 N519 R534 R536 W541 Y552 H553 K699 Y700 R156 E370 R409 S447 R457 S459 G464 N465 R480 R482 W487 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=0.024nM remove_due_to_license_issue Q04609 20726553 1770 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2xej A 1.78 BS04 OKD A 1 K207 R210 N257 E424 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 A701 K153 R156 N203 E370 L374 G464 N465 R480 R482 Y498 H499 K643 Y644 A645 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=1.34nM remove_due_to_license_issue Q04609 20726553 1768 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVQPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 2xel A 2.5 BS03 IA2 A 1 R428 L431 D590 N616 I617 S619 R620 R427 L430 D589 N615 I616 S618 R619 S181 G182 T186 N233 S236 S237 G457 E459 S180 G181 T185 N232 S235 S236 G456 E458 ? 0003774,0005524,0016459,0051015 remove_due_to_license_issue P08799 21680745 999 NPIHDRTSDYHKYLKVKQGDSDLFKLTVSDKRYIWYNPDPKERDSYECGEIVSETSDSFTFKTVDGQDRQVKKDDANQRNPIKFDGVEDMSELSYLNEPAVFHNLRVRYNQDLIYTYSGLFLVAVNPFKRIPIYTQEMVDIFKGRRRNEVAPHIFAISDVAYRSMLDDRQNQSLLITGESGAGKTENTKKVIQYLASVAGRNQANGSGVLEQQILQANPILEAFGNAKTTRNNNSSRFGKFIEIQFNSAGFISGASIQSYLLEKSRVVFQSETERNYHIFYQLLAGATAEEKKALHLAGPESFNYLNQSGCVDIKGVSDSEEFKITRQAMDIVGFSQEEQMSIFKIIAGILHLGNIKFEKGAGEGAVLKDKTALNAASTVFGVNPSVLEKALMEPRILAGRDLVAQHLNVEKSSSSRDALVKALYGRLFLWLVKKINNVLCQERKAYFIGVLDISGFEIFKVNSFEQLCINYTNEKLQQFFNHHMFKLEQEEYLKEKINWTFIDFGLDSQATIDLIDGRQPPGILALLDEQSVFPNATDNTLITKLHSHFSKKNAKYEEPRFSKTEFGVTHYAGQVMYEIQDWLEKNKDPLQQDLELCFKDSSDNVVTKLFNDPNIASRAKKGANFITVAAQYKEQLASLMATLETTNPHFVRCIIPNNKQLPAKLEDKVVLDQLRCNGVLEGIRITRKGFPNRIIYADFVKRYYLLAPNVPRDAEDSQKATDAVLKHLNIDPEQYRFGITKIFFRAGQLARIEEAREQRLESNEPPMDFDDDIPF 2xey A 2.7 BS01 YVQ A 1 L15 V23 C87 G90 L137 L10 V14 C70 G73 L120 D130 K132 E134 N135 D148 T170 D113 K115 E117 N118 D131 T153 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=154881662nM O14757 20561787 1270 VEDWDLVQTLGGEVQLAVNRVTEEAVAVKIVDENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2xez A 2.25 BS01 XEZ A 1 K38 C87 L137 K27 C66 L116 D130 K132 E134 N135 D148 T170 D109 K111 E113 N114 D127 T149 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.5uM remove_due_to_license_issue IC50=660693448nM O14757 20561787 1271 EDWDLVQTLGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2xf0 A 2.4 BS01 4UB A 1 L15 V23 Y86 C87 G90 L137 L12 V15 Y67 C68 G71 L118 D130 K132 E134 N135 D148 T170 D111 K113 E115 N116 D129 T151 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=30uM remove_due_to_license_issue IC50=33113112nM O14757 20561787 1271 PFVEDWDLVQTLGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2xfi A 1.73 BS01 XFI A 1 L91 D93 G95 S96 Y132 T133 Q134 F169 D289 G291 T292 T293 N294 R296 N446 L30 D32 G34 S35 Y71 T72 Q73 F108 D215 G217 T218 T219 N220 R222 N372 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D215 T218 3.4.23.46 0004190,0006508,0016020 ic50=15nM remove_due_to_license_issue P56817 20579874 1448 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2xfj A 1.8 BS01 VG5 A 1 L91 D93 G95 S96 Y132 T133 Q134 F169 W176 I179 D289 G291 T292 T293 N294 N446 L30 D32 G34 S35 Y71 T72 Q73 F108 W115 I118 D216 G218 T219 T220 N221 N373 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D216 T219 3.4.23.46 0004190,0006508,0016020 ic50=13nM remove_due_to_license_issue IC50=310nM P56817 20579874 500 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2xfk A 1.8 BS01 AA9 A 1 G72 L91 D93 G95 Y132 T133 Q134 F169 W176 D289 G291 T292 T293 N294 R296 N446 G11 L30 D32 G34 Y71 T72 Q73 F108 W115 D214 G216 T217 T218 N219 R221 N371 D93 S96 N98 A100 Y132 D289 T292 D32 S35 N37 A39 Y71 D214 T217 3.4.23.46 0004190,0006508,0016020 ic50=3nM remove_due_to_license_issue P56817 20579874 500 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPQVTVRANIAAITESDKFFIQGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTQQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 2xfm A -1.00 BS01 rna B 0 I308 Y313 K316 T317 Y318 R319 F333 K335 A381 M382 L393 I33 Y38 K41 T42 Y43 R44 F58 K60 A106 M107 L118 3.1.26.- 0003723 remove_due_to_license_issue Q9JMB7 21237665 1 ~ 8 RSETVLDFMFNLYQQTEEHKFQEQVSKELIGLIVLTKYNNKTYRVDDIDWDQNPKSTFKKADGSEVSFLEYYRKQYNQEITDLKQPVLVSQPKRRRGPGGTLPGPAMLIPELCYLTGLTD 2xg3 A 1.2 BS01 GAL B 1 H158 R162 N174 W181 E184 H46 R50 N62 W69 E72 ? 0030246 remove_due_to_license_issue P17931 20873837 2 ALIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 2xg5 A 2.0 BS01 EC2 A 1 P30 Y31 L32 V56 I93 P94 P95 P30 Y31 L32 V56 I93 P94 P95 ? 0005515,0030288,0042597,0043711,0061077,0071555 ic50=22uM remove_due_to_license_issue P15319 20586493 1219 AVSLDRTRAVFDGSEKSMTLDISNDNKQLPYLAQAWIENENQEKIITGPVIATPPVQRLEPGAKSMVRLSTTPDISKLPQDRESLFYFNLREIPPRSEKANVLQIALQTKIKLFYRPAAIKTRPNEVWQDQLILNKVSGGYRIENPTPYYVTVIGLGGSEKQAEEGEFETVMLSPRSEQTVKSANYNTPYLSYINDYGGRPVLSFICNGSRCSVKK 2xg9 A 1.8 BS01 NOJ A 1 E184 E378 A380 E182 E376 A378 D99 E184 T340 E378 L381 D97 E182 T338 E376 L379 3.2.1.2 0000272,0016161,0016798,0042802 remove_due_to_license_issue P16098 21085740 1490 VNVKGNYVQVYVMLPLDAVSVNNRFEKGDELRAQLRKLVEAGVDGVMVDVWWGLVEGKGPKAYDWSAYKQLFELVQKAGLKLQAIMSFHQCGGNVGDAVNIPIPQWVRDVGTRDPDIFYTDGHGTRNIEYLTLGVDNQPLFHGRSAVQMYADYMTSFRENMKEFLDAGVIVDIEVGLGPAGEMRYPSYPQSHGWSFPGIGEFICYDKYLQADFKAAAAAVGHPEWEFPNDVGQYNDTPERTQFFRDNGTYLSEKGRFFLAWYSNNLIKHGDRILDEANKVFLGYKVQLAIKISGIHWWYKVPSHAAELTAGYYNLHDRDGYRTIARMLKRHRASINFTCAEMRDSEQSSQAMSAPEELVQQVLSAGWREGLNVACENALPRYDPTAYNTILRNARPHGINQSGPPEHKLFGFTYLRLSNQLVEGQNYANFKTFVDRMHANLPRDPYVDPMAPLPRSGPEISIEMILQAAQPKLQPFPFQEHTDLPVG 2xg9 A 1.8 BS02 GLC A 1 M15 D51 H91 R418 M13 D49 H89 R416 D99 E184 T340 E378 L381 D97 E182 T338 E376 L379 3.2.1.2 0000272,0016161,0016798,0042802 remove_due_to_license_issue P16098 21085740 1491 VNVKGNYVQVYVMLPLDAVSVNNRFEKGDELRAQLRKLVEAGVDGVMVDVWWGLVEGKGPKAYDWSAYKQLFELVQKAGLKLQAIMSFHQCGGNVGDAVNIPIPQWVRDVGTRDPDIFYTDGHGTRNIEYLTLGVDNQPLFHGRSAVQMYADYMTSFRENMKEFLDAGVIVDIEVGLGPAGEMRYPSYPQSHGWSFPGIGEFICYDKYLQADFKAAAAAVGHPEWEFPNDVGQYNDTPERTQFFRDNGTYLSEKGRFFLAWYSNNLIKHGDRILDEANKVFLGYKVQLAIKISGIHWWYKVPSHAAELTAGYYNLHDRDGYRTIARMLKRHRASINFTCAEMRDSEQSSQAMSAPEELVQQVLSAGWREGLNVACENALPRYDPTAYNTILRNARPHGINQSGPPEHKLFGFTYLRLSNQLVEGQNYANFKTFVDRMHANLPRDPYVDPMAPLPRSGPEISIEMILQAAQPKLQPFPFQEHTDLPVG 2xgm A 2.55 BS01 LXN A 1 L442 H444 Y447 L386 H388 Y391 ? 0016757,0046872 remove_due_to_license_issue Q8PC69 20640461 1569 PEAVARLGRVRWTQQRHAEAAVLLQQASDAAPEHPGIALWLGHALEDAGQAEAAAAAYTRAHQLLPEEPYITAQLLNWRRRLCDWRALDVLSAQVRAAVAQGVGAVEPFAFLSEDASAAEQLACARTRAQAIAASVRPLAPTRVRSKGPLRVGFVSNGFGAHPTGLLTVALFEALQRRQPDLQMHLFATSGDDGSTLRTRLAQASTLHDVTALGHLATAKHIRHHGIDLLFDLRGWGGGGRPEVFALRPAPVQVNWLAYPGTSGAPWMDYVLGDAFALPPALEPFYSEHVLRLQGAFQPSDTSRVVAEPPSRTQCGLPEQGVVLCCFNNSYKLNPQSMARMLAVLREVPDSVLWLLSGPGEADARLRAFAHAQGVDAQRLVFMPKLPHPQYLARYRHADLFLDTHPYNAHTTASDALWTGCPVLTTPGETFAARVAGSLNHHLGLDEMNVADDAAFVAKAVALASDPAALTALHARVDVLRRASGVFHMDGFADDFGALLQALARRHGWLGI 2xgo A 2.6 BS01 ZKD A 1 P219 L222 N385 Y387 L412 L442 H444 Y447 T467 P199 L202 N365 Y367 L392 L422 H424 Y427 T447 ? 0016757,0046872 remove_due_to_license_issue Q8PC69 20640461 1569 QDFVAWLMLADAELGMGDTTAGEMAVQRGLALHPGHPEAVARLGRVRWTQQRHAEAAVLLQQASDAAPEHPGIALWLGHALEDAGQAEAAAAAYTRAHQLLPEEPYITAQLLNWRRRLCDWRALDVLSAQVRAAVAQGVGAVEPFAFLSEDASAAEQLACARTRAQAIAASVRPLAPTRVRSKGPLRVGFVSNGFGAHPTGLLTVALFEALQRRQPDLQMHLFATSGDDGSTLRTRLAQASTLHDVTALGHLATAKHIRHHGIDLLFDLRGWGGGGRPEVFALRPAPVQVNWLAYPGTSGAPWMDYVLGDAFALPPALEPFYSEHVLRLQGAFQPSDTSRVVAEPPSRTQCGLPEQGVVLCCFNNSYKLNPQSMARMLAVLREVPDSVLWLLSGPGEADARLRAFAHAQGVDAQRLVFMPKLPHPQYLARYRHADLFLDTHPYNAHTTASDALWTGCPVLTTPGETFAARVAGSLNHHLGLDEMNVADDAAFVAKAVALASDPAALTALHARVDVLRRASGVFHMDGFADDFGALLQALARRHGWLGI 2xgs A 2.39 BS01 44P A 1 P219 L222 N385 K388 K441 L442 H444 Y447 T467 D471 P193 L196 N359 K362 K415 L416 H418 Y421 T441 D445 ? 0016757,0046872 Kd=0.53mM remove_due_to_license_issue Q8PC69 20640461 1569 LMLADAELGMGDTTAGEMAVQRGLALHPGHPEAVARLGRVRWTQQRHAEAAVLLQQASDAAPEHPGIALWLGHALEDAGQAEAAAAAYTRAHQLLPEEPYITAQLLNWRRRLCDWRALDVLSAQVRAAVAQGVGAVEPFAFLSEDASAAEQLACARTRAQAIAASVRPLAPTRVRSKGPLRVGFVSNGFGAHPTGLLTVALFEALQRRQPDLQMHLFATSGDDGSTLRTRLAQASTLHDVTALGHLATAKHIRHHGIDLLFDLRGWGGGGRPEVFALRPAPVQVNWLAYPGTSGAPWMDYVLGDAFALPPALEPFYSEHVLRLQGAFQPSDTSRVVAEPPSRTQCGLPEQGVVLCCFNNSYKLNPQSMARMLAVLREVPDSVLWLLSGPGEADARLRAFAHAQGVDAQRLVFMPKLPHPQYLARYRHADLFLDTHPYNAHTTASDALWTGCPVLTTPGETFAARVAGSLNHHLGLDEMNVADDAAFVAKAVALASDPAALTALHARVDVLRRASGVFHMDGFADDFGALLQALARRHGWLGI 2xh5 A 2.72 BS02 X37 A 1 G161 A179 K181 M229 E230 A232 E236 T292 D293 F439 G16 A34 K36 M84 E85 A87 E91 T147 D148 F294 D275 K277 N280 D293 T313 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P31751 20151677 1480 KVTMNDFDYLKLLGKGTFGKVILVREKATGRYYAMKILRKEVIIAKDEVAHTVTESRVLQNTRHPFLTALKYAFQTHDRLCFVMEYANGGELFFHLSRERVFTEERARFYGAEIVSALEYLHSRDVVYRDIKLENLMLDKDGHIKITDFGLCKEGISDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHERLFELILMEEIRFPRTLSPEAKSLLAGLLKKDPKQRLGGGPSDAKEVMEHRFFLSINWQDVVQKKLLPPFKPQVTSEVDTRYFDDEFTAQSITQEMFEDFDYIADW 2xhi A 1.55 BS01 dna B 0 N149 R154 G202 Y203 R204 Q287 Q294 N140 R145 G193 Y194 R195 Q278 Q285 C249 N268 C240 N259 3.2.2.-,4.2.99.18 0000978,0003677,0003684,0003824,0004519,0005515,0005634,0005654,0005739,0005759,0005829,0006281,0006284,0006285,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045007,0045008,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O15527 21220122 2 ~ 15 RMGHRTLASTPALWASIPCPRSELRLDLVLPSGQSFRWREQSPAHWSGVLADQVWTLTQTEEQLHCTVYRGDKSQASRPTPDELEAVRKYFQLDVTLAQLYHHWGSVDSHFQEVAQKFQGVRLLRQDPIECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPSLQALAGPEVEAHLRKLGLGYRARYVSASARAILEEQGGLAWLQQLRESSYEEAHKALCILPGVGTCVADKICLMALDKPQAVPVNVHMWHIAQRDYSWHPTTSQAKGPSPQTNKELGNFFRSLWGPYAGWAQAVLFSADLRQ 2xhi A 1.55 BS02 dna C 0 G42 S147 S148 N149 N150 N151 I152 Y207 P244 G245 G247 C249 V250 K253 N268 H270 Q315 F319 G33 S138 S139 N140 N141 N142 I143 Y198 P235 G236 G238 C240 V241 K244 N259 H261 Q306 F310 C249 N268 C240 N259 3.2.2.-,4.2.99.18 0000978,0003677,0003684,0003824,0004519,0005515,0005634,0005654,0005739,0005759,0005829,0006281,0006284,0006285,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045007,0045008,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O15527 21220122 16 ~ 29 RMGHRTLASTPALWASIPCPRSELRLDLVLPSGQSFRWREQSPAHWSGVLADQVWTLTQTEEQLHCTVYRGDKSQASRPTPDELEAVRKYFQLDVTLAQLYHHWGSVDSHFQEVAQKFQGVRLLRQDPIECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPSLQALAGPEVEAHLRKLGLGYRARYVSASARAILEEQGGLAWLQQLRESSYEEAHKALCILPGVGTCVADKICLMALDKPQAVPVNVHMWHIAQRDYSWHPTTSQAKGPSPQTNKELGNFFRSLWGPYAGWAQAVLFSADLRQ 2xhm A 1.96 BS01 K26 A 1 H337 A338 S339 A340 W341 D342 Y344 H367 E368 H371 F375 H394 E395 Y496 V502 Y507 H321 A322 S323 A324 W325 D326 Y328 H351 E352 H355 F359 H378 E379 Y480 V486 Y491 H337 A338 H367 E368 H371 E395 H497 Y507 H321 A322 H351 E352 H355 E379 H481 Y491 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Q10714 20599761 1615 ALVKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 2xhr A 2.2 BS01 C0P A 1 A55 G97 M98 N106 L107 I110 G135 F138 A39 G81 M82 N90 L91 I94 G119 F122 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.0048uM remove_due_to_license_issue P07900 20718493 1001 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 2xht A 2.27 BS01 C0Y A 1 N51 S52 A55 K58 D93 M98 F138 T184 E223 N40 S41 A44 K47 D82 M87 F127 T173 E212 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=1.1uM remove_due_to_license_issue P07900 20718493 1224 MEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xhx A 2.801 BS01 T5M A 1 N51 S52 D54 A55 D93 I96 G97 F138 T184 E223 N41 S42 D44 A45 D83 I86 G87 F128 T174 E213 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 20718493 1224 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xi7 A 2.2 BS03 XI7 A 1 H34 D52 D79 D92 K94 H35 D53 D80 D93 K95 2.7.7.48,3.1.-.- remove_due_to_license_issue A5HC98 20862319 1186 GMDYQEYQQFLARINTARDACVAKDIDVDLLMARHDYFGRELCKSLNIEYRNDVPFIDIILDIRPEVDPLTIDAPHITPDNYLYINNVLYIIDYKVSVSNESSVITYDKYYELTRDISDRLSIPIEIVIIRIDPVSRDLHINSDRFKELYPTIVVDINFNQFFDLKQLLYEKFGDDEEFLLKVA 2xib B 2.2 BS01 DFU B 1 H66 E87 W88 H135 H136 Y178 D229 E288 W316 H32 E53 W54 H101 H102 Y144 D195 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Kd=55.1nM remove_due_to_license_issue Q8A3I4 20665773 1472 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRA 2xii A 1.8 BS02 TA9 A 1 H66 E87 W88 H135 H136 Y178 D229 W232 R262 H272 G286 E288 W316 H32 E53 W54 H101 H102 Y144 D195 W198 R228 H238 G252 E254 W282 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Kd=63.3nM remove_due_to_license_issue Q8A3I4 20665773 1002 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAA 2xix A 2.4 BS01 XIX A 1 A65 I185 A33 I153 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 21358046 1307 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2xiy A 2.2 BS01 XIY A 1 F49 V52 A65 L174 I185 D186 F17 V20 A33 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 21358046 1307 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2xiz A 2.21 BS01 XIZ A 1 A65 K67 L120 E121 L174 I185 D186 A33 K35 L88 E89 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 21358046 1307 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2xj0 A 3.1 BS01 XJ0 A 1 A65 K67 L120 L174 I185 D186 A300 E301 S306 A33 K35 L88 L142 I153 D154 A268 E269 S274 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 21358046 1307 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2xj1 A 2.13 BS01 XJ1 A 1 L44 F49 A65 K67 L120 E121 E171 N172 L174 I185 D186 L12 F17 A33 K35 L88 E89 E139 N140 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Kd=28nM remove_due_to_license_issue IC50=13nM P11309 21358046 1307 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2xj2 A 2.2 BS01 985 A 1 L44 F49 A65 K67 E121 L174 I185 D186 L12 F17 A33 K35 E89 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Kd=66nM remove_due_to_license_issue IC50=57nM P11309 21358046 1001 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 2xj7 A 2.0 BS01 GC2 A 1 G135 K166 D242 D243 Y282 W337 N339 D344 G132 K163 D239 D240 Y279 W334 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Kd=246nM remove_due_to_license_issue Q89ZI2 20851343 1000 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVERNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMPLQVKANRVLISPVEIELDAIYPGENIQILSAGLQKAPVKFVFVLTIEK 2xjg A 2.25 BS01 XJG A 1 N51 S52 D54 A55 I91 D93 I96 F138 T184 V186 N41 S42 D44 A45 I81 D83 I86 F128 T174 V176 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.015uM remove_due_to_license_issue P07900 20662534 1224 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xjj A 1.9 BS01 L81 A 1 N51 D54 A55 D93 I96 G97 M98 F138 T184 N35 D38 A39 D77 I80 G81 M82 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.31uM remove_due_to_license_issue P07900 20662534 1225 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDVQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2xjx A 1.66 BS01 XJX A 1 N51 D54 A55 D93 I96 G97 M98 F138 T184 N41 D44 A45 D83 I86 G87 M88 F128 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.71nM remove_due_to_license_issue IC50=20nM P07900 20662534 1232 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKERDKEVS 2xk1 A 2.8 BS01 EWB A 1 S49 Y147 S298 N300 L349 G412 T413 S49 Y147 S298 N300 L349 G412 T413 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue P39045 24900305 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 2xk3 A 2.2 BS01 XK3 A 1 I14 C22 V35 E87 C89 G92 F148 D159 F160 I12 C16 V29 E81 C83 G86 F134 D145 F146 D141 K143 A145 N146 D159 T179 D127 K129 A131 N132 D145 T150 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P51955 20936789 1280 SRAEDYEVLYTIGTRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFGVGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xk4 A 2.1 BS01 OL2 A 1 I14 V35 K37 M86 E87 C89 G92 F148 G158 D159 I12 V31 K33 M82 E83 C85 G88 F136 G146 D147 D141 K143 A145 N146 D159 T179 D129 K131 A133 N134 D147 T154 2.7.11.1 0004672,0005524,0006468 ic50=16.9uM remove_due_to_license_issue IC50=16900nM P51955 20936789 1280 SRAEDYEVLYTIGTYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFGLFVGTPYYMSPEQMNRMNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xk6 A 2.2 BS01 EQH A 1 I14 C22 V35 K37 Y70 M86 E87 Y88 C89 E90 G92 D93 F148 I11 C14 V27 K29 Y62 M78 E79 Y80 C81 E82 G84 D85 F132 D141 K143 A145 N146 D159 T179 D125 K127 A129 N130 D143 T146 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P51955 20936789 1280 RAEDYEVLYTIGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDVGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xk7 A 1.992 BS01 30E A 1 I14 M86 Y88 C89 G92 F148 D159 I12 M81 Y83 C84 G87 F135 D146 D141 K143 A145 N146 D159 T179 D128 K130 A132 N133 D146 T150 2.7.11.1 0004672,0005524,0006468 ic50=1.5uM remove_due_to_license_issue IC50=1500nM P51955 20936789 1280 SRAEDYEVLYTIGTGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFVGTPYYMSPEQMNNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xk8 A 2.001 BS01 5R1 A 1 I14 C22 K37 V68 Y70 M86 Y88 C89 G92 F148 D159 F160 I12 C16 K31 V62 Y64 M80 Y82 C83 G86 F134 D145 F146 D141 K143 A145 N146 D159 T179 D127 K129 A131 N132 D145 T150 2.7.11.1 0004672,0005524,0006468 ic50=2.4uM remove_due_to_license_issue IC50=1300nM P51955 20936789 1280 SRAEDYEVLYTIGTRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFFVGTPYYMSPEQMNNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xk9 A 2.35 BS01 XK9 A 1 L226 V234 K249 I251 E273 L301 M304 E305 G307 L354 T367 D368 L16 V23 K38 I40 E47 L75 M78 E79 G81 L128 T141 D142 D347 K349 N352 D368 T387 D121 K123 N126 D142 T161 2.7.11.1 0004672,0005524,0006468 ic50=0.03nM remove_due_to_license_issue O96017 21963792 1511 VYPKALRDEYIMSKTLGSGAGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2xkc A 2.5 BS01 4VQ A 1 I14 C22 V35 K37 M86 C89 G92 F148 G158 I12 C18 V31 K33 M82 C85 G88 F134 G144 K143 A145 N146 D159 T179 K129 A131 N132 D145 T147 2.7.11.1 0004672,0005524,0006468 ic50=2.6uM remove_due_to_license_issue IC50=2300nM P51955 20936789 1280 SRAEDYEVLYTIGTYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSLKPANVFLDGKQNVKLGDGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xkd A 1.96 BS01 T3M A 1 I14 C22 K37 Y70 M86 Y88 C89 G92 F148 D159 I12 C17 K32 Y65 M81 Y83 C84 G87 F134 D145 D141 K143 A145 N146 D159 T179 D127 K129 A131 N132 D145 T151 2.7.11.1 0004672,0005524,0006468 ic50=2.3uM remove_due_to_license_issue IC50=1600nM P51955 20936789 1280 SRAEDYEVLYTIGTGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSDLKPANVFLDGKQNVKLGDFTFVGTPYYMSPEQMNRMSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xke A 2.203 BS01 WI2 A 1 I14 C22 K37 Y70 M86 C89 G92 F148 D159 I12 C17 K32 Y65 M81 C84 G87 F134 D145 D141 K143 A145 N146 D159 T179 D127 K129 A131 N132 D145 T147 2.7.11.1 0004672,0005524,0006468 ic50=4.2uM remove_due_to_license_issue IC50=4200nM P51955 20936789 1280 SRAEDYEVLYTIGTGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSDLKPANVFLDGKQNVKLGDFTPYYMSPEQMNNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xkf A 2.35 BS01 BX1 A 1 I14 K37 Y70 M86 Y88 C89 G92 D93 F148 D159 I12 K32 Y65 M81 Y83 C84 G87 D88 F135 D146 D141 K143 A145 N146 D159 T179 D128 K130 A132 N133 D146 T151 2.7.11.1 0004672,0005524,0006468 ic50=0.87uM remove_due_to_license_issue IC50=410nM P51955 20936789 1280 SRAEDYEVLYTIGTGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFFVGTPYYMSPEQMNRSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xln A 2.4 BS01 EWA A 1 S49 K52 Y147 S298 N300 L349 T413 S49 K52 Y147 S298 N300 L349 T413 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue P39045 24900305 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 2xm1 A 2.0 BS01 LTM A 1 G135 K166 D242 D243 Y282 V314 W337 N339 D344 G132 K163 D239 D240 Y279 V311 W334 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Kd=8.5uM remove_due_to_license_issue Q89ZI2 20689974 1717 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVERNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMLPLQVKANRVLISPEIELDAIYPGENIQINFLSAGLQKAPVKFVRFQFVLTIEK 2xm2 A 1.95 BS01 LOG A 1 G135 K166 D242 D243 Y282 V314 W337 N339 D344 G125 K156 D232 D233 Y272 V304 W327 N329 D334 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=24uM remove_due_to_license_issue Q89ZI2 20689974 1000 LQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVERNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMLPLQVKANRVLISPEIELDAIYPGENIQINSAGLQKAPVKFVRFFVLTIEK 2xm8 A 3.4 BS01 B4W A 1 L226 G232 A247 L301 E302 L303 M304 E308 T367 L16 G17 A32 L68 E69 L70 M71 E75 T134 D347 K349 N352 D368 D114 K116 N119 D135 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=160nM O96017 21186793 1504 VYPKALRDEYIMSKTLGEVKLAFERKTCKKVAIKINVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEEN 2xm9 A 2.5 BS01 LWH A 1 L226 A247 K249 E273 I286 L301 M304 E308 E351 N352 L354 T367 D368 L16 A34 K36 E48 I61 L76 M79 E83 E126 N127 L129 T142 D143 D347 K349 N352 D368 T387 D122 K124 N127 D143 T162 2.7.11.1 0004672,0005524,0006468 ic50=0.009uM remove_due_to_license_issue O96017 21186793 1513 VYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 2xmy A 1.9 BS01 CDK A 1 I10 A31 F80 F82 L83 H84 D86 K89 L134 D145 I10 A31 F77 F79 L80 H81 D83 K86 L131 D142 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.11nM remove_due_to_license_issue Ki=0.11nM P24941 21035734 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2xn3 A 2.09 BS01 ID8 A 1 L246 L269 K270 N273 L228 L251 K252 N255 ? 0004867,0005615 Kd=89nM remove_due_to_license_issue P05543 21325280 1356 LYKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMEQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAGAMFLEAIPR 2xn3 B 2.09 BS01 ID8 A 1 R378 R381 R18 R21 ? remove_due_to_license_issue P05543 21325280 1356 LHPIIQIDRSFMLLILERSTRSILFLGKVVNPTEA 2xn5 A 1.7 BS01 FUN A 1 S23 S24 L269 K270 N273 S9 S10 L255 K256 N259 ? 0004867,0005615 Kd=123nM remove_due_to_license_issue P05543 21325280 1356 PNATLYKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMEQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAGAMFLEAIPR 2xn6 A 1.29 BS04 F6Y A 1 Y225 N273 Y207 N255 ? 0004867,0005615 remove_due_to_license_issue P05543 21325280 1369 LYKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMDQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAGAMFLEAIPR 2xn6 A 1.29 BS05 T44 A 1 S23 Q238 L246 L269 K270 N273 S5 Q220 L228 L251 K252 N255 ? 0004867,0005615 remove_due_to_license_issue P05543 21325280 1370 LYKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMDQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAGAMFLEAIPR 2xn6 B 1.29 BS01 T44 A 1 L376 R378 R381 L15 R17 R20 ? remove_due_to_license_issue P05543 21325280 1370 HPIIQIDRSFMLLILERSTRSILFLGKVVNPTEA 2xn7 A 1.43 BS01 T44 A 1 S24 Q238 L246 S266 L269 N273 S8 Q222 L230 S250 L253 N257 ? 0004867,0005615 remove_due_to_license_issue P05543 21325280 1355 ATLYKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMEQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAGAMFLEAIPR 2xn7 A 1.43 BS02 F6Z A 1 Y225 Q238 D240 Y209 Q222 D224 ? 0004867,0005615 remove_due_to_license_issue P05543 21325280 1356 ATLYKMSSINADFAFNLYRRFTVETPDKNIFFSPVSISAALVMLSFGACCSTQTEIVETLGFNLTDTPMVEIQHGFQHLICSLNFPKKELELQIGNALFIGKHLKPLAKFLNDVKTLYETEVFSTDFSNISAAKQEINSHVEMQTKGKVVGLIQDLKPNTIMVLVNYIHFKAQWANPFDPSKTEDSSSFLIDKTTTVQVPMMHQMEQYYHLVDMELNCTVLQMDYSKNALALFVLPKEGQMESVEAAMSSKTLKKWNRLLQKGWVDLFVPKFSISATYDLGATLLKMGIQHAYSENADFSGLTEDNGLKLSNAAHKAVLHIGEKGTEAAGAMFLEAIPR 2xn7 B 1.43 BS01 T44 A 1 L376 R378 R381 L15 R17 R20 ? remove_due_to_license_issue P05543 21325280 1355 HPIIQIDRSFMLLILERSTRSILFLGKVVNPTEA 2xnb A 1.85 BS01 Y8L A 1 I10 E12 V18 A31 K33 F82 L83 L134 D145 I10 E12 V18 A31 K33 F80 L81 L132 D143 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=149nM remove_due_to_license_issue P24941 21035734 1299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 2xne A 2.8 BS01 ASH A 1 R137 L139 G140 K141 A160 A213 P214 G216 T217 R11 L13 G14 K15 A34 A80 P81 G83 T84 D256 K258 E260 N261 N274 T292 D123 K125 E127 N128 N141 T150 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=190nM O14965 20833547 1389 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIANFGWSVHAPTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2xng A 2.605 BS01 A0H A 1 R137 L139 A160 A213 P214 G216 L263 K389 R11 L13 A34 A87 P88 G90 L137 K253 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 20833547 1391 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHATLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 2xni A 3.3 BS03 TR8 A 1 H57 L135 K136 G137 S139 R155 A156 A157 D168 H58 L136 K137 G138 S140 R156 A157 A158 D169 H57 D81 G137 S139 H58 D82 G138 S140 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 20801653 1181 GAPITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMR 2xnm A 1.85 BS01 WGZ A 1 I14 C22 K37 Y88 C89 D93 F148 G158 D159 I12 C20 K35 Y86 C87 D91 F137 G147 D148 D141 K143 A145 N146 D159 T179 D130 K132 A134 N135 D148 T159 2.7.11.1 0004672,0005524,0006468 ic50=0.16uM remove_due_to_license_issue IC50=25nM P51955 21366329 1280 SRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRRDLKPANVFLDGKQNVKLGDFGLARILFVGTPYYMSPEQMNRSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xnn A 2.5 BS01 430 A 1 I14 C22 K37 Y88 C89 D93 A145 F148 D159 I12 C18 K33 Y84 C85 D89 A133 F136 D147 D141 K143 A145 N146 D159 T179 D129 K131 A133 N134 D147 T153 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=>50000nM P51955 21366329 1280 SRAEDYEVLYTIGTYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFGFVGTPYYMSPEQMNRYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xno A 1.98 BS01 ED8 A 1 I14 C22 K37 M86 Y88 C89 D93 A145 F148 D159 I12 C20 K35 M84 Y86 C87 D91 A135 F138 D149 D141 K143 A145 N146 D159 T179 D131 K133 A135 N136 D149 T154 2.7.11.1 0004672,0005524,0006468 ic50=1.18uM remove_due_to_license_issue IC50=1180nM P51955 21366329 1280 SRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSRDLKPANVFLDGKQNVKLGDFFVGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xnp A 1.98 BS01 WCX A 1 I14 G15 Y19 C22 Y88 C89 E90 G92 D93 F148 G158 D159 F160 I12 G13 Y16 C19 Y85 C86 E87 G89 D90 F138 G148 D149 F150 D141 K143 A145 N146 D159 T179 D131 K133 A135 N136 D149 T156 2.7.11.1 0004672,0005524,0006468 ic50=0.36uM remove_due_to_license_issue IC50=570nM P51955 21366329 1280 SRAEDYEVLYTIGTGYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSHRDLKPANVFLDGKQNVKLGDFGLFVGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 2xnr A 1.6 BS01 rna C 0 R331 F333 N361 K363 F366 F368 I395 E397 S399 S400 S401 R4 F6 N34 K36 F39 F41 I68 E70 S72 S73 S74 ? 0003676,0003723 remove_due_to_license_issue P38996 20805243 0 ~ 4 MKSRLFIGNLPLKNVSKEDLFRIFSPYGHIMQINIKNAFGFIQFDNPQSVRDAIECESQEMNFGKKLILEVSSSN 2xo8 A 2.4 BS01 H70 A 1 K265 A424 G427 R428 L431 D590 K264 A423 G426 R427 L430 D589 S181 G182 T186 N233 S236 S237 G457 E459 S180 G181 T185 N232 S235 S236 G456 E458 ? 0003774,0005524,0016459,0051015 remove_due_to_license_issue P08799 21534527 1778 DPIHDRTSDYHKYLKVKQGDSDLFKLTVSDKRYIWYNPDPKERDSYECGEIVSETSDSFTFKTVDGQDRQVKKDDANQRNPIKFDGVEDMSELSYLNEPAVFHNLRVRYNQDLIYTYSGLFLVAVNPFKIIPIYTQEMVDIFKGRRRNEVAPHIFAISDVAYRSMLDDRQNQSLLITGESGAGKTENTKKVIQYLASVAGRNQANGSGVLEQQILQANPILEAFGNAKTTRNNNSSRFGKFIEIQFNSAGFISGASIQSYLLEKSRVVFQSETERNYHIFYQLLAGATAEEKKALHLAGPESFNYLNQSGCVDIKGVSDSEEFKITRQAMDIVGFSQEEQMSIFKIIAGILHLGNIKFEKGAGEGAVLKDKTALNAASTVFGVNPSVLEKALMEPRILAGRDLVAQHLNVEKSSSSRDALVKALYGRLFLWLVIKINNVLCQERKAYFIGVLDISGFEIFKVNSFEQLCINYTNEKLQQFFNHHMFKLEQEEYLKEKINWTFIDFGLDSQATIDLIDGRQPPGILALLDEQSVFPNATDNTLITKLHSHFSKKNAKYEEPRFSKTEFGVTHYAGQVMYEIQDWLEKNKDPLQQDLELCFKDSSDNVVTKLFNDPNIASRAKKGANFITVAAQYKEQLASLMATLETTNPHFVRCIIPNNKQLPAKLEDKVVLDQLRCNGVLEGIRITRKGFPNRIIYADFVKRYYLLAPNVPRDAEDSQKATDAVLKHLNIDPEQYRFGITKIFFRAGQLARIEEAREQRLESNEPPMDFDDDIPF 2xog A 1.72 BS01 SFB A 1 V43 N44 T45 N67 Q69 N71 A109 H119 F120 V40 N41 T42 N64 Q66 N68 A106 H116 F117 H12 K41 H119 F120 D121 H11 K38 H116 F117 D118 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=0.37mM remove_due_to_license_issue P61823 21205197 1125 ETAAAKFERQHMDSSTASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 2xoi A 1.72 BS01 SFB A 1 N44 T45 N67 N71 A109 H119 F120 N43 T44 N66 N70 A108 H118 F119 H12 K41 H119 F120 D121 H11 K40 H118 F119 D120 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=0.00046M remove_due_to_license_issue P61823 21205197 1125 ETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 2xow A 2.09 BS01 ISM A 1 H150 F197 G198 G199 S201 F245 M247 M249 A250 A253 H254 H59 F106 G107 G108 S110 F154 M156 M158 A159 A162 H163 3.4.21.105 0004252,0006508,0016020 remove_due_to_license_issue P09391 20890268 401 RAGPVTWVMMIACVVVFIAMQILGDQEVMLWLAWPFDPTLKFEFWRYFTHALMHFSLMHILFNLLWWWYLGGAVEKRLGSGKLIVITLISALLSGYVQQKFSGPWFGGLSGVVYALMGYVWLRGERDPQSGIYLQRGLIIFALIWIVAGWFDLFGMSMANGAHIAGLAVGLAMAFVDSL 2xp2 A 1.9 BS01 VGH A 1 A1148 M1199 A1200 G1202 P1215 N1254 L1256 G1269 I1399 E1400 A46 M97 A98 G100 P113 N149 L151 G164 I284 E285 D1249 A1251 R1253 N1254 D1270 D144 A146 R148 N149 D165 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 21812414 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 2xp3 A 2.0 BS01 B21 A 1 H59 K63 R68 C113 L122 Q131 F134 S154 H41 K45 R50 C95 L104 Q113 F116 S136 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 remove_due_to_license_issue IC50=>1000000nM Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xp4 A 1.8 BS01 G14 A 1 H59 L61 K63 R68 C113 L122 F134 S154 H157 H40 L42 K44 R49 C94 L103 F115 S135 H138 H59 C113 Q131 S154 H157 H40 C94 Q112 S135 H138 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=180uM remove_due_to_license_issue Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xp5 A 1.9 BS01 4FF A 1 H59 K63 R68 C113 L122 S154 H157 H41 K45 R50 C95 L104 S136 H139 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=360uM remove_due_to_license_issue Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xp6 A 1.9 BS01 4G2 A 1 H59 K63 R68 R69 C113 L122 F134 S154 H157 H41 K45 R50 R51 C95 L104 F116 S136 H139 H59 C113 A131 S154 H157 H41 C95 A113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=20uM remove_due_to_license_issue Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMAKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xp7 A 2.0 BS01 4F8 A 1 K63 R68 R69 C113 F134 S154 H157 K45 R50 R51 C95 F116 S136 H139 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 Kd=1.7uM remove_due_to_license_issue Kd=1700nM, IC50=1460nM Q13526 20932746 1164 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xp8 A 2.1 BS01 4FY A 1 H59 K63 R68 C113 Q131 S154 H157 H41 K45 R50 C95 Q113 S136 H139 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=15uM remove_due_to_license_issue IC50=15000nM Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xpa A 1.9 BS01 4G5 A 1 H59 K63 R68 R69 C113 L122 S154 H157 H42 K46 R51 R52 C96 L105 S137 H140 H59 C113 Q131 S154 H157 H42 C96 Q114 S137 H140 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=4.1uM remove_due_to_license_issue IC50=4100nM Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSGEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xpb A 2.0 BS01 4GE A 1 H59 K63 R68 R69 C113 L122 Q131 F134 S154 H157 H42 K46 R51 R52 C96 L105 Q114 F117 S137 H140 H59 C113 Q131 S154 H157 H42 C96 Q114 S137 H140 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=2uM remove_due_to_license_issue IC50=2000nM Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSGEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 2xpc A 1.49 BS01 051 A 1 D35 T36 R37 S71 G73 H183 K348 A414 S415 L416 N421 F422 D35 T36 R37 S71 G73 H183 K344 A410 S411 L412 N417 F418 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 Ki=125uM remove_due_to_license_issue P14900 21524830 500 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRRCVSFGVNMGDYHLNHQQGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2xpk A 2.4 BS01 Z0M A 1 G187 K218 D297 D298 C331 Y335 V370 W394 D401 G148 K179 D258 D259 C292 Y296 V331 W355 D362 3.2.1.169 Ki=0.005nM remove_due_to_license_issue Q0TR53 21095575 1625 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITCPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYDRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2xpk B 2.4 BS01 Z0M B 1 G187 K218 D297 D298 C331 Y335 T366 V370 W394 D401 G148 K179 D258 D259 C292 Y296 T327 V331 W355 D362 3.2.1.169 Ki=0.005nM remove_due_to_license_issue Q0TR53 21095575 1625 QVLVPNLNPTPENLEVVGDGFKITSSINLVGEEEADENAVNALREFLTANNIEINSENDPNSTTLIIGEVDDDIPELDEALNGTTAENLKEEGYALVSNDGKIAIEGKDGDGTFYGVQTFKQLVKESNIPEVNITDYPTVSARGIVEGFYGTPWTHQDRLDQIKFYGENKLNTYIYAPKDDPYHREKWREPYPESEMQRMQELINASAENKVDFVFGISPGIDIRFDGDAGEEDFNHLITKAESLYDMGVRSFAIYWDDIQDKSAAKHAQVLNRFNEEFVKAKGDVKPLITCPTEYDTGAMVSNGQPRAYTRIFAETVDPSIEVMWTGPGVVTNEIPLSDAQLISGIYDRNMAVWWNYPVTDYFKGKLALGPMHGLDKGLNQYVDFFTVNPMEHAELSKISIHTAADYSWNMDNYDYDKAWNRAIDMLYGDLAEDMKVFANHSTRMDNKTWAKSGREDAPELRAKMDELWNKLSSKEDASALIEELYGEFARMEEACNNLKANLPEVALEECSRQLDELITLAQGDKASLDMIVAQLNEDTEAYESAKEIAQNKLNTALSSFAVISEKVAQSFIQEALSFDLTLI 2xru A 2.9 BS01 400 A 1 L139 V147 A160 K162 L194 E211 Y212 A213 P214 L215 G216 N261 L263 D274 S388 L14 V22 A35 K37 L69 E86 Y87 A88 P89 L90 G91 N136 L138 D149 S253 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 20817473 1389 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 2xrz A 2.2 BS01 dna C 0 A160 H161 R164 N257 E301 W305 Y376 M379 W421 R429 W431 R441 Y442 M443 S444 R450 K451 A159 H160 R163 N245 E289 W293 Y364 M367 W409 R417 W419 R429 Y430 M431 S432 R438 K439 E301 W305 A335 G375 E289 W293 A323 G363 4.1.99.3 0000166,0000719,0003677,0003904,0006281,0016829 remove_due_to_license_issue Q8PYK9 21892138 3 ~ 14 HMNPKRIRALKSGKQGDGPVVYWMSRDQRAEDNWALLFSRAIAKEANVPVVVVFCLTDEFLEAGIRQYEFMLKGLQELEVSLSRKKIPSFFLRGDPGEKISRFVKDYNAGTLVTDFSPLRIKNQWIEKVISGISIPFFEVDAHNVVPCWEASQKHEYAAHTFRPKLYALLPEFLEEFPELEPNSVETLSDVLETGVKALLPERALLKNKDPLFEPWHFEPGEKAAKKVMESFIADRLDSYGALRNDPTKNMLSNLSPYLHFGQISSQRVVLEVEKAESNPGSKKAFLDEILIWKEISDNFCYYNPGYDGFESFPSWAKESLNAHRNDVRSHIYTLEEFEAGKTHDPLWNASQMELLSTGKMHGYTRMYWAKKILEWSESPEKALEIAICLNDRYELDGRDPNGYAGIAWSIGGVHDRAWGEREVTGKIRYMSYEGCKRKFDVKLYIEKYS 2xrz A 2.2 BS02 dna D 0 Y158 R429 A430 W431 Y157 R417 A418 W419 E301 W305 A335 G375 E289 W293 A323 G363 4.1.99.3 0000166,0000719,0003677,0003904,0006281,0016829 remove_due_to_license_issue Q8PYK9 21892138 1 ~ 14 HMNPKRIRALKSGKQGDGPVVYWMSRDQRAEDNWALLFSRAIAKEANVPVVVVFCLTDEFLEAGIRQYEFMLKGLQELEVSLSRKKIPSFFLRGDPGEKISRFVKDYNAGTLVTDFSPLRIKNQWIEKVISGISIPFFEVDAHNVVPCWEASQKHEYAAHTFRPKLYALLPEFLEEFPELEPNSVETLSDVLETGVKALLPERALLKNKDPLFEPWHFEPGEKAAKKVMESFIADRLDSYGALRNDPTKNMLSNLSPYLHFGQISSQRVVLEVEKAESNPGSKKAFLDEILIWKEISDNFCYYNPGYDGFESFPSWAKESLNAHRNDVRSHIYTLEEFEAGKTHDPLWNASQMELLSTGKMHGYTRMYWAKKILEWSESPEKALEIAICLNDRYELDGRDPNGYAGIAWSIGGVHDRAWGEREVTGKIRYMSYEGCKRKFDVKLYIEKYS 2xrz B 2.2 BS01 dna E 0 A160 H161 N257 E301 W305 M379 W421 R429 W431 R441 Y442 M443 S444 R450 K451 A165 H166 N229 E273 W277 M351 W393 R401 W403 R413 Y414 M415 S416 R422 K423 E301 W305 A335 G375 E273 W277 A307 G347 4.1.99.3 0000166,0000719,0003677,0003904,0006281,0016829 remove_due_to_license_issue Q8PYK9 21892138 4 ~ 14 LVPRGSHMNPKRIRALKSGKQGDGPVVYWMSRDQRAEDNWALLFSRAIAKEANVPVVVVFCLTDEFLEAGIRQYEFMLKGLQELEVSLSRKKIPSFFLRGDPGEKISRFVKDYNAGTLVTDFSPLRIKNQWIEKVISGISIPFFEVDAHNVVPCWEASQKHEYAAHTFRPKLYALLPEFLEEFPELEPNSVTKDPLFEPWHFEPGEKAAKKVMESFIADRLDSYGALRNDPTKNMLSNLSPYLHFGQISSQRVVLEVEKAESNPGSKKAFLDEILIWKEISDNFCYYNPGYDGFESFPSWAKESLNAHRNDVRSHIYTLEEFEAGKTHDPLWNASQMELLSTGKMHGYTRMYWAKKILEWSESPEKALEIAICLNDRYELDGRDPNGYAGIAWSIGGVHDRAWGEREVTGKIRYMSYEGCKRKFDVKLYIEKYS 2xrz B 2.2 BS02 dna F 0 Y158 R429 A430 W431 G432 E433 K439 R450 Y163 R401 A402 W403 G404 E405 K411 R422 E301 W305 A335 G375 E273 W277 A307 G347 4.1.99.3 0000166,0000719,0003677,0003904,0006281,0016829 remove_due_to_license_issue Q8PYK9 21892138 1 ~ 13 LVPRGSHMNPKRIRALKSGKQGDGPVVYWMSRDQRAEDNWALLFSRAIAKEANVPVVVVFCLTDEFLEAGIRQYEFMLKGLQELEVSLSRKKIPSFFLRGDPGEKISRFVKDYNAGTLVTDFSPLRIKNQWIEKVISGISIPFFEVDAHNVVPCWEASQKHEYAAHTFRPKLYALLPEFLEEFPELEPNSVTKDPLFEPWHFEPGEKAAKKVMESFIADRLDSYGALRNDPTKNMLSNLSPYLHFGQISSQRVVLEVEKAESNPGSKKAFLDEILIWKEISDNFCYYNPGYDGFESFPSWAKESLNAHRNDVRSHIYTLEEFEAGKTHDPLWNASQMELLSTGKMHGYTRMYWAKKILEWSESPEKALEIAICLNDRYELDGRDPNGYAGIAWSIGGVHDRAWGEREVTGKIRYMSYEGCKRKFDVKLYIEKYS 2xs2 A 1.35 BS01 rna B 0 F43 K70 I72 Y82 F84 K109 P112 A113 I114 R115 K116 H123 F12 K39 I41 Y51 F53 K78 P81 A82 I83 R84 K85 H87 ? 0003676,0003723,0003730 remove_due_to_license_issue Q64368 22021443 2 LPEGKIMPNTVFVGGIDVRMDETEIRSFFARYGSVKEVKIITDRTGVSKGYGFVSFYNDVDVQKIVESQINFHGKKLKLGPAIRKQH 2xsb A 2.11 BS01 GDL A 1 G8 Y160 I195 W219 N221 D226 N254 G8 Y158 I193 W217 N219 D224 N252 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0102571,1901135 ic50=11uM remove_due_to_license_issue Q2CEE3 20863279 1436 MLTGVIEGFYGRDWRRDERATVMDWIAAAGMNTYIYGPKDDVHVRARWRVPYDAAGLARLTELRDAAAARGMVFYVSLAPCLDVTYSDPQDRAALLARVDQLARAGLRNLVLLFDDIPSVLPEADRFDSFAEAQADLSNMVLRHLRGAGHVVFCPTEYCGRMAGGDPRGSAYLQRLGSTLDPAIDIFWTGPEIVSEEIVAAHLAAVGEVLRRRPVIWDNFHANDYDIRRVFAGPLGGRSRDILPLVAGWITNPNNEAEANFPAIHTTGAYLADPDYAPERAIAAAVAAWQPRFRLAFGDGAVPSDLVALLCDLFWQPFALGPETTRILSALRAALTVPRPDPSDPAWRAALEDLRDLKRRINKLFTLMTEIENRDLFHTFHNYLWEAQEEVGHLVAYCDWLDEAPPPGAVFPARGFGVAVQDIL 2xtk A 2.0 BS01 AZM A 1 Y34 D172 E174 Q230 Y232 N233 W312 Y7 D145 E147 Q203 Y205 N206 W285 3.2.1.14 0004553,0005975 ic50=164uM remove_due_to_license_issue B0Y2Y2 21044846 1339 FSNLAIYWGQGPNQLRLSHFCQETSLDIINIGFINYFPDMSPGHWPGSNFGNQCDGSVYVTNDGVVTKLLSGCHQIMEDIPICQAAGKKVLLSIGGAYPPDQSILSEDSAVAFATFLWGAFGPVAEGWEGPRPFGDVVVDGFDFDIEHNGGFGYATMVNTFRQYFNQVPERKFYLSAAPQCIIPDAQLSDAIFNAAFDFIWIQYYNTAACSAKSFIDTSLGTFNFDAWVTVLKASASKDAKLYVGLPASETAANQGYYLTPDEVESLVSTYMDRYPDTFGGIMLWEATASENNQIDGAPYADHMKDILLH 2xtn A 1.9 BS01 GTP A 1 T31 G32 G34 K35 S36 A37 S50 K51 L52 T56 L57 T58 H147 E149 N184 R185 T11 G12 G14 K15 S16 A17 S30 K31 L32 T36 L37 T38 H127 E129 N162 R163 ? 0005525 Kd=40nM remove_due_to_license_issue Q9UG22 21059949 1231 SELRIILVGKTGTGKSAAGNSILRKQAFESKLGSQTLTKTCSKSQGSWGNREIVIIDTPDMFSWKDHCEALYKEVQRCYLLSAPGPHVLLLVTQLGRYTSQDQQAAQRVKEIFGEDAMGHTIVLFTHKEDLGSLMDYMHDSDNKALSKLVAACGGRICAFNNRAEGSNQDDQVKELMDCIEDLLMEKNGDHYTNGLYSLIQRSKCGPV 2xto A 2.8 BS01 GDP A 1 G32 G34 K35 S36 A37 S50 K51 H147 E149 N183 N184 R185 G12 G14 K15 S16 A17 S30 K31 H127 E129 N163 N164 R165 ? 0005525 remove_due_to_license_issue Q9UG22 21059949 1256 SELRIILVGKTGTGKSAAGNSILRKQAFESKLGSQTLTKTCSKSQGSWGNREIVIIDTPDMFSWKDHCEALYKEVQRCYLLSAPGPHVLLLVTQLGRYTSQDQQAAQRVKEIFGEDAMGHTIVLFTHKEDLNGGSLMDYMHDSDNKALSKLVAACGGRICAFNNRAEGSNQDDQVKELMDCIEDLLMEKNGDHYTNGLYSLIQRVKEFKQSLIKYMETQRSYTA 2xu1 A 1.45 BS01 424 A 1 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A214 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A209 Q19 C25 H163 N187 Q19 C25 H163 N182 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21184410 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDAGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFENNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2xu3 A 0.9 BS01 XU3 A 1 G23 C25 G67 G68 L69 M70 A135 M161 D162 H163 A214 G23 C25 G67 G68 L69 M70 A135 M161 D162 H163 A214 Q19 C25 H163 N187 Q19 C25 H163 N187 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21184410 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2xu4 A 1.12 BS01 DJT A 1 G23 C25 E63 G67 G68 M70 A135 M161 D162 H163 A214 G23 C25 E63 G67 G68 M70 A135 M161 D162 H163 A211 Q19 C25 H163 N187 Q19 C25 H163 N184 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21184410 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2xu5 A 1.6 BS01 XU5 A 1 G23 C25 G67 G68 L69 M70 A135 M161 D162 G23 C25 G67 G68 L69 M70 A135 M161 D162 Q19 C25 H163 N187 Q19 C25 H163 N183 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21184410 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFEDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2xuc A 2.3 BS01 XRG A 1 Y34 D172 E174 Q230 Y232 W312 Y7 D145 E147 Q203 Y205 W285 3.2.1.14 0004553,0005975 ic50=79uM remove_due_to_license_issue Q873Y0 21168763 1338 FSNLAIYWGQGPNQLRLSHFCQETSLDIINIGFINYFPDMSPGHWPGSNFGNQCDGSVYVTNDGVVTKLLSGCHQIMEDIPICQAAGKKVLLSIGGAYPPDQSILSEDSAVAFATFLWGAFGPVAEGWEGPRPFGDVVVDGFDFDIEHNGGFGYATMVNTFRQYFNQVPERKFYLSAAPQCIIPDAQLSDAIFNAAFDFIWIQYYNTAACSAKSFIDTSLGTFNFDAWVTVLKASASKDAKLYVGLPASETAANQGYYLTPDEVESLVSTYMDRYPDTFGGIMLWEATASENNQIDGAPYADHMKDILLH 2xuc A 2.3 BS02 XRG A 2 Q37 N76 A124 W312 Q10 N49 A97 W285 3.2.1.14 0004553,0005975 ic50=79uM remove_due_to_license_issue Q873Y0 21168763 1339 FSNLAIYWGQGPNQLRLSHFCQETSLDIINIGFINYFPDMSPGHWPGSNFGNQCDGSVYVTNDGVVTKLLSGCHQIMEDIPICQAAGKKVLLSIGGAYPPDQSILSEDSAVAFATFLWGAFGPVAEGWEGPRPFGDVVVDGFDFDIEHNGGFGYATMVNTFRQYFNQVPERKFYLSAAPQCIIPDAQLSDAIFNAAFDFIWIQYYNTAACSAKSFIDTSLGTFNFDAWVTVLKASASKDAKLYVGLPASETAANQGYYLTPDEVESLVSTYMDRYPDTFGGIMLWEATASENNQIDGAPYADHMKDILLH 2xuf A 2.55 BS01 TZ4 A 1 Y72 W86 Y124 E202 W286 A337 F338 Y341 H447 Y70 W84 Y122 E200 W279 A330 F331 Y334 H440 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G119 G120 G152 S201 A202 G240 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 21090615 1545 REDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSAFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 2xui A 2.6 BS01 TZ5 A 1 Y72 W86 G121 Y124 W286 S293 A337 F338 Y341 W439 H447 Y72 W86 G121 Y124 W281 S288 A332 F333 Y336 W434 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Ki=0.410nM, Kd=0.00041nM P21836 21090615 1545 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSAFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 2xup A 2.7 BS02 TZ5 A 1 Y72 D74 W86 G121 Y124 E202 W286 S293 F338 Y341 W439 H447 Y72 D74 W86 G121 Y124 E202 W281 S288 F333 Y336 W434 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Ki=0.410nM, Kd=0.00041nM P21836 21090615 1548 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSAFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 2xuz A 1.9 BS01 EB4 A 1 K84 M85 K105 F106 R180 Y187 Q215 K66 M67 K87 F88 R162 Y169 Q197 ? 0005737,0005886,0006826,0030288,0045121,1901678 remove_due_to_license_issue P40409 21802011 1300 KKKIEYLDKTYEVTVPTDKIAITGSVESMEDAKLLDVHPQGAISFSGKFPDMFKDITDKAEPTGEKMEPNIEKILEMKPDVILASTKFPEKTLQKISTAGTTIPVSHISSNWKENMMLLAQLTGKEKKAKKIIADYEQDLKETKTKINDKAKDSKALVIRIRQGNIYIYPEQVYFNSTLYGDLGLKAPNEVKAAKAQELISLEKLSEMNPDHIFVQFSDDENADKPDALKDLEKNPIWKSLKAVKEDHVYVNSVDPLAQGGTAWSKVRFLKAAAEKLTQNK 2xv1 A 2.15 BS01 ECA A 1 K84 M85 K105 F106 R180 Y187 Q215 K67 M68 K88 F89 R163 Y170 Q198 ? 0005737,0005886,0006826,0030288,0045121,1901678 Kd=1.03uM remove_due_to_license_issue P40409 21802011 1301 EKKKIEYLDKTYEVTVPTDKIAITGSVESMEDAKLLDVHPQGAISFSGKFPDMFKDITDKAEPTGEKMEPNIEKILEMKPDVILASTKFPEKTLQKISTAGTTIPVSHISSNWKENMMLLAQLTGKEKKAKKIIADYEQDLKETKTKINDKAKDSKALVIRIRQGNIYIYPEQVYFNSTLYGDLGLKAPNEVKAAKAQELISLEKLSEMNPDHIFVQFSDDENADKPDALKDLEKNPIWKSLKAVKEDHVYVNSVDPLAQGGTAWSKVRFLKAAAEKLTQNKL 2xvd A 1.7 BS01 AS6 A 1 I621 V629 A645 K647 E664 T693 M696 E697 G699 L747 S757 D758 I15 V23 A39 K41 E55 T84 M87 E88 G90 L138 S148 D149 D740 A742 R744 N745 D758 K781 P783 D131 A133 R135 N136 D149 K163 P165 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.002uM remove_due_to_license_issue IC50=7nM P54760 21441027 1889 AKEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFLESSLGGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 2xvn A 2.35 BS01 KLS A 1 Y34 A124 D172 E174 Q230 Y232 W312 Y6 A96 D144 E146 Q202 Y204 W284 3.2.1.14 0004553,0005975 ic50=112uM remove_due_to_license_issue Q873Y0 21168763 1338 SNLAIYWGQGPNQLRLSHFCQETSLDIINIGFINYFPDMSPGHWPGSNFGNQCDGSVYVTNDGVVTKLLSGCHQIMEDIPICQAAGKKVLLSIGGAYPPDQSILSEDSAVAFATFLWGAFGPVAEGWEGPRPFGDVVVDGFDFDIEHNGGFGYATMVNTFRQYFNQVPERKFYLSAAPQCIIPDAQLSDAIFNAAFDFIWIQYYNTAACSAKSFIDTSLGTFNFDAWVTVLKASASKDAKLYVGLPASETAANQGYYLTPDEVESLVSTYMDRYPDTFGGIMLWEATASENNQIDGAPYADHMKDILLH 2xwd A 2.66 BS01 LGS A 1 D127 F128 E235 Y313 E340 W381 D123 F124 E231 Y309 E336 W377 E235 E340 C342 N370 E231 E336 C338 N366 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 remove_due_to_license_issue P04062 21483943 610 FARPCIPKSFGYSSVVCVCNATYCDSFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 2xwe A 2.31 BS01 AMF A 1 D127 F128 N234 E235 Y313 E340 C342 S345 W381 D126 F127 N233 E234 Y312 E339 C341 S344 W380 E235 E340 C342 N370 E234 E339 C341 N369 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 Ka=2113M^-1 remove_due_to_license_issue P04062 21483943 607 FARPCIPKSFGYSSVVCVCNATYCDSFDPPPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 2xwy A 2.53 BS01 IB8 A 1 V37 A395 A396 H428 G493 V494 P495 R503 V16 A371 A372 H404 G469 V470 P471 R479 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 21141896 1532 SMSYTWTGALITPCMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVK 2xx2 A 1.85 BS01 13C A 1 N37 A41 K44 D79 I82 M84 N92 F124 T171 L173 N37 A41 K44 D79 I82 M84 N92 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 21932796 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2xx4 A 2.199 BS01 13I A 1 N37 A41 K44 D79 I82 M84 N92 F124 T171 L173 N37 A41 K44 D79 I82 M84 N92 F121 T168 L170 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 21932796 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2xx5 A 2.0 BS01 13N A 1 N37 A41 D79 I82 M84 L89 N92 L93 F124 W148 T171 L173 N37 A41 D79 I82 M84 L89 N92 L93 F121 W145 T168 L170 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 21932796 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2xxr A 1.6 BS01 GLU A 1 Y488 A518 R523 G688 A689 T690 E738 Y57 A87 R92 G137 A138 T139 E187 ? 0015276,0016020 remove_due_to_license_issue P42260 21414913 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWW 2xxt A 1.9 BS01 KAI A 1 E440 Y488 P516 A518 R523 G688 A689 T690 E738 E9 Y57 P85 A87 R92 G137 A138 T139 E187 ? 0015276,0016020 remove_due_to_license_issue Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 21414913 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWW 2xxw A 2.3 BS01 GLU A 1 Y488 A518 R523 G688 A689 T690 E738 Y58 A88 R93 G138 A139 T140 E188 ? 0015276,0016020 remove_due_to_license_issue P42260 21414913 900 RSLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRKKITIAILQLQEEGKLHMMKEKWWR 2xxx A 2.098 BS01 GLU A 1 Y488 P516 L517 A518 R523 G688 A689 T690 E738 Y57 P85 L86 A87 R92 G137 A138 T139 E187 ? 0015276,0016020 remove_due_to_license_issue P42260 21414913 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRKKITIAILQLQEEGKLHMMKEKWW 2xxy A 3.0 BS01 KAI A 1 E440 Y488 P516 A518 R523 G688 A689 T690 E738 E9 Y57 P85 A87 R92 G137 A138 T139 E187 ? 0015276,0016020 remove_due_to_license_issue Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 21414913 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRKKITIAILQLQEEGKLHMMKEKWW 2xy9 A 1.97 BS03 3ES A 1 Q281 H353 A354 S355 A356 E376 V380 H383 E384 H387 F391 H410 F457 K511 F512 H513 V518 Y520 Y523 F527 Q242 H314 A315 S316 A317 E337 V341 H344 E345 H348 F352 H371 F414 K468 F469 H470 V475 Y477 Y480 F484 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H470 Y480 3.4.15.1 0006508,0008237,0008241,0016020 Ki=0.65nM remove_due_to_license_issue Ki=0.65nM P12821 21352096 1635 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPA 2xy9 A 1.97 BS04 3ES A 2 W59 Y62 N66 E123 W220 M223 W357 P519 R522 W20 Y23 N27 E84 W181 M184 W318 P476 R479 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H470 Y480 3.4.15.1 0006508,0008237,0008241,0016020 Ki=0.65nM remove_due_to_license_issue Ki=0.65nM P12821 21352096 1636 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPA 2xyd A 2.15 BS01 3ES A 1 Q259 H331 A332 S333 T358 H361 E362 H365 Y369 H388 E389 D393 F435 K489 F490 H491 T496 Y498 Y501 F505 Q256 H328 A329 S330 T355 H358 E359 H362 Y366 H385 E386 D390 F432 K486 F487 H488 T493 Y495 Y498 F502 H331 A332 H361 E362 H365 E389 H491 Y501 H328 A329 H358 E359 H362 E386 H488 Y498 3.4.15.1 0006508,0008237,0008241,0016020 Ki=150nM remove_due_to_license_issue Ki=0.65nM P12821 21352096 1611 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 2xye A 2.0 BS01 CXG B 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 T82 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 2xye B 2.0 BS01 CXG B 1 L123 D125 G127 A128 D129 G148 G149 I150 F153 P181 T182 L23 D25 G27 A28 D29 G48 G49 I50 F53 P81 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 2xyf A 1.8 BS01 G40 B 1 D25 G27 A28 D29 D30 G48 I50 P81 T82 D25 G27 A28 D29 D30 G48 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 2xyf B 1.8 BS01 G40 B 1 L123 D125 G127 A128 D129 G148 G149 F153 P181 T182 L23 D25 G27 A28 D29 G48 G49 F53 P81 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 2xyn A 2.81 BS01 VX6 A 1 L294 Y299 V302 A315 T361 E362 Y363 M364 P365 Y366 G367 L416 D427 L15 Y20 V23 A36 T80 E81 Y82 M83 P84 Y85 G86 L135 D146 D409 A411 R413 N414 D427 P448 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=4nM P42684 21417343 547 KWEMERTDITMKHKLGGGQYGEVYVGVWKKYSLTVAVKTLDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTLEPPFYIVTEYMPYGNLLDYLRECNREEVTAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHVVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNTFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYDLLEKGYRMEQPEGCPPKVYELMRACWKWSPADRPSFAETHQAFETMFHD 2xyr A 2.5 BS01 SFG A 1 N43 G71 G73 P80 G81 D99 L100 C115 D130 M131 Y132 N41 G69 G71 P78 G79 D97 L98 C113 D128 M129 Y130 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0004483 remove_due_to_license_issue P0C6X7 21637813 1298 QAWQPGVAMPNLYKMQRMLLEKCDLQNYGENAVIPKGIMMNVAKYTQLCQYLNTLTLAVPYNMRVIHFGAGSDKGVAPGTAVLRQWLPTGTLLVDSDLNDFVSDADSTLIGDCATVHTANKWDLIISDMYDPRTKENDSKEGFFTYLCGFIKQKLALGGSIAVKITEHSWNADLYKLMGHFSWWTAFVTNVNASSSEAFLIGANYLGKPKEQIDGYTMHANYIFWRNTNPIQLSSYSLFDMSKFPLKLRGTAVMSLKENQINDMIYSLLEKGRLIIRENNRVVVSS 2xys A 1.909 BS01 SY9 A 1 Y91 W145 C188 C189 Y193 Y91 W145 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Ki=38nM remove_due_to_license_issue Q8WSF8 21468359 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2xys A 1.909 BS02 SY9 E 2 Q55 I116 D162 Q55 I116 D162 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Ki=38nM remove_due_to_license_issue Q8WSF8 21468359 1207 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2xys B 1.909 BS01 SY9 A 1 Y53 Q55 I116 Y53 Q55 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Ki=38nM remove_due_to_license_issue Q8WSF8 21468359 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2xys B 1.909 BS02 SY9 B 1 Y91 W145 Y186 C188 C189 Y193 Y91 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Ki=38nM remove_due_to_license_issue Q8WSF8 21468359 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2xyt B 2.05 BS01 TC9 B 1 Y91 K141 Y186 Y91 K141 Y186 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Ki=509.2nM remove_due_to_license_issue Q8WSF8 21468359 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2xyt C 2.05 BS01 TC9 B 1 T34 Y53 Q55 S164 S165 T34 Y53 Q55 S164 S165 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21468359 1206 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2xyu A 2.117 BS01 Q9G A 1 A651 K653 M674 T699 Y701 M702 L753 S763 A40 K42 M63 T88 Y90 M91 L142 S152 D746 A748 R750 N751 D764 I786 D135 A137 R139 N140 D153 I155 2.7.10.1 0004672,0004713,0005524,0006468 ic50=4.5uM remove_due_to_license_issue Q03137 22137457 1898 FAKEIDASCIKIEKVIGVGEFGEVCSGRLKVPGKREICVAIKTLKAGYTDKQRRDFLSEASIMGQFDHPNIIHLEGVVTKCKPVMIITEYMENGSLDAFLRKNDGRFTVIQLVGMLRGIGSGMKYLSDMSYVHRDLAARNILVNSNLVCKVSDFIPIRWTAPEAIAYRKFTSASDVWSYGIVMWEVMSYGERPYWDMSNQDVIKAIEEGYRLPPPMDCPIALHQLMLDCWQKERSDRPKFGQIVNMLDKLIRNPNSLKRT 2xz5 A 2.8 BS01 ACH A 1 W145 Y186 Y193 W145 Y186 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21115477 1210 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYCEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2xz5 A 2.8 BS02 ACH A 2 W145 Y186 S187 C188 W145 Y186 S187 C188 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21115477 1211 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYCEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2xz5 A 2.8 BS04 ACH C 2 T34 S165 T34 S165 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21115477 1211 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYCEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2xz5 B 2.8 BS01 ACH B 1 Y91 W145 Y186 Y193 Y91 W145 Y186 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21115477 1210 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYCEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2xz5 B 2.8 BS02 ACH B 2 Y186 C188 Y186 C188 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21115477 1211 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYCEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRA 2xzc L 1.36 BS01 XOP L 1 Y37 G90 T91 W92 P98 F100 Y37 G90 T91 W92 P98 F100 remove_due_to_license_issue 21896761 1217 ESVLTQPPSVSAAPGQKVTISCSGSSSNIGNNYVSWYQQLPGTAPKLLIYDNNKRPSGIPDRFSGSKSGTSATLGITGLQTGDEADYYCGTWDSSLNPVFGGGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGE 2xzf A 1.799 BS01 dna B 0 P1 E2 K57 H72 R74 M75 K129 G170 N171 I172 Y238 K254 K256 R260 P1 E2 K57 H72 R74 M75 K129 G170 N171 I172 Y233 K249 K251 R255 P1 E2 P1 E2 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 21486746 1 ~ 14 PELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 2xzf A 1.799 BS02 dna C 0 K90 H91 V108 R109 F111 K90 H91 V108 R109 F111 P1 E2 P1 E2 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 21486746 15 ~ 28 PELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 2xzg A 1.7 BS01 VH1 A 1 R64 I66 L82 F91 I93 K96 R65 I67 L83 F92 I94 K97 ? 0005198,0006886,0016192,0030130,0030132 remove_due_to_license_issue IC50=18000nM Q00610 21816279 1362 FMAQILPIRFQEHLQLQNLGINPANIGFSTLTMESDKFICIREKVGEQAQVVIIDMNDPSNPIRRPISADSAIMNPASKVIALKAGKTLQIFNIEMKSKMKAHTMTDDVTFWKWISLNTVALVTDNAVYHWSMEGESQPVKMFDRHSSLAGCQIINYRTDAKQKWLLLTGISAQQNRVVGAMQLYSVDRKVSQPIEGHAASFAQFKMEGNAEESTLFCFAVRGQAGGKLHIIEVGTPPTGNQPFPKKAVDVFFPPEAQNDFPVAMQISEKHDVVFLITKYGYIHLYDLETGTCIYMNRISGETIFVTAPHEATAGIIGVNRKGQVLSVCVEEENIIPYITNVLQNPDLALRMAVRNNL 2xzl A 2.4 BS01 rna B 0 D297 E298 Y316 K354 T356 S357 P460 N462 A484 K485 S486 T553 V555 V605 L607 T698 S699 Y732 E733 S761 D763 G787 F788 D206 E207 Y225 K260 T262 S263 P366 N368 A390 K391 S392 T459 V461 V511 L513 T604 S605 Y638 E639 S667 D669 G693 F694 3.6.4.12,3.6.4.13 0000184,0003723,0003724,0004386,0005524,0005737,0008270,0016887 remove_due_to_license_issue P30771 21419344 1 ~ 9 NSCAYCGIDSAKCVIKCNSCKKWFCNTKNGTSSSHIVNHLVLSHHNVVSLHPDSDLGDTVLECYNCGRKNVFLLGFVSVVLLCRIPCAQTKWDTDQWQPLIEDRQLLSWVAEQPTEEEKLKARLITPSQISKLEAKWRSNKDATIPPLLLRYQDAYEYQRSYGPLIKLEADYDKQLKESQEHISVSWSLALNNRHLASFTKVAIGDEMILWYSGMQHPDWEGRGYIVRLPNDTFTLELKPSKTPPPTHLTTGFTAEFIWKGTSYDRMQDALKKFAIDKKSISGYLYYKILGHQVVDISFDVPLPKEFSIPNFAQLNSSQSNAVSHVLQRPLSLIQGPPGTGKTVTSATIVYHLSKIHKDRILVCAPSNVAVDHLAAKLRDLGLKVVRLTAKSREDVESSVSNLALHNLVGRGAKGELKNLLKLKDEVGELSASDTKRFVKLVRKTEAEILNKADVVCCTCVGAGDKRLDTKFRTVLIDESTQASEPECLIPIVKGAKQVILVGDHQQLGPVILERKAADAGLKQSLFERLISLGHVPIRLEVQYRMNPYLSEFPSNMFYEGSLQNGVTIEQRTVPNSKFPWPIRGIPMMFWANYGREEISANGTSFLNRIEAMNCERIITKLFRDGVKPEQIGVITPYEGQRAYILQYMQMNGSLDKDLYIKVEVASVDAFQGREKDYIILSCVRANEQQAIGFLRDPRRLNVGLTRAKYGLVILGNPRSLARNTLWNHLLIHFREKGCLVEGTLDNLQLCTVQLV 2xzw A 1.95 BS02 AKG A 1 G37 Q39 K40 G41 L56 K58 G87 G37 Q39 K40 G41 L50 K52 G81 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 remove_due_to_license_issue P0A3F4 21041661 201 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGRQKGQTEYTVEFLQKLKLEIVVEDAQVDTVIDKIVAAARTGEIGDGKIFVSPVDQTIRIRTGEKNADAISAW 2xzw B 1.95 BS03 AKG B 1 F36 G37 Q39 G41 L56 K58 G87 F36 G37 Q39 G41 L52 K54 G83 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 remove_due_to_license_issue P0A3F4 21041661 201 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGRQKGQTEREYTVEFLQKLKLEIVVEDAQVDTVIDKIVAAARTGEIGDGKIFVSPVDQTIRIRTGEKNADAISAW 2y0j A 2.43 BS01 AXC A 1 L665 I682 Y683 M703 Q716 F719 V723 L220 I237 Y238 M258 Q271 F274 V278 3.1.4.17 0004114,0007165,0008081 ic50=12nM remove_due_to_license_issue IC50=12nM Q9Y233 21602043 1760 WQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 2y1d A 2.05 BS01 34F A 1 D151 A176 S177 S213 N218 K219 S245 P265 D131 A156 S157 S183 N188 K189 S215 P235 0008299,0030604,0046872,0070402 remove_due_to_license_issue 21678907 1390 GRLRVVVLGSTGSIGTQALQVIADNPDRFEVVGLAAGGAHLDTLLRQRAQTGVTNIAVDIPYHGSDAATRLVEQTEADVVLNALVGALGLRPTLAALKTGARLALANKESLVAGGSLVLRAARPGQIVPVDSEHSALAQCLRGGTPDEVAKLVLTASGGPFRGWSAADLEHVTPEQAGNTLNSASLVNKGLEVIETHLLFGIPYDRIDVVVHPQSIIHSMVTFIDGSTIAQASPPDMKLPISLALGWPRRVSGAAAACDFHTASSWEFEPLDTDVFPAVELARQAGVAGGCMTAVYNAANEEAAAAFLAGRIGFPAIVGIIADVLHAADQWAVEPATVDDVLDAQRWARERAQRAVSGM 2y1g A 1.95 BS01 FM5 A 1 D151 A176 S177 S213 N218 K219 S245 P265 D141 A166 S167 S198 N203 K204 S230 P250 0008299,0030604,0046872,0070402 ic50=0.7uM remove_due_to_license_issue 21678907 1390 GRLRVVVLGSTGSIGTQALQVIADNPDRFEVVGLAAGGAHLDTLLRQRAQTGVTNIAVADEHAAQRVGDIPYHGSDAATRLVEQTEADVVLNALVGALGLRPTLAALKTGARLALANKESLVAGGSLVLRAARPGQIVPVDSEHSALAQCLRGGTPDEVAKLVLTASGGPFRGWSAADLEHVTPEQAGSMGPMNTLNSASLVNKGLEVIETHLLFGIPYDRIDVVVHPQSIIHSMVTFIDGSTIAQASPPDMKLPISLALGWPRRVSGAAAACDFHTASSWEFEPLDTDVFPAVELARQAGVAGGCMTAVYNAANEEAAAAFLAGRIGFPAIVGIIADVLHAADQWAVEPATVDDVLDAQRWARERAQRAVSGM 2y1o A 1.49 BS01 T26 A 1 D35 T36 R37 S71 G73 I139 F161 H183 A414 S415 N421 F422 D35 T36 R37 S71 G73 I139 F161 H183 A410 S411 N417 F418 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 remove_due_to_license_issue P14900 24900523 500 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRRCVSFGVNMGDYHLNHQQGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2y1w A 2.1 BS02 849 A 1 Q149 Y150 F153 Y154 M163 E258 P259 M260 Y262 E267 H415 W416 Q447 Q14 Y15 F18 Y19 M28 E123 P124 M125 Y127 E132 H280 W281 Q312 D166 E258 E267 H415 D31 E123 E132 H280 2.1.1.319 0016274,0018216 remove_due_to_license_issue IC50=30nM Q86X55 21410432 1005 SVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 2y1w C 2.1 BS02 849 C 1 Y150 F153 Y154 M163 E258 P259 M260 Y262 E267 H415 W416 Q447 Y15 F18 Y19 M28 E123 P124 M125 Y127 E132 H280 W281 Q312 D166 E258 E267 H415 D31 E123 E132 H280 2.1.1.319 0016274,0018216 remove_due_to_license_issue IC50=30nM Q86X55 21410432 1005 SVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 2y1x B 2.4 BS02 845 B 1 F153 Y154 N162 M163 E258 P259 M260 Y262 E267 H415 W416 F475 F18 Y19 N27 M28 E123 P124 M125 Y127 E132 H280 W281 F340 D166 E258 E267 H415 D31 E123 E132 H280 2.1.1.319 0016274,0018216 remove_due_to_license_issue Q86X55 21410432 1002 SVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRY 2y2h A 1.96 BS01 ZA2 A 1 A459 S460 S516 N518 M556 G558 G653 T654 A137 S138 S194 N196 M234 G236 G331 T332 2.4.1.129 0008658 remove_due_to_license_issue Q7CRA4 21732689 1000 SEITYSDGTVIASIDYLYFTTLAEAQERMYDYLAQRDNVSAKELKNEATQKFYRDLAAKEIENGGYKITTTIDQKIHSAMQSAVADYGYLLDDGTGRVEVGNVLMDNQTGAILGFVGGRNYQENQNNHAFDTKRSPASTTKPLLAYGIAIDQGLMGSETILSNYPTNFANGNPIMYANSKGTGMMTLGEALNYSWNIPAYWTYRMLRENGVDVKGYMEKMGYEIPEYGIESLPMGGGIEVTVAQHTNGYQTLANNGVYHQKHVISKIEAADGRVVYEYQDKPVQVYSKATATIMQGLLREVLSSRVTTTFKSNLTSLNPTLANADWIGKTGTTGQDENMWLMLSTPRLTLGGWIGHDDNHSLSQQAGYSNNSNYMAHLVNAIQQASPSIWGNERFALDPSVVKSEVLKSTGQKPGKVSVEGKEVEVTGSTVTSYWANKSGAPATSYRFAIGGSDADYQNAWSSIVGS 2y2i A 1.78 BS01 ZA3 A 1 A459 S460 K463 S516 N518 M556 G558 T654 A138 S139 K142 S195 N197 M235 G237 T333 2.4.1.129 0008658 remove_due_to_license_issue Q7CRA4 21732689 1000 ISEITYSDGTVIASIDYLYFTTLAEAQERMYDYLAQRDNVSAKELKNEATQKFYRDLAAKEIENGGYKITTTIDQKIHSAMQSAVADYGYLLDDGTGRVEVGNVLMDNQTGAILGFVGGRNYQENQNNHAFDTKRSPASTTKPLLAYGIAIDQGLMGSETILSNYPTNFANGNPIMYANSKGTGMMTLGEALNYSWNIPAYWTYRMLRENGVDVKGYMEKMGYEIPEYGIESLPMGGGIEVTVAQHTNGYQTLANNGVYHQKHVISKIEAADGRVVYEYQDKPVQVYSKATATIMQGLLREVLSSRVTTTFKSNLTSLNPTLANADWIGKTGTTGQDENMWLMLSTPRLTLGGWIGHDDNHSLSQQAGYSNNSNYMAHLVNAIQQASPSIWGNERFALDPSVVKSEVLKSTGQKPGKVSVEGKEVEVTGSTVTSYWANKSGAPATSYRFAIGGSDADYQNAWSSIVG 2y2j A 2.06 BS01 ZA4 A 1 A459 S460 K463 S516 N518 M556 G653 T654 A140 S141 K144 S197 N199 M237 G334 T335 2.4.1.129 0008658 remove_due_to_license_issue Q7CRA4 21732689 1000 ISEITYSDGTVIASISRDYLYFTTLAEAQERMYDYLAQRDNVSAKELKNEATQKFYRDLAAKEIENGGYKITTTIDQKIHSAMQSAVADYGYLLDDGTGRVEVGNVLMDNQTGAILGFVGGRNYQENQNNHAFDTKRSPASTTKPLLAYGIAIDQGLMGSETILSNYPTNFANGNPIMYANSKGTGMMTLGEALNYSWNIPAYWTYRMLRENGVDVKGYMEKMGYEIPEYGIESLPMGGGIEVTVAQHTNGYQTLANNGVYHQKHVISKIEAADGRVVYEYQDKPVQVYSKATATIMQGLLREVLSSRVTTTFKSNLTSLNPTLANADWIGKTGTTGQDENMWLMLSTPRLTLGGWIGHDDNHSLSQQAGYSNNSNYMAHLVNAIQQASPSIWGNERFALDPSVVKSEVLKSTGQKPGKVSVEGKEVEVTGSTVTSYWANKSGAPATSYRFAIGGSDADYQNAWSSIVGS 2y2k A 2.09 BS01 ZA5 A 1 A459 S460 K463 S516 N518 M556 T654 A138 S139 K142 S195 N197 M235 T333 2.4.1.129 0008658 remove_due_to_license_issue Q7CRA4 21732689 1000 SEITYSDGTVIASIRDYLYFTTLAEAQERMYDYLAQRDNVSAKELKNEATQKFYRDLAAKEIENGGYKITTTIDQKIHSAMQSAVADYGYLLDDGTGRVEVGNVLMDNQTGAILGFVGGRNYQENQNNHAFDTKRSPASTTKPLLAYGIAIDQGLMGSETILSNYPTNFANGNPIMYANSKGTGMMTLGEALNYSWNIPAYWTYRMLRENGVDVKGYMEKMGYEIPEYGIESLPMGGGIEVTVAQHTNGYQTLANNGVYHQKHVISKIEAADGRVVYEYQDKPVQVYSKATATIMQGLLREVLSSRVTTTFKSNLTSLNPTLANADWIGKTGTTGQDENMWLMLSTPRLTLGGWIGHDDNHSLSQQAGYSNNSNYMAHLVNAIQQASPSIWGNERFALDPSVVKSEVLKSTGQKPGKVSVEGKEVEVTGSTVTSYWANKSGAPATSYRFAIGGSDADYQNAWSSIVGSL 2y2n A 2.07 BS01 E07 A 1 S460 Y498 S516 N518 M556 G653 T654 T655 G656 D658 S139 Y177 S195 N197 M235 G332 T333 T334 G335 D337 2.4.1.129 0008658 remove_due_to_license_issue Q7CRA4 21732689 1000 ISEITYSDGTVIASIDYLYFTTLAEAQERMYDYLAQRDNVSAKELKNEATQKFYRDLAAKEIENGGYKITTTIDQKIHSAMQSAVADYGYLLDDGTGRVEVGNVLMDNQTGAILGFVGGRNYQENQNNHAFDTKRSPASTTKPLLAYGIAIDQGLMGSETILSNYPTNFANGNPIMYANSKGTGMMTLGEALNYSWNIPAYWTYRMLRENGVDVKGYMEKMGYEIPEYGIESLPMGGGIEVTVAQHTNGYQTLANNGVYHQKHVISKIEAADGRVVYEYQDKPVQVYSKATATIMQGLLREVLSSRVTTTFKSNLTSLNPTLANADWIGKTGTTGQDENMWLMLSTPRLTLGGWIGHDDNHSLSQQAGYSNNSNYMAHLVNAIQQASPSIWGNERFALDPSVVKSEVLKSTGQKPGKVSVEGKEVEVTGSTVTSYWANKSGAPATSYRFAIGGSDADYQNAWSSIVGS 2y2p A 1.62 BS01 Z10 A 1 S460 Y498 S516 N518 M556 G653 T654 T655 G656 D658 S139 Y177 S195 N197 M235 G332 T333 T334 G335 D337 2.4.1.129 0008658 remove_due_to_license_issue Q7CRA4 21732689 1000 ISEITYSDGTVIASIDYLYFTTLAEAQERMYDYLAQRDNVSAKELKNEATQKFYRDLAAKEIENGGYKITTTIDQKIHSAMQSAVADYGYLLDDGTGRVEVGNVLMDNQTGAILGFVGGRNYQENQNNHAFDTKRSPASTTKPLLAYGIAIDQGLMGSETILSNYPTNFANGNPIMYANSKGTGMMTLGEALNYSWNIPAYWTYRMLRENGVDVKGYMEKMGYEIPEYGIESLPMGGGIEVTVAQHTNGYQTLANNGVYHQKHVISKIEAADGRVVYEYQDKPVQVYSKATATIMQGLLREVLSSRVTTTFKSNLTSLNPTLANADWIGKTGTTGQDENMWLMLSTPRLTLGGWIGHDDNHSLSQQAGYSNNSNYMAHLVNAIQQASPSIWGNERFALDPSVVKSEVLKSTGQKPGKVSVEVEVTGSTVTSYWANKSGAPATSYRFAIGGSDADYQNAWSSIVGSL 2y34 A 2.01 BS02 UN9 A 1 D254 M299 Y303 Y310 H313 Y329 L343 H374 V376 R383 D68 M113 Y117 Y124 H127 Y143 L157 H188 V190 R197 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=300nM, EC50=79000nM, Kd=80nM Q9GZT9 21601578 601 PLPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVK 2y34 A 2.01 BS03 UN9 A 2 W258 T296 D320 F391 W72 T110 D134 F205 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=300nM, EC50=79000nM, Kd=80nM Q9GZT9 21601578 602 PLPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVK 2y3p A 2.62 BS01 SM8 A 1 K42 H45 R91 M92 N169 A175 K20 H23 R69 M70 N147 A153 5.6.2.2 0003677,0003918,0005524,0006259,0006265 remove_due_to_license_issue P0AES5 19965760 901 DYAMSVIVGRALPDVRDGLKPVHRRVLYAMNVLGNDWNKAYKKSARVVGDVIGKYHPHGDSAVYDTIVRMAQPFSLRYMLVDGQGNFGSIDGDSAAAMRYTEIRLAKIAHELMADLEKETVDFVDNYDGTEKIPDVMPTKIPNLLVNGSSGIAVGMATNIPPHNLTEVINGCLAYIDDEDISIEGLMEHIPGPDFPTAAIINGRRGIEEAYRTGRGKVYIRARAEVEVDAKTGRETIIVHEIPYQVNKARLIEKIAELVKEKRVEGISALRDESDKDGMRIVIEVKRDAVGEVVLNNLYSQTQLQVSFGINMVALHHGQPKIMNLKDIIAAFVRHRREVVTRRTIFELRKARDRAHILEALAVALANIDPIIELIRHAPTPAEAKTALVANPWQLGNVAAMLEDAARPEWLEPEFGVRDGLYYLTEQQAQAILDLRLQKLTGLEHEKLLDEYKELLDQIAELLRILGSADRLMEVIREELELVREQFGDKRRTEIT 2y4a A 2.7 BS01 BH6 A 1 A48 S49 Y147 S298 G412 T413 M414 A48 S49 Y147 S298 G412 T413 M414 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue IC50=85000nM, Ki=42000nM P39045 21574608 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 2y4k A 2.45 BS01 GDP A 1 P7 F8 E11 Q66 G75 K76 D100 A101 D102 W189 P6 F7 E10 Q65 G74 K75 D99 A100 D101 W188 2.4.1.217 0046872 remove_due_to_license_issue D0MI02 21288903 401 SLVVFPFKHEHPEVLLHNVRVAAAHPRVHEVLCIGYERDQTYEAVERAAPEISRATGTPVSVRLQERLGTLRPGKGDGMNTALRYFLEETQWERIHFYDADITSFGPDWITKAEEAADFGYGLVRHYFPRASTDAMITWMITRTGFALLWPHTELSWIEQPLGGELLMRREVAAMLYEDERVRRRSDWGIDTLYTFVTVAAGVSIYECYIPEGKAHRLYGGLDDLRTMLVECFAAIQSLQHEVVGQPAIHRQEHPHRVPVHIAERVGYDVEATLHRLMQHWTPRQVELLELFTTPVREGLRTCQRRPAFNFMDEMAWAATYHVLLEHFQPGDPDWEELLFKLWTTRVLNYTMTVALRGYDYAQQYLYRMLGRYRYQAALE 2y4l A 2.8 BS02 GDP A 1 P7 F8 E11 Y37 Q66 G75 K76 D100 A101 D102 W189 H217 R218 P6 F7 E10 Y36 Q65 G74 K75 D99 A100 D101 W188 H216 R217 2.4.1.217 0046872 remove_due_to_license_issue D0MI02 21288903 401 SLVVFPFKHEHPEVLLHNVRVAAAHPRVHEVLCIGYERDQTYEAVERAAPEISRATGTPVSVRLQERLGTLRPGKGDGMNTALRYFLEETQWERIHFYDADITSFGPDWITKAEEAADFGYGLVRHYFPRASTDAMITWMITRTGFALLWPHTELSWIEQPLGGELLMRREVAAMLYEDERVRRRSDWGIDTLYTFVTVAAGVSIYECYIPEGKAHRLYGGLDDLRTMLVECFAAIQSLQHEVVGQPAIHRQEHPHRVPVHIAERVGYDVEATLHRLMQHWTPRQVELLELFTTPVREGLRTCQRRPAFNFMDEMAWAATYHVLLEHFQPGDPDWEELLFKLWTTRVLNYTMTVALRGYDYAQQYLYRMLGRYRYQAALE 2y4m A 2.7 BS02 GDX A 1 P7 F8 K9 E11 I35 Q66 G75 K76 D100 A101 D102 L163 G165 W189 D192 H217 P6 F7 K8 E10 I34 Q65 G74 K75 D99 A100 D101 L162 G164 W188 D191 H216 2.4.1.217 0046872 remove_due_to_license_issue D0MI02 21288903 401 SLVVFPFKHEHPEVLLHNVRVAAAHPRVHEVLCIGYERDQTYEAVERAAPEISRATGTPVSVRLQERLGTLRPGKGDGMNTALRYFLEETQWERIHFYDADITSFGPDWITKAEEAADFGYGLVRHYFPRASTDAMITWMITRTGFALLWPHTELSWIEQPLGGELLMRREVAAMLYEDERVRRRSDWGIDTLYTFVTVAAGVSIYECYIPEGKAHRLLDDLRTMLVECFAAIQSLQHEVVGQPAIHRQEHPHRVPVHIAERVGYDVEATLHRLMQHWTPRQVELLELFTTPVREGLRTCQRRPAFNFMDEMAWAATYHVLLEHFQPGDPDWEELLFKLWTTRVLNYTMTVALRGYDYAQQYLYRMLGRYRYQAALE 2y54 A 3.65 BS01 V63 A 1 W145 C188 C189 Y193 W145 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=5011.87nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y54 A 3.65 BS02 V63 E 1 Q55 I116 Q55 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=5011.87nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y54 B 3.65 BS01 V63 A 1 Q55 I116 Q55 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=5011.87nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y54 B 3.65 BS02 V63 B 1 W145 C188 Y193 W145 C188 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=5011.87nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y55 A 2.6 BS01 FP5 A 1 A48 S49 K52 S298 N300 K410 T411 G412 T413 A48 S49 K52 S298 N300 K410 T411 G412 T413 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue Ki=125000nM, IC50=320000nM P39045 21574608 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 2y56 A 3.59 BS01 V11 A 1 Y91 K141 G143 S144 W145 C188 C189 Y193 Y91 K141 G143 S144 W145 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=100nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y56 B 3.59 BS01 V11 A 1 Y53 I116 Y53 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=100nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y56 B 3.59 BS02 V11 B 1 Y91 G143 W145 Y186 C188 C189 Y193 Y91 G143 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=100nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y57 A 3.3 BS01 V37 A 1 K141 G143 S144 W145 Y186 C188 C189 Y193 D195 K141 G143 S144 W145 Y186 C188 C189 Y193 D195 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=31.62nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y57 A 3.3 BS02 V37 E 1 Y53 Q55 M114 I116 Y53 Q55 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=31.62nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y57 B 3.3 BS01 V37 A 1 Y53 Q55 I116 Y53 Q55 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=31.62nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y57 B 3.3 BS02 V37 B 1 Y91 K141 G143 S144 W145 Y186 C188 C189 Y193 D195 Y91 K141 G143 S144 W145 Y186 C188 C189 Y193 D195 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Ki=31.62nM Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y58 A 3.25 BS01 V38 A 1 Y91 W145 Y186 C188 C189 Y193 Y91 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y58 A 3.25 BS02 V38 E 1 Q36 Y53 I116 Q36 Y53 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y58 B 3.25 BS01 V38 A 1 Q36 Y53 I116 Q36 Y53 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y58 B 3.25 BS02 V38 B 1 Y91 W145 Y186 C188 C189 Y193 Y91 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 21322593 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2y59 A 2.5 BS01 ZA3 A 1 A48 S49 Y147 S298 G412 T413 A48 S49 Y147 S298 G412 T413 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue P39045 21574608 501 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 2y5f A 1.29 BS01 XWG A 1 T98 Y99 F174 D189 A190 C191 Q192 V213 W215 G216 G226 I227 Y228 T84 Y85 F162 D179 A180 C181 Q182 V203 W205 G206 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=2nM remove_due_to_license_issue P00742 22162109 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2y5g A 1.29 BS01 FJD A 1 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G218 G226 I227 Y228 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=146nM remove_due_to_license_issue P00742 22162109 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2y5h A 1.33 BS01 Y5H A 1 T98 Y99 F174 A190 Q192 V213 W215 G216 C220 G226 I227 T84 Y85 F162 A180 Q182 V203 W205 G206 C209 G216 I217 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=1620nM remove_due_to_license_issue P00742 22162109 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGEQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2y5k A 2.1 BS01 YCU A 1 M18 G21 R22 G26 G28 L30 T31 M177 D178 M10 G13 R14 G18 G20 L22 T23 M161 D162 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM remove_due_to_license_issue IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k A 2.1 BS02 YCU C 1 T27 G28 T19 G20 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM remove_due_to_license_issue IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k C 2.1 BS01 YCU A 1 T27 T31 T19 T23 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM remove_due_to_license_issue IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k C 2.1 BS02 YCU C 1 M18 G21 R22 G26 G28 L30 T31 M177 D178 M10 G13 R14 G18 G20 L22 T23 M160 D161 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM remove_due_to_license_issue IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5l A 2.2 BS01 RO8 A 1 V17 M18 G21 R22 G26 G28 L30 T31 V9 M10 G13 R14 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.33uM remove_due_to_license_issue P09467 21550236 1000 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5l C 2.2 BS01 RO8 C 1 V17 M18 G21 R22 G26 G28 L30 T31 V9 M10 G13 R14 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.33uM remove_due_to_license_issue P09467 21550236 1000 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y67 A 1.85 BS01 N21 A 1 D35 T36 R37 S71 F161 H183 K348 A414 S415 N421 F422 D35 T36 R37 S71 F161 H183 K344 A410 S411 N417 F418 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=292uM remove_due_to_license_issue P14900 21963114 500 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIERCVSFGVNMGDYHLNHQQGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2y68 A 1.49 BS01 T04 A 1 G12 D35 T36 R37 S71 G73 F161 H183 K348 A414 S415 N421 F422 G12 D35 T36 R37 S71 G73 F161 H183 K344 A410 S411 N417 F418 K115 S116 N138 L147 H183 K115 S116 N138 L147 H183 6.3.2.9 0005515,0005524,0005737,0008360,0008764,0009058,0009252,0016874,0016881,0042802,0051301,0071555 ic50=253uM remove_due_to_license_issue P14900 21591605 500 ADYQGKNVVIIGLGLTGLSCVDFFLARGVTPRVMDTRMTPPGLDKLPEAVERHTGSLNDEWLMAADLIVASPGIALAHPSLSAAADAGIEIVGDIELFCREAQAPIVAITGSNGKSTVTTLVGEMAKAAGVNVGVGGNIGLPALMLLDDECELYVLELSSFQLETTSSLQAVAATILNVTEDHMDRYPFGLQQYRAAKLRIYENAKVCVVNADDALTMPIRRCVSFGVNMGDYHLNHQQGETWLRVKGEKVLNVKEMKLSGQHNYTNALAALALADAAGLPRASSLKALTTFTGLPHRFEVVLEHNGVRWINDSKATNVGSTEAALNGLHVDGTLHLLLGGDGKSADFSPLARYLNGDNVRLYCFGRDGAQLAALRPEVAEQTETMEQAMRLLAPRVQPGDMVLLSPACASLDQFKNFEQRGNEFARLAKELGSH 2y6c A 1.7 BS05 TQI A 1 L181 A182 H183 A184 A216 H219 E220 H223 H229 P239 L83 A84 H85 A86 A118 H121 E122 H125 H131 P141 H219 E220 H223 H229 H121 E122 H125 H131 3.4.24.23 0004222,0006508,0008237,0008270,0031012 ic50=0.0001M remove_due_to_license_issue Ki=10000nM P09237 21520417 1269 GYSLFPNSPKWTSKVVTYRIVSYTRDLPHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAFAPGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYPQNFKLSQDDIKGIQKLY 2y6d A 1.6 BS05 TQJ A 1 Y172 L181 A182 H183 Y215 H219 E220 H223 H229 V236 P239 T240 Y241 Y74 L83 A84 H85 Y117 H121 E122 H125 H131 V138 P141 T142 Y143 H219 E220 H223 H229 H121 E122 H125 H131 3.4.24.23 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=79nM P09237 21520417 1271 GYSLFPNSPKWTSKVVTYRIVSYTRDLPHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAFAPGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYFKLSQDDIKGIQKLYG 2y6o A 1.543 BS01 1N1 A 1 I627 A651 K653 M674 I697 T699 Y701 M702 E703 G705 L753 S763 I19 A43 K45 M66 I89 T91 Y93 M94 E95 G97 L145 S155 D746 A748 R750 N751 D764 I786 D138 A140 R142 N143 D156 I158 2.7.10.1 0004672,0004713,0005524,0006468 ic50=25nM remove_due_to_license_issue Q03137 22036717 1892 VREFAKEIDASCIKIEKVIGVGEFGEVCSGRLKVPGKREICVAIKTLKAGYTDKQRRDFLSEASIMGQFDHPNIIHLEGVVTKCKPVMIITEYMENGSLDAFLRKNDGRFTVIQLVGMLRGIGSGMKYLSDMSYVHRDLAARNILVNSNLVCKVSDFIPIRWTAPEAIAYRKFTSASDVWSYGIVMWEVMSYGERPYWDMSNQDVIKAIEEGYRLPPPMDCPIALHQLMLDCWQKERSDRPKFGQIVNMLDKLIRNPNSLKRT 2y71 A 1.5 BS01 CB6 A 1 N12 R15 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N10 R13 Y19 N70 G72 G73 H76 H96 I97 S98 R107 P11 N12 Y24 N75 G78 E99 H101 R108 P9 N10 Y19 N70 G73 E94 H96 R103 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=42.5nM remove_due_to_license_issue P9WPX7 21780742 1144 LIVNVINGPNLGRLGPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 2y76 A 2.5 BS01 CB7 A 1 N12 L13 N75 G77 G78 H81 H101 I102 S103 R112 N11 L12 N68 G70 G71 H74 H94 I95 S96 R105 P11 N12 N75 G78 E99 H101 R108 P10 N11 N68 G71 E92 H94 R101 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=440nM remove_due_to_license_issue P9WPX7 21780742 1144 ELIVNVINGPNLGRLGRGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 2y77 A 1.5 BS01 CB8 A 1 N12 N75 G77 G78 H81 H101 I102 S103 R112 N10 N66 G68 G69 H72 H92 I93 S94 R103 P11 N12 N75 G78 E99 H101 R108 P9 N10 N66 G69 E90 H92 R99 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=250nM remove_due_to_license_issue P9WPX7 21780742 1144 LIVNVINGPNLGRLGRGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 2y7i A 1.9 BS01 ARG A 1 Y33 E37 F71 A88 G89 D91 R96 E135 T138 T139 D177 Y16 E20 F54 A71 G72 D74 R79 E118 T121 T122 D160 ? 0015276,0016020,0030288,0030313,0034220,0046872 remove_due_to_license_issue Q8ZKA9 21560168 1245 ASVSARTLHFGTSATYAPYEFVDADNKIVGFDIDVANAVCKEMQAECSFTNQSFDSLIPSLRFKKFDAVIAGMDMTPKREQQVSFSQPYYEGLSAVVVTRKGAYHTFADLKGKKVGLENGTTHQRYLQDKQQAITPVAYDSYLNAFTDLKNNRLEGVFGDVAAIGKWLKNNPDYAIMDERASDPDYYGKGLGIAVRKDNDALLQEINAALDKVKASPEYAQMQEKWFT 2y7x A 1.9 BS01 MZA A 1 E97 T98 Y99 F174 D189 A190 Q192 S195 V213 W215 G216 G219 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 Q182 S185 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=1.3nM remove_due_to_license_issue Ki=1.3nM P00742 21349711 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2y7z A 1.84 BS01 C0Z A 1 E97 T98 Y99 F174 A190 Q192 S195 V213 W215 G216 G219 C220 G226 I227 Y228 E83 T84 Y85 F162 A180 Q182 S185 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=2nM remove_due_to_license_issue Ki=2nM P00742 21349710 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2y80 A 1.9 BS01 439 A 1 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=9nM remove_due_to_license_issue Ki=3nM P00742 21349710 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2y81 A 1.7 BS01 931 A 1 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=2nM remove_due_to_license_issue Ki=2nM P00742 21349710 1244 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 2y82 A 2.2 BS01 930 A 1 E97 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 E83 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=4nM remove_due_to_license_issue Ki=2nM P00742 21349710 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 2y8c A 2.1 BS01 DUQ A 1 F46 N103 Y112 I117 F46 N81 Y90 I95 S27 R91 S93 L99 D109 S27 R69 S71 L77 D87 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.4uM remove_due_to_license_issue Q8II92 21411327 400 MHLKIVCLSDEVREMYKNHKTHHEGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFGS 2y8c A 2.1 BS02 DUQ C 1 S92 S93 S70 S71 S27 R91 S93 L99 D109 S27 R69 S71 L77 D87 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.4uM remove_due_to_license_issue Q8II92 21411327 400 MHLKIVCLSDEVREMYKNHKTHHEGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFGS 2y8c B 2.1 BS01 DUQ B 1 F46 N103 G106 Y112 I117 F40 N72 G75 Y81 I86 S27 R91 S93 L99 D109 S21 R60 S62 L68 D78 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.4uM remove_due_to_license_issue Q8II92 21411327 400 MHLKIVCLSDEVREMYKNHDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEE 2y8i X 3.132 BS01 ADP X 1 N127 P128 G182 G184 K185 T186 E187 N233 N126 P127 G181 G183 K184 T185 E186 N232 S181 T186 S236 S237 S180 T185 S235 S236 3.6.4.1 0003774,0005524,0016459,0051015 remove_due_to_license_issue P08799 21841195 1001 NPIHDRTSDYHKYLKVKQGDSDLFKLTVSDKRYIWYNPDPKERDSYECGEIVSETSDSFTFKTVDGQDRQVKKDDANQRNPIKFDGVEDMSELSYLNEPAVFHNLRVRYNQDLIYTYSGLFLVAVNPFKRIPIYTQEMVDIFKGRRRNEVAPHIFAISDVAYRSMLDDRQNQSLLITGESGAGKTENTKKVIQYLASVAGRNQANGSGVLEQQILQANPILEAFGNAKTTRNNNSSRFGKFIEIQFNSAGFISGASIQSYLLEKSRVVFQSETERNYHIFYQLLAGATAEEKKALHLAGPESFNYLNQSGCVDIKGVSDSEEFKITRQAMDIVGFSQEEQMSIFKIIAGILHLGNIKFEKGAGEGAVLKDKTALNAASTVFGVNPSVLEKALMEPRILAGRDLVAQHLNVEKSSSSRDALVKALYGRLFLWLVKKINNVLCQERKAYFIGVLDISGFEIFKVNSFEQLCINYTNEKLQQFFNHHMFKLEQEEYLKEKINWTFIDFGLDSQATIDLIDGRQPPGILALLDEQSVFPNATDNTLITKLHSHFSKKNAKYEEPRFSKTEFGVTHYAGQVMYEIQDWLEKNKDPLQQDLELCFKDSSDNVVTKLFNDPNIASRAKKGANFITVAAQYKEQLASLMATLETTNPHFVRCIIPNNKQLPAKLEDKVVLDQLRCNAVLEGIRITRKGFPNRIIYADFVKRYYLLAPNVPRDAEDSQKATDAVLKHLNIDPEQYRFGITKIFFRAGQLARIEEARE 2y8l E 2.5 BS01 ADP E 1 M84 T86 T88 D89 L128 V129 I149 H150 R151 A320 G326 M62 T64 T66 D67 L106 V107 I127 H128 R129 A298 G304 ? 0004672,0004679,0005515,0005524,0005634,0005737,0005829,0006110,0006633,0010628,0016208,0019887,0019901,0031588,0031669,0032991,0042149,0043531,0043609,0044877,0045722,0051170 remove_due_to_license_issue P80385 21399626 1327 SNSSVYTTFMKSHRCYDLIPTSSKLVVFDTSLQVKKAFFALVTNGVRAAPLWDSKKQSFVGMLTITDFINILHRYYKSALVQIYELEEHKIETWREVYLQDSFKPLVCISPNASLFDAVSSLIRNKIHRLPVIDPESGNTLYILTHKRILKFLKLFITEFPKPEFMSKSLEELQIGTYANIAMVRTTTPVYVALGIFVQHRVSALPVVDEKGRVVDIYSKFDVINLAAEKTYNNLDVSVTKALQHRSHYFEGVLKCYLHETLEAIINRLVEAEVHRLVVVDEHDVVKGIVSLSDILQALVLTGG 2y8l E 2.5 BS02 ADP E 2 R69 K169 I239 S241 F243 D244 V275 L276 V296 H297 R298 R47 K147 I217 S219 F221 D222 V253 L254 V274 H275 R276 ? 0004672,0004679,0005515,0005524,0005634,0005737,0005829,0006110,0006633,0010628,0016208,0019887,0019901,0031588,0031669,0032991,0042149,0043531,0043609,0044877,0045722,0051170 remove_due_to_license_issue P80385 21399626 1328 SNSSVYTTFMKSHRCYDLIPTSSKLVVFDTSLQVKKAFFALVTNGVRAAPLWDSKKQSFVGMLTITDFINILHRYYKSALVQIYELEEHKIETWREVYLQDSFKPLVCISPNASLFDAVSSLIRNKIHRLPVIDPESGNTLYILTHKRILKFLKLFITEFPKPEFMSKSLEELQIGTYANIAMVRTTTPVYVALGIFVQHRVSALPVVDEKGRVVDIYSKFDVINLAAEKTYNNLDVSVTKALQHRSHYFEGVLKCYLHETLEAIINRLVEAEVHRLVVVDEHDVVKGIVSLSDILQALVLTGG 2y8q E 2.8 BS01 ADP E 1 M84 T86 T88 D89 L128 V129 I149 H150 R151 M62 T64 T66 D67 L106 V107 I127 H128 R129 ? 0004672,0004679,0005515,0005524,0005634,0005737,0005829,0006110,0006633,0010628,0016208,0019887,0019901,0031588,0031669,0032991,0042149,0043531,0043609,0044877,0045722,0051170 remove_due_to_license_issue P80385 21399626 1327 SNSSVYTTFMKSHRCYDLIPTSSKLVVFDTSLQVKKAFFALVTNGVRAAPLWDSKKQSFVGMLTITDFINILHRYYKSALVQIYELEEHKIETWREVYLQDSFKPLVCISPNASLFDAVSSLIRNKIHRLPVIDPESGNTLYILTHKRILKFLKLFITEFPKPEFMSKSLEELQIGTYANIAMVRTTTPVYVALGIFVQHRVSALPVVDEKGRVVDIYSKFDVINLAAEKTYNNLDVSVTKALQHRSHYFEGVLKCYLHETLEAIINRLVEAEVHRLVVVDEHDVVKGIVSLSDILQALVLTGG 2y8w A 1.8 BS01 rna B 0 R17 Y23 E24 H26 R27 T28 S30 K31 S34 E38 R43 K105 R106 A108 K112 R113 E121 R128 R129 R158 K160 D161 K167 L168 L169 Q170 V171 K200 R21 Y27 E28 H30 R31 T32 S34 K35 S38 E42 R47 K109 R110 A112 K116 R117 E125 R132 R133 R162 K164 D165 K171 L172 L173 Q174 V175 K204 3.1.-.- 0003723,0004519,0051607 remove_due_to_license_issue Q53WG9 21572442 5 ~ 24 GTGAMWLTKLVLNPASRAARRDLANPYEMHRTLSKAVSRALEEGRERLLWRLEPARGLEPPVVLVQTLTEPDWSVLDEGYAQVFPPKPFHPALKPGQRLRFRLRANPAKRLAATGKRVALKTPAEKVAWLERRLEEGGFRLLEGERGPWVQILQDTFLEVRRKKDGEEAGKLLQVQAVLFEGRLEVVDPERALATLRRGVGPGKALGLGLLSVAP 2ya6 A 2.0 BS01 DAN A 1 R332 I401 D402 F428 Y575 L583 Q587 R648 R706 Y737 R26 I95 D96 F122 Y269 L277 Q281 R342 R400 Y431 S356 D357 E632 Y737 S50 D51 E326 Y431 3.2.1.18 0004308 Ki=2uM remove_due_to_license_issue IC50=4800nM, Ki=1.6e+3nM P62575 21514303 1777 ALTEKTDIFESGRNGNPNKDGIKSYRIPALLKTDKGTLIAGADERRLHSSDWGDIGMVIRRSEDNGKTWGDRVTITNLRDNPKASDPSIGSPVNIDMVLVQDPETKRIFSIYDMFPEGKGIFGMSSQKEEAYKKIDGKTYQILYREGEKGAYTIRENGTVYTPDGKATDYRVVVDPVKPAYSDKGDLYKGDQLLGNIYFTTNKTSPFRIAKDSYLWMSYSDDDGKTWSAPQDITPMVKADWMKFLGVGPGTGIVLRNGPHKGRILIPVYTTNNVSHLDGSQSSRVIYSDDHGKTWHAGEAVNDNRQVDGQKIHSSTMNNRRAQNTESTVVQLNNGDVKLFMRGLTGDLQVATSKDGGVTWEKDIKRYPQVKDVYVQMSAIHTMHEGKEYIILSNAGGPKRENGMVHLARVEENGELTWLKHNPIQKGEFAYNSLQELGNGEYGILYEHTEKGQNAYTLSFRKFNWEFLSK 2ya7 A 1.89 BS01 ZMR A 1 R332 I333 D357 I401 D402 F428 Y575 Q587 R648 R706 Y737 R26 I27 D51 I95 D96 F122 Y269 Q281 R342 R400 Y431 S356 D357 E632 Y737 S50 D51 E326 Y431 3.2.1.18 0004308 Ki=0.72mM remove_due_to_license_issue Ki=7.20e+5nM P62575 21514303 1776 ALTEKTDIFESGRNGNPNKDGIKSYRIPALLKTDKGTLIAGADERRLHSSDWGDIGMVIRRSEDNGKTWGDRVTITNLRDNPKASDPSIGSPVNIDMVLVQDPETKRIFSIYDMFPEGKGIFGMSSQKEEAYKKIDGKTYQILYREGEKGAYTIRENGTVYTPDGKATDYRVVVDPVKPAYSDKGDLYKGDQLLGNIYFTTNKTSPFRIAKDSYLWMSYSDDDGKTWSAPQDITPMVKADWMKFLGVGPGTGIVLRNGPHKGRILIPVYTTNNVSHLDGSQSSRVIYSDDHGKTWHAGEAVNDNRQVDGQKIHSSTMNNRRAQNTESTVVQLNNGDVKLFMRGLTGDLQVATSKDGGVTWEKDIKRYPQVKDVYVQMSAIHTMHEGKEYIILSNAGGPKRENGMVHLARVEENGELTWLKHNPIQKGEFAYNSLQELGNGEYGILYEHTEKGQNAYTLSFRKFNWEFLS 2ya8 A 1.75 BS01 G39 A 1 R332 D357 I401 D402 F550 R648 R706 Y737 R26 D51 I95 D96 F244 R342 R400 Y431 S356 D357 E632 Y737 S50 D51 E326 Y431 3.2.1.18 0004308 Ki=1.77uM remove_due_to_license_issue Ki=1.77e+3nM P62575 21514303 1777 ALTEKTDIFESGRNGNPNKDGIKSYRIPALLKTDKGTLIAGADERRLHSSDWGDIGMVIRRSEDNGKTWGDRVTITNLRDNPKASDPSIGSPVNIDMVLVQDPETKRIFSIYDMFPEGKGIFGMSSQKEEAYKKIDGKTYQILYREGEKGAYTIRENGTVYTPDGKATDYRVVVDPVKPAYSDKGDLYKGDQLLGNIYFTTNKTSPFRIAKDSYLWMSYSDDDGKTWSAPQDITPMVKADWMKFLGVGPGTGIVLRNGPHKGRILIPVYTTNNVSHLDGSQSSRVIYSDDHGKTWHAGEAVNDNRQVDGQKIHSSTMNNRRAQNTESTVVQLNNGDVKLFMRGLTGDLQVATSKDGGVTWEKDIKRYPQVKDVYVQMSAIHTMHEGKEYIILSNAGGPKRENGMVHLARVEENGELTWLKHNPIQKGEFAYNSLQELGNGEYGILYEHTEKGQNAYTLSFRKFNWEFLSK 2yac A 2.2 BS01 937 A 1 R57 L59 G60 C67 A80 K82 L130 C133 R134 R136 S137 E140 F183 D194 A328 R19 L21 G22 C29 A42 K44 L92 C95 R96 R98 S99 E102 F145 D156 A290 D176 K178 G180 N181 D194 T214 D138 K140 G142 N143 D156 T176 2.7.11.21 0004672,0005524,0006468 ic50=0.002uM remove_due_to_license_issue IC50=3nM P53350 21470862 501 EIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKTLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 2yak A 2.2 BS01 OSV A 1 L19 S21 A25 V27 A40 K42 E64 I77 L93 V96 I160 D161 L18 S20 A24 V26 A39 K41 E63 I76 L92 V95 I159 D160 D139 K141 E143 N144 D161 T180 D138 K140 E142 N143 D160 T179 2.7.11.1 0004672,0005524,0006468 ic50=2nM remove_due_to_license_issue P53355 21446733 1279 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKPK 2yay A 1.86 BS01 DUP A 1 Q21 N25 I28 E48 E51 D79 H82 F83 K179 N183 R186 Y191 K198 Q14 N18 I21 E41 E44 D72 H75 F76 K172 N176 R179 Y184 K191 3.6.1.23 0004170,0005654,0016787,0046872 Kd=0.8uM remove_due_to_license_issue O15826 21454646 1265 NIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yaz A 2.4 BS01 UMP A 1 I28 W41 D79 H82 F83 N183 R186 Y191 I21 W34 D72 H75 F76 N176 R179 Y184 3.6.1.23 0004170,0005654,0016787,0046872 Kd=7.3uM remove_due_to_license_issue O15826 21454646 1265 NIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yaz A 2.4 BS03 UMP B 1 W60 W61 W53 W54 3.6.1.23 0004170,0005654,0016787,0046872 Kd=7.3uM remove_due_to_license_issue O15826 21454646 1265 NIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yaz B 2.4 BS01 UMP A 1 W60 W61 W59 W60 3.6.1.23 0004170,0005654,0016787,0046872 Kd=7.3uM remove_due_to_license_issue O15826 21454646 1265 KRARSANIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yaz B 2.4 BS02 UMP B 1 Q21 N25 I28 W41 D79 H82 F83 N183 R186 Y191 Q20 N24 I27 W40 D78 H81 F82 N182 R185 Y190 3.6.1.23 0004170,0005654,0016787,0046872 Kd=7.3uM remove_due_to_license_issue O15826 21454646 1265 KRARSANIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yb0 A 2.28 BS01 DUR A 1 N25 I28 W41 D79 H82 F83 N183 N19 I22 W35 D73 H76 F77 N177 3.6.1.23 0004170,0005654,0016787,0046872 Kd=140uM remove_due_to_license_issue O15826 21454646 1266 ANIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yb0 A 2.28 BS02 DUR B 1 W60 W61 W54 W55 3.6.1.23 0004170,0005654,0016787,0046872 Kd=140uM remove_due_to_license_issue O15826 21454646 1266 ANIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yb0 B 2.28 BS01 DUR A 1 W60 W61 W59 W60 3.6.1.23 0004170,0005654,0016787,0046872 Kd=140uM remove_due_to_license_issue O15826 21454646 1266 KRARSANIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yb0 B 2.28 BS02 DUR B 1 N25 I28 D79 H82 F83 N183 N24 I27 D78 H81 F82 N182 3.6.1.23 0004170,0005654,0016787,0046872 Kd=140uM remove_due_to_license_issue O15826 21454646 1266 KRARSANIPGAILHSLAELQDGLNAMIDPSWRAVRSLDNWALAITMESTELLDSYPWKWWKNLNATPDLANVRIELVDIFHFSLSGAMQMRSTPDDEIPAASLKPLKEVMTTFLPAKECTSDPYGFVFFPLTDTQNAIASFRNIIQLANAYRFDVIIECIIYAAEDLGFNLVAYYIAKHTLNCIRQLSGYKDGSYVKVNNGVEDNSLLHNCIKDVSLDEVLDADKYVQAWNSIMANVYEAFQIKESDRKDAERWFALAKENRL 2yb9 A 2.4 BS02 HA0 A 1 R102 F106 N542 A543 F544 H583 E584 E646 W693 G695 Y697 H711 R717 R49 F53 N489 A490 F491 H530 E531 E593 W640 G642 Y644 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 ic50=0.6nM remove_due_to_license_issue P08473 21515054 1751 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 2ybk A 2.4 BS02 2HG A 1 Y132 F185 H188 H276 Y126 F179 H182 H270 G170 Y177 H188 E190 H276 S288 G164 Y171 H182 E184 H270 S282 1.14.11.66,1.14.11.69 ic50=24uM remove_due_to_license_issue IC50=24000nM O75164 21460794 601 TLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 2ybp A 2.02 BS03 2HG A 1 Y132 F185 H188 S196 N198 K206 W208 H276 S288 Y126 F179 H182 S190 N192 K200 W202 H270 S282 G170 Y177 H188 E190 H276 S288 G164 Y171 H182 E184 H270 S282 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=24000nM O75164 21460794 1359 TLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 2ybs A 2.32 BS03 S2G A 1 Y132 F185 H188 N198 K206 H276 Y125 F178 H181 N191 K199 H269 G170 Y177 H188 E190 H276 S288 G163 Y170 H181 E183 H269 S281 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=26000nM O75164 21460794 1359 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 2ybt A 2.22 BS01 DW0 A 1 W31 F58 W99 N100 D138 E140 M210 Y212 W360 W11 F38 W79 N80 D118 E120 M190 Y192 W340 D136 D138 E140 Y212 D116 D118 E120 Y192 3.2.1.14 0004553,0005975,0008061 ic50=20uM remove_due_to_license_issue IC50=2.0e+4nM Q9BZP6 21609838 1399 AYQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNIKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTAP 2ybt A 2.22 BS02 DW0 A 2 W99 W218 W79 W198 D136 D138 E140 Y212 D116 D118 E120 Y192 3.2.1.14 0004553,0005975,0008061 ic50=20uM remove_due_to_license_issue IC50=2.0e+4nM Q9BZP6 21609838 1400 AYQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNIKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTAP 2ybu A 2.25 BS01 CX9 A 1 W31 F58 W99 N100 D138 E140 M210 Y212 W360 W11 F38 W79 N80 D118 E120 M190 Y192 W340 D136 D138 E140 Y212 D116 D118 E120 Y192 3.2.1.14 0004553,0005975,0008061 Ki=0.42uM remove_due_to_license_issue IC50=920nM Q9BZP6 21609838 1398 AYQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNIKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTA 2ybu A 2.25 BS02 CX9 A 2 W99 W218 W79 W198 D136 D138 E140 Y212 D116 D118 E120 Y192 3.2.1.14 0004553,0005975,0008061 Ki=0.42uM remove_due_to_license_issue IC50=920nM Q9BZP6 21609838 1399 AYQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNIKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTA 2yc0 A 2.15 BS02 2HG A 1 Y145 T196 H199 N205 F207 H279 I281 W296 Y145 T196 H199 N205 F207 H279 I281 W296 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=1500uM remove_due_to_license_issue Q9NWT6 21460794 601 MAATAAEAVASGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2yc3 A 1.4 BS01 MW5 A 1 I177 A203 Q238 V239 I240 D262 V263 I265 V266 I96 A122 Q157 V158 I159 D181 V182 I184 V185 2.7.7.60 0003824,0008299,0050518,0070567 ic50=0.14uM remove_due_to_license_issue P69834 21766403 1301 MEKSVSVILLAGGQGPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLDRKTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILSE 2yc5 A 1.6 BS01 6BC A 1 R157 Q158 I177 A203 Q238 V239 I240 D262 V263 I265 V266 V273 R75 Q76 I95 A121 Q156 V157 I158 D180 V181 I183 V184 V191 2.7.7.60 0003824,0008299,0050518,0070567 ic50=0.035uM remove_due_to_license_issue IC50=35nM P69834 21766403 1300 MEKSVSVILLAGSMPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLDRKTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILS 2ycf A 1.77 BS01 YCF A 1 L226 C231 V234 I251 E273 M304 E305 G307 L354 T367 D368 L17 C22 V25 I42 E49 M80 E81 G83 L130 T143 D144 D347 K349 N352 D368 T387 D123 K125 N128 D144 T163 2.7.11.1 0004672,0005524,0006468 ic50=0.03nM remove_due_to_license_issue O96017 21963792 600 SVYPKALRDEYIMSKTLGSGACGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2ych A 2.2 BS02 ATP A 1 E19 G21 A22 S23 K26 K173 G199 A200 E201 E242 K245 R246 G314 G315 G316 L319 E9 G11 A12 S13 K16 K162 G188 A189 E190 E231 K234 R235 G275 G276 G277 L280 ? 0005524,0046872 remove_due_to_license_issue Q72IW8 21596754 502 PRVEALGLEIGASALKLVEVSGNPPALKALASRPTPPGLLMEGMVAEPAALAQEIKELLLEARTRKRYVVTALSNLAVILRPIQVPKMPLKEMEEAVRWEAERYIPFPIEVVLDFAPLTPLSEVQEGEQVQVMVAAARQEAVAGVLEALRGAGLVPVVLDVKPFAGLYPLEARLAEEPDRVFLVLDIGAESTSLVLLRGDKPLAVRVLTLSGKDFTEAIARSFNLDLLAAEEVKRTYGRIYDAIRPVLVELTQELRRSLEFFRIQLSPEVGYLLGGGSKLRGLASLLTDTLGVNLEPVNPWEAVAVDPKRFESEQLQEIGPEFAVALGLALRGVEP 2ycm A 1.8 BS01 30A A 1 R157 Q158 A203 Q238 V259 D261 D262 V263 S264 I265 V266 V273 R73 Q74 A119 Q151 V172 D174 D175 V176 S177 I178 V179 V186 2.7.7.60 0003824,0008299,0050518,0070567 ic50=274uM remove_due_to_license_issue P69834 21766403 1306 EKSVSVILLAGMPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILSE 2ycq A 2.05 BS01 UPX A 1 V234 K249 E273 L303 M304 G307 L354 T367 D368 V24 K39 E48 L78 M79 G82 L129 T142 D143 D347 K349 N352 D368 T387 D122 K124 N127 D143 T162 2.7.11.1 0004672,0005524,0006468 ic50=0.14nM remove_due_to_license_issue O96017 21963792 600 VYPKALRDEYIMSKTLGSGACGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2ycr A 2.2 BS01 HCW A 1 L226 V234 K249 E273 L301 M304 E305 G307 L354 T367 D368 L16 V21 K36 E45 L73 M76 E77 G79 L126 T139 D140 D347 K349 N352 D368 T387 D119 K121 N124 D140 T159 2.7.11.1 0004672,0005524,0006468 ic50=69.6nM remove_due_to_license_issue O96017 21963792 600 VYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTAKPQ 2ycs A 2.35 BS01 NXP A 1 V234 K249 E273 L301 M304 G307 E308 L354 T367 D368 V22 K37 E46 L74 M77 G80 E81 L127 T140 D141 D347 K349 N352 D368 T387 D120 K122 N125 D141 T158 2.7.11.1 0004672,0005524,0006468 ic50=1.36nM remove_due_to_license_issue O96017 21963792 600 SVYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2yde A 2.28 BS02 S2G A 1 Y145 L188 T196 H199 N205 F207 K214 H279 I281 N294 W296 Y145 L188 T196 H199 N205 F207 K214 H279 I281 N294 W296 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=189uM remove_due_to_license_issue Q9NWT6 21460794 601 MAATAAEAVASGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2ydf A 2.75 BS01 IO3 A 1 Y150 K199 L219 R222 L238 H242 R257 A291 Y137 K186 L206 R209 L225 H229 R244 A278 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 21501503 2001 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVAADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAA 2ydf A 2.75 BS02 IO3 A 2 L387 I388 N391 L407 R410 Y411 V433 L453 R485 S489 L374 I375 N378 L394 R397 Y398 V420 L440 R472 S476 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 21501503 2002 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVAADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAA 2ydf A 2.75 BS03 IO3 A 3 L115 I142 H146 L185 R186 K190 L102 I129 H133 L172 R173 K177 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 21501503 2003 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVAADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAA 2ydf A 2.75 BS04 IO3 A 4 V409 R410 K541 V396 R397 K528 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 21501503 2004 SEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVAADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAA 2ydi A 1.6 BS01 YDI A 1 L15 A36 E85 Y86 C87 S88 G90 L137 L14 A35 E84 Y85 C86 S87 G89 L136 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=150nM O14757 22551018 1282 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 2ydj A 1.85 BS01 YDJ A 1 L15 Y20 A36 E85 Y86 C87 E134 N135 L137 D148 L8 Y13 A29 E70 Y71 C72 E119 N120 L122 D133 D130 K132 E134 N135 D148 T170 D115 K117 E119 N120 D133 T155 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.005uM remove_due_to_license_issue IC50=6.0nM, EC50=10nM O14757 22551018 1270 DWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2ydk A 1.9 BS01 YDK A 1 L15 A36 E85 Y86 C87 G90 E134 N135 L137 D148 L13 A34 E78 Y79 C80 G83 E127 N128 L130 D141 D130 K132 E134 N135 D148 T170 D123 K125 E127 N128 D141 T163 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.007uM remove_due_to_license_issue IC50=7nM, EC50=20nM O14757 22551018 1277 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2ydm A 2.44 BS02 SLC A 1 Q281 H353 H383 E384 K511 H513 Y520 Y523 Q242 H314 H344 E345 K468 H470 Y477 Y480 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H470 Y480 3.4.15.1 0006508,0008237,0008241,0016020 ic50=36.4nM remove_due_to_license_issue P12821 21810173 1626 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWQ 2ydo A 3.0 BS01 ADN A 1 F168 E169 N253 S277 H278 F163 E164 N238 S262 H263 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue EC50=700nM, Ki=700nM P29274 21593763 400 SSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSAAAADILVGVLAIPFAIAISTGFCAACHGCLFIACFVLVLTASSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMESTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLRQQEPFKAAAAENLYF 2ydt A 1.6 BS01 EDG A 1 W169 E170 Q195 M226 W148 E149 Q174 M205 3.2.1.55 0016798,0046556,0046872 remove_due_to_license_issue B8ZY56 21773614 500 GKTFSNVEIFDPPTNYRDPQVLYARPLELSDGTLLGTWENYSPEPPNVWFPIVKSKDGGKTWKEISKVKDTQNNWGLRYQPQLYELPRAFGKYPKGTVLCSGSSIPSDLSETLIEVYASRDKGYTWEFVSHVALGGEALPNPGLTPVWEPFLMTYKEKLILYYSDQRDNATHSQKLVHQTTTDLKKWSKVVDDTKYANYYARPGMPTVAKLPNNEYIYVYEYGGGPNPPAGSDYWFPVYYRLSKDPQKFLNKAHHQIVSNDGTTPAGSPYVVWTPYGGKNGTIVVSCGTRSEIFTNQALGDASAWKKWDVPQPTAYTRSLLTFQKDPDLLMIMGAGILPPAGGKNTVSASVVRLSEVMK 2ydt A 1.6 BS02 AHR A 1 E60 Q101 E39 Q80 3.2.1.55 0016798,0046556,0046872 remove_due_to_license_issue B8ZY56 21773614 501 GKTFSNVEIFDPPTNYRDPQVLYARPLELSDGTLLGTWENYSPEPPNVWFPIVKSKDGGKTWKEISKVKDTQNNWGLRYQPQLYELPRAFGKYPKGTVLCSGSSIPSDLSETLIEVYASRDKGYTWEFVSHVALGGEALPNPGLTPVWEPFLMTYKEKLILYYSDQRDNATHSQKLVHQTTTDLKKWSKVVDDTKYANYYARPGMPTVAKLPNNEYIYVYEYGGGPNPPAGSDYWFPVYYRLSKDPQKFLNKAHHQIVSNDGTTPAGSPYVVWTPYGGKNGTIVVSCGTRSEIFTNQALGDASAWKKWDVPQPTAYTRSLLTFQKDPDLLMIMGAGILPPAGGKNTVSASVVRLSEVMK 2ydv A 2.6 BS01 NEC A 1 L85 T88 F168 N181 W246 L249 H250 N253 H278 L83 T86 F166 N179 W236 L239 H240 N243 H268 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue Ki=16nM, IC50=3.7nM, EC50=251nM P29274 21593763 400 IMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSAAAADILVGVLAIPFAIAISTGFCAACHGCLFIACFVLVLTASSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMESQSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLRQQEPFKAAAAENLYFQ 2ydw B 1.9 BS01 WSH B 1 W97 P98 V103 L108 L110 Y155 N156 I162 W21 P22 V27 L32 L34 Y79 N80 I86 ? Kd=46nM remove_due_to_license_issue Kd=52nM, IC50=29.9nM P25440 21568322 1182 NQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMP 2ye9 A 2.2 BS01 2D4 A 1 N51 A55 K58 D93 I96 G97 M98 L107 T109 F138 T184 E223 N36 A40 K43 D78 I81 G82 M83 L92 T94 F123 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21561141 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2yek A 1.98 BS01 EAM A 1 W97 P98 V103 L108 L110 N156 I162 W24 P25 V30 L35 L37 N83 I89 ? ic50=32.5nM remove_due_to_license_issue IC50=32.5nM, Ki=74nM, Kd=100nM P25440 21568322 1188 RVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQEL 2yel A 1.65 BS01 WSH A 1 W81 P82 L92 L94 N140 I146 W40 P41 L51 L53 N99 I105 ? ic50=15.5nM remove_due_to_license_issue Kd=19nM, IC50=15.5nM O60885 21568322 1170 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 2yem A 2.3 BS01 WSH A 1 W374 P375 L387 N433 V439 W26 P27 L39 N85 V91 ? ic50=15.5nM remove_due_to_license_issue Kd=19nM, IC50=15.5nM O60885 21568322 1459 KVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMP 2yer A 1.83 BS01 TQ1 A 1 L15 A36 E85 Y86 C87 G90 E91 L137 L14 A35 E84 Y85 C86 G89 E90 L136 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.02uM remove_due_to_license_issue O14757 22342147 1270 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2yex A 1.3 BS01 YEX A 1 L15 V23 A36 E85 Y86 C87 G90 L137 L14 V22 A35 E84 Y85 C86 G89 L136 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.0001uM remove_due_to_license_issue IC50=0.100000nM O14757 22342147 1278 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2yfe A 2.0 BS01 YFE A 1 R280 I281 C285 R288 L330 I341 S342 M348 R68 I69 C73 R76 L118 I129 S130 M136 ? 0003677,0004879,0005634,0006355 Ki=0.236uM remove_due_to_license_issue EC50=458nM, Kd=236nM P37231 22509006 999 DQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKISKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2yfx A 1.7 BS01 VGH A 1 A1148 M1196 M1199 A1200 G1202 N1254 L1256 G1269 D1270 I1399 E1400 A46 M94 M97 A98 G100 N152 L154 G167 D168 I291 E292 D1249 A1251 R1253 N1254 D1270 L1291 D147 A149 R151 N152 D168 L183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 24432909 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILMELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 2yga A 2.37 BS01 GDM A 1 N37 D40 K44 M84 L92 K98 G121 V122 F124 N37 D40 K44 M84 L92 K98 G121 V122 F124 ? 0005524,0006457,0016887,0051082,0140662 Kd=24.5uM remove_due_to_license_issue P02829 21778327 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAGLINLLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2yge A 1.956 BS01 GDM A 1 N37 D40 A41 D79 M84 N92 N98 G121 V122 F124 N37 D40 A41 D79 M84 N92 N98 G121 V122 F124 ? 0005524,0006457,0016887,0051082,0140662 Kd=8.62uM remove_due_to_license_issue P02829 21778327 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDRIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIANSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2ygf A 2.0 BS01 GDM A 1 N37 D40 A41 K44 D79 N92 K98 G121 V122 F124 N36 D39 A40 K43 D78 N91 K97 G120 V121 F123 ? 0005524,0006457,0016887,0051082,0140662 Kd~10uM remove_due_to_license_issue P02829 21778327 1215 ASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAEVINNIGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQMISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 2yh1 A -1.00 BS01 rna B 0 R150 Y152 K195 N196 F197 F199 K225 R227 R228 P229 H230 D231 K260 F262 G264 G265 N289 V291 S294 T296 K300 Y302 F304 L331 R3 Y5 K48 N49 F50 F52 K78 R80 R81 P82 H83 D84 K113 F115 G117 G118 N142 V144 S147 T149 K153 Y155 F157 L184 ? 0003676,0003723,0005634,0006397 remove_due_to_license_issue P26368 21753750 601 ~ 609 ARRLYVGNIPFGITEEAMMDFFNAQMRLGGLTQAPGNPVLAVQINQDKNFAFLEFRSVDETTQAMAFDGIIFQGQSLKIRRPHDYQPLPGMSENPSVYVPGVVSTVVPDSAHKLFIGGLPNYLNDDQVKELLTSFGPLKAFNLVKDSATGLSKGYAFCEYVDINVTDQAIAGLNGMQLGDKKLLVQRASVGAKNA 2yhd A 2.2 BS02 AV6 A 1 K720 V730 Q733 M734 Q738 M894 I898 K50 V60 Q63 M64 Q68 M224 I228 ? Ki=23uM remove_due_to_license_issue IC50=18640nM P10275 21846139 1921 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2yi0 A 1.6 BS01 YI0 A 1 N51 S52 A55 K58 D93 G97 M98 L107 G108 F138 T184 N36 S37 A40 K43 D78 G82 M83 L92 G93 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=7.5nM remove_due_to_license_issue Kd=13nM P07900 22984537 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 2yi5 A 2.5 BS01 YI5 A 1 N51 S52 A55 D93 G97 M98 F138 T184 N36 S37 A40 D78 G82 M83 F120 T166 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=39nM remove_due_to_license_issue Kd=34nM P07900 22984537 1226 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 2yi7 A 1.4 BS01 BZ8 A 1 N51 A55 D93 I96 G97 M98 F138 T184 N36 A40 D78 I81 G82 M83 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=4.8nM remove_due_to_license_issue Kd=6.3nM P07900 22984537 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 2yig A 1.7 BS01 5EL A 1 L184 L185 L218 H222 E223 G237 L239 F241 P242 I243 Y244 T245 T247 L81 L82 L115 H119 E120 G134 L136 F138 P139 I140 Y141 T142 T144 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=79.4nM remove_due_to_license_issue IC50=125.89nM P45452 21669521 301 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKFMLPDDDVQGIQSLYGPGDED 2yiq A 1.89 BS01 YIQ A 1 L226 V234 I251 E273 M304 G307 L354 T367 D368 L16 V20 I37 E43 M74 G77 L124 T137 D138 D347 K349 N352 D368 T387 D117 K119 N122 D138 T157 2.7.11.1 0004672,0005524,0006468 ic50=12.67nM remove_due_to_license_issue O96017 21907711 600 VYPKALRDEYIMSKTLGGEVKLAFERKTCKKVAIKIISKVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2yir A 2.1 BS01 YIR A 1 L226 V234 K249 I251 E273 L301 L303 M304 G307 L354 T367 D368 L17 V25 K40 I42 E50 L78 L80 M81 G84 L131 T144 D145 D347 K349 N352 D368 T387 D124 K126 N129 D145 T164 2.7.11.1 0004672,0005524,0006468 ic50=0.17nM remove_due_to_license_issue O96017 21907711 600 SVYPKALRDEYIMSKTLGSGACGEVKLAFERKTCKKVAIKIISKLNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALP 2yis A 2.0 BS01 YIS A 1 A51 K53 E71 L75 I84 L104 T106 M109 G110 H148 L167 D168 F169 P351 P352 A44 K46 E64 L68 I77 L97 T99 M102 G103 H133 L152 D153 F154 P324 P325 D150 K152 N155 D168 T185 D135 K137 N140 D153 T158 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Kd=0.001000nM Q16539 21888439 1353 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2yit A 2.2 BS01 YIT A 1 L226 V234 K249 E273 E305 G307 L354 T367 D368 L16 V24 K39 E49 E81 G83 L130 T143 D144 D347 K349 N352 D368 T387 D123 K125 N128 D144 T163 2.7.11.1 0004672,0005524,0006468 ic50=0.29nM remove_due_to_license_issue O96017 21907711 600 VYPKALRDEYIMSKTLGSGACGEVKLAFERKTCKKVAIKIISKLNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ 2yiu A 2.7 BS03 SMA A 1 F144 M154 G158 V161 L180 I292 P294 E295 F298 Y302 M336 F142 M152 G156 V159 L178 I290 P292 E293 F296 Y300 M334 H217 N221 K251 D252 E295 H215 N219 K249 D250 E293 1.10.2.2 0005886,0008121,0009055,0016020,0016491,0022904,0045275,0046872,1902600 remove_due_to_license_issue P05418 21996020 502 GIPHDHYEPKTGFERWLHRRLPIVSLVYDTLMIPTPKNLNWWWIWGIVLAFCLVLQIATGIVLVMHYTPHVDLAFASVEHIMRDVNGGYMLRYLHANGASLFFLAVYIHIFRGLYYGSYKAPREVTWIVGMLIYLMMMGTAFMGYVLPWGQMSFWGATVITGLFGAIPGVGEAIQTWLLGGPAVDNPTLNRFFSLHYLLPFVIAALVVVHIWAFHTTGNNNPTGVEVRRGSKEEAKKDTLPFWPYFVIKDLFALAVVLVVFFAIVGFMPNYLGHPDNYIEANPLVTPAHIVPEWYFLPFYAILRAFTADVWVVMLVNWLSFGIIDAKFFGVIAMFGAILVMALVPWLDTSRVRSGQYRPLFKWWFWLLAVDFVVLMWVGAMPAEGIYPYIALAGSAYWFAYFLIILPLLGIIEKPDAMPQTIEEDFNA 2yiu D 2.7 BS03 SMA D 1 M140 F144 M145 V161 I292 P294 E295 F298 Y302 M138 F142 M143 V159 I290 P292 E293 F296 Y300 H217 N221 K251 D252 E295 H215 N219 K249 D250 E293 1.10.2.2 0005886,0008121,0009055,0016020,0016491,0022904,0045275,0046872,1902600 remove_due_to_license_issue P05418 21996020 502 GIPHDHYEPKTGFERWLHRRLPIVSLVYDTLMIPTPKNLNWWWIWGIVLAFCLVLQIATGIVLVMHYTPHVDLAFASVEHIMRDVNGGYMLRYLHANGASLFFLAVYIHIFRGLYYGSYKAPREVTWIVGMLIYLMMMGTAFMGYVLPWGQMSFWGATVITGLFGAIPGVGEAIQTWLLGGPAVDNPTLNRFFSLHYLLPFVIAALVVVHIWAFHTTGNNNPTGVEVRRGSKEEAKKDTLPFWPYFVIKDLFALAVVLVVFFAIVGFMPNYLGHPDNYIEANPLVTPAHIVPEWYFLPFYAILRAFTADVWVVMLVNWLSFGIIDAKFFGVIAMFGAILVMALVPWLDTSRVRSGQYRPLFKWWFWLLAVDFVVLMWVGAMPAEGIYPYIALAGSAYWFAYFLIILPLLGIIEKPDAMPQTIEEDFNA 2yiu F 2.7 BS01 SMA A 1 C154 H155 C138 H139 H155 H139 7.1.1.8 0005886,0008121,0016020,0046872,0051537,1902600 remove_due_to_license_issue P05417 21996020 502 DFLYYATAGAGTVAAGAAAWTLVNQMNPSADVQALASIQVDVSGVETGTQLTVKWLGKPVFIRRRTEDEIQAGREVDLGQLIDRSAQNSNKPDAPATDENRTMDEAGEWLVMIGVCTHLGCVPIGDGAGDFGGWFCPCHGSHYDTSGRIRRGPAPQNLHIPVAEFLDDTTIKLG 2yiv X 1.28 BS06 NBN X 1 L82 V565 I586 F608 L81 V564 I585 F607 1.2.7.4 0003824,0004601,0005737,0005886,0006091,0016151,0016491,0042542,0043885,0046872,0050418,0051539,0098869 remove_due_to_license_issue Q9F8A8 21904889 5005 ARQNLKSTDRAVQQMLDKAKREGIQTVWDRYEAMKPQCGFGETGLCCRHCLQGPCRINPFGDEPKVGICGATAEVIVARGLDRSIAAGAAGHSGHAKHLAHTLKKAVQGKAASYMIKDRTKLHSIAKRLGIPTEGQKDEDIALEVAKAALADFHEKDTPVLWVTTVLPPSRVKVLSAHGLIPAGIDHEIAEIMHRTSMGCDADAQNLLLGGLRCSLADLAGCYMGTDLADILFGTPAPVVTESNLGVLKADAVNVAVHGHNPVLSDIIVSVSKEMENEARAAGATGINVVGICCTGNEVLMRHGIPACTHSVSQEMAMITGALDAMILDYQCIQPSVATIAECTGTTVITTMEMSKITGATHVNFAEEAAVENAKQILRLAIDTFKRRKGKPVEIPNIKTKVVAGFSTEAIINALSKLNANDPLKPLIDNVVNGNIRGVCLFAGCNNVKVPQDQNFTTIARKLLKQNVLVVATGCGAGALMRHGFMDPANVDELCGDGLKAVLTAIGEANGLGGPLPPVLHMGSCVDNSRAVALVAALANRLGVDLDRLPVVASAAEAMHEKAVAIGTWAVTIGLPTHIGVLPPITGSLPVTQILTSSVKDITGGYFIVELDPETAADKLLAAINERRAGLGLPW 2yiw A 2.0 BS01 YIW A 1 V30 V38 A51 K53 E71 L75 I84 L104 T106 M109 G110 A111 L167 D168 F169 P352 V26 V31 A44 K46 E64 L68 I77 L97 T99 M102 G103 A104 L152 D153 F154 P325 D150 K152 N155 D168 T185 D135 K137 N140 D153 T158 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Kd=0.400000nM Q16539 21888439 1353 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2yix A 2.3 BS01 YIX A 1 Y35 E71 L74 L75 I84 T106 H107 L108 M109 A111 L167 D168 F169 L171 Y32 E68 L71 L72 I81 T103 H104 L105 M106 A108 L164 D165 F166 L168 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=3.3nM remove_due_to_license_issue Kd=3.3nM, IC50=58nM Q16539 21888439 1355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 2yj2 A 1.15 BS01 YJ2 A 1 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A214 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A213 Q19 C25 H163 N187 Q19 C25 H163 N186 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21898833 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTSDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2yj8 A 1.3 BS01 YJ8 A 1 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A214 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A213 Q19 C25 H163 N187 Q19 C25 H163 N186 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21898833 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTSDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2yj9 A 1.35 BS01 YJ9 A 1 G23 C25 G61 E63 G67 G68 L69 M70 A135 M161 D162 H163 A214 G23 C25 G61 E63 G67 G68 L69 M70 A135 M161 D162 H163 A210 Q19 C25 H163 N187 Q19 C25 H163 N183 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21898833 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFEDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2yjb A 1.4 BS01 YJ9 A 1 G23 C25 G61 E63 G67 G68 L69 M70 Y72 A135 M161 D162 H163 G164 A214 G23 C25 G61 E63 G67 G68 L69 M70 Y72 A135 M161 D162 H163 G164 A214 Q19 C25 H163 N187 Q19 C25 H163 N187 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21898833 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2yjc A 1.14 BS01 424 A 1 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 Q19 C25 H163 N187 Q19 C25 H163 N186 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 21898833 1221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTSDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 2yjq A 2.25 BS01 BGC C 1 N48 R49 D65 N42 R43 D59 3.2.1.151','3.2.1.4 remove_due_to_license_issue Q1A2D0 21795708 1 AKTITIKVDTFKDRKPISPYIYGTNQDLAGDENMAARRLGGNRMTGYNWENNMSNAGSDWQHSSDNYLCSNGGLTQAECEKPGAVVTSFHDQSLKLGTYSLVTLPMAGYVAADGNGSVQESEAAPSARWNQVVNAKNAPFQLQPDLNDNYVYVDEFVHFLVNKYGTASTKAGVKGYALDNEPALWSHTHPRIHPEKVGAKELVDRSVSLSKAVKAIDAGAEVFGPVLYGFGAYKDLQTAPDWDSVKGNYSWFVDYYLDQMRLSSQVEGKRLLDVFDVHWYPEAMGGGIRITNEVGNDETKKARMQAPRTLWDPTYKEDSWIAQWFSEFLPILPRLKQSVDKYYPGTKLAMTSYSYGGENDISGGIAMTDVLGILGKNDVYMANYWKLKDGVNNYVSAAYKLYRNYDGKNSTFGDTSVSAQTSDIVNSSVHASVTNSDKELHLVVMNKSMDSAFDAQFDLSGAKTYISGKVWGFDKNSSQIKEAAPITQISGNRFTYTVPPLTAYHIVLTT 2yjq A 2.25 BS02 BGC C 2 R49 W66 R43 W60 3.2.1.151','3.2.1.4 remove_due_to_license_issue Q1A2D0 21795708 2 AKTITIKVDTFKDRKPISPYIYGTNQDLAGDENMAARRLGGNRMTGYNWENNMSNAGSDWQHSSDNYLCSNGGLTQAECEKPGAVVTSFHDQSLKLGTYSLVTLPMAGYVAADGNGSVQESEAAPSARWNQVVNAKNAPFQLQPDLNDNYVYVDEFVHFLVNKYGTASTKAGVKGYALDNEPALWSHTHPRIHPEKVGAKELVDRSVSLSKAVKAIDAGAEVFGPVLYGFGAYKDLQTAPDWDSVKGNYSWFVDYYLDQMRLSSQVEGKRLLDVFDVHWYPEAMGGGIRITNEVGNDETKKARMQAPRTLWDPTYKEDSWIAQWFSEFLPILPRLKQSVDKYYPGTKLAMTSYSYGGENDISGGIAMTDVLGILGKNDVYMANYWKLKDGVNNYVSAAYKLYRNYDGKNSTFGDTSVSAQTSDIVNSSVHASVTNSDKELHLVVMNKSMDSAFDAQFDLSGAKTYISGKVWGFDKNSSQIKEAAPITQISGNRFTYTVPPLTAYHIVLTT 2yjq A 2.25 BS03 OXZ A 1 G47 N48 E187 Y286 W391 G41 N42 E181 Y280 W385 3.2.1.151','3.2.1.4 remove_due_to_license_issue Q1A2D0 21795708 1518 AKTITIKVDTFKDRKPISPYIYGTNQDLAGDENMAARRLGGNRMTGYNWENNMSNAGSDWQHSSDNYLCSNGGLTQAECEKPGAVVTSFHDQSLKLGTYSLVTLPMAGYVAADGNGSVQESEAAPSARWNQVVNAKNAPFQLQPDLNDNYVYVDEFVHFLVNKYGTASTKAGVKGYALDNEPALWSHTHPRIHPEKVGAKELVDRSVSLSKAVKAIDAGAEVFGPVLYGFGAYKDLQTAPDWDSVKGNYSWFVDYYLDQMRLSSQVEGKRLLDVFDVHWYPEAMGGGIRITNEVGNDETKKARMQAPRTLWDPTYKEDSWIAQWFSEFLPILPRLKQSVDKYYPGTKLAMTSYSYGGENDISGGIAMTDVLGILGKNDVYMANYWKLKDGVNNYVSAAYKLYRNYDGKNSTFGDTSVSAQTSDIVNSSVHASVTNSDKELHLVVMNKSMDSAFDAQFDLSGAKTYISGKVWGFDKNSSQIKEAAPITQISGNRFTYTVPPLTAYHIVLTT 2yjw A 1.61 BS01 YJW A 1 N51 A55 K58 D93 G97 M98 L107 G108 T184 N35 A39 K42 D77 G81 M82 L91 G92 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2yjx A 1.83 BS01 YJX A 1 F22 L103 L107 G108 F138 Y139 W162 F170 F6 L87 L91 G92 F122 Y123 W146 F154 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2yk1 H 1.85 BS01 NCT H 1 I29 G31 S50 V93 E101 I27 G29 S44 V90 E103 Kd=7.4nM remove_due_to_license_issue 22079050 300 QLLESGPGLVKPSETLSLTCTVSGGSIWGWIRQPPGKGLEWIGSIYSSGSTYYNPSLKSRVTTSVDTSKNQFSLRLSSVTAADTAVYYCVAWFGDLLSLKGVELWGQGTLVTVSSASTKGPSVFPLALGCLVKDYFPEPVTVSWNLTSGVHTFPAVLQSSGLYSLSSVVTCNVDHKPSNTKV 2yk1 L 1.85 BS01 NCT H 1 Y34 Y36 W96 Y33 Y35 W97 remove_due_to_license_issue 22079050 300 ELTQPPSASGTPGQRVTISCSGSSSNIGSNYVYWYQQLPGTAPKLLIYRNNQRPSGVPDRFSGSKSGTSASLAISGLRSEDEADYYCAAWDDSLSAWVFGGGTQLDILGQPKAAPSVTLFPPSPKATLVCLISDFYPGAVTVAAGVETTTPSKQSNNKYAASSYLSLTPEQWSYSCQVTHEGSTVEKT 2yk9 A 1.32 BS01 YK9 A 1 F22 I26 L103 L107 G108 F138 Y139 W162 F170 F6 I10 L87 L91 G92 F122 Y123 W146 F154 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2ykb A 1.93 BS01 YKB A 1 F22 I26 A55 M98 L103 I104 L107 G108 F138 Y139 W162 F170 F6 I10 A39 M82 L87 I88 L91 G92 F122 Y123 W146 F154 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2ykc A 1.67 BS01 YKC A 1 F22 M98 L103 L107 G108 F138 Y139 W162 F170 T184 F6 M82 L87 L91 G92 F122 Y123 W146 F154 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2yke A 1.43 BS01 YKE A 1 F22 N51 A55 D93 M98 L103 L107 G108 F138 Y139 W162 F170 T184 F6 N35 A39 D77 M82 L87 L91 G92 F122 Y123 W146 F154 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2yki A 1.67 BS01 YKI A 1 F22 N51 D93 M98 L103 L107 G108 F138 Y139 W162 F170 F6 N35 D77 M82 L87 L91 G92 F122 Y123 W146 F154 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.35nM remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2ykj A 1.46 BS01 YKJ A 1 F22 M98 L103 L107 G108 F138 Y139 W162 F170 T184 F6 M82 L87 L91 G92 F122 Y123 W146 F154 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21972823 1224 METFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 2ylc A 1.3 BS01 U A 1 F42 H57 F38 H53 ? 0003723,0006355 remove_due_to_license_issue P0A1R0 21737752 1073 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPSRPVSH 2yln A 1.12 BS01 CYS A 1 W97 N114 R123 S165 N166 W62 N79 R88 S130 N131 ? Kd=0.021uM remove_due_to_license_issue Q5F9M1 22138345 500 AISGSLIERINNKGTVTVGTEGTYAPFTYHDKDGKLTGYDVEVTRAVAEKLGVKVEFKETQWDSMMAGLKAGRFDVVANQVGLTSPERQATFDKSEPYSWSGAVLVAHNDSNIKSIADIKGVKTAQSLTSNYGEKAKAAGAQLVPVDGLAQSLTLIEQKRADATLNDELAVLDYLKKNPNAGVKIVWSAPADEKVGSGLIVNKGNDEAVAKFSTAINELKADGTLKKLGEQFFGKDISVQ 2yln A 1.12 BS02 CYS A 2 E56 Y59 W97 S162 G183 L184 N201 E21 Y24 W62 S127 G148 L149 N166 ? Kd=0.021uM remove_due_to_license_issue Q5F9M1 22138345 600 AISGSLIERINNKGTVTVGTEGTYAPFTYHDKDGKLTGYDVEVTRAVAEKLGVKVEFKETQWDSMMAGLKAGRFDVVANQVGLTSPERQATFDKSEPYSWSGAVLVAHNDSNIKSIADIKGVKTAQSLTSNYGEKAKAAGAQLVPVDGLAQSLTLIEQKRADATLNDELAVLDYLKKNPNAGVKIVWSAPADEKVGSGLIVNKGNDEAVAKFSTAINELKADGTLKKLGEQFFGKDISVQ 2ylo A 2.5 BS02 YLO A 1 P723 G724 R726 N727 F826 E829 L830 N833 Y834 P54 G55 R57 N58 F157 E160 L161 N164 Y165 ? remove_due_to_license_issue IC50=13100nM P10275 22047606 1922 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ylp A 2.3 BS02 056 A 1 F673 N727 F826 E829 L830 N833 Y834 E837 F3 N57 F156 E159 L160 N163 Y164 E167 ? remove_due_to_license_issue P10275 22047606 1922 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ylp A 2.3 BS03 056 A 2 V716 V730 Q733 M734 V46 V60 Q63 M64 ? remove_due_to_license_issue P10275 22047606 1923 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ylq A 2.4 BS02 YLQ A 1 F673 N727 F826 E829 L830 N833 E837 F3 N57 F156 E159 L160 N163 E167 ? remove_due_to_license_issue IC50=>10000nM P10275 22047606 1922 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2ym3 A 2.007 BS01 YM3 A 1 L15 G16 V23 A36 E85 Y86 C87 G90 E91 L137 L8 G9 V11 A24 E62 Y63 C64 G67 E68 L114 D130 K132 E134 N135 D148 T170 D107 K109 E111 N112 D125 T147 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.2uM remove_due_to_license_issue IC50=1200nM O14757 22111927 1271 DWDLVQTLGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2ym4 A 2.35 BS01 4YM A 1 L15 G16 K38 E85 Y86 C87 E91 L137 S147 L12 G13 K35 E66 Y67 C68 E72 L118 S128 D130 K132 E134 N135 D148 T170 D111 K113 E115 N116 D129 T151 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.5uM remove_due_to_license_issue IC50=1500nM O14757 22111927 1271 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVNIKKEICINKMLNHENVVKFYGHQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2ym5 A 2.03 BS01 YM5 A 1 V23 A36 E85 Y86 C87 E91 L137 S147 V11 A24 E63 Y64 C65 E69 L115 S125 D130 K132 E134 N135 D148 T170 D108 K110 E112 N113 D126 T148 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.43uM remove_due_to_license_issue IC50=430nM O14757 22111927 1271 DWDLVQTLGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2ym6 A 2.01 BS01 YM6 A 1 L15 V23 L84 E85 C87 E91 L137 L9 V17 L67 E68 C70 E74 L120 D130 K132 E134 N135 D148 T170 D113 K115 E117 N118 D131 T153 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.88uM remove_due_to_license_issue IC50=880nM O14757 22111927 1271 EDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2ym7 A 1.81 BS01 YM7 A 1 L15 A36 K38 L84 E85 Y86 C87 E91 E134 L137 S147 D148 L9 A25 K27 L61 E62 Y63 C64 E68 E111 L114 S124 D125 D130 K132 E134 N135 D148 T170 D107 K109 E111 N112 D125 T147 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.13uM remove_due_to_license_issue IC50=130nM O14757 22111927 1272 EDWDLVQTLGEVQLAVNRVTEEAVAVKIVNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 2ym7 A 1.81 BS02 YM7 A 2 W9 E33 Y71 R74 F83 W3 E22 Y50 R53 F60 D130 K132 E134 N135 D148 T170 D107 K109 E111 N112 D125 T147 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.13uM remove_due_to_license_issue IC50=130nM O14757 22111927 1273 EDWDLVQTLGEVQLAVNRVTEEAVAVKIVNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 2ym8 A 2.07 BS01 YM8 A 1 A36 L84 E85 Y86 C87 E134 L137 S147 D148 A24 L60 E61 Y62 C63 E110 L113 S123 D124 D130 K132 E134 N135 D148 T170 D106 K108 E110 N111 D124 T146 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.013uM remove_due_to_license_issue IC50=13nM O14757 22111927 1271 DWDLVQTLGEVQLAVNRVTEEAVAVKIVNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2ymd A 1.96 BS01 SRO A 1 Y91 W145 V146 C188 C189 Y193 Y91 W145 V146 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=693uM remove_due_to_license_issue Q8WSF8 23196367 1213 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYESTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCALTFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAGNGFF 2ymd A 1.96 BS02 SRO E 1 I104 V106 M114 I116 I104 V106 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=693uM remove_due_to_license_issue Q8WSF8 23196367 1213 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYESTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCALTFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAGNGFF 2ymd B 1.96 BS01 SRO A 1 I104 V106 M114 I116 I104 V106 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=693uM remove_due_to_license_issue Q8WSF8 23196367 1213 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYESTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCALTFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAGNG 2ymd B 1.96 BS02 SRO B 1 Y91 W145 V146 C188 C189 Y193 Y91 W145 V146 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=693uM remove_due_to_license_issue Q8WSF8 23196367 1212 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYESTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCALTFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAGNG 2yme F 2.4 BS01 CWB F 1 W145 Y186 C188 Y193 W145 Y186 C188 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=343uM remove_due_to_license_issue Q8WSF8 23196367 1207 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2yme G 2.4 BS01 CWB F 1 W53 R55 I116 W53 R55 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=343uM remove_due_to_license_issue Q8WSF8 23196367 1207 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2yme G 2.4 BS02 CWB G 1 Y91 W145 C188 C189 Y193 Y91 W145 C188 C189 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 Kd=343uM remove_due_to_license_issue Q8WSF8 23196367 1207 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 2ynd A 1.89 BS02 646 A 1 D98 F103 F105 G199 Y211 H213 F226 S319 Y334 L388 L410 D73 F78 F80 G174 Y186 H188 F201 S294 Y309 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=32nM remove_due_to_license_issue A5K1A2 24451586 1001 IDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 2yne A 1.72 BS02 YNE A 1 E97 F105 Y211 Y315 Y334 S335 N365 A366 L367 L388 L409 L410 E71 F79 Y185 Y289 Y308 S309 N339 A340 L341 L362 L383 L384 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=2.7nM remove_due_to_license_issue A5K1A2 24451586 1001 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 2yof A 1.82 BS01 74W A 1 D17 R18 F44 P45 R47 F74 R78 R99 G104 Y107 E151 Y153 E154 D15 R16 F42 P43 R45 F72 R76 R97 G102 Y105 E141 Y143 E144 2.7.4.8,2.7.4.9 0004385,0004550,0004798,0005524,0005634,0005737,0005739,0006177,0006227,0006233,0006235,0009165,0016301,0046710,0046940,0050316 Ki=25uM remove_due_to_license_issue Ki=25000nM Q8I4S1 23240776 211 DDKKKGKFIVFEGLDRSGKSTQSKLLVEYLKNNNVEVKHLYFPNRETGIGQIISKYLKMENSMSNETIHLLFSANRWEHMNEIKSLLLKGIWVVCDRYAYSGVAYSSGALNLNKTWCMNPDQGLIKPDVVFYLNVPPNYEEIYEKVETQKKIYETYKHFAHEDYWINIDATRKIEDIHNDIVKEVTKIKVEPEEFNFLWS 2yog A 1.5 BS01 74X A 1 F44 P45 L59 F74 R78 R99 S103 G104 Y107 F41 P42 L56 F71 R75 R96 S100 G101 Y104 2.7.4.8,2.7.4.9 0004385,0004550,0004798,0005524,0005634,0005737,0005739,0006177,0006227,0006233,0006235,0009165,0016301,0046710,0046940,0050316 Ki=31uM remove_due_to_license_issue Ki=31000nM Q8I4S1 23240776 211 DKKKGKFIVFEGLDRSGKSTQSKLLVEYLKNNNVEVKHLYFPNRETGIGQIISKYLKMENSMSNETIHLLFSANRWEHMNEIKSLLLKGIWVVCDRYAYSGVAYSSGALNLNKTWCMNPDQGLIKPDVVFYLNVPPNYIYEKVETQKKIYETYKHFAHEDYWINIDATRKIEDIHNDIVKEVTKIKVEPEEFNFLWS 2yoh A 1.6 BS01 WMJ A 1 D17 R18 F44 P45 L59 F74 R78 R99 S103 G104 Y107 E151 D14 R15 F41 P42 L56 F71 R75 R96 S100 G101 Y104 E140 2.7.4.8,2.7.4.9 0004385,0004550,0004798,0005524,0005634,0005737,0005739,0006177,0006227,0006233,0006235,0009165,0016301,0046710,0046940,0050316 Ki=11uM remove_due_to_license_issue Ki=11000nM Q8I4S1 23240776 211 DKKKGKFIVFEGLDRSGKSTQSKLLVEYLKNNNVEVKHLYFPNRETGIGQIISKYLKMENSMSNETIHLLFSANRWEHMNEIKSLLLKGIWVVCDRYAYSGVAYSSGALNLNKTWCMNPDQGLIKPDVVFYLNVPPNYEEIYEKVETQKKIYETYKHFAHEDYWINIDATRKIEDIHNDIVKEVTKIKVEPEEFNFLWS 2yoj A 1.76 BS01 8Y6 A 1 R200 C366 S367 G410 M414 Y415 Q446 I447 Y448 R195 C361 S362 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=5nM remove_due_to_license_issue O92972 24900812 1569 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 2yol A 3.2 BS01 EBN A 1 G83 F85 H1051 D1075 D1129 Y1130 T1132 G1151 N1152 G1153 I1155 Y1161 G37 F39 H94 D118 D172 Y173 T175 G194 N195 G196 I198 Y204 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue Ki=130nM P06935 23307694 2170 SHMTDMWIERTADITWESDAEITGSSERVDVRLDDDGNFQLMNDPGVLWDTSPKEYKKGDTTTGVYRIMTRGLLGSYQAGAGVMVEGVFHTLWHTTKGAALMSGEGRLDPYWGSVKEDRLCYGGPWKLQHKWNGHDEVQMIVVEPGKNVKNVQTKPGVFKTPEGEIGAVTLDYPTGTSGSPIVDKNGDVIGLYGNGVIMPNGSYISAIVQGE 2ypf A 2.55 BS01 dna B 0 R266 V269 D301 Q305 G336 Q339 I369 Q407 I437 Q441 I471 G472 Q475 I505 Q509 D539 Q543 D573 Q577 Q611 I641 G642 I675 G676 Q679 D709 K712 Q713 D743 G744 Q747 G778 Q781 K814 Q815 K848 Q849 R80 V83 D115 Q119 G150 Q153 I183 Q221 I251 Q255 I285 G286 Q289 I319 Q323 D353 Q357 D387 Q391 Q425 I455 G456 I489 G490 Q493 D523 K526 Q527 D557 G558 Q561 G592 Q595 K628 Q629 K662 Q663 ? remove_due_to_license_issue Q3ZD73 23999294 -2 ~ 19 AFTHAHIVALSQHPAALATVAVKYQDMIAALPEATHEAIVAVAKQWSGARALEALLTVAGELRGPPLQLDTGQLLKIAKRGGVTAVEAVHAWRNALTGAPLNLTPEQVVAIASHDGGKQALETVQRLLPVLCQAHGLTPQQVVAIASNGGGKQALETVQRLLPVLCQAHGLTPEQVVAIASNIGGKQALETVQALLPVLCQAHGLTPQQVVAIASNGGGKQALETVQRLLPVLCQAHGLTPEQVVAIASNIGGKQALETVQALLPVLCQAHGLTPEQVVAIASNIGGKQALETVQALLPVLCQAHGLTPEQVVAIASNIGGKQALETVQALLPVLCQAHGLTPEQVVAIASHDGGKQALETVQRLLPVLCQAHGLTPEQVVAIASHDGGKQALETVQRLLPVLCQAHGLTPQQVVAIASNGGGKQALETVQRLLPVLCQAHGLTPEQVVAIASNIGGKQALETVQALLPVLCQAHGLTPEQVVAIASNIGGKQALETVQALLPVLCQAHGLTPEQVVAIASHDGGKQALETVQRLLPVLCQAHGLTPEQVVAIASHDGGKQALETVQRLLPVLCQAHGLTPEQVVAIASHDGGKQALETVQRLLPVLCQAHGLTPQQVVAIASNGGGKQALETVQRLLPVLCQAAGLTPEQVVAIASHDGGKQALETVQRLLPVL 2ypi A 2.5 BS01 PGA A 1 N10 K12 H95 E165 I170 G171 S211 G232 N9 K11 H94 E164 I169 G170 S210 G231 N10 K12 H95 E97 E165 G171 S211 N9 K11 H94 E96 E164 G170 S210 5.3.1.1 0004807,0005737,0005739,0005829,0005886,0006094,0006096,0016853,0019563,0046166 Ki=15uM remove_due_to_license_issue P00942 2204418 249 ARTFFVGGNFKLNGSKQSIKEIVERLNTASIPENVEVVICPPATYLDYSVSLVKKPQVTVGAQNAYLKASGAFTGENSVDQIKDVGAKWVILGHSERRSYFHEDDKFIADKTKFALGQGVGVILCIGETLEEKKAGKTLDVVERQLNAVLEEVKDWTNVVVAYEPVWAIGTGLAATPEDAQDIHASIRKFLASKLGDKAASELRILYGGSANGSNAVTFKDKADVDGFLVGGASLKPEFVDIINSRN 2ypi B 2.5 BS01 PGA B 1 K12 H95 E165 A169 I170 G171 G210 S211 L230 G232 K11 H94 E164 A168 I169 G170 G209 S210 L229 G231 N10 K12 H95 E97 E165 G171 S211 N9 K11 H94 E96 E164 G170 S210 5.3.1.1 0004807,0005737,0005739,0005829,0005886,0006094,0006096,0016853,0019563,0046166 Ki=15uM remove_due_to_license_issue P00942 2204418 249 ARTFFVGGNFKLNGSKQSIKEIVERLNTASIPENVEVVICPPATYLDYSVSLVKKPQVTVGAQNAYLKASGAFTGENSVDQIKDVGAKWVILGHSERRSYFHEDDKFIADKTKFALGQGVGVILCIGETLEEKKAGKTLDVVERQLNAVLEEVKDWTNVVVAYEPVWAIGTGLAATPEDAQDIHASIRKFLASKLGDKAASELRILYGGSANGSNAVTFKDKADVDGFLVGGASLKPEFVDIINSRN 2ypo A 2.0 BS02 PHE A 1 F91 M92 R171 A174 N175 F87 M88 R167 A170 N171 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=21uM remove_due_to_license_issue O53512 23274137 900 MNWTVDIPIDLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypo B 2.0 BS01 PHE A 1 V5 V55 V5 V50 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=21uM remove_due_to_license_issue O53512 23274137 900 MNWTVDIPILPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypo B 2.0 BS03 PHE B 1 F91 R171 A174 N175 F86 R166 A169 N170 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=21uM remove_due_to_license_issue O53512 23274137 900 MNWTVDIPILPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypp A 2.3 BS01 TYR A 1 F91 R171 N175 F89 R169 N173 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=39uM remove_due_to_license_issue O53512 23274137 800 MNWTVDIPIDPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypp A 2.3 BS03 TYR B 1 V55 Y173 A174 V53 Y171 A172 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=39uM remove_due_to_license_issue O53512 23274137 800 MNWTVDIPIDPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypp B 2.3 BS01 TYR A 1 V55 Y173 A174 V52 Y170 A171 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=39uM remove_due_to_license_issue O53512 23274137 800 MNWTVDIPIPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypp B 2.3 BS03 TYR B 1 F91 R171 A174 N175 F88 R168 A171 N172 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=39uM remove_due_to_license_issue O53512 23274137 800 MNWTVDIPIPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ypp B 2.3 BS04 TYR B 2 L15 P16 L18 R23 E53 R256 L12 P13 L15 R20 E50 R253 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=39uM remove_due_to_license_issue O53512 23274137 801 MNWTVDIPIPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 2ywp A 2.9 BS01 A42 A 1 L15 G16 A36 K38 Y86 C87 L137 D148 L14 G15 A35 K37 Y85 C86 L136 D147 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=7nM O14757 16446090 1 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 2yxj A 2.2 BS01 N3C A 1 F97 Y101 F105 V126 E129 L130 G138 R139 V141 Y195 F37 Y41 F45 V66 E69 L70 G78 R79 V81 Y135 ? 0042981 ic50=9nM remove_due_to_license_issue Ki=<1.000000nM, IC50=6nM, Kd=0.37nM, EC50=30nM Q07817 17572662 1001 SNRELVVDFLSYKLSQKGYSWSSEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGN 2yz3 A 2.3 BS03 M5P A 1 F42 Y47 H96 D98 H159 R185 N190 H220 F31 Y36 H85 D87 H148 R174 N179 H209 H94 H96 D98 H159 C178 Y181 N190 H220 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 Ki=220nM remove_due_to_license_issue Q7BJM5 18052313 401 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVV 2z1w A 1.63 BS02 BDI A 1 Y106 D156 C158 Q203 G229 G230 M260 Y96 D135 C137 Q182 G208 G209 M239 D102 D280 C318 C320 C323 H349 D92 D259 C297 C299 C302 H328 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 remove_due_to_license_issue P28720 17949745 600 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLTKQSEEGVTFKMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGQGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 2z3h A 1.5 BS02 BLO A 1 E25 S28 V29 N45 Y47 C54 A55 E56 R82 P87 C88 E23 S26 V27 N43 Y45 C52 A53 E54 R80 P85 C86 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 2500 LSQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLPS 2z3h B 1.5 BS01 BLO A 1 Y126 W128 Y124 W126 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 2500 LSQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLPSGYVW 2z3h B 1.5 BS03 BLO B 1 E25 S28 V29 N45 Y47 C54 A55 E56 R82 P87 C88 E23 S26 V27 N43 Y45 C52 A53 E54 R80 P85 C86 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 2501 LSQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLPSGYVW 2z3h C 1.5 BS02 BLO C 1 E25 D26 S28 V29 N45 Y47 C54 E56 R82 P87 C88 E23 D24 S26 V27 N43 Y45 C52 E54 R80 P85 C86 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 2502 LSQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLPS 2z3h D 1.5 BS02 BLO D 1 E25 D26 S28 V29 N45 Y47 C54 E56 R82 P87 C88 E23 D24 S26 V27 N43 Y45 C52 E54 R80 P85 C86 3.5.4.23 0003824,0004126,0005737,0005829,0008270,0009972,0016787,0042802,0046677,0046872,0047711,0055086,0072527,1901135 remove_due_to_license_issue P0C2P0 17959604 2503 LSQEESTLIERATATINSIPISEDYSVASAALSSDGRIFTGVNVYHFTGGPCAELVVLGTAAAAAAGNLTCIVAIGNENRGILSPCGRCRQVLLDLHPGIKAIVKDSDGQPTAVGIRELLP 2z3z A 1.95 BS01 AIO A 1 Q203 E205 Y518 H522 S603 Y604 Y635 Y639 H710 Q132 E134 Y441 H445 S522 Y523 Y554 Y558 H629 Y518 S603 Y604 D678 H710 Y441 S522 Y523 D597 H629 3.4.14.12 0004177,0006508,0008236,0008239 remove_due_to_license_issue Q7MUW6 18042490 801 VVGLQWMGDNYVFIEGDDLVFNKTTRFSAADLNALMFPSFRTLDAGRGLVVLFTQGGLVGFDMLARKVTYLFDTNEETASLDFSPVGDRVAYVRNHNLYIARGGKLGEGMSRAIAVTIDGTETLVYGQAVHQREFGIEKGTFWSPKGSCLAFYRMDQSMVKPTPIVDYHPLEAESKPLYYPMAGTPSHHVTVGIYHLATGKTVYLQTGEPKEKFLTNLSWSPDENILYVAEVNRAQNECKVNAYDAETGRFVRTLFVETDKHYVEPLHPLTFLPGSNNQFIWQSRRDGWNHLYLYDTTGRLIRQVTKGEWEVTNFAGFDPKGTRLYFESTEASPLERHFYCIDIKGGKTKDLTPESGMHRTQLSPDGSAIIDIFQSPTVPRKVTVTNIGKGSHTLLEAKAMPEIRTGTIMAADGQTPLYYKLTMPLHFDPAKKYPVIVYVYGGPHAQLVTKTWGGWDIYMAQKGYAVFTVDSRGSANRGAAFEQVIHRRLGQTEMADQMCGVDFLKSQSWVDADRIGVHGWSYGGFMTTNLMLTHGDVFKVGVAGGPVIDWNRYAIMYGERYFDAPQENPEGYDAANLLKRAGDLKGRLMLIHGAIDPVVVWQHSLLFLDACVKARTYPDYYVYPSHEHNVMGPDRVHLYETITRYFTDHL 2z4b A 2.34 BS01 DC8 A 1 M295 E305 M336 L339 I376 F377 H475 L476 M29 E39 M70 L73 I110 F111 H202 L203 ? 0003677,0004879,0006355 Ki=0.44nM remove_due_to_license_issue Ki=0.44nM Q92731 17614275 80 DALSPEQLVLTLLEAEPPHVLISRPASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMKVPVYDLLLEMLNAH 2z4o A 1.6 BS01 065 B 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2z4o B 1.6 BS01 065 B 1 D125 G127 A128 D129 G148 G149 I150 D25 G27 A28 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.27nM remove_due_to_license_issue P03367 17696515 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2z4r A 3.05 BS02 ADP A 1 Y102 F107 V108 V139 G140 L141 G142 K143 T144 H145 I271 L299 R300 Y7 F12 V13 V44 G45 L46 G47 K48 T49 H50 I176 L204 R205 ? 0003677,0003688,0005524,0005737,0005886,0006260,0006270,0006275,0016887,0043565 remove_due_to_license_issue P46798 18216012 501 TPLNPDYTFENFVVGPGNSFAYHAALEVAKHPGRYNPLFIYGGVGLGKTHLLQSIGNYVVQNEPDLRVMYITSEKFLNDLVDSMKEGKLNEFREKYRKKVDILLIDDVQFLIGKTGVQTELFHTFNELHDSGKQIVICSDREPQKLSEFQDRLVSRFQMGLVAKLEPPDEETRKSIARKMLEIEHGELPEEVLNFVAENVDDNLRRLRGAIIKLLVYKETTGKEVDLKEAILLLKDFIKP 2z4w A 2.45 BS03 749 A 1 R44 H73 D80 R89 L143 Q147 K174 Y210 D214 K238 R38 H67 D74 R83 L137 Q141 K168 Y201 D205 K223 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.98uM remove_due_to_license_issue Q12051 18800762 1101 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSGHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2z4w B 2.45 BS03 749 B 1 H73 S76 D80 R89 L143 Q147 K174 F179 Y210 D214 K238 H65 S68 D72 R81 L135 Q139 K166 F171 Y198 D202 K220 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.98uM remove_due_to_license_issue Q12051 18800762 1102 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLP 2z4y A 2.1 BS01 252 A 1 D80 R89 L143 K174 Q211 D214 K238 D74 R83 L137 K168 Q199 D202 K222 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM remove_due_to_license_issue Q12051 18800762 1201 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2z4y A 2.1 BS02 252 A 2 G40 R44 H73 R89 R90 G37 R38 H67 R83 R84 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM remove_due_to_license_issue Q12051 18800762 1202 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKND 2z4y B 2.1 BS01 252 B 1 S76 D80 R89 L143 H144 Q147 K174 Q211 D214 K238 S63 D67 R76 L130 H131 Q134 K161 Q193 D196 K214 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.71uM remove_due_to_license_issue Q12051 18800762 1203 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSLVPFINLLGIIYQIRDDYLNLKDFGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN 2z4z A 2.09 BS01 SC0 A 1 R44 H73 D80 R89 L143 K174 T175 Y210 Q211 D214 K238 L340 R41 H70 D77 R86 L140 K171 T172 Y205 Q206 D209 K227 L315 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=1.86uM remove_due_to_license_issue Q12051 18800762 1201 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHGHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPELLYIIDHLSEL 2z4z B 2.09 BS01 SC0 B 1 D80 R89 L143 Q147 K174 Y210 Q211 D214 K238 D74 R83 L137 Q141 K168 Y202 Q203 D206 K224 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=1.86uM remove_due_to_license_issue Q12051 18800762 1202 KMEAKIDELINNDPVWSSQNESLISKPYNHILLKKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHGHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPLYIIDHL 2z50 A 2.01 BS01 028 A 1 D80 R89 Q147 K174 Q211 K238 D68 R77 Q135 K162 Q193 K214 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=11.22uM remove_due_to_license_issue Q12051 18800762 1201 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN 2z50 B 2.01 BS01 028 B 1 D80 R89 Q147 K174 Q211 K238 D65 R74 Q132 K159 Q191 K212 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=11.22uM remove_due_to_license_issue Q12051 18800762 1202 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKN 2z52 A 2.13 BS03 H23 A 1 S76 D80 R89 Y112 L140 H144 Q147 K174 K238 S68 D72 R81 Y104 L132 H136 Q139 K166 K222 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Q12051 18800762 1001 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHGHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNKYLP 2z52 B 2.13 BS03 H23 B 1 S76 D80 R89 Y112 H144 Q147 K174 K238 S68 D72 R81 Y104 H136 Q139 K166 K220 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=2.69uM remove_due_to_license_issue Q12051 18800762 1002 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLP 2z60 A 1.95 BS01 P3Y A 1 L248 G249 Y253 V256 A269 F317 M318 G321 N322 L370 L21 G22 Y26 V29 A42 F87 M88 G91 N92 L140 D363 A365 R367 N368 D381 P402 D133 A135 R137 N138 D151 P172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 17718712 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG 2z78 A 2.1 BS01 H86 A 1 I48 H73 S76 I79 D80 R89 L143 Q147 T175 F179 Y210 Q211 D214 K238 I45 H70 S73 I76 D77 R86 L140 Q144 T172 F176 Y207 Q208 D211 K233 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Q12051 18800762 1300 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSHHGHSLVPFINLLGIIYQIRDDYLNLKDFQMSKGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPELLYIIDHLSEL 2z78 B 2.1 BS01 H86 B 1 L47 H73 S76 L77 D80 R89 L143 Q147 K174 L178 T182 Y210 Q211 D214 K238 L44 H70 S73 L74 D77 R86 L140 Q144 K171 L175 T179 Y204 Q205 D208 K229 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 remove_due_to_license_issue Q12051 18800762 1301 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSSHSLVPFINLLGIIYQIRDDYLNLKDFQMSGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPELLYIIDHLSEL 2z7g A 2.52 BS02 EH9 A 1 H14 D16 F62 D293 H14 D16 F62 D293 H12 H14 H211 E214 H235 D292 H12 H14 H211 E214 H235 D292 3.5.4.4 0004000,0005515,0005737,0005764,0005829,0005886,0006154,0007155,0008270,0009117,0009168,0009897,0016787,0019239,0031410,0042110,0043103,0046103,0046872,0046936,0060169,0060205,0070161 remove_due_to_license_issue Ki=0.82nM P56658 18549808 356 TPAFDKPKVELHVHLDGAIKPETILYYGKRRGIALPADTPEELQNIIGMDKPLTLPDFLAKFDYYMPAIAGCRDAIKRIAYEFVEMKAKDGVVYVEVRYSPHLLANSKVEPIPWNQAEGDLTPDEVVSLVNQGLQEGERDFGVKVRSILCCMRHQPSWSSEVVELCKKYREQTVVAIDLAGDETIEGSSLFPGHVQAYAEAVKSGVHRTVHAGEVGSANVVKEAVDTLKTERLGHGYHTLEDTTLYNRLRQENMHFEICPWSSYLTGAWKPDTEHAVIRFKNDQVNYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEDEKKELLDLLYKAYR 2z7h A 2.08 BS02 GG3 A 1 R44 H73 D80 R89 K174 F179 Y210 D214 K238 R35 H64 D71 R80 K165 F170 Y198 D202 K222 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 Ki=115nM remove_due_to_license_issue Q12051 18442135 1302 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSGHSLVPFINLLGIIYQIRDDYLNLKDFQMGFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNDNENKYLPELLYIIDHLS 2z7i A 2.1 BS02 742 A 1 R44 H73 D80 R89 K174 F179 T182 I203 Q211 D214 K238 R41 H70 D77 R86 K171 F176 T179 I197 Q205 D208 K226 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005737,0005739,0008299,0015031,0016114,0016740,0033384,0033386,0045337,0046872 ic50=0.1uM remove_due_to_license_issue Q12051 18800762 1302 NKMEAKIDELINNDPVWSSQNESLISKPYNHILLKPGKNFRLNLIVQINRVMNLPKDQLAIVSQIVELLHNSSLLIDDIEDNAPLRRGQTTSHLIFGVPSTINTANYMYFRAMQLVSQLTTKEPLYHNLITIFNEELINLHRGQGLDIYWRDFLPEIIPTQEMYLNMVMNKTGGLFRLTLRLMEALSPSGHSLVPFINLLGIIYQIRDDYLNLKDFQFAEDITEGKLSFPIVHALNFTKTKGQTEQHNEILRILLLRTSDKDIKLKLIQILEFDTNSLAYTKNFINQLVNMIKNENKYLPDELLYIIDHLSEL 2z7r A 2.0 BS01 STU A 1 L68 G69 A92 K94 D142 F143 L144 D148 E191 N192 L194 T204 L16 G17 A40 K42 D79 F80 L81 D85 E128 N129 L131 T141 D187 K189 E191 N192 D205 T225 D124 K126 E128 N129 D142 T150 2.7.11.1 0004672,0004674,0005524,0006468 ic50~0.4nM remove_due_to_license_issue Q15418 17965187 1 GSEKADPSHFELLKVLGQGSFGKVFLVRKVTRPDSGHLYAMKVLKKATLKVILADVNHPFVVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALGLDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKEGTVEYMAPEVVNRQGHSHSADWWSYGVLMFEMLTGSLPFQGKDRKETMTLILKAKLGMPQFLSTEAQSLLRALFKRNPANRLGSGPDGAEEIKRHVFYSTIDWNKLYRREIKPPFKP 2z92 A 2.3 BS01 ENE A 1 H35A I37 W47 N58 D95 W103 H34 I36 W46 N57 D97 W104 Kd=0.8nM remove_due_to_license_issue 18463096 1 QLLESGPDLVKPSQSLSLTCTVTGYSITSGYNWHWIRQFPGNKLEWMGYIHYRGTTNYNTSLKSRISITRDSSKNQFFLQLNSVTTEDTATYYCACDDFYSDYWGQGTIVTVSSAKTTPPSVYPLAPSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVP 2z92 B 2.3 BS01 ENE A 1 Y36 R46 W91 N94 P96 Y35 R45 W90 N93 P95 remove_due_to_license_issue 18463096 1 ELVMTQTPAIMSASPGEKVTMTCSASSSVSSVHWYQQKSGTSPKRWIYDTSKLPSGVPGRFSGSGSGTSYSLTISSMEAEDAATYYCQQWSSNPPTFGAGTKLEVKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 2z94 A 1.78 BS02 TLD A 1 H41 C145 H41 C145 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=1400nM P0C6X7 17981158 902 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 2z97 A 1.8 BS01 7HE A 1 T101 R112 L244 G248 T252 T349 F350 G351 H355 C357 G359 T92 R103 L235 G239 T243 T340 F341 G342 H346 C348 G350 R186 G248 D251 T252 V253 C357 L358 G359 E366 V396 R177 G239 D242 T243 V244 C348 L349 G350 E357 V387 1.14.15.1 0004497,0005506,0005515,0005737,0016705,0018683,0019383,0020037,0046872 remove_due_to_license_issue P00183 19133773 417 NLAPLPPHVPEHLVFDFDMYNPSNLSAGVQEAWAVLQESNVPDLVWTRCNGGHWIATRGQLIREAYEDYRHFSSECPFIPREAGEAYDFIPTSMDPPEQRQFRALANQVVGMPVVDKLENRIQELACSLIESLRPQGQCNFTEDYAEPFPIRIFMLLAGLPEEDIPHLKYLTDQMTRPDGSMTFAEAKEALYDYLIPIIEQRRQKPGTDAISIVANGQVNGRPITSDEAKRMCGLLLVGGLDTVVNFLSFSMEFLAKSPEHRQELIERPERIPAACEELLRRFSLVADGRILTSDYEFHGVQLKKGDQILLPQMLSGLDERENACPMHVDFSRQKVSHTTFGHGSHLCLGQHLARREIIVTLKEWLTRIPDFSIAPGAQIQHKSGIVSGVQALPLVWDPATTKAV 2za0 A 1.7 BS03 MGI A 1 H127 M158 E173 H124 M155 E170 Q34 E100 H127 E173 Q31 E97 H124 E170 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 Ki=0.23uM remove_due_to_license_issue Q9CPU0 18695250 300 PQPASSGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIATI 2za0 A 1.7 BS04 MGI A 2 Q34 F68 L70 F93 E100 Q31 F65 L67 F90 E97 Q34 E100 H127 E173 Q31 E97 H124 E170 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 Ki=0.23uM remove_due_to_license_issue Q9CPU0 18695250 400 PQPASSGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIATI 2za0 B 1.7 BS03 MGI A 1 Q34 M66 L70 E100 Q26 M58 L62 E92 Q34 E100 H127 E173 Q26 E92 H119 E165 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 remove_due_to_license_issue Q9CPU0 18695250 300 SGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIATII 2za0 B 1.7 BS04 MGI A 2 H127 E173 H119 E165 Q34 E100 H127 E173 Q26 E92 H119 E165 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 remove_due_to_license_issue Q9CPU0 18695250 400 SGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIATII 2za3 A 2.65 BS01 U5P A 1 D23 N104 D136 K138 T194 T195 P264 Q269 G293 R294 D23 N101 D133 K135 T191 T192 P261 Q266 G290 R291 4.1.1.23 0004590,0006207,0006221,0016831,0044205 remove_due_to_license_issue Q8T6J6 17981823 500 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNEEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILK 2za3 A 2.65 BS02 U5P B 1 D141 I142 D138 I139 4.1.1.23 0004590,0006207,0006221,0016831,0044205 remove_due_to_license_issue Q8T6J6 17981823 600 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNEEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILK 2za3 B 2.65 BS01 U5P B 1 D23 K102 N104 D136 T194 T195 P264 G293 R294 D23 K100 N102 D134 T192 T193 P262 G291 R292 4.1.1.23 0004590,0006207,0006221,0016831,0044205 remove_due_to_license_issue Q8T6J6 17981823 600 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIRKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILK 2za5 A 2.3 BS01 2FF A 1 Y177 D203 S204 C205 Q206 V227 W229 G230 E231 G232 R238 Y162 D188 S189 C190 Q191 V212 W214 G215 E216 G217 R223 H59 D106 Q206 G207 D208 S209 G210 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=3.7nM remove_due_to_license_issue P20231 18272363 4 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 2za5 C 2.3 BS01 2FF C 1 Y177 D203 S204 C205 Q206 W229 G230 E231 G232 R238 Y162 D188 S189 C190 Q191 W214 G215 E216 G217 R223 H59 D106 Q206 G207 D208 S209 G210 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=3.7nM remove_due_to_license_issue P20231 18272363 2 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 2zas A 2.0 BS01 1OH A 1 L268 E275 M306 L309 Y326 L345 I349 F435 L37 E44 M75 L78 Y95 L114 I118 F204 ? ic50=13.9nM remove_due_to_license_issue IC50=13.9nM P62508 18582436 460 KPYNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAKV 2zaz A 1.8 BS01 GK1 A 1 V30 A51 K53 T106 M109 D168 V27 A44 K46 T99 M102 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T178 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=0.4uM remove_due_to_license_issue Ki=400nM, IC50=2500nM Q16539 18006306 362 ERPTFYRQELNKTIWEVPERYQNLSPVGGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2zb0 A 2.1 BS01 GK3 A 1 V30 A51 E71 T106 L108 M109 D168 F169 L171 V27 A48 E68 T103 L105 M106 D165 F166 L168 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=0.24uM remove_due_to_license_issue Ki=240nM, IC50=1500nM Q16539 18006306 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2zb1 A 2.5 BS01 GK4 A 1 Y35 A51 K53 L75 T106 M109 A111 L167 D168 F169 Y30 A46 K48 L70 T101 M104 A106 L162 D163 F164 D150 K152 N155 D168 T185 D145 K147 N150 D163 T178 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=0.48uM remove_due_to_license_issue IC50=3000nM, Ki=480nM Q16539 18006306 361 ERPTFYRQELNKTIWEVPERYQNLSPVGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 2zbk B 3.56 BS01 RDC B 1 D76 G80 I81 V112 T170 V172 D63 G67 I68 V99 T157 V159 5.6.2.2 0003676,0003677,0003916,0003918,0005515,0005524,0006265,0006268,0009330,0034335,0042802 remove_due_to_license_issue O05207 18334211 531 EFFKRNPELAGFPNPARALYQTVRELIENSLDATDVHGILPNIKITIDLIDDARQIYKVNVVDNGIGIPPQEVPNAFGRVLYSSKYVNRQTRGMYGLGVKAAVLYSQMHQDKPIEIETSPVNSKRIYTFKLKIDINKNEPIIVERGSVENTRGFHGTSVAISIPGDWPKAKSRIYEYIKRTYIITPYAEFIFKDPEGNVTYYPRLTNKIPKPPQEVKPHPYGVDREEIKILINNLKRDYTIKEFLVNEFQSIGDTTADKILELAGLKPNKKVKNLTEEEITRLVETFKKDEDFRSPSADSLSVIGEDLIELGLKKIFNPDFAASITRKPKAYQGHPFIVEAGVAFGGSIPVGEEPIVLRYANKIPLIYDEKSDVIWKVVEELDWKRYGIESDQYQMVVMVHLCSTKIPYKSAGKESIAEVENIEKEIKNALMEVARKLKQYLSEKRKEQEAKKKLLAYLKYIPEVSRSLATFLASGNKELVSKYQNEISEGLFKLISKKLDLINIE 2zc9 H 1.58 BS03 22U H 1 Y60A W60D N98 A190 C191 V213 S214 W215 G216 F227 Y47 W50 N95 A193 C194 V218 S219 W220 G221 F232 3.4.21.5 0004252,0005509,0006508,0007596 Ki=180nM remove_due_to_license_issue Ki=250nM P00734 19520086 1501 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2zcq A 2.38 BS01 B65 A 1 F22 Y41 R45 D48 V133 V137 Q165 N168 F22 Y41 R45 D48 V133 V137 Q165 N168 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=1.5nM remove_due_to_license_issue A9JQL9 18276850 451 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 2zcr A 1.92 BS01 B69 A 1 H18 F22 V137 L141 A157 L160 G161 L164 Q165 N168 R171 F233 H18 F22 V134 L138 A154 L157 G158 L161 Q162 N165 R168 F230 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=135nM remove_due_to_license_issue A9JQL9 18276850 668 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 2zcs A 2.03 BS01 B70 A 1 H18 F22 F26 Y41 V137 G138 L145 A157 L160 G161 L164 Q165 N168 Y248 H18 F22 F26 Y41 V137 G138 L145 A157 L160 G161 L164 Q165 N168 Y248 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=6nM remove_due_to_license_issue A9JQL9 18276850 640 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 2zda H 1.73 BS03 32U H 1 Y60A L99 I174 D189 A190 V213 W215 G216 Y47 L96 I172 D192 A193 V218 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 19520086 1000 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2zdk A 1.67 BS02 50U A 1 H57 N97 T98 D189 S190 C191 Q192 V213 S214 W215 G216 G219 H40 N79 T80 D171 S172 C173 Q174 V191 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zdl A 1.8 BS02 45U A 1 H57 N97 T98 L99 D189 S190 C191 Q192 S214 W215 G216 G219 H40 N79 T80 L81 D171 S172 C173 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zdm A 1.93 BS02 46U A 1 H57 T98 L99 D189 S190 C191 Q192 W215 G216 G219 H40 T80 L81 D171 S172 C173 Q174 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zdn A 1.98 BS02 49U A 1 N97 T98 D189 S190 C191 Q192 S195 V213 S214 W215 G216 N79 T80 D171 S172 C173 Q174 S177 V191 S192 W193 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zdt A 2.0 BS01 46C A 1 K68 I70 G71 V78 A91 E147 M149 D150 A151 N152 S193 V196 L206 K24 I26 G27 V34 A47 E103 M105 D106 A107 N108 S149 V152 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 18313930 901 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPREHTIEEWKELIYKEVMN 2zdx A 2.54 BS01 P4A A 1 N258 A262 D293 V298 L306 F330 T358 N229 A233 D264 V269 L277 F282 T310 H250 E254 K257 N258 H221 E225 K228 N229 2.7.11.2 0004672,0004740,0005515,0005524,0005739,0005759,0006885,0008286,0009267,0010510,0010565,0010906,0016301,0042304,0042593,0042594,0045124,0046320,0071398,0072593,2000811 remove_due_to_license_issue Q16654 21904029 500 VPREVEHFSRYSPSPLSMKQLLDFGSENACERTSFAFLRQELPVRLANILKEIDILPTQLVNTSSVQLVKSWYIQSLMDLVEFHEKSPDDQKALSDFVDTLIKVRNRHHNVVPTMAQGIIEYNQNLQYFLDRFYMNRISTRMLMNQHILIFSDSQTGNPSHIGSIDPNCDVVAVVQDAFECSRMLCDQYYLSSPELKLTQVNGKFPDQPIHIVYVPSHLHHMLFELFKNAMRATVEHQENQPSLTPIEVIVVLGKEDLTIKISDRGGGVPLRIIDRLFSYTFGYGLPISRLYAKYFQGDLNLYSLSGYGTDAIIYLKALSSESIEKLPVFNKSAFKH 2zdz A 2.0 BS01 310 A 1 G73 Q74 G75 L92 D94 G96 Y133 W138 F170 I172 W177 I180 D290 G292 T294 G14 Q15 G16 L33 D35 G37 Y74 W79 F111 I113 W118 I121 D225 G227 T229 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D225 T228 3.4.23.46 0004190,0006508,0016020 ic50=0.7uM remove_due_to_license_issue IC50=700nM P56817 18162398 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLMEDCGY 2ze1 A 2.2 BS01 411 A 1 Q74 G75 D94 G96 S97 V131 Y133 W138 F170 W177 D290 G292 T293 T294 Q10 G11 D30 G32 S33 V67 Y69 W74 F106 W113 D217 G219 T220 T221 D94 S97 N99 A101 Y133 D290 T293 D30 S33 N35 A37 Y69 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=0.6uM remove_due_to_license_issue IC50=600nM P56817 18162398 1 FVEMVDNLRQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTEDCGY 2zfp H 2.25 BS03 19U H 1 H57 Y60A A190 S195 V213 S214 W215 G216 G226 F227 H43 Y47 A193 S198 V218 S219 W220 G221 G231 F232 3.4.21.5 0004252,0005509,0006508,0007596 Ki=6.8uM remove_due_to_license_issue Ki=13000nM P00734 19520086 801 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2zfs A 1.51 BS02 12U A 1 H57 N97 L99 Q175 D189 S190 C191 Q192 W215 G216 G219 H40 N79 L81 Q155 D171 S172 C173 Q174 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zft A 1.76 BS02 10U A 1 H57 N97 T98 L99 D189 S190 C191 Q192 S214 W215 G216 G219 H40 N79 T80 L81 D171 S172 C173 Q174 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zg1 A 2.7 BS01 SIA A 1 R124 K132 Y133 S134 R100 K108 Y109 S110 ? remove_due_to_license_issue O15389 18022638 241 VYELQVQKSVTVQEGLCVLVPCSFSYPWRSWYSSPPLYVYWFRDGEIPYYAEVVATNNPDRRVKPETQGRFRLLGDVQKKNCSLSIGDARMEDTGSYFFRVERGRDVKYSYQQNKLNLEVTALIEKPDIHEPLESGRPTRLSCSLPGSCEAGPPLTFSWTGNALSPLDPETTRSSELTLTPRPEDHGTNLTCQMKRQTTERTVQLNVS 2zg3 A 3.0 BS01 SIA B 1 R124 K132 Y133 S134 R100 K108 Y109 S110 ? remove_due_to_license_issue O15389 18022638 3 VYELQVQKSVTVQEGLCVLVPCSFSYPWRSWYSSPPLYVYWFRDGEIPYYAEVVATNNPDRRVKPETQGRFRLLGDVQKKNCSLSIGDARMEDTGSYFFRVERGRDVKYSYQQNKLNLEVTALIEKPDIHFLEPLESGRPTRLSCSLPGSCEAGPPLTFSWTGNALSPLDPETTRSSELTLTPRPEDHGTNLTCQMKRQTTERTVQLNVS 2zga A 1.65 BS01 YDP A 1 R8 D25 V82 R8 D25 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.48uM remove_due_to_license_issue P03367 21762812 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2zgx H 1.8 BS03 29U H 1 H57 Y60A W60D D189 A190 V213 W215 G216 H43 Y47 W50 D191 A192 V217 W219 G220 3.4.21.5 0004252,0005509,0006508,0007596 Ki=180nM remove_due_to_license_issue Ki=180nM, Kd=110nM P00734 19520086 1601 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2zhd A 1.94 BS02 12U A 1 H57 T98 L99 Q175 D189 S190 Q192 V213 S214 W215 G216 G219 H40 T80 L81 Q155 D171 S172 Q174 V191 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zi0 A 2.82 BS01 rna C 0 K21 Q25 R28 H29 N32 R33 R36 H38 S40 P41 S42 R46 K17 Q21 R24 H25 N28 R29 R32 H34 S36 P37 S38 R42 ? remove_due_to_license_issue Q8UYT3 18600235 1 ~ 20 EIPLHEIIRKLERMNQKKQAQRKRHKLNRKERGHKSPSEQRRSELWHARQVELSAINSDN 2zi0 A 2.82 BS02 rna D 0 R26 K30 K39 R46 W50 H51 R22 K26 K35 R42 W46 H47 ? remove_due_to_license_issue Q8UYT3 18600235 1 ~ 20 EIPLHEIIRKLERMNQKKQAQRKRHKLNRKERGHKSPSEQRRSELWHARQVELSAINSDN 2zi0 B 2.82 BS01 rna C 0 R26 K34 K39 R46 W50 H51 R23 K31 K36 R43 W47 H48 ? remove_due_to_license_issue Q8UYT3 18600235 1 ~ 20 IEIPLHEIIRKLERMNQKKQAQRKRHKLNRKERGHKSPSEQRRSELWHARQVELS 2zi0 B 2.82 BS02 rna D 0 R28 H29 N32 R33 R36 H38 S40 P41 S42 R46 R25 H26 N29 R30 R33 H35 S37 P38 S39 R43 ? remove_due_to_license_issue Q8UYT3 18600235 1 ~ 20 IEIPLHEIIRKLERMNQKKQAQRKRHKLNRKERGHKSPSEQRRSELWHARQVELS 2zif A 2.4 BS01 SAM A 1 D28 A29 S47 P49 F220 F243 A244 G245 T248 E264 L265 D8 A9 S27 P29 F169 F192 A193 G194 T197 E213 L214 S47 P48 V96 S27 P28 V70 2.1.1.-,2.1.1.113 0003677,0005737,0008168,0008170,0009007,0009307,0015667,0032259 Kd=43uM remove_due_to_license_issue Q5SL84 18618709 298 VHRLHVGDAREVLASFPEASVHLVVTSPPYWTLPGQLGHIEDYEAFLDELDRVWREVFRLLVPGGRLVIVVGDVAVARFGRHLVFPLHADIQVRCRKLGFDNLNPIIWHKHTNPYEPGAIIKTEIEYILMQRKPGGYRKPTQEQREKSRLPKEDFHRFFRQIWDDIPPFPLELAERLVRMFSFVGDVVLDPFAGTGTTLIAAARWGRRALGVELVPRYAQLAKERFAREVPGFSLEVLD 2zir B 2.4 BS03 NH7 B 1 Y93 L96 W102 W106 D297 C299 Y300 D359 Y361 H362 Y73 L76 W82 W86 D277 C279 Y280 D339 Y341 H342 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H228 R271 K274 D277 C279 Y280 D332 D339 H342 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=6.4nM remove_due_to_license_issue Q02293 19217288 903 EPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPG 2zis B 2.6 BS03 NH8 B 1 L96 W102 W106 R202 D297 C299 D359 Y361 H362 L75 W81 W85 R181 D276 C278 D338 Y340 H341 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H227 R270 K273 D276 C278 Y279 D331 D338 H341 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 19217288 903 PLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPG 2zjf A 2.4 BS01 BSU A 1 D104 W105 I137 Y164 V193 Y272 H333 W334 D101 W102 I134 Y161 V190 Y262 H323 W324 F36 D104 W105 I127 Y164 Y272 D302 H333 F33 D101 W102 I124 Y161 Y262 D292 H323 3.3.2.10 0003824,0004301,0009636,0016787,0042803 ic50=19nM remove_due_to_license_issue IC50=19nM P95276 18585390 360 VHRILNCRGTRIHAVADSPPDQQGPLVVLLHGFPESWYSWRHQIPALAGAGYRVVAIDQRGYGRSSKYRVQKAYRIKELVGDVVGVLDSYGAEQAFVVGHDWGAPVAWTFAWLHPDRCAGVVGISVPFAGRGVIGLPGSPFGERRPSDYHLELAGPGRVWYQDYFAVQDGIITEIEEDLRGWLLGLTYTVSGEGMMAATKAAVSMDPIDVIRAGPLCMAEGARLKDAFVYPETMPAWFTEADLDFYTGEFERSGFGGPLSFYHNIDNDWHDLADQQGKPLTPPALFIGGQYDVGTIWGAQAIERAHEVMPNYRGTHMIADVGHWIQQEAPEETNRLLLDFLGGLRP 2zju A 2.58 BS01 IM4 A 1 W143 Y185 Y192 W144 Y186 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=970nM P58154 18338186 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGR 2zju A 2.58 BS02 IM4 E 1 W53 A103 R104 L112 M114 W54 A104 R105 L113 M115 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=970nM P58154 18338186 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGR 2zju B 2.58 BS01 IM4 A 1 W53 A103 R104 L112 M114 W54 A104 R105 L113 M115 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=970nM P58154 18338186 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 2zju B 2.58 BS02 IM4 C 1 W143 Y185 Y192 W144 Y186 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=970nM P58154 18338186 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 2zjv A 2.7 BS01 CT4 A 1 W143 Y185 C187 Y192 W144 Y186 C188 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue P58154 18338186 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 2zjv A 2.7 BS02 CT4 E 1 W53 A103 R104 L112 M114 W54 A104 R105 L113 M115 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue P58154 18338186 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 2zjv B 2.7 BS01 CT4 A 1 R104 L112 M114 R104 L112 M114 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue P58154 18338186 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 2zjv B 2.7 BS02 CT4 B 1 W143 T144 Y185 C187 Y192 W143 T144 Y185 C187 Y192 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue P58154 18338186 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 2zjw A 2.4 BS01 REF A 1 L45 V53 V66 K68 F113 I174 D175 L45 V53 V66 K68 F113 I174 D175 D156 K158 N161 D175 P184 S194 D156 K158 N161 D175 P184 S194 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.02uM remove_due_to_license_issue Ki=20nM, IC50=40nM P68400 19414254 336 MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 2zkj A 2.0 BS01 ADP A 1 N258 R261 A262 V298 L306 S312 T313 A328 G331 L334 N229 R232 A233 V269 L277 S283 T284 A291 G294 L297 H250 E254 K257 N258 H221 E225 K228 N229 2.7.11.2 0004672,0004740,0005515,0005524,0005739,0005759,0006885,0008286,0009267,0010510,0010565,0010906,0016301,0042304,0042593,0042594,0045124,0046320,0071398,0072593,2000811 Kd=3.3uM remove_due_to_license_issue Q16654 18658136 501 VPREVEHFSRYSPSPLSMKQLLDFGSCERTSFAFLRQELPVRLANILKEIDILPTQLVNTSSVQLVKSWYIQSLMDLVEFHEKSPDDQKALSDFVDTLIKVRNRHHNVVPTMAQGIIEYKDACTVDPVTNQNLQYFLDRFYMNRISTRMLMNQHILIFSSHIGSIDPNCDVVAVVQDAFECSRMLCDQYYLSSPELKLTQVNGKFPDQPIHIVYVPSHLHHMLFELFKNAMRATVEHQENQPSLTPIEVIVVLGKEDLTIKISDRGGGVPLRIIDRLFSYTYSTAPTAPLAGFGYGLPISRLYAKYFQGDLNLYSLSGYGTDAIIYLKALSSESIEKLPVFNKSAFKHYQDDWCI 2zlg A 2.52 BS01 MRT A 1 Q692 K693 M721 S726 Y730 Q600 K601 M629 S634 Y638 C218 N426 C428 E430 C443 Y741 Y742 C143 N343 C345 E347 C360 Y649 Y650 1.17.4.1 0000166,0004748,0005515,0005524,0005634,0005737,0005971,0009263,0016491,0042802 remove_due_to_license_issue P21524 18610997 889 TLAARIAISNLHKQTTKQFSKVVEDLYRYVNAATGKPAPMISDDVYNIVMENKDKLNSAIVYDRDFQYSYFGFKTLERSYLLRINGQVAERPQHLIMRVALGIHGRDIEAALETYNLMSLKYFTHASPTLFNAGTPKPQMSSCFLVAMKEDSIEGIYDTLKECALISKTAGGIGLHIHNIRSTGSYIAGTNGTSNGLIPMIRVFNNTARYVGAFALYLEPWHADIFDFIDIRKNHGKEEIRARDLFPALWIPDLFMKRVEENGTWTLFSPTSAPGLSDCYGDEFEALYTRYEKEGRGKTIKAQKLWYSILEAQTETGTPFVVYKDACNRKSNQKNLGVIKSSNLCCEIVEYSAPDETAVCNLASVALPAFIETSEDGKTSTYNFKKLHEIAKVVTRNLNRVIDRNYYPVEEARKSNMRHRPIALGVQGLADTFMLLRLPFDSEEARLLNIQIFETIYHASMEASCELAQKDGPYETFQGSPASQGILQFDMWDQKPYGMWDWDTLRKDIMKHGVRNSLTMAPMPTASTSQILGYNECFEPVTSNMFQVVNPYLLRDLVDLGIWDEGMKQYLITQNGSIQGLPNVPQELKDLYKTVWEISQKTIINMAADRSVYIDQSHSLNLFLRAPTMGKLTSMHFYGWKKGLKTGMYYLRTQ 2zm1 A 2.1 BS01 KSF A 1 A271 K273 E288 M292 T316 M319 L371 A41 K43 E58 M62 T86 M89 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=220nM remove_due_to_license_issue IC50=220nM P06239 18977146 513 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 2zm3 A 2.5 BS01 575 A 1 L1005 Q1007 V1013 A1031 M1079 L1081 M1082 T1083 G1085 M1142 L26 Q28 V34 A52 M100 L102 M103 T104 G106 M160 D1135 R1139 N1140 D1153 E1162 D153 R157 N158 D171 E180 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd=0.614uM remove_due_to_license_issue IC50=2420nM P08069 18501599 1 SFSAADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPENPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEEN 2zmd A 2.88 BS01 537 A 1 I531 A551 I586 M602 E603 G605 L654 I16 A36 I71 M87 E88 G90 L139 N556 L565 D647 K649 N652 D664 A686 N41 L50 D132 K134 N137 D149 A162 2.7.12.1 0004672,0005524,0005975,0006468 remove_due_to_license_issue IC50=98nM P33981 18480048 900 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMDSQVGAVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 2zmj A 2.35 BS02 MI4 A 1 Y143 V230 S233 S271 S274 W282 C284 V296 A299 H301 H393 Y397 L410 F418 Y21 V50 S53 S91 S94 W102 C104 V116 A119 H121 H213 Y217 L230 F238 ? 0003677,0004879,0006355 ic50=30nM remove_due_to_license_issue P13053 18710208 1 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 2zmm A 2.1 BS01 35B A 1 Y46 D48 V49 K120 F182 S216 A217 I219 G220 R221 Q262 Y45 D47 V48 K119 F181 S215 A216 I218 G219 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=25nM remove_due_to_license_issue P18031 18798205 307 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2zn7 A 2.1 BS01 410 A 1 Y46 D48 K120 F182 S216 I219 R221 Q262 Y45 D47 K119 F181 S215 I218 R220 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=13nM remove_due_to_license_issue P18031 18798205 300 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 2zns A 2.0 BS01 GLU A 1 Y474 L502 T503 R508 G673 S674 T675 E723 Y60 L88 T89 R94 G139 S140 T141 E189 ? 0015276,0016020 remove_due_to_license_issue P39086 21893069 301 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGC 2znt A 1.6 BS01 DYH A 1 E426 Y474 P501 L502 T503 R508 V670 G673 S674 T675 S706 M722 E723 S726 E12 Y60 P87 L88 T89 R94 V136 G139 S140 T141 S172 M188 E189 S192 ? 0015276,0016020 Ki=0.5nM remove_due_to_license_issue Ki=0.740000nM P39086 21893069 1 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGC 2znu A 1.8 BS01 NDZ A 1 E426 Y474 T503 R508 V670 G673 S674 T675 S706 M722 E723 S726 E12 Y60 T89 R94 V136 G139 S140 T141 S172 M188 E189 S192 ? 0015276,0016020 Ki=7.7nM remove_due_to_license_issue P39086 21893069 1 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGC 2zo3 H 1.7 BS03 33U H 1 H57 Y60A W60D N98 L99 I174 D189 A190 V213 W215 G216 E217 H43 Y47 W50 N95 L96 I171 D191 A192 V217 W219 G220 E221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.1nM remove_due_to_license_issue Ki=0.036000nM P00734 19520086 2501 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 2zof A 2.3 BS03 BES A 1 D132 E166 E167 D195 R343 E414 G416 S417 H445 D136 E170 E171 D199 R347 E418 G420 S421 H449 3.4.13.18 0004180,0005654,0005737,0005829,0006508,0008233,0008237,0016787,0016805,0046872,0070573 ic50=7nM remove_due_to_license_issue Q9D1A2 18550540 1080 SPNSMSALKAVFQYIDENQDRYVKKLAEWVAIQSVSAWPEKRGEIRRMMEVAAADVQRLGGSVELVDIGKQKLPDGSEIPLPPILLGKLGSDPQKKTVCIYGHLDVQPAALEDGWDSEPFTLVEREGKLYGRGSTDDKGPVAGWMNALEAYQKTGQEIPVNLRFCLEGMEESGSEGLDELIFAQKDKFFKDVDYVCISDNYWLGKNKPCITYGLRGICYFFIEVECSDKDLHSGVYGGSVHEAMTDLISLMGCLVDKKGKILIPGINDAVAPVTDEEHALYDHIDFDMEEFAKDVGAETLLHSCKKDILMHRWRYPSLSLHGIEGAFSGSGAKTVIPRKVVGKFSIRLVPDMIPEVVSEQVSSYLSKKFAELQSPNKFKVYMGHGGKPWVSDFNHPHYQAGRRALKTVFGVEPDLTREGGSIPVTLTFQEATGKNVMLLPVGSADDGAHSQNEKLNRLNYIEGTKMLAAYLYEVSQLK 2zof A 2.3 BS04 BES B 1 H228 T330 H232 T334 3.4.13.18 0004180,0005654,0005737,0005829,0006508,0008233,0008237,0016787,0016805,0046872,0070573 ic50=7nM remove_due_to_license_issue Q9D1A2 18550540 1081 SPNSMSALKAVFQYIDENQDRYVKKLAEWVAIQSVSAWPEKRGEIRRMMEVAAADVQRLGGSVELVDIGKQKLPDGSEIPLPPILLGKLGSDPQKKTVCIYGHLDVQPAALEDGWDSEPFTLVEREGKLYGRGSTDDKGPVAGWMNALEAYQKTGQEIPVNLRFCLEGMEESGSEGLDELIFAQKDKFFKDVDYVCISDNYWLGKNKPCITYGLRGICYFFIEVECSDKDLHSGVYGGSVHEAMTDLISLMGCLVDKKGKILIPGINDAVAPVTDEEHALYDHIDFDMEEFAKDVGAETLLHSCKKDILMHRWRYPSLSLHGIEGAFSGSGAKTVIPRKVVGKFSIRLVPDMIPEVVSEQVSSYLSKKFAELQSPNKFKVYMGHGGKPWVSDFNHPHYQAGRRALKTVFGVEPDLTREGGSIPVTLTFQEATGKNVMLLPVGSADDGAHSQNEKLNRLNYIEGTKMLAAYLYEVSQLK 2zof B 2.3 BS01 BES A 1 H228 T330 H232 T334 3.4.13.18 0004180,0005654,0005737,0005829,0006508,0008233,0008237,0016787,0016805,0046872,0070573 ic50=7nM remove_due_to_license_issue Q9D1A2 18550540 1080 SPNSMSALKAVFQYIDENQDRYVKKLAEWVAIQSVSAWPEKRGEIRRMMEVAAADVQRLGGSVELVDIGKQKLPDGSEIPLPPILLGKLGSDPQKKTVCIYGHLDVQPAALEDGWDSEPFTLVEREGKLYGRGSTDDKGPVAGWMNALEAYQKTGQEIPVNLRFCLEGMEESGSEGLDELIFAQKDKFFKDVDYVCISDNYWLGKNKPCITYGLRGICYFFIEVECSDKDLHSGVYGGSVHEAMTDLISLMGCLVDKKGKILIPGINDAVAPVTDEEHALYDHIDFDMEEFAKDVGAETLLHSCKKDILMHRWRYPSLSLHGIEGAFSGSGAKTVIPRKVVGKFSIRLVPDMIPEVVSEQVSSYLSKKFAELQSPNKFKVYMGHGGKPWVSDFNHPHYQAGRRALKTVFGVEPDLTREGGSIPVTLTFQEATGKNVMLLPVGSADDGAHSQNEKLNRLNYIEGTKMLAAYLYEVSQLK 2zof B 2.3 BS04 BES B 1 D132 E166 E167 D195 R343 E414 G416 S417 H445 D136 E170 E171 D199 R347 E418 G420 S421 H449 3.4.13.18 0004180,0005654,0005737,0005829,0006508,0008233,0008237,0016787,0016805,0046872,0070573 ic50=7nM remove_due_to_license_issue Q9D1A2 18550540 1081 SPNSMSALKAVFQYIDENQDRYVKKLAEWVAIQSVSAWPEKRGEIRRMMEVAAADVQRLGGSVELVDIGKQKLPDGSEIPLPPILLGKLGSDPQKKTVCIYGHLDVQPAALEDGWDSEPFTLVEREGKLYGRGSTDDKGPVAGWMNALEAYQKTGQEIPVNLRFCLEGMEESGSEGLDELIFAQKDKFFKDVDYVCISDNYWLGKNKPCITYGLRGICYFFIEVECSDKDLHSGVYGGSVHEAMTDLISLMGCLVDKKGKILIPGINDAVAPVTDEEHALYDHIDFDMEEFAKDVGAETLLHSCKKDILMHRWRYPSLSLHGIEGAFSGSGAKTVIPRKVVGKFSIRLVPDMIPEVVSEQVSSYLSKKFAELQSPNKFKVYMGHGGKPWVSDFNHPHYQAGRRALKTVFGVEPDLTREGGSIPVTLTFQEATGKNVMLLPVGSADDGAHSQNEKLNRLNYIEGTKMLAAYLYEVSQLK 2zoq A 2.39 BS01 5ID A 1 I48 E50 V56 A69 Q122 M125 S170 L173 I25 E27 V33 A46 Q99 M102 S147 L150 D166 K168 S170 N171 D184 T207 D143 K145 S147 N148 D161 T184 2.7.11.24 0000165,0001784,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005635,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005829,0005856,0005886,0005901,0005925,0006351,0006468,0006915,0006974,0007254,0008286,0009887,0010759,0014032,0014044,0016020,0016310,0019233,0019902,0030278,0030509,0030641,0030878,0031143,0031281,0031663,0032206,0032496,0032872,0033554,0034198,0035556,0038083,0038133,0042473,0042552,0042770,0042802,0043330,0045944,0048009,0048538,0050804,0051216,0051403,0051493,0060020,0060324,0060425,0060440,0061308,0070161,0070371,0070374,0070498,0070849,0071260,0071356,0072584,0090170,0098792,0098978,0106310,0120041,0140297,1904262,1904417,2000641 ic50=0.9uM remove_due_to_license_issue P27361 18983981 382 VPGEVEMVKGQPFDVGPRYTQLQYIGEGAYGMVSSAYDHVRKTRVAIKKISPFEHQTYCQRTLREIQILLRFRHENVIGIRDILRASTLEAMRDVYIVQDLMETDLYKLLKSQQLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLINTTCDLKICDFGLARIADPEHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINMKARNYLQSLPSKTKVAWAKLFPKSDSKALDLLDRMLTFNPNKRITVEEALAHPYLEQYYDPTDEPVAEEPFTFAMELDDLPKERLKELIFQETARFQPGV 2zp0 H 2.7 BS02 PI0 H 1 H57 D60 G97 T98 P170I D189 S190 C191 K192 S195 V213 S214 W215 G216 G219 H41 D44 G85 T86 P169 D186 S187 C188 K189 S192 V210 S211 W212 G213 G215 3.4.21.21 0004252,0006508 remove_due_to_license_issue P08709 1001 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 2zq1 A 1.68 BS02 11U A 1 H57 N97 T98 L99 D189 S190 C191 S214 W215 G216 G219 H40 N79 T80 L81 D171 S172 C173 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zq2 A 1.4 BS02 13U A 1 T98 L99 D189 S190 C191 Q192 V213 W215 G216 G219 T80 L81 D171 S172 C173 Q174 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=276nM remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 2zsc A 1.3 BS01 BTN A 1 S18 Y34 S36 V38 W69 S76 T78 W96 D116 S17 Y33 S35 V37 W68 S75 T77 W95 D115 ? 0005576,0009374 remove_due_to_license_issue B9A0T7 19187241 301 SDVQSSLTGTWYNELNSKMELTANKDGTLTGKYLSKVGDVYVPYPLSGRYNLQPPAGQGVALGWAVSWENSKIHSATTWSGQFFSESSPVILTQWLLSSSTARGDVWESTLVGNDSFTKTAPT 2zsc B 1.3 BS01 BTN B 1 S18 Y34 S36 V38 W69 S76 T78 W96 D116 S17 Y33 S35 V37 W68 S75 T77 W95 D115 ? 0005576,0009374 remove_due_to_license_issue B9A0T7 19187241 301 SDVQSSLTGTWYNELNSKMELTANKDGTLTGKYLSKVGDVYVPYPLSGRYNLQPPAGQGVALGWAVSWENSKIHSATTWSGQFFSESSPVILTQWLLSSSTARGDVWESTLVGNDSFTKTAPT 2zu3 A 1.75 BS01 ZU3 A 1 H40 E71 L127 G128 T142 A144 G145 C147 H161 V162 G163 G164 N165 H40 E71 L127 G128 T142 A144 G145 C147 H161 V162 G163 G164 N165 H40 E71 G145 C147 H40 E71 G145 C147 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue P03313 19144641 501 GPAFEFAVAMMKRNSSTVKTEYGEFTMLGIYDRWAVLPRHAKPGPTILMNDQEVGVLDAKELVDKDGTNLELTLLKLNRNEKFRDIRGFLAKEEVEVNEAVLAINTSKFPNMYIPVGQVTEYGFLNLGGTPTKRMLMYNFPTRAGQCGGVLMSTGKVLGIHVGGNGHQGFSAALLKHYFN 2zu4 A 1.93 BS01 ZU3 A 1 L27 H41 F140 N142 G143 C145 H163 H164 M165 E166 P168 Q189 T190 A191 Q192 L27 H41 F140 N142 G143 C145 H163 H164 M165 E166 P168 Q189 T190 A191 Q192 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=38nM P0C6X7 19144641 501 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 2zu5 A 1.65 BS01 ZU5 A 1 L27 H41 M49 F140 G143 C145 H163 H164 M165 E166 P168 D187 Q189 T190 A191 Q192 L27 H41 M49 F140 G143 C145 H163 H164 M165 E166 P168 D187 Q189 T190 A191 Q192 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue Ki=99nM P0C6X7 19144641 2001 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 2zv2 A 2.4 BS01 609 A 1 I172 V180 A193 K195 F268 V271 G274 L320 D331 I12 V18 A31 K33 F75 V78 G81 L127 D138 D313 K315 N318 D331 T351 D120 K122 N125 D138 T158 2.7.11.17 0004672,0005524,0006468 remove_due_to_license_issue IC50=5.0e+2nM Q96RR4 21504895 501 VQLNQYTLKDEIGKYGVVKLAYNENDNTYYAMKVLSKKEQVYQEIAILKKLDHPNVVKLVEVLDDPNEDHLYMVFELVNQGPVMEVPTLKPLSEDQARFYFQDLIKGIEYLHYQKIIHRDIKPSNLLVGEDGHIKIADFGVSNEFKGSDALLSNTVGTPAFMAPESLSETRKIFSGKALDVWAMGVTLYCFVFGQCPFMDERIMCLHSKIKSQALEFPDQPDIAEDLKDLITRMLDKNPESRIVVPEIKLHPWVTR 2zv9 A 2.76 BS01 PP2 A 1 V261 A273 E290 M294 T319 M322 L374 V24 A36 E53 M57 T82 M85 L137 D367 R369 A371 N372 D385 F405 D130 R132 A134 N135 D148 F160 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P25911 18984583 513 PAWEIPRESIKLVKKLGAGQFGEVWMGYYNNSTKVAVKTLKPGTMSVQAFLEEANLMKTLQHDKLVRLYAVVTKEEPIYIITEFMAKGSLLDFLKSDEGGKVLLPKLIDFSAQIAEGMAYIERKNYIHRDLRAANVLVSESLMCKIADFGLARVIEGAKFPIKWTAPEAINFGCFTIKSNVWSFGILLYEIVTYGKIPYPGRTNADVMSALSQGYRMPRMENCPDELYDIMKMCWKEKAEERPTFDYLQSVLDDFY 2zva A 2.6 BS01 1N1 A 1 L253 A273 K275 E290 M294 V303 I317 T319 M322 A323 G325 L374 A384 L16 A36 K38 E53 M57 V66 I80 T82 M85 A86 G88 L137 A147 D367 R369 A371 N372 D385 F405 D130 R132 A134 N135 D148 F164 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P25911 18984583 513 PAWEIPRESIKLVKKLGAGQFGEVWMGYYNNSTKVAVKTLKPGTMSVQAFLEEANLMKTLQHDKLVRLYAVVTKEEPIYIITEFMAKGSLLDFLKSDEGGKVLLPKLIDFSAQIAEGMAYIERKNYIHRDLRAANVLVSESLMCKIADFGLARVIETAREGAKFPIKWTAPEAINFGCFTIKSNVWSFGILLYEIVTYGKIPYPGRTNADVMSALSQGYRMPRMENCPDELYDIMKMCWKEKAEERPTFDYLQSVLDDFYT 2zvj A 2.3 BS03 KOM A 1 W38 M40 D141 W143 K144 N170 P174 E199 W36 M38 D139 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 19056347 302 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQG 2zwz A 2.36 BS01 ZWZ A 1 H34 Y64 E66 W67 H128 H129 D224 R254 E266 F290 H28 Y58 E60 W61 H122 H123 D218 R248 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=16.3nM remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAV 2zx5 A 2.65 BS01 ZX5 A 1 H34 F59 E66 W67 H128 H129 Y171 D224 M225 R254 E266 F290 H28 F53 E60 W61 H122 H123 Y165 D218 M219 R248 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAV 2zx6 A 2.42 BS01 ZX6 A 1 H34 Y64 E66 W67 H128 H129 D224 M225 R254 E266 F290 H28 Y58 E60 W61 H122 H123 D218 M219 R248 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=0.475nM remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAVE 2zx6 B 2.42 BS01 ZX6 B 1 H34 Y64 E66 W67 H128 H129 D224 M225 R254 E266 F290 H28 Y58 E60 W61 H122 H123 D218 M219 R248 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=0.475nM remove_due_to_license_issue Q9WYE2 19967696 902 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAVE 2zx7 A 2.48 BS01 ZX7 A 1 H34 Y64 E66 W67 H128 H129 D224 M225 R254 E266 V269 N270 F290 H28 Y58 E60 W61 H122 H123 D218 M219 R248 E260 V263 N264 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=0.427nM remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAVE 2zx8 A 2.33 BS01 ZX8 A 1 H34 Y64 E66 W67 H128 H129 D224 M225 R254 T264 E266 V269 N270 F290 H28 Y58 E60 W61 H122 H123 D218 M219 R248 T258 E260 V263 N264 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=0.441nM remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAV 2zx9 A 2.62 BS01 ZX9 A 1 H34 L50 E66 W67 H128 H129 D224 R254 E266 F290 H28 L44 E60 W61 H122 H123 D218 R248 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAVE 2zxa A 2.57 BS01 ZXA A 1 H34 E66 W67 H128 H129 D224 M225 R254 E266 F290 H28 E60 W61 H122 H123 D218 M219 R248 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAVE 2zxb A 2.61 BS01 ZXB A 1 H34 Y64 E66 H128 E266 H28 Y58 E60 H122 E260 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAVE 2zxd A 2.15 BS01 ZXD A 1 F32 H34 E66 W67 H128 H129 Y171 D224 E266 F290 F26 H28 E60 W61 H122 H123 Y165 D218 E260 F284 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=6uM remove_due_to_license_issue Q9WYE2 19967696 901 RYKPDWESLREHTVPKWFDKAKFGIFIHWGIYSVPGWATPTGELGKVPMDAWFFQNPYAEWYENSLRIKESPTWEYHVKTYGENFEYEKFADLFTAEKWDPQEWADLFKKAGAKYVIPTTKHHDGFCLWGTKYTDFNSVKRGPKRDLVGDLAKAVREAGLRFGVYYSGGLDWRFTTEPIRYPEDLSYIRPNTYEYADYAYKQVMELVDLYLPDVLWNDMGWPEKGKEDLKYLFAYYYNKHPEGSVNDRWGVPHWDFKTAEYHVNYPGDLPGYKWEFTRGIGLSFGYNRNEGPEHMLSVEQLVYTLVDVVSKGGNLLLNVGPKGDGTIPDLQKERLLGLGEWLRKYGDAIYGTSVWERCCAKTEDGTEIRFTRKCNRIFVIFLGIPTGEKIVIEDLNLSAGTVRHFLTGERLSFKNVGKNLEITVPKKLLETDSITLVLEAV 2zxg A 1.55 BS02 S23 A 1 E121 M260 G261 A262 M263 E264 V294 H297 E298 E320 Y376 Y381 R825 E117 M256 G257 A258 M259 E260 V290 H293 E294 E316 Y372 Y377 R821 E264 H297 E298 H301 E320 N373 Y381 E260 H293 E294 H297 E316 N369 Y377 3.4.11.2 0004177,0005515,0005886,0006508,0008237,0008270,0042802,0046872 Ki=0.00000079M remove_due_to_license_issue P04825 19622865 901 PQAKYRHDYRAPDYQITDIDLTFDLDAQKTVVTAVSQAVRHGASDAPLRLNGEDLKLVSVHINDEPWTAWKEEEGALVISNLPERFTLKIINEISPAANTALEGLYQSGDALCTQCEAEGFRHITYYLDRPDVLARFTTKIIADKIKYPFLLSNGNRVAQGELENGRHWVQWQDPFPKPCYLFALVAGDFDVLRDTFTTRSGREVALELYVDRGNLDRAPWAMTSLKNSMKWDEERFGLEYDLDIYMIVAVDFFNMGAMENKGLNIFNSKYVLARTDTATDKDYLDIERVIGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSSDLGSRAVNRINNVRTMRGLQFAEDASPMAHPIRPDMVIEMNNFYTLTVYEKGAEVIRMIHTLLGEENFQKGMQLYFERHDGSAATCDDFVQAMEDASNVDLSHFRRWYSQSGTPIVTVKDDYNPETEQYTLTISQRTPATPDQAEKQPLHIPFAIELYDNEGKVIPLQKGGHPVNSVLNVTQAEQTFVFDNVYFQPVPALLCEFSAPVKLEYKWSDQQLTFLMRHARNDFSRWDAAQSLLATYIKLNVARHQQGQPLSLPVHVADAFRAVLLDEKIDPALAAEILTLPSVNEMAELFDIIDPIAIAEVREALTRTLATELADELLAIYNANYQSEYRVEHEDIAKRTLRNACLRFLAFGETHLADVLVSKQFHEANNMTDALAALSAAVAAQLPCRDALMQEYDDKWHQNGLVMDKWFILQATSPAANVLETVRGLLQHRSFTMSNPNRIRSLIGAFAGSNPAAFHAEDGSGYLFLVEMLTDLNSRNPQVASRLIEPLIRLKRYDAKRQEKMRAALEQLKGLENLSGDLYEKITKALA 2zy1 A 1.78 BS01 830 A 1 F22 R45 D48 V137 L160 G161 L164 Q165 F22 R45 D48 V132 L155 G156 L159 Q160 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=0.04uM remove_due_to_license_issue A9JQL9 19456099 808 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 2zyb A 2.55 BS01 KSL A 1 A271 T316 L371 A41 T86 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=20nM P06239 18977146 511 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 2zz2 A 1.53 BS01 6CN A 1 D20 K42 D70 M126 S127 P180 Q185 G202 R203 D10 K32 D60 M116 S117 P170 Q175 G192 R193 K42 D70 A72 D75 K32 D60 A62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=29000nM O26232 19236876 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFAVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz2 A 1.53 BS02 6CN B 1 D75 I76 T79 D65 I66 T69 K42 D70 A72 D75 K32 D60 A62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=29000nM O26232 19236876 302 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFAVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz2 B 1.53 BS01 6CN A 1 D75 I76 T79 D65 I66 T69 K42 D70 A72 D75 K32 D60 A62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=29000nM O26232 19236876 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFAVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz2 B 1.53 BS02 6CN B 1 D20 K42 D70 M126 S127 P180 Q185 G202 R203 D10 K32 D60 M116 S117 P170 Q175 G192 R193 K42 D70 A72 D75 K32 D60 A62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=29000nM O26232 19236876 302 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFAVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz6 A 1.66 BS01 6AZ A 1 D20 K72 M126 S127 P180 Q185 G202 R203 D10 K62 M116 S117 P170 Q175 G192 R193 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=190nM O26232 19236876 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz6 A 1.66 BS02 6AZ B 1 D75 I76 T79 D65 I66 T69 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=190nM O26232 19236876 302 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz6 B 1.66 BS01 6AZ A 1 D75 I76 T79 D65 I66 T69 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=190nM O26232 19236876 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zz6 B 1.66 BS02 6AZ B 1 D20 K72 M126 S127 P180 Q185 G202 R203 D10 K62 M116 S117 P170 Q175 G192 R193 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=190nM O26232 19236876 302 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 2zzu H 2.5 BS01 359 H 1 H57 D60 G97 T98 T99 S170H P170I D189 S190 C191 K192 S195 S214 W215 G216 Q217 G219 H41 D44 G85 T86 T87 S168 P169 D186 S187 C188 K189 S192 S211 W212 G213 Q214 G215 3.4.21.21 0004252,0006508 ic50=39nM remove_due_to_license_issue P08709 20045964 1 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 3a1c A 1.85 BS01 ACP A 1 D424 T426 E457 H462 I464 G490 E491 G492 N502 V532 T572 G573 D574 K600 D25 T27 E58 H63 I65 G91 E92 G93 N103 V133 T173 G174 D175 K201 D424 D618 D622 D25 D219 D223 7.2.2.8 0000166,0005215,0005524,0016020,0016887 Kd~0.1mM remove_due_to_license_issue O29777 19478797 997 AELGILIKNADALEVAEKVTAVIFDKTGTLTKGKPEVTDLVPLNGDERELLRLAAIAERRSEHPIAEAIVKKALEHGIELGEPEKVEVIAGEGVVADGILVGNKRLMEDFGVAVSNEVELALEKLEREAKTAVIVARNGRVEGIIAVSDTLKESAKPAVQELKRMGIKVGMITGDNWRSAEAISRELNLDLVIAEVLPHQKSEEVKKLQAKEVVAFVGDGINDAPALAQADLGIAVGSGSDVAVESGDIVLIRDDLRDVVAAIQLSR 3a1d A 1.85 BS01 ADP A 1 E457 H462 I464 E491 G492 N502 G573 D574 K600 E58 H63 I65 E92 G93 N103 G174 D175 K201 D424 D618 D622 D25 D219 D223 7.2.2.8 0000166,0005215,0005524,0016020,0016887 remove_due_to_license_issue O29777 19478797 997 AELGILIKNADALEVAEKVTAVIFDKTGTLTKGKPEVTDLVPLNGDERELLRLAAIAERRSEHPIAEAIVKKALEHGIELGEPEKVEVIAGEGVVADGILVGNKRLMEDFGVAVSNEVELALEKLEREAKTAVIVARNGRVEGIIAVSDTLKESAKPAVQELKRMGIKVGMITGDNWRSAEAISRELNLDLVIAEVLPHQKSEEVKKLQAKEVVAFVGDGINDAPALAQADLGIAVGSGSDVAVESGDIVLIRDDLRDVVAAIQLSRK 3a1e A 1.95 BS01 ACP A 1 D424 T426 E457 Q462 I464 E491 G492 N502 V532 T572 G573 D574 K600 D25 T27 E58 Q63 I65 E92 G93 N103 V133 T173 G174 D175 K201 D424 D618 D622 D25 D219 D223 7.2.2.8 0000166,0005215,0005524,0016020,0016887 Kd~2.2mM remove_due_to_license_issue O29777 19478797 997 AELGILIKNADALEVAEKVTAVIFDKTGTLTKGKPEVTDLVPLNGDERELLRLAAIAERRSEQPIAEAIVKKALEHGIELGEPEKVEVIAGEGVVADGILVGNKRLMEDFGVAVSNEVELALEKLEREAKTAVIVARNGRVEGIIAVSDTLKESAKPAVQELKRMGIKVGMITGDNWRSAEAISRELNLDLVIAEVLPHQKSEEVKKLQAKEVVAFVGDGINDAPALAQADLGIAVGSGSDVAVESGDIVLIRDDLRDVVAAIQLSRK 3a1s A 1.5 BS01 GDP A 1 N26 G28 K29 T30 S31 A130 D132 S158 S159 V160 N13 G15 K16 T17 S18 A117 D119 S145 S146 V147 ? 0005525 Kd=14.8uM remove_due_to_license_issue Q9WXQ8 19733088 1 LHMVKVALAGCPNVGKTSLFNALTGTKQYVANWPGVTVEKKEGVFTYKGYTINLIDLPGTYSLGYSSIDEKIARDYLLKGDADLVILVADSVNPEQSLYLLLEILEMEKKVILAMTAIDEAKKTGMKIDRYELQKHLGIPVVFTSSVTGEGLEELKEKIVEYAQKNTILHRMILDYGEKVESEIKKVENFLRDKKLRINPRYFALKYLSGDPEFYSEGVKLGLPELSEEERIGYRLLIAKRKREYVENVVKEAFA 3a1t A 1.8 BS01 GDP A 1 N26 G28 K29 T30 S31 A130 D132 S158 V160 N12 G14 K15 T16 S17 A116 D118 S144 V146 ? 0005525 Kd=14.8uM remove_due_to_license_issue Q9WXQ8 19733088 1 HMVKVALAGCPNVGKTSLFNALTGTKQYVANWPGVTVEKKEGVFTYKGYTINLIDLPGTYSLGYSSIDEKIARDYLLKGDADLVILVADSVNPEQSLYLLLEILEMEKKVILAMTAIDEAKKTGMKIDRYELQKHLGIPVVFTSSVTGEGLEELKEKIVEYAQKNTILHRMILDYGEKVESEIKKVENFLRDKKLRINPRYFALKYLSGDPEFYSEGVKLGLPELSEEERIGYRLLIAKRKREYVENVVKEAFA 3a29 A 2.6 BS01 2T0 A 1 V17 G21 A24 G26 T27 G28 E29 L30 T31 K112 Y113 R140 M177 V9 G13 A16 G18 T19 G20 E21 L22 T23 K96 Y97 R124 M161 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=13nM P09467 19762234 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3a29 C 2.6 BS01 2T0 C 1 V17 G21 A24 T27 G28 L30 T31 K112 Y113 M177 V9 G13 A16 T19 G20 L22 T23 K95 Y96 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=13nM P09467 19762234 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3a2c A 2.9 BS01 PDY A 1 V78 Q80 C140 L141 E190 N191 L193 D207 V32 Q34 C94 L95 E144 N145 L147 D161 D186 K188 E190 N191 D207 S216 D140 K142 E144 N145 D161 S170 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=130nM P49137 20057052 1 HVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSVAPEVLYDKSCDMWSLGVIMYILLCGYPPFYSPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKE 3a2c A 2.9 BS02 PDY A 2 Y260 P261 Y264 Y197 P198 Y201 D186 K188 E190 N191 D207 S216 D140 K142 E144 N145 D161 S170 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=130nM P49137 20057052 2 HVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSVAPEVLYDKSCDMWSLGVIMYILLCGYPPFYSPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKE 3a2o A 0.88 BS01 KNJ B 1 D25 G27 A28 G48 I50 V82 I84 D25 G27 A28 G48 I50 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 19954246 999 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3a2o B 0.88 BS01 KNJ B 1 D125 G127 A128 D129 D130 I147 G149 I150 I184 D25 G27 A28 D29 D30 I47 G49 I50 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.83nM remove_due_to_license_issue P03367 19954246 999 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3a3y A 2.8 BS06 OBN A 1 F323 G326 I327 I328 V329 A330 F790 T804 F292 G295 I296 I297 V298 A299 F759 T773 D376 D717 D721 D345 D686 D690 ? 0000166,0005215,0005391,0005524,0005886,0006813,0006814,0006883,0008556,0010248,0016020,0016887,0030007,0036376,0046872,1902600,1990573 remove_due_to_license_issue Q4H132 19666591 6000 LDELKKEVSMDDHKLSLDELHNKYGTDLTRGLTNARAKEILARDGPNSLTPPPTTPEWIKFCRQLFGGFSILLWIGAILCFLAYGIQAATEDEPANDNLYLGVVLSTVVIVTGCFSYYQEAKSSRIMDSFKNMVPQQALVIRDGEKSTINAEFVVAGDLVEVKGGDRIPADLRIISAHGCKVDNSSLTGESEPQTRSPEFSSENPLETRNIAFFSTNCVEGTARGVVVYTGDRTVMGRIATLASGLEVGRTPIAIEIEHFIHIITGVAVFLGVSFFILSLILGYSWLEAVIFLIGIIVANVPEGLLATVTVCLTLTAKRMARKNCLVKNLEAVETLGSTSTICSDKTGTLTQNRMTVAHMWFDNQIHEADTTENQSGAAFDKTSATWSALSRIAALCNRAVFQAGQDNVPILKRSVAGDASESALLKCIELCCGSVQGMRDRNPKIVEIPFNSTNKYQLSIHENEKSSESRYLLVMKGAPERILDRCSTILLNGAEEPLKEDMKEAFQNAYLELGGLGERVLGFCHFALPEDKYNEGYPFDADEPNFPTTDLCFVGLMAMIDPPRAAVPDAVGKCRSAGIKVIMVTGDHPITAKAIAKGVGIISEGNETIEDIAARLNIPIGQVNPRDAKACVVHGSDLKDLSTEVLDDILHYHTEIVFARTSPQQKLIIVEGCQRQGAIVAVTGDGVNDSPALKKADIGVAMGISGSDVSKQAADMILLDDNFASIVTGVEEGRLIFDNLKKSIAYTLTSNIPEITPFLVFIIGNVPLPLGTVTILCIDLGTDMVPAISLAYEQAESDIMKRQPRNPKTDKLVNERLISMAYGQIGMIQALGGFFSYFVILAENGFLPMDLIGKRVRWDDRWISDVEDSFGQQWTYEQRKIVEFTCHTSFFISIVVVQWADLIICKTRRNSIFQQGMKNKILIFGLFEETALAAFLSYCPGTDVALRMYPLKPSWWFCAFPYSLIIFLYDEMRRFIIRRSPGGWVEQETYY 3a46 A 2.2 BS01 dna C 0 Y95 M113 R114 F116 S272 G273 K274 N275 Y94 M112 R113 F115 S271 G272 K273 N274 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0140078 remove_due_to_license_issue Q5UQ00 19625256 1 ~ 13 PEGPEVALTADILEKYFKGKTLEYIDFISGRYSKSEPEGYDDFIANLPLKVSNVDTKGKFLWFELFDPNDKSNKWYIWNTFGLTGMWSLFEAKYTRAVLSFDNELMAYFSDMRNFGTFKFSNSEKELKRKLNELGPDFLKNDDIDISKIKKYKQPIVALLMDQKKIGSGLGNYLVAEILYRAKIDPHKLGSNLTDQEIENLWYWIKYETKLAYDSNHIGYMVNLENESSKIGRKNYHPNIHPTEKEFDFLVYRKKKDPNGNKVIADKIIGSGKNKRTTYWAPAIQKLE 3a46 A 2.2 BS02 dna D 0 E3 K60 G83 L84 R114 F116 G172 N173 Y221 Y253 R254 N275 R277 T278 Y280 E2 K59 G82 L83 R113 F115 G171 N172 Y220 Y252 R253 N274 R276 T277 Y279 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0140078 remove_due_to_license_issue Q5UQ00 19625256 14 ~ 26 PEGPEVALTADILEKYFKGKTLEYIDFISGRYSKSEPEGYDDFIANLPLKVSNVDTKGKFLWFELFDPNDKSNKWYIWNTFGLTGMWSLFEAKYTRAVLSFDNELMAYFSDMRNFGTFKFSNSEKELKRKLNELGPDFLKNDDIDISKIKKYKQPIVALLMDQKKIGSGLGNYLVAEILYRAKIDPHKLGSNLTDQEIENLWYWIKYETKLAYDSNHIGYMVNLENESSKIGRKNYHPNIHPTEKEFDFLVYRKKKDPNGNKVIADKIIGSGKNKRTTYWAPAIQKLE 3a46 B 2.2 BS01 dna E 0 Y95 M113 R114 N115 F116 S272 G273 K274 N275 Y94 M112 R113 N114 F115 S271 G272 K273 N274 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0140078 remove_due_to_license_issue Q5UQ00 19625256 1 ~ 13 PEGPEVALTADILEKYFKGKTLEYIDFISGRYSKSEPEGYDDFIANLPLKVSNVDTKGKFLWFELFDPNDKSNKWYIWNTFGLTGMWSLFEAKYTRAVLSFDNELMAYFSDMRNFGTFKFSNSEKELKRKLNELGPDFLKNDDIDISKIKKYKQPIVALLMDQKKIGSGLGNYLVAEILYRAKIDPHKLGSNLTDQEIENLWYWIKYETKLAYDSNHIGYMVNLENESSKIGRKNYHPNIHPTEKEFDFLVYRKKKDPNGNKVIADKIIGSGKNKRTTYWAPAIQKLE 3a46 B 2.2 BS02 dna F 0 P2 E3 K60 G83 L84 R114 F116 G172 N173 Y221 Y253 R254 K268 N275 R277 T278 Y280 P1 E2 K59 G82 L83 R113 F115 G171 N172 Y220 Y252 R253 K267 N274 R276 T277 Y279 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0140078 remove_due_to_license_issue Q5UQ00 19625256 14 ~ 26 PEGPEVALTADILEKYFKGKTLEYIDFISGRYSKSEPEGYDDFIANLPLKVSNVDTKGKFLWFELFDPNDKSNKWYIWNTFGLTGMWSLFEAKYTRAVLSFDNELMAYFSDMRNFGTFKFSNSEKELKRKLNELGPDFLKNDDIDISKIKKYKQPIVALLMDQKKIGSGLGNYLVAEILYRAKIDPHKLGSNLTDQEIENLWYWIKYETKLAYDSNHIGYMVNLENESSKIGRKNYHPNIHPTEKEFDFLVYRKKKDPNGNKVIADKIIGSGKNKRTTYWAPAIQKLE 3a4o X 3.0 BS01 STU X 1 L22 V30 K44 E89 Y90 M91 G94 A140 L143 L16 V24 K38 E83 Y84 M85 G88 A134 L137 N141 D154 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P07948 19857964 902 DAWEIPRESIKLVKRLGAGQFGEVWMGYYNNSTKVAVKTLKPGTMSVQAFLEEANLMKTLQHDKLVRLYAVVTREEPIYIITEYMAKGSLLDFLKSDEGGKVLLPKLIDFSAQIAEGMAYIERKNYIHRDLRAANVLVSESLMCKIADFGLARVEGAKFPIKWTAPEAINFGCFTIKSDVWSFGILLYEIVTYGKIPYPGRTNADVMTALSQGYRMPRVENCPDELYDIMKMCWKEKAEERPTFDYLQSVLDDFYTATE 3a4p A 2.54 BS01 DFQ A 1 V1092 A1108 L1157 Y1159 M1160 K1161 G1163 M1211 A1221 Y1230 V30 A43 L92 Y94 M95 K96 G98 M146 A156 Y165 D1204 A1206 R1208 N1209 D1222 A1243 D139 A141 R143 N144 D157 A168 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=28nM P08581 20093027 1362 VQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3a5y A 1.9 BS01 KAA A 1 S76 E78 R100 H108 N109 F112 M114 Y118 E244 L245 N247 F249 E251 G296 A298 G300 R303 S72 E74 R96 H104 N105 F108 M110 Y114 E216 L217 N219 F221 E223 G268 A270 G272 R275 6.3.1.- 0000049,0000166,0004812,0004824,0005515,0005524,0005737,0005829,0006418,0006430,0016874,0016880,0042803,0043687,0052868,0071468 Kd=11nM remove_due_to_license_issue P0A8N7 20729861 1990 ASWQPSASIPNLLKRAAIMAEIRRFFADRGVLEVETPCMSQATVTDIHLVPFETRFVGPGHSQGMNLWLMTSPEYHMKRLLVAGCGPVFQLCRSFRNEEMGRYHNPEFTMLEWYRPHYDMYRLMNEVDDLLQQVLDCPAAESLSYQQAFLRYLEIDPLSADTLLQLLFTFGVEPNIGKEKPTFVYHFPASQASLAQISTEDHRVAERFEVYYKGIELANGFHELTDAREQQQRFEQDNRKRAARGLPQHPIDQNLIEALKVGMPDCSGVALGVDRLVMLALGAETLAEVIAFSVDRA 3a5y B 1.9 BS01 KAA B 1 S76 E78 R100 H108 N109 F112 M114 Y118 E244 L245 A246 N247 F249 E251 G296 A298 G300 R303 S74 E76 R98 H106 N107 F110 M112 Y116 E229 L230 A231 N232 F234 E236 G281 A283 G285 R288 6.3.1.- 0000049,0000166,0004812,0004824,0005515,0005524,0005737,0005829,0006418,0006430,0016874,0016880,0042803,0043687,0052868,0071468 Kd=11nM remove_due_to_license_issue P0A8N7 20729861 1991 ETASWQPSASIPNLLKRAAIMAEIRRFFADRGVLEVETPCMSQATVTDIHLVPFETRFVGPGHSQGMNLWLMTSPEYHMKRLLVAGCGPVFQLCRSFRNEEMGRYHNPEFTMLEWYRPHYDMYRLMNEVDDLLQQVLDCPAAESLSYQQAFLRYLEIDPLSADKTQLREEEDRDTLLQLLFTFGVEPNIGKEKPTFVYHFPASQASLAQISTEDHRVAERFEVYYKGIELANGFHELTDAREQQQRFEQDNRKRAARGLPQHPIDQNLIEALKVGMPDCSGVALGVDRLVMLALGAETLAEVIAFSVDRA 3a6t A 1.96 BS02 8OG A 1 I6 V8 R23 H28 E34 F35 G37 I80 L82 P116 N119 I4 V6 R21 H26 E32 F33 G35 I78 L80 P114 N117 3.6.1.55 0000287,0005515,0006203,0006260,0006281,0006289,0008413,0016787,0030145,0035539,0044715,0044716,0046067,0046872,0047693 Kd=52nM remove_due_to_license_issue P08337 19864691 134 KLQIAVGIIRNENNEIFITRRAADAHMANKLEFPGGKIEMGETPEQAVVRELQEEVGITPQHFSLFEKLEYEFPDRHITLWFWLVERWEGEPWGKEGQPGEWMSLVGLNADDFPPANEPVIAKLKRL 3a73 A 2.19 BS01 PJ2 A 1 M123 Y138 I142 A158 Y161 F165 M122 Y137 I141 A157 Y160 F164 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 20014793 1011 AHKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCCFAEEGKKLVAASQAALG 3a73 A 2.19 BS02 PJ2 A 2 R114 H146 R113 H145 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 20014793 1012 AHKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCCFAEEGKKLVAASQAALG 3a9i A 1.8 BS02 LYS A 1 R12 D92 S135 T166 H195 H197 R11 D91 S128 T159 H188 H190 2.3.3.14 0003824,0004410,0005737,0009085,0016740,0019752,0019878,0036440,0046872,0046912 remove_due_to_license_issue O87198 19996101 378 REWKIIDSTLREGEQFEKANFSTQDKVEIAKALDEFGIEYIEVTTPVASPQSRKDAEVLASLGLKAKVVTHIQCRLDAAKVAVETGVQGIDLLFGTSKYLDIPRIIEEAKEVIAYIREAAPHVEVRFSAEDTFRSEEQDLLAVYEAVAPYVDRVGLADTVGVATPRQVYALVREVRRVVGPRVDIEFHGHNDTGCAIANAYEAIEAGATHVDTTILGIGERNGITPLGGFLARMYTLQPEYVRRKYKLEMLPELDRMVARMVGVEIPFNNYITGETAFSHKAGMHLKAIYINPEAYEPYPPEVFGVKGLHYGEEELHRVTQHIKALADRGQLTLEELDRILREWITA 3aaf A 1.9 BS01 dna C 0 K976 F977 G978 R993 Y1034 F1037 M1038 K1039 K21 F22 G23 R38 Y79 F82 M83 K84 3.1.-.-,5.6.2.4 0006260,0006281,0043138 remove_due_to_license_issue Q14191 20159463 1 ~ 14 SWDFGPQAFKLLSAVDILGEKFGIGLPILFLRGSNSQRLADQYRRHSLFGTGKDQTESWWKAFSRQLITEGFLVEVSRYNKFMKICALTKKGRNWLHKANTESQSLILQ 3aaf A 1.9 BS02 dna D 0 R987 S989 N990 S991 Q992 K1036 F1037 R32 S34 N35 S36 Q37 K81 F82 3.1.-.-,5.6.2.4 0006260,0006281,0043138 remove_due_to_license_issue Q14191 20159463 1 ~ 14 SWDFGPQAFKLLSAVDILGEKFGIGLPILFLRGSNSQRLADQYRRHSLFGTGKDQTESWWKAFSRQLITEGFLVEVSRYNKFMKICALTKKGRNWLHKANTESQSLILQ 3aaf B 1.9 BS01 dna C 0 R987 S989 N990 S991 Q992 K1036 F1037 R32 S34 N35 S36 Q37 K81 F82 3.1.-.-,5.6.2.4 0006260,0006281,0043138 remove_due_to_license_issue Q14191 20159463 1 ~ 14 SWDFGPQAFKLLSAVDILGEKFGIGLPILFLRGSNSQRLADQYRRHSLFGTGKDQTESWWKAFSRQLITEGFLVEVSRYNKFMKICALTKKGRNWLHKANTESQSLILQ 3aaf B 1.9 BS02 dna D 0 K976 F977 G978 R993 Y1034 F1037 M1038 K1039 K21 F22 G23 R38 Y79 F82 M83 K84 3.1.-.-,5.6.2.4 0006260,0006281,0043138 remove_due_to_license_issue Q14191 20159463 1 ~ 14 SWDFGPQAFKLLSAVDILGEKFGIGLPILFLRGSNSQRLADQYRRHSLFGTGKDQTESWWKAFSRQLITEGFLVEVSRYNKFMKICALTKKGRNWLHKANTESQSLILQ 3aaq A 2.0 BS01 ARU A 1 G51 S52 T53 R56 G188 G189 Q231 G299 N302 Y346 Y350 G11 S12 T13 R16 G144 G145 Q187 G255 N258 Y302 Y306 ? 0000166,0009134,0016020,0016787,0017110,0046872 Ki=0.5mM remove_due_to_license_issue Q5ZUA2 20159467 1 KHSCIAVIDAGSTGSRLHIYSYDTDDTNTPIHIEEIWNKKIKPGFASIQPNSVTIDAYLTMLLADAPIHNIPVYFYATAGMRLLPQSQQKKYYDELEYWFRQQSQWQLVEAKTITGNDEALFDWLAVNYKLDTLKSSVGVMDMGGASVQIVFPMPKNAEISKHNQVELNIYGQNINLYVHSFLGLGQTEMSHQFLNSPSCFANDYPLPDGESGQGNAPSCKEEVTSLMNSVHKVNQQIQPLLALNPVNEWYSIGGISNLASSQLFHFENSELTNQSLLQQGDNQICHQQWDILNGQYPDDEYLYQYCLLSSYYYALMVDGYGINPNQTIHYIPPEQNLDWTIGVVLHRA 3aas A 1.75 BS01 GUS A 1 H40 D171 Q174 S177 V191 S192 G194 G196 H40 D171 Q174 S177 V191 S192 G194 G196 H40 D84 Q174 G175 D176 S177 G178 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=31uM remove_due_to_license_issue P00760 20202854 1001 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3aau A 1.8 BS01 GZC A 1 C25 H40 C41 K43 D171 S172 S177 V191 S192 G194 G196 C25 H40 C41 K43 D171 S172 S177 V191 S192 G194 G196 H40 D84 Q174 G175 D176 S177 G178 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 20202854 3001 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3aav A 1.7 BS01 A2C A 1 F24 H40 D171 S172 C173 G175 D176 S177 V191 G196 C197 F24 H40 D171 S172 C173 G175 D176 S177 V191 G196 C197 H40 D84 Q174 G175 D176 S177 G178 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 20202854 1001 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3abt A 3.2 BS01 2PF A 1 G285 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 V590 L625 P626 W751 W756 S760 Y761 G800 E801 A809 T810 V811 A814 G114 G116 S118 L136 E137 A138 R139 G144 R145 G159 A160 M161 V162 V411 L446 P447 W572 W577 S581 Y582 G612 E613 A621 T622 V623 A626 T335 D553 K661 T164 D374 K482 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 20568732 1 SGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLG 3abu A 3.1 BS01 12F A 1 G285 S286 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 F538 A539 H564 A589 V590 L625 W751 W756 S760 Y761 G800 E801 A809 T810 V811 A814 G114 S115 G116 S118 L136 E137 A138 R139 G144 R145 G159 A160 M161 V162 F358 A359 H384 A409 V410 L445 W571 W576 S580 Y581 G611 E612 A620 T621 V622 A625 T335 D553 K661 T164 D373 K481 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 20568732 1 SGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAM 3acl A 2.35 BS02 3F1 A 1 D43 F53 H56 S65 Y66 M73 Q115 W117 D41 F51 H54 S63 Y64 M71 Q113 W115 1.13.11.24 0003712,0005515,0005634,0005654,0005737,0005829,0006366,0007586,0008127,0016604,0030099,0030224,0046872,0051213 Kd=0.6uM remove_due_to_license_issue O00625 20711196 302 SSKKVTLSVLSREQSEGVGARVRRSIGRPELKNLDPFLLFDEFKGGRPGGFPDHPHRGFETVSYLLEGGSMAHEDFCGHTGKMNPGDLQWMTAGRGILHAEMPCSEEPAHGLQLWVNLRSSEKMVEPQYQELKSEEIPKPSKDGVTVAVISGEALGIKSKVYTRTPTLYLDFKLDPGAKHSQPIPKGWTSFIYTISGDVYIGPDDAQQKIEPHHTAVLGEGDSVQVENKDPKRSHFVLIAGEPLREPVIQHGPFVMNTNEEISQAILDFRNAKNGFERAKTWKSKIGN 3acw A 1.63 BS01 651 A 1 F22 F26 G138 L145 L160 L164 Q165 N168 F22 F26 G138 L145 L160 L164 Q165 N168 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 remove_due_to_license_issue A9JQL9 21098670 1001 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 3acx A 1.31 BS01 673 A 1 H18 F22 F26 Y41 A134 V137 G138 L141 L145 A157 L160 G161 H18 F22 F26 Y41 A134 V137 G138 L141 L145 A157 L160 G161 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 remove_due_to_license_issue A9JQL9 21098670 1001 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 3ad7 B 2.2 BS03 MTG B 1 I67 R69 M264 Y271 T354 K358 V402 I67 R69 M264 Y271 T354 K358 V402 A62 T65 T66 G326 K358 A62 T65 T66 G326 K358 1.5.3.24 0000166,0005737,0008115,0016491,0046653 Kd=3.01mM remove_due_to_license_issue Q50LF2 20675294 801 ADLLPEHPEFLWNNPEPKKSYDVVIVGGGGHGLATAYYLAKNHGITNVAVLEKGWLAGGNMARNTTIIRSNYLWDESAGIYEKSLKLWEELPEELEYDFLFSQRGVLNLAHTLGDVRESIRRVEANKFNGVDAEWLTPEQVKEVCPIINTGDNIRYPVMGATYQPRAGIAKHDHVAWAFARKANEMGVDIIQNCEVTGFLKDGEKVTGVKTTRGTILAGKVALAGAGHSSVLAELAGFELPIQSHPLQALVSELFEPVHPTVVMSNHIHVYVSQAHKGELVMGAGIDSYNGYGQRGAFHVIEEQMAAAVELFPIFARAHVLRTWGGIVDTTMDASPIISKTPIQNLYVNCGWGTGGFKGTPGAGYTLAHTIAHDEPHKLNAPFALERFETGHLIDEHGAAAVAH 3ad8 B 2.2 BS03 PYC B 1 T65 I67 R69 M264 Y271 T354 K358 V402 T65 I67 R69 M264 Y271 T354 K358 V402 A62 T65 T66 G326 K358 A62 T65 T66 G326 K358 1.5.3.24 0000166,0005737,0008115,0016491,0046653 Kd=0.69mM remove_due_to_license_issue Q50LF2 20675294 801 ADLLPEHPEFLWNNPEPKKSYDVVIVGGGGHGLATAYYLAKNHGITNVAVLEKGWLAGGNMARNTTIIRSNYLWDESAGIYEKSLKLWEELPEELEYDFLFSQRGVLNLAHTLGDVRESIRRVEANKFNGVDAEWLTPEQVKEVCPIINTGDNIRYPVMGATYQPRAGIAKHDHVAWAFARKANEMGVDIIQNCEVTGFLKDGEKVTGVKTTRGTILAGKVALAGAGHSSVLAELAGFELPIQSHPLQALVSELFEPVHPTVVMSNHIHVYVSQAHKGELVMGAGIDSYNGYGQRGAFHVIEEQMAAAVELFPIFARAHVLRTWGGIVDTTMDASPIISKTPIQNLYVNCGWGTGGFKGTPGAGYTLAHTIAHDEPHKLNAPFALERFETGHLIDEHGAAAVAH 3adb A 2.8 BS01 rna C 0 Y79 K91 I120 V124 M128 K138 N181 D191 R195 S199 I202 K203 K209 I212 V216 R219 K220 K224 K227 Y81 K93 I122 V126 M130 K140 N183 D193 R197 S201 I204 K205 K211 I214 V218 R221 K222 K226 K229 2.7.1.164 0001717,0002098,0005524,0016301,0016773,0043915 remove_due_to_license_issue Q58933 20705242 1 ~ 76 HHMLIILTGLPGVGKSTFSKNLAKILSKNNIDVIVLGSDLIRESFPVWKEKYEEFIKKSTYRLIDSALKNYWVIVDDTNYYNSMRRDLINIAKKYNKNYAIIYLKASLDVLIRRNIERGEKIPNEVIKKMYEKFDEPGKKYKWDEPFLIIDTTKDIDFNEIAKKLIEKSKEIPKFYVLEENKNKNNNISDKIDKETRKIVSEYIKSKKLDKDKIKEVVELRKEFLKKIKKMEEVDADRVLKEFKDLLNSY 3adb B 2.8 BS01 rna D 0 W46 E48 E51 K55 Y78 Y79 N80 S81 M82 R84 I120 V124 M128 D133 K137 K138 Y139 K140 W141 D188 D191 R195 S199 I202 I212 V216 R219 K220 K227 K228 W53 E55 E58 K62 Y85 Y86 N87 S88 M89 R91 I127 V131 M135 D140 K144 K145 Y146 K147 W148 D187 D190 R194 S198 I201 I211 V215 R218 K219 K226 K227 2.7.1.164 0001717,0002098,0005524,0016301,0016773,0043915 remove_due_to_license_issue Q58933 20705242 1 ~ 76 MNHHHHHMLIILTGLPGVGKSTFSKNLAKILSKNNIDVIVLGSDLIRESFPVWKEKYEEFIKKSTYRLIDSALKNYWVIVDDTNYYNSMRRDLINIAKKYNKNYAIIYLKASLDVLIRRNIERGEKIPNEVIKKMYEKFDEPGKKYKWDEPFLIIDTTKDIDFNEIAKKLIEKSKEIPKFKNNNISDKIDKETRKIVSEYIKSKKLDKDKIKEVVELRKEFLKKIKKMEEVDADRVLKEFKDLLNSY 3ads A 2.25 BS01 IMN A 1 R280 G284 C285 R288 I341 S342 M348 R66 G70 C71 R74 I127 S128 M134 ? 0003677,0004879,0005634,0006355 Kd=9.73uM remove_due_to_license_issue EC50=50000nM P37231 20717101 1 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3ads A 2.25 BS02 IMN A 2 I281 F282 C285 S289 H323 F360 F363 M364 H449 L469 Y473 I67 F68 C71 S75 H109 F146 F149 M150 H235 L255 Y259 ? 0003677,0004879,0005634,0006355 Kd=9.73uM remove_due_to_license_issue EC50=50000nM P37231 20717101 2 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3adt A 2.7 BS01 HID A 1 C285 Q286 S289 H323 L330 F363 M364 H449 Y473 C68 Q69 S72 H106 L113 F146 M147 H232 Y256 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 20717101 2 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3adt A 2.7 BS02 HID A 2 Y222 P227 L228 K230 R288 M329 S332 L333 Y20 P25 L26 K28 R71 M112 S115 L116 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 20717101 3 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3adu A 2.77 BS01 MYI A 1 C285 R288 L330 L333 C68 R71 L113 L116 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 20717101 1 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3adu A 2.77 BS02 MYI A 2 F282 C285 S289 H323 Y327 F363 H449 Y473 F65 C68 S72 H106 Y110 F146 H232 Y256 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 20717101 2 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3adv A 2.27 BS01 SRO A 1 C285 S289 Y327 L330 M364 H449 C71 S75 Y113 L116 M150 H235 ? 0003677,0004879,0005634,0006355 Kd=933uM remove_due_to_license_issue P37231 20717101 1 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3adv A 2.27 BS02 SRO A 2 L228 R288 E295 M329 L333 E343 L26 R74 E81 M115 L119 E129 ? 0003677,0004879,0005634,0006355 Kd=933uM remove_due_to_license_issue P37231 20717101 3 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3afk A 1.95 BS01 GAL C 1 N43 H59 R63 W80 E83 N44 H60 R64 W81 E84 3.1.21.- 0004518,0004536,0006259,0006915,0030246,0030247,0043065 remove_due_to_license_issue Q6WY08 20530247 2 MQGVNIYNISAGTSVDLAAPVTTGDIVTFFSSALNLNAGAGNPNNTTLNLFAENGAYLLHIAFRLQENVIIFNSRQPDGPWLVEQRVSDVANQFAGIDGKAMVTVFDHGDKYQVVINEKTVIQYTKQISGLTSSLSYNATEETSIFSTVVEAVTYTGLALEHHHHHH 3ag9 B 2.0 BS01 A02 B 1 G52 S53 F54 G55 A70 Y122 V123 F129 D166 E170 L173 F187 E230 G38 S39 F40 G41 A56 Y108 V109 F115 D152 E156 L159 F173 E216 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Ki=9nM remove_due_to_license_issue P00517 20732331 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKIRVSINEKCGKEFSEF 3agl A 2.1 BS01 A03 A 1 G52 S53 F54 G55 V57 A70 M120 E121 V123 E127 P169 E170 L173 T183 E203 E230 F327 Y330 G43 S44 F45 G46 V48 A61 M111 E112 V114 E118 P160 E161 L164 T174 E194 E221 F318 Y321 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 Ki=16nM remove_due_to_license_issue P17612 20732331 351 SEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3ahn A 1.8 BS01 3A1 A 1 G327 Y328 C329 H356 E357 H360 W377 C383 F420 R476 Q477 H479 Y486 Y487 Y490 G327 Y328 C329 H356 E357 H360 W377 C383 F420 R476 Q477 H479 Y486 Y487 Y490 ? 0004222,0006508,0006518,0046872 Ki=90.1nM remove_due_to_license_issue Q4W803 20817732 565 MKFSEFRYERPNIEKLKASFQQALQSFQKASNAEEQNEAMKEINQLRNDFSTMAQICYIRHTIDTNDEFYKQEQDFFDEVEPIVKGLVNDYYRALVSSPFRSQLEGKWGKQLFALAEAELKTYSPDIVEDLQLENKLTSEYTKLVASAKIFFEGEERTLAQLQPFVESPDRDMRKRASEARFTFFQEHEEKFDEIYDQLVKVRTAIAQKLGFKNFVELGYARLGRTDYNAEMVAKFRKQVEKHIVPIAVKLRERQRERIGVEKLKYYDEAFVFPTGNPMPKGDANWIIENGKKMYEELSPETGEFFRYMIEHELMDLVAKKGKASGGYCTYIENYKAPFIFSNFTGTSGDIDVLTHEAGHAFQVYESRHYEIPEYNWPTLEACEIHSMSMEFFTWPWMKLFFKEDAEKYQFYHLSDALLFLPYGVAVDEFQHFVYENPNATPAERKQAWRAIERKYMPTKDYDGNDYLERGGFWQRQSHIYTTAFYYIDYTLAQICAFQFWKRSRENYKEAWNDYLTLCRQGGSKPFTELVRVANLISPFEDGCVQSVVGGIEGWLNSVDDQSL 3aho A 1.88 BS02 3A2 A 1 G327 Y328 C329 H356 E357 H360 W377 L380 E384 R476 Q477 H479 Y486 Y487 Y490 G327 Y328 C329 H356 E357 H360 W377 L380 E384 R476 Q477 H479 Y486 Y487 Y490 ? 0004222,0006508,0006518,0046872 Ki=88.9nM remove_due_to_license_issue Q4W803 20817732 566 MKFSEFRYERPNIEKLKASFQQALQSFQKASNAEEQNEAMKEINQLRNDFSTMAQICYIRHTIDTNDEFYKQEQDFFDEVEPIVKGLVNDYYRALVSSPFRSQLEGKWGKQLFALAEAELKTYSPDIVEDLQLENKLTSEYTKLVASAKIFFEGEERTLAQLQPFVESPDRDMRKRASEARFTFFQEHEEKFDEIYDQLVKVRTAIAQKLGFKNFVELGYARLGRTDYNAEMVAKFRKQVEKHIVPIAVKLRERQRERIGVEKLKYYDEAFVFPTGNPMPKGDANWIIENGKKMYEELSPETGEFFRYMIEHELMDLVAKKGKASGGYCTYIENYKAPFIFSNFTGTSGDIDVLTHEAGHAFQVYESRHYEIPEYNWPTLEACEIHSMSMEFFTWPWMKLFFKEDAEKYQFYHLSDALLFLPYGVAVDEFQHFVYENPNATPAERKQAWRAIERKYMPTKDYDGNDYLERGGFWQRQSHIYTTAFYYIDYTLAQICAFQFWKRSRENYKEAWNDYLTLCRQGGSKPFTELVRVANLISPFEDGCVQSVVGGIEGWLNSVDDQSL 3ai8 B 2.11 BS01 HNQ B 1 Q23 G24 S25 C26 H110 H111 C119 G121 W221 Q25 G26 S27 C28 H112 H113 C121 G123 W223 Q23 C29 H199 N219 Q25 C31 H201 N221 3.4.22.1 0006508,0008234 Ki=271.8uM remove_due_to_license_issue Ki=271800nM P07858 21598397 255 LKLPASFDAREQWPQCPTIKEIRDQGSCGSCWAFGAVEAISDRICIHTNAHVSVEVSAEDLLTCCGSMCGDGCNGGYPAEAWNFWTRKGLVSGGLYESHVGCRPYSIPPCEHHVNGSRPPCTGEGDTPKCSKICEPGYSPTYKQDKHYGYNSYSVSNSEKDIMAEIYKNGPVEGAFSVYSDFLLYKSGVYQHVTGEMMGGHAIRILGWGVENGTPYWLVANSWNTDWGDNGFFKILRGQDHCGIESEVVAGIPRTD 3aid A 2.5 BS01 ARQ A 1 D25 G27 A28 I50 D25 G27 A28 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=137nM remove_due_to_license_issue P03369 8894111 401 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3aid B 2.5 BS01 ARQ A 1 D25 G27 G48 G49 I50 D25 G27 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 8894111 401 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3aig A 2.8 BS03 0ZC A 1 K106 I107 I108 T139 H142 E143 I165 P168 G169 L170 K105 I106 I107 T138 H141 E142 I164 P167 G168 L169 3.4.24.46 0004222,0005576,0005886,0006508,0008237,0046872 remove_due_to_license_issue P34179 9521103 1000 NLPQRYIELVVVADRRVFMKYNSDLNIIRTRVHEIVNIINEFYRSLNIRVSLTDLEIWSGQDFITIQSSSSNTLNSFGEWRERVLLTRKRHDNAQLLTAINFEGKIIGKAYTSSMCNPRSSVGIVKDHSPINLLVAVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTPGRSYEFSDDSMGYYQKFLNQYKPQCILNKP 3aje A 1.8 BS01 THR A 1 T36 V37 G39 H68 R122 A142 E181 S182 T35 V36 G38 H67 R121 A141 E180 S181 2.7.7.87 0000049,0003725,0005524,0005737,0006450,0008033,0016779,0061710 remove_due_to_license_issue Q970S6 21538543 353 TQIIKIDPLNPEIDKIKIAADVIRNGGTVAFPTETVYGLGANAFDGNACLKIFQAKNRPVDNPLIVHIADFNQLFEVAKDIPDKVLEIAQIVWPGPLTFVLKKTERVPKEVTAGLDTVAVRMPAHPIALQLIRESGVPIAAPSANLATRPSPTKAEDVIVDLNGRVDVIIDGGHTFFGVESTIINVTVEPPVLLRPGPFTIEELKKLFGEIVIPHYAPNTRLLLVENRNIFKDVVSLLSKKYKVALLIPKELSKEFEGLQQIILGSDENLYEVARNLFDSFRELDKLNVDLGIMIGFPERGIGFAIMNRARKASGFSIIKAISDVYKYV 3am1 A 2.4 BS01 rna B 0 Y83 N84 S85 R88 D137 K141 K142 Y143 K144 W145 S191 D192 D195 K196 R199 S203 I206 I216 R223 Y81 N82 S83 R86 D135 K139 K140 Y141 K142 W143 S178 D179 D182 K183 R186 S190 I193 I203 R210 2.7.1.164 0001717,0002098,0005524,0016301,0016773,0043915 remove_due_to_license_issue Q58933 20870747 1 ~ 81 DIMLIILTGLPGVGKSTFSKNLAKILSKNNIDVIVLGSDLIRESFPVWKEKYEEFIKKSTYRLIDSALKNYWVIVDDTNYYNSMRRDLINIAKKYNKNYAIIYLKASLDVLIRRNIERGEKIPNEVIKKMYEKFDEPGKKYKWDEPFLIIDTTKDIDFNEIAKKLIEKSKEIPKFNISDKIDKETRKIVSEYIKSKKLDKDKIKEVVELRKEFLKKIKKVDADRVLKEFKDLLNSY 3ama A 1.75 BS02 SKE A 1 L49 V57 A70 Y122 A123 G126 L173 F327 L49 V57 A70 Y122 A123 G126 L173 F322 D166 K168 E170 N171 D184 T201 D166 K168 E170 N171 D184 T201 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 Ki=0.297uM remove_due_to_license_issue Kd=>10000nM P17612 21774789 351 GNAAAAKKGSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIRTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRIQQAVNFPFLVKLEFSFKDNSNLYMVLEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKSNFDDYEEEEIRVSINEKCGKEFSEF 3amb A 2.25 BS02 VX6 A 1 V57 A70 K72 Y122 A123 P124 G126 L173 D184 N326 V55 A68 K70 Y120 A121 P122 G124 L171 D182 N319 D166 K168 E170 N171 D184 T201 D164 K166 E168 N169 D182 T199 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 Ki=0.66uM remove_due_to_license_issue Kd=>10000nM P17612 21774789 351 AAAAKKGSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIRTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRIQQAVNFPFLVKLEFSFKDNSNLYMVLEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKSNFDDYEEEEIRVSINEKCGKEFSEF 3amv A 2.1 BS03 BIN A 1 I68 Q71 Q72 Y75 R193 F196 R242 R309 R310 I64 Q67 Q68 Y71 R189 F192 R238 R296 R297 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=10.8nM remove_due_to_license_issue P00489 10548038 930 SDQEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLP 3anq A 2.6 BS01 EHB A 1 F170 A186 K188 F238 L241 D307 F37 A53 K55 F105 L108 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=240nM Q13627 20981014 1 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 3anr A 2.6 BS01 HRM A 1 A186 K188 F238 L241 L294 D307 A53 K55 F105 L108 L161 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=80nM, Ki=33nM Q13627 20981014 1 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 3ans A 1.98 BS01 S38 A 1 F267 D335 W336 M339 Y383 M419 Y466 H524 F36 D104 W105 M108 Y152 M188 Y235 H293 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F36 H103 D104 W105 N128 N147 Y152 Y235 D265 H293 3.1.3.76,3.3.2.10 0003824 ic50=565nM remove_due_to_license_issue IC50=565nM P34913 21192659 601 CNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD 3ant A 2.4 BS01 S82 A 1 F267 D335 W336 M339 Y383 L408 Y466 H524 F36 D104 W105 M108 Y152 L177 Y235 H293 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F36 H103 D104 W105 N128 N147 Y152 Y235 D265 H293 3.1.3.76,3.3.2.10 0003824 ic50=8.5nM remove_due_to_license_issue IC50=6.1nM P34913 21192659 601 CNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD 3ao1 A 1.9 BS01 BZX A 1 H185 G197 H119 G131 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.5mM remove_due_to_license_issue Q72498 21275048 213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEDGIPSMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATD 3ao1 A 1.9 BS02 BZX B 1 G106 R107 W108 P109 G50 R51 W52 P53 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.5mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEDGIPSMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATD 3ao1 B 1.9 BS01 BZX A 1 G106 R107 P109 G50 R51 P53 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.5mM remove_due_to_license_issue Q72498 21275048 213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATDI 3ao1 B 1.9 BS02 BZX B 1 H185 G197 H119 G131 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.5mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATDI 3ao2 A 1.8 BS02 AVX A 1 H185 S195 G197 E198 V201 H116 S124 G126 E127 V130 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=0.17mM remove_due_to_license_issue P04585 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQ 3ao2 A 1.8 BS03 AVX B 1 G106 R107 W108 P109 G50 R51 W52 P53 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=0.17mM remove_due_to_license_issue P04585 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQ 3ao2 B 1.8 BS01 AVX A 1 G106 R107 W108 P109 G50 R51 W52 P53 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=0.17mM remove_due_to_license_issue P04585 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 3ao2 B 1.8 BS02 AVX B 1 H185 R187 G197 E198 V201 H115 R117 G122 E123 V126 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=0.17mM remove_due_to_license_issue P04585 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 3ao4 A 1.95 BS01 833 A 1 H185 G197 E198 H117 G129 E130 3.1.13.2,3.1.26.13 0003676,0015074 Kd=8.5mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATD 3ao4 A 1.95 BS02 833 B 1 G106 R107 W108 P109 I204 D207 G50 R51 W52 P53 I136 D139 3.1.13.2,3.1.26.13 0003676,0015074 Kd=8.5mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATD 3ao4 B 1.95 BS01 833 A 1 G106 R107 W108 P109 I204 D207 G50 R51 W52 P53 I130 D133 3.1.13.2,3.1.26.13 0003676,0015074 Kd=8.5mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKYSAGERIVDIIATD 3ao4 B 1.95 BS02 833 B 1 H185 G197 E198 H116 G123 E124 3.1.13.2,3.1.26.13 0003676,0015074 Kd=8.5mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKYSAGERIVDIIATD 3ao5 A 1.8 BS02 BBY A 1 H185 R187 S195 G197 E198 V201 H115 R117 S122 G124 E125 V128 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.9mM remove_due_to_license_issue Q72498 21275048 213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDI 3ao5 A 1.8 BS03 BBY B 1 G106 R107 W108 P109 G50 R51 W52 P53 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.9mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDI 3ao5 B 1.8 BS03 BBY A 1 G106 R107 W108 P109 G50 R51 W52 P53 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.9mM remove_due_to_license_issue Q72498 21275048 213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEDGSMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATDI 3ao5 B 1.8 BS04 BBY B 1 H185 R187 S195 G197 E198 V201 H117 R119 S127 G129 E130 V133 3.1.13.2,3.1.26.13 0003676,0015074 Kd=5.9mM remove_due_to_license_issue Q72498 21275048 1 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTGATVRAACDWAGIKQEDGSMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATDI 3aox A 1.75 BS01 EMH A 1 L1122 A1148 L1196 L1198 M1199 A1200 L1256 G1269 L37 A52 L100 L102 M103 A104 L160 G173 D1249 A1251 R1253 N1254 D1270 R1279 D153 A155 R157 N158 D174 R183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd=2.4nM remove_due_to_license_issue IC50=1.9nM Q9UM73 21575866 901 STIMTDYNPNYCFAGKTSSISDLKEVPRKNITLIRGLGGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRACAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 3ap7 A 1.53 BS03 SIA B 1 R59 W86 R56 W83 ? 0030246 remove_due_to_license_issue O00214 21288902 3 SLNNLQNIIYNPVIPFVGTIPDQLDPGTLIVIRGHVPSDADRFQVDLQNGSSVKPRADVAFHFNPRFKRAGCIVCNTLINEKWGREEITYDTPFKREKSFEIVIMVLKDKFQVAVNGKHTLLYGHRIGPEKIDTLGIYGKVNIHSIGFSFS 3apc A 2.544 BS01 MMD A 1 M804 I831 K833 D836 I879 E880 I881 V882 M953 I963 D964 M558 I585 K587 D590 I633 E634 I635 V636 M707 I717 D718 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=36nM P48736 21316229 1 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMASEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLG 3aqa A 2.3 BS01 BYH A 1 W97 P98 L108 N156 M165 W25 P26 L36 N84 M93 ? remove_due_to_license_issue Kd=28000nM, IC50=28000nM P25440 21513886 201 GRVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQE 3aqt A 2.5 BS01 RCO A 1 S110 L114 R145 A146 D149 S87 L91 R122 A123 D126 ? 0003677,0006355 Kd=0.19uM remove_due_to_license_issue Q8NR95 21559286 230 RAQKREQTRARLITSARTLMAERGVDNVGIAEITEGANIGTGTFYNYFPDREQLLQAVAEDAFESVGIALDQVLTKLDDPAEVFAGSLRHLVRHSLEDRIWGGFFIQMGAAHPVLMRILGPRARRDLLHGLETGRFTIEDLDLATTCTFGSLIAAIQMALSDDKDQIFAAAMLRMVGVQAAEAREIASRPLPEIS 3ara A 1.7 BS01 MKH A 1 V65 G99 V100 Y105 G110 V42 G76 V77 Y82 G87 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=0.32uM remove_due_to_license_issue IC50=480nM P33316 22404301 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3ara A 1.7 BS02 MKH B 1 S86 A90 S63 A67 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=0.32uM remove_due_to_license_issue IC50=480nM P33316 22404301 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3ara C 1.7 BS01 MKH A 1 S86 A90 S63 A67 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=0.32uM remove_due_to_license_issue IC50=480nM P33316 22404301 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3ara C 1.7 BS02 MKH C 1 V65 G99 V100 Y105 V109 G110 V42 G76 V77 Y82 V86 G87 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=0.32uM remove_due_to_license_issue IC50=480nM P33316 22404301 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3arb A 2.7 BS01 FEE A 1 C12 F70 Y73 S76 F77 D80 W133 D153 T156 F171 C7 F65 Y68 S71 F72 D75 W126 D146 T149 F164 ? remove_due_to_license_issue P11609 21376639 601 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYWGSLHHILDAQKMVWNHRHHHHHH 3arb C 2.7 BS01 FEE A 1 P28 N30 R95 P28 N30 R94 ? remove_due_to_license_issue P01848 21376639 601 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKDFACANAFNNSIIPEDTFFPSP 3ard A 3.01 BS01 3GH A 1 S28 M69 F70 Y73 S76 F77 D80 W133 D153 T156 F171 S23 M64 F65 Y68 S71 F72 D75 W127 D147 T150 F165 ? remove_due_to_license_issue P11609 21376639 307 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYWGSLHHILDAQKMVWNHRHHHH 3ard C 3.01 BS01 3GH A 1 P28 N30 R95 G96 P28 N30 R94 G95 ? remove_due_to_license_issue P01848 21376639 307 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKFACANAFNNSIIPEDTFFPSP 3are A 2.8 BS01 4GH A 1 F70 Y73 S76 F77 D80 V118 W133 L150 D153 G155 T156 F171 F64 Y67 S70 F71 D74 V110 W125 L142 D145 G147 T148 F163 ? remove_due_to_license_issue P11609 21376639 601 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSKEDYPIEIQLSAGCEMYGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYWGSLHHILDAQKMVWNHRHHHH 3are C 2.8 BS01 4GH A 1 P28 R95 P28 R94 ? remove_due_to_license_issue P01848 21376639 601 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKDFACANAFNNSIIPEDTFFPSP 3arf A 2.9 BS01 DB3 A 1 C12 Q14 V30 F70 Y73 S76 F77 D80 W133 D153 T156 C6 Q8 V24 F64 Y67 S70 F71 D74 W126 D146 T149 ? remove_due_to_license_issue P11609 21376639 650 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYWGSLHHILDAQKMVWNHRHHHH 3arf C 2.9 BS01 DB3 A 1 P28 N30 R95 G96 P28 N30 R94 G95 ? remove_due_to_license_issue P01848 21376639 650 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKDFACANAFNNSIIPEDTFFPSP 3arg A 3.0 BS01 DB6 A 1 C12 F70 Y73 S76 F77 D80 W133 D153 G155 T156 V160 C6 F64 Y67 S70 F71 D74 W124 D144 G146 T147 V151 ? remove_due_to_license_issue P11609 21376639 650 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMPKEDYPIEIQLSAGCEMYNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNDETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYWGSLHHILDAQKMVWNHRHHHH 3arg C 3.0 BS01 DB6 A 1 P28 R95 P28 R94 ? remove_due_to_license_issue P01848 21376639 650 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSAGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKDFACANAFNNSIIPEDTFFPSP 3arn A 1.8 BS01 MSJ A 1 G99 V100 Y105 G110 V112 G76 V77 Y82 G87 V89 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=3.9uM remove_due_to_license_issue IC50=9.48e+3nM P33316 22339362 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3arn A 1.8 BS02 MSJ B 1 S86 G87 A90 S63 G64 A67 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=3.9uM remove_due_to_license_issue IC50=9.48e+3nM P33316 22339362 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3arn C 1.8 BS01 MSJ A 1 S86 G87 A90 K91 S63 G64 A67 K68 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=3.9uM remove_due_to_license_issue IC50=9.48e+3nM P33316 22339362 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3arn C 1.8 BS02 MSJ C 1 G99 V100 Y105 V109 G110 V112 G76 V77 Y82 V86 G87 V89 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 ic50=3.9uM remove_due_to_license_issue IC50=9.48e+3nM P33316 22339362 165 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQAL 3arp A 1.55 BS01 DEQ A 1 W168 V205 W275 T276 W397 W147 V184 W254 T255 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPP 3arq A 1.5 BS01 DM5 A 1 W275 G320 D392 W397 Y435 W254 G299 D371 W376 Y414 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3arr A 1.65 BS01 PNX A 1 W275 G367 K370 W397 Y435 W254 G346 K349 W376 Y414 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMA 3arr A 1.65 BS02 PNX A 2 W168 V205 H228 W570 W147 V184 H207 W549 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMA 3art A 2.23 BS01 DEQ A 1 G320 G321 A322 W397 G299 G300 A301 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3art A 2.23 BS02 DEQ A 2 W168 Y171 N208 S209 D229 W231 W147 Y150 N187 S188 D208 W210 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3art A 2.23 BS03 DEQ A 3 V146 P148 N150 P181 D183 R262 V125 P127 N129 P160 D162 R241 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 608 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3aru A 1.9 BS01 PNX A 1 F316 G367 K370 D392 F393 W397 Y435 F295 G346 K349 D371 F372 W376 Y414 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3aru A 1.9 BS02 PNX A 2 V205 E315 F316 G321 A322 V184 E294 F295 G300 A301 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3aru A 1.9 BS03 PNX A 3 W168 N208 A212 H228 D229 W147 N187 A191 H207 D208 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 608 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3arv A 1.5 BS01 SAU A 1 W275 W397 W254 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3arv A 1.5 BS02 SAU A 2 W168 Y171 V205 S209 T276 W147 Y150 V184 S188 T255 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3arw A 1.5 BS01 CTI A 1 W275 W397 W254 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3arx A 1.16 BS01 POY A 1 W275 G367 K370 D392 W397 Y435 W254 G346 K349 D371 W376 Y414 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3arx A 1.16 BS02 POY A 2 W168 V205 S209 A212 H228 D229 W147 V184 S188 A191 H207 D208 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3ary A 1.35 BS01 I5I A 1 W275 W397 W254 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3ary A 1.35 BS02 I5I A 2 W168 Y171 V205 W147 Y150 V184 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGVVTPPN 3arz A 1.82 BS01 I5I A 1 W275 D392 W397 W254 D371 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMA 3arz A 1.82 BS02 I5I A 2 W168 Y171 V205 W147 Y150 V184 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGWTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMA 3as0 A 2.0 BS01 SAU A 1 D392 W397 D371 W376 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3as0 A 2.0 BS02 SAU A 2 E315 F316 G320 G321 A322 E294 F295 G299 G300 A301 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3as1 A 2.0 BS01 CTI A 1 G320 G321 A322 G299 G300 A301 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3as2 A 1.8 BS01 POY A 1 G367 K370 D392 W397 Y435 G346 K349 D371 W376 Y414 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3as2 A 1.8 BS02 POY A 2 N208 S209 N187 S188 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3as2 A 1.8 BS03 POY A 3 E42 A44 N52 D53 M54 K56 E21 A23 N31 D32 M33 K35 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 608 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMAGGV 3as3 A 2.4 BS01 I5I A 1 W397 R463 W376 R442 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 606 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMA 3as3 A 2.4 BS02 I5I A 2 G321 A322 G300 A301 D311 D313 E315 Y391 D290 D292 E294 Y370 3.2.1.14 0004553,0004568,0005975,0006032,0008061 remove_due_to_license_issue Q9AMP1 21531720 607 APTAPSIDMYGSNNLQFSKIELAMETTSGYNDMVKYHELAKIKVKFNQWSGTSGDTYNVYFDGVKVATGAITGSQTTASFEYGQGGLYQMEIEACDATGCSKSAPVEITIADTDGSHLKPLTMNVDPNNKSYNTDPSIVMGTYFVEWGIYGRDYTVDNMPVDNLTHILYGFIPICGPNESVKSVGGNSFNALQTACRGVNDYEVVIHDPWAAYQKSFPQAGHEYSTPIKGNYAMLMALKQRNPDLKIIPSIGGGTLSDPFYDFVDKKNRDTFVASVKKFLKTWKFYDGVDIDWEFPGGGGAAADKGDPVNDGPAYIALMRELRVMLDELEAETGRTYELTSAIGVGYDKIEDVDYADAVQYMDYIFAMTYDFYGGWNNVPGHQTALYCGSFMRPGQCDGGGVDENGEPYKGPAYTADNGIQLLLAQGVPANKLVLGTAMYGRGWEGVTPDTLTDPNDPMTGTATGKLKGSTAQGVWEDGVIDYKGIKSFMLGANNTGINGFEYGYDAQAEAPWVWNRSTGELITFDDHRSVLAKGNYAKSLGLAGLFSWEIDADNGDILNAMHEGMA 3asx A 2.0 BS01 D99 A 1 F54 V179 L183 L211 F288 C289 P292 F19 V144 L148 L176 F253 C254 P257 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=20nM remove_due_to_license_issue P37268 21353782 1 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVKIRKGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQN 3at1 A 2.8 BS01 PCT A 1 S52 T53 R54 T55 R105 S52 T53 R54 T55 R105 R54 T55 K84 R105 H134 Q137 T228 P266 G292 R54 T55 K84 R105 H134 Q137 T228 P266 G292 2.1.3.2 0004070,0004088,0005515,0005737,0005829,0006207,0006221,0006520,0006541,0009347,0016597,0016740,0016743,0042802,0044205,0070207 remove_due_to_license_issue P0A786 2405902 311 ANPLYQKHIISINDLSRDDLNLVLATAAKLKANPQPELLKHKVIASCFFEASTRTRLSFQTSMHRLGASVVGFSDSANTSLGKKGETLADTISVISTYVDAIVMRHPQEGAARLATEFSGNVPVLNAGDGSNQHPTQTLLDLFTIQQTEGRLDNLHVAMVGDLKYGRTVHSLTQALAKFDGNRFYFIAPDALAMPEYILDMLDEKGIAWSLHSSIEEVMAEVDILYMTRVQKERLDPSEYANVKAQFVLRASDLHNAKANMKVLHPLPRVDEIATDVDKTPHAWYFQQAGNGIFARQALLALVLNRDLVL 3at3 A 2.6 BS01 ATK A 1 L45 V53 V66 K68 F113 V116 M163 I174 D175 L45 V53 V66 K68 F113 V116 M163 I174 D175 D156 K158 N161 D175 P184 S194 D156 K158 N161 D175 P184 S194 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=110nM P68400 21735094 336 MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 3at4 A 2.2 BS01 CCK A 1 L45 V53 V66 K68 F113 H115 V116 M163 I174 D175 L44 V52 V65 K67 F112 H114 V115 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=2.26nM remove_due_to_license_issue P68400 21735094 336 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 3ati A 1.71 BS02 SZ4 A 1 D189 S190 C191 V209 G214 D171 S172 C173 V191 G196 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 6 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3atk A 1.74 BS02 SZ1 A 1 S190 S195 V209 C215 S172 S177 V191 C197 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 4 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3atm A 1.72 BS02 TSS A 1 S190 C191 Q192 S195 W211 C215 S172 C173 Q174 S177 W193 C197 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 5 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3atp A 2.5 BS01 SER A 1 R64 N68 F151 F152 Q154 T156 R26 N30 F113 F114 Q116 T118 ? 0006935,0007165 remove_due_to_license_issue P02942 21979954 201 NFTVLQTIRQQQSTLNGSWVALLQTRNTLNRAGIRYMMDQNNIGSGSTVAELMESASISLKQAEKNWADYEALPRDPRQSTAAAAEIKRNYDIYHNALAELIQLLGAGKINEFFDQPTQGYQDGFEKQYVAYMEQNDRLHDIAVSDNNASY 3atp B 2.5 BS01 SER B 1 R64 N68 F151 F152 T156 R27 N31 F114 F115 T119 ? 0006935,0007165 remove_due_to_license_issue P02942 21979954 201 ENFTVLQTIRQQQSTLNGSWVALLQTRNTLNRAGIRYMMDQNNIGSGSTVAELMESASISLKQAEKNWADYEALPRDPRQSTAAAAEIKRNYDIYHNALAELIQLLGAGKINEFFDQPTQGYQDGFEKQYVAYMEQNDRLHDIAVSDNNAS 3atu A 1.65 BS01 ADP A 1 T14 Y15 G201 G202 E268 K271 R272 S275 G338 G339 R342 D366 T11 Y12 G198 G199 E265 K268 R269 S272 G335 G336 R339 D363 D10 K71 E175 D199 D7 K68 E172 D196 ? 0005524,0140662 remove_due_to_license_issue P0DMV8 21608060 1452 AAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILMG 3atv A 1.58 BS01 ADP A 1 G12 T14 Y15 G201 G202 E268 K271 R272 S275 G338 G339 R342 D366 G10 T12 Y13 G199 G200 E266 K269 R270 S273 G336 G337 R340 D364 D10 K71 E175 D199 D8 K69 E173 D197 ? 0005524,0140662 remove_due_to_license_issue P0DMV8 21608060 1452 KAAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILMG 3au6 A 3.3 BS02 DG3 A 1 R157 G187 S188 R191 V196 G197 D198 D200 Y258 K263 R270 R150 G180 S181 R184 V189 G190 D191 D193 Y251 K256 R263 2.7.7.7,4.2.99.18 0003677,0003824,0003887,0005737,0005829,0006259,0006260,0006281,0008270,0042578,0046872,0071897 remove_due_to_license_issue Q5SJ64 22306405 576 MRNQELARIFEEIGLMSEFLGDNPFRVRAYHQAARTLYDLDTPIEEIAEKGKEALMELPGVGPDLAEKILEFLRTGKVRKHEELSRKVPRGVLEVMEVPGVGPKTARLLYEGLGIDSLEKLKAALDRGFGPKRAERIREGLALAQAAGKRRPLGAVLSLARSLLEAIRALPGVERAELCGSARRYKDTVGDLDFLVASREGERAVEGFVRLPQVKEVYAKGKERATVFLKNGLQVDLRVVPPESYGAGLQYLTGSKAHSIRLRALAQEKGLKLSEYGVFRGEKRIAGETEEEVYAALGLPWIPPPLREDQGEVEAALEGRLPKLLELPQVKGDLQVHSTYSDGQNTLEELWEAAKTMGYRYLAVTDHSPAVRVGPSPEEALKRVGEIRRFNETHGPPYLLAGAEVDIHPDGTLDYPDWVLRELDLVLVSVHSRFNLPKADQTKRLLKALENPFVHVLAHPTARLLGRRAPIEADWEAVFQKAKEKGVAVEIDGYYDRMDLPDDLARMAYGMGLWISLSTDAHQTDHLRFMELAVGTAQRAWIGPERVLNTLDYEDLLSWLKA 3axm A 1.65 BS02 6PG A 1 K175 K201 R295 H298 S379 K159 K185 R279 H282 S360 K175 K201 D202 D203 E204 H294 H327 K334 K159 K185 D186 D187 E188 H278 H311 K318 4.1.1.39 0000166,0000287,0004497,0009507,0009536,0009853,0015977,0015979,0016829,0016984,0019253,0046872 Ki=8.5uM remove_due_to_license_issue P0C512 22609438 479 GFKAGVTYYTPEYETKDTDILAAFRVTPQPGVPPEEAGAAVAAESSTGTWTTVWTDGLTSLDRYKGRCYHIEPVVGEDNQYIAYVAYPLDLFEEGSVTNMFTSIVGNVFGFKALRALRLEDLRIPPTYSKTFQGPPHGIQVERDKLNKYGRPLLGCTIKPKLGLSAKNYGRACYECLRGGLDFTKDDENVNSQPFMRWRDRFVFCAEAIYKSQAETGEIKGHYLNATAGTCEEMIKRAVFARELGVPIVMHDYLTGGFTANTSLAHYCRDNGLLLHIHRAMHAVIDRQKNHGMHFRVLAKALRMSGGDHIHAGTVVGKEREMTLGFVDLLRDDFIEKDRARGIFFTQDWVSMPGVIPVASGGIHVWHMPALTEIFGDDSVLQFGGGTLGHPWGNAPGAAANRVALEACVQARNEGRDLAREGNEIIRSACKWSPELAAACEIWK 3axm B 1.65 BS02 6PG B 1 K175 K201 R295 H298 S379 K161 K187 R281 H284 S359 D203 E204 H294 H327 D189 E190 H280 H313 4.1.1.39 0000166,0000287,0004497,0009507,0009536,0009853,0015977,0015979,0016829,0016984,0019253,0046872 Ki=8.5uM remove_due_to_license_issue P0C512 22609438 479 GFKAGVKLTYYTPEYETKDTDILAAFRVTPQPGVPPEEAGAAVAAESSTGTWTTVWTDGLTSLDRYKGRCYHIEPVVGEDNQYIAYVAYPLDLFEEGSVTNMFTSIVGNVFGFKALRALRLEDLRIPPTYSKTFQGPPHGIQVERDKLNKYGRPLLGCTIKPKLGLSAKNYGRACYECLRGGLDFTKDDENVNSQPFMRWRDRFVFCAEAIYKSQAETGEIKGHYLNATAGTCEEMIKRAVFARELGVPIVMHDYLTGGFTANTSLAHYCRDNGLLLHIHRAMHAVIDRQKNHGMHFRVLAKALRMSGGDHIHAGTVEREMTLGFVDLLRDDFIEKDRARGIFFTQDWVSMPGVIPVASGGIHVWHMPALTEIFGDDSVLQFGGGTLGHPWGNAPGAAANRVALEACVQARNEGRDLAREGNEIIRSACKWSPELAAACEIWK 3axz A 2.25 BS01 ADN A 1 Y86 L87 S88 P89 G113 L138 G140 P144 Y92 L93 S94 P95 G119 L144 G146 P150 P89 E116 R154 P95 E122 R160 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=372uM remove_due_to_license_issue P43912 21602303 401 VPRGSHMWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLADGLLDCPHYTRPEVLEGLTVPPVLMSGHHEEIRKWRLKQSLQRTWLRRPELLEGLALTDEQRKLLKEAQAEHNS 3ay0 A 3.05 BS02 ADN A 1 Y177 F203 D223 I224 D251 V252 F273 Y161 F187 D207 I208 D235 V236 F257 2.1.1.228 0002939,0005737,0008033,0008168,0008175,0016740,0030488,0032259,0052906 remove_due_to_license_issue Q58293 21602303 401 PLCLKINKKHGEQTRRILIENNLLNKDYKITSEGNYLYLPIKDVDEDILKSILNIEFELVDKELEEKSFREIISKKYRKEIDEGLISLSYDVVGDLVILQISDEVDEKIRKEIGELAYKLIPCKGVFRRVRELEHLAGENRTLTIHKENGYRLWVDIAKVYFSPRLGGERARIMKKVSLNDVVVDMFAGVGPFSIACKNAKKIYAIDINPHAIELLKKNIKLNKLEHKIIPILSDVREVDVKGNRVIMNLPKFAHKFIDKALDIVEEGGVIHYYTIGKDFDKAIKLFEKKCDCEVLEKRIVKSYAPREYILALDFKINKK 3ay9 A 1.75 BS01 ADP A 1 T13 T14 Y15 G201 G202 E268 K271 R272 S275 G338 G339 R342 D366 T10 T11 Y12 G198 G199 E265 K268 R269 S272 G335 G336 R339 D363 D10 K71 E175 D199 D7 K68 E172 D196 ? 0005524,0140662 remove_due_to_license_issue P0DMV8 21608060 1452 AAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILMG 3aya A 2.0 BS01 GAL C 1 H158 R162 W181 E184 H43 R47 W66 E69 ? 0030246 remove_due_to_license_issue P17931 21949831 2 MPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 3ayc B 1.8 BS01 GAL C 1 H158 R162 N174 W181 E184 H43 R47 N59 W66 E69 ? 0030246 remove_due_to_license_issue P17931 21949831 4 MPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 3ayd A 1.9 BS01 GAL B 1 H158 R162 N174 W181 E184 H43 R47 N59 W66 E69 ? 0030246 remove_due_to_license_issue P17931 21949831 2 MPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 3az8 C 3.1 BS01 S21 D 1 H133 G142 W179 H49 G58 W95 H133 I139 G142 V143 E147 H49 I55 G58 V59 E63 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 231 TSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFAL 3az8 D 3.1 BS01 S21 D 1 H98 E147 F169 L170 F171 H15 E64 F86 L87 F88 H133 I139 G142 V143 E147 H50 I56 G59 V60 E64 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 231 DTSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKIAKLSGVGYVNGKVVINISEMTFA 3az9 C 2.75 BS01 K91 C 1 H98 E147 A150 F169 L170 F171 F226 H14 E63 A66 F85 L86 F87 F142 H133 I139 G142 V143 E147 H49 I55 G58 V59 E63 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 2 TSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFAL 3az9 C 2.75 BS02 K91 D 1 H133 F134 P141 G142 H49 F50 P57 G58 H133 I139 G142 V143 E147 H49 I55 G58 V59 E63 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 1 TSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFAL 3az9 D 2.75 BS01 K91 C 1 H133 P141 G142 V143 H50 P58 G59 V60 H133 I139 G142 V143 E147 H50 I56 G59 V60 E64 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 2 DTSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFA 3az9 D 2.75 BS02 K91 D 1 H98 E147 A150 Q151 F169 L170 F171 H15 E64 A67 Q68 F86 L87 F88 H133 I139 G142 V143 E147 H50 I56 G59 V60 E64 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 1 DTSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFA 3aza A 2.7 BS01 KM0 B 1 H133 F134 G142 H50 F51 G59 H133 I139 G142 V143 E147 H50 I56 G59 V60 E64 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 2 DTSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFALS 3aza B 2.7 BS01 KM0 B 1 H98 E147 A150 Q151 F169 L170 F171 F226 H14 E63 A66 Q67 F85 L86 F87 F138 H133 I139 G142 V143 E147 H49 I55 G58 V59 E63 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 2 TSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKIAKLSGVGYVNGKVVINISEMTFAL 3azb C 2.6 BS01 KM1 D 1 H133 F134 P141 G142 H49 F50 P57 G58 H133 I139 G142 V143 E147 H49 I55 G58 V59 E63 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 1 TSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKSSLGIAKLSGVGYVNGKVVINISEMTFAL 3azb D 2.6 BS01 KM1 D 1 L96 P97 H98 A150 Q151 G154 N167 F169 L170 F171 F226 L13 P14 H15 A67 Q68 G71 N84 F86 L87 F88 F139 H133 I139 G142 V143 E147 H50 I56 G59 V60 E64 4.2.1.59 0006633,0016836 remove_due_to_license_issue Q965D7 21843645 1 DTSIDIEDIKKILPHRYPFLLVDKVIYMQPNKTIIGLKQVSTNEPFFNGHFPQKQIMPGVLQIEALAQLAGILCLKSDDSQKNNLFLFAGVDGVRWKKPVLPGDTLTMQANLISFKIAKLSGVGYVNGKVVINISEMTFA 3b0w A 2.2 BS01 DGX A 1 L287 C320 M365 A368 F377 F388 H479 L23 C56 M101 A104 F113 F124 H215 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=2000nM, Kd=109nM P51449 21733845 1 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQH 3b1m A 1.6 BS02 KRC A 1 G284 C285 F287 R288 S289 L330 M334 I341 L353 M364 K367 G67 C68 F70 R71 S72 L113 M117 I124 L136 M147 K150 ? 0003677,0004879,0005634,0006355 Ki=3.3nM remove_due_to_license_issue P37231 21720019 1 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3b1t A 2.5 BS01 YCL A 1 W347 D350 R374 V469 H471 D473 R639 C645 W311 D314 R338 V433 H435 D437 R600 C606 D350 H471 D473 C645 D314 H435 D437 C606 3.5.3.15 0004668,0005509,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0006338,0016787,0019827,0032991,0036211,0042802,0043687,0045087,0046872,0140794,0140795,0140796,0140797,0140798,0140809,0140810,0140811 remove_due_to_license_issue Q9UM07 21882827 800 GTLIRVTPEQPTHAVCVLGTLTQLDICSSAPTSFSINASPGVVVDITWPLDPGVEVTLTMKAASGSTGDQKVQISYYGPKTPPVKALLYLTAVEISLCADITRTGKQRTWTWGPCGQGAILLVNCDRDNLESSAMDCEDDEVLDSEDLQDMSLMTLSTKTPKDFFTNHTLVLHVARSEMDKVRVFQATCSVVLGPKWPSHYLMVPGGKHNMDFYVEALAFPDTDFPGLITLTISLLDTSNLELPEAVVFQDSVVFRVAPWIMTPNTQPPQEVYACSIFENEDFLKSVTTLAMKAKCKLTICPEEENMDDQWMQDEMEIGYIQAPHKTLPVVFDSPRNRGLKEFPIKRVMGPDFGYVTRGPQTGGISGLDSFGNLEVSPPVTVRGKEYPLGRILFGDSCYPSNDSRQMHQALQDFLSAQQVQAPVKLYSDWLSVGHVDEFLSFVPAPDRKGFRLLLASPRSCYKLFQEQQNEGHGEALLFEGKKQQKIKNILSNKTLREHNSFVERCIDWNRELLKRELGLAESDIIDIPQLFKLKEFSKAEAFFPNMVNMLVLGKHLGIPKPFGPVINGRCCLEEKVCSLLEPLGLQCTFINDFFTYHIRHGEVHCGTNVRRKPFSFKWWNMVP 3b1u A 2.1 BS01 YFF A 1 W347 D350 R374 V469 H471 D473 R639 H640 C645 W312 D315 R339 V434 H436 D438 R604 H605 C610 D350 H471 D473 C645 D315 H436 D438 C610 3.5.3.15 0004668,0005509,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0006338,0016787,0019827,0032991,0036211,0042802,0043687,0045087,0046872,0140794,0140795,0140796,0140797,0140798,0140809,0140810,0140811 remove_due_to_license_issue Q9UM07 21882827 800 GTLIRVTPEQPTHAVCVLGTLTQLDICSSAPETSFSINASPGVVVDITWPLDPGVEVTLTMKAASGSTGDQKVQISYYGPKTPPVKALLYLTAVEISLCADITRTGKQRTWTWGPCGQGAILLVNCDRDNLESSAMDCEDDEVLDSEDLQDMSLMTLSTKTPKDFFTNHTLVLHVARSEMDKVRVFQATCSVVLGPKWPSHYLMVPGGKHNMDFYVEALAFPDTDFPGLITLTISLLDTSNLELPEAVVFQDSVVFRVAPWIMTPNTQPPQEVYACSIFENEDFLKSVTTLAMKAKCKLTICPEEENMDDQWMQDEMEIGYIQAPHKTLPVVFDSPRNRGLKEFPIKRVMGPDFGYVTRGPQTGGISGLDSFGNLEVSPPVTVRGKEYPLGRILFGDSCYPSNDSRQMHQALQDFLSAQQVQAPVKLYSDWLSVGHVDEFLSFVPAPDRKGFRLLLASPRSCYKLFQEQQNEGHGEALLFEGIKKKKQQKIKNILSNKTLREHNSFVERCIDWNRELLKRELGLAESDIIDIPQLFKLKEFSKAEAFFPNMVNMLVLGKHLGIPKPFGPVINGRCCLEEKVCSLLEPLGLQCTFINDFFTYHIRHGEVHCGTNVRRKPFSFKWWNMVP 3b24 A 1.7 BS01 B2J A 1 A55 K58 I96 G97 M98 A40 K43 I81 G82 M83 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.042mM remove_due_to_license_issue Kd=42000nM P07900 21875802 237 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3b25 A 1.75 BS01 B2K A 1 N51 A55 G97 M98 L107 F138 W162 N36 A40 G82 M83 L92 F123 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.86uM remove_due_to_license_issue Kd=8.6E2nM, IC50=9600nM P07900 21875802 1 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3b26 A 2.1 BS01 B2L A 1 A55 G97 M98 N106 L107 F138 Y139 A40 G82 M83 N91 L92 F123 Y124 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.23uM remove_due_to_license_issue IC50=6900nM, Kd=2.3E2nM P07900 21875802 1 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3b27 A 1.5 BS01 B2T A 1 A55 I96 G97 M98 L107 F138 A46 I87 G88 M89 L98 F129 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=6.9uM remove_due_to_license_issue IC50=750nM, Kd=6.9E3nM P07900 21875802 1 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3b28 A 1.35 BS01 B2X A 1 A55 G97 M98 N106 L107 F138 Y139 A40 G82 M83 N91 L92 F123 Y124 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.0034uM remove_due_to_license_issue Kd=3.4nM, IC50=3000nM P07900 21875802 237 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3b2q A 2.1 BS01 ATP A 1 F149 S318 I321 V327 V328 R330 P345 F128 S297 I300 V306 V307 R309 P324 H156 I185 T186 R349 H135 I164 T165 R328 3.6.3.14 0005524,0006754,0015986,0033178,0042777,0046034,0046933,1902600 remove_due_to_license_issue Q60187 19003877 461 IAGPLIFVEKTEPVGYNEIVNIKMGDGTVRRGQVLDSSADIVVVQVFEIFTGETLKLPASVDLLGRILSGSGEPRDGGPRIVPDQLLDINGAAMNPYARLPPKDFIQTGISTIDGTNTLVRGQKLPIFSASGLPHNEIALQIARQASVPGSESAFAVVFAAMGITNEEAQYFMSDFEKTGALERAVVFLNLADDPAVERIVTPRMALTAAEYLAYEHGMHVLVILTDITNYAEALRQMGAARNEVPGRRGYPGYMYTDLATLYERAGIVKGAKGSVTQIPILSMPGDDITHPIPDLSGYITEGQIVVARELHRKGIYPPINVLPSLSRLMNSGIGAGKTREDHKAVSDQMYAGYAEGRDLRGLVAIVGKEALSERDTKFLEFADLFEDKFVRQGWNENRTIEDTLEIGWQILTHLPENQLGRIDNKYIQKYHPAHR 3b2q B 2.1 BS01 ATP A 1 F149 P315 D316 Q325 P345 F129 P286 D287 Q296 P316 H156 I185 T186 R349 H136 I165 T166 R320 3.6.3.14 0005524,0006754,0015986,0033178,0042777,0046034,0046933,1902600 remove_due_to_license_issue Q60187 19003877 461 AGPLIFVEKTEPVGYNEIVNIKMGDGTVRRGQVLDSSADIVVVQVFEGVIFTGETLKLPASVDLLGRILSGSGEPRDGGPRIVPDQLLDINGAAMNPYARLPPKDFIQTGISTIDGTNTLVRGQKLPIFSASGLPHNEIALQIARQASVPGSESAFAVVFAAMGITNEEAQYFMSDFEKTGALERAVVFLNLADDPAVERIVTPRMALTAAEYLAYEHGMHVLVILTDITNYAEALRQMGRGYPGYMYTDLATLYERAGIVKGAKGSVTQIPILSMPGDDITHPIPDLSGYITEGQIVVARELHRKGIYPPINVLPSLSRLMNSGIGAGKTREDHKAVSDQMYAGYAEGRDLRGLVAIVGKEALSERDTKFLEFADLFEDKFVRQGWNENRTIEDTLEIGWQILTHLPENQLGRIDNKYIQKYHPAHRKAK 3b2t A 1.8 BS01 M33 A 1 L487 G490 A515 A567 L633 L24 G27 A49 A101 L153 D626 T628 R630 N631 D644 D146 T148 R150 N151 D164 2.7.10.1 0004672,0005524,0006468 remove_due_to_license_issue P21802 18056630 1996 SEYELPEDPKWEFPRDKLTLGKPLGEGCFGQVVMAEAVGIDPKEAVTVAVKMLKDDATEKDLSDLVSEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLRARRPPQMTFKDLVSCTYQLARGMEYLASQKCIHRDLTARNVLVTENNVMKIADFGLARDINNIDYYKKTTNGRLPVKWMAPEALFDRVYTHQSDVWSFGVLMWEIFTLGGSPYPGIPVEELFKLLKEGHRMDKPANCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRILTLTTNQE 3b2t B 1.8 BS01 M33 B 1 L487 V495 A515 A567 L633 L30 V34 A52 A104 L156 D626 T628 R630 N631 D644 D149 T151 R153 N154 D167 2.7.10.1 0004672,0005524,0006468 remove_due_to_license_issue P21802 18056630 1996 PMLAGVSEYELPEDPKWEFPRDKLTLGKPLFGQVVMAEAVGIDKPKEAVTVAVKMLKDDATEKDLSDLVSEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLRARRPPQMTFKDLVSCTYQLARGMEYLASQKCIHRDLTARNVLVTENNVMKIADFGLARDINNIDYYKKTTNGRLPVKWMAPEALFDRVYTHQSDVWSFGVLMWEIFTLGGSPYPGIPVEELFKLLKEGHRMDKPANCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRILTLT 3b2w A 2.3 BS01 9NH A 1 V259 A271 K273 E288 M292 L300 T316 Y318 M319 G322 L371 A381 D382 F383 V22 A34 K36 E51 M55 L63 T79 Y81 M82 G85 L134 A144 D145 F146 D364 R366 A368 N369 D382 A400 F402 D127 R129 A131 N132 D145 A161 F163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM remove_due_to_license_issue P06239 18083554 601 WEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTA 3b3c A 1.46 BS03 PLU A 1 H97 D117 E151 E152 D179 C227 Y251 H256 H97 D117 E151 E152 D179 C227 Y251 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=105uM remove_due_to_license_issue Q01693 18576673 500 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDATNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 3b3s A 1.18 BS03 LEU A 1 D179 Y225 C227 F248 H256 D179 Y225 C227 F248 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 remove_due_to_license_issue Q01693 18576673 304 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDATNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 3b3w A 1.75 BS03 LEU A 1 D117 E151 E152 D179 C227 H256 D117 E151 E152 D179 C227 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 remove_due_to_license_issue Q01693 18576673 297 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACADHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 3b3x A 2.5 BS01 A33 A 1 S70 S130 T235 G236 A237 R244 Y274 S39 S97 T202 G203 A204 R210 Y239 S70 K73 S130 E166 K234 A237 S39 K42 S97 E133 K201 A204 3.5.2.6 0005886,0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P00808 18515103 300 DDFAKLEEQFDAKLGIFALDTGTNRTVTYRPDERFAFASTIKALTVGVLLQQKSIEDLNQRITYTRDDLVNYNPITEKHVDTGMTLKELADASLRYSDNTAQNLILKQIGGPESLKKELRKIGDEVTNPERFEPELNEVNPGETQDTSTARALATSLQAFALEDKLPSEKRELLIDWMKRNTTGDALIRAGVPEGWEVADKTGAGSYGTRNDIAIIWPPKGDPVVLAVLSSRDKKDAKYDDKLIAEATKVVVKAL 3b4f A 1.89 BS02 TUO A 1 N62 H64 N67 H94 H119 L198 T199 T200 W209 N59 H61 N64 H91 H116 L194 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.2nM remove_due_to_license_issue Ki=7.2nM P00918 18024029 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3b4p A 1.7 BS01 3B4 A 1 L53 H73 F81 W84 E140 Q147 L45 H65 F73 W76 E132 Q139 ? 0017000 Kd=4uM remove_due_to_license_issue Q396C9 19053436 500 NTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLPS 3b4p B 1.7 BS01 3B4 B 1 L53 H73 F81 W84 E140 Q147 L46 H66 F74 W77 E133 Q140 ? 0017000 Kd=4uM remove_due_to_license_issue Q396C9 19053436 500 ENTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLPS 3b50 A 1.4 BS01 SLB A 1 N10 D49 F65 E67 R70 R127 R147 F170 N187 Q214 N10 D49 F65 E67 R70 R127 R147 F170 N187 Q214 ? 0030288,0042597,0055085 Kd=28nM remove_due_to_license_issue P44542 17947229 311 ADYDLKFGMNAGTSSNEYKAAEMFAKEVKEKSQGKIEISLYPSSQLGDDRAMLKQLKDGSLDFTFAESARFQLFYPEAAVFALPYVISNYNVAQKALFDTEFGKDLIKKMDKDLGVTLLSQAYNGTRQTTSNRAINSIADMKGLKLRVPNAATNLAYAKYVGASPTPMAFSEVYLALQTNAVDGQENPLAAVQAQKFYEVQKFLAMTNHILNDQLYLVSNETYKELPEDLQKVVKDAAENAAKYHTKLFVDGEKDLVTFFEKQGVKITHPDLVPFKESMKPYYAEFVKQTGQKGESALKQIEAINPKGEA 3b5j A 2.0 BS01 12D A 1 Y477 I484 G505 S506 G507 K508 S509 T510 Y13 I20 G41 S42 G43 K44 S45 T46 ? 0005524,0016887 Kd=2.1uM remove_due_to_license_issue P08716 18155559 708 HHDITFRNIRFRYKPDSPVILDNINLSIKQGEVIGIVGRAGSGKSTLTKLIQRFYIPENGQVLIDGHDLALADPNWLRRQVGVVLQDNVLLNRSIIDNISLANPGMSVEKVIYAAKLAGAHDFISELREGYNTIVGEQGAGLSGGQRQRIAIARALVNNPKILIFDEATSALDYESEHVIMRNMHKICKGRTVIIIAHRLSTVKNADRIIVMEKGKIVEQGKHKELLSEPESLYSYLYQLQSD 3b5r A 1.8 BS01 B5R A 1 L704 N705 L707 G708 W741 M742 M745 V746 M749 F764 T877 M895 V903 L34 N35 L37 G38 W71 M72 M75 V76 M79 F94 T207 M225 V233 ? remove_due_to_license_issue Ki=1.7nM P10275 18805694 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 3b65 A 1.8 BS01 3B6 A 1 L704 N705 L707 G708 W741 M742 M745 V746 M749 F764 T877 M895 V903 L34 N35 L37 G38 W71 M72 M75 V76 M79 F94 T207 M225 V233 ? remove_due_to_license_issue P10275 18805694 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 3b66 A 1.65 BS01 B66 A 1 L704 N705 G708 W741 M742 M745 V746 M749 F764 T877 M895 L34 N35 G38 W71 M72 M75 V76 M79 F94 T207 M225 ? remove_due_to_license_issue P10275 18805694 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 3b67 A 1.9 BS01 B67 A 1 L704 N705 Q711 W741 M742 M745 V746 M749 F764 T877 M895 I899 L34 N35 Q41 W71 M72 M75 V76 M79 F94 T207 M225 I229 ? remove_due_to_license_issue P10275 18805694 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 3b68 A 1.9 BS01 B68 A 1 L704 N705 L707 G708 Q711 W741 M742 M745 V746 M749 F764 T877 M895 I899 V903 L34 N35 L37 G38 Q41 W71 M72 M75 V76 M79 F94 T207 M225 I229 V233 ? remove_due_to_license_issue Ki=4nM P10275 18805694 1 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 3b7i A 1.75 BS03 PLU A 1 H97 D117 E151 E152 C227 F248 H256 H97 D117 E151 E152 C227 F248 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=1.5uM remove_due_to_license_issue Q01693 18576673 500 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACADHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 3b7j A 2.4 BS01 JUG B 1 I64 F109 R110 I111 P112 I57 F102 R103 I104 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 18565285 163 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3b7r L 1.811 BS02 BIR L 1 Q136 Y267 G268 G269 E271 N291 V292 H295 E296 E318 Y378 Y383 R563 K565 Q136 Y267 G268 G269 E271 N291 V292 H295 E296 E318 Y378 Y383 R563 K565 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 Ki=20nM remove_due_to_license_issue P09960 18804029 1001 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3b7u X 1.9 BS02 KEL X 1 Y267 G268 G269 E271 V292 H295 E296 H299 E318 Y378 Y383 R563 K565 Y267 G268 G269 E271 V292 H295 E296 H299 E318 Y378 Y383 R563 K565 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=5nM, Ki=10nM P09960 18804029 707 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3b8q A 2.75 BS01 900 A 1 L840 V848 A866 K868 E885 L889 T916 C919 L1035 C1045 D1046 F1047 L23 V31 A49 K51 E68 L72 T99 C102 L168 C178 D179 F180 D1028 A1030 R1032 N1033 D1046 D161 A163 R165 N166 D179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=0.480000nM P35968 18324761 501 ERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3b8r A 2.7 BS01 887 A 1 L840 V848 A866 K868 E885 L889 T916 C919 L1035 C1045 D1046 F1047 L23 V26 A44 K46 E63 L67 T94 C97 L163 C173 D174 F175 D1028 A1030 R1032 N1033 D1046 D156 A158 R160 N161 D174 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=0.600000nM P35968 18324759 201 ERLPYDASKWEFPRDRLKLGKPLGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3b8z A 1.4 BS05 294 A 1 T378 L379 G380 H410 E411 H414 H420 S441 L443 T444 S445 I446 T115 L116 G117 H147 E148 H151 H157 S178 L180 T181 S182 I183 3.4.24.- 0004222,0006508,0008237 ic50=0.29uM remove_due_to_license_issue Q9UNA0 17991750 801 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3b92 A 2.0 BS02 440 A 1 G349 E398 L401 H405 E406 H409 H415 P437 A439 V440 G134 E183 L186 H190 E191 H194 H200 P222 A224 V225 3.4.24.86 0004222,0006508,0008237 Ki=10nM remove_due_to_license_issue Ki=10nM P78536 18054488 501 ADPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYVGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3b9g A 1.4 BS02 IMH A 1 N12 D14 D40 M164 E184 N186 W250 D251 N12 D14 D40 M164 E184 N186 W250 D251 D10 D15 D40 W83 T137 W185 N186 W250 D251 D10 D15 D40 W83 T137 W185 N186 W250 D251 3.2.2.1 0005829,0006139,0006152,0008477,0016798,0016799,0046872 Ki=19uM remove_due_to_license_issue Q9GPQ4 18519562 501 SAKNVVLDHDGNLDDFVAMVLLASNTEKVRLIGALCTDADCFVENGFNVTGKIMCLMHNNMNLPLFPIGKSAATAVNPFPKEWRCLAKNMDDMPILNIPENVELWDKIKAENEKYEGQQLLADLVMNSEEKVTICVTGPLSNVAWCIDKYGEKFTSKVEECVIMGGAVDVRGNVFLPSTDGTAEWNIYWDPASAKTVFGCPGLRRIMFSLDSTNTVPVRSPYVQRFGEQTNFLLSILVGTMWAMGGGYAWDALTAAYVVDQKVANVDPVPIDVVVDKQPNEGATVRTDAENYPLTFVARNPEAEFFLDMLLRSARAC 3b9s A 1.8 BS01 RW1 A 1 P1 M2 V106 P1 M2 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 18794110 118 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3b9s B 1.8 BS01 RW1 A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 18794110 118 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3b9s B 1.8 BS02 RW1 B 1 P1 M2 V106 P1 M2 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 18794110 116 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3bb1 A 2.8 BS01 GNP A 1 G49 V50 G51 K52 S53 S54 S68 P69 S72 G96 H163 E210 N211 G48 V49 G50 K51 S52 S53 S67 P68 S71 G95 H162 E204 N205 3.6.5.- 0005525,0006886,0009707,0015450 remove_due_to_license_issue Q41009 18400179 281 ASQQQTVRGWSGINTFAPATQTKLLELLGNLKQEDVNSLTILVMGKGGVGKSSTVNSIIGERVVSISPFQSEGPRPVMVSRSRAGFTLNIIDTPGLIEGGYINDMALNIIKSFLLDKTIDVLLYVDRLDAYRVDNLDKLVAKAITDSFGKGIWNKAIVALTHAQFSPPDGLPYDEFFSKRSEALLQVVRSGASLKSDIPVVLIENSGRCNKNDSDEKVLPNGIAWIPHLVQTITEVALNKSESIFVDKNLID 3bb1 A 2.8 BS02 GNP B 1 Y132 R133 P169 Y131 R132 P168 3.6.5.- 0005525,0006886,0009707,0015450 remove_due_to_license_issue Q41009 18400179 281 ASQQQTVRGWSGINTFAPATQTKLLELLGNLKQEDVNSLTILVMGKGGVGKSSTVNSIIGERVVSISPFQSEGPRPVMVSRSRAGFTLNIIDTPGLIEGGYINDMALNIIKSFLLDKTIDVLLYVDRLDAYRVDNLDKLVAKAITDSFGKGIWNKAIVALTHAQFSPPDGLPYDEFFSKRSEALLQVVRSGASLKSDIPVVLIENSGRCNKNDSDEKVLPNGIAWIPHLVQTITEVALNKSESIFVDKNLID 3bb1 B 2.8 BS01 GNP A 1 Y132 R133 P169 Y124 R125 P161 3.6.5.- 0005525,0006886,0009707,0015450 remove_due_to_license_issue Q41009 18400179 281 VRGWSGINTFAPATQTKLLELLGNLKQEDVNSLTILVMGKGGVGKSSTVNSIIGERVVSISPFQSGPRPVMVSRSRAGFTLNIIDTPGLIEGGYINDMALNIIKSFLLDKTIDVLLYVDRLDAYRVDNLDKLVAKAITDSFGKGIWNKAIVALTHAQFSPPDGLPYDEFFSKRSEALLQVVRSGASLASDIPVVLIENSGRCNSDEKVLPNGIAWIPHLVQTITEVALNKSESIFVDKNLIDG 3bb1 B 2.8 BS02 GNP B 1 G49 G51 K52 S53 S54 P69 S72 H163 E210 N211 G42 G44 K45 S46 S47 P62 S65 H155 E197 N198 3.6.5.- 0005525,0006886,0009707,0015450 remove_due_to_license_issue Q41009 18400179 281 VRGWSGINTFAPATQTKLLELLGNLKQEDVNSLTILVMGKGGVGKSSTVNSIIGERVVSISPFQSGPRPVMVSRSRAGFTLNIIDTPGLIEGGYINDMALNIIKSFLLDKTIDVLLYVDRLDAYRVDNLDKLVAKAITDSFGKGIWNKAIVALTHAQFSPPDGLPYDEFFSKRSEALLQVVRSGASLASDIPVVLIENSGRCNSDEKVLPNGIAWIPHLVQTITEVALNKSESIFVDKNLIDG 3bbb C 1.3 BS01 DA C 1 K12 Y52 V112 K8 Y48 V108 K12 Y52 N115 H118 E129 K8 Y48 N111 H114 E125 2.7.13.3,2.7.4.6 0000155,0000160,0001726,0003677,0003713,0004550,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 remove_due_to_license_issue P22392 19435876 153 ERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbb C 1.3 BS02 DG C 1 L55 F60 L64 T94 L51 F56 L60 T90 K12 Y52 N115 H118 E129 K8 Y48 N111 H114 E125 2.7.13.3,2.7.4.6 0000155,0000160,0001726,0003677,0003713,0004550,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 remove_due_to_license_issue P22392 19435876 154 ERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbf A 1.7 BS01 GDP A 1 K12 L55 F60 L64 R88 T94 V112 G113 N115 K11 L54 F59 L63 R87 T93 V111 G112 N114 K12 Y52 N115 H118 E129 K11 Y51 N114 H117 E128 2.7.13.3,2.7.4.6 0000155,0000160,0001726,0003677,0003713,0004550,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 remove_due_to_license_issue P22392 19435876 160 ANLERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbf B 1.7 BS01 GDP B 1 K12 L55 F60 R88 T94 V112 G113 N115 K11 L54 F59 R87 T93 V111 G112 N114 K12 Y52 N115 H118 E129 K11 Y51 N114 H117 E128 2.7.13.3,2.7.4.6 0000155,0000160,0001726,0003677,0003713,0004550,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 remove_due_to_license_issue P22392 19435876 160 ANLERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbt B 2.8 BS01 FMM B 1 V707 A724 K726 M747 T771 L825 T835 D836 F837 V25 A42 K44 M63 T87 L141 T151 D152 F153 D818 A820 R822 N823 D836 D134 A136 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=54nM, IC50=>1000nM Q15303 18334220 91 AQLRILKETELKRVKVLGSGAFGTVYKGIWVPEGETVKIPVAIKILNEGPKANVEFMDEALIMASMDHPHLVRLLGVCLSPTIQLVTQLMPHGCLLEYVHEHKDNIGSQLLLNWCVQIAKGMMYLEERRLVHRDLAARNVLVKSPNHVKITDFGLARLLPIKWMALECIHYRKFTHQSDVWSYGVTIWELMTFGGKPYDGIPTREIPDLLEKGERLPQPPICTIDVYMVMVKCWMIDADSRPKFKELAAEFSRMARDPQRYLVIQDDRMKLPSP 3bc3 A 2.2 BS01 OPT A 1 Q19 A25 G61 E63 G67 G68 L69 M70 A135 L144 M161 D162 H163 W189 A214 Q19 A25 G61 E63 G67 G68 L69 M70 A135 L144 M161 D162 H163 W184 A209 Q19 C25 H163 N187 Q19 C25 H163 N182 3.4.22.15 0006508,0008234 Ki=0.155uM remove_due_to_license_issue P07711 18278855 300 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3bc4 A 1.82 BS01 LLG A 1 D25 G27 V82 D25 G27 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.5uM remove_due_to_license_issue P04587 18720485 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 3bc4 A 1.82 BS02 LLG A 2 G48 I50 G52 G48 I50 G52 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.5uM remove_due_to_license_issue P04587 18720485 2502 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 3bc5 A 2.27 BS01 ZAA A 1 F282 G284 C285 I341 F360 F363 M364 H449 Y473 F70 G72 C73 I129 F148 F151 M152 H237 Y259 ? 0003677,0004879,0005634,0006355 ic50=0.005uM remove_due_to_license_issue EC50=4nM, IC50=5nM P37231 19201606 1 MQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTSPFVIYDMNSLMMGEDKIKFKHKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTEMSLHPLLQEIYKDLY 3bcn A 2.85 BS01 E64 A 1 G23 C25 W26 G65 G66 N156 H157 G23 C25 W26 G65 G66 N156 H157 Q19 C25 H157 N173 Q19 C25 H157 N173 3.4.22.- 0005576,0006508,0008234 remove_due_to_license_issue A5YVK8 18167146 214 LPEHVDWRAKGAVIPLKNQGKCGSCWAFSTVTTVESINQIRTGNLISLSEQQLVDCSKKNHGCKGGYFDRAYQYIIANGGIDTEANYPYKAFQGPCRAAKKVVRIDGCKGVPQCNENALKNAVASQPSVVAIDASSKQFQHYKGGIFTGPCGTKLNHGVVIVGYGKDYWIVRNSWGRHWGEQGYTRMKRVGGCGLCGIARLPFYPTKAA 3bcs A 2.0 BS01 CJB A 1 G135 L136 D283 N284 H377 N484 E672 A673 S674 G675 G124 L125 D266 N267 H351 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=6100nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3be2 A 1.75 BS01 RAJ A 1 V848 A866 E885 T916 F918 C919 H1026 L1035 I1044 C1045 D1046 F1047 V34 A49 E68 T99 F101 C102 H159 L168 I177 C178 D179 F180 D1028 A1030 R1032 N1033 D1046 D161 A163 R165 N166 D179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=2nM remove_due_to_license_issue IC50=2nM P35968 18324761 501 EHAERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDTCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHH 3be9 A 2.0 BS01 P04 A 1 V45 R47 V53 I66 K68 F113 V116 M163 I174 D175 V40 R42 V48 I61 K63 F108 V111 M158 I169 D170 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=24nM remove_due_to_license_issue Ki=24nM P28523 18055206 501 MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNAYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 3bea A 2.02 BS01 IXH A 1 L588 G589 A614 K616 T663 Y665 C666 G669 L785 F797 A800 R801 L42 G43 A68 K70 T117 Y119 C120 G123 L174 F186 A189 R190 D778 A780 R782 N783 D796 N805 N814 D167 A169 R171 N172 D185 N194 N203 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=0.007uM remove_due_to_license_issue P07333,Q02763 18342505 923 QVRWKIIESYEGNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKSRVLSTLSTRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGNARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQAQEDRRER 3bel A 2.3 BS01 POX A 1 A743 K745 C775 R776 L788 T790 M793 D800 L844 T854 D855 F856 A38 K40 C64 R65 L77 T79 M82 D89 L133 T143 D144 F145 D837 A839 R841 N842 D855 D126 A128 R130 N131 D144 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.014uM remove_due_to_license_issue IC50=14nM P00533 18508264 1 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPVKIPVAIKELKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERNFYRALMVVDADE 3bep A 1.92 BS01 dna D 0 E8 L11 K12 E8 L11 K12 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 remove_due_to_license_issue P0A988 18191219 11 ~ 24 MKFTVEREHLLKPLQQVSGPLGGRPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 3bep B 1.92 BS01 dna C 0 H148 K198 H148 K198 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 remove_due_to_license_issue P0A988 18191219 2 ~ 11 MKFTVEREHLLKPLQQVSGPLGGRPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 3bet A 1.85 BS02 CTF A 1 H94 V121 F131 L198 T199 T200 P201 P202 H92 V119 F128 L195 T196 T197 P198 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=1.5uM remove_due_to_license_issue IC50=1500nM, Ki=1470nM P00918 18260615 264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3bex A 1.51 BS01 PAU A 1 E101 V102 G103 D105 R106 E104 V105 G106 D108 R109 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 Kd=2.7uM remove_due_to_license_issue Q9WZY5 18186650 248 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bex A 1.51 BS02 PAU B 1 K162 T179 K165 T182 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 Kd=2.7uM remove_due_to_license_issue Q9WZY5 18186650 248 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bex B 1.51 BS01 PAU A 1 K162 T179 K165 T182 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 Kd=2.7uM remove_due_to_license_issue Q9WZY5 18186650 248 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bex B 1.51 BS02 PAU B 1 E101 V102 G103 D105 R106 T131 E104 V105 G106 D108 R109 T134 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 Kd=2.7uM remove_due_to_license_issue Q9WZY5 18186650 248 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bf1 A 2.3 BS01 ADP A 1 T10 H11 R27 G127 T128 F150 Q217 T13 H14 R30 G130 T131 F153 Q220 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 remove_due_to_license_issue Q9WZY5 18186650 247 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bf1 A 2.3 BS04 ADP D 1 V32 F33 V35 F36 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 remove_due_to_license_issue Q9WZY5 18186650 247 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bf1 B 2.3 BS02 ADP B 1 T10 H11 R27 T128 F150 Q217 T13 H14 R30 T131 F153 Q220 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 remove_due_to_license_issue Q9WZY5 18186650 247 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bf1 B 2.3 BS04 ADP E 1 V32 F33 V35 F36 2.7.1.33 0004594,0005524,0005737,0015937,0016301,0043169,0046872 remove_due_to_license_issue Q9WZY5 18186650 247 MDPMYLLVDVGNTHSVFSITEDGKTFRRWRLSTGVFQTEDELFSHLHPLLGDAMREIKGIGVASVVPTQNTVIERFSQKYFHISPIWVKAKNGCVKWNVKNPSEVGADRVANVVAFVKEYGKNGIIIDMGTATTVDLVVNGSYEGGAILPGFFMMVHSLFRGTAKLPLVEVKPADFVVGKDTEENIRLGVVNGSVYALEGIIGRIKEVYGDLPVVLTGGQSKIVKDMIKHEIFDEDLTIKGVYHFCFG 3bft A 2.27 BS01 S2P A 1 Y61 T91 R96 G141 S142 T143 E193 M196 Y59 T89 R94 G139 S140 T141 E191 M194 ? 0015276,0016020 Ki=323nM remove_due_to_license_issue P19491 18269227 1009 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3bfu A 1.95 BS01 R2P A 1 Y61 T91 R96 G141 S142 T143 E193 M196 Y61 T91 R96 G141 S142 T143 E193 M196 ? 0015276,0016020 Ki=531nM remove_due_to_license_issue P19491 18269227 264 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 3bgb A 1.9 BS01 LJG B 1 D25 G27 D30 I50 P81 I84 D25 G27 D30 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18760609 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3bgb B 1.9 BS01 LJG B 1 D25 G27 A28 D30 V32 G48 G49 I50 P81 D25 G27 A28 D30 V32 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.9uM remove_due_to_license_issue P04587 18760609 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3bgc A 1.8 BS01 LJH A 1 D25 G27 A28 D30 G48 I50 V82 I84 D25 G27 A28 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=9.6uM remove_due_to_license_issue P04587 18760609 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3bgc B 1.8 BS01 LJH A 1 D25 A28 D30 V32 G48 G49 I50 V82 I84 D25 A28 D30 V32 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18760609 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3bgl A 2.225 BS01 RID A 1 R590 S661 S684 D690 K692 R150 S221 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=4.5nM remove_due_to_license_issue P04035 18155906 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3bgl A 2.225 BS02 RID B 1 E559 C561 K735 A751 N755 L853 A856 H861 E119 C121 K295 A311 N315 L413 A416 H421 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=4.5nM remove_due_to_license_issue P04035 18155906 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3bgl B 2.225 BS01 RID A 1 E559 C561 S565 K735 A751 L853 A856 L857 E119 C121 S125 K295 A311 L413 A416 L417 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=4.5nM remove_due_to_license_issue P04035 18155906 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3bgl B 2.225 BS02 RID B 1 R590 V683 S684 D690 K692 R150 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 ic50=4.5nM remove_due_to_license_issue P04035 18155906 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3bgp A 2.8 BS01 VX1 A 1 F49 V52 A65 K67 L120 L174 D186 F17 V20 A33 K35 L88 L142 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue Ki=91nM P11309 18290603 314 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3bgq A 2.0 BS01 VX2 A 1 L44 F49 A65 K67 I104 E121 R122 L174 I185 D186 L12 F17 A33 K35 I72 E89 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=11nM remove_due_to_license_issue Ki=11nM P11309 18290603 314 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3bgs A 2.099 BS01 DIH A 1 A116 A117 G118 F200 E201 V217 M219 N243 A116 A117 G118 F200 E201 V217 M219 N243 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 Ki=380pM remove_due_to_license_issue P00491 18154341 301 MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPD 3bgz A 2.4 BS01 VX3 A 1 L44 G45 F49 V52 K67 I104 I185 D186 L12 G13 F17 V20 K35 I67 I148 D149 D167 K169 N172 D186 L193 T204 D130 K132 N135 D149 L156 T167 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=0.55uM remove_due_to_license_issue IC50=550nM, Ki=550nM P11309 18290603 314 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGERVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3bh3 A 2.1 BS01 PNH A 1 R30 Y75 K116 R30 Y75 K116 4.1.1.4 0016829,0016831,0047602 remove_due_to_license_issue Q7NSA6 19458715 247 MKQQEVRQRAFAMPLTSPAFPPGPYRFVNREYMIITYRTDPAAIEAVLPEPLQMAEPVVRYEFIRMPDSTGFGDYSESGQVIPVTFRGERGSYTLAMFLDDQPPLAGGRELWGFPKKAGKPRLEVHQDTLVGSLDFGPVRIATGTMGYKYEALDRSALLASLAEPNFLLKIIPHVDGSPRICELVRYHTTDVAIKGAWSAPGSLELHPHALAPVAALPVLEVLSARHFVCDLTLDLGTVVFDYL 3bhx A 1.6 BS04 BHX A 1 R210 N257 D387 E424 E425 D453 G518 N519 Y552 H553 K699 Y700 R156 N203 D333 E370 E371 D399 G464 N465 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.7nM remove_due_to_license_issue Q04609 18234225 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3bi0 A 1.67 BS04 BIX A 1 R210 N257 D387 E424 E425 D453 G518 N519 R534 Y552 H553 K699 Y700 R156 N203 D333 E370 E371 D399 G464 N465 R480 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=14nM remove_due_to_license_issue Q04609 18234225 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3bi1 A 1.5 BS04 3BI A 1 K207 R210 N257 D387 E424 E425 D453 R463 G518 N519 R534 R536 K539 W541 N544 F546 Y552 H553 K699 Y700 K153 R156 N203 D333 E370 E371 D399 R409 G464 N465 R480 R482 K485 W487 N490 F492 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.12nM remove_due_to_license_issue Q04609 18234225 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3bi6 A 2.2 BS01 396 A 1 I305 A326 K328 V360 N376 E377 Y378 C379 G381 G382 F433 D463 I13 A34 K36 V68 N84 E85 Y86 C87 G89 G90 F141 D151 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 ic50=15nM remove_due_to_license_issue IC50=15nM P30291 18191399 901 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVLL 3biz A 2.2 BS01 61E A 1 I305 V313 A326 K328 V360 N376 E377 Y378 C379 G382 F433 D463 I13 V17 A30 K32 V61 N77 E78 Y79 C80 G83 F134 D144 D426 K428 D127 K129 2.7.10.2 0004672,0005524,0006468 ic50=58nM remove_due_to_license_issue IC50=58nM P30291 18191399 576 SRYTTEFHELEKIGSSVFKCVKRLDGCIYAIKRSKKPSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVL 3bjc A 2.0 BS03 WAN A 1 H613 A783 F786 M816 Q817 F820 H79 A249 F252 M267 Q268 F271 3.1.4.35 0004112,0004114,0004115,0004117,0005515,0005829,0007165,0008081,0010613,0010749,0016787,0019933,0030553,0042098,0042130,0046068,0046069,0046872,0047555,0048101,0048599,0055118,0055119,0060282 ic50=0.11uM remove_due_to_license_issue IC50=110nM O76074 18346713 901 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 3bki P 1.87 BS01 FQX P 1 Y16 Y61 P89 L90 T91 R96 E193 M196 Y220 Y12 Y57 P85 L86 T87 R92 E189 M192 Y216 ? 0015276,0016020 ic50=7.6uM remove_due_to_license_issue P19491 18754610 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3bkk A 2.17 BS03 KAF A 1 Q281 H353 A354 S355 A356 H383 E384 H387 F391 E411 K511 F512 H513 V518 Y520 Y523 Q244 H316 A317 S318 A319 H346 E347 H350 F354 E374 K474 F475 H476 V481 Y483 Y486 H353 A354 H383 E384 H387 E411 H513 Y523 H316 A317 H346 E347 H350 E374 H476 Y486 3.4.15.1 0006508,0008237,0008241,0016020 Ki=0.83uM remove_due_to_license_issue P12821 18457420 704 VTDEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTP 3bkl A 2.18 BS03 KAW A 1 H353 A354 S355 A356 H383 E384 H387 F391 E411 D415 F457 K511 F512 H513 V518 Y520 Y523 H313 A314 S315 A316 H343 E344 H347 F351 E371 D375 F415 K469 F470 H471 V476 Y478 Y481 H353 A354 H383 E384 H387 E411 H513 Y523 H313 A314 H343 E344 H347 E371 H471 Y481 3.4.15.1 0006508,0008237,0008241,0016020 Ki=0.679uM remove_due_to_license_issue P12821 18457420 800 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSASMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPN 3bl0 A 1.9 BS02 BL0 A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=121nM remove_due_to_license_issue P00918 18162396 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3bl1 A 2.1 BS02 BL1 A 1 H64 H94 H119 F131 V143 L198 T199 W209 H61 H91 H116 F127 V139 L194 T195 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2520nM remove_due_to_license_issue Kd=300nM, Ki=2520nM P00918 18374572 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3bl7 A 2.31 BS01 DD1 A 1 K142 Y143 W175 E185 D205 L206 S272 K94 Y95 W127 E137 D157 L158 S224 3.6.1.59 0000290,0016787 ic50=7.62nM remove_due_to_license_issue IC50=0.030000nM, EC50=4.0nM Q96C86 18839960 901 LPFSGFRLQKVLRESARDKIIFLHGKVNEEDAVVILEKTPFQVEQVAQLLTGSPELQLQFSNDIYSTYHLFPPRQLNDVKTTVVYPATEKHLQKYLRQDLRLIRETGDDYRNITLPHLESQSLSIQWVYNILDKKAEADRIVFENPDPSDGFVLIPDLKWNQQQLDDLYLIAICHRRGIRSLRDLTPEHLPLLRNILHQGQEAILQRYRMKGDHLRVYLHYLPSYYHLHVHFTALGFEAPGSGVERAHLLAEVIENLECDPRHYQQRTLTFALRADDPLLKLLQEA 3bl9 A 1.8 BS01 DD2 A 1 R54 F63 K142 Y143 W175 E185 D205 L206 R13 F22 K94 Y95 W127 E137 D157 L158 3.6.1.59 0000290,0016787 ic50=43.94nM remove_due_to_license_issue IC50=43.94nM, EC50=67nM Q96C86 18839960 901 LPFSGFRLQKVLRESARDKIIFLHGKVNEEDAVVILEKTPFQVEQVAQLLTGSPELQLQFSNDIYSTYHLFPPRQLNDVKTTVVYPATEKHLQKYLRQDLRLIRETGDDYRNITLPHLESQSLSIQWVYNILDKKAEADRIVFENPDPSDGFVLIPDLKWNQQQLDDLYLIAICHRRGIRSLRDLTPEHLPLLRNILHQGQEAILQRYRMKGDHLRVYLHYLPSYYHLHVHFTALGFEAPGSGVERAHLLAEVIENLECDPRHYQQRTLTFALRADDPLLKLLQEA 3bla A 2.6 BS01 DD3 A 1 Y143 W175 E185 D205 L206 Y273 Y95 W127 E137 D157 L158 Y225 3.6.1.59 0000290,0016787 remove_due_to_license_issue Q96C86 18839960 1 LPFSGFRLQKVLRESARDKIIFLHGKVNEEDAVVILEKTPFQVEQVAQLLTGSPELQLQFSNDIYSTYHLFPPRQLNDVKTTVVYPATEKHLQKYLRQDLRLIRETGDDYRNITLPHLESQSLSIQWVYNILDKKAEADRIVFENPDPSDGFVLIPDLKWNQQQLDDLYLIAICHRRGIRSLRDLTPEHLPLLRNILHQGQEAILQRYRMKGDHLRVYLHYLPSYYHLHVHFTALGFEAPGSGVERAHLLAEVIENLECDPRHYQQRTLTFALRADDPLLKLLQEA 3bla B 2.6 BS01 DD3 B 1 W175 E185 D205 L206 W128 E138 D158 L159 3.6.1.59 0000290,0016787 remove_due_to_license_issue Q96C86 18839960 2 VRLPFSGFRLQKVLRESARDKIIFLHGKVNEDAVVILEKTPFQVEQVAQLLTGSPELQLQFSNDIYSTYHLFPPRQLNDVKTTVVYPATEKHLQKYLRQDLRLIRETGDDYRNITLPHLESQSLSIQWVYNILDKKAEADRIVFENPDPSDGFVLIPDLKWNQQQLDDLYLIAICHRRGIRSLRDLTPEHLPLLRNILHQGQEAILQRYRMKGDHLRVYLHYLPSYYHLHVHFTALGFEAPGSGVERAHLLAEVIENLECDPRHYQQRTLTFALRADDPLLKLLQEAQQ 3blr A 2.8 BS01 CPB A 1 I25 F30 A46 K48 F103 C106 N154 L156 D167 I19 F24 A40 K42 F87 C90 N138 L140 D151 D149 K151 A153 N154 D167 T191 D133 K135 A137 N138 D151 T171 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=20nM, Kd=6.4nM, Ki=3.0nM P50750 18566585 940 SVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKG 3bls A 2.3 BS01 APB A 1 S64 Y150 T316 G317 A318 N346 R349 S61 Y147 T313 G314 A315 N343 R346 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=7300nM P00811 9819201 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNAL 3blt A 2.2 BS01 PSY A 1 D356 C403 R404 A405 G406 V407 G408 R409 T410 Q446 D170 C217 R218 A219 G220 V221 G222 R223 T224 Q260 E290 W354 D356 H402 C403 R409 T410 E104 W168 D170 H216 C217 R223 T224 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P15273 18528979 501 SPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCRRQTAVRADLNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGLGDGIMADMYTLTIREAGQKTISVPVVHVGNWPDQTAVSSEVTKALASLVDQTAETKRNMYESKGSSAVADDSKLRPVIHCRAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS 3blu A 2.0 BS01 PVS A 1 F229 D356 C403 R404 A405 G406 V407 G408 R409 T410 Q446 F43 D170 C217 R218 A219 G220 V221 G222 R223 T224 Q260 E290 W354 D356 H402 C403 R409 T410 E104 W168 D170 H216 C217 R223 T224 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P15273 18528979 501 SPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCRRQTAVRADLNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGLGDGIMADMYTLTIREAGQKTISVPVVHVGNWPDQTAVSSEVTKALASLVDQTAETKRNMYESKGSSAVADDSKLRPVIHCRAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS 3bm6 A 2.1 BS01 C9P A 1 S64 Q120 Y150 N152 Y221 G317 A318 T319 S61 Q117 Y147 N149 Y218 G314 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 20452208 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3bm8 A 2.7 BS01 PSY A 1 F229 C403 R404 A405 G406 V407 G408 R409 Q446 F43 C217 R218 A219 G220 V221 G222 R223 Q260 E290 W354 A356 H402 C403 R409 T410 E104 W168 A170 H216 C217 R223 T224 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P15273 18528979 501 SPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCRRQTAVRADLNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGLGDGIMADMYTLTIREAGQKTISVPVVHVGNWPAQTAVSSEVTKALASLVDQTAETKRNMYESKGSSAVADDSKLRPVIHCRAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS 3bm9 A 1.6 BS01 BXZ A 1 N51 A55 K58 D93 I96 G97 M98 F138 T184 N35 A39 K42 D77 I80 G81 M82 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.19uM remove_due_to_license_issue IC50=190nM P07900 18197612 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3bmn A 1.98 BS02 AX3 A 1 S95 F97 Y174 P210 S94 F96 Y157 P193 R14 D161 Y174 K178 R13 D144 Y157 K161 ? 0000166,0016491,0047040 Ki>35uM remove_due_to_license_issue O76290 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmo A 1.6 BS02 AX4 A 1 S95 F97 Y174 L209 P210 W221 S94 F96 Y161 L196 P197 W208 R14 D161 Y174 K178 R13 D148 Y161 K165 ? 0000166,0016491,0047040 Ki=5.4uM remove_due_to_license_issue O76290 19916554 274 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQKGTTSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq A 1.7 BS02 AX5 A 1 S95 F97 Y174 L208 P210 M213 S94 F96 Y159 L193 P195 M198 R14 D161 Y174 K178 R13 D146 Y159 K163 ? 0000166,0016491,0047040 Ki=3.2uM remove_due_to_license_issue O76290 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQKGSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmy A 1.6 BS01 CXZ A 1 N51 A55 D93 I96 G97 M98 F138 T184 N41 A45 D83 I86 G87 M88 F128 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.03uM remove_due_to_license_issue IC50=30nM P07900 18197612 1 QPMEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3bpc A 1.85 BS01 KDA C 1 S91 R95 S97 R101 remove_due_to_license_issue 18272175 1 DIVMSQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTITSVQAEDLAVYYCKQSYNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSEGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 3bpc A 1.85 BS02 KDB C 1 N30A R30C N31 R33 remove_due_to_license_issue 18272175 2 DIVMSQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTITSVQAEDLAVYYCKQSYNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSEGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 3bpc B 1.85 BS01 KDA C 1 Y33 R52 N52D E100A Y33 R52 N56 E107 remove_due_to_license_issue 18272175 1 EVKLVESGGGLVQSGGSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKANGYTTEYSPSVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDHDGYYERFSYWGQGTLVTVSAAKTTPPSVYPLAPSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVP 3bpr A 2.8 BS01 OLP A 1 A617 F673 M674 K675 G677 D678 M730 A43 F88 M89 K90 G92 D93 M145 D723 A725 R727 N728 D741 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q12866 19028587 900 NKLEDVVIDRNLLILGKILGEGEFGSVMEGNLKQEDGTSLKVAVKTMKREIEEFLSEAACMKDFSHPNVIRLLGVCIEMSSPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFGLSPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESLPD 3bqc A 1.5 BS01 EMO A 1 V53 V66 K68 I95 F113 V116 N118 M163 I174 D175 V51 V64 K66 I93 F111 V114 N116 M161 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 ic50~2uM remove_due_to_license_issue Ki=1850nM, IC50=580nM P68400 18242640 400 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 3bqn B 1.8 BS01 BQN B 1 F153 V157 Y166 I235 Y257 I259 F285 K287 E301 L302 K305 F26 V30 Y39 I108 Y130 I132 F158 K160 E174 L175 K178 ? ic50=2.5nM remove_due_to_license_issue IC50=2.5nM P20701 18783948 1 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 3br9 A 2.3 BS01 DEY A 1 F193 P197 S288 N291 N316 G317 D318 C366 L384 G410 M414 Y415 Q446 Y448 G449 S556 F188 P192 S283 N286 N311 G312 D313 C361 L379 G405 M409 Y410 Q441 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.062uM remove_due_to_license_issue EC50=210nM, IC50=62nM P26663 18242088 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3bra A 2.3 BS01 AEF A 1 D32 F108 D37 F113 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 Kd=2000uM remove_due_to_license_issue Kd=2000000nM P56817 18226904 394 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3brd A 2.21 BS01 dna B 0 K233 R234 F235 K368 R397 S400 T402 K476 K39 R40 F41 K143 R167 S170 T172 K242 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue V6CLJ5 18381292 1 ~ 15 VQSLTSDRMIDFLSNKEKYECVISIFHAKVAQKSYGNEKRFFCPPPCIYLIGQGWKLKKDRVAQLYKTLQQATELVAYIGIGSDTSERQQLDFPNIYDYCAAKTLYISDSDKRKYFDLNAQFFYGCGMEIGGFVSQRIKVISKPSKKKTDCKYLCIASGTKVALFNRLRSQTVSTRYLHVEGNAFHASSTKWGAFTIHLFDDQETDNFAVRDGFVYYGSVVKLVDSVTGIALPRLRIRKVDKQQVILDASCSEEPVSQLHKCAFQMIDNELVYLCLSHDKIIQHQATAINEHRHQINDGAAWTIISTDKAEYRFFEAMGQVANPISPCPVVGSLEVDGHGEASRVELHGRDFKPNLKVWFGATPVETTFRSEESLHCSIPPVSQVRNEQTHWMFTNRTTGDVEVPISLVRDDGVVYSSGLTFSYKSL 3brd A 2.21 BS02 dna C 0 K227 Y229 S367 R399 Q401 K33 Y35 S142 R169 Q171 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue V6CLJ5 18381292 1 ~ 15 VQSLTSDRMIDFLSNKEKYECVISIFHAKVAQKSYGNEKRFFCPPPCIYLIGQGWKLKKDRVAQLYKTLQQATELVAYIGIGSDTSERQQLDFPNIYDYCAAKTLYISDSDKRKYFDLNAQFFYGCGMEIGGFVSQRIKVISKPSKKKTDCKYLCIASGTKVALFNRLRSQTVSTRYLHVEGNAFHASSTKWGAFTIHLFDDQETDNFAVRDGFVYYGSVVKLVDSVTGIALPRLRIRKVDKQQVILDASCSEEPVSQLHKCAFQMIDNELVYLCLSHDKIIQHQATAINEHRHQINDGAAWTIISTDKAEYRFFEAMGQVANPISPCPVVGSLEVDGHGEASRVELHGRDFKPNLKVWFGATPVETTFRSEESLHCSIPPVSQVRNEQTHWMFTNRTTGDVEVPISLVRDDGVVYSSGLTFSYKSL 3brf A 2.47 BS01 dna B 0 K233 R234 F235 K368 R397 S400 K476 K495 K37 R38 F39 K138 R163 S166 K239 K258 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue 18381292 1 ~ 15 SLTSDRMIDFLSNKEKYECVISIFHAKVAQKSYGNEKRFFCPPPCIYLIGQGWKLKKDRVAQLYKTLTELVAYIGIGSDTSERQQLDFPNIYDYCAAKTLYISDSDKRKYFDLNAQFFYGCGMEIGGFVSQRIKVISKPSKKKQSDCKYLCIASGTKVALFNRLRSQTVSTRYLHVEGNAFHASSTKWGAFTIHLFDDEQETDNFAVRDGFVYYGSVVKLVDSVTGIALPRLRIRKVDKQQVILDASCSEEPVSQLHKCAFQMIDNELVYLCLSHDKIIQHQATAINEHRHQINDGAAWTIISTDKAEYRFFEAMGQVANPISPCPVVGSLEVDGHGEASRVELHGRDFKPNLKVWFGATPVETTFRSEESLHCSIPPVSQVRNEQTHWMFTNRTTGDVEVPISLVRDDGVVYSSGLTFSYKS 3brf A 2.47 BS02 dna C 0 K227 Y229 S367 K368 S370 K373 R399 Q401 T402 K31 Y33 S137 K138 S140 K143 R165 Q167 T168 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue 18381292 1 ~ 15 SLTSDRMIDFLSNKEKYECVISIFHAKVAQKSYGNEKRFFCPPPCIYLIGQGWKLKKDRVAQLYKTLTELVAYIGIGSDTSERQQLDFPNIYDYCAAKTLYISDSDKRKYFDLNAQFFYGCGMEIGGFVSQRIKVISKPSKKKQSDCKYLCIASGTKVALFNRLRSQTVSTRYLHVEGNAFHASSTKWGAFTIHLFDDEQETDNFAVRDGFVYYGSVVKLVDSVTGIALPRLRIRKVDKQQVILDASCSEEPVSQLHKCAFQMIDNELVYLCLSHDKIIQHQATAINEHRHQINDGAAWTIISTDKAEYRFFEAMGQVANPISPCPVVGSLEVDGHGEASRVELHGRDFKPNLKVWFGATPVETTFRSEESLHCSIPPVSQVRNEQTHWMFTNRTTGDVEVPISLVRDDGVVYSSGLTFSYKS 3brg C 2.2 BS01 dna A 0 K84 Y86 S191 K192 R220 S221 Q222 K32 Y34 S139 K140 R166 S167 Q168 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 18381292 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMERDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDETVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTPEP 3brg C 2.2 BS02 dna B 0 K90 R91 F92 K192 R218 R220 K295 K311 K38 R39 F40 K140 R164 R166 K235 K251 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 18381292 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMERDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDETVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTPEP 3brn A 2.0 BS01 SRO A 1 S18 Y27 V43 I82 V84 D106 M108 W118 S14 Y23 V39 I78 V80 D102 M104 W114 ? 0030682,0043176 Kd<2nM remove_due_to_license_issue Q09JR9 18445596 158 AQCDFGGPFQAYKSVNGPGNGGYYLRKTTKPGTPECAYVLVPQNTLSEGQSTSFTYGKLQNGQMIQLTATVTVNGDKIEVTGAGQDLSGTTTVLFSDYRSCDVMRGPDGNYELWVHSSAINLQSYGCCDTKFAQVAGGRPIHHTWQTYCPPLP 3bs1 A 1.6 BS01 dna B 0 S164 H169 N185 L186 K187 N201 S202 S29 H34 N50 L51 K52 N66 S67 ? 0000156,0003677 remove_due_to_license_issue P0A0I7 18462677 1 ~ 16 MDNSVETIELKRGSNSVYVQYDDIMFFESSTKSHRLIAHLDNRQIEFYGNLKELSQLDDRFFRCHNSFVVNRHNIESIDSKERIVYFKNKEHCYASVRNVKKI 3bs1 A 1.6 BS02 dna C 0 R170 Y183 H200 N201 S231 V232 R233 R35 Y48 H65 N66 S96 V97 R98 ? 0000156,0003677 remove_due_to_license_issue P0A0I7 18462677 1 ~ 16 MDNSVETIELKRGSNSVYVQYDDIMFFESSTKSHRLIAHLDNRQIEFYGNLKELSQLDDRFFRCHNSFVVNRHNIESIDSKERIVYFKNKEHCYASVRNVKKI 3bsb B 2.8 BS01 rna C 0 Q867 F897 N899 Y900 Y933 C935 R936 Q939 Q968 H972 Q975 R1008 Q1011 Y1041 N1043 Y1044 K1076 N1080 E1083 Y1120 N1122 Y1123 Q1126 Y1156 H1159 Q40 F70 N72 Y73 Y106 C108 R109 Q112 Q141 H145 Q148 R181 Q184 Y214 N216 Y217 K249 N253 E256 Y293 N295 Y296 Q299 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 18328718 1 ~ 9 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 3bsc A 2.65 BS01 2PD A 1 F193 P197 R200 N316 D318 C366 L384 G410 M414 Q446 Y448 S556 F188 P192 R195 N311 D313 C361 L379 G405 M409 Q441 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue IC50=33000nM P26663 18242088 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3bsu A 2.1 BS01 rna D 0 D51 R52 A55 D26 R27 A30 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 HMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu A 2.1 BS02 dna E 0 Y29 W43 F58 K60 Y4 W18 F33 K35 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 HMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu B 2.1 BS01 rna D 0 M27 D51 R52 F53 P54 A55 M2 D26 R27 F28 P29 A30 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 HMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu B 2.1 BS02 dna E 0 Y29 W43 F58 K59 K60 Y4 W18 F33 K34 K35 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 HMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu C 2.1 BS01 rna D 0 D51 R52 P54 A55 D25 R26 P28 A29 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 MFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRKS 3bsu C 2.1 BS02 dna E 0 Y29 W43 F58 K60 Y3 W17 F32 K34 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 MFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRKS 3bsu F 2.1 BS01 rna I 0 R52 A55 R28 A31 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 SHMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu F 2.1 BS02 dna J 0 Y29 W43 F58 K60 Y5 W19 F34 K36 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 SHMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu G 2.1 BS01 rna I 0 G24 D51 R52 F53 P54 A55 G1 D28 R29 F30 P31 A32 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 GSHMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu G 2.1 BS02 dna J 0 Y29 W43 F58 K60 Y6 W20 F35 K37 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 GSHMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVRK 3bsu H 2.1 BS01 rna I 0 R52 F53 A55 R27 F28 A30 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 HMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVR 3bsu H 2.1 BS02 dna J 0 W43 F58 K60 W18 F33 K35 3.1.26.4 remove_due_to_license_issue O60930 18337749 1 ~ 12 HMFYAVRRGRKTGVFLTWNECRAQVDRFPAARFKKFATEDEAWAFVR 3bsx A 2.32 BS01 rna C 0 Q860 Q867 F897 N899 Y900 Q903 R936 Q939 Q968 H972 Q975 Y1005 R1008 Q1011 N1043 Y1044 F1077 S1079 N1080 E1083 N1122 Y1123 Q1126 Y1156 H1159 Q33 Q40 F70 N72 Y73 Q76 R109 Q112 Q141 H145 Q148 Y178 R181 Q184 N216 Y217 F250 S252 N253 E256 N295 Y296 Q299 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 18328718 1 ~ 10 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 3bsx B 2.32 BS01 rna D 0 Q867 N899 Y900 Q903 R936 Q939 H972 Q975 Y1005 R1008 Q1011 Y1041 N1043 Y1044 F1077 S1079 N1080 E1083 N1122 Y1123 Y1156 H1159 Q40 N72 Y73 Q76 R109 Q112 H145 Q148 Y178 R181 Q184 Y214 N216 Y217 F250 S252 N253 E256 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 18328718 2 ~ 10 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 3bt9 A 2.75 BS01 DEQ A 1 Q57 E58 W61 T89 Y93 Y103 Y107 E120 Q56 E57 W60 T88 Y92 Y102 Y106 E119 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 201 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIQESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3bt9 B 2.75 BS01 DEQ A 1 N97 F162 N96 F161 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 201 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIQESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3btc A 2.9 BS01 MGR A 1 W61 E90 Y103 E120 Y123 I124 A153 N154 N157 W60 E89 Y102 E119 Y122 I123 A152 N153 N156 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 200 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIQESKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3bti A 2.85 BS01 BER A 1 E57 W61 Q64 S86 T89 Y93 E120 Y123 E56 W60 Q63 S85 T88 Y92 E119 Y122 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 802 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEQSKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3btj A 2.98 BS01 DEQ A 1 E57 W61 T89 Y93 I100 Y103 L119 E56 W60 T88 Y92 I99 Y102 L118 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 201 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEQSKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3btj B 2.98 BS01 DEQ A 1 N97 I100 T161 F162 N96 I99 T160 F161 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 201 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEQSKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3btl A 2.9 BS01 MGR A 1 W61 E90 Y93 Y103 E120 I124 A153 N154 N157 W60 E89 Y92 Y102 E119 I123 A152 N153 N156 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 18616285 200 NLKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEQSKWQEQWKKEQIKAKTNREKFYLYNELSLTTEYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3bu1 A 1.4 BS01 HSM A 1 S12 Y21 V37 Y51 D94 W105 S9 Y18 V34 Y48 D91 W102 ? 0030682,0043176 Kd=7.1nM remove_due_to_license_issue Q09JX9 18445596 301 CDTVSAWQSLRGPGTGGYYLFKTTEGGKTDCTYVKGSNFNDAAQTATYTYGNLGSGNQLTQQTASASISGNAIVVGTDHSEVLYSDGSTCDVVRLNGQIELWIHSSATSNTGNLNSCCTDKFNQEKGSRPEHVVYRSTCPNLPQ 3buf A 2.3 BS01 AEG A 1 D32 F108 G230 D37 F113 G223 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 Kd=800uM remove_due_to_license_issue P56817 18226904 394 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSFPDGFWLGEQLVCWQAWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHRTAAVEGPFVTLDMEDCGYNI 3bug A 2.5 BS01 AEH A 1 Q12 F108 W115 Q14 F110 W117 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D218 T221 3.4.23.46 0004190,0006508,0016020 Kd=660uM remove_due_to_license_issue Kd=660000nM P56817 18226904 394 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEFPDGFWLGEQLVCWPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHRTAAVEGPFVTLDMEDCGYNI 3buh A 2.3 BS01 AED A 1 G11 G13 D32 F108 G16 G18 D37 F113 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 Kd=220uM remove_due_to_license_issue Kd=220000nM P56817 18226904 394 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3bv2 A 2.4 BS01 P38 A 1 V30 A51 K53 E71 L75 I84 L104 T106 L108 M109 G110 A111 H148 L167 D168 F169 L171 R173 V26 A47 K49 E67 L71 I80 L100 T102 L104 M105 G106 A107 H144 L163 D164 F165 L167 R169 D150 K152 N155 D168 T185 D146 K148 N151 D164 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.44nM remove_due_to_license_issue Q16539 18364256 501 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 3bv3 A 2.59 BS01 P39 A 1 A51 K53 E71 I84 L104 T106 L108 M109 A111 I141 H148 D168 F169 G170 L171 A47 K49 E67 I80 L100 T102 L104 M105 A107 I137 H144 D164 F165 G166 L167 D150 K152 N155 D168 T185 D146 K148 N151 D164 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Ki=0.46nM Q16539 18364256 501 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3bva A 1.05 BS01 2NC B 1 N25 G27 A28 D29 G48 I50 V82 I84 N25 G27 A28 D29 G48 I50 V82 I84 N25 T26 G27 N25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18281688 200 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bva B 1.05 BS01 2NC B 1 N25 G27 A28 D29 D30 I47 G48 G49 I50 N25 G27 A28 D29 D30 I47 G48 G49 I50 N25 T26 G27 N25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ka=3300000M^-1 remove_due_to_license_issue P03367 18281688 200 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bvb A 1.3 BS01 017 B 1 N25 D30 V32 V82 I84 N25 D30 V32 V82 I84 N25 T26 G27 N25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18281688 401 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bvb B 1.3 BS01 017 B 1 N25 G27 A28 D29 G48 G49 I50 N25 G27 A28 D29 G48 G49 I50 N25 T26 G27 N25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ka=3170000M^-1 remove_due_to_license_issue P03367 18281688 401 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bwf A 2.35 BS01 DWC A 1 L44 G45 F49 V52 A65 K67 I104 L120 E121 R122 E171 L174 I185 D186 L12 G13 F17 V20 A33 K35 I72 L88 E89 R90 E139 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=200pM remove_due_to_license_issue P11309 18425743 315 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3bwj A 2.3 BS01 ARX A 1 T51 G52 S53 F54 G55 V57 A70 M120 Y122 V123 E127 D166 K168 E170 L173 T183 F187 F327 T42 G43 S44 F45 G46 V48 A61 M111 Y113 V114 E118 D157 K159 E161 L164 T174 F178 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=0.319uM remove_due_to_license_issue P00517 19143565 351 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3bwj A 2.3 BS02 ARX A 2 G136 R137 S139 G234 Y235 G127 R128 S130 G225 Y226 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 Kd=0.319uM remove_due_to_license_issue P00517 19143565 352 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3bwk A 2.42 BS01 C1P A 1 Q45 G49 C51 N87 Y90 G91 G92 Y93 N182 H183 W215 Q38 G42 C44 N80 Y83 G84 G85 Y86 N175 H176 W208 Q45 C51 H183 N213 Q38 C44 H176 N206 3.4.22.- 0006508,0008234 remove_due_to_license_issue Q8IIL0 19620707 300 YEANYEDVIKKYKPADAKLDRIAYDWRLHGGVTPVKDQALCGSCWAFSSVGSVESQYAIRKKALFLFSEQELVDCSVKNNGCYGGYITNAFDDMIDLGGLCSQDDYPYVSNLPETCNLKRCNERYTIKSYVSIPDDKFKEALRYLGPISISIAASDDFAFYRGGFYDGECGAAPNHAVILVGYGMKDIYNEDTGRMEKFYYYIIKNSWGSDWGEGGYINLETDENGYKKTCSIGTEAYVPLL 3bwk C 2.42 BS01 C1P C 1 Q45 G49 C51 N87 Y90 G91 G92 Y93 P181 N182 H183 W215 Q38 G42 C44 N80 Y83 G84 G85 Y86 P174 N175 H176 W200 Q45 C51 H183 N213 Q38 C44 H176 N198 3.4.22.- 0006508,0008234 remove_due_to_license_issue Q8IIL0 19620707 300 YEANYEDVIKKYKPADAKLDRIAYDWRLHGGVTPVKDQALCGSCWAFSSVGSVESQYAIRKKALFLFSEQELVDCSVKNNGCYGGYITNAFDDMIDLGGLCSQDDYPYVSNLPETCNLKRCNERYTIKSYVSIPDDKFKEALRYLGPISISIAASDDFAFYRGGFYDGECGAAPNHAVILVGYGMKDIEKFYYYIIKNSWGSDWGEGGYINLETDENGYKKTCSIGTEAYVPLL 3bx2 A 2.84 BS01 rna C 0 R579 Q582 N614 Y615 Q618 H648 R651 Q654 L684 H688 N759 Y760 N800 E803 Y836 N838 Y839 Q842 H876 R879 R20 Q23 N55 Y56 Q59 H89 R92 Q95 L125 H129 N200 Y201 N241 E244 Y277 N279 Y280 Q283 H317 R320 ? 0003723 remove_due_to_license_issue P25339 18327269 1 ~ 9 VLDQYIGSIHSLCKDQHGCRFLQKQLDILGSKAADAIFEETKDYTVELMTDSFGNYLIQKLLEEVTTEQRIVLTKISSPHFVEISLNPHGTRALQKLIECIKTDEEAQIVVDSLRPYTVQLSKDLNGNHVIQKCLQRLKPENFQFIFDAISDSCIDIATHRHGCCVLQRCLDHGTTEQCDNLCDKLLALVDKLTLDPFGNYVVQYIITKEAEKNKYDYTHKIVHLLKPRAIELSIHKFGSNVIEKILKTAIVSEPMILEILNNGGETGIQSLLNDSYGNYVLQTALDISHKQNDYLYKRLSEIVAPLLVGPIRNTPHGKRIIGMLHLD 3bx2 B 2.84 BS01 rna D 0 Q575 R579 Q582 N614 Y615 R651 Q654 L684 H688 N759 Y760 S799 N800 E803 Y836 N838 Y839 Q842 H876 Q14 R18 Q21 N53 Y54 R90 Q93 L123 H127 N198 Y199 S238 N239 E242 Y275 N277 Y278 Q281 H315 ? 0003723 remove_due_to_license_issue P25339 18327269 1 ~ 9 DQYIGSIHSLCKDQHGCRFLQKQLDILGSKAADAIFEETKDYTVELMTDSFGNYLIQKLLEEVTTEQRIVLTKISSPHFVEISLNPHGTRALQKLIECIKTDEEAQIVVDSLRPYTVQLSKDLNGNHVIQKCLQRLKPENFQFIFDAISDSCIDIATHRHGCCVLQRCLDHGTTEQCDNLCDKLLALVDKLTLDPFGNYVVQYIITKEAEKNKYDYTHKIVHLLKPRAIELSIHKFGSNVIEKILKTAIVSEPMILEILNNGGETGIQSLLNDSYGNYVLQTALDISHKQNDYLYKRLSEIVAPLLVGPIRNTPHGKRIIGML 3bx3 A 3.0 BS01 rna C 0 Q575 R579 N614 Y615 Q618 H648 R651 Q654 L684 H688 R720 C723 R724 Q727 F757 N759 Y760 S799 N800 E803 N838 Y839 H876 R879 Q14 R18 N53 Y54 Q57 H87 R90 Q93 L123 H127 R159 C162 R163 Q166 F196 N198 Y199 S238 N239 E242 N277 Y278 H315 R318 ? 0003723 remove_due_to_license_issue P25339 18327269 1 ~ 8 DQYIGSIHSLCKDQHGCRFLQKQLDILGSKAADAIFEETKDYTVELMTDSFGNYLIQKLLEEVTTEQRIVLTKISSPHFVEISLNPHGCRALQKLIECIKTDEEAQIVVDSLRPYTVQLSKDLNGNHVIQKCLQRLKPENFQFIFDAISDSCIDIATHRHGCRVLQRCLDHGTTEQCDNLCDKLLALVDKLTLDPFGNYVVQYIITKEAEKNKYDYTHKIVHLLKPRAIELSIHKFGSNVIEKILKTAIVSEPMILEILNNGGETGIQSLLNDSYGNYVLQTALDISHKQNDYLYKRLSEIVAPLLVGPIRNTPHGKRIIGMLHL 3bx3 B 3.0 BS01 rna D 0 F612 N614 Y615 Q618 H648 R651 Q654 L684 H688 R720 R724 Q727 F757 N759 Y760 N800 E803 N838 Y839 R879 F27 N29 Y30 Q33 H63 R66 Q69 L99 H103 R135 R139 Q142 F172 N174 Y175 N215 E218 N253 Y254 R294 ? 0003723 remove_due_to_license_issue P25339 18327269 1 ~ 8 DILGSKAADAIFEETKDYTVELMTDSFGNYLIQKLLEEVTTEQRIVLTKISSPHFVEISLNPHGCRALQKLIECIKTDEEAQIVVDSLRPYTVQLSKDLNGNHVIQKCLQRLKPENFQFIFDAISDSCIDIATHRHGCRVLQRCLDHGTTEQCDNLCDKLLALVDKLTLDPFGNYVVQYIITKEAEKNKYDYTHKIVHLLKPRAIELSIHKFGSNVIEKILKTAIVSEPMILEILNNGGETGIQSLLNDSYGNYVLQTALDISHKQNDYLYKRLSEIVAPLLVGPIRNTPHGKRIIGMLH 3bx5 A 2.4 BS01 304 A 1 Y35 A51 K53 E71 L75 T106 L108 M109 A111 A157 L167 D168 Y31 A47 K49 E67 L71 T102 L104 M105 A107 A153 L163 D164 D150 K152 N155 D168 T185 D146 K148 N151 D164 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=3.5nM remove_due_to_license_issue IC50=3.5nM Q16539 18313298 501 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3bxf A 1.7 BS01 FBP A 1 T148 G149 T151 T152 R175 Q185 G242 M247 R250 R251 E269 K310 T63 G64 T66 T67 R90 Q100 G157 M162 R165 R166 E184 K225 ? 0030246 Kd=2.87uM remove_due_to_license_issue O32253 18554327 401 SNAKDVLGLTLLEKTLKERLNLKDAIIVSGDSDQSPWVKKEMGRAAVACMKKRFSGKNIVAVTGGTTIEAVAEMMTPDSKNRELLFVPARGGLGEDVKNQANTICAHMAEKASGTYRLLFVPGQLSQGAYSSIIEEPSVKEVLNTIKSASMLVHGIGEAKTMAQRRNTPLEDLKKIDDNDAVTEAFGYYFNADGEVVHKVHSVGMQLDDIDAIPDIIAVAGGSSKAEAIEAYFKKPRNTVLVTDEGAAKKLLR 3bxg A 1.8 BS01 BG6 A 1 T148 G150 T151 T152 E180 G240 I241 M247 R250 R251 E269 F271 K310 T56 G58 T59 T60 E88 G148 I149 M155 R158 R159 E177 F179 K218 ? 0030246 Kd=10.98uM remove_due_to_license_issue O32253 18554327 401 GLTLLEKTLKERLNLKDAIIVSGDSDQSPWVKKEMGRAAVACMKKRFSGKNIVAVTGGTTIEAVAEMMTPDSKNRELLFVPARGGLGEDVKNQANTICAHMAEKASGTYRLLFVPGQLSQGAYSSIIEEPSVKEVLNTIKSASMLVHGIGEAKTMAQRRNTPLEDLKKIDDNDAVTEAFGYYFNADGEVVHKVHSVGMQLDDIDAIPDIIAVAGGSSKAEAIEAYFKKPRNTVLVTDEGAAKKLLRD 3bxh A 1.85 BS01 F6P A 1 T148 G149 T151 T152 E180 G242 M247 R250 R251 E269 F271 K310 T56 G57 T59 T60 E88 G150 M155 R158 R159 E177 F179 K218 ? 0030246 Kd=94.34uM remove_due_to_license_issue O32253 18554327 401 GLTLLEKTLKERLNLKDAIIVSGDSDQSPWVKKEMGRAAVACMKKRFSGKNIVAVTGGTTIEAVAEMMTPDSKNRELLFVPARGGLGEDVKNQANTICAHMAEKASGTYRLLFVPGQLSQGAYSSIIEEPSVKEVLNTIKSASMLVHGIGEAKTMAQRRNTPLEDLKKIDDNDAVTEAFGYYFNADGEVVHKVHSVGMQLDDIDAIPDIIAVAGGSSKAEAIEAYFKKPRNTVLVTDEGAAKKLLRDE 3bxs A 1.6 BS01 DRS A 1 D25 G27 D29 G48 D25 G27 D29 G48 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8uM remove_due_to_license_issue P03369 18311928 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bxs A 1.6 BS02 DRS B 1 D25 P81 V82 I84 D25 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8uM remove_due_to_license_issue P03369 18311928 203 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bxs B 1.6 BS01 DRS A 1 D125 P181 I184 D25 P81 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8uM remove_due_to_license_issue P03369 18311928 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bxs B 1.6 BS02 DRS B 1 G127 A128 D129 G148 G27 A28 D29 G48 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8uM remove_due_to_license_issue P03369 18311928 203 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3bxz A 3.0 BS01 ADP A 1 M81 F84 Q87 G105 G107 K108 T109 M71 F74 Q77 G95 G97 K98 T99 7.4.2.8 0005524,0006605,0006886,0016020,0017038 remove_due_to_license_issue P10408 18761349 901 GSRNDRTLRRMRKVVNIINAMEPEMEKLSDEELKGKTAEFRARLEKGEVLENLIPEAFAVVREASKRVFGMRHFDVQLLGGMVLNERCIAEMRTGEGKTLTATLPAYLNALTGKGVHVVTVNDYLAQRDAENNRPLFEFLGLTVGINLPGMPAPAKREAYAADITYGTNNEYGFDYLRDNMAFSPEERVQRKLHYALVDEVDSILIDEARTPLIILASITFQNYFRLYEKLAGMTGTADTEAFEFSSIYKLDTVVVPTNRPMIRKDLPDLVYMTEAEKIQAIIEDIKERTAKGQPVLVGTISIEKSELVSNELTKAGIKHNVLNAKFHANEAAIVAQAGYPAAVTIATNMAGRGTDIVLGGSWQAEVAALENPTAEQIEKIKADWQVRHDAVLEAGGLHIIGTERHESRRIDNQLRGRSGRQGDAGSSRFYLSMEDAL 3bym A 2.0 BS01 AM0 A 1 V259 A271 E288 M292 Y318 M319 G322 L371 V30 A42 E59 M63 Y89 M90 G93 L142 D364 R366 A368 N369 D382 A400 F402 D135 R137 A139 N140 D153 A171 F173 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.006uM remove_due_to_license_issue IC50=6nM P06239 18278858 1 QKPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 3byo A 2.0 BS01 AM9 A 1 L251 V259 A271 K273 E288 T316 Y318 M319 G322 L371 L21 V29 A41 K43 E58 T86 Y88 M89 G92 L141 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM remove_due_to_license_issue IC50=1600nM P06239 18278858 1 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 3bys A 2.2 BS01 AM5 A 1 A271 K273 E288 M292 I314 T316 Y318 M319 G322 L371 I380 A381 D382 A42 K44 E59 M63 I85 T87 Y89 M90 G93 L142 I151 A152 D153 D364 R366 A368 N369 D382 D135 R137 A139 N140 D153 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5nM remove_due_to_license_issue IC50=0.5nM P06239 18321037 1 QKPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 3byu A 2.3 BS01 AM6 A 1 A271 V272 K273 E288 M292 T316 Y318 M319 G322 L371 A381 D382 F383 A41 V42 K43 E58 M62 T86 Y88 M89 G92 L141 A151 D152 F153 D364 R366 A368 N369 D382 F402 D134 R136 A138 N139 D152 F157 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.8nM remove_due_to_license_issue IC50=0.8nM P06239 18321037 1 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 3bz3 A 2.2 BS01 YAM A 1 R426 I428 V436 A452 E500 L501 C502 G505 L553 D564 L567 S568 R13 I15 V23 A35 E83 L84 C85 G88 L136 D147 L150 S151 D546 A548 R550 N551 D564 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.5nM remove_due_to_license_issue IC50=1.5nM Q05397 18339875 1 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPLAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSRYLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQQEE 3c0z A 2.1 BS03 SHH A 1 H669 H670 F679 D707 H709 F738 H152 H153 F162 D190 H192 F221 3.5.1.-,3.5.1.98 ic50=113uM remove_due_to_license_issue IC50=>10000nM, Ki=129nM, Kd=36000nM Q8WUI4 18285338 301 TLPFTTGLIYDSVMLKHQCSCGDNSRHPEHAGRIQSIWSRLQERGLRSQCECLRGRKASLEELQSVHSERHVLLYGTNPLSRLKLDNGKLAGLLAQVMLPCGGVGVDTDTIWNELHSSNAARWAAGSVTDLAFKVASRELKNGFAVVRPPGHHADHSTAMGFCFFNSVAIACRQLQQQSKASKILIVDWDVHHGNGTQQTFYQDPSVLYISLHRHDDGNFFPGSGAVDEVGAGSGEGFNVNVAWAGGLDPPMGDPEYLAAFRIVVMPIAREFSPDLVLVSAGFDAAEGHPAPLGGYHVSAKCFGYMTQQLMNLAGGAVVLALEGGHDLTAICDASEACVAALLGNRVDPLSEEGWKQKPNLNAIRSLEAVIRVHSKYWGCMQR 3c10 A 2.0 BS03 TSN A 1 H669 H670 F679 D707 H709 F738 L810 H152 H153 F162 D190 H192 F221 L293 3.5.1.-,3.5.1.98 ic50=0.3uM remove_due_to_license_issue IC50=22nM, Ki=195nM Q8WUI4 18285338 301 TLPFTTGLIYDSVMLKHQCSCGDNSRHPEHAGRIQSIWSRLQERGLRSQCECLRGRKASLEELQSVHSERHVLLYGTNPLSRLKLDNGKLAGLLAQVMLPCGGVGVDTDTIWNELHSSNAARWAAGSVTDLAFKVASRELKNGFAVVRPPGHHADHSTAMGFCFFNSVAIACRQLQQQSKASKILIVDWDVHHGNGTQQTFYQDPSVLYISLHRHDDGNFFPGSGAVDEVGAGSGEGFNVNVAWAGGLDPPMGDPEYLAAFRIVVMPIAREFSPDLVLVSAGFDAAEGHPAPLGGYHVSAKCFGYMTQQLMNLAGGAVVLALEGGHDLTAICDASEACVAALLGNRVDPLSEEGWKQKPNLNAIRSLEAVIRVHSKYWGCMQR 3c1k A 1.84 BS02 T15 A 1 H57 Y60A L99 C191 E192 S195 S214 W215 G216 E217 G219 C220 H69 Y73 L122 C219 E220 S223 S244 W245 G246 E247 G248 C249 H57 D102 E192 G193 D194 S195 G196 H69 D125 E220 G221 D222 S223 G224 3.4.21.5 0004252,0005509,0005576,0006508,0007596 Ki=0.36nM remove_due_to_license_issue P00734 18291642 403 DCGLRPLFEKKSLEDKTERELLESYIIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3c1x A 2.17 BS01 CKK A 1 A1108 E1127 M1131 F1134 L1140 L1157 M1160 D1164 F1200 M1211 A1221 D1222 F1223 A59 E78 M82 F85 L91 L108 M111 D115 F151 M162 A172 D173 F174 D1204 A1206 R1208 N1209 D1222 D155 A157 R159 N160 D173 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.045uM remove_due_to_license_issue IC50=45nM P08581 18289854 1500 TVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3c2f A 2.35 BS01 PRP A 1 K144 S256 G257 T277 S278 K143 S234 G235 T249 S250 R107 K144 K176 E206 D227 R106 K143 K175 E205 D226 2.4.2.19 0004514,0005634,0005737,0009435,0016757,0016763,0019363,0034213,0034354 Kd=10.1mM remove_due_to_license_issue P43619 18321072 300 PVYEHLLPVNGAWRQDVTNWLSEDVPSFDFGGYVVGSDLKEANLYCKQDGMLCGVPFAQEVFNQCELQVEWLFKEGSFLEPSKNDSGKIVVAKITGPAKNILLAERTALNILSRSSGIATASHKIISLARSTGYKGTIAGTRKTTPGLRRLEKYSMLVGGCDTHRYDLSSMVMLKDNHIWATGSITNAVKNARAVCGFAVKIEVECLSEDEATEAIEAGADVIMLDNHFLLECSGGLNLLCDDIDIYSTSSIHQGTPVIDFSLKLAH 3c2o A 2.3 BS01 NTM A 1 T142 R143 H165 R166 M174 S276 T141 R142 H164 R165 M173 S247 R107 K144 K176 E206 D227 R106 K143 K175 E205 D226 2.4.2.19 0004514,0005634,0005737,0009435,0016757,0016763,0019363,0034213,0034354 Kd=0.45mM remove_due_to_license_issue P43619 18321072 300 PVYEHLLPVNGAWRQDVTNWLSEDVPSFDFGGYVVGSDLKEANLYCKQDGMLCGVPFAQEVFNQCELQVEWLFKEGSFLEPSKNDSGKIVVAKITGPAKNILLAERTALNILSRSSGIATASHKIISLARSTGYKGTIAGTRKTTPGLRRLEKYSMLVGGCDTHRYDLSSMVMLKDNHIWATGSITNAVKNARAVCGFAVKIEVECLSEDEATEAIEAGADVIMLDNHFLLECSGGLNLCDDIDIYSTSSIHQGTPVIDFSLKLA 3c2r A 2.4 BS01 PHT A 1 T142 R143 H165 R166 M174 T141 R142 H164 R165 M173 R107 K144 K176 E206 D227 R106 K143 K175 E205 D226 2.4.2.19 0004514,0005634,0005737,0009435,0016757,0016763,0019363,0034213,0034354 Kd=0.78mM remove_due_to_license_issue P43619 18321072 300 PVYEHLLPVNGAWRQDVTNWLSEDVPSFDFGGYVVGSDLKEANLYCKQDGMLCGVPFAQEVFNQCELQVEWLFKEGSFLEPSKNDSGKIVVAKITGPAKNILLAERTALNILSRSSGIATASHKIISLARSTGYKGTIAGTRKTTPGLRRLEKYSMLVGGCDTHRYDLSSMVMLKDNHIWATGSITNAVKNARAVCGFAVKIEVECLSEDEATEAIEAGADVIMLDNHFLLECSGGLNLLCDDIDIYSTSSIHQGTPVIDFSLKLAH 3c2r B 2.4 BS01 PHT B 1 T142 R143 H165 R166 M174 T141 R142 H164 R165 M173 R107 K144 K176 E206 D227 R106 K143 K175 E205 D226 2.4.2.19 0004514,0005634,0005737,0009435,0016757,0016763,0019363,0034213,0034354 Kd=0.78mM remove_due_to_license_issue P43619 18321072 301 PVYEHLLPVNGAWRQDVTNWLSEDVPSFDFGGYVVGSDLKEANLYCKQDGMLCGVPFAQEVFNQCELQVEWLFKEGSFLEPSKNDSGKIVVAKITGPAKNILLAERTALNILSRSSGIATASHKIISLARSTGYKGTIAGTRKTTPGLRRLEKYSMLVGGCDTHRYDLSSMVMLKDNHIWATGSITNAVKNARAVCGFAVKIEVECLSEDEATEAIEAGADVIMLDNHFLLECSGGLNLLCDDIDIYSTSSIHQGTPVIDFSLKLAH 3c43 A 2.3 BS01 315 A 1 E205 E206 Y547 S552 Q553 K554 S630 Y631 Y662 Y666 V711 E167 E168 Y509 S514 Q515 K516 S592 Y593 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.019uM remove_due_to_license_issue IC50=19nM P27487 18331795 804 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3c45 A 2.05 BS01 317 A 1 E205 E206 F357 Y547 S552 Q553 K554 S630 Y662 Y666 E167 E168 F319 Y509 S514 Q515 K516 S592 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.00021uM remove_due_to_license_issue IC50=12nM P27487 18331795 805 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3c49 A 2.8 BS01 KU8 A 1 H384 G385 R400 Y414 K421 S422 Y425 E514 H209 G210 R225 Y239 K246 S247 Y250 E339 S422 Y425 E514 S247 Y250 E339 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 19354255 601 SMKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKGPTDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 3c4c A 2.57 BS01 324 A 1 A481 K483 L514 I527 T529 Q530 W531 C532 F583 D594 F595 A34 K36 L67 I80 T82 Q83 W84 C85 F136 D147 F148 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=13nM, Ki=2.6nM, Kd=100nM P15056 18287029 2 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGSGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARELS 3c4e A 1.98 BS01 C4E A 1 F49 A65 K67 L174 D186 F17 A33 K35 L142 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50~100uM remove_due_to_license_issue P11309 18287029 306 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3c4f A 2.07 BS01 C4F A 1 F489 A512 I545 E562 A564 L630 A640 D641 F26 A49 I82 E99 A101 L155 A165 D166 D623 A625 R627 N628 D641 D148 A150 R152 N153 D166 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=1.9uM remove_due_to_license_issue IC50=1900nM P11362 18287029 1 ELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 3c4h A 2.1 BS01 DRL A 1 H384 G385 Y414 S422 Y425 E514 H209 G210 Y239 S247 Y250 E339 S422 Y425 E514 S247 Y250 E339 2.4.2.- 0003950 Kd=2uM remove_due_to_license_issue Q9Y6F1 19354255 601 SMKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKGPTDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 3c52 A 2.3 BS03 PGH A 1 D82 H83 H180 K184 H210 G211 S213 N253 D255 T256 D82 H83 H169 K173 H199 G200 S202 N242 D244 T245 C69 E70 G136 H180 A226 N253 C69 E70 G136 H169 A215 N242 4.1.2.13 0004332,0005975,0006096,0008270,0016829,0016832,0030388,0046872 remove_due_to_license_issue P56109 18688832 404 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMGIVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3c52 B 2.3 BS03 PGH B 1 D82 H83 H180 K184 H210 G211 S213 N253 D255 T256 D82 H83 H168 K172 H198 G199 S201 N241 D243 T244 C69 E70 G136 H180 A226 N253 C69 E70 G136 H168 A214 N241 4.1.2.13 0004332,0005975,0006096,0008270,0016829,0016832,0030388,0046872 remove_due_to_license_issue P56109 18688832 404 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMGILVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3c56 A 2.3 BS02 PH4 A 1 N23 S49 D82 H180 K184 G211 S213 N253 D255 T256 R259 N23 S49 D82 H170 K174 G201 S203 N243 D245 T246 R249 C69 E70 G136 H180 A226 N253 C69 E70 G136 H170 A216 N243 4.1.2.13 0004332,0005975,0006096,0008270,0016829,0016832,0030388,0046872 Ki=0.013uM remove_due_to_license_issue Ki=13nM P56109 18688832 309 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMGIAVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3c56 B 2.3 BS02 PH4 B 1 N23 S49 D82 H180 K184 H210 G211 A212 S213 N253 D255 T256 R259 N23 S49 D82 H167 K171 H197 G198 A199 S200 N240 D242 T243 R246 C69 E70 G136 H180 A226 N253 C69 E70 G136 H167 A213 N240 4.1.2.13 0004332,0005975,0006096,0008270,0016829,0016832,0030388,0046872 Ki=0.013uM remove_due_to_license_issue Ki=13nM P56109 18688832 309 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3c58 A 1.9 BS01 dna C 0 K90 H91 V108 R109 K110 F111 K90 H91 V108 R109 K110 F111 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 18635007 15 ~ 28 PELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSIRSALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 3c58 A 1.9 BS02 dna B 0 P1 E2 E5 K57 H72 R74 M75 R109 K129 Q163 G170 N171 I172 S217 I219 Y238 K254 K256 R260 G261 P1 E2 E5 K57 H72 R74 M75 R109 K129 Q163 G170 N171 I172 S217 I219 Y236 K252 K254 R258 G259 3.2.2.23,4.2.99.18 0003676,0003677,0003684,0003906,0006281,0006284,0008270,0008534,0016787,0016798,0016799,0016829,0019104,0034039,0046872,0140078 remove_due_to_license_issue P42371 18635007 1 ~ 14 PELPEVETVRRELEKRIVGQKIISIEATYPRMVLTGFEQLKKELTGKTIQGISRRGKYLIFEIGDDFRLISHLRMEGKYRLATLDAPREKHDHLTMKFADGQLIYADVRKFGTWELISTDQVLPYFLKKKIGPEPTYEDFDEKLFREKLRKSTKKIKPYLLEQTLVAGLGNIYVDEVLWLAKIHPEKETNQLIESSIHLLHDSIIEILQKAIKLGGSSIRSALGSTGKMQNELQVYGKTGEKCSRCGAEIQKIKVAGRGTHFCPVCQQK 3c5u A 2.8 BS01 P41 A 1 P191 E192 L195 H228 L232 P242 I250 Y258 I259 P177 E178 L181 H214 L218 P228 I236 Y244 I245 D150 K152 N155 D168 T185 D147 K149 N152 D165 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=6.4nM Q16539 18296051 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3c5u A 2.8 BS02 P41 A 2 V30 Y35 A51 K53 L75 L104 T106 L108 M109 G110 L167 V27 Y32 A48 K50 L72 L101 T103 L105 M106 G107 L164 D150 K152 N155 D168 T185 D147 K149 N152 D165 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=6.4nM Q16539 18296051 362 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3c6t A 2.7 BS01 M14 A 1 P95 K102 K103 V106 Y181 Y188 F227 W229 P236 Y318 P97 K104 K105 V108 Y183 Y190 F229 W231 P238 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 18396399 561 NSPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3c6u A 2.7 BS01 M22 A 1 L100 K103 V106 Y181 Y188 G190 F227 W229 L234 H235 P236 Y318 L101 K104 V107 Y182 Y189 G191 F228 W230 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 18396399 561 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3c72 B 2.3 BS03 CX1 B 1 R144 H190 G192 Q193 Y195 C196 Y241 W244 R137 H183 G185 Q186 Y188 C189 Y234 W237 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=22.7uM remove_due_to_license_issue Q08603 18399557 334 DVTIKSDAPDTLLLEKHADYIASYGSKDDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3c79 A 2.48 BS01 IM4 A 1 W147 Y188 C190 Y195 W150 Y191 C193 Y198 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=63nM remove_due_to_license_issue Ki=19nM Q8WSF8 18477694 301 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 3c79 A 2.48 BS02 IM4 B 1 Y55 V108 M116 Y58 V111 M119 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=63nM remove_due_to_license_issue Ki=19nM Q8WSF8 18477694 302 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 3c79 E 2.48 BS01 IM4 A 1 Y55 V108 M116 I118 Y58 V111 M119 I121 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=19nM Q8WSF8 18477694 301 DDKLHSQANLMRLKSDLFNRSMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 3c7n A 3.115 BS01 ADP A 1 G10 N11 N12 N13 G205 H206 E272 K275 K276 S279 G343 T344 R346 G10 N11 N12 N13 G205 H206 E272 K275 K276 S279 G343 T344 R346 D8 K69 D174 D203 D8 K69 D174 D203 ? 0000774,0005515,0005516,0005524,0005634,0005737,0005829,0006457,0006914,0010499,0042026,0042277,0043161,0140662 remove_due_to_license_issue P32589 18550409 672 MSTPFGLDLGNNNSVLAVARNRGIDIVVNEVSNRSTPSVVGFGPKNRYLGETGKNKQTSNIKNTVANLKRIIGLDYHHPDFEQESKHFTSKLVELDDKKTGAEVRFAGEKHVFSATQLAAMFIDKVKDTVKQDTKANITDVCIAVPPWYTEEQRYNIADAARIAGLNPVRIVNDVTAAGVSYGIFKTDLPEGEEKPRIVAFVDIGHSSYTCSIMAFKKGQLKVLGTACDKHFGGRDFDLAITEHFADEFKTKYKIDIRENPKAYNRILTAAEKLKKVLSANTNAPFSVESVMNDVDVSSQLSREELEELVKPLLERVTEPVTKALAQAKLSAEEVDFVEIIGGTTRIPTLKQSISEAFGKPLSTTLNQDEAIAKGAAFICAIHSPTLRVRPFKFEDIHPYSVSYSWDKQVEDEDHMEVFPAGSSFPSTKLITLNRTGDFSMAASYTDITQLPPNTPEQIANWEITGVQLPEGQDSVPVKLKLRCDPSGLHTIEEAYTIEDIEVEEPIPLPEDAPEDAEQEFKKVTKTVKKDDLTIVAHTFGLDAKKLNELIEKENEMLAQDKLVAETEDRKNTLEEYIYTLRGKLEEEYAPFASDAEKTKLQGMLNKAEEWLYDEGFDSIKAKYIAKYEELASLGNIIRGRYLAKEEEK 3c7n B 3.115 BS01 ADP B 1 G201 G202 E268 K271 R272 S275 G338 G339 R342 I343 G199 G200 E266 K269 R270 S273 G336 G337 R340 I341 D10 K71 E175 D199 D8 K69 E173 D197 3.6.4.10 0005524,0140662 remove_due_to_license_issue P19120 18550409 560 KGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILSGDKDLLLLDVTPLSLGIETAGGVMTVLIKRNTTIPTKQTQTFTTYSDNQPGVLIQVYEGERAMTKDNNLLGKFELTGIPPAPRGVPQIEVTFDIDANGILNVSAVDKSTGKENKITITNDKGRLSKEDIERMVQEAEKYKAEDEKQRDKVSSKNSLESYAF 3c7p A 1.7 BS02 POF A 1 H94 H119 F131 G132 V135 Q136 L198 T199 T200 H92 H117 F128 G129 V132 Q133 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=0.1nM remove_due_to_license_issue P00918 18723489 265 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3c7q A 2.1 BS01 XIN A 1 L840 E850 V899 V916 F918 C919 K920 G922 L1035 C1045 L22 E32 V81 V98 F100 C101 K102 G104 L159 C169 D1028 A1030 R1032 N1033 D1046 K1055 D1064 D152 A154 R156 N157 D170 K175 D184 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=21nM remove_due_to_license_issue IC50=21nM, Kd=2.9nM, Ki=3.80nM P35968 18559524 1172 RLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQD 3c84 A 1.94 BS01 TH4 A 1 W147 Y188 C190 Y195 W150 Y191 C193 Y198 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=14nM remove_due_to_license_issue Ki=3.9nM Q8WSF8 18477694 301 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3c84 A 1.94 BS02 TH4 B 1 Y55 M116 I118 Y58 M119 I121 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=14nM remove_due_to_license_issue Ki=3.9nM Q8WSF8 18477694 302 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3c84 E 1.94 BS01 TH4 A 1 Y55 M116 I118 Y53 M114 I116 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=3.9nM Q8WSF8 18477694 301 DKLHSQANLMRLKSDLFYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3c8e A 1.5 BS01 GSH A 1 T52 N54 I82 Q87 K100 I101 E117 S118 T48 N50 I78 Q83 K96 I97 E113 S114 1.11.1.-,1.8.4.- 0004364,0004601,0005737,0015036,0042803,0098869 Kd=0.07mM remove_due_to_license_issue Q46845 21222452 289 TYQPAKVWTWDKSAGGAFANINRPVSGPTHEKTLPVGKHPLQLYSLGTPNGQKVTIMLEELLALGVTGAEYDAWLIRIGDGDQFSSGFVEVNPNSKIPALRDHTHNPPIRVFESGSILLYLAEKFGYFLPQDLAKRTETMNWLFWLQGAAPFLGGGFGHFYHYAPVKIEYAINRFTMEAKRLLDVLDKQLAQHKFVAGDEYTIADMAIWPWFGNVVLGGVYDAAEFLDAGSYKHVQRWAKEVGERPAVKRGRIVNRTNGPLNEQLHERHDASDFETNTEDKRQG 3c8e A 1.5 BS02 GSH A 2 F22 N26 T52 N54 P155 G158 W215 F18 N22 T48 N50 P151 G154 W211 1.11.1.-,1.8.4.- 0004364,0004601,0005737,0015036,0042803,0098869 Kd=0.07mM remove_due_to_license_issue Q46845 21222452 290 TYQPAKVWTWDKSAGGAFANINRPVSGPTHEKTLPVGKHPLQLYSLGTPNGQKVTIMLEELLALGVTGAEYDAWLIRIGDGDQFSSGFVEVNPNSKIPALRDHTHNPPIRVFESGSILLYLAEKFGYFLPQDLAKRTETMNWLFWLQGAAPFLGGGFGHFYHYAPVKIEYAINRFTMEAKRLLDVLDKQLAQHKFVAGDEYTIADMAIWPWFGNVVLGGVYDAAEFLDAGSYKHVQRWAKEVGERPAVKRGRIVNRTNGPLNEQLHERHDASDFETNTEDKRQG 3c8e B 1.5 BS01 GSH B 1 T52 N54 Q87 K100 I101 E117 S118 T47 N49 Q82 K95 I96 E112 S113 1.11.1.-,1.8.4.- 0004364,0004601,0005737,0015036,0042803,0098869 Kd=0.07mM remove_due_to_license_issue Q46845 21222452 289 YQPAKVWTWDKSAGGAFANINRPVSGPTHEKTLPVGKHPLQLYSLGTPNGQKVTIMLEELLALGVTGAEYDAWLIRIGDGDQFSSGFVEVNPNSKIPALRDHTHNPPIRVFESGSILLYLAEKFGYFLPQDLAKRTETMNWLFWLQGAAPFLGGGFGHFYHYAPVKIEYAINRFTMEAKRLLDVLDKQLAQHKFVAGDEYTIADMAIWPWFGNVVLGGVYDAAEFLDAGSYKHVQRWAKEVGERPAVKRGRIVNRTNGPLNEQLHERHDASDFETNTEDKRQG 3c8e B 1.5 BS02 GSH B 2 F22 N26 T52 N54 P155 G158 W215 F17 N21 T47 N49 P150 G153 W210 1.11.1.-,1.8.4.- 0004364,0004601,0005737,0015036,0042803,0098869 Kd=0.07mM remove_due_to_license_issue Q46845 21222452 290 YQPAKVWTWDKSAGGAFANINRPVSGPTHEKTLPVGKHPLQLYSLGTPNGQKVTIMLEELLALGVTGAEYDAWLIRIGDGDQFSSGFVEVNPNSKIPALRDHTHNPPIRVFESGSILLYLAEKFGYFLPQDLAKRTETMNWLFWLQGAAPFLGGGFGHFYHYAPVKIEYAINRFTMEAKRLLDVLDKQLAQHKFVAGDEYTIADMAIWPWFGNVVLGGVYDAAEFLDAGSYKHVQRWAKEVGERPAVKRGRIVNRTNGPLNEQLHERHDASDFETNTEDKRQG 3c9e A 1.8 BS07 E64 A 1 Q19 G23 C25 E59 N60 G65 G66 Y67 L160 H162 Q19 G23 C25 E59 N60 G65 G66 Y67 L160 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 18692071 308 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3caj A 1.8 BS02 EZL A 1 H94 H119 L198 T199 T200 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8nM remove_due_to_license_issue Ki=8nM, IC50=3nM, Kd=0.71nM P00918 18359629 265 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3cbp A 1.42 BS02 SFG A 1 A226 E228 G264 N265 H293 K294 N296 H297 Y335 W352 E356 A110 E112 G148 N149 H177 K178 N180 H181 Y219 W228 E232 Y245 H293 H297 Y305 Y335 Y129 H177 H181 Y189 Y219 2.1.1.364 0005694,0006355,0016279,0140945 remove_due_to_license_issue IC50=2500nM Q8WTS6 18471979 1501 GVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDERTALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCISTNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITHQEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPNCIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHEAPEWYQVELKAFQAT 3cbs A 2.0 BS01 R12 A 1 L28 A36 T54 V58 L121 R132 Y134 L28 A36 T54 V58 L121 R132 Y134 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 ic50=58nM remove_due_to_license_issue P29373 10531482 200 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKTSTTVRTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTRELTNDGELILTMTADDVVCTRVYVRE 3cc4 1 2.7 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 F39 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 F39 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18455733 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3cc4 2 2.7 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 N16 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R35 H37 K38 R40 H41 W42 R43 T47 E49 G1 K2 K3 K5 A6 K8 R10 L11 K13 N16 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R32 H34 K35 R37 H38 W39 R40 T44 E46 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18455733 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 3cc4 3 2.7 BS01 rna 0 0 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 D66 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 D66 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18455733 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3cc4 A 2.7 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 G203 G204 G205 R206 Q207 H208 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 G203 G204 G205 R206 Q207 H208 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18455733 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3cc4 B 2.7 BS01 rna 0 0 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 Q94 R95 P96 L97 E99 W101 R111 T112 L113 D114 V115 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 K267 D281 G282 V285 N286 G288 E289 S300 V301 P302 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 Q94 R95 P96 L97 E99 W101 R111 T112 L113 D114 V115 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 K267 D281 G282 V285 N286 G288 E289 S300 V301 P302 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18455733 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3cc4 C 2.7 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 P71 Q73 D74 R76 A77 R78 V80 P81 Q82 V84 K85 R87 H90 P92 K93 T94 E95 K96 D97 L100 D101 N103 D104 K105 E106 R107 Q108 R127 G128 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 R182 R184 Y186 R187 R188 P189 A190 T202 R205 N206 A213 T214 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 P71 Q73 D74 R76 A77 R78 V80 P81 Q82 V84 K85 R87 H90 P92 K93 T94 E95 K96 D97 L100 D101 N103 D104 K105 E106 R107 Q108 R127 G128 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 R182 R184 Y186 R187 R188 P189 A190 T202 R205 N206 A213 T214 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18455733 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKQDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3cc4 D 2.7 BS01 rna 0 0 K20 V22 H24 T52 A54 R56 E60 K72 S96 Q97 F98 D99 D100 T101 S105 F106 G107 D129 N133 R156 K11 V13 H15 T38 A40 R42 E46 K58 S82 Q83 F84 D85 D86 T87 S91 F92 G93 D95 N99 R122 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3cc4 D 2.7 BS02 rna 9 0 E12 M13 R14 Q47 M48 V50 V73 T74 R76 P137 G138 R140 V141 K143 R144 D145 R149 P152 K154 H155 E3 M4 R5 Q33 M34 V36 V59 T60 R62 P103 G104 R106 V107 K109 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3cc4 E 2.7 BS01 rna 0 0 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 G142 Q143 A146 Q150 R153 N155 K157 D158 R160 V161 F162 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 G142 Q143 A146 Q150 R153 N155 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18455733 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3cc4 F 2.7 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18455733 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 3cc4 H 2.7 BS01 rna 0 0 K4 A6 M8 R10 K14 P15 A16 Y17 T18 R19 R20 E21 Y22 K35 K39 Q40 R61 S64 A67 R74 R91 K92 F93 H95 R99 E100 N101 M116 R117 A118 A119 F120 R154 R155 Y157 N158 K159 I160 T161 S163 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 K36 Q37 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M102 R103 A104 A105 F106 R140 R141 Y143 N144 K145 I146 T147 S149 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3cc4 H 2.7 BS02 rna 9 0 D11 E56 D8 E53 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 1 ~ 122 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3cc4 I 2.7 BS01 rna 0 0 P69 T70 T82 G83 S84 P87 D110 L111 L112 S113 Y114 N118 K121 E122 G125 T126 S129 P4 T5 T17 G18 S19 P22 D45 L46 L47 S48 Y49 N53 K56 E57 G60 T61 S64 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 18455733 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 3cc4 J 2.7 BS01 rna 0 0 I18 G20 R21 S24 L31 I46 T47 G48 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R74 K80 T82 R84 G85 M86 P88 H89 K90 K91 R95 E99 R102 V103 I127 K128 G140 I15 G17 R18 S21 L28 I43 T44 G45 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R71 K77 T79 R81 G82 M83 P85 H86 K87 K88 R92 E96 R99 V100 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18455733 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3cc4 K 2.7 BS01 rna 0 0 M1 A3 D7 T9 G11 E13 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 P45 T54 S56 R66 R77 K78 R81 R87 M1 A3 D7 T9 G11 E13 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 P45 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18455733 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3cc4 L 2.7 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 G34 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 K132 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 G34 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 K127 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18455733 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3cc4 M 2.7 BS01 rna 0 0 A1 S3 Y5 R9 K13 P15 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 T108 F109 P110 N111 N116 G124 K127 D135 N137 H138 P139 N143 D146 W149 Q155 A156 D157 F160 R161 L163 G165 R168 N170 R171 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 G192 K193 A1 S3 Y5 R9 K13 P15 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 T108 F109 P110 N111 N116 G124 K127 D135 N137 H138 P139 N143 D146 W149 Q155 A156 D157 F160 R161 L163 G165 R168 N170 R171 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 G192 K193 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 18455733 10 ~ 2914 ARSAYSYIRDAWKNPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKG 3cc4 N 2.7 BS01 rna 0 0 P4 R5 Y6 K7 P9 R13 A16 T18 H21 Q22 R25 L26 K28 S29 V101 I104 P109 F116 P130 N132 V135 P4 R5 Y6 K7 P9 R13 A16 T18 H21 Q22 R25 L26 K28 S29 V101 I104 P109 F116 P130 N132 V135 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3cc4 N 2.7 BS02 rna 9 0 A1 G3 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3cc4 O 2.7 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 S109 H110 V111 R112 I114 R115 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 S109 H110 V111 R112 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18455733 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3cc4 P 2.7 BS01 rna 0 0 T1 D2 L3 K7 R8 L9 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G127 G128 E130 S133 V134 T1 D2 L3 K7 R8 L9 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G127 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18455733 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3cc4 Q 2.7 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 R21 G22 T23 K38 H40 K42 S46 P48 G50 H53 R55 F56 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 R21 G22 T23 K38 H40 K42 S46 P48 G50 H53 R55 F56 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3cc4 Q 2.7 BS02 rna 9 0 R19 P25 Q27 R19 P25 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3cc4 R 2.7 BS01 rna 0 0 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18455733 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3cc4 S 2.7 BS01 rna 0 0 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18455733 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3cc4 T 2.7 BS01 rna 0 0 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 P90 S94 N95 R97 D105 K107 R111 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 P90 S94 N95 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18455733 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3cc4 U 2.7 BS01 rna 0 0 S34 K35 N38 L42 R44 E50 W51 R56 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18455733 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3cc4 V 2.7 BS01 rna 0 0 T1 H4 V5 E7 R9 Q34 P43 G44 K47 R50 K51 A54 R55 K57 T58 E62 T1 H4 V5 E7 R9 Q34 P43 G44 K47 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18455733 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3cc4 W 2.7 BS01 rna 0 0 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3cc4 W 2.7 BS02 rna 9 0 R8 H14 D50 F51 K129 H130 P131 K133 E134 R8 H14 D50 F51 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3cc4 X 2.7 BS01 rna 0 0 R8 T11 P13 R15 D16 R18 A19 P21 N22 H23 D27 K28 R34 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 S68 R2 T5 P7 R9 D10 R12 A13 P15 N16 H17 D21 K22 R28 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18455733 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3cc4 Y 2.7 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 N230 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 N136 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18455733 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3cc4 Z 2.7 BS01 rna 0 0 S34 G36 R37 G39 A40 R41 Y42 G43 R44 V45 R47 R70 R73 T76 Y83 Y93 S1 G3 R4 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 T43 Y50 Y60 ? 0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P60619 18455733 10 ~ 2914 SSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 3cc7 1 2.7 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 Q51 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 Q51 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18455733 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3cc7 2 2.7 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 R20 P22 W24 V25 K28 T29 D30 H37 K38 R40 H41 W42 R43 T47 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 R20 P22 W24 V25 K28 T29 D30 H34 K35 R37 H38 W39 R40 T44 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18455733 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 3cc7 3 2.7 BS01 rna 0 0 M1 Q2 M3 P4 N8 T9 Y10 H13 N15 E16 H17 V25 G28 R29 T31 M33 K34 W35 I36 R38 Q39 R42 N43 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 M1 Q2 M3 P4 N8 T9 Y10 H13 N15 E16 H17 V25 G28 R29 T31 M33 K34 W35 I36 R38 Q39 R42 N43 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18455733 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3cc7 A 2.7 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 R17 A18 S20 H21 Y23 K24 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 F201 G203 G204 R206 Q207 H208 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 R17 A18 S20 H21 Y23 K24 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 F201 G203 G204 R206 Q207 H208 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18455733 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3cc7 B 2.7 BS01 rna 0 0 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 Q94 R95 P96 L97 T98 E99 R111 T112 L113 D114 V115 P116 E117 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 S300 V301 P302 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 Q94 R95 P96 L97 T98 E99 R111 T112 L113 D114 V115 P116 E117 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 S300 V301 P302 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18455733 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3cc7 C 2.7 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 Q73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 S88 H90 P92 K93 T94 E95 K96 D97 L100 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 Q73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 S88 H90 P92 K93 T94 E95 K96 D97 L100 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18455733 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKQDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3cc7 D 2.7 BS01 rna 0 0 K20 V22 H24 T52 A54 R56 E60 K72 S96 Q97 D99 D100 T101 S105 F106 G107 D129 R156 K11 V13 H15 T38 A40 R42 E46 K58 S82 Q83 D85 D86 T87 S91 F92 G93 D95 R122 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3cc7 D 2.7 BS02 rna 9 0 E12 M13 R14 Q47 M48 V50 T74 R76 P137 G138 R140 V141 R144 D145 R149 P152 K154 H155 E3 M4 R5 Q33 M34 V36 T60 R62 P103 G104 R106 V107 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3cc7 E 2.7 BS01 rna 0 0 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 E110 K111 A112 H119 E139 G142 Q143 A146 R153 N155 K157 D158 R160 V161 F162 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 E110 K111 A112 H119 E139 G142 Q143 A146 R153 N155 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18455733 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3cc7 F 2.7 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18455733 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 3cc7 H 2.7 BS01 rna 0 0 K4 A6 M8 R10 K14 P15 A16 Y17 T18 R19 R20 E21 Y22 K35 R61 S64 A67 R74 R91 K92 F93 H95 R99 E100 N101 M116 R117 A118 A119 F120 G121 R154 R155 Y157 N158 K159 T161 S163 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M102 R103 A104 A105 F106 G107 R140 R141 Y143 N144 K145 T147 S149 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3cc7 H 2.7 BS02 rna 9 0 D11 E56 D8 E53 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 1 ~ 122 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3cc7 I 2.7 BS01 rna 0 0 P69 T70 G83 S84 E86 P87 E89 K107 D110 L111 L112 S113 Y114 N118 K121 E122 G125 T126 S129 L130 P4 T5 G18 S19 E21 P22 E24 K42 D45 L46 L47 S48 Y49 N53 K56 E57 G60 T61 S64 L65 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 18455733 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 3cc7 J 2.7 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 G48 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R74 K80 T82 R84 G85 M86 P88 K90 K91 R95 R102 V103 I127 K128 G140 I15 G17 R18 S21 L28 T44 G45 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R71 K77 T79 R81 G82 M83 P85 K87 K88 R92 R99 V100 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18455733 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3cc7 K 2.7 BS01 rna 0 0 M1 A3 D7 T9 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 M1 A3 D7 T9 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18455733 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3cc7 L 2.7 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 K132 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 K127 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18455733 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3cc7 M 2.7 BS01 rna 0 0 A1 S3 Y5 R9 K13 P15 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 N111 N116 G124 K127 D135 N137 H138 P139 A140 W149 A156 D157 F160 R161 L163 G165 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 A1 S3 Y5 R9 K13 P15 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 N111 N116 G124 K127 D135 N137 H138 P139 A140 W149 A156 D157 F160 R161 L163 G165 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 18455733 10 ~ 2914 ARSAYSYIRDAWKNPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKG 3cc7 N 2.7 BS01 rna 0 0 P4 Y6 K7 P9 R13 A16 T18 R25 L26 K28 S29 V101 P109 F116 P130 N132 V135 P4 Y6 K7 P9 R13 A16 T18 R25 L26 K28 S29 V101 P109 F116 P130 N132 V135 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3cc7 N 2.7 BS02 rna 9 0 A1 G3 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 K38 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 K38 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3cc7 O 2.7 BS01 rna 0 0 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R50 Y51 K63 L65 G66 S67 G68 S82 S109 H110 V111 R112 I114 R115 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R50 Y51 K63 L65 G66 S67 G68 S82 S109 H110 V111 R112 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18455733 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3cc7 P 2.7 BS01 rna 0 0 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 G60 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S117 Y119 R120 Y123 D124 G127 G128 E130 S133 V134 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 G60 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S117 Y119 R120 Y123 D124 G127 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18455733 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3cc7 Q 2.7 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 R21 G22 T23 K38 H40 K42 S46 P48 G50 H53 R55 F56 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 R21 G22 T23 K38 H40 K42 S46 P48 G50 H53 R55 F56 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3cc7 Q 2.7 BS02 rna 9 0 R19 Q27 R19 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3cc7 R 2.7 BS01 rna 0 0 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 A133 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 A133 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18455733 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3cc7 S 2.7 BS01 rna 0 0 S1 H9 T11 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 S1 H9 T11 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18455733 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3cc7 T 2.7 BS01 rna 0 0 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18455733 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3cc7 U 2.7 BS01 rna 0 0 S34 K35 N38 L42 R44 E50 W51 R56 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18455733 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3cc7 V 2.7 BS01 rna 0 0 T1 H4 V5 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 T1 H4 V5 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18455733 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3cc7 W 2.7 BS01 rna 0 0 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3cc7 W 2.7 BS02 rna 9 0 R8 H14 D50 K129 H130 P131 K133 E134 R8 H14 D50 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3cc7 X 2.7 BS01 rna 0 0 R8 T11 P13 R15 D16 R18 A19 P21 N22 H23 D27 K28 M30 R34 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 S68 K69 R2 T5 P7 R9 D10 R12 A13 P15 N16 H17 D21 K22 M24 R28 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 S62 K63 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18455733 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3cc7 Y 2.7 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 N230 P231 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 N136 P137 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18455733 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3cc7 Z 2.7 BS01 rna 0 0 S34 G36 R37 G39 A40 R41 Y42 G43 R44 V45 R47 R70 R73 T76 Y83 Y93 S1 G3 R4 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 T43 Y50 Y60 ? 0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P60619 18455733 10 ~ 2914 SSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 3ccb A 2.49 BS01 B2Y A 1 R125 E205 E206 Y547 S630 Y662 Y666 R83 E163 E164 Y505 S588 Y620 Y624 Y547 S630 Y631 D708 H740 Y505 S588 Y589 D666 H698 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=30uM remove_due_to_license_issue IC50=30000nM P27487 18346892 800 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3ccc A 2.71 BS01 7AC A 1 E205 E206 Y547 S630 Y631 Y662 Y666 N710 E163 E164 Y505 S588 Y589 Y620 Y624 N668 Y547 S630 Y631 D708 H740 Y505 S588 Y589 D666 H698 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=8nM P27487 18346892 800 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3ccm 1 2.55 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 F39 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 K25 S26 Y27 H28 T29 K30 K31 K32 S35 F39 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18455733 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3ccm 2 2.55 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R31 N36 H37 K38 R40 H41 W42 R43 D46 T47 E49 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R31 N33 H34 K35 R37 H38 W39 R40 D43 T44 E46 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18455733 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 3ccm 3 2.55 BS01 rna 0 0 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 S27 G28 R29 T31 M33 K34 W35 I36 R38 Q39 R42 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 D66 K68 K76 A77 L79 R80 G82 R84 G86 Q91 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 S27 G28 R29 T31 M33 K34 W35 I36 R38 Q39 R42 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 D66 K68 K76 A77 L79 R80 G82 R84 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18455733 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3ccm A 2.55 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S110 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 F201 G203 G204 G205 R206 Q207 H208 P209 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G237 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S110 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 F201 G203 G204 G205 R206 Q207 H208 P209 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G237 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18455733 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3ccm B 2.55 BS01 rna 0 0 P1 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 Q94 P96 L97 E99 R111 T112 L113 D114 V115 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 V220 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 K267 G282 V285 N286 G288 S300 V301 P302 G303 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 P1 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 Q94 P96 L97 E99 R111 T112 L113 D114 V115 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 V220 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 K267 G282 V285 N286 G288 S300 V301 P302 G303 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18455733 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3ccm C 2.55 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 R65 G66 Q67 A68 H69 Q73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 S88 H90 P92 K93 T94 K96 D97 L100 D101 N103 D104 K105 E106 R107 Q108 R127 V148 K149 T150 Q151 R168 K173 I174 K175 A176 G177 Q178 R182 R184 Y186 R187 R188 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 R65 G66 Q67 A68 H69 Q73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 S88 H90 P92 K93 T94 K96 D97 L100 D101 N103 D104 K105 E106 R107 Q108 R127 V148 K149 T150 Q151 R168 K173 I174 K175 A176 G177 Q178 R182 R184 Y186 R187 R188 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18455733 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKQDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3ccm D 2.55 BS01 rna 0 0 K20 H24 T52 R56 E60 K72 S96 Q97 D99 D100 T101 S105 F106 G107 D129 R156 K11 H15 T38 R42 E46 K58 S82 Q83 D85 D86 T87 S91 F92 G93 D95 R122 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccm D 2.55 BS02 rna 9 0 E12 M13 R14 Q47 M48 V50 T74 R76 P137 R140 V141 K143 R144 D145 R149 P152 K154 H155 E3 M4 R5 Q33 M34 V36 T60 R62 P103 R106 V107 K109 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccm E 2.55 BS01 rna 0 0 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 Q143 A146 D147 Q150 R153 N155 K157 D158 R160 V161 F162 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 Q143 A146 D147 Q150 R153 N155 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18455733 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3ccm F 2.55 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18455733 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 3ccm H 2.55 BS01 rna 0 0 K4 A6 M8 R10 K14 P15 A16 Y17 T18 R19 R20 E21 Y22 K35 K39 Q40 R61 S64 A67 R74 R91 K92 F93 H95 R99 E100 N101 M116 R117 A118 A119 F120 R154 R155 Y157 N158 K159 I160 T161 S163 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 K36 Q37 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M102 R103 A104 A105 F106 R140 R141 Y143 N144 K145 I146 T147 S149 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3ccm I 2.55 BS01 rna 0 0 P69 T70 T82 G83 G85 E86 P87 E89 D110 L111 S113 Y114 N118 K121 E122 G125 S129 L130 P4 T5 T17 G18 G20 E21 P22 E24 D45 L46 S48 Y49 N53 K56 E57 G60 S64 L65 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 18455733 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 3ccm J 2.55 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 G48 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 K80 R81 T82 R84 G85 M86 P88 K90 R95 E99 R102 V103 Y104 I127 K128 G140 I15 G17 R18 S21 L28 T44 G45 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 K77 R78 T79 R81 G82 M83 P85 K87 R92 E96 R99 V100 Y101 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18455733 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3ccm K 2.55 BS01 rna 0 0 M1 A3 D7 T9 G11 E13 K14 S16 K30 I32 S33 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 M1 A3 D7 T9 G11 E13 K14 S16 K30 I32 S33 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18455733 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3ccm L 2.55 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 T63 D65 R67 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 K132 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 T63 D65 R67 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 K127 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18455733 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3ccm M 2.55 BS01 rna 0 0 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 N111 N116 G124 K127 D135 N137 H138 P139 A140 N143 W149 A156 D157 F160 R161 L163 G165 R168 N170 R171 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 N111 N116 G124 K127 D135 N137 H138 P139 A140 N143 W149 A156 D157 F160 R161 L163 G165 R168 N170 R171 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 18455733 10 ~ 2914 ARSAYSYIRDAWKNPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKG 3ccm N 2.55 BS01 rna 0 0 P4 Y6 K7 P9 R13 A16 T18 H21 Q22 R25 L26 K28 S29 V101 P109 F116 P130 N132 P4 Y6 K7 P9 R13 A16 T18 H21 Q22 R25 L26 K28 S29 V101 P109 F116 P130 N132 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccm N 2.55 BS02 rna 9 0 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccm O 2.55 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 V111 R112 V113 I114 R115 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 V111 R112 V113 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18455733 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3ccm P 2.55 BS01 rna 0 0 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18455733 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3ccm Q 2.55 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 N16 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 N16 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccm Q 2.55 BS02 rna 9 0 R19 P25 Q27 R19 P25 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccm R 2.55 BS01 rna 0 0 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K60 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 P81 E82 K83 E93 N94 N98 H101 H113 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K60 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 P81 E82 K83 E93 N94 N98 H101 H113 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18455733 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3ccm S 2.55 BS01 rna 0 0 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18455733 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3ccm T 2.55 BS01 rna 0 0 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 D83 V87 R89 S94 N95 R97 D105 K107 R111 D116 D117 S118 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 D83 V87 R89 S94 N95 R97 D105 K107 R111 D116 D117 S118 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18455733 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3ccm U 2.55 BS01 rna 0 0 G18 S34 K35 N38 L42 R44 E50 W51 R56 G15 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18455733 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3ccm V 2.55 BS01 rna 0 0 T1 H4 V5 R9 Q34 G44 R50 K51 A54 R55 K57 T58 E62 T1 H4 V5 R9 Q34 G44 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18455733 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3ccm W 2.55 BS01 rna 0 0 R8 G9 V11 N12 H14 T15 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 G75 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 R8 G9 V11 N12 H14 T15 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 G75 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccm W 2.55 BS02 rna 9 0 R8 H14 D50 F51 K129 H130 P131 K133 E134 R8 H14 D50 F51 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccm X 2.55 BS01 rna 0 0 T11 P13 R15 R18 A19 P21 N22 H23 D27 K28 M30 R34 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 S68 T5 P7 R9 R12 A13 P15 N16 H17 D21 K22 M24 R28 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18455733 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3ccm Y 2.55 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 R204 A206 S207 K208 G210 A211 R212 K213 N230 P231 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 R110 A112 S113 K114 G116 A117 R118 K119 N136 P137 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18455733 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3ccm Z 2.55 BS01 rna 0 0 S34 G36 R37 G39 A40 R41 Y42 G43 R44 V45 R47 R70 R73 T76 Y83 S1 G3 R4 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 T43 Y50 ? 0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P60619 18455733 10 ~ 2914 SSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 3ccn A 1.9 BS01 LKG A 1 A1108 L1157 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 A48 L87 M90 D94 R138 M141 A151 D152 Y160 D1204 A1206 R1208 N1209 D1222 A1243 D134 A136 R138 N139 D152 A172 2.7.10.1 0004672,0004713,0005524,0006468 ic50=120nM remove_due_to_license_issue IC50=120nM P08581 18426196 1 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNREVSQFLTEGIIMKDFSHPNVLSLLGICLPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 3ccq 1 2.9 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18455733 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3ccq 2 2.9 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R35 N36 H37 K38 R40 H41 W42 R43 R44 T47 E49 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R32 N33 H34 K35 R37 H38 W39 R40 R41 T44 E46 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18455733 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 3ccq 3 2.9 BS01 rna 0 0 M1 Q2 M3 P4 N8 T9 Y10 N15 E16 H17 V25 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 M1 Q2 M3 P4 N8 T9 Y10 N15 E16 H17 V25 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18455733 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3ccq A 2.9 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 F201 G203 G204 R206 Q207 H208 P209 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 F201 G203 G204 R206 Q207 H208 P209 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18455733 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3ccq B 2.9 BS01 rna 0 0 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 G93 Q94 P96 L97 T98 E99 W101 R111 T112 L113 D114 V115 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 R217 Q221 K222 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 S300 V301 P302 G303 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 G93 Q94 P96 L97 T98 E99 W101 R111 T112 L113 D114 V115 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 R217 Q221 K222 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 S300 V301 P302 G303 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18455733 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3ccq C 2.9 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 P71 Q73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 H90 P92 K93 E95 K96 L100 D101 N103 D104 K105 E106 R107 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 P189 A190 T202 R205 N206 A213 T214 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 P71 Q73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 H90 P92 K93 E95 K96 L100 D101 N103 D104 K105 E106 R107 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 P189 A190 T202 R205 N206 A213 T214 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18455733 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKQDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3ccq D 2.9 BS01 rna 0 0 K20 V22 H24 T52 A54 R56 E60 K72 S96 Q97 D99 D100 T101 S105 F106 D129 T131 N133 R156 K11 V13 H15 T38 A40 R42 E46 K58 S82 Q83 D85 D86 T87 S91 F92 D95 T97 N99 R122 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccq D 2.9 BS02 rna 9 0 M13 R14 Q47 M48 V50 V73 T74 R76 P137 G138 R140 V141 R144 D145 R149 P152 K154 H155 M4 R5 Q33 M34 V36 V59 T60 R62 P103 G104 R106 V107 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccq E 2.9 BS01 rna 0 0 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 E139 G142 Q143 A146 Q150 R153 N155 K157 D158 R160 V161 F162 Y35 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 E139 G142 Q143 A146 Q150 R153 N155 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18455733 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3ccq F 2.9 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18455733 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 3ccq H 2.9 BS01 rna 0 0 K4 A6 M8 R10 K14 P15 A16 Y17 T18 R19 R20 E21 Y22 K35 K39 Q40 R61 S64 A67 R74 R91 K92 F93 H95 R99 E100 N101 M116 R117 A118 A119 F120 G121 R154 R155 Y157 N158 K159 I160 T161 S163 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 K36 Q37 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M102 R103 A104 A105 F106 G107 R140 R141 Y143 N144 K145 I146 T147 S149 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3ccq I 2.9 BS01 rna 0 0 P69 T70 G83 S84 E86 P87 E89 K107 D110 L111 L112 S113 Y114 N118 K121 E122 G125 S129 L130 P4 T5 G18 S19 E21 P22 E24 K42 D45 L46 L47 S48 Y49 N53 K56 E57 G60 S64 L65 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 18455733 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 3ccq J 2.9 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 G48 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R74 K80 T82 R84 G85 M86 P88 K90 K91 R95 E99 R102 V103 Y104 I127 K128 G140 I15 G17 R18 S21 L28 T44 G45 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R71 K77 T79 R81 G82 M83 P85 K87 K88 R92 E96 R99 V100 Y101 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18455733 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3ccq K 2.9 BS01 rna 0 0 M1 A3 T9 G11 E13 S16 K30 I32 S33 V34 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 M1 A3 T9 G11 E13 S16 K30 I32 S33 V34 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18455733 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3ccq L 2.9 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 T63 D65 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 T63 D65 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18455733 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3ccq M 2.9 BS01 rna 0 0 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 H77 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 P110 N111 N116 G124 R125 K127 D135 N137 H138 P139 A140 N143 W149 D157 F160 R161 L163 G165 R168 N170 R171 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 S189 G191 K193 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 H77 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 V100 R104 R107 F109 P110 N111 N116 G124 R125 K127 D135 N137 H138 P139 A140 N143 W149 D157 F160 R161 L163 G165 R168 N170 R171 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 S189 G191 K193 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 18455733 10 ~ 2914 ARSAYSYIRDAWKNPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKG 3ccq N 2.9 BS01 rna 0 0 Y6 K7 R13 T18 H21 Q22 R25 L26 K28 S29 V101 I104 P109 P130 N132 Y6 K7 R13 T18 H21 Q22 R25 L26 K28 S29 V101 I104 P109 P130 N132 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccq N 2.9 BS02 rna 9 0 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccq O 2.9 BS01 rna 0 0 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 G83 T84 S109 H110 V111 R112 I114 R115 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 G83 T84 S109 H110 V111 R112 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18455733 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3ccq P 2.9 BS01 rna 0 0 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 G60 R61 R63 R65 Q66 K68 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 G60 R61 R63 R65 Q66 K68 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18455733 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3ccq Q 2.9 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 H53 R55 F56 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 H53 R55 F56 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccq Q 2.9 BS02 rna 9 0 R19 P25 Q27 R19 P25 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccq R 2.9 BS01 rna 0 0 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18455733 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3ccq S 2.9 BS01 rna 0 0 S1 H9 T11 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 S1 H9 T11 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18455733 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3ccq T 2.9 BS01 rna 0 0 S1 K2 Q3 P4 D5 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 S1 K2 Q3 P4 D5 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18455733 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3ccq U 2.9 BS01 rna 0 0 T17 S34 K35 N38 L42 R44 E50 W51 R56 T14 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18455733 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3ccq V 2.9 BS01 rna 0 0 T1 H4 V5 E7 R9 Q34 P43 R50 K51 A54 R55 K57 T58 E62 T1 H4 V5 E7 R9 Q34 P43 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18455733 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3ccq W 2.9 BS01 rna 0 0 R8 G9 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 R8 G9 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccq W 2.9 BS02 rna 9 0 R8 H14 D50 K129 H130 P131 K133 E134 R8 H14 D50 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccq X 2.9 BS01 rna 0 0 R8 T11 R15 D16 R18 A19 P21 N22 H23 D27 K28 R34 K39 H40 R49 L50 N55 E56 W59 R61 R63 S68 R2 T5 R9 D10 R12 A13 P15 N16 H17 D21 K22 R28 K33 H34 R43 L44 N49 E50 W53 R55 R57 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18455733 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3ccq Y 2.9 BS01 rna 0 0 R115 Q119 R120 H121 R122 V123 K125 P126 Q127 F128 R130 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 N230 P231 Y233 R21 Q25 R26 H27 R28 V29 K31 P32 Q33 F34 R36 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 N136 P137 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18455733 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3ccq Z 2.9 BS01 rna 0 0 S34 G36 R37 G39 A40 R41 Y42 G43 R44 V45 R47 R70 R73 G75 T76 Y83 Y93 S1 G3 R4 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 G42 T43 Y50 Y60 ? 0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P60619 18455733 10 ~ 2914 SSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 3ccr 1 3.0 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 G23 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 G23 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18455733 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3ccr 2 3.0 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 K9 R10 L11 K13 N16 Q17 S19 V21 P22 W24 V25 L27 K28 T29 D30 R35 H37 K38 R40 H41 W42 R43 T47 G1 K2 K3 K5 A6 K8 K9 R10 L11 K13 N16 Q17 S19 V21 P22 W24 V25 L27 K28 T29 D30 R32 H34 K35 R37 H38 W39 R40 T44 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18455733 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 3ccr 3 3.0 BS01 rna 0 0 M1 Q2 N8 Y10 H13 E16 H17 S27 G28 R29 Q30 T31 M33 W35 I36 R38 Q39 R42 G45 I46 G47 N48 D49 G50 K51 K54 G58 D59 K60 P61 T62 K63 K64 T65 K68 K76 L79 R80 E81 G82 W83 R84 G86 Q91 M1 Q2 N8 Y10 H13 E16 H17 S27 G28 R29 Q30 T31 M33 W35 I36 R38 Q39 R42 G45 I46 G47 N48 D49 G50 K51 K54 G58 D59 K60 P61 T62 K63 K64 T65 K68 K76 L79 R80 E81 G82 W83 R84 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18455733 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3ccr A 3.0 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 S20 H21 R22 Y23 A25 D26 K31 H47 P49 R51 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 A196 V197 D198 H199 F201 G203 G204 R206 Q207 H208 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 V225 G226 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 S20 H21 R22 Y23 A25 D26 K31 H47 P49 R51 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 A196 V197 D198 H199 F201 G203 G204 R206 Q207 H208 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 V225 G226 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18455733 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3ccr B 3.0 BS01 rna 0 0 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 P15 R16 K17 R18 T20 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 Q94 R95 P96 L97 T98 E99 W101 R111 T112 L113 D114 V115 P116 E117 R141 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 G255 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 K298 S300 V301 P302 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 P15 R16 K17 R18 T20 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 Q94 R95 P96 L97 T98 E99 W101 R111 T112 L113 D114 V115 P116 E117 R141 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 G255 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 K298 S300 V301 P302 P304 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18455733 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3ccr C 3.0 BS01 rna 0 0 R27 L30 A38 N41 R42 K43 Q44 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 Q73 D74 R76 A77 R78 V80 P81 Q82 A83 V84 K85 R87 S88 H90 P92 K93 T94 K96 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 R188 P189 A190 T202 R205 N206 A208 A213 E217 V218 N219 D222 P225 G226 R246 R27 L30 A38 N41 R42 K43 Q44 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 Q73 D74 R76 A77 R78 V80 P81 Q82 A83 V84 K85 R87 S88 H90 P92 K93 T94 K96 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 R188 P189 A190 T202 R205 N206 A208 A213 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18455733 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKQDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3ccr D 3.0 BS01 rna 0 0 K20 V22 H24 T52 R56 E60 K72 S96 Q97 T101 F104 S105 F106 G107 D129 N133 K11 V13 H15 T38 R42 E46 K58 S82 Q83 T87 F90 S91 F92 G93 D95 N99 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccr D 3.0 BS02 rna 9 0 E12 M13 R14 M48 P49 V50 K72 V73 T74 R76 P137 G138 R140 V141 K143 R144 D145 R149 P152 K154 H155 E3 M4 R5 M34 P35 V36 K58 V59 T60 R62 P103 G104 R106 V107 K109 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccr E 3.0 BS01 rna 0 0 Y35 N55 A56 K57 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 I138 E139 Q143 A146 R153 K157 D158 R160 V161 F162 Y35 N55 A56 K57 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 I138 E139 Q143 A146 R153 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18455733 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3ccr F 3.0 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 E90 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 E90 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18455733 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 3ccr H 3.0 BS01 rna 0 0 K4 A6 M8 R10 K14 P15 A16 Y17 T18 R19 R20 Y22 K35 K39 R61 G63 S64 A67 R74 R91 K92 F93 H95 R99 E100 M116 R117 A118 A119 F120 R154 R155 Y157 N158 K159 I160 T161 S163 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 Y19 K32 K36 R58 G60 S61 A64 R71 R88 K89 F90 H92 R96 E97 M102 R103 A104 A105 F106 R140 R141 Y143 N144 K145 I146 T147 S149 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3ccr H 3.0 BS02 rna 9 0 D11 E56 D8 E53 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 1 ~ 122 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3ccr I 3.0 BS01 rna 0 0 P69 T70 T82 G83 S84 P87 Q88 E89 D110 L111 L112 S113 Y114 K121 E122 G125 S129 L130 P4 T5 T17 G18 S19 P22 Q23 E24 D45 L46 L47 S48 Y49 K56 E57 G60 S64 L65 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 18455733 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 3ccr J 3.0 BS01 rna 0 0 I18 G20 R21 S24 T47 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R81 T82 R84 G85 M86 P88 H89 K90 K91 R93 R95 E99 R102 V103 I127 K128 G140 I15 G17 R18 S21 T44 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R78 T79 R81 G82 M83 P85 H86 K87 K88 R90 R92 E96 R99 V100 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18455733 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3ccr K 3.0 BS01 rna 0 0 M1 A3 D7 T9 Q10 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 M1 A3 D7 T9 Q10 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18455733 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3ccr L 3.0 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 R30 G31 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 Q55 K56 V57 T63 D65 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 K132 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 R30 G31 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 Q55 K56 V57 T63 D65 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 K127 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18455733 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3ccr M 3.0 BS01 rna 0 0 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 A56 K57 Q58 I61 R68 G70 S71 R73 K74 R76 K78 G80 R81 R82 S83 K84 R85 Q86 V88 R90 I91 T92 R93 R94 K95 D96 I97 R99 R104 R107 F109 P110 N111 N116 G124 D135 N137 H138 P139 A140 D146 W149 D157 F160 R161 L163 G165 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 A56 K57 Q58 I61 R68 G70 S71 R73 K74 R76 K78 G80 R81 R82 S83 K84 R85 Q86 V88 R90 I91 T92 R93 R94 K95 D96 I97 R99 R104 R107 F109 P110 N111 N116 G124 D135 N137 H138 P139 A140 D146 W149 D157 F160 R161 L163 G165 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 K193 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 18455733 10 ~ 2914 ARSAYSYIRDAWKNPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKG 3ccr N 3.0 BS01 rna 0 0 P4 R5 Y6 K7 R13 A16 T18 D19 H21 Q22 R25 L26 K28 S29 I104 L106 P109 F116 P130 N132 V135 P4 R5 Y6 K7 R13 A16 T18 D19 H21 Q22 R25 L26 K28 S29 I104 L106 P109 F116 P130 N132 V135 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccr N 3.0 BS02 rna 9 0 A1 G3 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 G112 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 G112 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccr O 3.0 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 G46 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 V111 R112 V113 I114 R115 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 G46 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 V111 R112 V113 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18455733 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3ccr P 3.0 BS01 rna 0 0 T1 D2 K7 R8 L9 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S117 Y119 R120 Y123 D124 K125 G128 E130 S133 V134 T1 D2 K7 R8 L9 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S117 Y119 R120 Y123 D124 K125 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18455733 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3ccr Q 3.0 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 N16 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 G12 K13 K15 N16 R21 G22 T23 K38 H40 K42 P45 S46 P48 G50 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccr Q 3.0 BS02 rna 9 0 R19 P25 Q27 R19 P25 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccr R 3.0 BS01 rna 0 0 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 V66 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 A115 A116 H117 V119 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 K15 M17 R19 S24 F25 K26 K29 K36 K60 Q61 H62 S64 G65 V66 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 A115 A116 H117 V119 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18455733 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3ccr S 3.0 BS01 rna 0 0 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 S1 H9 T11 E12 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18455733 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3ccr T 3.0 BS01 rna 0 0 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 D116 S1 K2 Q3 P4 D5 K6 Q7 R8 K9 Q11 R12 R13 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 D116 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18455733 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3ccr U 3.0 BS01 rna 0 0 T17 S34 K35 N38 L42 R44 E50 W51 R56 T14 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18455733 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3ccr V 3.0 BS01 rna 0 0 T1 H4 V5 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 T1 H4 V5 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18455733 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3ccr W 3.0 BS01 rna 0 0 R8 G9 E10 V11 N12 T15 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 R8 G9 E10 V11 N12 T15 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccr W 3.0 BS02 rna 9 0 R8 H14 N49 D50 F51 K129 H130 P131 K133 E134 R8 H14 N49 D50 F51 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccr X 3.0 BS01 rna 0 0 T11 R15 D16 R18 A19 P21 N22 H23 D27 K28 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 N65 S68 T5 R9 D10 R12 A13 P15 N16 H17 D21 K22 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 N59 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18455733 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3ccr Y 3.0 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18455733 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3ccr Z 3.0 BS01 rna 0 0 S34 G36 R37 F38 G39 A40 R41 Y42 G43 R44 V45 R47 R70 R73 T76 Y83 Y93 S1 G3 R4 F5 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 T43 Y50 Y60 ? 0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P60619 18455733 10 ~ 2914 SSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 3cct A 2.12 BS01 3HI B 1 E559 C561 S565 R568 K735 A751 L853 A856 L857 H861 E119 C121 S125 R128 K295 A311 L413 A416 L417 H421 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cct A 2.12 BS02 3HI B 2 R590 V683 S684 D690 K691 K692 R150 V243 S244 D250 K251 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cct B 2.12 BS01 3HI B 1 R590 V683 S684 D690 K692 R150 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=27.4nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cct B 2.12 BS02 3HI B 2 E559 C561 S565 R568 K735 A751 L853 A856 L857 E119 C121 S125 R128 K295 A311 L413 A416 L417 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=27.4nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3ccv 1 2.9 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 C22 G23 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 A43 K44 R45 R46 Y48 E49 W50 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18455733 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3ccv 2 2.9 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 N36 H37 K38 R40 H41 W42 R43 R44 T47 E49 G1 K2 K3 K5 A6 K8 R10 L11 K13 Q17 S19 P22 W24 V25 L27 K28 T29 D30 N33 H34 K35 R37 H38 W39 R40 R41 T44 E46 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18455733 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDRRNHKRRHWRRNDTDE 3ccv 3 2.9 BS01 rna 0 0 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 K68 K76 A77 L79 R80 E81 G82 R84 A85 G86 Q91 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 T65 K68 K76 A77 L79 R80 E81 G82 R84 A85 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18455733 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3ccv A 2.9 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 K24 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 G203 G204 R206 Q207 H208 P209 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 R22 Y23 K24 A25 D26 K31 H47 R51 S52 S111 G113 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 M194 N195 V197 D198 H199 G203 G204 R206 Q207 H208 P209 G210 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 D227 I228 A229 S230 K231 R232 T233 G234 R235 G236 G237 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18455733 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVSAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVAGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3ccv B 2.9 BS01 rna 0 0 P1 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 G93 Q94 P96 L97 T98 E99 W101 R111 T112 L113 D114 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 S300 V301 P302 G303 P304 R307 R312 R316 N318 S334 N335 Q336 G337 P1 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 G14 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 P70 R85 Y87 Y92 G93 Q94 P96 L97 T98 E99 W101 R111 T112 L113 D114 P116 E117 H119 R141 P155 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 D281 G282 V285 N286 G288 E289 S300 V301 P302 G303 P304 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18455733 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3ccv C 2.9 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 P71 Q73 D74 R76 A77 V80 P81 Q82 V84 K85 R87 S88 H90 P92 K93 T94 E95 K96 L100 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 A190 T202 R205 N206 A213 T214 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 V70 P71 Q73 D74 R76 A77 V80 P81 Q82 V84 K85 R87 S88 H90 P92 K93 T94 E95 K96 L100 D101 N103 D104 K105 E106 R107 Q108 R127 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 A190 T202 R205 N206 A213 T214 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18455733 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKQDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3ccv D 2.9 BS01 rna 0 0 K20 H24 T52 K53 A54 R56 E60 K72 S96 Q97 D99 D100 T101 S105 F106 G107 D129 T131 N133 K11 H15 T38 K39 A40 R42 E46 K58 S82 Q83 D85 D86 T87 S91 F92 G93 D95 T97 N99 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccv D 2.9 BS02 rna 9 0 E12 M13 Q47 M48 P49 V50 V73 T74 R76 P137 G138 R140 V141 R144 D145 P152 K154 H155 E3 M4 Q33 M34 P35 V36 V59 T60 R62 P103 G104 R106 V107 R110 D111 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18455733 1 ~ 122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3ccv E 2.9 BS01 rna 0 0 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 Q143 A146 Q150 R153 K157 D158 R160 V161 F162 N55 A56 S60 G63 T64 S67 H68 N71 Y82 H90 F91 G109 E110 K111 A112 H119 E139 Q143 A146 Q150 R153 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18455733 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3ccv F 2.9 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18455733 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGEADADVEDIADKVEELR 3ccv H 2.9 BS01 rna 0 0 K4 A6 M8 R10 K14 P15 A16 Y17 T18 R19 R20 E21 Y22 K35 K39 Q40 R61 S64 A67 R74 R91 K92 F93 H95 R99 E100 N101 M116 R117 A118 A119 F120 G121 R154 R155 Y157 N158 K159 T161 S163 L174 K1 A3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 E18 Y19 K32 K36 Q37 R58 S61 A64 R71 R88 K89 F90 H92 R96 E97 N98 M102 R103 A104 A105 F106 G107 R140 R141 Y143 N144 K145 T147 S149 L160 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 10 ~ 2914 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3ccv H 2.9 BS02 rna 9 0 D11 E56 D8 E53 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P60617 18455733 1 ~ 122 KPASMYRDIDKPAYTRREYITGIPGSKIAQHKMGRKQKDADDYPVQISLIVEETVQLRHGSLEASRLSANRHLIKELGEEGDYKMTLRKFPHQVLRENKDGMRAAFGKIVGTAARVQAGEQLFTAYCNVEDAEHVKEAFRRAYNKITPSCRIKVERGEEL 3ccv I 2.9 BS01 rna 0 0 P69 T70 G83 S84 E86 P87 E89 K107 D110 L111 L112 S113 Y114 N118 K121 E122 G125 T126 S129 L130 P4 T5 G18 S19 E21 P22 E24 K42 D45 L46 L47 S48 Y49 N53 K56 E57 G60 T61 S64 L65 ? 0003735,0005840,0006412,0015934,0019843,0070180,1990904 remove_due_to_license_issue P14122 18455733 10 ~ 2914 GVPPTAELIKDEAGFETGSGEPQEDFVADLSVDQVKQIAEQKHPDLLSYDLTNAAKEVVGTCTSLGVTIE 3ccv J 2.9 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R74 K80 T82 R84 G85 M86 P88 K90 K91 R93 R95 E99 R102 V103 I127 K128 G140 I15 G17 R18 S21 L28 T44 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R71 K77 T79 R81 G82 M83 P85 K87 K88 R90 R92 E96 R99 V100 I124 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18455733 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3ccv K 2.9 BS01 rna 0 0 M1 A3 T9 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 M1 A3 T9 G11 E13 K14 S16 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 T54 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18455733 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3ccv L 2.9 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 A33 G34 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 Q55 K56 V57 D65 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 K132 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 A33 G34 R35 K37 H38 E39 F40 H41 L46 G47 K48 G50 F51 K52 R53 P54 Q55 K56 V57 D65 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 K127 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18455733 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3ccv M 2.9 BS01 rna 0 0 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 R104 R107 F109 P110 N111 N116 G124 K127 D135 N137 H138 P139 A140 N143 D146 W149 D157 F160 R161 L163 G165 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 G192 K193 A1 S3 Y5 R9 K13 W25 Q29 R32 G35 A36 R39 R42 R45 L46 K48 R50 S51 Q52 K55 A56 Q58 I61 R68 K69 G70 S71 R73 K74 R75 R76 K78 A79 G80 R81 R82 S83 K84 R85 Q86 V88 T89 R90 T92 R93 R94 K95 D96 I97 R99 R104 R107 F109 P110 N111 N116 G124 K127 D135 N137 H138 P139 A140 N143 D146 W149 D157 F160 R161 L163 G165 R168 N170 R171 G172 K176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 G192 K193 ? 0002181,0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P60618 18455733 10 ~ 2914 ARSAYSYIRDAWKNPGDGQLAELQWQRQQEWRNEGAVERIERPTRLDKARSQGYKAKQGVIVARVSVRKGSARKRRHKAGRRSKRQGVTRITRRKDIQRVAEERASRTFPNLRVLNSYSVGQDGRQKWHEVILIDPNHPAIQNDDDLSWICADDQADRVFRGLTGAGRRNRGLSGKGKGSEKTRPSLRSNGGKG 3ccv N 2.9 BS01 rna 0 0 P4 R5 Y6 K7 R13 A16 T18 D19 H21 Q22 R25 L26 K28 S29 V101 I104 P109 F116 P130 N132 V135 P4 R5 Y6 K7 R13 A16 T18 D19 H21 Q22 R25 L26 K28 S29 V101 I104 P109 F116 P130 N132 V135 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccv N 2.9 BS02 rna 9 0 A1 G3 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 K38 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 A1 G3 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 K38 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 S60 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18455733 1 ~ 122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3ccv O 2.9 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 G83 S109 H110 V111 R112 I114 R115 S1 K2 T3 N4 A12 K15 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 R47 R50 Y51 K63 L65 G66 S67 G68 S82 G83 S109 H110 V111 R112 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18455733 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3ccv P 2.9 BS01 rna 0 0 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 G60 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 G60 R61 R63 R65 Q66 K68 R69 A70 Y71 H73 Q74 K75 G76 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G128 E130 S133 V134 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18455733 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAYGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3ccv Q 2.9 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 N16 R21 G22 T23 K38 H40 K42 S46 P48 G50 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 N16 R21 G22 T23 K38 H40 K42 S46 P48 G50 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccv Q 2.9 BS02 rna 9 0 R19 Q27 R19 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18455733 1 ~ 122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3ccv R 2.9 BS01 rna 0 0 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K36 K60 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K36 K60 H62 S64 G65 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18455733 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3ccv S 2.9 BS01 rna 0 0 S1 H9 T11 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 S1 H9 T11 K13 Q21 K23 S33 K34 N53 T54 Q55 N56 M58 K62 K63 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18455733 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3ccv T 2.9 BS01 rna 0 0 S1 K2 Q3 P4 D5 K6 Q7 R8 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 S1 K2 Q3 P4 D5 K6 Q7 R8 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 K69 L79 K81 T82 V87 R89 S94 N95 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18455733 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3ccv U 2.9 BS01 rna 0 0 T17 S34 K35 N38 L42 R44 E50 W51 R56 T14 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18455733 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3ccv V 2.9 BS01 rna 0 0 T1 H4 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 T1 H4 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18455733 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3ccv W 2.9 BS01 rna 0 0 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 R8 G9 E10 V11 N12 T15 D16 D19 T20 M23 N25 H27 H28 V29 N30 H31 D39 A40 Y41 G43 M44 K47 R69 E74 G75 R108 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccv W 2.9 BS02 rna 9 0 R8 H14 D50 K129 H130 P131 K133 E134 R8 H14 D50 K129 H130 P131 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18455733 1 ~ 122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3ccv X 2.9 BS01 rna 0 0 T11 R15 D16 R18 A19 P21 N22 H23 D27 K28 M30 R34 K39 H40 R49 L50 P52 N55 E56 W59 R61 R63 S68 T5 R9 D10 R12 A13 P15 N16 H17 D21 K22 M24 R28 K33 H34 R43 L44 P46 N49 E50 W53 R55 R57 S62 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18455733 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3ccv Y 2.9 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 N230 P231 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 N136 P137 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18455733 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3ccv Z 2.9 BS01 rna 0 0 S34 G36 R37 G39 A40 R41 Y42 G43 R44 V45 R47 R70 R73 G75 T76 Y83 Y93 S1 G3 R4 G6 A7 R8 Y9 G10 R11 V12 R14 R37 R40 G42 T43 Y50 Y60 ? 0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P60619 18455733 10 ~ 2914 SSGRFGARYGRVSRRRVAEIESEMNEDHACPNCGEDRVDRQGTGIWQCSYCDYKFTGGSYKPETPGGKTVRRS 3ccw A 2.1 BS01 4HI B 1 E559 C561 S565 R568 K735 A751 L853 E119 C121 S125 R128 K295 A311 L413 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3ccw A 2.1 BS02 4HI B 2 R590 S661 S684 D690 K692 R150 S221 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3ccw B 2.1 BS01 4HI B 1 R590 S661 V683 S684 D690 K692 R150 S221 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=13.5nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3ccw B 2.1 BS02 4HI B 2 E559 S565 K735 A751 H752 L853 E119 S125 K295 A311 H312 L413 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=13.5nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3ccz A 1.7 BS01 5HI A 1 R590 S661 S684 D690 K692 R150 S221 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=51.7nM remove_due_to_license_issue P04035 18540668 876 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 3ccz A 1.7 BS02 5HI B 1 E559 C561 A564 S565 K735 A751 L853 A856 E119 C121 A124 S125 K295 A311 L413 A416 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=51.7nM remove_due_to_license_issue P04035 18540668 876 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 3ccz B 1.7 BS01 5HI A 1 E559 C561 A564 S565 K735 A751 L853 A856 E104 C106 A109 S110 K280 A296 L398 A401 E559 K691 D767 E104 K236 D312 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=51.7nM remove_due_to_license_issue P04035 18540668 876 EPRPNEECLQILAKFLSDAEIIQLVNAKLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 3ccz B 1.7 BS02 5HI B 1 R590 S661 V683 S684 D690 K692 R135 S206 V228 S229 D235 K237 E559 K691 D767 E104 K236 D312 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=51.7nM remove_due_to_license_issue P04035 18540668 876 EPRPNEECLQILAKFLSDAEIIQLVNAKLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAG 3cd0 A 2.4 BS01 6HI B 1 E559 C561 A564 S565 K735 A751 L853 L857 H861 E119 C121 A124 S125 K295 A311 L413 L417 H421 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd0 A 2.4 BS02 6HI B 2 R590 S661 S684 D690 K692 R150 S221 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd0 B 2.4 BS01 6HI B 1 R590 S661 V683 S684 D690 K692 R150 S221 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=26.9nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd0 B 2.4 BS02 6HI B 2 E559 A564 S565 R568 K735 A751 L853 E119 A124 S125 R128 K295 A311 L413 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=26.9nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd5 A 2.39 BS01 7HI A 1 E559 A564 S565 R568 K735 A751 L853 E119 A124 S125 R128 K295 A311 L413 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=12.7nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLVKS 3cd5 A 2.39 BS02 7HI B 1 R590 S684 D690 K692 R150 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=12.7nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLVKS 3cd5 B 2.39 BS01 7HI A 1 R590 S684 D690 K692 R150 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=12.7nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLVKS 3cd5 B 2.39 BS02 7HI B 1 E559 S565 R568 K735 A751 H752 L853 L857 E119 S125 R128 K295 A311 H312 L413 L417 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=12.7nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHLVKS 3cd7 A 2.05 BS01 882 A 1 E559 C561 L562 S565 R568 K735 A751 N755 L853 A856 H861 E90 C92 L93 S96 R99 K266 A282 N286 L384 A387 H392 E559 K691 D767 E90 K222 D298 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=14.3nM remove_due_to_license_issue IC50=1.8nM P04035 18540668 1 AKFLSDAEIIQLVNAIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd7 A 2.05 BS02 882 A 2 R590 S684 D690 K692 R121 S215 D221 K223 E559 K691 D767 E90 K222 D298 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=14.3nM remove_due_to_license_issue IC50=1.8nM P04035 18540668 2 AKFLSDAEIIQLVNAIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd7 B 2.05 BS01 882 A 1 R590 S661 V683 S684 D690 K692 R130 S201 V223 S224 D230 K232 E559 K691 D767 E99 K231 D307 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue IC50=1.8nM P04035 18540668 1 AKFLSDAEIIQLVNAKHIPAYKLETLIHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd7 B 2.05 BS02 882 A 2 E559 C561 L562 S565 K735 H752 L853 A856 G860 E99 C101 L102 S105 K275 H292 L393 A396 G400 E559 K691 D767 E99 K231 D307 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue IC50=1.8nM P04035 18540668 2 AKFLSDAEIIQLVNAKHIPAYKLETLIHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cd8 A 2.0 BS01 L5G A 1 I1084 V1092 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I31 V39 A49 Y92 M93 D97 R141 M144 A154 D155 Y163 D1204 A1206 R1208 N1209 D1222 A1243 D137 A139 R141 N142 D155 A175 2.7.10.1 0004672,0004713,0005524,0006468 ic50=9nM remove_due_to_license_issue IC50=9nM P08581 18426196 1 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNRIGEVSQFLTEGIIMKDFSHPNVLSLLGICSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 3cda A 2.07 BS01 8HI A 1 R590 S661 V683 S684 D690 K692 R150 S221 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=26.3nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHL 3cda A 2.07 BS02 8HI B 1 E559 C561 S565 R568 K735 A751 N755 L853 A856 L857 E119 C121 S125 R128 K295 A311 N315 L413 A416 L417 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=26.3nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGHL 3cda B 2.07 BS01 8HI A 1 E559 C561 S565 R568 K735 A751 H752 N755 L853 A856 E119 C121 S125 R128 K295 A311 H312 N315 L413 A416 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=26.3nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cda B 2.07 BS02 8HI B 1 R590 V683 S684 D690 K692 R150 V243 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=26.3nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cdb A 2.3 BS01 9HI A 1 E559 C561 S565 K735 A751 L853 A856 L857 H861 E119 C121 S125 K295 A311 L413 A416 L417 H421 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=95.7nM remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cdb A 2.3 BS02 9HI A 2 R590 S684 D690 K692 R150 S244 D250 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 Kd=95.7nM remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cdb B 2.3 BS01 9HI A 1 R590 V683 S684 D690 K691 K692 R150 V243 S244 D250 K251 K252 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 1 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cdb B 2.3 BS02 9HI A 2 E559 C561 K735 A751 H752 L853 A856 E119 C121 K295 A311 H312 L413 A416 E559 K691 D767 E119 K251 D327 1.1.1.34 0004420,0005789,0008299,0015936,0016616,0050661 remove_due_to_license_issue P04035 18540668 2 EPRPNEECLQILGNAEKGAKFLSDAEIIQLVNAKHIPAYKLETLIETHERGVSIRRQLLSKKLSEPSSLQYLPYRDYNYSLVMGACCENVIGYMPIPVGVAGPLCLDEKEFQVPMATTEGCLVASTNRGCRAIGLGGGASSRVLADGMTRGPVVRLPRACDSAEVKAWLETSEGFAVIKEAFDSTSRFARLQKLHTSIAGRNLYIRFQSRSGDAMGMNMISKGTEKALSKLHEYFPEMQILAVSGNYCTDKKPAAINWIEGRGKSVVCEAVIPAKVVREVLKTTTEAMIEVNINKNLVGSAMAGSIGGYNAHAANIVTAIYIACGQDAAQNVGSSNCITLMEASGPTNEDLYISCTMPSIEIGTVGGGTNLLPQQACLQMLGVQGACKDNPGENARQLARIVCGTVMAGELSLMAALAAGH 3cde A 2.1 BS01 N3H A 1 F193 N291 D318 C366 S368 L384 G410 N411 M414 Y415 Q446 Y448 S556 F188 N286 D313 C361 S363 L379 G405 N406 M409 Y410 Q441 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50<0.01uM remove_due_to_license_issue IC50=<10nM, EC50=5nM P26663 18457949 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3ce0 A 2.8 BS01 P34 A 1 D284 H384 G385 Y414 F415 S422 Y425 E514 D104 H204 G205 Y234 F235 S242 Y245 E334 S422 Y425 E514 S242 Y245 E334 2.4.2.- 0003950 remove_due_to_license_issue IC50=1430nM Q9Y6F1 19354255 601 KRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 3ce3 A 2.4 BS01 1FN A 1 I1084 A1108 K1110 M1131 L1157 M1160 M1211 V1220 A1221 D1222 F1223 I31 A55 K57 M78 L104 M107 M158 V167 A168 D169 F170 D1204 A1206 R1208 N1209 D1222 A1243 D151 A153 R155 N156 D169 A176 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1.8nM remove_due_to_license_issue IC50=1.8nM P08581 18690676 1401 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3cen A 1.6 BS01 FXA A 1 E97 T98 Y99 F174 A190 C191 Q192 V213 W215 G216 G218 C220 I227 Y228 E83 T84 Y85 F162 A180 C181 Q182 V203 W205 G206 G208 C209 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=5.5nM remove_due_to_license_issue Ki=5.5nM P00742 18424044 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3cf1 A 4.4 BS01 ADP A 1 I206 G207 G248 T249 G250 K251 T252 L253 H384 G408 A409 I186 G187 G228 T229 G230 K231 T232 L233 H364 G388 A389 K251 T252 D304 N348 R453 K524 T525 D577 E578 D609 A685 K231 T232 D284 N328 R433 K504 T505 D557 E558 D585 A661 3.6.4.6 0000502,0003689,0005515,0005524,0005634,0005654,0005737,0005783,0005789,0005811,0005829,0006281,0006302,0006338,0006511,0006734,0006888,0006914,0006974,0008289,0010494,0010498,0010918,0016236,0016567,0016787,0016887,0019079,0019903,0019904,0019985,0030970,0031334,0031593,0031625,0032436,0032510,0032991,0033554,0034098,0034605,0035331,0035617,0035800,0035861,0036297,0036435,0036503,0036513,0042288,0042802,0043161,0043209,0043531,0044389,0044877,0045202,0045732,0045879,0046034,0048471,0050807,0061775,0061857,0070842,0071218,0072389,0090263,0097352,0098978,0106300,0120186,0140036,0140455,0140584,0140588,0140665,0140849,1901224,1903006,1903715,1903843,1903862,1904288,1904949,1905634,1990381,1990730,2000060,2001171 remove_due_to_license_issue Q01853 18462676 807 NRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSALRETVVEVPQVTWEDIGGLEDVKRELQELVQYPVEHPDKFLKFGMTPSKGVLFYGPPGCGKTLLAKAIANECQANFISIKGPELLTMWFGESEANVREIFDKARQAAPCVLFFDELDSIAKARGDGGGAADRVINQILTEMDGMSTKKNVFIIGATNRPDIIDPAILRPGRLDQLIYIPLPDEKSRVAILKANLRKSPVAKDVDLEFLAKMTNGFSGADLTEICQRACKLAIRESIESEIVPEIRRDHFEEAMRFARRSVSDNDIRKYEMFAQTLQ 3cf1 A 4.4 BS02 ADP A 2 D478 I479 C522 G523 K524 T525 L526 I656 G684 A685 D458 I459 C502 G503 K504 T505 L506 I632 G660 A661 K251 T252 D304 N348 R453 K524 T525 D577 E578 D609 A685 K231 T232 D284 N328 R433 K504 T505 D557 E558 D585 A661 3.6.4.6 0000502,0003689,0005515,0005524,0005634,0005654,0005737,0005783,0005789,0005811,0005829,0006281,0006302,0006338,0006511,0006734,0006888,0006914,0006974,0008289,0010494,0010498,0010918,0016236,0016567,0016787,0016887,0019079,0019903,0019904,0019985,0030970,0031334,0031593,0031625,0032436,0032510,0032991,0033554,0034098,0034605,0035331,0035617,0035800,0035861,0036297,0036435,0036503,0036513,0042288,0042802,0043161,0043209,0043531,0044389,0044877,0045202,0045732,0045879,0046034,0048471,0050807,0061775,0061857,0070842,0071218,0072389,0090263,0097352,0098978,0106300,0120186,0140036,0140455,0140584,0140588,0140665,0140849,1901224,1903006,1903715,1903843,1903862,1904288,1904949,1905634,1990381,1990730,2000060,2001171 remove_due_to_license_issue Q01853 18462676 900 NRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSALRETVVEVPQVTWEDIGGLEDVKRELQELVQYPVEHPDKFLKFGMTPSKGVLFYGPPGCGKTLLAKAIANECQANFISIKGPELLTMWFGESEANVREIFDKARQAAPCVLFFDELDSIAKARGDGGGAADRVINQILTEMDGMSTKKNVFIIGATNRPDIIDPAILRPGRLDQLIYIPLPDEKSRVAILKANLRKSPVAKDVDLEFLAKMTNGFSGADLTEICQRACKLAIRESIESEIVPEIRRDHFEEAMRFARRSVSDNDIRKYEMFAQTLQ 3cf8 A 2.4 BS01 QUE A 1 F59 K62 I111 P112 F52 K55 I104 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 Ki=12.7uM remove_due_to_license_issue Q5G940 18780820 164 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3cf8 B 2.4 BS01 QUE A 1 I98 Y100 I88 Y90 H58 I64 G67 V68 E72 H48 I54 G57 V58 E62 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 18780820 164 QFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3cf9 A 2.6 BS01 AGI A 1 F59 K62 F109 R110 F52 K55 F102 R103 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 18780820 161 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3cf9 B 2.6 BS01 AGI A 1 I98 Y100 I88 Y90 H58 I64 G67 V68 E72 H48 I54 G57 V58 E62 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 18780820 161 QFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3cfn A 1.87 BS01 2AN A 1 K15 A108 T119 V121 K6 A99 T110 V112 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=4.3uM remove_due_to_license_issue Kd=1100nM P02766 19954984 1 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3cfn B 1.87 BS01 2AN B 1 K15 V16 L17 K6 V7 L8 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=4.3uM remove_due_to_license_issue Kd=1100nM P02766 19954984 1 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3cft A 1.87 BS01 5NS A 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=64uM remove_due_to_license_issue Kd=64000nM P02766 19954984 1 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3cft B 1.87 BS01 5NS B 1 L17 A108 L110 L8 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=64uM remove_due_to_license_issue Kd=64000nM P02766 19954984 1 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3cft B 1.87 BS02 5NS B 2 K15 L17 A108 K6 L8 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=64uM remove_due_to_license_issue Kd=64000nM P02766 19954984 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3cgf A 3.0 BS01 JNF A 1 I70 V78 K93 M149 N152 S193 L206 I26 V34 K49 M105 N108 S149 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=3nM P53779 18482836 523 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQLDEREHTIEEWKELIYKEVMN 3cgo A 3.0 BS01 JNO A 1 I70 V78 M149 D150 A151 Q155 I26 V34 M105 D106 A107 Q111 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue IC50=270nM P53779 18482836 510 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYREHTIEEWKELIYKEVMN 3cgy A 2.6 BS01 RDC A 1 N390 Y394 D416 G420 I421 V445 L447 R451 A471 N60 Y64 D86 G90 I91 V93 L95 R99 A119 2.7.13.3,3.1.3.- 0016310,0016772 remove_due_to_license_issue Kd=715000nM P0DM80 18440021 700 SVLLSRELHPVAPLLDNLISALNKVYQRKGVNISMDISPEISFVGEQNDFVEVMGNVLDNACKYCLEFVEISARQTDDHLHIFVEDDGPGIPVGLAVAREITEQYAGQIIASDSLLGGARMEVVFGRQHPTQK 3ch9 A 2.2 BS01 XRG A 1 Y48 W137 D175 E177 M243 Y245 D246 W384 Y10 W99 D137 E139 M205 Y207 D208 W346 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 ic50=500uM remove_due_to_license_issue Q873X9 18355729 439 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQT 3chc A 1.9 BS01 ZRG A 1 Y48 W137 D175 E177 M243 Y245 D246 E322 W384 Y10 W99 D137 E139 M205 Y207 D208 E284 W346 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 ic50=81uM remove_due_to_license_issue Q873X9 18355729 439 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQT 3chd A 2.0 BS01 WRG A 1 Y48 W137 D175 E177 M243 Y245 D246 F251 R301 E322 W384 Y10 W99 D137 E139 M205 Y207 D208 F213 R263 E284 W346 D173 D175 E177 Y245 D135 D137 E139 Y207 3.2.1.14 0004553,0005975,0008061 ic50=12uM remove_due_to_license_issue IC50=1.2e+4nM Q873X9 18355729 800 ASSGYRSVVYFVNWAIYGRNHNPQDLPVERLTHVLYAFANVRPETGEVYMTDSWADIEKHYPGDSWSDTGNNVYGCIKQLYLLKKQNRNLKVLLSIGGWTYSPNFAPAASTDAGRKNFAKTAVKLLQDLGFDGLDIDWEYPENDQQANDFVLLLKEVRTALDSYSAANAGGQHFLLTVASPAGPDKIKVLHLKDMDQQLDFWNLMAYDYAGSFSSLSGHQANVYNDTSNPLSTPFNTQTALDLYRAGGVPANKIVLGMPLYGRSFANTDGPGKPYNGVGQGSWENGVWDYKALPQAGATEHVLPDIMASYSYDATNKFLISYDNPQVANLKSGYIKSLGLGGAMWWDSSSDKTGSDSLITTVVNALGGTGVFEQSQNELDYPVSQYDNLRNGMQT 3chg D 2.8 BS01 313 D 1 G26 I27 W72 W178 W225 T229 H230 G11 I12 W57 W163 W210 T214 H215 ? 0005886,0006865,0022857,0043190,0045121,0055085 remove_due_to_license_issue P46922 18567662 1 KTIIGIDPGSGIMSLTDKAMKDYDLNDWTLISASSAAMTATLKKSYDRKKPIIITGWTPHWMFSRYKLKYLDDPKQSYGSAEEIHTITRKGFSKEQPNAAKLLSQFKWTQDEMGEIMIKVEEGEKPAKVAAEYVNKHKDQIAEWTKGVQKVKGDKINLAYVAWDSEIASTNVIGKVLEDLGYEVTLTQVEAGPMWTAIATGSADASLSAWLPNTHKAYAAKYKGKYDDIGTSMTGVKMGLVVPQYMKNVNSIEDLKK 3cho A 1.8 BS02 4BG A 1 Q136 A137 Y267 W311 F314 V367 A377 Y378 Q136 A137 Y267 W311 F314 V367 A377 Y378 E271 H295 E296 H299 E318 D375 Y383 E271 H295 E296 H299 E318 D375 Y383 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=280nM remove_due_to_license_issue IC50=300nM P09960 18394906 901 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3chp A 2.1 BS02 4BO A 1 Q136 A137 Y267 E271 F314 E318 P374 A377 Y378 Y383 Q134 A135 Y265 E269 F312 E316 P372 A375 Y376 Y381 E271 H295 E296 H299 E318 D375 Y383 E269 H293 E294 H297 E316 D373 Y381 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=5400nM remove_due_to_license_issue IC50=5400nM P09960 18394906 901 IVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3chq A 2.09 BS02 4BQ A 1 Q136 A137 Y267 G269 M270 E271 E296 W311 F314 E318 L369 P374 A377 Y378 Y383 Q134 A135 Y265 G267 M268 E269 E294 W309 F312 E316 L367 P372 A375 Y376 Y381 E271 H295 E296 H299 E318 D375 Y383 E269 H293 E294 H297 E316 D373 Y381 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=20nM remove_due_to_license_issue IC50=20nM P09960 18394906 901 IVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3chr A 2.2 BS02 4BS A 1 Q136 A137 Y267 G269 E271 W311 F314 L369 P374 A377 Y378 Q136 A137 Y267 G269 E271 W311 F314 L369 P374 A377 Y378 E271 H295 E296 H299 E318 D375 Y383 E271 H295 E296 H299 E318 D375 Y383 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=61nM remove_due_to_license_issue IC50=61nM P09960 18394906 613 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3chs A 2.55 BS02 4BU A 1 Q136 Y267 G269 E271 H295 E296 W311 F314 E318 V367 P374 A377 Y378 P382 Q136 Y267 G269 E271 H295 E296 W311 F314 E318 V367 P374 A377 Y378 P382 E271 H295 E296 H299 E318 D375 Y383 E271 H295 E296 H299 E318 D375 Y383 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue P09960 18394906 901 PEIVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3cib A 1.72 BS01 314 A 1 G72 D93 G95 Y132 T133 Q134 F169 Y259 D289 G291 T293 G15 D36 G38 Y75 T76 Q77 F112 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=14nM remove_due_to_license_issue IC50=522nM P56817 18468890 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3cic A 1.75 BS01 316 A 1 G72 Q73 D93 G95 S96 Y132 T133 Q134 F169 Y259 D289 G291 T293 G15 Q16 D36 G38 S39 Y75 T76 Q77 F112 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=3nM remove_due_to_license_issue IC50=300nM, Ki=3nM P56817 18468890 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3cid A 1.8 BS01 318 A 1 G72 D93 G95 S96 P131 Y132 T133 Q134 G135 F169 Y259 D289 G291 T293 G15 D36 G38 S39 P74 Y75 T76 Q77 G78 F112 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=5nM remove_due_to_license_issue IC50=5nM P56817 18468890 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3cj2 A 1.75 BS01 SX3 A 1 R422 M423 R501 W528 R417 M418 R496 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=14uM remove_due_to_license_issue P26663 18400495 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3cj3 A 1.87 BS01 SX4 A 1 L419 R422 M423 H475 S476 Y477 R501 W528 L416 R419 M420 H472 S473 Y474 R498 W525 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=57uM remove_due_to_license_issue P26663 18400495 572 HHMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYHS 3cj4 A 2.07 BS01 SX5 A 1 L419 R422 M423 H475 S476 I482 R501 W528 L415 R418 M419 H471 S472 I478 R497 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.31uM remove_due_to_license_issue P26663 18400495 571 HHMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3cj5 A 1.92 BS01 SX6 A 1 R422 M423 H475 S476 L497 R498 R501 W528 R421 M422 H474 S475 L496 R497 R500 W527 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.46uM remove_due_to_license_issue P26663 18400495 571 HHMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYHS 3cjf A 2.15 BS01 SAV A 1 L838 A864 F916 C917 K918 G920 L1033 L24 A50 F102 C103 K104 G106 L162 D1026 A1028 R1030 N1031 D1044 K1053 D155 A157 R159 N160 D173 K180 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=6.3nM remove_due_to_license_issue IC50=6.3nM P35968 18620382 1167 CERLPYDASKWEFPRDRLNLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDLARDIYKPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 3cjo A 2.28 BS02 K30 A 1 E116 G117 E118 R119 W127 A133 I136 Y211 L214 E215 G217 A218 R221 E99 G100 E101 R102 W110 A116 I119 Y194 L197 E198 G200 A201 R204 ? 0003777,0005524,0007018,0008017 ic50=2.2nM remove_due_to_license_issue P52732 18578472 1 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 3cke A 2.4 BS01 FDF A 1 Y67 F87 D90 F153 L184 N219 W308 R314 Y315 Y55 F75 D78 F141 L172 N207 W286 R292 Y293 Y67 F87 F153 K181 W308 Y55 F75 F141 K169 W286 4.2.3.9 0010333,0016829,0016838,0045483,0046872 remove_due_to_license_issue Q9UR08 18385128 400 SLEPPPSTFQPLCHPLVEEVSKEVDGYFLQHWNFPNEKARKKFVAAGFSRVTCLYFPKALDDRIHFACRLLTVLFLIDDLLEYMSFEEGSAYNEKLIPISRGDVLPDRSIPVEYIIYDLWESMRAHDREMADEILEPVFLFMRAQTDRTRARPMGLGGYLEYRERDVGKELLAALMRFSMGLKLSPSELQRVREIDANCSKHLSVVNDIYSYEKELYTLCTSVQILAQEADVTAEAAKRVLFVMCREWELRHQLLVARLSAEGLETPGLAAYVEGLEYQMSGNELWSQTTLRYSV 3ckp A 2.3 BS01 012 A 1 Q12 G13 L30 D32 G34 P70 Y71 T72 F108 R128 Y198 D228 G230 T231 T232 Q18 G19 L36 D38 G40 P76 Y77 T78 F114 R134 Y195 D225 G227 T228 T229 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D225 T228 3.4.23.46 0004190,0006508,0016020 Ki=0.449uM remove_due_to_license_issue P56817 18434152 501 KKGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3ckr A 2.7 BS01 009 A 1 Q12 G13 D32 G34 Y71 T72 Q73 F108 I110 R128 Y198 D228 G230 T231 T232 Q18 G19 D38 G40 Y77 T78 Q79 F114 I116 R134 Y195 D225 G227 T228 T229 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D225 T228 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 18434152 501 KKGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3ckt A 1.65 BS01 YDP A 1 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.48uM remove_due_to_license_issue P03367 21762812 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ckt B 1.65 BS01 YDP A 1 D25 G27 A28 D30 G48 D25 G27 A28 D30 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 21762812 2501 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ckz A 1.9 BS02 ZMR A 1 R118 E119 D151 R152 W178 E227 S246 E276 R292 R371 Y406 R36 E37 D69 R70 W97 E146 S165 E195 R211 R286 Y320 D151 E277 R292 R371 Y406 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=0.19nM remove_due_to_license_issue Q6DPL2 18480754 469 VKLAGNSSLCPINGWAVYSKDNSIRIGSKGDVFVIREPFISCSHLECRTFFLTQGALLNDKHSNGTVKDRSPHRTLMSCPVGEAPSPYNSRFESVAWSASACHDGTSWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFKMEKGKVVKSVELDAPNYYYEECSCYPNAGEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGVFGDNPRPNDGTGSCGPVSSNGAYGVKGFSFKYGNGVWIGRTKSTNSRSGFEMIWDPNGWTETDSSFSVKQDIVAITDWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKESTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTI 3cl0 A 2.2 BS01 G39 A 1 R118 E119 D151 R152 W178 E276 R292 N294 Y347 R371 Y406 R36 E37 D69 R70 W97 E195 R211 N213 Y262 R286 Y320 D151 E277 R292 R371 Y406 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=84.8nM remove_due_to_license_issue Q6DPL2 18480754 800 VKLAGNSSLCPINGWAVYSKDNSIRIGSKGDVFVIREPFISCSHLECRTFFLTQGALLNDKHSNGTVKDRSPHRTLMSCPVGEAPSPYNSRFESVAWSASACHDGTSWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFKMEKGKVVKSVELDAPNYYYEECSCYPNAGEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGVFGDNPRPNDGTGSCGPVSSNGAYGVKGFSFKYGNGVWIGRTKSTNSRSGFEMIWDPNGWTETDSSFSVKQDIVAITDWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKESTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTI 3cl2 A 2.538 BS01 G39 A 1 E119 D151 W178 S246 R292 Y347 R371 Y406 E37 D69 W97 S165 R211 Y262 R286 Y320 D151 E277 R292 R371 Y406 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue Q6DPL2 18480754 800 VKLAGNSSLCPINGWAVYSKDNSIRIGSKGDVFVIREPFISCSHLECRTFFLTQGALLNDKHSNGTVKDRSPHRTLMSCPVGEAPSPYNSRFESVAWSASACHDGTSWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFKMEKGKVVKSVELDAPNYHYEECSCYPNAGEITCVCRDSWHGSNRPWVSFNQNLEYQIGYICSGVFGDNPRPNDGTGSCGPVSSNGAYGVKGFSFKYGNGVWIGRTKSTNSRSGFEMIWDPNGWTETDSSFSVKQDIVAITDWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKESTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTI 3clp A 2.0 BS01 CMP A 1 V282 T284 F296 G297 E298 M299 A300 S308 A309 V311 R348 V65 T67 F79 G80 E81 M82 A83 S91 A92 V94 R131 ? 0005221 remove_due_to_license_issue Q98GN8 18619611 1 VRRGDFVRNWQLVAAVPLFQKLGPAVLVEIVRALRARTVPAGAVICRIGEPGDRMFFVVEGSVSVATPNPVELGPGAFFGEMALISGEPESATVSAATTVSLLSLHSADFQMLCSSSPEIAEIFRKTALERR 3cm2 D 2.5 BS02 X23 D 1 L292 K297 V298 G306 L307 T308 D309 W310 E314 Q319 L39 K44 V45 G53 L54 T55 D56 W57 E61 Q66 2.3.2.27 Ki=340nM remove_due_to_license_issue IC50=110nM P98170 18851976 600 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVRT 3cm7 B 3.1 BS02 X22 B 1 K299 G306 L307 T308 D309 W310 E314 Q319 W323 K45 G52 L53 T54 D55 W56 E60 Q65 W69 2.3.2.27 remove_due_to_license_issue IC50=290nM P98170 18851976 600 NLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVRT 3cn0 A 1.52 BS01 LJ1 A 1 K15 L110 S117 T118 K5 L100 S107 T108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=3080nM P02766 18811132 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3cn0 B 1.52 BS01 LJ1 B 1 K15 L110 S117 T118 K5 L100 S107 T108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=3080nM P02766 18811132 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3co6 C 2.1 BS01 dna A 0 L183 R214 H215 S218 R225 S234 S235 W237 L30 R61 H62 S65 R72 S81 S82 W84 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 -4 ~ 12 SSRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNPEGG 3co6 C 2.1 BS02 dna B 0 N158 S164 Y165 N211 H215 G232 N5 S11 Y12 N58 H62 G79 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 13 ~ 28 SSRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNPEGG 3co7 C 2.91 BS01 dna A 0 L183 R214 H215 S218 R225 S234 S235 W237 L29 R60 H61 S64 R71 S80 S81 W83 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 -2 ~ 14 SRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3co7 C 2.91 BS02 dna B 0 R157 S164 Y165 N211 H215 G232 R3 S10 Y11 N57 H61 G78 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 15 ~ 30 SRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3co7 F 2.91 BS01 dna D 0 L183 R214 H215 S218 R225 S234 S235 W237 L29 R60 H61 S64 R71 S80 S81 W83 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 -2 ~ 14 SRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3co7 F 2.91 BS02 dna E 0 R157 S164 Y165 N211 H215 G232 R3 S10 Y11 N57 H61 G78 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 15 ~ 30 SRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3co9 A 2.1 BS01 3MS A 1 F193 N291 D318 C366 S368 L384 M414 Y415 I447 Y448 G449 S556 F193 N291 D318 C366 S368 L384 M414 Y415 I447 Y448 G449 S556 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue IC50=<10nM, EC50=8.5nM P26663 18487044 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3coa C 2.2 BS01 dna A 0 L183 R214 H215 S218 R225 S234 S235 W237 L28 R59 H60 S63 R70 S79 S80 W82 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 -4 ~ 12 RRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3coa C 2.2 BS02 dna B 0 S164 Y165 N211 H215 G232 S9 Y10 N56 H60 G77 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 13 ~ 28 RRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3coa F 2.2 BS01 dna D 0 L183 R214 H215 S218 R225 S234 S235 W237 L29 R60 H61 S64 R71 S80 S81 W83 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 -4 ~ 12 SRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3coa F 2.2 BS02 dna E 0 S164 Y165 N211 H215 G232 S10 Y11 N57 H61 G78 ? 0003700,0006355,0043565 remove_due_to_license_issue Q12778 18786403 13 ~ 28 SRRNAWGNLSYADLITKAIESSAEKRLTLSQIYEWMVKSVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIRVQNEGTGKSSWWMLNP 3coh A 2.7 BS01 83H A 1 L139 V147 A160 L194 Y212 A213 P214 G216 L263 L12 V20 A33 L67 Y85 A86 P87 G89 L136 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T151 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 18630890 1 WALEDFEIGRPLGKGKFGNVYLAREKNSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDSTRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKKVIHRDIKPENLLLGSAGELKIADLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQDTYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3coq A 2.4 BS01 dna D 0 K17 K18 L49 T50 R51 K10 K11 L42 T43 R44 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P04386 18611375 1 ~ 20 EQACDICRLKKLKCSKEKPKCAKCLKNNWECRYSPKTKRSPLTRAHLTEVESRLERLEQLFLLIFPREDLDMILKMDSLQDIKALLTGL 3coq A 2.4 BS02 dna E 0 Q9 A10 R15 K18 K20 C21 K23 L49 Q2 A3 R8 K11 K13 C14 K16 L42 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P04386 18611375 21 ~ 40 EQACDICRLKKLKCSKEKPKCAKCLKNNWECRYSPKTKRSPLTRAHLTEVESRLERLEQLFLLIFPREDLDMILKMDSLQDIKALLTGL 3coq B 2.4 BS01 dna D 0 A10 R15 K18 K20 K23 R46 L49 A3 R8 K11 K13 K16 R39 L42 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P04386 18611375 1 ~ 20 EQACDICRLKKLKCSKEKPKCAKCLKNNWECRYSPKTKRSPLTRAHLTEVESRLERLEQLFLLIFPREDLDMILKMDSLQDIKALLTGL 3coq B 2.4 BS02 dna E 0 K17 K18 L49 T50 R51 K10 K11 L42 T43 R44 ? 0000981,0003700,0006355,0008270 remove_due_to_license_issue P04386 18611375 21 ~ 40 EQACDICRLKKLKCSKEKPKCAKCLKNNWECRYSPKTKRSPLTRAHLTEVESRLERLEQLFLLIFPREDLDMILKMDSLQDIKALLTGL 3cow A 1.8 BS01 52H A 1 P38 T39 M40 G46 H47 L50 Q72 F157 G158 K160 D161 Q164 T186 V187 M195 P36 T37 M38 G44 H45 L48 Q70 F155 G156 K158 D159 Q162 T184 V185 M193 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=0.125uM remove_due_to_license_issue Ki=270nM P9WIL5 18821554 401 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIG 3coy A 2.03 BS01 53H A 1 P38 T39 M40 G46 H47 L50 Q72 F157 G158 K160 D161 Q164 T186 V187 M195 P36 T37 M38 G44 H45 L48 Q70 F149 G150 K152 D153 Q156 T178 V179 M187 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D80 D81 Q84 K152 S188 S189 R190 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=0.96uM remove_due_to_license_issue Ki=300nM P9WIL5 18821554 301 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMNGSGRLLVAARLGTTRLLDNIAIEIGTF 3coz A 2.0 BS01 54H A 1 P38 T39 M40 H44 G46 H47 L50 F157 G158 D161 Q164 T186 V187 M195 P36 T37 M38 H42 G44 H45 L48 F155 G156 D159 Q162 T184 V185 M193 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=2.7uM remove_due_to_license_issue P9WIL5 18821554 401 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3cp9 A 2.5 BS01 C19 A 1 L840 V848 A866 K868 E885 L889 V898 T916 C919 L1035 C1045 D1046 F1047 L24 V26 A44 K46 E63 L67 V76 T94 C97 L163 C173 D174 F175 D1028 A1030 R1032 N1033 D1046 D156 A158 R160 N161 D174 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=48nM P35968 18447379 501 AERLPYDASKWEFPRDRLKLGKPLQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3cpb A 2.7 BS01 C92 A 1 A866 K868 E885 V914 T916 F918 C919 L1035 C1045 D1046 F1047 A42 K44 E61 V90 T92 F94 C95 L161 C171 D172 F173 D1028 A1030 R1032 N1033 D1046 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=>25000nM P35968 18447379 1 RLPYDASKWEFPRDRLKLGKPLQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3cpc A 2.4 BS01 C52 A 1 V848 A866 K868 E885 L889 V899 T916 C919 L1035 C1045 D1046 F1047 V23 A41 K43 E60 L64 V74 T91 C94 L160 C170 D171 F172 D1028 A1030 R1032 N1033 D1046 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=>5000nM P35968 18447379 1 LPYDASKWEFPRDRLKLGKPLQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3cph A 2.9 BS01 GDP A 1 S29 G30 V31 G32 K33 S34 C35 F45 F49 N133 K134 D136 M137 S162 A163 K164 S10 G11 V12 G13 K14 S15 C16 F26 F30 N114 K115 D117 M118 S143 A144 K145 Q79 Q60 ? 0000131,0003924,0005515,0005525,0005737,0005739,0005741,0005768,0005783,0005886,0005935,0006887,0006893,0006906,0006914,0007107,0015031,0030133,0030658,0031321,0031410,0031982,0043332 remove_due_to_license_issue P07560 18426803 302 IMKILLIGDSGVGKSCLLVRFVEDKFNPSFITTIGIDFKIKTVDINGKKVKLQLWDTAGQERFRTITTAYYRGAMGIILVYDVTDERTFTNIKQWFKTVNEHANDEAQLLLVGNKSDMETRVVTADQGEALAKELGIPFIESSAKNDDNVNEIFFTLAKLIQEKIDSNKLVGVGN 3cpj B 2.35 BS01 GDP B 1 G23 G25 K26 S27 N28 F38 N39 M40 N126 K127 D129 L130 A157 L158 G14 G16 K17 S18 N19 F29 N30 M31 N108 K109 D111 L112 A139 L140 ? 0000139,0003924,0005515,0005525,0005739,0005741,0005768,0005794,0005802,0005829,0006887,0006914,0015031,0016020,0016192,0034498,0055037 remove_due_to_license_issue P38555 18426803 1207 YDLLFKIVLIGDSGVGKSNLLSRFTKNEFNMGVEFATRTLEIEGKRIKAQIWDTAGQERYRAITSAYYRGAVGALIVYDSKSSSYENCNHWLSELRENADVAVGLIGNKSDLAHLRAVPTEESKTFAQENQLLFTETSALSENVDKAFEELINTIYQKVPTISL 3cqu A 2.2 BS02 CQU A 1 L156 F161 V164 A177 E228 Y229 A230 E234 M281 T291 D292 F438 L13 F18 V21 A34 E85 Y86 A87 E91 M138 T148 D149 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 ic50=151nM remove_due_to_license_issue IC50=151nM P31749 18456494 999 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMSERRPHFPQFDYSASS 3cqw A 2.0 BS03 CQW A 1 A177 M227 A230 E234 E278 M281 D292 F438 A34 M84 A87 E91 E135 M138 D149 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 ic50=42nM remove_due_to_license_issue P31749 18456494 999 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMIERRPHFPQFDYSASS 3cr4 X 2.15 BS01 PNT X 1 C84 H85 F87 C85 H86 F88 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=53uM remove_due_to_license_issue P02638 18602402 101 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 3cr4 X 2.15 BS02 PNT X 2 H42 F43 F88 H43 F44 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=53uM remove_due_to_license_issue P02638 18602402 102 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 3cr5 X 1.85 BS01 PNT X 1 C84 F88 C85 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=64uM remove_due_to_license_issue P02638 18602402 94 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFEH 3cr5 X 1.85 BS02 PNT X 2 F43 C84 F87 F88 F44 C85 F88 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=64uM remove_due_to_license_issue P02638 18602402 95 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFEH 3cs7 A 2.2 BS02 LG0 A 1 E97 T98 Y99 A190 C191 Q192 V213 W215 G216 C220 E83 T84 Y85 A180 C181 Q182 V203 W205 G206 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.021nM remove_due_to_license_issue Ki=0.021nM P00742 18550370 298 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3cso A 2.71 BS01 XNI A 1 P197 R200 N316 C366 L384 N411 M414 Y415 Y448 P195 R198 N314 C364 L382 N409 M412 Y413 Y446 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 18852280 579 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPEGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3cst A 3.2 BS01 E52 A 1 M804 A805 W812 Y867 V882 D884 A885 T887 K890 M953 M567 A568 W575 Y630 V645 D647 A648 T650 K653 M715 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 18484710 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 3cth A 2.3 BS01 319 A 1 A1108 K1110 E1127 M1131 F1134 L1157 Y1159 M1160 H1202 M1211 A1221 D1222 F1223 A57 K59 E76 M80 F83 L106 Y108 M109 H151 M160 A170 D171 F172 D1204 A1206 R1208 N1209 D1222 A1243 D153 A155 R157 N158 D171 A178 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.035uM remove_due_to_license_issue IC50=35nM P08581 18479916 2001 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3ctj A 2.5 BS01 320 A 1 A1108 M1131 L1157 Y1159 M1160 M1211 V1220 A1221 D1222 F1223 A58 M81 L107 Y109 M110 M161 V170 A171 D172 F173 D1204 A1206 R1208 N1209 D1222 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.11uM remove_due_to_license_issue IC50=110nM P08581 18479916 2001 VHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3ctq A 1.95 BS01 337 A 1 Y35 A51 K53 R70 E71 L74 L75 M78 T106 L108 M109 G110 A111 D112 L167 D168 F169 Y31 A47 K49 R66 E67 L70 L71 M74 T102 L104 M105 G106 A107 D108 L163 D164 F165 D150 K152 N155 D168 T185 D146 K148 N151 D164 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=40nM remove_due_to_license_issue Q16539 18462940 1 RPTFYRQELAKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCAKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3ctr A 2.1 BS01 MGP A 1 W456 W475 D477 D478 W17 W36 D38 D39 3.1.13.4 0003676,0003723,0004535,0005634,0005737,0006402,0046872 Kd=6.94uM remove_due_to_license_issue O95453 18694759 1 GPLGSDHVLHVTFPKEWKTSDLYQLFSAFGNIQISWIDDTSAFVSLSQPEQVKIAVNTSKYAESYRIQTYAEYMG 3ctt A 2.1 BS01 3CU A 1 Y299 D327 W441 D443 R526 D542 F575 H600 Y293 D321 W435 D437 R520 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=0.45uM remove_due_to_license_issue O43451 19123216 1001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3cvk A 2.31 BS01 N34 A 1 F193 R200 S288 N291 G317 D318 C366 S368 M414 I447 Y448 G449 S556 F188 R195 S283 N286 G312 D313 C361 S363 M409 I442 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50<0.01uM remove_due_to_license_issue P26663 18722768 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3cvv A 2.1 BS01 dna C 0 K246 P247 P293 Q299 W302 H365 L366 H369 W409 Q418 R421 Y423 S424 F428 K431 K260 P261 P307 Q313 W316 H379 L380 H383 W423 Q432 R435 Y437 S438 F442 K445 Q299 W302 W330 H365 W384 W407 Q313 W316 W344 H379 W398 W421 ? 0000166,0003677,0003904,0005634,0005737,0032922,0043153,0071949 remove_due_to_license_issue Q8SXK5 19570997 1 ~ 15 EKGASTSLYKKAGLMDSQRSTLVHWFRKGLRLHDNPALSHIFTAANAAPGRYFVRPIFILDPGILDWMQVGANRWRFLQQTLEDLDNQLRKLNSRLFVVRGKPAEVFPRIFKSWRVEMLTFETDIEPYSVTRDAAVQKLAKAEGVRVETHCSHTIYNPELVIAKNLGKAPITYQKFLGIVEQLKVPKVLGVPEKLKNMPTPPKDEVEQKDSAAYDCPTMKQLVKRPEELGPNKFPGGETEALRRMEESLKDEIWVARFEKPNTAPNSLEPSTTVLSPYLKFGCLSARLFNQKLKEIIKRQPKHSQPPVSLIGQLMWREFYYTVAAAEPNFDRMLGNVYCMQIPWQEHPDHLEAWTHGRTGYPFIDAIMRQLRQEGWIHHLARHAVACFLTRGDLWISWEEGQRVFEQLLLDQDWALNAGNWMWLSASAFFHQYFRVYSPVAFGKKTDPQGHYIRKYVPELSKYPAGCIYEPWKASLVDQRAYGCVLGTDYPHRIVKHEVVHKENIKRMGAAYKVNREVR 3cvv A 2.1 BS02 dna D 0 I157 H417 Y419 F420 R502 R505 I171 H431 Y433 F434 R516 R519 Q299 W302 W330 H365 W384 W407 Q313 W316 W344 H379 W398 W421 ? 0000166,0003677,0003904,0005634,0005737,0032922,0043153,0071949 remove_due_to_license_issue Q8SXK5 19570997 1 ~ 15 EKGASTSLYKKAGLMDSQRSTLVHWFRKGLRLHDNPALSHIFTAANAAPGRYFVRPIFILDPGILDWMQVGANRWRFLQQTLEDLDNQLRKLNSRLFVVRGKPAEVFPRIFKSWRVEMLTFETDIEPYSVTRDAAVQKLAKAEGVRVETHCSHTIYNPELVIAKNLGKAPITYQKFLGIVEQLKVPKVLGVPEKLKNMPTPPKDEVEQKDSAAYDCPTMKQLVKRPEELGPNKFPGGETEALRRMEESLKDEIWVARFEKPNTAPNSLEPSTTVLSPYLKFGCLSARLFNQKLKEIIKRQPKHSQPPVSLIGQLMWREFYYTVAAAEPNFDRMLGNVYCMQIPWQEHPDHLEAWTHGRTGYPFIDAIMRQLRQEGWIHHLARHAVACFLTRGDLWISWEEGQRVFEQLLLDQDWALNAGNWMWLSASAFFHQYFRVYSPVAFGKKTDPQGHYIRKYVPELSKYPAGCIYEPWKASLVDQRAYGCVLGTDYPHRIVKHEVVHKENIKRMGAAYKVNREVR 3cwe A 1.6 BS01 825 A 1 Y546 D548 D681 F682 C715 S716 A717 I719 G720 R721 Q762 Y53 D55 D183 F184 C217 S218 A219 I221 G222 R223 Q264 D681 C715 R721 S722 Q762 D183 C217 R223 S224 Q264 3.1.3.48 0004725,0006470,0016311 ic50=0.12uM remove_due_to_license_issue IC50=120nM, EC50=1200nM P18031 18477508 784 AADKLEFMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 3cwj A 2.4 BS01 321 A 1 F193 P197 S288 N291 N316 D318 C366 L384 G410 N411 M414 Y415 Q446 Y448 S556 F188 P192 S283 N286 N311 D313 C361 L379 G405 N406 M409 Y410 Q441 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50<0.01uM remove_due_to_license_issue IC50=<10nM, EC50=11nM P26663 18662878 1001 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3cwk A 1.6 BS01 REA A 1 A32 V54 V58 R59 E121 K132 A32 V54 V58 R59 E121 K132 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 Kd=250nM remove_due_to_license_issue P29373 19018099 300 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKVSTTVRTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTLELTNDGELIETMTADDVVCTKVFVRE 3cx9 A 2.8 BS01 LPX A 1 Y150 E153 Q196 K199 W214 L219 R222 L238 V241 H242 C245 R257 L260 Y148 E151 Q194 K197 W212 L217 R220 L236 V239 H240 C243 R255 L258 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 remove_due_to_license_issue P02768 19601929 2001 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATLRETYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPKEFNAETFTFHADICTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAALG 3cxc 1 3.0 BS01 rna 0 0 G1 K2 K3 K5 A6 K8 R10 L11 K13 N16 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R35 H37 R40 H41 W42 R43 N45 T47 G1 K2 K3 K5 A6 K8 R10 L11 K13 N16 Q17 S19 P22 W24 V25 L27 K28 T29 D30 R32 H34 R37 H38 W39 R40 N42 T44 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P22452 18947996 10 ~ 2914 GKKSKATKKRLAKLDNQNSRVPAWVMLKTDERNHKRRHWRRNDTDE 3cxc 2 3.0 BS01 rna 0 0 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 S27 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 N43 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 D66 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 M1 Q2 P4 N8 T9 Y10 H13 N15 E16 H17 V25 S27 G28 R29 Q30 T31 M33 K34 W35 I36 R38 Q39 R42 N43 G45 I46 G47 N48 G50 K51 S53 K54 G58 D59 K60 P61 T62 K63 K64 D66 K68 K76 A77 L79 R80 G82 R84 A85 G86 Q91 ? 0000049,0003735,0005840,0006412,0008270,0019843,0046872,0070180,1990904 remove_due_to_license_issue P32411 18947996 10 ~ 2914 MQMPRRFNTYCPHCNEHQEHEVEKVRSGRQTGMKWIDRQRERNSGIGNDGKFSKVPGGDKPTKKTDLKYRCGECGKAHLREGWRAGRLEFQE 3cxc A 3.0 BS01 rna 0 0 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 Y23 K24 A25 D26 K31 H47 P49 R51 S52 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 A193 M194 N195 V197 D198 H199 G203 G204 G205 R206 Q207 H208 P209 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 I228 A229 S230 K231 R232 T233 G234 R235 G236 G1 R2 R3 G6 Q7 R8 R9 G10 R11 G12 T13 S14 T15 F16 R17 A18 S20 H21 Y23 K24 A25 D26 K31 H47 P49 R51 S52 K117 F118 A119 R120 A121 S122 G123 V124 L140 P141 S142 E144 K146 G162 G163 R164 T165 K167 P168 F169 V170 K171 A172 G173 K175 H176 H177 K178 K180 R182 G183 T184 K185 W186 P187 N188 V189 R190 G191 V192 A193 M194 N195 V197 D198 H199 G203 G204 G205 R206 Q207 H208 P209 K211 P212 K213 S214 I215 S216 R217 N218 P220 P221 G222 R223 K224 V225 G226 I228 A229 S230 K231 R232 T233 G234 R235 G236 ? 0002181,0003723,0003735,0005840,0006412,0015934,0019843,0022625,0022626,1990904 remove_due_to_license_issue P20276 18947996 10 ~ 2914 GRRIQGQRRGRGTSTFRAPSHRYKADLEHRKVEDGDVIAGTVVDIEHDPARSAPVAAVEFEDGDRRLILAPEGVGVGDELQVGVDAEIAPGNTLPLAEIPEGVPVCNVESSPGDGGKFARASGVNAQLLTHDRNVAVVKLPSGEMKRLDPQCRATIGVVGGGGRTDKPFVKAGNKHHKMKARGTKWPNVRGVAMNAVDHPFGGGGRQHPGKPKSISRNAPPGRKVGDIASKRTGRGG 3cxc B 3.0 BS01 rna 0 0 P1 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 Q94 P96 L97 T98 E99 W101 R111 T112 L113 D114 V115 P116 E117 R141 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 G282 V285 N286 G288 E289 S300 V301 P302 K306 R307 R312 R316 N318 S334 N335 Q336 G337 P1 Q2 P3 S4 R5 P6 R7 K8 G9 S10 L11 G12 F13 P15 R16 K17 R18 R25 N27 S28 K45 M48 T49 H50 N59 P70 R85 Y87 Y92 Q94 P96 L97 T98 E99 W101 R111 T112 L113 D114 V115 P116 E117 R141 K156 K157 K158 V161 E163 T206 K207 G208 K209 G210 T211 Q212 G213 K216 R217 Q221 K222 R223 K224 G225 K226 H227 R229 Q230 G231 W232 R233 R234 R235 G237 N238 L239 G240 P241 W242 N243 P244 S245 R246 V247 R248 S249 T250 V251 P252 Q253 Q254 Q256 Y259 Q261 R262 T263 E264 L265 N266 G282 V285 N286 G288 E289 S300 V301 P302 K306 R307 R312 R316 N318 S334 N335 Q336 G337 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P20279 18947996 10 ~ 2914 PQPSRPRKGSLGFGPRKRSTSETPRFNSWPSDDGQPGVQGFAGYKAGMTHVVLVNDEPNSPREGMEETVPVTVIETPPMRAVALRAYEDTPYGQRPLTEVWTDEFHSELDRTLDVPEDHDPDAAEEQIRDAHEAGDLGDLRLITHTVPDAVPSVPKKKPDVMETRVGGGSVSDRLDHALDIVEDGGEHAMNDIFRAGEYADVAGVTKGKGTQGPVKRWGVQKRKGKHARQGWRRRIGNLGPWNPSRVRSTVPQQGQTGYHQRTELNKRLIDIGEGDEPTVDGGFVNYGEVDGPYTLVKGSVPGPDKRLVRFRPAVRPNDQPRLDPEVRYVSNESNQG 3cxc C 3.0 BS01 rna 0 0 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 P71 L73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 H90 P92 K93 E95 K96 D97 L100 D101 N103 D104 K105 E106 R107 R127 V148 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 R188 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 R27 R36 A38 N41 R42 K43 Q44 D45 Y46 G47 S48 D49 A52 G53 R55 T56 P57 S60 S63 G64 G66 Q67 A68 H69 P71 L73 D74 R76 A77 V80 P81 Q82 A83 V84 K85 R87 H90 P92 K93 E95 K96 D97 L100 D101 N103 D104 K105 E106 R107 R127 V148 K149 T150 Q151 R168 D170 K173 I174 K175 A176 G177 Q178 G179 R182 R184 Y186 R187 R188 A190 T202 R205 N206 A213 E217 V218 N219 D222 P225 G226 R246 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12735 18947996 10 ~ 2914 MQATIYDLDGNTDGEVDLPDVFETPVRSDLIGKAVRAAQANRKQDYGSDEYAGLRTPAESFGSGRGQAHVPKLDGRARRVPQAVKGRSAHPPKTEKDRSLDLNDKERQLAVRSALAATADADLVADRGHEFDRDEVPVVVSDDFEDLVKTQEVVSLLEALDVHADIDRADETKIKAGQGSARGRKYRRPASILFVTSDEPSTAARNLAGADVATASEVNTEDLAPGGAPGRLTVFTESALAEVAER 3cxc D 3.0 BS01 rna 0 0 K20 V22 H24 T52 A54 R56 E60 K72 Q97 D99 D100 T101 N103 S105 G107 D129 K11 V13 H15 T38 A40 R42 E46 K58 Q83 D85 D86 T87 N89 S91 G93 D95 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18947996 10 ~ 2914 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3cxc D 3.0 BS02 rna 9 0 E12 M13 R14 R17 Q47 M48 V50 R51 K72 V73 T74 R76 P137 G138 R140 V141 R144 D145 R149 P152 K154 H155 E3 M4 R5 R8 Q33 M34 V36 R37 K58 V59 T60 R62 P103 G104 R106 V107 R110 D111 R115 P118 K120 H121 ? 0000049,0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P14124 18947996 3001 ~ 3122 FHEMREPRIEKVVVHMGIGHANAEDILGEITGQMPVRTKAKRTVGEFDIREGDPIGAKVTLRDEMAEEFLQTALPLAELATSQFDDTGNFSFGLDVTVNLVRPGYRVAKRDKASRSIPTKHRLNPADAVAFIESTYDVEV 3cxc E 3.0 BS01 rna 0 0 Y35 N55 S60 G63 T64 S67 H68 N71 Y82 H90 F91 E110 K111 A112 H119 E139 Q143 A146 Q150 R153 N155 K157 D158 R160 V161 F162 Y35 N55 S60 G63 T64 S67 H68 N71 Y82 H90 F91 E110 K111 A112 H119 E139 Q143 A146 Q150 R153 N155 K157 D158 R160 V161 F162 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P14135 18947996 10 ~ 2914 PRVELEIPEDVDAEQDHLDITVEGDNGSVTRRLWYPDIDVSVDGDTVVIESDEDNAKTMSTIGTFQSHIENMFHGVTEGWEYGMEVFYSHFPMQVNVEGDEVVIENFLGEKAPRRTTIHGDTDVEIDGEELTVSGPDIEAVGQTAADIEQLTRINDKDVRVFQDGVYITRKP 3cxc F 3.0 BS01 rna 0 0 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 K31 G32 T33 N34 E35 K38 R42 V54 Q55 I59 Q80 L89 V91 G92 S93 A94 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue P12743 18947996 10 ~ 2914 PVYVDFDVPADLEDDALEALEVARDTGAVKKGTNETTKSIERGSAELVFVAEDVQPEEIVMHIPELADEKGVPFIFVEQQDDLGHAAGLEVGSAAAAVTDAGAAATVLEEIADKVEELR 3cxc H 3.0 BS01 rna 0 0 K1 G3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 Y19 D32 R57 A60 A63 R70 R84 R86 K87 F88 F90 R94 E95 N96 M111 R112 A113 P114 F115 G116 R147 R148 M151 K152 T154 T156 K1 G3 M5 R7 K11 P12 A13 Y14 T15 R16 R17 Y19 D32 R57 A60 A63 R70 R84 R86 K87 F88 F90 R94 E95 N96 M100 R101 A102 P103 F104 G105 R136 R137 M140 K141 T143 T145 0003735,0005840,0006412 remove_due_to_license_issue 18947996 10 ~ 2914 KPGAMYRNSSKPAYTRREYISGIPGKKIAQFDMGNNGAGPTYPAQVELVVEKPVQIRHNALEAARVAANRYVQNSGAAANYKFRIRKFPFHVIRENKDGMRAPFGKPVGTAARVHGANHIFIAWVNPDPNVEEAWRRAKMKVTPTINIDSSPAGNA 3cxc I 3.0 BS01 rna 0 0 I18 G20 R21 S24 L31 T47 G48 R49 Q52 K59 R60 I63 N65 N67 G68 Y69 F70 P72 K73 R74 K80 T82 R84 G85 M86 H89 K90 K91 R95 E99 R102 V103 Y104 K128 G140 I15 G17 R18 S21 L28 T44 G45 R46 Q49 K56 R57 I60 N62 N64 G65 Y66 F67 P69 K70 R71 K77 T79 R81 G82 M83 H86 K87 K88 R92 E96 R99 V100 Y101 K125 G137 ? 0003729,0003735,0005840,0006412,0015934,0017148,0019843,0022625,1990904 remove_due_to_license_issue P29198 18947996 10 ~ 2914 AEFDADVIVDARDCIMGRVASQVAEQALDGETVAVVNAERAVITGREEQIVEKYEKRVDIGNDNGYFYPKRPDGIFKRTIRGMLPHKKQRGREAFESVRVYLGNPYDEDGEVLDGTSLDRLSNIKFVTLGEISETLGANKTW 3cxc J 3.0 BS01 rna 0 0 M1 A3 T9 G11 E13 S16 L17 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 S56 R66 R77 K78 R81 R87 M1 A3 T9 G11 E13 S16 L17 K30 I32 S33 V34 H35 G36 Y37 S38 G39 T40 K41 N42 R43 H44 S56 R66 R77 K78 R81 R87 ? 0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P22450 18947996 10 ~ 2914 MEALGADVTQGLEKGSLITCADNTGARELKVISVHGYSGTKNRHPKAGLGDKITVSVTKGTPEMRRQVLEAVVVRQRKPIRRPDGTRVKFEDNAAVIVDENEDPRGTELKGPIAREVAQRFGSVASAATMIV 3cxc K 3.0 BS01 rna 0 0 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 R67 D70 E71 K107 L109 G110 A111 G112 Q113 R115 S126 T1 K3 K4 K5 R6 R8 G9 R11 T12 H13 G14 G16 H18 K19 N20 R21 R22 G23 A24 G25 H26 R27 G28 G29 R30 G31 D32 R35 K37 H38 E39 H41 L46 G47 K48 G50 F51 K52 R53 P54 K56 V57 D65 R67 D70 E71 K102 L104 G105 A106 G107 Q108 R110 S121 ? 0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P12737 18947996 10 ~ 2914 TSKKKRQRGSRTHGGGSHKNRRGAGHRGGRGDAGRDKHEFHNHEPLGKSGFKRPQKVQEEAATIDVREIDENVTLLAADDVAEFRVDVRDVVEEADDADYVKVLGAGQVRHELTLIADDFSEGAREKVEGAGGSVELTDLGEERQ 3cxc L 3.0 BS01 rna 0 0 A1 S3 Y5 R9 K13 K16 W25 Q29 R32 P35 A36 R39 R42 R45 L46 R48 R50 S51 L52 K55 A56 Q58 R68 K69 G70 S71 R73 R74 T75 R76 F77 N78 K79 G80 R81 R82 S83 K84 R85 M86 V88 N89 R90 T92 R93 K94 K95 N96 I97 R99 I100 R104 R107 K108 F109 P110 N111 N116 G124 R125 K127 D135 D137 H138 P139 A140 Q146 W149 T153 R154 R156 L157 F160 R161 L163 S165 R168 C170 R171 G172 R174 Q176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 A192 K193 A194 A1 S3 Y5 R9 K13 K16 W25 Q29 R32 P35 A36 R39 R42 R45 L46 R48 R50 S51 L52 K55 A56 Q58 R68 K69 G70 S71 R73 R74 T75 R76 F77 N78 K79 G80 R81 R82 S83 K84 R85 M86 V88 N89 R90 T92 R93 K94 K95 N96 I97 R99 I100 R104 R107 K108 F109 P110 N111 N116 G124 R125 K127 D135 D137 H138 P139 A140 Q146 W149 T153 R154 R156 L157 F160 R161 L163 S165 R168 C170 R171 G172 R174 Q176 G177 K178 G179 E181 K182 R184 P185 S186 L187 R188 G191 A192 K193 A194 0003735,0005840,0006412 remove_due_to_license_issue 18947996 10 ~ 2914 ARSAYSYIREAWKRPKEGQIAELMWHRMQEWRNEPAVVRIERPTRLDRARSLGYKAKQGIIVVRVAIRKGSSRRTRFNKGRRSKRMMVNRITRKKNIQRIAEERANRKFPNLRVLNSYSVGEDGRHKWHEVILIDPDHPAIKSDDQLSWISRTRHRLRTFRGLTSAGRRCRGLRGQGKGSEKVRPSLRVNGAKA 3cxc M 3.0 BS01 rna 0 0 P4 R5 Y6 K7 P9 R13 A16 T18 D19 H21 Q22 R25 L26 K28 S29 V101 P109 F116 N132 V135 P4 R5 Y6 K7 P9 R13 A16 T18 D19 H21 Q22 R25 L26 K28 S29 V101 P109 F116 N132 V135 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18947996 10 ~ 2914 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3cxc M 3.0 BS02 rna 9 0 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 D162 A1 G3 P4 Y6 V8 M10 R11 R12 R14 R17 T18 Y20 R23 R33 V35 R37 S39 N40 K41 H42 R44 Q46 N53 G54 D55 D56 T57 N77 M78 S108 T110 P111 S113 K114 R141 H146 I147 Y150 Q153 Y159 S160 D162 ? 0000027,0003735,0005840,0006412,0008097,0019843,0022625,1990904 remove_due_to_license_issue P14123 18947996 3001 ~ 3122 ATGPRYKVPMRRRREARTDYHQRLRLLKSGKPRLVARKSNKHVRAQLVTLGPNGDDTLASAHSSDLAEYGWEAPTGNMPSAYLTGLLAGLRAQEAGVEEAVLDIGLNSPTPGSKVFAIQEGAIDAGLDIPHNDDVLADWQRTRGAHIAEYDEQLEEPLYSGDFDAADLPEHFDELRETLLDGDIEL 3cxc N 3.0 BS01 rna 0 0 S1 K2 T3 N4 A12 K15 S16 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 G46 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 R112 V113 I114 R115 S1 K2 T3 N4 A12 K15 S16 R19 A24 V25 D28 K35 P36 R37 R38 E42 N44 G46 R47 R50 Y51 K63 L65 G66 S67 G68 S82 T84 S109 H110 R112 V113 I114 R115 ? 0003723,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12733 18947996 10 ~ 2914 SKTNPRLSSLIADLKSAARSSGGAVWGDVAERLEKPRRTHAEVNLGRIERYAQEDETVVVPGKVLGSGVLQKDVTVAAVDFSGTAETKIDQVGEAVSLEQAIENNPEGSHVRVIR 3cxc O 3.0 BS01 rna 0 0 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 K71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G127 G128 E130 S133 T1 D2 L3 K7 R8 G17 K18 N19 R20 W22 F23 P25 Q28 T36 R37 R41 K52 K54 K55 G56 N57 S58 R59 R61 R63 R65 Q66 K68 R69 A70 K71 H73 Q74 K75 G76 A77 G78 R80 K81 G82 K83 A84 G85 A86 R87 Q88 K91 W94 E95 S96 R99 A100 R102 R109 S116 S117 Y119 R120 Y123 D124 G127 G128 E130 S133 ? 0003723,0003735,0005840,0006412,0019843,0022625,0070180,1990904 remove_due_to_license_issue P14119 18947996 10 ~ 2914 TDLSAQKRLAADVLDVGKNRVWFNPERQGDIADAITREDVRELVDEGAIQAKDKKGNSRGRARERQKKRAKGHQKGAGSRKGKAGARQNSKEDWESRIRAQRTKLRELRDEGTLSSSQYRDLYDKAGGGEFDSVADLERYIDA 3cxc P 3.0 BS01 rna 0 0 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 R21 G22 T23 K38 H40 K42 P45 S46 P48 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 P1 S2 S3 N4 G5 P6 L7 E8 G9 R11 K13 K15 R21 G22 T23 K38 H40 K42 P45 S46 P48 H53 R55 G58 Q59 T60 Q67 G68 D69 A70 D77 G79 K80 K82 T83 I85 Q94 E95 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18947996 10 ~ 2914 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3cxc P 3.0 BS02 rna 9 0 R19 Q27 R19 Q27 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12734 18947996 3001 ~ 3122 PSSNGPLEGTRGKLKNKPRDRGTSPPQRAVEEFDDGEKVHLKIDPSVPNGRFHPRFDGQTGTVEGKQGDAYKVDIVDGGKEKTIIVTAAHLRRQE 3cxc Q 3.0 BS01 rna 0 0 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K36 K60 H62 S64 G65 V66 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 A133 S134 A135 W136 N137 S138 G1 I2 S3 Y4 S5 M17 R19 S24 F25 K26 K29 K36 K60 H62 S64 G65 V66 G67 H68 K69 S70 K71 G74 W75 D76 R79 Y80 E82 K83 N94 N98 H101 H113 A115 A116 H117 V119 Q122 K126 P127 R128 A129 M130 G131 R132 A133 S134 A135 W136 N137 S138 ? 0002181,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P10970 18947996 10 ~ 2914 GISYSVEADPDTTAKAMLRERQMSFKHSKAIAREIKGKTAGEAVDYLEAVIEGDQPVPFKQHNSGVGHKSKVDGWDAGRYPEKASKAFLDLLENAVGNADHQGFDGEAMTIKHVAAHKVGEQQGRKPRAMGRASAWNSPQVDVELILEEP 3cxc R 3.0 BS01 rna 0 0 S1 H9 T11 E12 K13 Q21 K23 R31 S33 K34 N53 Q55 N56 M58 K62 K63 S1 H9 T11 E12 K13 Q21 K23 R31 S33 K34 N53 Q55 N56 M58 K62 K63 ? 0003735,0005840,0006412,0019843,1990904 remove_due_to_license_issue P12732 18947996 10 ~ 2914 SWDVIKHPHVTEKAMNDMDFQNKLQFAVDDRASKGEVADAVEEQYDVTVEQVNTQNTMDGEKKAVVRLSEDDDAQEVASRI 3cxc S 3.0 BS01 rna 0 0 S1 K2 Q3 P4 D5 Q7 R8 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 L79 K81 T82 D83 R89 S94 N95 R97 D105 K107 R111 S1 K2 Q3 P4 D5 Q7 R8 Q11 R12 R13 P15 L16 H17 H20 K21 R24 T26 R32 R38 N39 R41 N43 A44 R52 G53 D54 V65 L67 L79 K81 T82 D83 R89 S94 N95 R97 D105 K107 R111 ? 0003723,0003735,0005840,0006412,0015934,0019843,1990904 remove_due_to_license_issue P10972 18947996 10 ~ 2914 SKQPDKQRKSQRRAPLHERHKQVRATLSADLREEYGQRNVRVNAGDTVEVLRGDFAGEEGEVINVDLDKAVIHVEDVTLEKTDGEEVPRPLDTSNVRVTDLDLEDEKREARLESEDDSA 3cxc T 3.0 BS01 rna 0 0 S34 K35 N38 L42 R44 E50 W51 R56 S31 K32 N35 L39 R41 E47 W48 R53 ? 0003735,0005840,0006412,0008270,0019843,0046872,1990904 remove_due_to_license_issue P14116 18947996 10 ~ 2914 RECDYCGTDIEPGTGTMFVHKDGATTHFCSSKCENNADLGREARNLEWTDTAR 3cxc U 3.0 BS01 rna 0 0 T1 H4 V5 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 T1 H4 V5 E7 R9 Q34 P43 G44 R50 K51 A54 R55 K57 T58 E62 ? 0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P10971 18947996 10 ~ 2914 TVLHVQEIRDMTPAEREAELDDLKTELLNARAVQAAGGAPENPGRIKELRKAIARIKTIQGEEGD 3cxc V 3.0 BS01 rna 0 0 R8 G9 E10 V11 N12 H14 T15 D19 T20 M23 N25 H27 H28 V29 H31 A40 Y41 G43 M44 K47 R69 E74 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 R8 G9 E10 V11 N12 H14 T15 D19 T20 M23 N25 H27 H28 V29 H31 A40 Y41 G43 M44 K47 R69 E74 R108 S113 R117 L118 H119 P120 P121 R122 G123 G124 H125 G127 V128 K129 R154 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18947996 10 ~ 2914 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3cxc V 3.0 BS02 rna 9 0 R8 H14 D50 K129 H130 K133 E134 R8 H14 D50 K129 H130 K133 E134 ? 0000463,0003723,0003735,0005840,0006412,0015934,0019843,0022625,1990904 remove_due_to_license_issue P14121 18947996 3001 ~ 3122 MHALVQLRGEVNMHTDIQDTLEMLNIHHVNHCTLVPETDAYRGMVAKVNDFVAFGEPSQETLETVLATRAEPLEGDADVDDEWVAEHTDYDDISGLAFALLSEETTLREQGLSPTLRLHPPRGGHDGVKHPVKEGGQLGKHDTEGIDDLLEAMR 3cxc W 3.0 BS01 rna 0 0 R8 T11 P13 R15 R18 A19 E20 P21 N22 H23 D27 K28 M30 R34 K39 H40 R49 L50 N55 E56 W59 R61 R63 S68 K69 R2 T5 P7 R9 R12 A13 E14 P15 N16 H17 D21 K22 M24 R28 K33 H34 R43 L44 N49 E50 W53 R55 R57 S62 K63 ? 0002181,0003735,0005840,0006412,0019843,0022625,1990904 remove_due_to_license_issue P18138 18947996 10 ~ 2914 ERVVTIPLRDARAEPNHKRADKAMILIREHLAKHFSVDEDAVRLDPSINEAAWARGRANTPSKIRVRAARFEEEGEAIVEAE 3cxc X 3.0 BS01 rna 0 0 R115 Q119 R120 H121 R122 K125 P126 Q127 F128 R130 Q131 D132 H134 K135 K136 K137 R138 V139 S142 W143 R144 K145 R147 G148 Q149 L150 S151 K152 R154 R155 G156 I157 K158 G159 K160 V164 E165 A166 G167 F168 R169 S170 P171 T172 R175 G176 H178 P179 R186 H188 N189 R204 A206 S207 K208 V209 G210 A211 R212 K213 E215 N230 Y233 R21 Q25 R26 H27 R28 K31 P32 Q33 F34 R36 Q37 D38 H40 K41 K42 K43 R44 V45 S48 W49 R50 K51 R53 G54 Q55 L56 S57 K58 R60 R61 G62 I63 K64 G65 K66 V70 E71 A72 G73 F74 R75 S76 P77 T78 R81 G82 H84 P85 R92 H94 N95 R110 A112 S113 K114 V115 G116 A117 R118 K119 E121 N136 Y139 ? 0000166,0003677,0003735,0005840,0006281,0006412,0019843,0022625,1990904 remove_due_to_license_issue P12736 18947996 10 ~ 2914 TELQARGLTEKTPDLSDEDARLLTQRHRVGKPQFNRQDHHKKKRVSTSWRKPRGQLSKQRRGIKGKGDTVEAGFRSPTAVRGKHPSGFEEVRVHNVDDLEGVDGDTEAVRIASKVGARKRERIEEEAEDAGIRVLNPTYVEV 3cxc Y 3.0 BS01 rna 0 0 R10 G12 R13 G15 P16 R17 Y18 G19 L20 K21 I22 R23 K46 R49 T52 R1 G3 R4 G6 P7 R8 Y9 G10 L11 K12 I13 R14 K37 R40 T43 0003735,0005840,0006412 remove_due_to_license_issue 18947996 10 ~ 2914 RTGRFGPRYGLKIRVRVADVEIKHKKKHKCPVCGFKKLKRAGTGIWMCGHCGYKIAGGCYQPETVAGKAVMKA 3cxc Z 3.0 BS01 rna 0 0 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 G23 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 K44 R46 Y48 E49 W50 Q51 K53 A54 T1 G2 A3 G4 T5 P6 S7 Q8 G9 K10 K11 N12 T13 T14 T15 H16 T17 K18 C19 R20 R21 G23 S26 Y27 H28 T29 K30 K31 K32 S35 K41 S42 K44 R46 Y48 E49 W50 Q51 K53 A54 ? 0003723,0003735,0005840,0006412,0008270,0019843,0022625,0046872,1990904 remove_due_to_license_issue P32410 18947996 10 ~ 2914 TGAGTPSQGKKNTTTHTKCRRCGEKSYHTKKKVCSSCGFGKSAKRRDYEWQSKAGE 3cy2 A 2.01 BS02 MB9 A 1 F49 V52 A65 K67 R122 N172 L174 I185 D186 F17 V20 A33 K35 R88 N138 L140 I151 D152 D167 K169 N172 D186 L193 T204 D133 K135 N138 D152 L159 T170 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=60nM remove_due_to_license_issue P11309 22136433 501 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3cyu A 1.7 BS02 0CR A 1 H94 H119 F131 G132 Q136 L198 T199 T200 P202 H91 H116 F127 G128 Q132 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=60nM remove_due_to_license_issue P00918 18461940 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3cyw A 1.4 BS01 017 A 1 D25 G27 A28 D30 V32 V48 P81 V82 I84 D25 G27 A28 D30 V32 V48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=17nM remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIVGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3cyw B 1.4 BS01 017 A 1 D25 G27 A28 D29 V48 G49 I50 D25 G27 A28 D29 V48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIVGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3cyx A 1.2 BS01 ROC A 1 D25 G27 D29 D30 G48 G49 V50 P81 D25 G27 D29 D30 G48 G49 V50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=10nM remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3cyx B 1.2 BS01 ROC A 1 R8 D25 G27 G48 P81 V82 I84 R8 D25 G27 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3cyz A 1.8 BS01 9OD A 1 M49 M86 F117 I119 M46 M83 F114 I116 ? 0005549,0005615,0007608 Kd=60nM remove_due_to_license_issue Q9U9J6 19481550 124 WVPPEVFDLVAEDKARCMSEHGTTQAQIDDVDKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3cyz B 1.8 BS01 9OD B 1 L53 F117 L49 F113 ? 0005549,0005615,0007608 Kd=60nM remove_due_to_license_issue Q9U9J6 19481550 121 VPPEVFDLVAEDKARCMSEHGTTQAQIDDVDKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3cyz B 1.8 BS02 9OD B 2 K17 D35 Y48 M49 L52 L104 A105 K13 D31 Y44 M45 L48 L100 A101 ? 0005549,0005615,0007608 Kd=60nM remove_due_to_license_issue Q9U9J6 19481550 122 VPPEVFDLVAEDKARCMSEHGTTQAQIDDVDKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3cz1 A 1.5 BS01 NBB A 1 L52 I119 L50 I117 ? 0005549,0005615,0007608 Kd=55nM remove_due_to_license_issue Q9U9J6 19481550 122 DWVPPEVFDLVAEDKARCMSEHGTTQAQIDDVDKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3cz1 B 1.5 BS01 NBB B 1 M49 L52 L53 I119 M45 L48 L49 I115 ? 0005549,0005615,0007608 Kd=55nM remove_due_to_license_issue Q9U9J6 19481550 122 VPPEVFDLVAEDKARCMSEHGTTQAQIDDVDKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3cz1 B 1.5 BS02 NBB B 2 L73 R81 M86 V108 F117 L69 R77 M82 V104 F113 ? 0005549,0005615,0007608 Kd=55nM remove_due_to_license_issue Q9U9J6 19481550 123 VPPEVFDLVAEDKARCMSEHGTTQAQIDDVDKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3czv A 2.0 BS02 AZM A 1 H94 F131 L198 T199 V200 H91 F128 L195 T196 V197 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Ki=16nM remove_due_to_license_issue Ki=17nM, Kd=50nM Q8N1Q1 18618712 263 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 3d04 A 2.4 BS01 SAK A 1 F59 R110 I111 P112 F52 R103 I104 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 Ki=0.9uM remove_due_to_license_issue Q5G940 18780820 163 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3d04 B 2.4 BS01 SAK A 1 I98 Y100 R158 I89 Y91 R149 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 18780820 163 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAER 3d0b A 1.74 BS01 SNX A 1 A55 M98 L107 F138 Y139 W162 A40 M83 L92 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.29uM remove_due_to_license_issue P07900 18511277 233 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3d0e A 2.0 BS01 G93 A 1 V166 A179 K181 E200 L204 F227 M229 Y231 A232 E236 E279 M282 D293 F294 F439 V21 A34 K36 E55 L59 F82 M84 Y86 A87 E91 E134 M137 D148 F149 F294 D275 K277 N280 D293 T313 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 ic50=13nM remove_due_to_license_issue IC50=13nM, Kd=2.1nM, Ki=4nM P31751 18800763 1 KVTMNDFDYLKLLGKGTFGKVILVREKATGRYYAMKILRKEVIIAKDEVAHTVTESRVLQNTRHPFLTALKYAFQTHDRLCFVMEYANGGELFFHLSRERVFTEERARFYGAEIVSALEYLHSRDVVYRDIKLENLMLDKDGHIKITDFGLCKEGISDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHERLFELILMEEIRFPRTLSPEAKSLLAGLLKKDPKQRLGGGPSDAKEVMEHRFFLSINWQDVVQKKLLPPFKPQVTSEVDTRYFDDEFTAQSITITPPDQRTHFPQFDYSASIR 3d14 A 1.9 BS01 AK1 A 1 F157 V160 K175 V187 Q190 L191 E194 L223 A226 L276 D287 F24 V27 K42 V54 Q57 L58 E61 L90 A93 L143 D154 D269 K271 E273 N274 D287 T305 D136 K138 E140 N141 D154 T166 2.7.11.1 0004672,0005524,0006468 ic50=22nM remove_due_to_license_issue IC50=22nM P97477 18678489 1 GPLGSRQWTLEDFDIGRPLGKGKFGNVYLARERQSKFILALKVLFKTQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSRFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSNGELKIADFGWSVHAPSCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGMPPFEAHTYQETYRRISRVEFTFPDFVTEGARDLISRLLKHNASQRLTLAEVLEHPWIKANSS 3d1g A 1.64 BS01 322 A 1 R152 G174 H175 P242 D243 V247 S346 V360 M362 R152 G174 H175 P242 D243 V247 S346 V360 M362 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki~10uM remove_due_to_license_issue P0A988 18678908 501 MKFTVEREHLLKPLQQVSGPLGGRPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 3d1v A 2.7 BS01 D1V A 1 A116 G118 F200 E201 V217 T242 N243 A115 G117 F199 E200 V216 T241 N242 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S32 H63 H85 Y87 E88 A115 M218 S219 N242 V244 H256 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 18790691 293 ENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS 3d1x A 1.05 BS01 ROC A 1 D25 G27 D29 D30 G48 G49 I50 I84 D25 G27 D29 D30 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2.2nM remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d1x B 1.05 BS01 ROC A 1 R8 D25 G27 G48 G49 P81 V82 I84 R8 D25 G27 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d1y A 1.05 BS01 ROC A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=6nM remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFVKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d1y B 1.05 BS01 ROC A 1 R108 D125 G127 G148 I150 P181 I184 R8 D25 G27 G48 I50 P81 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFVKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d1z A 1.3 BS01 017 B 1 D25 G27 A28 D30 V82 I84 D25 G27 A28 D30 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d1z B 1.3 BS01 017 B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.6nM remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d20 A 1.05 BS01 017 A 1 R8 D25 A28 D30 P81 V82 I84 R8 D25 A28 D30 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=5nM remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFVKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d20 B 1.05 BS01 017 A 1 D125 G127 A128 D129 G148 I150 D25 G27 A28 D29 G48 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04587 18597780 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFVKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3d27 A 2.2 BS03 W29 A 1 Y62 Y65 H79 D97 D108 H171 H178 E204 Y59 Y62 H76 D94 D105 H168 H175 E201 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H76 D94 D105 H168 R172 H175 Q179 E201 N205 Q230 E232 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0070006 ic50=55.7uM remove_due_to_license_issue P0AE18 18785729 265 SIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 3d28 A 2.3 BS01 B34 A 1 F193 N316 C366 M414 Y415 Y448 G449 S556 F188 N311 C361 M409 Y410 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=1.4uM remove_due_to_license_issue P26663 18554907 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3d2e A 2.35 BS01 ATP A 1 G10 N11 N12 N13 K69 G205 H206 S207 E272 K275 S279 G342 G343 T344 R346 G9 N10 N11 N12 K68 G204 H205 S206 E271 K274 S278 G341 G342 T343 R345 D8 K69 D174 D203 D7 K68 D173 D202 ? 0005524,0140662 remove_due_to_license_issue P32589 18555782 1001 STPFGLDLGNNNSVLAVARNRGIDIVVNEVSNRSTPSVVGFGPKNRYLGETGKNKQTSNIKNTVANLKRIIGLDYHHPDFEQESKHFTSKLVELDDKKTGAEVRFAGEKHVFSATQLAAMFIDKVKDTVKQDTKANITDVCIAVPPWYTEEQRYNIADAARIAGLNPVRIVNDVTAAGVSYGIFKTDLPEGEEKPRIVAFVDIGHSSYTCSIMAFKKGQLKVLGTACDKHFGGRDFDLAITEHFADEFKTKYKIDIRENPKAYNRILTAAEKLKKVLSANTNAPFSVESVMNDVDVSSQLSREELEELVKPLLERVTEPVTKALAQAKLSAEEVDFVEIIGGTTRIPTLKQSISEAFGKPLSTTLNQDEAIAKGAAFICAIHSPTLRVRPFKFEDIHPYSVSYSWDKQVEDEDHMEVFPAGSSFPSTKLITLNRTGDFSMAASYTDITQLPPNTPEQIANWEITGVQLPEGQDSVPVKLKLRCDPSGLHTIEEAYTIEDTKTVKKDDLTIVAHTFGLDAKKLNELIEKENEMLAQDKLVAETEDRKNTLEEYIYTLRGKLEEEYAPFASDAEKTKLQGMLNKAEEWLYDEGFDSIKAKYIAKYEELASLGNIIRGRYLAKEEEKKQAIR 3d2r A 2.03 BS01 ADP A 1 N258 A262 V298 L306 S312 T313 A328 G331 L334 N229 A233 V269 L277 S283 T284 A291 G294 L297 H250 E254 K257 N258 H221 E225 K228 N229 2.7.11.2 0004672,0004740,0005515,0005524,0005739,0005759,0006885,0008286,0009267,0010510,0010565,0010906,0016301,0042304,0042593,0042594,0045124,0046320,0071398,0072593,2000811 Kd=3.3uM remove_due_to_license_issue Q16654 18658136 501 PREVEHFSRYSPSPLSMKQLLDFGSENCERTSFAFLRQELPVRLANILKEIDILPTQLVNTSSVQLVKSWYIQSLMDLVEFHEKSPDDQKALSDFVDTLIKVRNRHHNVVPTMAQGIIEYKDACDPVTNQNLQYFLDRFYMNRISTRMLMNQHILIFSDSHIGSIDPNCDVVAVVQDAFECSRMLCDQYYLSSPELKLTQVNGKFPDQPIHIVYVPSHLHHMLFELFKNAMRATVEHQENQPSLTPIEVIVVLGKEDLTIKISDRGGGVPLRIIDRLFSYTYSTAPTAPLAGFGYGLPISRLYAKYFQGDLNLYSLSGYGTDAIIYLKALSSESIEKLPVFNKSAFKHYDDWCI 3d2s A 1.7 BS01 rna E 0 E187 N192 R195 C200 R201 E9 N14 R17 C22 R23 ? 0046872 remove_due_to_license_issue Q9NR56 19043415 1 ~ 6 TDRLEVCREYQRGNCNRGENDCRFAHPADSTMIDTNDNTVTVCMDYIKGRCSREKCKYFHPPAHLQA 3d2s B 1.7 BS01 rna F 0 E183 R186 E187 R195 C200 R201 F202 E6 R9 E10 R18 C23 R24 F25 ? 0046872 remove_due_to_license_issue Q9NR56 19043415 1 ~ 5 RTDRLEVCREYQRGNCNRGENDCRFAHPADSTMIDTNDNTVTVCMDYIKGRCSREKCKYFHPPAHLQA 3d2s C 1.7 BS01 rna G 0 E187 N192 R195 C200 R201 F202 E9 N14 R17 C22 R23 F24 ? 0046872 remove_due_to_license_issue Q9NR56 19043415 1 ~ 6 TDRLEVCREYQRGNCNRGENDCRFAHPADSTMIDTNDNTVTVCMDYIKGRCSREKCKYFHPPAHLQA 3d2s D 1.7 BS01 rna H 0 E183 R186 E187 R190 R195 C200 R201 F202 E6 R9 E10 R13 R18 C23 R24 F25 ? 0046872 remove_due_to_license_issue Q9NR56 19043415 1 ~ 5 RTDRLEVCREYQRGNCNRGENDCRFAHPADSTMIDTNDNTVTVCMDYIKGRCSREKCKYFHPPAHLQA 3d2t A 1.85 BS01 1FL A 1 K15 A108 L110 T119 K6 A99 L101 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=75nM remove_due_to_license_issue IC50=12000nM, Kd=407nM, EC50=5600nM P02766 14711308 502 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3d2t B 1.85 BS01 1FL B 1 A108 L110 T119 A94 L96 T105 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=75nM remove_due_to_license_issue IC50=12000nM, Kd=407nM, EC50=5600nM P02766 14711308 500 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANRYTIAALLSPYSYSTTAVVT 3d2w A 1.65 BS01 dna B 0 K192 F194 R197 F221 R227 F229 F231 S258 E261 K3 F5 R8 F32 R38 F40 F42 S69 E72 ? 0003676,0003723 remove_due_to_license_issue Q921F2 19174564 2 GSKVFVGRCTEDMTAEELQQFFCQYGEVVDVFIPKPFRAFAFVTFADDKVAQSLCGEDLIIKGISVHISNAE 3d3p A 1.75 BS02 20A A 1 M347 L393 N395 T407 I410 F414 M431 Q443 F446 M196 L242 N244 T256 I259 F263 M280 Q292 F295 3.1.4.53 0004114,0007165,0008081 ic50=3.1nM remove_due_to_license_issue IC50=3.16nM Q07343 18539455 505 SISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIPQA 3d45 A 3.0 BS01 7MG A 1 K319 N333 W449 W468 D470 D471 K212 N226 W329 W348 D350 D351 3.1.13.4 0003676,0003723,0004535,0005634,0005737,0006402,0046872 remove_due_to_license_issue Q8VDG3 19217398 651 GPMEIIRSNFKINLHKVYQAIEEADFFAIDGEFSGISDSGFDTPEERYQKLKKHSMDFLLFQFGLCAFKYDHTDSKHVTKSFNFYVFPKPFSRSSPDVKFVCQSSSIDFLASQGFDFNKVFCSGIPYLNQEEERQLREQFDEYTKEQEELNDAVGFSRVIHAIANSGKLVVGHNMLLDVMHTIHQFYCPLPADLNEFKEMAICVFPRLLDTKLMASTQPFKDIINNTSLAELEKRLKETPFDPPKVESAEGFPSYDQLHEAGYDAYITGLCFISMANYLGSSARSKLIEPFFNKLFLMRVMDIPYLNLEGPDLQPKRDHVLHVTFPKEWKTSDLYQLFSAFGNIQISWIDDTSAFVSLSQPEQVQIAVNTSKYAESYRIQTYA 3d45 B 3.0 BS01 7MG B 1 W449 W468 D470 D471 W317 W336 D338 D339 3.1.13.4 0003676,0003723,0004535,0005634,0005737,0006402,0046872 remove_due_to_license_issue Q8VDG3 19217398 1152 GPMEIIRSNFKINLHKVYQAIEEADFFAIDGEFSGISDGPSVTALTSGFDTPEERYQKLKKHSMDFLLFQFGLCAFKYDHTDSKHVTKSFNFYVFPKPFSRSSPDVKFVCQSSSIDFLASQGFDFNKVFCSGIPYLNQEEERQLRETKEQEELNDAVGFSRVIHAIANSGKLVVGHNMLLDVMHTIHQFYCPLPADLNEFKEMAICVFPRLLDTKLMASTQPFKDIINNTSLAELEKRLKETPFDPPKVESAEHEAGYDAYITGLCFISMANYLGSKLIEPFFNKLFLMRIPYLNLEGPDLQPKRDHVLHVTFPKEWKTSDLYQLFSAFGNIQISWIDDTSAFVSLSQPEQVQIAVNTSKYAESYRIQTYAEY 3d4f A 1.55 BS02 LN1 A 1 S70 S130 V216 L220 T235 G236 A237 R244 N276 S45 S105 V191 L195 T210 G211 A212 R218 N249 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 18955486 601 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3d4l A 2.0 BS01 605 A 1 E205 E206 S209 F357 R358 S630 Y662 Y666 N710 V711 E167 E168 S171 F319 R320 S592 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=32nM remove_due_to_license_issue IC50=32nM P27487 18524582 1521 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3d4q A 2.8 BS01 SM5 A 1 I463 G464 S465 V471 A481 K483 E501 W531 C532 F583 D594 I16 G17 S18 V24 A34 K36 E54 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.030000nM P15056 18676143 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3d4y A 1.52 BS02 MVL A 1 H90 D92 W95 D204 F206 Y269 D341 W415 H471 D472 Y727 R876 H61 D63 W66 D175 F177 Y240 D312 W386 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=2uM remove_due_to_license_issue Q24451 18759458 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3d4z A 1.39 BS02 GIM A 1 H90 D92 W95 D204 D341 W415 H471 D472 Y727 R876 H61 D63 W66 D175 D312 W386 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=13uM remove_due_to_license_issue Q24451 18759458 1048 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3d50 A 1.79 BS02 OEV A 1 H90 D92 W95 D204 F206 D341 H471 D472 Y727 R876 H61 D63 W66 D175 F177 D312 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=17uM remove_due_to_license_issue Q24451 18759458 1048 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3d51 A 1.43 BS02 GOX A 1 H90 D92 W95 D204 D341 H471 D472 Y727 R876 H61 D63 W66 D175 D312 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=70uM remove_due_to_license_issue Q24451 18759458 1048 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3d52 A 1.6 BS02 GHR A 1 H90 D92 W95 D204 F206 D341 H471 D472 Y727 R876 H61 D63 W66 D175 F177 D312 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=520uM remove_due_to_license_issue Q24451 18759458 1048 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3d5m A 2.2 BS01 4MS A 1 F193 P197 S288 N291 G317 D318 C366 L384 M414 Y415 Y448 G449 S556 F190 P194 S285 N288 G314 D315 C363 L381 M411 Y412 Y445 G446 S553 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50<0.01uM remove_due_to_license_issue P26663 18554907 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3d62 A 2.7 BS01 959 A 1 H41 M49 G143 C145 M165 R188 Q189 H39 M47 G141 C143 M163 R186 Q187 H41 G143 C145 H39 G141 C143 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue P0C6X7 18611220 350 FRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCS 3d67 A 3.4 BS02 GEM A 1 H159 E162 R217 N234 R235 H288 S299 Y341 D348 E363 H159 E162 R217 N234 R235 H288 S299 Y341 D348 E363 H159 E162 R217 H288 E363 H159 E162 R217 H288 E363 3.4.17.20 0003331,0004180,0004181,0005576,0005615,0006508,0007596,0008237,0008270,0009410,0010757,0030163,0042730,0046872,0051918,0070062,0071333,0097421,2000346 remove_due_to_license_issue Q96IY4 18559974 660 AQSGQVLAALPRTSRQVQVLQNLTTTYEIVLWQPVTADLIVKKKQVHFFVNASDVDNVKAHLNVSGIPCSVLLADVEDLIQQQISNDTVSPRASASYYEQYHSLNEIYSWIEFITERHPDMLTKIHIGSSFEKYPLYVLKVSGKEQTAKNAIWIDCGIHAREWISPAFCLWFIGHITQFYGIIGQYTNLLRLVDFYVMPVVNVDGYDYSWKKNRMWRKNRSFYANNHCIGTDLNRNFASKHWCEEGASSSSCSETYCGLYPESEPEVKAVASFLRRNINQIKAYISMHSYSQHIVFPYSYTRSKSKDHEELSLVASEAVRAIEKTSKNTRYTHGHGSETLYLAPGGGDDWIYDLGIKYSFTIELRDTGTYGFLLPERYIKPTCREAFAAVSKIAWHVIRNV 3d6o A 1.58 BS01 U1S A 1 H12 K41 N44 T45 F120 H12 K41 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=77uM remove_due_to_license_issue P61823 19173562 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3d6p A 1.6 BS01 U2S A 1 H12 K41 N44 T45 F120 H12 K41 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=179uM remove_due_to_license_issue P61823 19173562 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3d6q A 1.6 BS01 U3S A 1 H12 K41 N44 T45 F120 H12 K41 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=172uM remove_due_to_license_issue P61823 19173562 127 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3d6y A 2.7 BS01 dna B 0 S7 I8 G9 R23 Y42 R43 S6 I7 G8 R22 Y41 R42 ? 0003677,0003700,0006355 remove_due_to_license_issue P39075 18658145 -13 ~ 12 KESYYSIGEVSKLANVSIKALRYYDKIDLFKPAYVDPDTSYRYYTDSQLIHLDLIKSLKYIGTPLEEMKKAQDLEMEELFAFYTEQERQIREKLDFLSALEQTISLVKKRMKRQMEYPALGEVFVLDEEEIRIIQTEAEGIGPENVLNASYSKLKKFIESADGFTNNSYGATFSFQPYTSIDEMTYRHIFTPVLTNKQISSITPDMEITTIPKGRYACIAYNFSPEHYFLNLQKLIKYIADRQLTVVSDVYELIIPIHYSPKKQEEYRVEMKIEILD 3d6z A 2.6 BS01 dna B 0 S7 I8 G9 R23 Y42 R43 S6 I7 G8 R22 Y41 R42 ? 0003677,0003700,0006355 remove_due_to_license_issue P39075 18658145 -13 ~ 12 KESYYSIGEVSKLANVSIKALRYYDKIDLFKPAYVDPDTSYRYYTDSQLIHLDLIKSLKYIGTPLEEMKKAQDLEMEELFAFYTEQERQIREKLDFLSALEQTISLVKKRMKRQMEYPALGEVFVLDEEEIRIIQTEAEGIGPENVLNASYSKLKKFIESADGFTNNSYGATFSFQPYTSIDEMTYRHIFTPVLTNKQISSITPDMEITTIPKGRYACIAYNFSPEHYFLNLQKLIKYIADRQLTVVSDVYELIIPIHYSPKKQEEYRVEMKIEILD 3d78 A 1.6 BS01 NBB A 1 M49 L52 W116 F117 V118 I119 M49 L52 W116 F117 V118 I119 ? 0005549,0005615,0007608 Kd=23nM remove_due_to_license_issue Q9U9J6 19481550 120 APDWVPPEVFDLVAEDKARCMSEHGTTQAQIDDVNKGNLVNEPSITCYMYCLLEAFSLVDDEANVDEDIMLGLLPDQLQERAQSVMGKCLPTSGSDNCNKIYNLAKCVQESAPDVWFVI 3d7b A 1.6 BS01 U4S A 1 H12 K41 N44 T45 F120 H12 K41 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=203uM remove_due_to_license_issue P61823 19173562 127 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3d7d A 1.69 BS04 FBD A 1 R210 N257 E424 L428 E457 R463 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 L374 E403 R409 G464 N465 R480 R482 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=14nM remove_due_to_license_issue Ki=50.0nM Q04609 19053759 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3d7f A 1.54 BS04 YBY A 1 R210 N257 E424 L428 E457 R463 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 L374 E403 R409 G464 N465 R480 R482 Y495 H496 K640 Y641 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.5nM remove_due_to_license_issue Kd=143nM Q04609 19053759 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3d7g A 1.75 BS04 MUD A 1 R210 N257 E424 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 G464 N465 R480 R482 Y495 H496 K640 Y641 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=17nM remove_due_to_license_issue Q04609 19053759 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3d7h A 1.55 BS04 YC2 A 1 R210 E424 R463 D465 G518 N519 R534 R536 F546 Y552 H553 K699 Y700 R156 E370 R409 D411 G464 N465 R480 R482 F492 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.06nM remove_due_to_license_issue Ki=0.01nM, IC50=0.021000nM Q04609 19053759 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3d7k A 2.49 BS02 D7K A 1 G393 A394 L395 T396 G419 M421 G447 D448 G449 S450 Y453 N475 S477 W478 G479 A480 T481 G392 A393 L394 T395 G418 M420 G446 D447 G448 S449 Y452 N474 S476 W477 G478 A479 T480 L25 G27 A28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 A27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 18570438 572 AMITGGELVVRTLIKAGVEHLFGLHGAHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3d7k A 2.49 BS03 D7K B 1 H26 G27 A28 E50 T73 Q113 H25 G26 A27 E49 T72 Q112 L25 G27 A28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 A27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 18570438 572 AMITGGELVVRTLIKAGVEHLFGLHGAHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3d7k B 2.49 BS01 D7K A 1 H26 G27 A28 E50 T73 Q113 H25 G26 A27 E49 T72 Q112 L25 G27 A28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 A27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 18570438 572 AMITGGELVVRTLIKAGVEHLFGLHGAHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3d7k B 2.49 BS03 D7K B 1 G393 A394 L395 T396 G419 M421 G447 D448 G449 S450 Y453 N475 S477 W478 G479 A480 T481 G392 A393 L394 T395 G418 M420 G446 D447 G448 S449 Y452 N474 S476 W477 G478 A479 T480 L25 G27 A28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 A27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 18570438 572 AMITGGELVVRTLIKAGVEHLFGLHGAHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3d7m A 2.9 BS03 GDP A 1 E43 S44 G45 K46 S47 T48 S151 R176 T177 R178 N269 K270 D272 L273 C325 A326 E10 S11 G12 K13 S14 T15 S109 R134 T135 R136 N227 K228 D230 L231 C283 A284 E43 T48 R178 D200 Q204 E10 T15 R136 D158 Q162 ? 0000287,0001664,0003924,0003925,0005515,0005525,0005634,0005737,0005813,0005829,0005834,0005856,0005886,0005938,0007165,0007186,0007188,0007193,0007198,0010854,0016787,0019001,0019003,0030496,0031683,0031749,0031821,0032794,0032991,0034695,0045542,0046872,0050805,0051301,0060236,0072678,0098794,0098978,0099645,1904322,1904778 remove_due_to_license_issue P10824 19222191 355 VKLLLLGAGESGKSTIVKQMKICHEAGYSEEECKQYKAVVYSNTIQSIIAIIRAMGRLKIDFGDAARADDARQLFVLAAELAGVIKRLWKDSGVQACFNRSREYQLNDSAAYYLNDLDRIAQPNYIPTQQDVLRTRVKTTGIVETHFTFKDLHFKMFDVGGQRSERKKWIHCFEGVTAIIFCVALSDYDLVLAEDEEMNRMHESMKLFDSICNNKWFTDTSIILFLNKKDLFEEKIKKSPLTICYPEYAGSNTYEEAAAYIQCQFEDLNKRKDTKEIYTHFTCATDTKNVCFVFDAVTDVIIKNN 3d7z A 2.1 BS01 GK5 A 1 A51 K53 E71 L75 T106 M109 A111 L167 D168 F169 L171 A48 K50 E68 L72 T103 M106 A108 L164 D165 F166 L168 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=12nM remove_due_to_license_issue Ki=12nM, IC50=75nM Q16539 18614366 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3d83 A 1.9 BS01 GK6 A 1 A51 K53 E71 T106 M109 I141 H148 D168 F169 A48 K50 E68 T103 M106 I138 H145 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=4.4nM remove_due_to_license_issue IC50=6.0nM, Ki=4.4nM Q16539 18602262 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3d8w A 1.7 BS02 D8W A 1 Q92 H94 H96 F131 L198 T199 T200 Q89 H91 H93 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7nM remove_due_to_license_issue P00918 19170619 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3d8y A 1.72 BS01 T3S A 1 K41 V43 N44 T45 F120 K41 V43 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=396uM remove_due_to_license_issue Ki=396000nM P61823 19173562 127 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3d8z A 1.98 BS01 TXS A 1 H12 V43 N44 T45 H119 F120 H12 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=423uM remove_due_to_license_issue P61823 19173562 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3d91 A 2.2 BS01 REM A 1 Q19 D38 G40 Y83 S84 T85 F124 D226 G228 A229 S230 S233 M303 A314 Q16 D35 G37 Y80 S81 T82 F121 D219 G221 A222 S223 S226 M296 A307 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 Kd=131pM remove_due_to_license_issue IC50=1nM, Ki=0.7nM, Kd=131nM P00797 350 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALARH 3d94 A 2.3 BS02 D94 A 1 L975 Q977 F980 V983 A1001 K1003 F1017 M1024 V1033 M1049 M1052 D1056 X1112 G1122 D1123 F1124 L20 Q22 F25 V28 A46 K48 F62 M69 V78 M94 M97 D101 X146 G156 D157 F158 D1105 R1109 N1110 D1123 E1132 D139 R143 N144 D157 E166 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=157nM remove_due_to_license_issue IC50=19nM P08069 18566589 1 VYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLLELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEEN 3d9v A 3.3 BS01 H52 A 1 R84 V90 A103 M153 M156 L205 A215 F368 R79 V85 A98 M148 M151 L200 A210 F363 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=6nM, IC50=30nM Q13464 16249185 416 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSNRRY 3d9z A 1.65 BS02 D9Z A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2nM remove_due_to_license_issue Ki=12nM P00918 19170619 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3da6 A 2.0 BS01 BZ9 A 1 G71 V78 A91 K93 L95 E111 L144 M146 M149 L206 G26 V31 A44 K46 L48 E64 L97 M99 M102 L159 D189 K191 N194 D207 T226 D142 K144 N147 D160 T169 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 19062275 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSGGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAREHTIEEWKELIYKEVMNS 3da9 B 1.8 BS03 44U B 1 Y83 N131 L132 I209 C231 S235 S256 W257 G258 E259 Y47 N95 L96 I172 C194 S198 S219 W220 G221 E222 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Kd=3.1uM remove_due_to_license_issue Kd=3100nM, IC50=18000nM P00734 19371038 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3daj A 2.0 BS01 FXG A 1 L139 K141 G142 K143 F144 N146 V147 A160 K162 L194 Y212 A213 L263 F275 L13 K15 G16 K17 F18 N20 V21 A34 K36 L68 Y86 A87 L137 F149 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T153 2.7.11.1 0004672,0005524,0006468 ic50=2.9uM remove_due_to_license_issue P97477 18579375 1 QWTLEDFDIGRPLGKGKFGNVYLARERQSKFILALKVLFKTQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSRFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSNGELKIADFGWSTLDYLPPEMIHDEKVDLWSLGVLCYEFLVGMPPFEAHTYQETYRRISRVEFTFPDFVTEGARDLISRLLKHNASQRLTLAEVLEHPWIKANSS 3daz A 1.6 BS02 MZM A 1 Q92 H94 H119 V121 F131 L198 T199 Q89 H91 H116 V118 F127 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11.8nM remove_due_to_license_issue Ki=14nM, IC50=21nM, EC50=4e+1nM P00918 19170619 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3db6 A 2.85 BS01 FRS A 1 L45 G46 C53 A66 K68 E87 V100 V114 C119 F169 G179 D180 L22 G23 C30 A43 K45 E64 V77 V91 C96 F146 G156 D157 D162 K164 G166 N167 D180 T200 D139 K141 G143 N144 D157 T177 2.7.11.21 0004672,0005524,0006468 remove_due_to_license_issue Q4KMI8 18678933 1 KEIPDVLVDPRTMKRYMRGRFLGKGGFAKCYEITDMDTKEVFAGKVVPKSMLLKPHQKEKMSTEIAIHKSLDNPHVVGFHGFFEDDDFVYVVLEICRRRSLLELHKRRKAVTEPEARYFMRQTIQGVQYLHNNRVIHRDLKLGNLFLNDDMDVKIGDFGLATKIEFDGERKKDLCGTPNYIAPEVLCKKGHSFEVDIWSLGCILYTLLVGKPPFETSCLKETYIRIKKNEYSVPRHINPVASALIRRMLHADPTLRPSVAELLTDEFFTSGYAPMRLPTSCLTVPPR 3db8 A 3.15 BS01 1FR A 1 K47 A51 C53 A66 K68 C119 R122 F169 K24 A28 C30 A43 K45 C96 R99 F146 D162 K164 G166 N167 D180 D139 K141 G143 N144 D157 2.7.11.21 0004672,0005524,0006468 remove_due_to_license_issue Q4KMI8 18790636 313 KEIPDVLVDPRTMKRYMRGRFLGKGGFAKCYEITDMDTKEVFAGKVVPKSMLLKPHQKEKMSTEIAIHKSLDNPHVVGFHGFFEDDDFVYVVLEICRRRSLLELHKRRKAVTEPEARYFMRQTIQGVQYLHNNRVIHRDLKLGNLFLNDDMDVKIGDFGLATKIHSFEVDIWSLGCILYTLLVGKPPFETSCLKETYIRIKKNEYSVPRHINPVASALIRRMLHADPTLRPSVAELLTDEFFTSGYAPMRLPTSCLTVPPR 3dba A 2.57 BS01 35G A 1 S97 F99 L115 N116 I142 A143 F164 S165 L168 Y174 T176 L197 S43 F45 L61 N62 I88 A89 F110 S111 L114 Y120 T122 L143 3.1.4.35 remove_due_to_license_issue P52731 18614542 1 RLEECNILFELLTEIQDEAGSMEKIVHKTLQRLSQLLAADRCSMFICRSRNGIPEVATRLLNVTPTSKFEDNLVNPDKETVFPLDIGIAGWVAHTKKFFNIPDVKKNNHFSDYLDKKTGYTTVNMMAIPITQGKEVLAVVMALNKLNASEFSKEDEEVFKKYLNFISLVLR 3dba B 2.57 BS01 35G B 1 S97 F99 L115 N116 I142 A143 F164 S165 L168 T176 M179 L197 S43 F45 L61 N62 I88 A89 F110 S111 L114 T122 M125 L143 3.1.4.35 remove_due_to_license_issue P52731 18614542 2 RLEECNILFELLTEIQDEAGSMEKIVHKTLQRLSQLLAADRCSMFICRSRNGIPEVATRLLNVTPTSKFEDNLVNPDKETVFPLDIGIAGWVAHTKKFFNIPDVKKNNHFSDYLDKKTGYTTVNMMAIPITQGKEVLAVVMALNKLNASEFSKEDEEVFKKYLNFISLVLR 3dbd A 3.05 BS01 3FR A 1 L45 K47 C53 K68 L116 C119 R122 F169 L22 K24 C30 K45 L93 C96 R99 F146 D162 K164 G166 N167 D180 D139 K141 G143 N144 D157 2.7.11.21 0004672,0005524,0006468 remove_due_to_license_issue Q4KMI8 18793847 313 KEIPDVLVDPRTMKRYMRGRFLGKGGFAKCYEITDMDTKEVFAGKVVPKSMLLKPHQKEKMSTEIAIHKSLDNPHVVGFHGFFEDDDFVYVVLEICRRRSLLELHKRRKAVTEPEARYFMRQTIQGVQYLHNNRVIHRDLKLGNLFLNDDMDVKIGDFGLATKIHSFEVDIWSLGCILYTLLVGKPPFETSCLKETYIRIKKNEYSVPRHINPVASALIRRMLHADPTLRPSVAELLTDEFFTSGYAPMRLPTSCLTVPPR 3dbs A 2.8 BS01 GD9 A 1 K802 M804 A805 I831 Y867 I879 E880 I881 V882 M953 I963 D964 K565 M567 A568 I594 Y630 I642 E643 I644 V645 M716 I726 D727 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=13nM, Ki=41.8nM, Kd=48nM P48736 18754654 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3dbu A 1.7 BS02 D8W A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8.8nM remove_due_to_license_issue P00918 19170619 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3dc3 A 1.7 BS02 AZM A 1 H94 H119 V121 F131 L198 T199 T200 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=4.9nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 19170619 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3dcc A 1.6 BS02 D9Z A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.1nM remove_due_to_license_issue Ki=12nM P00918 19170619 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3dcq A 1.8 BS03 2G0 A 1 S22 S23 G24 N70 D96 D99 D101 D104 S22 S23 G24 N70 D96 D99 D101 D104 ? 0030246,0044010,0046872 ic50=5.94uM remove_due_to_license_issue Q9HYN5 19101469 201 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 3dcq B 1.8 BS03 2G0 B 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 ic50=5.94uM remove_due_to_license_issue Q9HYN5 19101469 201 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 3dcr A 1.4 BS01 KVS B 1 R8 D25 G27 A28 D29 G48 I84 R8 D25 G27 A28 D29 G48 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue O38732 18657969 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3dcr B 1.4 BS01 KVS B 1 D25 G27 A28 D29 D30 I47 G48 D25 G27 A28 D29 D30 I47 G48 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 ic50=6.3nM remove_due_to_license_issue O38732 18657969 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3dcs A 1.8 BS02 MZM A 1 Q92 H94 H119 V121 F131 L198 T199 Q89 H91 H116 V118 F127 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11.4nM remove_due_to_license_issue Ki=14nM, IC50=21nM, EC50=4e+1nM P00918 19170619 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3dct A 2.5 BS02 064 A 1 M265 F284 L287 T288 M290 H294 M328 F329 R331 I335 H447 W454 W469 M22 F41 L44 T45 M47 H51 M85 F86 R88 I92 H204 W211 W226 ? 0004879,0032052,0038183 remove_due_to_license_issue EC50=65nM, IC50=20nM Q96RI1 18621523 1 ELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEEFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEERIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3dcv A 2.7 BS01 55E A 1 F49 A65 K67 L120 E121 R122 L174 I185 D186 F18 A34 K36 L89 E90 R91 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 18672368 500 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3dcw A 1.5 BS02 EZL A 1 H94 H119 L198 T199 T200 P202 H91 H116 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki<1nM remove_due_to_license_issue Ki=8nM, IC50=3nM, Kd=0.71nM P00918 19170619 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3dd0 A 1.48 BS02 EZL A 1 H94 H119 L198 T199 T200 P201 H92 H117 L195 T196 T197 P198 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki<1nM remove_due_to_license_issue Ki=8nM, IC50=3nM, Kd=0.71nM P00918 19170619 301 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3dd8 A 1.9 BS02 2C7 A 1 H94 H119 V121 L198 T199 P202 H91 H116 V118 L194 T195 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=14nM remove_due_to_license_issue Ki=14nM P00918 18640037 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3ddf A 1.2 BS02 GB6 A 1 H90 D92 W95 D204 Y269 D340 D341 H471 D472 Y727 G877 H60 D62 W65 D174 Y239 D310 D311 H441 D442 Y697 G847 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=67uM remove_due_to_license_issue Q24451 18599296 4001 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ddg A 1.74 BS02 GB7 A 1 H90 D92 W95 D204 Y269 D340 D341 H471 D472 Y727 G877 H60 D62 W65 D174 Y239 D310 D311 H441 D442 Y697 G847 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=1uM remove_due_to_license_issue Q24451 18599296 5001 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ddp C 2.7 BS01 RC8 C 1 E8 K9 I10 G11 A31 F80 L83 H84 Q85 L134 E9 K10 I11 G12 A32 F81 L84 H85 Q86 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=62nM P24941 18574471 299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ddq C 1.8 BS01 RRC C 1 I10 V18 A31 F80 F82 L83 L134 I11 V19 A32 F81 F83 L84 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.21uM remove_due_to_license_issue IC50=700nM, Kd=3400nM, Ki=250nM P24941 18574471 299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 3ddu A 1.56 BS01 552 A 1 F173 M235 R252 C255 F476 S554 W595 R643 V644 F172 M234 R251 C254 F473 S551 W592 R640 V641 Y473 S554 D641 H680 Y470 S551 D638 H677 3.4.21.26 0004252,0005515,0005634,0005737,0005829,0006508,0008236,0016020,0070012 ic50=40nM remove_due_to_license_issue P48147 18606544 901 LSFQYPDVYRDETAVQDYHGHKICDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNSYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESSGIAGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRVINIDFTDPEESKWKVLVPEHEKDVLEWIACVRSNFLVLCYLHDVKNTLQLHDLTTGALLKIFPLDVGSIVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVVKIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGILAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVAACANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLVKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNVDWIP 3deh C 2.5 BS01 RXA C 1 T166 L168 T133 L135 T62 S63 H121 G122 C163 R164 T29 S30 H88 G89 C130 R131 3.4.22.56 0001554,0001666,0001782,0001818,0002020,0004175,0004190,0004197,0004861,0005123,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0006974,0007413,0007507,0007605,0007611,0008047,0008233,0008234,0008627,0009410,0009411,0009611,0009749,0010038,0010165,0014069,0014070,0016005,0016241,0016485,0021766,0030163,0030182,0030216,0030218,0030220,0030889,0031264,0031647,0032025,0032355,0032496,0034349,0034612,0035094,0035556,0042542,0043025,0043029,0043065,0043200,0043525,0044346,0044877,0045165,0045786,0046007,0048011,0051146,0051384,0051402,0051604,0061713,0070269,0071407,0071887,0072734,0097153,0097190,0097193,0097194,0097200,0098693,0098978,0140639,1902004,1904019 ic50=149nM remove_due_to_license_issue IC50=149nM P42574 18768468 300 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIETKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH 3dei C 2.8 BS01 RXB C 1 T166 L168 T255 T134 L136 T212 T62 S63 H121 G122 C163 R164 T30 S31 H89 G90 C131 R132 3.4.22.56 0001554,0001666,0001782,0001818,0002020,0004175,0004190,0004197,0004861,0005123,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0006974,0007413,0007507,0007605,0007611,0008047,0008233,0008234,0008627,0009410,0009411,0009611,0009749,0010038,0010165,0014069,0014070,0016005,0016241,0016485,0021766,0030163,0030182,0030216,0030218,0030220,0030889,0031264,0031647,0032025,0032355,0032496,0034349,0034612,0035094,0035556,0042542,0043025,0043029,0043065,0043200,0043525,0044346,0044877,0045165,0045786,0046007,0048011,0051146,0051384,0051402,0051604,0061713,0070269,0071407,0071887,0072734,0097153,0097190,0097193,0097194,0097200,0098693,0098978,0140639,1902004,1904019 remove_due_to_license_issue IC50=40nM P42574 18768468 300 LDNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIEHKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH 3dej C 2.6 BS01 RXC C 1 T166 E167 L168 T255 T133 E134 L135 T211 T62 S63 H121 G122 C163 R164 T29 S30 H88 G89 C130 R131 3.4.22.56 0001554,0001666,0001782,0001818,0002020,0004175,0004190,0004197,0004861,0005123,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0006974,0007413,0007507,0007605,0007611,0008047,0008233,0008234,0008627,0009410,0009411,0009611,0009749,0010038,0010165,0014069,0014070,0016005,0016241,0016485,0021766,0030163,0030182,0030216,0030218,0030220,0030889,0031264,0031647,0032025,0032355,0032496,0034349,0034612,0035094,0035556,0042542,0043025,0043029,0043065,0043200,0043525,0044346,0044877,0045165,0045786,0046007,0048011,0051146,0051384,0051402,0051604,0061713,0070269,0071407,0071887,0072734,0097153,0097190,0097193,0097194,0097200,0098693,0098978,0140639,1902004,1904019 remove_due_to_license_issue P42574 18768468 300 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIETKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH 3dek A 2.4 BS01 RXD A 1 E123 C163 G165 T166 L168 E90 C130 G132 T133 L135 T62 S63 H121 G122 C163 R164 T29 S30 H88 G89 C130 R131 3.4.22.56 0001554,0001666,0001782,0001818,0002020,0004175,0004190,0004197,0004861,0005123,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0006974,0007413,0007507,0007605,0007611,0008047,0008233,0008234,0008627,0009410,0009411,0009611,0009749,0010038,0010165,0014069,0014070,0016005,0016241,0016485,0021766,0030163,0030182,0030216,0030218,0030220,0030889,0031264,0031647,0032025,0032355,0032496,0034349,0034612,0035094,0035556,0042542,0043025,0043029,0043065,0043200,0043525,0044346,0044877,0045165,0045786,0046007,0048011,0051146,0051384,0051402,0051604,0061713,0070269,0071407,0071887,0072734,0097153,0097190,0097193,0097194,0097200,0098693,0098978,0140639,1902004,1904019 ic50=27nM remove_due_to_license_issue P42574 18768468 300 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIETKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH 3dg8 A 2.58 BS01 RJ6 A 1 C15 A16 L46 D54 F58 N108 I112 L119 L164 C15 A16 L46 D54 F58 N98 I102 L109 L154 L46 D54 L46 D54 1.5.1.3,2.1.1.45 0004146,0046654,0050661 remove_due_to_license_issue P13922 19146480 609 MMEQVCDVFDIYAICACCKVESKNEGKKNEVFNNYTFRGLGNKGVLPWKCISLDMKYFRAVTTYVNESKYEKLKYKRCKYLNKETKKLQNVVVMGRTNWESIPKKFKPLSNRINVILSRTLKKEDFDEDVYIINKVEDLIVLLGKLNYYKCFILGGSVVYQEFLEKKLIKKIYFTRINSTYECDVFFPEINENEYQIISVSDVYTSNNTTLDFIIYKKTNN 3dga A 2.7 BS01 RJ1 A 1 C15 D54 M55 F58 I112 I164 C15 D54 M55 F58 I101 I153 L46 D54 L46 D54 1.5.1.3,2.1.1.45 0004146,0046654,0050661 remove_due_to_license_issue P13922 19146480 609 MMEQVCDVFDIYAICACCKVESKNEGKKNEVFNNYTFRGLGNKGVLPWKCNSLDMKYFCAVTTYVNESKYEKLKYKRCKYLNKEKKLQNVVVMGRTSWESIPKKFKPLSNRINVILSRTLKKEDFDEDVYIINKVEDLIVLLGKLNYYKCFIIGGSVVYQEFLEKKLIKKIYFTRINSTYECDVFFPEINENEYQIISVSDVYTSNNTTLDFIIYKKTN 3dgl A 1.8 BS02 ATP A 1 Y43 M45 F50 H62 G63 Y39 M41 F46 H58 G59 Kd=250nM remove_due_to_license_issue 19522480 81 DDDDKKTNWLKRIYRVRPCVKCKVAPRDWKVKNKHLRIYNMCKTCFNNSIDIGDDTYHGHVDWLMYADS 3dgn A 2.7 BS02 ADP A 1 R41 Y43 M45 F50 H62 G63 H64 R37 Y39 M41 F46 H58 G59 H60 remove_due_to_license_issue 19522480 81 DDDDKKTNWLKRIYRVRPCVKCKVAPRDWKVKNKHLRIYNMCKTCFNNSIDIGDDTYHGHVDWLMYADS 3dgo A 2.5 BS02 ATP A 1 K34 F43 M45 F50 H62 G63 K30 F39 M41 F46 H58 G59 Kd=180nM remove_due_to_license_issue 19522480 82 DDDDKKTNWLKRIYRVRPCVKCKVAPRDWKVKNKHLRIFNMCKTCFNNSIDIGDDTYHGHVDWLMYADS 3dgq A 1.6 BS01 EAA A 1 Y7 R13 I104 Y108 T109 Y8 R14 I105 Y109 T110 Y7 R13 Y8 R14 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 ic50=12uM remove_due_to_license_issue IC50=2.6e+4nM P09211 19396894 211 MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3dhk H 1.73 BS03 23U H 1 Y60A W60D A190 C191 S195 V213 S214 W215 G216 E217 F227 Y47 W50 A192 C193 S197 V217 S218 W219 G220 E221 F231 3.4.21.5 0004252,0005509,0006508,0007596 Ki=47nM remove_due_to_license_issue IC50=12nM P00734 19520086 1601 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3di6 A 2.65 BS01 PDZ A 1 L100 K103 V106 Y181 Y188 W229 L234 H235 P236 Y318 L96 K99 V102 Y177 Y184 W225 L230 H231 P232 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 18632268 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAG 3djf A 2.302 BS01 BC3 A 1 A118 A119 G120 Y202 E203 V219 G220 M221 N245 H259 A111 A112 G113 Y195 E196 V212 G213 M214 N238 H252 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 H259 S31 H59 H81 Y83 E84 A111 M214 S215 N238 S240 H252 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 ic50=0.8uM remove_due_to_license_issue Q9BMI9 20129792 290 VTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESDLKPNHEEVLATGAQRAELMQSWFEKIIEKLPKD 3djf B 2.302 BS01 BC3 B 1 A118 A119 G120 Y202 E203 V219 G220 M221 N245 A112 A113 G114 Y196 E197 V213 G214 M215 N239 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 S32 H60 H82 Y84 E85 A112 M215 S216 N239 S241 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 ic50=0.8uM remove_due_to_license_issue Q9BMI9 20129792 289 SVTANIENVKKVAHHIQKLTSIVPEIGIICGSGLADGVKDKITIPYTKIPNFPQTSVVGHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESAQRAELMQSWFEKIIEKLPKD 3djk A 1.0 BS01 G55 B 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18783203 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3djk B 1.0 BS01 G55 B 1 D125 G127 A128 D129 D130 G148 G149 I150 D25 G27 A28 D29 D30 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=26pM remove_due_to_license_issue P03367 18783203 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3djo A 1.6 BS01 U2P A 1 V43 N44 T45 K66 R85 F120 D121 V43 N44 T45 K66 R85 F120 D121 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=40.8uM remove_due_to_license_issue Ki=40800nM P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djo A 1.6 BS02 U2P B 1 Q11 H12 Q11 H12 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=40.8uM remove_due_to_license_issue Ki=40800nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djo B 1.6 BS01 U2P B 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=40.8uM remove_due_to_license_issue Ki=40800nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djp A 1.6 BS01 UA3 A 1 K41 N44 T45 H119 F120 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=63.2uM remove_due_to_license_issue P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djp B 1.6 BS01 UA3 B 1 V43 N44 T45 H119 F120 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=63.2uM remove_due_to_license_issue P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djq A 1.53 BS01 UDP A 1 V43 N44 T45 H119 F120 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=1046.4uM remove_due_to_license_issue Ki=1046400nM P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djq B 1.53 BS01 UDP B 1 V43 N44 T45 H119 F120 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=1046.4uM remove_due_to_license_issue Ki=1046400nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djv A 1.6 BS01 C3P A 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=27.9uM remove_due_to_license_issue Ki=27900nM P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djv B 1.6 BS01 C3P B 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=27.9uM remove_due_to_license_issue Ki=27900nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djx A 1.69 BS01 C5P A 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=1557.9uM remove_due_to_license_issue P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djx B 1.69 BS01 C5P B 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=1557.9uM remove_due_to_license_issue P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3dk1 A 1.07 BS01 G05 B 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 18843400 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3dk1 B 1.07 BS01 G05 B 1 D125 G127 A128 D129 G148 G149 I150 D25 G27 A28 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.18nM remove_due_to_license_issue P03367 18843400 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3dkf A 1.8 BS01 SX8 A 1 I1084 A1108 L1157 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I35 A54 L103 Y105 M106 D110 R154 M157 A167 D168 Y176 D1204 A1206 R1208 N1209 D1222 D150 A152 R154 N155 D168 2.7.10.1 0004672,0004713,0005524,0006468 Ki=2.7nM remove_due_to_license_issue IC50=4.0nM, Kd=0.820000nM P08581 19934279 1 TVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVKE 3dkg A 1.91 BS01 SX8 A 1 I1084 A1108 L1157 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 A1226 I35 A50 L99 Y101 M102 D106 R150 M153 A163 D164 A168 D1204 A1206 R1208 N1209 D1222 D146 A148 R150 N151 D164 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=4.0nM, Kd=0.820000nM P08581 19934279 1 TVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVICVYHGTLLDKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATY 3dkj A 2.0 BS01 PRP A 1 R196 R311 D313 G353 G383 G384 R176 R291 D293 G333 G363 G364 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 19666527 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 3dkj A 2.0 BS03 PRP B 1 R40 R392 K400 K423 R32 R372 K380 K403 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 19666527 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 3dkj B 2.0 BS01 PRP A 1 R40 R392 K400 K423 R32 R372 K380 K403 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 19666527 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 3dkj B 2.0 BS02 PRP B 1 R196 D313 G353 G383 G384 R176 D293 G333 G363 G364 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 19666527 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 3dln A 1.91 BS01 GLU A 1 Y61 L90 T91 R96 G141 S142 T143 E193 Y58 L87 T88 R93 G138 S139 T140 E190 ? 0015276,0016020 remove_due_to_license_issue P19492 19003990 374 RTIVVTTILESPYVMYKKNHEQLEGNERYEGYCVDLAYEIAKHVRIKYKLSIVGDGKYGARDPETKIWNGMVGELVYGRADIAVAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWSYMKSAEPSVFTKTTADGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSALGTPVNLAVLKLSEQGILDKLKNKWWYDKGEC 3dm6 A 2.6 BS01 757 A 1 G11 Q12 G13 D32 G34 S35 P70 Y71 T72 Q73 G74 F108 Y198 D228 G230 T231 T232 N233 R235 G14 Q15 G16 D35 G37 S38 P73 Y74 T75 Q76 G77 F111 Y189 D219 G221 T222 T223 N224 R226 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D219 T222 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=37nM P56817 18842420 1000 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGYN 3dnd A 2.26 BS02 LL2 A 1 L49 A70 E127 E170 L173 T183 F327 L35 A56 E113 E156 L159 T169 F313 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 18767090 351 VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3dne A 2.0 BS02 LL1 A 1 L49 V57 A70 E121 Y122 V123 L173 T183 D184 F327 L37 V45 A58 E109 Y110 V111 L161 T171 D172 F315 D166 K168 E170 N171 D184 T201 D154 K156 E158 N159 D172 T189 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 18767090 351 ESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3dng A 2.0 BS05 AXA A 1 L193 H197 L214 Y216 P217 N218 Y219 A220 F221 R222 Y227 P230 L114 H118 L135 Y137 P138 N139 Y140 A141 F142 R143 Y148 P151 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=7.4nM remove_due_to_license_issue IC50=7.4nM P22894 19173605 1 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dnt A 1.66 BS01 ATP A 1 V98 A152 G153 A154 Q155 K157 I179 K181 R235 F236 D237 H311 Y331 D332 V97 A143 G144 A145 Q146 K148 I170 K172 R213 F214 D215 H289 Y309 D310 2.7.11.1 0000287,0000976,0001217,0003677,0004674,0004676,0004677,0004679,0004711,0005515,0005524,0005829,0006338,0006355,0022611,0032993,0035175,0035402,0035403,0035979,0040008,0043565,0044010,0044022,0044023,0044024,0044025,0045892,0046677,0072354,0072371,0072518,0106310,0110001,0140823,0140855,0140857,1990244 Kd=18uM remove_due_to_license_issue P23874 19150849 500 PKLVTWMNNQRVGELTKLANGAHTFKYAPEWLASRYARPLSLSLPLQRGNITSDAVFNFFDNLLPDSPIVRDRIVKRYHAKSRQPFDLLSEIGRDSVGAVTLIPIMAWEKLTEARLEEVLTAYKADIPLGMIREENDFRISVAGAQEKTALLRIGNDWCIPKGITPTTHIIKLPIQSVDNEYYCLLLAKELGLNVPDAEIIKAGNVRALAVERFDRRWNAERTVLLRLPQEDMCQTFGLPSSVKYESDGGPGIARIMAFLMGSSEALKDRYDFMKFQVFQWLIGATQGHAKNFSVFIQAGGSYRLTPFYDIISAFPVLGGTGIHISDLKLAMGLNASKGKKTAIDKIYPRHFLATAKVLRFPEVQMHEILSDFARMIPAALDNVKTSLPTDFPENVVTAVESNVLRLHGRLSREY 3dog C 2.7 BS01 NNN C 1 I10 E12 G13 A31 F80 L83 Q85 L134 I11 E13 G14 A32 F81 L84 Q86 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=40nM P24941 18790752 299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 3doy A 2.4 BS01 2BE A 1 F59 K62 F109 I111 P112 F52 K55 F102 I104 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 ic50=1.52uM remove_due_to_license_issue Q5G940 19309082 3001 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3doy B 2.4 BS01 2BE A 1 I98 Y100 R158 I89 Y91 R149 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 3001 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAER 3doz A 2.5 BS01 3BE B 1 F59 K62 I64 R110 F51 K54 I56 R102 H58 I64 G67 V68 E72 H50 I56 G59 V60 E64 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 163 QSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3doz B 2.5 BS01 3BE B 1 I98 Y100 R158 I89 Y91 R149 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 ic50=1.98uM remove_due_to_license_issue Q5G940 19309082 163 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3doz D 2.5 BS01 3BE C 1 F59 I64 F51 I56 H58 I64 G67 V68 E72 H50 I56 G59 V60 E64 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 162 QSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAE 3dp0 A 2.5 BS01 2BC B 1 F59 K62 F109 R110 F52 K55 F102 R103 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 162 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3dp0 B 2.5 BS01 2BC B 1 I98 Y100 R158 E159 I89 Y91 R149 E150 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 ic50=1.42uM remove_due_to_license_issue Q5G940 19309082 162 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3dp1 A 2.3 BS01 2RB B 1 F59 K62 F109 R110 F51 K54 F101 R102 H58 I64 G67 V68 E72 H50 I56 G59 V60 E64 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 162 QSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3dp1 B 2.3 BS01 2RB B 1 I98 R158 I89 R149 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 ic50=9.92uM remove_due_to_license_issue Q5G940 19309082 162 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAER 3dp1 D 2.3 BS01 2RB C 1 F59 I64 F50 I55 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 161 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAER 3dp2 A 2.4 BS01 4BE B 1 F59 K62 F109 R110 F52 K55 F102 R103 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 162 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3dp2 B 2.4 BS01 4BE B 1 I98 Y100 R158 E159 I89 Y91 R149 E150 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 ic50=1.5uM remove_due_to_license_issue Q5G940 19309082 162 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3dp3 A 2.3 BS01 4BB A 1 F59 K62 I64 F109 R110 I111 P112 F52 K55 I57 F102 R103 I104 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 ic50=1.52uM remove_due_to_license_issue Q5G940 19309082 163 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3dp3 B 2.3 BS01 4BB A 1 Y100 R158 Y91 R149 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 163 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAER 3dp3 D 2.3 BS01 4BB C 1 F59 I64 F52 I57 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19309082 162 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAER 3dp4 A 2.11 BS01 AMQ A 1 Y61 L90 T91 R96 G141 S142 T143 L192 E193 M196 Y58 L87 T88 R93 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 Kd=43nM remove_due_to_license_issue Ki=21nM P19492 19003990 374 RTIVVTTILESPYVMYKKNHEQLEGNERYEGYCVDLAYEIAKHVRIKYKLSIVGDGKYGARDPETKIWNGMVGELVYGRADIAVAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWSYMKSAEPSVFTKTTADGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSALGTPVNLAVLKLSEQGILDKLKNKWWYDKGEC 3dp9 A 2.3 BS01 BIG A 1 I50 S76 A77 G78 F152 V153 V172 E173 M174 E175 D198 F208 I49 S75 A76 G77 F151 V152 V171 E172 M173 E174 D197 F207 3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509 Kd=208pM remove_due_to_license_issue Q9KPI8 19270684 301 KIGIIGAMQQEVAILKDLIEDVQEVNQAGCTFYSGQIQGVDVVLLQSGIGKVSAALGTALLISQYAPDVVINTGSAGGFDASLNVGDVVISSEVRHHDADVTAFGYEIGQMAGQPAAFKADEKLMTVAEQALAQLPNTHAVRGLICTGDAFVCTAERQQFIRQHFPSVVAVEMEASAIAQTCHQFKVPFVVVRAISDVADKESPLSFEEFLPLAAKSSSAMVLKMVELL 3dp9 C 2.3 BS01 BIG C 1 I50 S76 A77 G78 F152 V153 V172 E173 M174 E175 D198 F208 I50 S76 A77 G78 F152 V153 V172 E173 M174 E175 D198 F208 3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509 Kd=208pM remove_due_to_license_issue Q9KPI8 19270684 301 MKIGIIGAMQQEVAILKDLIEDVQEVNQAGCTFYSGQIQGVDVVLLQSGIGKVSAALGTALLISQYAPDVVINTGSAGGFDASLNVGDVVISSEVRHHDADVTAFGYEIGQMAGQPAAFKADEKLMTVAEQALAQLPNTHAVRGLICTGDAFVCTAERQQFIRQHFPSVVAVEMEASAIAQTCHQFKVPFVVVRAISDVADKESPLSFEEFLPLAAKSSSAMVLKMVELL 3dpd A 2.85 BS01 41A A 1 K833 Y867 E880 I881 V882 M953 I963 D964 K597 Y631 E644 I645 V646 M717 I727 D728 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=3453nM P48736 18644721 2040 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGRLLYYVNLLLIDHRFLLRRGEYVLHMWQISFNADKLTSATNPDKENSMSISILLDNYCHPIALPKHEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGNKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLGI 3dpe A 1.6 BS05 AXB A 1 I159 L160 A161 L193 H197 L214 Y216 P217 N218 Y219 A220 R222 Y227 S228 P230 I80 L81 A82 L114 H118 L135 Y137 P138 N139 Y140 A141 R143 Y148 S149 P151 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=57nM remove_due_to_license_issue IC50=57nM P22894 19173605 1 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dpf A 2.1 BS05 AXB A 1 I159 L160 A161 L193 H197 L214 Y216 P217 N218 Y219 A220 R222 T224 Y227 S228 P230 I80 L81 A82 L114 H118 L135 Y137 P138 N139 Y140 A141 R143 T145 Y148 S149 P151 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=57nM P22894 19173605 1 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dpk A 1.95 BS01 8C5 A 1 A614 K616 E633 M637 T663 Y665 C666 G669 L785 F797 A56 K58 E75 M79 T105 Y107 C108 G111 L156 F168 D778 A780 R782 N783 D796 N805 D149 A151 R153 N154 D167 N176 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=4.1nM remove_due_to_license_issue P07333,P11362 19193011 923 VRWKIIESSYTFIDPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRQLSSRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVRLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQE 3drp A 2.6 BS01 R8E A 1 K101 K102 K103 V106 V179 Y181 Y188 V189 P225 F227 W229 L234 H235 P236 Y318 K102 K103 K104 V107 V180 Y182 Y189 V190 P226 F228 W230 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 18826204 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3drr A 2.89 BS01 R8E A 1 L100 K101 K103 V106 Y188 V189 P225 F227 W229 L234 H235 P236 Y318 L101 K102 K104 V107 Y189 V190 P226 F228 W230 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 18826204 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3drs A 3.15 BS01 R8D A 1 L100 K101 N103 V106 V108 Y181 Y188 F227 L234 H235 P236 Y318 L101 K102 N104 V107 V109 Y182 Y189 F228 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 18826204 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQV 3ds6 A 2.9 BS01 A17 A 1 V30 Y35 K53 E71 L75 H107 L108 M109 G110 L167 D168 F169 V27 Y32 K50 E68 L72 H104 L105 M106 G107 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T176 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=0.8nM, Ki=0.400000nM Q16539 18817365 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3dst B 1.9 BS01 GRG B 1 H190 G192 C196 R232 K235 Y241 W244 F293 H184 G186 C190 R226 K229 Y235 W238 F287 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H184 R226 K229 D232 C234 Y235 D274 D281 H284 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 Kd=0.83nM remove_due_to_license_issue Q08603 18756270 334 QKDVTIKSDAPDTLLLEKHADYIASYGSKDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3dsu B 1.9 BS01 FPP B 1 F147 H190 G192 C196 Y241 W244 F293 F141 H184 G186 C190 Y235 W238 F287 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H184 R226 K229 D232 C234 Y235 D274 D281 H284 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 Kd=94nM remove_due_to_license_issue Q08603 18756270 334 QKDVTIKSDAPDTLLLEKHADYIASYGSKKYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3dsz A 2.0 BS01 LIZ A 1 Q33 R36 T52 Q54 V66 A68 R70 D77 L79 Y106 F123 T136 Q27 R30 T46 Q48 V60 A62 R64 D71 L73 Y100 F117 T130 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 Kd=17.1nM remove_due_to_license_issue P80188 19227970 187 LIPAPPLSKVPLQQNFQDNQFHGKWYQVGRAGNAALREDKDPQKMTAQIYELKEDKSYNVTAVRFRKKKCDYLTMTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFSITLLGRTKELASELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 3dt1 A 2.8 BS01 P40 A 1 A51 K53 E71 L75 T106 M109 D168 F169 A55 K57 E75 L79 T110 M113 D172 F173 D150 K152 N155 D168 T185 D154 K156 N159 D172 T189 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=0.900000nM Q16539 18817365 361 HMLEMSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3dtc A 2.6 BS01 VIN A 1 I150 F155 V158 A169 K171 M220 F222 A223 R224 G226 L275 T293 D294 I15 F20 V23 A34 K36 M73 F75 A76 R77 G79 L128 T146 D147 D268 K270 S272 N273 D294 A312 D121 K123 S125 N126 D147 A152 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue P80192 18714982 6331 LLEIDFAELTLEEIIGIGGFGKVYRAFWIGDEVAVKAATIENVRQEAKLFAMLKHPNIIALRGVCLKELCLVMEFARGGPLNRVLSGKRIPPDILVNWAVQIARGMNYLHDEAIVPIIHRDLKSSNILILQKVENGDLSNKILKITDFGLGAYAWMAPEVIRASMFSKGSDVWSYGVLLWELLTGEVPFRGIDGLAVAYGVAMNKLALPIPSTCPEPFAKLMEDCWNPDPHSRPSFTNILDQLTT 3du8 A 2.2 BS01 553 A 1 F67 A83 K85 Y134 V135 L188 C199 D200 F33 A49 K51 Y94 V95 L148 C159 D160 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=0.146uM remove_due_to_license_issue P49841 19115845 553 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 3dux H 1.6 BS03 64U H 1 H57 Y60A W60D A190 C191 S195 V213 S214 W215 G216 G226 F227 H43 Y47 W50 A191 C192 S196 V216 S217 W218 G219 G229 F230 3.4.21.5 0004252,0005509,0006508,0007596 Ki=100nM remove_due_to_license_issue Ki=100nM P00734 19520086 901 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3duy A 1.97 BS01 AFJ A 1 D32 G34 Y71 T72 Q73 F108 D228 G230 T231 T232 D35 G37 Y74 T75 Q76 F111 D220 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=1.4uM remove_due_to_license_issue IC50=>10000nM P56817 19195886 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3dv1 A 2.1 BS01 AR9 A 1 Q12 L30 D32 G34 Y71 T72 Q73 F108 I110 Y198 D228 G230 T231 T232 Q15 L33 D35 G37 Y74 T75 Q76 F111 I113 Y190 D220 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.59uM remove_due_to_license_issue IC50=>10000nM P56817 19195887 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3dv5 A 2.1 BS01 BAV A 1 Q12 L30 D32 G34 Y71 T72 Q73 W115 Y198 D228 G230 T231 T232 Q15 L33 D35 G37 Y74 T75 Q76 W118 Y190 D220 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.027uM remove_due_to_license_issue IC50=45nM P56817 19195887 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3dwb A 2.38 BS03 RDF A 1 F149 V565 N566 A567 V604 H607 E608 H611 E667 H732 R738 F49 V455 N456 A457 V494 H497 E498 H501 E557 H622 R628 H607 E608 H611 E667 D671 H732 R738 H497 E498 H501 E557 D561 H622 R628 3.4.24.71 0004222,0006508,0008237 ic50=0.65uM remove_due_to_license_issue IC50=1200nM P42892 18992253 817 SEACVSVTSSILSSMDPTVDPCHDFFSYACGGWIKANPVPDGHSRWGTFSNLWEHNQAIIKHLLENSTASVSEAERKAQVYYRACMNETRIEELRAKPLMELIERLGGWNITGPWAKDNFQDTLQVVTAHYRTSPFFSVYVSADSKNSNSNVIQVDQSGLGLPSRDYYLNKTENEKVLTGYLNYMVQLGKLLGGGDEEAIRPQMQQILDFETALANITIPQEKRRDEELIYHKVTAAELQTLAPAINWLPFLNTIFYPVEINESEPIVVYDKEYLEQISTLINTTDRCLLNNYMIWNLVRKTSSFLDQRFQDADEKFMEVMWKFCVSDTENNLGFALGPMFVKATFAEDSKSIATEIILEIKKAFEESLSTLKWMDEETRKSAKEKADAIYNMIGYPNFIMDPKELDKVFNDYTAVPDLYFENAMRFFNFSWRVTADQLRKAPNRDQWSMTPPMVNAYYSPTKNEIVFPAGILQAPFYTRSSPKALNFGGIGVVVGHELTHAFDDQGREYDKDGNLRPWWKNSSVEAFKRQTECMVEQYSNYSVNGEPVNGRHTLGENIADNGGLKAAYRAYQNWVKKNGAEHSLPTLGLTNNQLFFLGFAQVWCSVRTPESSHEGLITDPHSPSRFRVIGSLSNSKEFSEHFRCPPGSPMNPPHKCEVW 3dx0 A 1.7 BS02 MSN A 1 H90 D92 W95 D204 F206 R228 D341 W415 H471 D472 Y727 H60 D62 W65 D174 F176 R198 D311 W385 H441 D442 Y697 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=36nM remove_due_to_license_issue Ki=36nM Q24451 19101978 1049 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3dx1 A 1.21 BS02 YHO A 1 H90 D92 W95 D204 D341 H471 D472 Y727 H61 D63 W66 D175 D312 H442 D443 Y698 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=265uM remove_due_to_license_issue Ki=2.65e+5nM Q24451 19101978 1050 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3dx2 A 1.4 BS02 MZB A 1 H90 D92 W95 D204 F206 R228 D341 W415 H471 D472 Y727 H61 D63 W66 D175 F177 R199 D312 W386 H442 D443 Y698 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=150nM remove_due_to_license_issue Q24451 19101978 1048 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3dx3 A 1.42 BS02 YTB A 1 H90 D92 W95 D204 D341 H471 D472 Y727 H60 D62 W65 D174 D311 H441 D442 Y697 H90 D92 D204 D341 H471 H60 D62 D174 D311 H441 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=300nM remove_due_to_license_issue Ki=300nM Q24451 19101978 1050 CQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3dx4 A 1.38 BS02 GOO A 1 H90 D92 W95 D204 R228 D341 W415 H471 D472 Y727 H61 D63 W66 D175 R199 D312 W386 H442 D443 Y698 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=76nM remove_due_to_license_issue Ki=76nM Q24451 19101978 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3dxg A 1.39 BS01 U5P A 1 H12 V43 N44 T45 H119 F120 H12 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue P61823 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3dxg A 1.39 BS02 U5P A 2 C65 N67 Q69 N71 A109 E111 V118 H119 C65 N67 Q69 N71 A109 E111 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue P61823 126 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3dxh A 1.4 BS01 UDP A 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue Ki=647000nM P61823 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3dxh A 1.4 BS02 UDP A 2 C65 N67 Q69 N71 A109 E111 V118 H119 C65 N67 Q69 N71 A109 E111 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue Ki=647000nM P61823 126 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3dxh A 1.4 BS03 UDP B 2 Y76 H105 Y76 H105 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue Ki=647000nM P61823 126 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3dxj C 3.0 BS01 NE6 D 1 V1037 W1038 E1041 V1037 W1038 E1041 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue Q8RQE9 18957204 1529 MEIKRFGRIREVIPLPPLTEIQVESYRRALQADVPPEKRENVGIQAAFRETFPIEEEDKGKGGLVLDFLEYRLGEPPFPQDECREKDLTYQAPLYARLQLIHKDTGLIKEDEVFLGHIPLMTEDGSFIINGADRVIVSQIHRSPGVYFTPDPARPGRYIASIIPLPKRGPWIDLEVEPNGVVSMKVNKRKFPLVLLLRVLGYDQETLARELGAYGELVQGLMDESVFAMRPEEALIRLFTLLRPGDPPKRDKAVAYVYGLIADPRRYDLGEAGRYKAEEKLGIRLSGRTLARFEDGEFKDEVFLPTLRYLFALTAGVPGHEVDDIDHLGNRRIRTVGELMTDQFRVGLARLARGVRERMLMGSEDSLTPAKLVNSRPLEAAIREFFSRSQLSQFKDETNPLSSLRHKRRISALGPGGLTRERAGFDVRDVHRTHYGRICPVETPEGANIGLITSLAAYARVDELGFIRTPYRRVVGGVVTDEVVYMTATEEDRYTIAQANTPLEGNRIAAERVVARRKGEPVIVSPEEVEFMDVSPKQVFSVNTNLIPFLEHDDANRALMGSNMQTQAVPLIRAQAPVVMTGLEERVVRDSLAALYAEEDGEVAKVDGNRIVVRYEDGRLVEYPLRRFYRSNQGTALDQRPRVVVGQRVRKGDLLADGPASENGFLALGQNVLVAIMPFDGYNFEDAIVISEELLKRDFYTSIHIERYEIEARDTKLGPERITRDIPHLSEAALRDLDEEGVVRIGAEVKPGDILVGRTSFKGESEPTPEERLLRSIFGEKARDVKDTSLRVPPGEGGIVVRTVRLRRGDPGVELKPGVREVVRVYVAQKRKLQVGDKLANRHGNKGVVAKILPVEDMPHLPDGTPVDVILNPLGVPSRMNLGQILETHLGLAGYFLGQRYISPIFDGAKEPEIKELLAQAFEVYFGKRKGEGFGVDKREVEVLRRAEKLGLVTPGKTPEEQLKELFLQGKVVLYDGRTGEPIEGPIVVGQMFIMKLYHMVEDKMHARSTGPYSLITQQPLGGKAQFGGQRFGEMEVWALEAYGAAHTLQEMLTLKSDDIEGRNAAYEAIIKGEDVPEPSVPESFRVLVKELQALALDVQTLDEKDNPVDIFEGLASKR 3dxj D 3.0 BS05 NE6 D 1 F614 L619 G620 V1099 H1103 A1438 S1439 K1463 I1467 F613 L618 G619 V1098 H1102 A1437 S1438 K1462 I1466 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0006351,0006360,0006366,0006383,0008270,0016779,0034062,0042793,0046872 remove_due_to_license_issue Q8RQE8 18957204 1529 KKEVRKVRIALASPEKIRSWSYGEVEKPETINYRTLKPERDGLFDERIFGPIKDYECACGKYKRQRFEGKVCERCGVEVTKSIVRRYRMGHIELATPAAHIWFVKDVPSKIGTLLDLSATELEQVLYFSKYIVLDPKGAILNGVPVEKRQLLTDEEYRELRYGKQETYPLPPGVDALVKDGEEVVKGQELAPGVVSRLDGVALYRFPRRVRVEYVKKERAGLRLPLAAWVEKEAYKPGEILAELPEPYLFRAEEEGVVELKELEEGAFLVLRREDEPVATYFLPVGMTPLVVHGEIVEKGQPLAEAKGLLRMPRQVRAAQVEAEEEGETVYLTLFLEWTEPKDYRVQPHMNVVVPEGARVEAGDKIVAAIDPEEEVIAEAEGVVHLHEPASILVVKARVYPFEDDVEVSTGDRVAPGDVLADGGKVKSDVYGRVEVDLVRNVVRVVESYDIDARMGAEAIQQLLKELDLEALEKELLEEMKHPSRARRAKARKRLEVVRAFLDSGNRPEWMILEAVPVLPPDLRPMVQVDGGRFATSDLNDLYRRLINRNNRLKKLLAQGAPEIIIRNEKRMLQEAVDALLDNGRRGAPVTNPGSDRPLRSLTDILSGKQGRFRQNLLGKRVDYSGRSVIVVGPQLKLHQCGLPKRMALELFKPFLLKKMEEKGIAPNVKAARRMLERQRDIKDEVWDALEEVIHGKVVLLNRAPTLHRLGIQAFQPVLVEGQSIQLHPLVCEAFNADFDGDQMAVHVPLSSFAQAEARIQMLSAHNLLSPASGEPLAKPSRDIILGLYYITQVRKEKKGAGLEFATPEEALAAHERGEVALNAPIKVAGRETSVGRLKYVFANPDEALLAVAHGIVDLQDVVTVRYMGKRLETSPGRILFARIVAEAVEDEKVAWELIQLDVPQEKNSLKDLVYQAFLRLGMEKTARLLDALKYYGFTFSTTSGITIGIDDAVIPEEKKQYLEEADRKLLQIEQAYEMGFLTDRERYDQILQLWTETTEKVTQAVFKNFEENYPFNPLYVMAQSGARGNPQQIRQLCGLRGLMQKPSGETFEVPVRSSFREGLTVLEYFISSHGARKGGADTALRTADSGYLTRKLVDVTHEIVVREADCGTTNYISVPLFQPDEVTRSLRLRKRADIEAGLYGRVLAREVEVLGVRLEEGRYLSMDDVHLLIKAAEAGEIQEVPVRSPLTCQTRYGVCQKCYGYDLSMARPVSIGEAVGIVAAQSIGEPGTQLTMRTFHTGGVAGAADITQGLPRVIELFEARRPKAKAVISEIDGVVRIEETEEKLSVFVESEGFSKEYKLPKEARLLVKDGDYVEAGQPLTRGAIDPHQLLEAKGPEAVERYLVEEIQKVYRAQGVKLHDKHIEIVVRQMMKYVEVTDPGDSRLLEGQVLEKWDVEALNERLIAEGKTPVAWKPLLMGVTKSALSTKSWLSAASFQNTTHVLTEAAIAGKKDELIGLKENVILGRLIPAGTGSDFVRFTQVVDQKTLKAIEEARKEAVEA 3dxk A 2.7 BS01 N23 B 1 L117 S188 L106 S174 ? 0003779,0005515,0005524,0005634,0005737,0005829,0005856,0005885,0010592,0030030,0034314,0035861,0042995,0045944,0051015,0060271 remove_due_to_license_issue P61157 19648907 395 AGRLPACVVDCGTGYTKLGYAGNTEPQFIIPSCIAIKESVMKGVDDLDFFIGDEAIEKPTYATKWPIRHGIVEDWDLMERFMEQVIFKYLRAEPEDHYFLLTEPPLNTPENREYTAEIMFESFNVPGLYIAVQAVLALAASWTSRERTLTGTVIDSGDGVTHVIPVAEGYVIGSCIKHIPIAGRDITYFIQQLLRDREVGIPPEQSLETAKAVKERYSYVCPDLVKEFNKYDTDGSKWIKQYTGINAISKKFSIDVGYERFLGPEIFFHPEFANPDFTQPISEVVDEVIQNCPIDVRRPLYKNIVLSGGSTMFRDFGRRLQRDLKRTVDARLKLSEELSKPKPIDVQVITHHMQRYAVWFGGSMLASTPEFYQVCHTKKDYEEIGPSICRHNPVFGV 3dxk B 2.7 BS01 N23 B 1 Y202 A203 F204 D209 L246 P247 D248 R250 Y61 A62 F63 D68 L105 P106 D107 R109 ? 0003779,0005515,0005524,0005634,0005737,0005829,0005856,0005885,0005938,0010592,0034314,0035861,0042995,0045944,0051015,1905168,2001032 remove_due_to_license_issue A7MB62 19648907 395 QAVLTLYAQGLLGVVVDSGDGVTHICPVYEGFSLPHLTRRLDIAGRDITRYLIKLLLLRGYAFNHSADFETVRMIKEKLCYVGYNIEQEQKLALETTVLVESYTLPDGRIIKVGGERFEAPEALFQPHLINVEGVGVAELLFNTIQAADIDTRSEFYKHIVLSGGSTMYPGLPSRLERELKQLYLERVLKGDVEKLSKFKIRIEDPPRRKH 3dxm A 2.85 BS01 N24 A 1 C12 E84 M89 M93 T113 N118 T126 C10 E71 M76 M80 T100 N105 T113 ? 0003779,0005515,0005524,0005634,0005737,0005829,0005856,0005885,0010592,0030030,0034314,0035861,0042995,0045944,0051015,0060271 remove_due_to_license_issue P61157 19648907 419 GRLPACVVDCGTGYTKLGYAGNTEPQFIIPSCIAIKEVMKGVDDLDFFIGDEAIEKPTYATKWPIRHGIVEDWDLMERFMEQVIFKYLRAEPEDHYFLLTEPPLNTPENREYTAEIMFESFNVPGLYIAVQAVLALAASWTSRQVGERTLTGTVIDSGDGVTHVIPVAEGYVIGSCIKHIPIAGRDITYFIQQLLRDREVGIPPEQSLETAKAVKERYSYVCPDLVKEFNKYDTDGSKWIKQYTGINAISKKEFSIDVGYERFLGPEIFFHPEFANPDFTQPISEVVDEVIQNCPIDVRRPLYKNIVLSGGSTMFRDFGRRLQRDLKRTVDARLKLSEELSKPKPIDVQVITHHMQRYAVWFGGSMLASTPEFYQVCHTKKDYEEIGPSICRHNPVFGV 3dy6 A 2.9 BS01 DY6 A 1 W264 R284 C285 T288 T289 F327 L330 L339 V341 V348 H449 Y473 W51 R66 C67 T70 T71 F109 L112 L121 V123 V130 H231 Y255 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=1259nM, IC50=126nM Q03181 18722772 478 VADLKAFSKHIYNAYLKNFNMTKKKARSILTAPFVIHDIETLWQAEKGLVWGLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKD 3dya A 2.3 BS01 PZL A 1 K102 K103 V106 Y188 V189 F227 W229 L234 H235 P236 Y318 K98 K99 V102 Y184 V185 F223 W225 L230 H231 P232 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=3nM remove_due_to_license_issue EC50=1nM, IC50=3nM P04585 19007201 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAG 3dyo A 1.8 BS03 IPT A 1 N102 D201 E461 E537 H540 N604 W999 N90 D189 E449 E525 H528 N592 W987 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo A 1.8 BS04 IPT A 2 E304 P306 R645 D648 Q702 W708 E292 P294 R633 D636 Q690 W696 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2002 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo A 1.8 BS05 IPT A 3 R230 F231 N232 R237 A238 R218 F219 N220 R225 A226 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2003 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo A 1.8 BS06 IPT B 1 D507 E508 D495 E496 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2004 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo D 1.8 BS01 IPT C 3 D507 E508 D495 E496 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2004 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo D 1.8 BS04 IPT D 1 R230 F231 N232 A238 V239 R218 F219 N220 A226 V227 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2003 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo D 1.8 BS05 IPT D 2 N102 D201 E461 H540 N604 W999 N90 D189 E449 H528 N592 W987 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dyo D 1.8 BS06 IPT D 3 E304 R645 D648 Q702 W708 E292 R633 D636 Q690 W696 D201 H357 H391 E416 N418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 N406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5mM remove_due_to_license_issue Ki=7.6e+4nM P00722 19472413 2002 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETNGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3dz2 A 1.86 BS01 A8M A 1 X68 C82 F223 N224 C226 G227 Y228 H243 I244 T245 E247 X1 C15 F152 N153 C155 G156 Y157 H172 I173 T174 E176 S229 H243 S157 H171 4.1.1.50 0004014,0006597,0008295 ic50=70uM remove_due_to_license_issue IC50=70000nM P17707 19209891 368 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAAYCMGRMNSDCWYLYTLDFPESQPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQSSKCEGFKRLDCQSAMFNDYNFVFTSFAK 3dz2 B 1.86 BS01 A8M A 1 F7 E11 S66 E67 F4 E8 S59 E60 E67 E60 4.1.1.50 0004014,0008295 remove_due_to_license_issue IC50=70000nM P17707 19209891 368 AHFFEGTEKLLEVWFSRQQQGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 3dz4 A 1.84 BS01 C8M A 1 X68 C82 F223 N224 C226 G227 S229 I244 T245 E247 X1 C15 F150 N151 C153 G154 S156 I171 T172 E174 S229 H243 S155 H169 4.1.1.50 0004014,0006597,0008295 ic50=400nM remove_due_to_license_issue IC50=400nM P17707 19209891 368 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAAYCMGRMNSDCWYLYTLDFSQPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQSSKCRKIEGFKRLDCQSAMFNDYNFVFTSFAK 3dz4 B 1.84 BS01 C8M A 1 F7 S66 E67 F4 S60 E61 E67 E61 4.1.1.50 0004014,0008295 remove_due_to_license_issue IC50=400nM P17707 19209891 368 AHFFEGTEKLLEVWFSRQQPQGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 3dz5 A 2.43 BS01 M8M A 1 X68 F223 C226 G227 Y228 S229 H243 I244 T245 E247 X1 F149 C152 G153 Y154 S155 H169 I170 T171 E173 S229 H243 S154 H168 4.1.1.50 0004014,0006597,0008295 remove_due_to_license_issue IC50=7nM P17707 19209891 368 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAAYCMGRMNSDCWYLYTLDSQPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQSSQKIEGFKRLDCQSAMFNDYNFVFTSFAKK 3dz5 B 2.43 BS01 M8M A 1 F7 S66 E67 F4 S54 E55 E67 E55 4.1.1.50 0004014,0008295 remove_due_to_license_issue IC50=7nM P17707 19209891 368 AHFFEGTEKLLEVWFGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 3dz6 A 1.83 BS01 M8E A 1 X68 C82 F223 N224 C226 G227 Y228 I244 T245 E247 X1 C15 F147 N148 C150 G151 Y152 I168 T169 E171 S229 H243 S152 H166 4.1.1.50 0004014,0006597,0008295 ic50=15nM remove_due_to_license_issue P17707 19209891 368 cSMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAAYCMGRMNSDCWYLYTLDFDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNIEGFKRLDCQSAMFNDYNFVFTSFAKK 3dz6 B 1.83 BS01 M8E A 1 F7 L65 S66 E67 F3 L54 S55 E56 E67 E56 4.1.1.50 0004014,0008295 remove_due_to_license_issue P17707 19209891 368 HFFEGTEKLLEVWFSRGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 3dzt A 1.8 BS01 EAH A 1 F13 M17 W34 W37 N39 Y113 G130 K149 F13 M17 W34 W37 N39 Y113 G130 K149 ? 0005549,0005576,0005615,0007608,0019863,0035821,0042311,0050688,0090729 Kd=60.2nM remove_due_to_license_issue P18153 19234127 305 MGPFDPEEMLFIFTRCMEDNLEDGANRLPMLAKWKEWINEPVDSPATQCFGKCVLVRTGLYDPVAQKFDASVIQEQFKAYPSLGEKSKVEAYANAVKQLPSTNNDCAAVFKAYDPVHKAHKDTSKNLFHGNKELTKGLYEKLGKDIRQKKQSYFEFCENKYYPAGSDKRQQLCQIRQYTVLDDALFKEHTDCVMKGIRYITKDNQLDVEEVKRDFKLVNKDTKALEEVLNDCKSKEPSNAKEKSWHYYKCLVESSVKDDFKEAFDYREVRSQIYAFNLPKNQAYSKPAVMEIDGKQCP 3e01 A 2.95 BS01 PZ2 A 1 L100 K103 V106 Y188 F227 W229 H235 P236 Y318 L96 K99 V102 Y184 F223 W225 H231 P232 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue EC50=17nM P04585 19007201 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGI 3e0p B 1.7 BS01 B3C B 1 H57 S99 Q100 D102 P172I A190 C191 Q192 G193 S195 V213 S214 W215 G216 D217 A218 H41 S87 Q88 D90 P170 A189 C190 Q191 G192 S194 V212 S213 W214 G215 D216 A217 D102 D90 3.4.21.- 0004252,0006508 remove_due_to_license_issue Q16651 18752942 1 ITGGSSAVAGQWPWQVSITYEGVHVCGGSLVSEQWVLSAAHCFPSEHHKEAYEVKLGAHQLDSYSEDAKVSTLKDIIPHPSYLQEGSQGDIALLQLSRPITFSRYIRPISLPAAQASFPNGLHCTVTGWGHVAPSVSLLTPKPLQQLEVPLISRETCNSLYNIDAKPEEPHFVQEDMVCAGYVEGGKDACQGDSGGPLSCPVEGLWYLTGIVSWGDACGARNRPGVYTLASSYASWIQSKVTELQP 3e0q A 1.9 BS01 JFD A 1 A119 G120 Y202 E203 V219 G220 M221 N245 A112 G113 Y195 E196 V212 G213 M214 N238 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 H259 S31 H59 H81 Y83 E84 A111 M214 S215 N238 S240 H252 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 remove_due_to_license_issue Q9BMI9 20122887 400 VTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESDLKPNHEEVLATGAQRAELMQSWFEKIIEKLPKD 3e0q B 1.9 BS01 JFD B 1 G120 Y202 E203 G220 N245 G114 Y196 E197 G214 N239 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 S32 H60 H82 Y84 E85 A112 M215 S216 N239 S241 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 remove_due_to_license_issue Q9BMI9 20122887 401 SVTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVEQRAELMQSWFEKIIEKLPKD 3e12 A 1.7 BS03 KD0 A 1 K41 K46 N48 R49 S50 Q99 K124 H185 D233 K40 K45 N47 R48 S49 Q98 K123 H184 D227 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0046364 remove_due_to_license_issue O66496 19228070 268 EKFLVIAGPCAIESEELLLKVGEEIKRLSEKFKEVEFVFKSSFDKANRSSIHSFRGHGLEYGVKALRKVKEEFGLKITTDIHESWQAEPVAEVADIIQIPAFLCRQTDLLLAAAKTGRAVNVKKGQFLAPWDTKNVVEKLKFGGAKEIYLTERGTTFGYNNLVVDFRSLPIMKQWAKVIYDATHSVQLPGGGGMREFIFPLIRAAVAVGCDGVFMETHPEPEKALSDASTQLPLSQLEGIIEAILEIREVASKYYETI 3e12 B 1.7 BS03 KD0 B 1 K41 K46 N48 R49 S50 Q99 K124 H185 D233 K39 K44 N46 R47 S48 Q97 K122 H183 D225 2.5.1.55 0005737,0005829,0008676,0009058,0009103,0016740,0019294,0046364 remove_due_to_license_issue O66496 19228070 268 KFLVIAGPCAIESEELLLKVGEEIKRLSEKFKEVEFVFKSSFDKANRSSIHSFRGHGLEYGVKALRKVKEEFGLKITTDIHESWQAEPVAEVADIIQIPAFLCRQTDLLLAAAKTGRAVNVKKGQFLAPWDTKNVVEKLKFGGAKEIYLTERGTTFGYNNLVVDFRSLPIMKQWAKVIYDATHSVQLPGGGMREFIFPLIRAAVAVGCDGVFMETHPEPEKALSDASTQLPLSQLEGIIEAILEIREVASKYYETI 3e16 B 1.6 BS01 B4C B 1 H57 E97 G98 P172I H172J F172K A190 Q192 G193 S195 V213 W215 G216 D217 H41 E85 G86 P170 H171 F172 A189 Q191 G192 S194 V212 W214 G215 D216 D102 D90 3.4.21.- 0004252,0006508 remove_due_to_license_issue Q16651 18752942 1 ITGGSSAVAGQWPWQVSITYEGVHVCGGSLVSEQWVLSAAHCFPSEHHKEAYEVKLGAHQLDSYSEDAKVSTLKDIIPHPSYLQEGSQGDIALLQLSRPITFSRYIRPISLPAAQASFPNGLHCTVTGWGHVAPSVSLLTPKPLQQLEVPLISRETCNSLYNIDAKPEEPHFVQEDMVCAGYVEGGKDACQGDSGGPLSCPVEGLWYLTGIVSWGDACGARNRPGVYTLASSYASWIQSKVTELQPR 3e2m A 2.0 BS01 E2M A 1 F153 Y166 Y257 I259 E284 F285 K287 L302 F26 Y39 Y130 I132 E157 F158 K160 L175 ? ic50=0.4nM remove_due_to_license_issue IC50=0.4nM P20701 18783948 1 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 3e2m B 2.0 BS01 E2M A 1 V308 I309 V181 I182 ? ic50=0.4nM remove_due_to_license_issue IC50=0.4nM P20701 18783948 1 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 3e2m B 2.0 BS02 E2M B 1 F153 Y166 I235 Y257 I259 E284 F285 K287 E301 L302 F26 Y39 I108 Y130 I132 E157 F158 K160 E174 L175 ? ic50=0.4nM remove_due_to_license_issue IC50=0.4nM P20701 18783948 1 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIYVI 3e37 B 1.8 BS03 ED5 B 1 W104 Y156 R204 Y207 G252 C256 D299 W305 D361 Y363 H364 W88 Y140 R188 Y191 G236 C240 D283 W289 D345 Y347 H348 H250 R293 K296 D299 C301 Y302 D354 D361 H364 H234 R277 K280 D283 C285 Y286 D338 D345 H348 2.5.1.58 0003824,0004659,0004660,0005515,0005829,0005875,0005965,0006629,0008270,0008318,0018343,0046872 ic50=4050nM remove_due_to_license_issue P49356 19246009 1 SSPVWSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPEGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYDIINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKRERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVLGVPENALQPTHPVYNIGPDKVIQATTYFLQKPVPGFE 3e3b X 3.2 BS01 CCK X 1 L46 V54 V67 K69 F114 I117 M164 I175 D176 L46 V54 V67 K69 F114 I117 M164 I175 D176 N162 D176 S195 N162 D176 S195 2.7.11.1 0000785,0001669,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005829,0005956,0006302,0006338,0006468,0006915,0006974,0007283,0016055,0021987,0031519,0032435,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0097421,0106310,0140823,0140855,0140857,1901524,1903955,1905818,1990244,2001234 remove_due_to_license_issue P19784 19193990 351 MPGPAAGSRARVYAEVNSLRSREYWDYEAHVPSWGNQDDYQLVRKLGRGKYSEVFEAINITNNERVVVKILKPVKKKKIKREVKILENLRGGTNIIKLIDTVKDPVSKTPALVFEYINNTDFKQLYQILTDFDIRFYMYELLKALDYCHSKGIMHRDVKPHNVMIDHQQKKLRLIDWGLAEFYHPAQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRREPFFHGQDNYDQLVRIAKVLGTEELYGYLKKYHIDLDPHFNDILGQHSRKRWENFIHSENRHLVSPEALDLLDKLLRYDHQQRLTAKEAMEHPYFYPVVKEQSQ 3e3c A 2.5 BS01 HHG A 1 F12 L24 S38 Y40 S63 V64 Y71 F19 L31 S45 Y47 S70 V71 Y78 ? remove_due_to_license_issue Q7DB61 19228114 150 GLVPRGSMIMKDGIYSIIFISNEDSCGEGILIKNGNMITGGDIASVYQGVLSEDEDIILHVHRYNYEIPSVLNIEQDYQLVIPKKVLSNDNNLTLHCHVRGNEKLFVDVYAKFIEPLV 3e3u A 1.56 BS01 NVC A 1 G49 V50 G51 Q56 G105 C106 L107 L141 H148 E149 H152 F195 G48 V49 G50 Q55 G104 C105 L106 L140 H147 E148 H151 F194 G51 Q56 C106 L107 H148 E149 H152 G50 Q55 C105 L106 H147 E148 H151 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=0.013uM remove_due_to_license_issue IC50=13nM P9WIJ3 19008098 201 AVVPIRIVGDPVLHTATTPVTVAADGSLPADLAQLIATMYDTMDAANGVGLAANQIGCSLRLFVYDCAADRAMTARRRGVVINPVLETSEIPETMPDPDTDDEGCLSVPGESFPTGRAKWARVTGLDADGSPVSIEGTGLFARMLQHETGHLDGFLYLDRLIGRYARNAKRAVKSHGWGVPGLSWLPGEDPDPFGH 3e3u A 1.56 BS02 NVC A 2 V4 P5 Q35 T39 V3 P4 Q34 T38 G51 Q56 C106 L107 H148 E149 H152 G50 Q55 C105 L106 H147 E148 H151 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=0.013uM remove_due_to_license_issue IC50=13nM P9WIJ3 19008098 202 AVVPIRIVGDPVLHTATTPVTVAADGSLPADLAQLIATMYDTMDAANGVGLAANQIGCSLRLFVYDCAADRAMTARRRGVVINPVLETSEIPETMPDPDTDDEGCLSVPGESFPTGRAKWARVTGLDADGSPVSIEGTGLFARMLQHETGHLDGFLYLDRLIGRYARNAKRAVKSHGWGVPGLSWLPGEDPDPFGH 3e3u A 1.56 BS03 NVC A 3 V13 T19 C59 S60 V12 T18 C58 S59 G51 Q56 C106 L107 H148 E149 H152 G50 Q55 C105 L106 H147 E148 H151 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=0.013uM remove_due_to_license_issue IC50=13nM P9WIJ3 19008098 203 AVVPIRIVGDPVLHTATTPVTVAADGSLPADLAQLIATMYDTMDAANGVGLAANQIGCSLRLFVYDCAADRAMTARRRGVVINPVLETSEIPETMPDPDTDDEGCLSVPGESFPTGRAKWARVTGLDADGSPVSIEGTGLFARMLQHETGHLDGFLYLDRLIGRYARNAKRAVKSHGWGVPGLSWLPGEDPDPFGH 3e4a A 2.6 BS03 QIX A 1 H108 Q111 H112 F115 L116 N139 A140 E189 F820 R824 Y831 H66 Q69 H70 F73 L74 N97 A98 E147 F778 R782 Y789 Q111 Q69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 20498699 2001 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNPVVGNLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 3e51 A 1.9 BS01 N35 A 1 F193 N291 D318 C366 S368 L384 G410 M414 Y415 Q446 Y448 S556 F188 N286 D313 C361 S363 L379 G405 M409 Y410 Q441 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.014uM remove_due_to_license_issue P26663 18796353 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3e5a A 2.3 BS01 VX6 A 1 L139 F144 A160 E211 Y212 A213 P214 G216 T217 L263 A273 D274 L15 F20 A36 E87 Y88 A89 P90 G92 T93 L139 A149 D150 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Ki=5.9nM remove_due_to_license_issue Ki=0.600000nM, IC50=20nM, Kd=4.1nM O14965 18662907 500 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3e5u C 1.83 BS01 3C4 C 1 Y76 I84 G85 K86 T90 N92 I94 K133 Y68 I76 G77 K78 T82 N84 I86 K125 ? 0003677,0006355 remove_due_to_license_issue B8FW11 18717788 504 DFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLASLKRENILDKKKNKIIVYNLGELKHLSE 3e5u C 1.83 BS02 3C4 D 1 L131 V134 L123 V126 ? 0003677,0006355 remove_due_to_license_issue B8FW11 18717788 502 DFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLASLKRENILDKKKNKIIVYNLGELKHLSE 3e5u D 1.83 BS01 3C4 C 1 L131 V134 L123 V126 ? 0003677,0006355 remove_due_to_license_issue B8FW11 18717788 504 DFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLASLKRENILDKKKNKIIVYNLGELKHLSEQ 3e5u D 1.83 BS02 3C4 D 1 Y76 I84 G85 K86 T90 N92 K133 Y68 I76 G77 K78 T82 N84 K125 ? 0003677,0006355 remove_due_to_license_issue B8FW11 18717788 502 DFCGAIIPDNFFPIEKLRNYTQMGLIRDFAKGSAVIMPGEEITSMIFLVEGKIKLDIIFEDGSEKLLYYAGGNSLIGKLYPTGNNIYATAMEPTRTCWFSEKSLRTVFRTDEDMIFEIFKNYLTKVAYYARQVAEMNTYNPTIRILRLFYELCSSQGKRVGDTYEITMPLSQKSIGEITGVHHVTVSRVLASLKRENILDKKKNKIIVYNLGELKHLSEQ 3e62 A 1.922 BS01 5B1 A 1 V863 A880 M929 E930 Y931 L932 L983 V25 A42 M91 E92 Y93 L94 L145 D976 A978 R980 N981 D994 S1016 D138 A140 R142 N143 D156 S178 2.7.10.2 0004672,0004713,0005524,0006468 ic50=40.9uM remove_due_to_license_issue IC50=40900nM O60674 19019674 1 RDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 3e63 A 1.9 BS01 5B2 A 1 L855 G856 K857 V863 A880 M929 E930 Y931 L932 L983 L16 G17 K18 V24 A41 M90 E91 Y92 L93 L144 D976 A978 R980 N981 D994 S1016 D137 A139 R141 N142 D155 S177 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.6uM remove_due_to_license_issue IC50=1600nM O60674 19019674 1 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 3e64 A 1.8 BS01 5B3 A 1 G861 V863 A880 M929 E930 Y931 L932 L983 D994 G23 V25 A42 M91 E92 Y93 L94 L145 D156 D976 A978 R980 N981 D994 S1016 D138 A140 R142 N143 D156 S178 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.078uM remove_due_to_license_issue IC50=78nM O60674 19019674 1 RDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 3e6k A 2.1 BS03 ABH A 1 D124 H126 D128 N130 S137 H141 D232 E277 D119 H121 D123 N125 S132 H136 D227 E272 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=7000nM remove_due_to_license_issue P05089 19093830 552 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVAPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHK 3e6v A 1.72 BS03 ABH A 1 D124 D128 S137 H141 D232 E277 D119 D123 S132 H136 D227 E272 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=147nM remove_due_to_license_issue P05089 19093830 552 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVNPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 3e6y A 2.5 BS02 CW1 A 1 N49 F126 K129 P174 D222 N45 F122 K125 P170 D218 ? 0005737,0007165,0008104 Kd=2.5uM remove_due_to_license_issue P93343 19244612 261 PTAREENVYMAKLAEQAERYEEMVEFMEKVSNSLGSEELTVEERNLLSVAYKNVIGARRASWRIISSIEQKEESRGNEEHVNSIREYRSKIENELSKICDGILKLLDAKLIPSAASGDSKVFYLKMKGDYHRYLAEFKTGAERKEAAESTLTAYKAAQDIATTELAPTHPIRLGLALNFSVFYYEILNSPDRACNLAKQAFDEAIAELDTLGEESYKDSTLIMQLLRDNLTLWT 3e73 A 2.8 BS02 GSH A 1 R4 L272 H274 K317 H323 R364 P366 D367 E374 R10 L278 H280 K323 H329 R370 P372 D373 E380 2.5.1.18 0004364,0004930,0005515,0005737,0005886,0005975,0007186,0008270,0016740,0017124,0031179,0043295,0046872,0050750,1990748 remove_due_to_license_issue O43813 19528316 502 SMDIEFMAQRAFPNPYADYNKSLAEGYFDAAGRLTPEFSQRLTNKIRELLQQMERGLKSADPRDGTGYTGWAGIAVLYLHLYDVFGDPAYLQLAHGYVKQSLNCLTKRSITFLCGDAGPLAVAAVLYHKMNNEKQAEDCITRLIHLNKIDPHAPNEMLYGRIGYIYALLFVNKNFGVEKIPQSHIQQICETILTSGENLARKRNFTAKSPLMYEWYQEYYVGAAHGLAGIYYYLMQPSLQVSQGKLHSLVKPSVDYVCQLKFPSGNYPPCIGDNRDLLVHWCHGAPGVIYMLIQAYKVFREEKYLCDAYQCADVIWQYGLLKKGYGLCHGSAGNAYAFLTLYNLTQDMKYLYRACKFAEWCLEYGEHGCRTPDTPFSLFEGMAGTIYFLADLLVPTKARFPAFEL 3e7b A 1.7 BS03 E7B A 1 R96 C127 I130 Y134 D197 W206 D220 R221 V223 H248 Y272 F276 R91 C122 I125 Y129 D192 W201 D215 R216 V218 H243 Y267 F271 D64 H66 D92 D95 R96 N124 H125 H173 R221 H248 D59 H61 D87 D90 R91 N119 H120 H168 R216 H243 3.1.3.16 0016787 ic50=0.16nM remove_due_to_license_issue P62136 18992256 500 SLNLDSIIGRLLEVQGSRPGKNVQLTENEIRGLCLKSREIFLSQPILLELEAPLKICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFLLRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDLQSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVQGWGENDRGVSFTFGAEVVAKFLHKHDLDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYCGEFDNAGAMMSVDETLMCSFQILKPA 3e7o A 2.14 BS01 35F A 1 I32 V40 A53 M108 E109 L110 M111 D112 A113 L168 I24 V32 A45 M100 E101 L102 M103 D104 A105 L160 D151 K153 N156 D169 T188 D143 K145 N148 D161 T180 2.7.11.24 0004672,0004707,0005524,0006468 ic50=120nM remove_due_to_license_issue P45984 18801372 1 QFYSVQVADSTFTVLKRYQQLKPIGSGAQGIVCAAFDTVLGINVAVKKLSRPFQNQTHAKRAYRELVLLKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIHMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTASTNFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGELVKGSVIFQGTDHIDQWNKVIEQLGTPSAEFMAALQPTVRNYVENRPAYPGIAFEELFPDWIFPSERDKIKTSQARDLLSKMLVIDPDKRISVDEALRHPYITVWYDPAEAEAPPPQIHAIEEWKELIYKEVM 3e81 A 1.629 BS03 SLB A 1 M20 E56 M20 E56 3.1.3.103 0016787,0016788,0046872 remove_due_to_license_issue Q8A712 18986982 171 MKEIKLILTDIDGVWTDGGMFYDQTGNEWKKFNTSDSAGIFWAHNKGIPVGILTGEKTEIVRRRAEKLKVDYLFQGVVDKLSAAEELCNELGINLEQVAYIGDDLNDAKLLKRVGIAGVPASAPFYIRRLSTIFLEKRGGEGVFREFVEKVLGINLEDFIAVIQ 3e81 A 1.629 BS04 SLB C 1 T34 S37 R64 K67 T34 S37 R64 K67 3.1.3.103 0016787,0016788,0046872 remove_due_to_license_issue Q8A712 18986982 171 MKEIKLILTDIDGVWTDGGMFYDQTGNEWKKFNTSDSAGIFWAHNKGIPVGILTGEKTEIVRRRAEKLKVDYLFQGVVDKLSAAEELCNELGINLEQVAYIGDDLNDAKLLKRVGIAGVPASAPFYIRRLSTIFLEKRGGEGVFREFVEKVLGINLEDFIAVIQ 3e81 B 1.629 BS01 SLB A 1 T34 R64 K67 T34 R64 K67 3.1.3.103 0016787,0016788,0046872 remove_due_to_license_issue Q8A712 18986982 171 MKEIKLILTDIDGVWTDGGMFYDQTGNEWKKFNTSDSAGIFWAHNKGIPVGILTGEKTEIVRRRAEKLKVDYLFQGVVDKLSAAEELCNELGINLEQVAYIGDDLNDAKLLKRVGIAGVPASAPFYIRRLSTIFLEKRGGEGVFREFVEKVLGINLEDFIAVIQ 3e81 B 1.629 BS04 SLB B 1 M20 E56 M20 E56 3.1.3.103 0016787,0016788,0046872 remove_due_to_license_issue Q8A712 18986982 171 MKEIKLILTDIDGVWTDGGMFYDQTGNEWKKFNTSDSAGIFWAHNKGIPVGILTGEKTEIVRRRAEKLKVDYLFQGVVDKLSAAEELCNELGINLEQVAYIGDDLNDAKLLKRVGIAGVPASAPFYIRRLSTIFLEKRGGEGVFREFVEKVLGINLEDFIAVIQ 3e85 A 1.95 BS01 BSU A 1 L22 V23 L55 H68 Y80 F142 L22 V23 L55 H68 Y80 F142 3.1.27.- 0004518,0004540,0004864,0005509,0005634,0005737,0005829,0006952,0009738,0010427,0038023,0044373,0046872,1904408 Kd=4.2uM remove_due_to_license_issue Q9LLQ2 19220853 158 GVFTFQDEYTSTIAPAKLYKALVTDADIIIPKAVETIQSVEIVEGNGGPGTIKKLTFIEGGESKYVLHKIEAIDEANLGYNYSIVGGVGLPDTIEKISFETKLVEGANGGSIGKVTIKIETKGDAQPNEEEGKAAKARGDAFFKAIESYLSAHP 3e85 A 1.95 BS02 BSU A 2 I37 F57 R138 I37 F57 R138 3.1.27.- 0004518,0004540,0004864,0005509,0005634,0005737,0005829,0006952,0009738,0010427,0038023,0044373,0046872,1904408 Kd=4.2uM remove_due_to_license_issue Q9LLQ2 19220853 159 GVFTFQDEYTSTIAPAKLYKALVTDADIIIPKAVETIQSVEIVEGNGGPGTIKKLTFIEGGESKYVLHKIEAIDEANLGYNYSIVGGVGLPDTIEKISFETKLVEGANGGSIGKVTIKIETKGDAQPNEEEGKAAKARGDAFFKAIESYLSAHP 3e85 A 1.95 BS03 BSU A 3 Y9 F99 V115 F143 Y9 F99 V115 F143 3.1.27.- 0004518,0004540,0004864,0005509,0005634,0005737,0005829,0006952,0009738,0010427,0038023,0044373,0046872,1904408 Kd=4.2uM remove_due_to_license_issue Q9LLQ2 19220853 160 GVFTFQDEYTSTIAPAKLYKALVTDADIIIPKAVETIQSVEIVEGNGGPGTIKKLTFIEGGESKYVLHKIEAIDEANLGYNYSIVGGVGLPDTIEKISFETKLVEGANGGSIGKVTIKIETKGDAQPNEEEGKAAKARGDAFFKAIESYLSAHP 3e85 A 1.95 BS04 BSU A 4 F5 G89 G132 A135 R138 F5 G89 G132 A135 R138 3.1.27.- 0004518,0004540,0004864,0005509,0005634,0005737,0005829,0006952,0009738,0010427,0038023,0044373,0046872,1904408 Kd=4.2uM remove_due_to_license_issue Q9LLQ2 19220853 161 GVFTFQDEYTSTIAPAKLYKALVTDADIIIPKAVETIQSVEIVEGNGGPGTIKKLTFIEGGESKYVLHKIEAIDEANLGYNYSIVGGVGLPDTIEKISFETKLVEGANGGSIGKVTIKIETKGDAQPNEEEGKAAKARGDAFFKAIESYLSAHP 3e8n A 2.5 BS03 VRA A 1 G79 K97 I99 V127 I141 D208 F209 V211 S212 L215 M219 G19 K37 I39 V67 I81 D148 F149 V151 S152 L155 M159 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T165 2.7.12.2 0004672,0005524,0006468 ic50=19nM remove_due_to_license_issue Q02750 19706763 1001 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3e8r A 1.9 BS02 615 A 1 T347 L348 G349 E398 L401 H405 E406 H409 H415 Y433 V434 P437 A439 T130 L131 G132 E177 L180 H184 E185 H188 H194 Y212 V213 P216 A218 3.4.24.86 0004222,0006508,0008237 remove_due_to_license_issue Ki=0.180000nM P78536 18835710 486 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3e90 A 2.45 BS01 NKK B 1 G83 F85 Q86 G33 F35 Q36 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004252,0044423 remove_due_to_license_issue P06935 19059417 195 DMWIERTADISWESDAEITGSSERVDVRLDDDGNFQLMNDPGAGGGG 3e90 B 2.45 BS01 NKK B 1 H51 D129 F130 G133 S135 G151 N152 G153 Y161 H49 D127 F128 G131 S133 G149 N150 G151 Y159 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0005524 remove_due_to_license_issue P06935 19059417 195 GGGVLWDTKEYKKGDTTTGVYRIMTRGLLGSYQAGAGVMVEGVFHTLWHTTKGAALMSGEGRLDPYWGSVKEDRLCYGGPWKLQHKWNGQDEVQMIVVEPGKNVKNVRTKPGVFKTPEGEIGAVTLDFPTGTSGSPIVDKNGDVIGLYGNGVIMPNGSYISAIVQGKRMDEPI 3e92 A 2.0 BS01 G6A A 1 Y35 E71 I84 T106 M109 G110 A111 L167 D168 F169 Y33 E69 I82 T104 M107 G108 A109 L165 D166 F167 D150 K152 N155 D168 T185 D148 K150 N153 D166 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=10nM remove_due_to_license_issue Ki=10.0nM Q16539 18789685 361 QERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3e93 A 2.0 BS01 19B A 1 A51 K53 E71 L74 T106 L108 M109 H148 L167 D168 F169 A48 K50 E68 L71 T103 L105 M106 H145 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T179 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=1.4nM remove_due_to_license_issue Ki=1.4nM Q16539 18789685 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3e9b A 2.15 BS03 S2C A 1 D124 H126 D128 N130 S137 H141 D183 E186 D232 D119 H121 D123 N125 S132 H136 D178 E181 D227 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0001889,0001938,0002250,0004053,0005615,0005737,0005741,0005829,0006525,0007565,0009410,0009635,0010042,0010043,0010269,0014075,0016787,0016813,0019547,0030145,0030324,0032496,0032964,0033189,0033197,0042130,0042802,0042832,0043025,0043200,0043434,0045087,0046007,0046686,0046872,0048545,0048678,0051597,0060056,0060135,0060336,0070301,0070965,0071222,0071353,0071377,0071549,0071560,1905541,2000552 Ki=4500nM remove_due_to_license_issue P07824 19093830 502 KPIEIIGAPFSKGQPRGGVEKGPAALRKAGLVEKLKETEYNVRDHGDLAFVDVPNDSPFQIVKNPRSVGKANEQLAAVVAETQKNGTISVVLGGDHSMAIGSISGHARVHPDLCVIWVDAHTDINTPLTASSGNLHGQPVAFLLKELKGKFPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYIIKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPVFTPATGTPVVGGLSYREGLYITEEIYKTGLLSGLDIMEVNPTLGKTPEEVTRTVNTAVALTLSCFGTKREGNHK 3e9h A 2.1 BS02 KAA A 1 E231 R253 H261 N262 F265 M267 E269 Y271 E411 H412 N414 F416 E418 G463 G467 R470 E223 R245 H253 N254 F257 M259 E261 Y263 E403 H404 N406 F408 E410 G455 G459 R462 R253 E255 R260 H261 E411 N414 R470 R245 E247 R252 H253 E403 N406 R462 6.1.1.6 0000049,0000166,0000287,0003676,0004812,0004824,0005524,0005737,0005829,0006412,0006418,0006430,0016740,0046872 remove_due_to_license_issue Q9RHV9 19174549 2002 ELNDQLRVRREKLKKIEELGVDPFGKRFERTHKAEELFELYGDLSKEELEEQQIEVAVAGRIMTKRGMGKAGFAHIQDVTGQIQIYVRQDDVGEQQYELFKISDLGDIVGVRGTMFKTKVGELSIKVSSYEFLTKALRPLPEKDIEQRYRQRYLDLIMNPESKKTFITRSLIIQSMRRYLDSHGYLEVETPMMHAVAGGAAARPFITHHNALDMTLYMRIAIELHLKRLIVGGLEKVYEIGRVFRNEGISTRHNPEFTMLELYEAYADFRDIMKLTENLIAHIATEVLGTTKIQYGEHLVDLTPEWRRLHMVDAIKEYVGVDFWRQMSDEEARELAKEHGVEVAPHMTFGHIVNEFFEQKVEDKLIQPTFIYGHPVEISPLAKKNPDDPRFTDRFELFIVGREHANAFTELNDPIDQRQRFEEQLKEREQGNDEAHEMDEDFLEALEYGMPPTGGLGIGVDRLVMLLTNSPSIRDVLLFPQMRH 3e9i A 2.2 BS01 XAH A 1 G207 E231 R253 H261 N262 F265 M267 E269 Y271 E411 H412 N414 F416 E418 G467 G199 E223 R245 H253 N254 F257 M259 E261 Y263 E403 H404 N406 F408 E410 G459 R253 E255 R260 H261 E411 N414 R470 R245 E247 R252 H253 E403 N406 R462 6.1.1.6 0000049,0000166,0000287,0003676,0004812,0004824,0005524,0005737,0005829,0006412,0006418,0006430,0016740,0046872 remove_due_to_license_issue Q9RHV9 19174549 1001 ELNDQLRVRREKLKKIEELGVDPFGKRFERTHKAEELFELYGDLSKEELEEQQIEVAVAGRIMTKRGMGKAGFAHIQDVTGQIQIYVRQDDVGEQQYELFKISDLGDIVGVRGTMFKTKVGELSIKVSSYEFLTKALRPLPEKDIEQRYRQRYLDLIMNPESKKTFITRSLIIQSMRRYLDSHGYLEVETPMMHAVAGGAAARPFITHHNALDMTLYMRIAIELHLKRLIVGGLEKVYEIGRVFRNEGISTRHNPEFTMLELYEAYADFRDIMKLTENLIAHIATEVLGTTKIQYGEHLVDLTPEWRRLHMVDAIKEYVGVDFWRQMSDEEARELAKEHGVEVAPHMTFGHIVNEFFEQKVEDKLIQPTFIYGHPVEISPLAKKNPDDPRFTDRFELFIVGREHANAFTELNDPIDQRQRFEEQLKEREQGNDEAHEMDEDFLEALEYGMPPTGGLGIGVDRLVMLLTNSPSIRDVLLFPQMRH 3eax A 1.9 BS01 LZP A 1 Y46 D48 A217 G220 R221 Q262 Q266 Y45 D47 A216 G219 R220 Q261 Q265 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=12uM remove_due_to_license_issue P18031 19012396 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG 3eb1 A 2.4 BS01 LZQ A 1 Y46 D48 A217 G220 Q262 Q266 Y45 D47 A216 G219 Q261 Q265 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=16.3uM remove_due_to_license_issue IC50=20000nM P18031 19012396 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGD 3ebh A 1.65 BS02 BES A 1 E319 V459 G460 A461 E463 H496 E497 H500 E519 Y575 Y580 E124 V264 G265 A266 E268 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=478.2nM remove_due_to_license_issue Ki=190nM, IC50=284nM O96935 19196988 1085 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 3ebi A 2.0 BS02 BEY A 1 Q317 E319 V459 G460 A461 M462 E463 R489 V493 H496 E497 E519 Y575 Y580 M1034 Q122 E124 V264 G265 A266 M267 E268 R294 V298 H301 E302 E324 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=79nM remove_due_to_license_issue O96935 19196988 1085 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 3ebl A 1.9 BS01 GA4 A 1 F27 G122 S123 I133 Y134 S198 R251 Y254 V326 G327 F13 G92 S93 I103 Y104 S168 R221 Y224 V296 G297 3.-.-.- 0005634,0005737,0009739,0009740,0009939,0010325,0010331,0016787,0048444 Kd=0.5uM remove_due_to_license_issue Q6L545 19037316 401 VVPLHTWVLISNFKLSYNILRRADGTFERDLGEYLDRRVPANARPLEGVSSFDHIIDQSVGLEVRIYRAALEFLTDAPAAEPFPVIIFFHGGSFVHSSASSTIYDSLCRRFVKLSKGVVVSVNYRRAPEHRYPCAYDDGWTALKWVMSQPFMRSGGDAQARVFLSGDSSGGNIAHHVAVRAADEGVKVCGNILLNAMFGGTERTESERRLDGKYFVTLQDRDWYWKAYLPEDADRDHPACNPFGPNGRRLGGLPFAKSLIIVSGLDLTCDRQLAYADALREDGHHVKVVQCENATVGFYLLPNTVHYHEVMEEISDFLNANLY 3ebo A 1.9 BS01 57D A 1 F285 E382 A610 G612 Y613 F268 E356 A584 G586 Y587 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 23279842 940 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ebp A 2.0 BS01 CPB A 1 N284 F285 L380 E382 A610 G612 Y613 N267 F268 L354 E356 A584 G586 Y587 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue IC50=1200nM P00489 23279842 940 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ecn A 2.1 BS01 IBM A 1 M670 Y748 Q778 F781 F785 M189 Y267 Q297 F300 F304 3.1.4.53 0004114,0007165,0008081 ic50=698uM remove_due_to_license_issue IC50=700000nM O60658 18983167 3 DDVPPRIARAMENEEYWDFDIFELEAATHNRPLIYLGLKMFARFGICEFLHCSESTLRSWLQIIEANYHSSNPYHNSTHSADVLHATAYFLSKERIKETLDPIDEVAALIAATIHDVDHPGRTNSFLCNAGSELAILYNDTAVLESHHAALAFQLTTGDDKCNIFKNMERNDYRTLRQGIIDMVLATEMTKHFEHVNKFVNSINKPLATLEENGETDKNQEVINTMLRTPENRTLIKRMLIKCADVSNPCRPLQYCIEWAARISEEYFSQTDEEKQQGLPVVMPVFDRNTCSIPKSQISFIDYFITDMFDAWDAFVDLPDLMQHLDNNFKYWKGLDEM 3ed0 A 2.3 BS01 EMO A 1 F59 R110 I111 P112 F52 R103 I104 P105 H58 I64 G67 V68 E72 H51 I57 G60 V61 E65 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 Kd=0.45uM remove_due_to_license_issue Q5G940 19433000 163 LQSQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3ed0 B 2.3 BS01 EMO A 1 I98 Y100 I89 Y91 H58 I64 G67 V68 E72 H49 I55 G58 V59 E63 4.2.1.59 0005737,0006633,0009245,0016020,0016829,0016836,0019171 remove_due_to_license_issue Q5G940 19433000 163 SQFFIEHILQILPHRYPMLLVDRITELQANQKIVAYKNITFNEDVFNGHFPNKPIFPGVLIVEGMAQSGGFLAFTSLWGFDPEIAKTKIVYFMTIDKVKFRIPVTPGDRLEYHLEVLKHKGMIWQVGGTAQVDGKVVAEAELKAMIAERE 3ee2 A 1.91 BS02 NZO A 1 R14 M99 W104 Y152 R13 M98 W103 Y151 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50~65uM remove_due_to_license_issue O60760 19939518 201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAIANWIKRRPQTKL 3eeb A 2.1 BS01 IHP A 1 T28 R29 K54 H55 R85 S136 S169 R171 R182 K183 K195 K200 T28 R29 K54 H55 R85 S136 S169 R171 R182 K183 K195 K200 2.3.1.-,3.4.22.-,6.3.2.- Kd=1.3uM remove_due_to_license_issue Q9KS12 18845756 210 ADGKILHNQNVNSWGPITVTPTTDGGETRFDGQIIVQMENDPVVAKAAANLAGKHAESSVVVQLDSDGNYRVVYGDPSKLDGKLRWQLVGHGRDHSETNNTRLSGYSADELAVKLAKFQQSFNQAENINNKPDHISIVGCSLVSDDKQKGFGHQFINAMDANGLRVDVSVRSSELAVDEAGRKHTKDANGDWVQKAENNKVSLSW 3efj A 2.6 BS01 MT3 A 1 I1084 F1089 V1092 A1108 K1110 F1124 G1128 M1131 L1157 Y1159 M1160 G1163 M1211 F1223 I31 F36 V39 A55 K57 F71 G75 M78 L104 Y106 M107 G110 M158 F170 D1204 A1206 R1208 N1209 D1222 D151 A153 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=39nM, Ki=39nM P08581 18763753 1 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 3efj B 2.6 BS01 MT3 B 1 I1084 F1089 V1092 A1108 F1124 G1128 M1131 L1140 L1157 Y1159 M1160 G1163 M1211 I31 F36 V39 A55 F71 G75 M78 L87 L104 Y106 M107 G110 M158 D1204 A1206 R1208 N1209 D1222 D151 A153 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=39nM, Ki=39nM P08581 18763753 2 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 3efk A 2.2 BS01 MT4 A 1 I1084 F1089 A1108 F1124 E1127 G1128 M1131 L1140 L1142 L1157 Y1159 M1160 G1163 M1211 D1222 F1223 I31 F36 A55 F71 E74 G75 M78 L87 L89 L104 Y106 M107 G110 M158 D169 F170 D1204 A1206 R1208 N1209 D1222 D151 A153 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 Ki=14nM remove_due_to_license_issue Ki=14nM, IC50=14nM P08581 18763753 1 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 3efk B 2.2 BS01 MT4 B 1 I1084 F1089 A1108 F1124 E1127 G1128 M1131 L1140 L1142 L1157 Y1159 M1160 G1163 M1211 A1221 D1222 F1223 I31 F36 A55 F67 E70 G71 M74 L83 L85 L100 Y102 M103 G106 M154 A164 D165 F166 D1204 A1206 R1208 N1209 D1222 D147 A149 R151 N152 D165 2.7.10.1 0004672,0004713,0005524,0006468 Ki=14nM remove_due_to_license_issue Ki=14nM, IC50=14nM P08581 18763753 2 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 3efr A 2.55 BS01 BTN A 1 S13 T14 Q15 Q34 G37 R38 G40 L46 Y53 F54 G106 L108 G119 I120 G121 S13 T14 Q15 Q34 G37 R38 G40 L46 Y53 F54 G106 L108 G119 I120 G121 G40 K103 R231 G40 K103 R231 6.3.4.15 0004077,0005524,0005737,0016874,0036211 remove_due_to_license_issue O66837 19385043 1001 MFKNLIWLKEVDSTQERLKEWNVSYGTALVADRQTKGRGGLGRKWLSQEGGLYFSFLLNPKEFENLLQLPLVLGLSVSEALEEITEIPFSLKWPNDVYFQEKKVSGVLRELSKDKLIVGIGINVNQREIPEEIKDRATTLYEITGKDWDRKEVLLKVLKRISENLKKFKEKSFKEFKGKIESKMLYLGEEVKLLGEGKITGKLVGLSEKGGALILTEEGIKEILSGEFSLRRS 3efs A 2.3 BS01 ATP A 1 R40 R43 W45 L46 K92 K103 N123 S229 L230 R231 R39 R42 W44 L45 K91 K102 N122 S228 L229 R230 R40 K103 R231 R39 K102 R230 6.3.4.15 0004077,0005524,0005737,0016874,0036211 Kd=7.2uM remove_due_to_license_issue O66837 19385043 1001 FKNLIWLKEVDSTQERLKEWNVSYGTALVADRQTKGRGRLGRKWLSQEGGLYFSFLLNPKEFENLLQLPLVLGLSVSEALEEITEIPFSLKWPNDVYFQEKKVSGVLRELSKDKLIVGIGINVNQREIPEEIKDRATTLYEITGKDWDRKEVLLKVLKRISENLKKFKEKSFKEFKGKIESKMLYLGEEVKLLGEGKITGKLVGLSEKGGALILTEEGIKEILSGEFSLRRS 3efs A 2.3 BS03 ATP B 1 K192 S233 K191 S232 R40 K103 R231 R39 K102 R230 6.3.4.15 0004077,0005524,0005737,0016874,0036211 Kd=7.2uM remove_due_to_license_issue O66837 19385043 1001 FKNLIWLKEVDSTQERLKEWNVSYGTALVADRQTKGRGRLGRKWLSQEGGLYFSFLLNPKEFENLLQLPLVLGLSVSEALEEITEIPFSLKWPNDVYFQEKKVSGVLRELSKDKLIVGIGINVNQREIPEEIKDRATTLYEITGKDWDRKEVLLKVLKRISENLKKFKEKSFKEFKGKIESKMLYLGEEVKLLGEGKITGKLVGLSEKGGALILTEEGIKEILSGEFSLRRS 3eft A 1.85 BS02 3BS A 1 H94 V121 F131 L198 T199 T200 H91 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=12nM remove_due_to_license_issue P00918 19778001 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3efw A 2.29 BS01 AK8 A 1 F144 V147 K162 V174 L178 Y212 A213 L263 A273 F275 F19 V22 K37 V49 L53 Y87 A88 L138 A148 F150 D256 K258 E260 N261 D274 D131 K133 E135 N136 D149 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 19062275 404 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFLDYLPPEMIEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3egk H 2.2 BS03 M18 H 1 H57 Y60A W60D L99 A190 C191 V213 W215 G216 G226 F227 H43 Y47 W50 L96 A191 C192 V216 W218 G219 G229 F230 3.4.21.5 0004252,0005509,0006508,0007596 Ki=22uM remove_due_to_license_issue P00734 17955562 601 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3egt A 2.0 BS03 722 A 1 Y99 D103 M106 R112 T168 Q172 K212 D255 K269 Y90 D94 M97 R103 T159 Q163 K203 D246 K260 M1 E20 E22 D28 C43 K47 Y48 V54 I55 D56 V57 A58 L62 H98 D103 D107 R112 R160 T167 D175 D188 Y211 K212 F251 D255 D256 V270 A277 A293 E297 S304 E308 E318 M1 E20 E22 D28 C43 K47 Y48 V54 I55 D56 V57 A58 L62 H89 D94 D98 R103 R151 T158 D166 D179 Y202 K203 F242 D246 D247 V261 A268 A284 E288 S295 E299 E309 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Ki=1.26nM remove_due_to_license_issue Q86C09 19309137 3001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSLDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 3egt B 2.0 BS01 722 A 1 N131 L134 N123 L126 M1 E20 E22 D28 C43 K47 Y48 V54 I55 D56 V57 A58 L62 H98 D103 D107 R112 R160 T167 D175 D188 Y211 K212 F251 D255 D256 V270 A277 A293 E297 S304 E308 E318 M1 E20 E22 D28 C43 K47 Y48 V54 I55 D56 V57 A58 L62 H90 D95 D99 R104 R152 T159 D167 D180 Y203 K204 F243 D247 D248 V262 A269 A285 E289 S296 E300 E310 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Ki=1.26nM remove_due_to_license_issue Q86C09 19309137 3001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSLDDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 3egt B 2.0 BS04 722 B 1 Y99 E102 D103 M106 D107 R112 Q172 K212 D255 K269 Y91 E94 D95 M98 D99 R104 Q164 K204 D247 K261 M1 E20 E22 D28 C43 K47 Y48 V54 I55 D56 V57 A58 L62 H98 D103 D107 R112 R160 T167 D175 D188 Y211 K212 F251 D255 D256 V270 A277 A293 E297 S304 E308 E318 M1 E20 E22 D28 C43 K47 Y48 V54 I55 D56 V57 A58 L62 H90 D95 D99 R104 R152 T159 D167 D180 Y203 K204 F243 D247 D248 V262 A269 A285 E289 S296 E300 E310 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Ki=1.26nM remove_due_to_license_issue Q86C09 19309137 4001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSLDDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 3egz A 2.2 BS01 rna B 0 Y208 N210 N211 E214 K217 S243 L244 K245 M246 R247 Q249 F251 K275 R278 Q280 K283 D285 S286 D287 Y8 N10 N11 E14 K17 S43 L44 K45 M46 R47 Q49 F51 K75 R78 Q80 K83 D85 S86 D87 ? 0003676,0003723 remove_due_to_license_issue P09012 18940672 1 ~ 65 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAK 3eh8 A 2.7 BS01 dna B 0 K24 Y27 I55 R59 R61 R70 R72 K74 Y111 A147 E148 C150 S152 Y154 D168 A170 Q171 R172 K200 K202 K24 Y27 I55 R59 R61 R70 R72 K74 Y111 A147 E148 C150 S152 Y154 D168 A170 Q171 R172 K200 K202 3.1.-.- 0004519 remove_due_to_license_issue P03880 19103658 1 ~ 31 GSDLTYAYLVGLYEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSKILPIFEKYPMFSNKQYDYLRFRNALLSGIIYLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYKLWLKQLRKISRYSEKIKIPSNY 3eh8 A 2.7 BS02 dna C 0 G15 D16 Y18 S20 T22 K23 E35 S37 I64 M66 K94 L156 Y162 T189 K190 Y192 R243 G15 D16 Y18 S20 T22 K23 E35 S37 I64 M66 K94 L156 Y162 T189 K190 Y192 R243 3.1.-.- 0004519 remove_due_to_license_issue P03880 19103658 1 ~ 31 GSDLTYAYLVGLYEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSKILPIFEKYPMFSNKQYDYLRFRNALLSGIIYLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYKLWLKQLRKISRYSEKIKIPSNY 3eh8 D 2.7 BS01 dna E 0 K24 Y27 I55 R59 R61 R70 R72 D73 K74 I110 Y111 E148 C150 S152 Y154 K158 D168 Q171 R172 K200 K202 Q230 K24 Y27 I55 R59 R61 R70 R72 D73 K74 I110 Y111 E148 C150 S152 Y154 K158 D168 Q171 R172 K200 K202 Q230 3.1.-.- 0004519 remove_due_to_license_issue P03880 19103658 1 ~ 31 GSDLTYAYLVGLYEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSKILPIFEKYPMFSNKQYDYLRFRNALLSGIIYLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYKLWLKQLRKISRYSEKIKIPSNY 3eh8 D 2.7 BS02 dna F 0 G15 D16 G17 Y18 S20 T22 K23 E35 L36 S37 I64 M66 R70 K94 E148 L156 Y162 T189 K190 Y192 V206 R243 G15 D16 G17 Y18 S20 T22 K23 E35 L36 S37 I64 M66 R70 K94 E148 L156 Y162 T189 K190 Y192 V206 R243 3.1.-.- 0004519 remove_due_to_license_issue P03880 19103658 1 ~ 31 GSDLTYAYLVGLYEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSKILPIFEKYPMFSNKQYDYLRFRNALLSGIIYLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYKLWLKQLRKISRYSEKIKIPSNY 3eh8 G 2.7 BS01 dna H 0 K24 Y27 I55 R59 R61 R70 R72 K74 Y111 E148 C150 S152 Y154 D168 A170 Q171 R172 K200 K202 Q230 K24 Y27 I55 R59 R61 R70 R72 K74 Y111 E148 C150 S152 Y154 D168 A170 Q171 R172 K200 K202 Q230 3.1.-.- 0004519 remove_due_to_license_issue P03880 19103658 1 ~ 31 GSDLTYAYLVGLYEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSKILPIFEKYPMFSNKQYDYLRFRNALLSGIIYLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYKLWLKQLRKISRYSEKIKIPSNY 3eh8 G 2.7 BS02 dna I 0 G15 D16 G17 Y18 S20 T22 K23 K24 E35 L36 S37 I64 M66 K94 Y162 K190 Y192 V206 R243 G15 D16 G17 Y18 S20 T22 K23 K24 E35 L36 S37 I64 M66 K94 Y162 K190 Y192 V206 R243 3.1.-.- 0004519 remove_due_to_license_issue P03880 19103658 1 ~ 31 GSDLTYAYLVGLYEGDGYFSITKKGKYLTYELGIELSIKDVQLIYKIKKILGIGIVSFRKRNEIEMVALRIRDKNHLKSKILPIFEKYPMFSNKQYDYLRFRNALLSGIIYLEDLPDYTRSDEPLNSIESIINTSYFSAWLVGFIEAEGCFSVYKLNKDDDYLIASFDIAQRDGDILISAIRKYLSFTTKVYLDKTNCSKLKVTSVRSVENIIKFLQNAPVKLLGNKKLQYKLWLKQLRKISRYSEKIKIPSNY 3ehw A 1.8 BS01 DUP A 1 R153 G157 F158 G159 S160 T161 R130 G134 F135 G136 S137 T138 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw A 1.8 BS02 DUP B 1 A98 G99 V100 I101 D102 Y105 G110 A75 G76 V77 I78 D79 Y82 G87 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw A 1.8 BS03 DUP C 1 R85 S86 G87 R62 S63 G64 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw B 1.8 BS01 DUP A 1 R85 S86 G87 Q131 R61 S62 G63 Q107 A46 R85 G87 I94 D102 A22 R61 G63 I70 D78 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 QLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw B 1.8 BS02 DUP B 1 R153 G157 F158 G159 S160 T161 R129 G133 F134 G135 S136 T137 A46 R85 G87 I94 D102 A22 R61 G63 I70 D78 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 QLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw B 1.8 BS03 DUP C 1 A98 G99 V100 I101 D102 Y105 G110 A74 G75 V76 I77 D78 Y81 G86 A46 R85 G87 I94 D102 A22 R61 G63 I70 D78 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 QLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw C 1.8 BS01 DUP A 1 A98 G99 V100 I101 D102 Y105 G110 A74 G75 V76 I77 D78 Y81 G86 A46 R85 G87 I94 D102 A22 R61 G63 I70 D78 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 QLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw C 1.8 BS02 DUP B 1 R85 S86 G87 R61 S62 G63 A46 R85 G87 I94 D102 A22 R61 G63 I70 D78 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 QLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehw C 1.8 BS03 DUP C 1 R153 G157 F158 G159 S160 T161 R129 G133 F134 G135 S136 T137 A46 R85 G87 I94 D102 A22 R61 G63 I70 D78 3.6.1.23 0000287,0004170,0006226,0046081 remove_due_to_license_issue P33316 777 QLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALDDTERGSGGFGSTGKN 3ehx A 1.9 BS06 BDL A 1 I180 L181 A182 H218 E219 H222 H228 V235 F237 P238 T239 Y240 I75 L76 A77 H113 E114 H117 H123 V130 F132 P133 T134 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=25nM remove_due_to_license_issue P39900 19275207 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3ehy A 1.9 BS06 TBL A 1 I180 L181 A182 L214 H218 E219 H222 H228 Y240 I75 L76 A77 L109 H113 E114 H117 H123 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=1.4uM remove_due_to_license_issue P39900 19275207 1 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3eid A 3.15 BS01 PO5 A 1 I10 E12 A31 K33 F80 L83 L134 I10 E12 A31 K33 F77 L80 L131 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T160 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=450nM P24941 18835709 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 3eig A 1.7 BS01 MTX A 1 I7 V8 L22 E30 R31 R32 F34 E35 N64 L67 R70 V115 I7 V8 L22 E30 R31 R32 F34 E35 N64 L67 R70 V115 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=21nM remove_due_to_license_issue IC50=22nM, Kd=0.194984nM, Ki=4420nM, EC50=13.3nM P00374 19478082 200 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNERRYFERMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3eio A 2.0 BS01 AJH A 1 E205 E206 F357 Y585 S630 Y662 Y666 V711 E167 E168 F319 Y547 S592 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=223nM remove_due_to_license_issue IC50=223nM P27487 18996694 1 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 3ej1 A 3.22 BS01 5BP A 1 I10 A31 K33 F80 L83 H84 L134 D145 I10 A31 K33 F77 L80 H81 L131 D142 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=120nM P24941 18835709 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ej5 X 2.5 BS01 EJ5 X 1 Y80 V81 G121 Y123 I172 E177 R180 Y76 V77 G117 Y119 I168 E173 R176 V81 V77 3.2.2.22 0017148,0030598 ic50=0.27mM remove_due_to_license_issue P02879 19138659 300 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLAISFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAP 3ejp A 1.32 BS02 HN2 A 1 H90 D92 W95 D204 F206 R228 D341 H471 D472 Y727 R876 H61 D63 W66 D175 F177 R199 D312 H442 D443 Y698 R847 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=2.8nM remove_due_to_license_issue Q24451 20209559 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ejq A 1.45 BS02 HN3 A 1 H90 D92 W95 D204 F206 R228 D341 H471 D472 Y727 E875 R876 G877 H61 D63 W66 D175 F177 R199 D312 H442 D443 Y698 E846 R847 G848 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=2.7nM remove_due_to_license_issue Q24451 20209559 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ejr A 1.27 BS02 HN4 A 1 H90 D92 W95 D204 F206 R228 D341 H471 D472 Y727 E875 R876 G877 H61 D63 W66 D175 F177 R199 D312 H442 D443 Y698 E846 R847 G848 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 Ki=2.7nM remove_due_to_license_issue Q24451 20209559 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ejs A 1.35 BS02 HN5 A 1 H90 D92 W95 D204 F206 R228 D341 H471 D472 Y727 E875 R876 G877 H61 D63 W66 D175 F177 R199 D312 H442 D443 Y698 E846 R847 G848 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=250nM remove_due_to_license_issue Q24451 20209559 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ejt A 1.35 BS02 HN6 A 1 H90 D92 W95 D204 F206 R228 Y269 D341 H471 D472 Y727 R876 G877 H61 D63 W66 D175 F177 R199 Y240 D312 H442 D443 Y698 R847 G848 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=44nM remove_due_to_license_issue Q24451 20209559 1050 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3eju A 1.32 BS02 HN7 A 1 H90 D92 W95 D204 F206 R228 D341 H471 D472 Y727 E875 R876 G877 H61 D63 W66 D175 F177 R199 D312 H442 D443 Y698 E846 R847 G848 H90 D92 D204 D341 H471 H61 D63 D175 D312 H442 3.2.1.114 0000139,0003824,0004559,0004572,0005783,0005794,0005795,0005975,0006013,0006486,0006491,0015923,0016020,0016063,0016787,0016798,0030246,0035010,0046872 ic50=250nM remove_due_to_license_issue Q24451 20209559 1049 QCQDVVQDVPNVDVQMLELYDRMSFKDIDGGVWKQGWNIKYDPLKYNAHHKLKVFVVPHSHNDPGWIQTFEEYYQHDTKHILSNALRHLHDNPEMKFIWAEISYFARFYHDLGENKKLQMKSIVKNGQLEFVTGGWVMPDEANSHWRNVLLQLTEGQTWLKQFMNVTPTASWAIDPFGHSPTMPYILQKSGFKNMLIQRTHYSVKKELAQQRQLEFLWRQIWDNKGDTALFTHMMPFYSYDIPHTCGPDPKVCCQFDFKRMGSFGLSCPWKVPPRTISDQNVAARSDLLVDQWKKKAELYRTNVLLIPLGDDFRFKQNTEWDVQRVNYERLFEHINSQAHFNVQAQFGTLQEYFDAVHQAERAGQAEFPTLSGDFFTYADRSDNYWSGYYTSRPYHKRMDRVLMHYVRAAEMLSAWHSWDGMARIEERLEQARRELSLFQHHDGITGTAKTHVVVDYEQRMQEALKACQMVMQQSVYRLLTKPSIYSPDFSFSYFTLDDSRWPGSGVEDSRTTIILGEDILPSKHVVMHNTLPHWREQLVDFYVSSPFVSVTDLANNPVEAQVSPVWSWHHDTLTKTIHPQGSTTKYRIIFKARVPPMGLATYVLTISDSKPEHTSYASNLLLRKNPTSLPLGQYPEDVKFGDPREISLRVGNGPTLAFSEQGLLKSIQLTQDSPHVPVHFKFLKYGVRSHGDRSGAYLFLPNGPASPVELGQPVVLVTKGKLESSVSVGLPSVVHQTIMRGGAPEIRNLVDIGSLDNTEIVMRLETHIDSGDIFYTDLNGLQFIKRRRLDKLPLQANYYPIPSGMFIEDANTRLTLLTGQPLGGSSLASGELEIMQDRRLASDDERGLGQGVLDNKPVLHIYRLVLEKVNNCVRPSKLHPAGYLTSAAHKASQSLLDPLDKFIFAENEWIGAQGQFGGDHPSAREDLDVSVMRRLTKSSAKTQRVGYVLHRTNLMQCGTPEEHTQKLDVCHLLPNVARCERTTLTFLQNLEHLDGMVAPEVCPMETAAYVSSHSS 3ekn A 2.2 BS01 GS3 A 1 L1002 G1003 Q1004 V1010 A1028 V1060 M1076 M1079 G1082 M1139 L19 G20 Q21 V27 A45 V77 M93 M96 G99 M156 N1132 R1136 N1137 D1150 N149 R153 N154 D167 2.7.10.1 0004672,0004714,0005524,0006468,0007169,0016020 ic50=2nM remove_due_to_license_issue P06213 19071018 1 YVPDEWEVSREKITLLRELGQGSFGMVYEGNARDIIKGEAETRVAVKTVNESASLRERIEFLNEASVMKGFTCHHVVRLLGVVSKGQPTLVVMELMAHGDLKSYLRSLRPEAENNPGRPPPTLQEMIQMAAEIADGMAYLNAKKFVHRNLAARNCMVAHDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMAPESLKDGVFTTSSDMWSFGVVLWEITSLAEQPYQGLSNEQVLKFVMDGGYLDQPDNCPERVTDLMRMCWQFNPNMRPTFLEIVNLLKDDLHPSFPEVSFFHSEENK 3eko A 1.55 BS01 PYU A 1 N51 A55 K58 D93 I96 M98 T184 N42 A46 K49 D84 I87 M89 T175 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.2uM remove_due_to_license_issue P07900 18929486 901 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKEL 3ekp A 2.15 BS01 478 B 1 D25 G27 A28 G49 I50 D25 G27 A28 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 200 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3ekp B 2.15 BS01 478 B 1 D25 G27 A28 D30 V48 I50 P81 D25 G27 A28 D30 V48 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=1.3nM remove_due_to_license_issue P03369 22712830 200 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3ekq A 2.2 BS01 ROC A 1 D25 G27 A28 D29 D30 V48 G49 I50 I84 D25 G27 A28 D29 D30 V48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=176nM remove_due_to_license_issue P03369 22712830 100 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPTNIIGRNLLTQIGCTLNF 3ekq B 2.2 BS01 ROC A 1 R8 L23 D25 G27 V48 P81 I84 R8 L23 D25 G27 V48 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 100 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPTNIIGRNLLTQIGCTLNF 3ekr A 2.0 BS01 PY9 A 1 N51 A55 K58 D93 I96 G97 M98 T184 N42 A46 K49 D84 I87 G88 M89 T175 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.03uM remove_due_to_license_issue P07900 18929486 901 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKEL 3eks A 1.8 BS03 CY9 A 1 Y133 A135 I136 Y143 Y169 A170 P172 M355 F375 Y132 A134 I135 Y142 Y168 A169 P171 M354 F374 3.6.4.- 0000281,0005515,0005524,0005737,0005856,0006338,0007291,0016787,0030723,0031011,0032507,0035060,0035148 remove_due_to_license_issue P10987 18938176 903 DEEVAALVVDNGSGMCKAGFAGDDAPRAVFPSIVGRPRHQGVMVGMGQKDSYVGDEAQSKRGILTLKYPIEHGIVTNWDDMEKIWHHTFYNELRVAPEEHPVLLTEAPLNPKANREKMTQIMFETFNTPAMYVAIQAVLSLYASGRTTGIVLDSGDGVSHTVPIYEGYALPHAILRLDLAGRDLTDYLMKILTERGYSFTTTEEREIVRDIKEKLCYVALDFEQEMATAASSSSLEKSYELKDGQVITIGNERFRCPEALFQPSFLGMEACGIHETTYNSIMKCDVDIRKDLYANTVLSGGTTMYPGIADRMQKEITALAPSTMKIKIIAPPERKYSVWIGGSILASLSTFQQMWISKQEYDESGPSIVHRKCF 3ekt A 1.97 BS01 017 B 1 D25 G27 A28 D29 D30 V48 G49 I50 D25 G27 A28 D29 D30 V48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 200 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3ekt B 1.97 BS01 017 B 1 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.026nM remove_due_to_license_issue P03369 22712830 200 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3ekv A 1.75 BS01 478 A 1 D25 G27 A28 D30 G48 G49 I50 D25 G27 A28 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.39nM remove_due_to_license_issue P03369 22712830 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ekv B 1.75 BS01 478 A 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ekw A 1.6 BS01 DR7 B 1 D25 G27 D29 V48 G49 I50 D25 G27 D29 V48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 100 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3ekw B 1.6 BS01 DR7 B 1 R8 L23 D25 G27 A28 D29 V48 G49 I50 P81 R8 L23 D25 G27 A28 D29 V48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=10.9nM remove_due_to_license_issue P03369 22712830 100 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3ekx A 1.97 BS01 1UN B 1 D25 G27 D30 G49 I84 D25 G27 D30 G49 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ekx B 1.97 BS01 1UN B 1 R8 D25 G27 G49 I50 P81 R8 D25 G27 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.39nM remove_due_to_license_issue P03369 22712830 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3eky A 1.8 BS01 DR7 A 1 R8 D25 G27 D29 G48 G49 I50 P81 V82 I84 R8 D25 G27 D29 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.23nM remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3eky B 1.8 BS01 DR7 A 1 D25 G27 D29 G48 G49 I50 P81 V82 I84 D25 G27 D29 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3el0 A 2.0 BS01 1UN A 1 D25 G27 A28 D29 D30 P81 I84 D25 G27 A28 D29 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=34.1nM remove_due_to_license_issue P03369 22712830 201 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3el0 B 2.0 BS01 1UN A 1 D25 I47 V48 I50 A82 D25 I47 V48 I50 A82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 201 PQITLWKRPIVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIVGIGGFVKVRQYDQIPIEICGHKAIGTVLVGPTPANIIGRNLLTQIGCTLNF 3el1 A 1.7 BS01 DR7 A 1 D25 G27 D29 G48 G49 P81 I84 D25 G27 D29 G48 G49 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.23nM remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3el1 B 1.7 BS01 DR7 A 1 R8 D25 G27 A28 D29 G49 I50 P81 V82 R8 D25 G27 A28 D29 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3el4 A 2.0 BS01 ROC A 1 D25 G27 A28 D29 D30 G48 G49 I50 T82 D25 G27 A28 D29 D30 G48 G49 I50 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=67.4nM remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3el4 B 2.0 BS01 ROC A 1 R8 D25 G27 P81 R8 D25 G27 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3el5 A 1.6 BS01 1UN B 1 D25 G27 D30 G48 G49 I50 P81 T82 D25 G27 D30 G48 G49 I50 P81 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3el5 B 1.6 BS01 1UN B 1 D25 G27 D29 D30 I50 P81 D25 G27 D29 D30 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=18.9nM remove_due_to_license_issue P03369 22712830 201 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3el7 A 2.8 BS01 PD3 A 1 A293 K295 E310 M314 Y340 M341 L393 V402 A403 D404 A35 K37 E51 M55 Y79 M80 L132 V141 A142 D143 D386 R388 A390 N391 D404 D125 R127 A129 N130 D143 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 18940662 601 KDAWEIPRESLRLEVKLGQGGEVWMGTWNGTTRVAIKTLKPTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3el8 A 2.3 BS01 PD5 A 1 V281 A293 E310 M314 Y340 M341 L393 A403 D404 V24 A36 E53 M57 Y83 M84 L136 A146 D147 D386 R388 A390 N391 D404 F424 D129 R131 A133 N134 D147 F154 2.7.10.2 0004672,0004713,0005524,0006468 ic50=25nM remove_due_to_license_issue P00523 18940662 601 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3el9 A 1.6 BS01 DR7 A 1 D25 A28 D29 G48 G49 I50 P81 T82 D25 A28 D29 G48 G49 I50 P81 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=4nM remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3el9 B 1.6 BS01 DR7 A 1 D25 G27 A28 D29 G48 G49 I50 P81 D25 G27 A28 D29 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 22712830 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3elc A 2.5 BS02 F01 A 1 A100 K104 M105 L106 A131 T132 T133 A101 K105 M106 L107 A132 T133 T134 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=2.02mM remove_due_to_license_issue Kd=2020000nM P62617 19320487 901 EMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 3elc A 2.5 BS03 F01 B 1 D56 G58 D57 G59 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=2.02mM remove_due_to_license_issue Kd=2020000nM P62617 19320487 902 EMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 3elc C 2.5 BS02 F01 C 1 A100 K104 M105 L106 A131 T132 T133 A101 K105 M106 L107 A132 T133 T134 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=2.02mM remove_due_to_license_issue Kd=2020000nM P62617 19320487 903 EMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 3elj A 1.8 BS01 GS7 A 1 I32 G33 S34 G35 V40 A53 M108 E109 M111 D112 A113 N114 Q117 L168 I26 G27 S28 G29 V34 A47 M102 E103 M105 D106 A107 N108 Q111 L162 D151 K153 N156 D169 T188 D145 K147 N150 D163 T176 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P45983 19071018 365 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLSFMMTPYVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPEREHTIEEWKELIYKEVMDLE 3elm A 1.9 BS07 24F A 1 Y176 L184 A186 H187 A188 V219 H222 E223 H226 H232 L239 F241 I243 Y244 Y73 L81 A83 H84 A85 V116 H119 E120 H123 H129 L136 F138 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.19nM remove_due_to_license_issue IC50=0.5nM, Ki=0.19nM P45452 19422229 400 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYFMLPDDDVQGIQSLYGPGDED 3elm B 1.9 BS06 24F B 1 L184 L185 A186 H187 F189 H222 E223 H226 H232 L239 F241 I243 Y244 L81 L82 A83 H84 F86 H119 E120 H123 H129 L136 F138 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.19nM remove_due_to_license_issue IC50=0.5nM, Ki=0.19nM P45452 19422229 400 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 3emg A 2.6 BS01 685 A 1 L377 F382 V385 A400 K402 M448 M450 A451 G454 L501 D512 L13 F18 V21 A35 K37 M76 M78 A79 G82 L129 D140 D494 A496 R498 N499 D512 K533 D122 A124 R126 N127 D140 K157 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=6.0nM, Ki=9nM P43405 18938080 685 LDRKLLTLEDKELGSGNFGTVKKGYYQMKVVKTVAVKILKLKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYY 3eml A 2.6 BS01 ZMA A 1 L85 F168 M177 W246 L249 N253 M270 L83 F159 M168 W384 L387 N391 M408 E1011 D1020 E209 D218 ?,3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P29274 18832607 401 IMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYRSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLRQ 3ens B 2.3 BS01 ENS B 1 T98 Y99 E147 D189 A190 Q192 V213 W215 G216 G218 C220 G226 T84 Y85 E135 D179 A180 Q182 V203 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=8.9nM remove_due_to_license_issue P00742 18998662 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTRGLP 3eoc A 3.2 BS01 T2A A 1 I10 G11 V18 F80 F82 L83 H84 Q85 D86 K89 L134 I10 G11 V18 F77 F79 L80 H81 Q82 D83 K86 L131 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=230nM P24941 18929484 501 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3eor A 2.9 BS02 CFV A 1 A100 P103 K104 M105 L106 A131 A101 P104 K105 M106 L107 A132 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 remove_due_to_license_issue P62617 19320487 901 EMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 3eos A 1.78 BS02 PK2 A 1 V45 N70 D102 Y106 Q107 D156 C158 G229 G230 A232 M260 G261 D280 V35 N60 D92 Y96 Q97 D134 C136 G207 G208 A210 M238 G239 D258 D102 D280 C318 C320 C323 H349 D92 D258 C291 C293 C296 H322 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=4nM remove_due_to_license_issue P28720 19894214 400 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLKQSEEGVTFHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 3eou A 1.93 BS02 PK3 A 1 D102 Y106 D156 C158 G229 G230 L231 A232 M260 G261 D280 D92 Y96 D129 C131 G202 G203 L204 A205 M233 G234 D253 D102 D280 C318 C320 C323 H349 D92 D253 C285 C287 C290 H316 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=97nM remove_due_to_license_issue P28720 19894214 500 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMQSEEGVTFLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 3eq7 A 2.89 BS01 X99 A 1 F173 C255 F476 S554 W595 R643 F170 C252 F473 S551 W592 R640 Y473 S554 D641 H680 Y470 S551 D638 H677 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 19006380 711 FQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 3eq8 A 2.73 BS01 X98 A 1 F173 M235 G254 C255 F476 S554 W595 R643 V644 F172 M234 G253 C254 F475 S553 W594 R642 V643 Y473 S554 D641 H680 Y472 S553 D640 H679 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 19006380 711 LSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 3eq9 A 2.47 BS01 X97 A 1 F173 M235 R252 G254 C255 F476 S554 W595 R643 V644 F171 M233 R250 G252 C253 F474 S552 W593 R641 V642 Y473 S554 D641 H680 Y471 S552 D639 H678 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 ic50=41nM remove_due_to_license_issue P23687 19006380 711 SFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 3eqb A 2.62 BS03 LUG A 1 N78 K97 V127 I141 D208 F209 V211 S212 L215 N18 K37 V67 I81 D148 F149 V151 S152 L155 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T163 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue Q02750 18951019 1 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3eql C 2.7 BS01 MXP D 1 E1034 W1038 S1084 L1088 E1034 W1038 S1084 L1088 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue Q8RQE9 18946472 1527 MEIKRFGRIREVIPLPPLTEIQVESYRRALQADVPPEKRENVGIQAAFRETFPIEEEDKGKGGLVLDFLEYRLGEPPFPQDECREKDLTYQAPLYARLQLIHKDTGLIKEDEVFLGHIPLMTEDGSFIINGADRVIVSQIHRSPGVYFTPDPARPGRYIASIIPLPKRGPWIDLEVEPNGVVSMKVNKRKFPLVLLLRVLGYDQETLARELGAYGELVQGLMDESVFAMRPEEALIRLFTLLRPGDPPKRDKAVAYVYGLIADPRRYDLGEAGRYKAEEKLGIRLSGRTLARFEDGEFKDEVFLPTLRYLFALTAGVPGHEVDDIDHLGNRRIRTVGELMTDQFRVGLARLARGVRERMLMGSEDSLTPAKLVNSRPLEAAIREFFSRSQLSQFKDETNPLSSLRHKRRISALGPGGLTRERAGFDVRDVHRTHYGRICPVETPEGANIGLITSLAAYARVDELGFIRTPYRRVVGGVVTDEVVYMTATEEDRYTIAQANTPLEGNRIAAERVVARRKGEPVIVSPEEVEFMDVSPKQVFSVNTNLIPFLEHDDANRALMGSNMQTQAVPLIRAQAPVVMTGLEERVVRDSLAALYAEEDGEVAKVDGNRIVVRYEDGRLVEYPLRRFYRSNQGTALDQRPRVVVGQRVRKGDLLADGPASENGFLALGQNVLVAIMPFDGYNFEDAIVISEELLKRDFYTSIHIERYEIEARDTKLGPERITRDIPHLSEAALRDLDEEGVVRIGAEVKPGDILVGRTSFKGESEPTPEERLLRSIFGEKARDVKDTSLRVPPGEGGIVVRTVRLRRGDPGVELKPGVREVVRVYVAQKRKLQVGDKLANRHGNKGVVAKILPVEDMPHLPDGTPVDVILNPLGVPSRMNLGQILETHLGLAGYFLGQRYISPIFDGAKEPEIKELLAQAFEVYFGKRKGEGFGVDKREVEVLRRAEKLGLVTPGKTPEEQLKELFLQGKVVLYDGRTGEPIEGPIVVGQMFIMKLYHMVEDKMHARSTGPYSLITQQPLGGKAQFGGQRFGEMEVWALEAYGAAHTLQEMLTLKSDDIEGRNAAYEAIIKGEDVPEPSVPESFRVLVKELQALALDVQTLDEKDNPVDIFEGLASKR 3eql D 2.7 BS03 MXP D 1 K610 Q611 L619 G620 K1463 I1467 K426 Q427 L435 G436 K1279 I1283 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0006351,0006360,0006366,0006383,0008270,0016779,0034062,0042793,0046872 remove_due_to_license_issue Q8RQE8 18946472 1527 KKEVRKVRIALASPEKIRSWSYGEVEKPETINYRTLKPERDGLFDERIFGPIKDYECACGKYKRQRFEGKVCERCGVEVTKSIVRRYRMGHIELATPAAHIWFVKDVPSKIGTLLDLSATELEQVLYFSKYIVLDPKGAILNGVPVEKRQLLTDEEYRELRYGKQETYPLPPGVDALVKDGEEVVKGQELAPGVVSRLDGVALYRFASILVVKARVYPFEDDVEVSTGDRVAPGDVLADGGKVKSDVYGRVEVDLVRNVVRVVESYDIDARMGAEAIQQLLKELDLEALEKELLEEMKHPSRARRAKARKRLEVVRAFLDSGNRPEWMILEAVPVLPPDLRPMVQVDGGRFATSDLNDLYRRLINRNNRLKKLLAQGAPEIIIRNEKRMLQEAVDALLDNGRRGAPVTNPGSDRPLRSLTDILSGKQGRFRQNLLGKRVDYSGRSVIVVGPQLKLHQCGLPKRMALELFKPFLLKKMEEKGIAPNVKAARRMLERQRDIKDEVWDALEEVIHGKVVLLNRAPTLHRLGIQAFQPVLVEGQSIQLHPLVCEAFNADFDGDQMAVHVPLSSFAQAEARIQMLSAHNLLSPASGEPLAKPSRDIILGLYYITQVRKEKKGAGLEFATPEEALAAHERGEVALNAPIKVAGRETSVGRLKYVFANPDEALLAVAHGIVDLQDVVTVRYMGKRLETSPGRILFARIVAEAVEDEKVAWELIQLDVPQEKNSLKDLVYQAFLRLGMEKTARLLDALKYYGFTFSTTSGITIGIDDAVIPEEKKQYLEEADRKLLQIEQAYEMGFLTDRERYDQILQLWTETTEKVTQAVFKNFEENYPFNPLYVMAQSGARGNPQQIRQLCGLRGLMQKPSGETFEVPVRSSFREGLTVLEYFISSHGARKGGADTALRTADSGYLTRKLVDVTHEIVVREADCGTTNYISVPLFQPDEVTRSLRLRKRADIEAGLYGRVLAREVEVLGVRLEEGRYLSMDDVHLLIKAAEAGEIQEVPVRSPLTCQTRYGVCQKCYGYDLSMARPVSIGEAVGIVAAQSIGEPGTQLTMRTFHTGGVAGAADITQGLPRVIELFEARRPKAKAVISEIDGVVRIEETEEKLSVFVESEGFSKEYKLPKEARLLVKDGDYVEAGQPLTRGAIDPHQLLEAKGPEAVERYLVEEIQKVYRAQGVKLHDKHIEIVVRQMMKYVEVTDPGDSRLLEGQVLEKWDVEALNERLIAEGKTPVAWKPLLMGVTKSALSTKSWLSAASFQNTTHVLTEAAIAGKKDELIGLKENVILGRLIPAGTGSDFVRFTQVVDQKTLKAIEEARKEAVEA 3eqr A 2.0 BS01 T74 A 1 L132 V140 A156 K158 E177 I190 T205 L207 A208 G211 L259 G269 L16 V24 A40 K42 E55 I68 T83 L85 A86 G89 L137 G147 D252 A254 R256 N257 D270 V292 D130 A132 R134 N135 D148 V170 2.7.10.2,2.7.11.1 0004672,0004713,0005524,0006468 Ki=0.002uM remove_due_to_license_issue IC50=20nM, Ki=2nM Q07912 18993068 1 LTCLIGEKDLRLLEKLGDGSFGVVRRGEWDAPSGKTVSVAVKCLKPEAMDDFIREVNAMHSLDHRNLIRLYGVVLTPPMKMVTELAPLGSLLDRLRKHQGHFLLGTLSRYAVQVAEGMGYLESKRFIHRDLAARNLLLATRDLVKIGDFGLMRALPQNDDHYVMQEHRKVPFAWCAPESLKTRTFSHASDTWMFGVTLWEMFTYGQEPWIGLNGSQILHKIDKEGERLPRPEDCPQDIYNVMVQCWAHKPEDRPTFVALRDFLLEAQPTD 3eqt A 2.0 BS01 rna C 0 T575 H576 I597 L621 K634 K651 W652 S653 T30 H31 I52 L76 K89 K106 W107 S108 3.6.4.13 remove_due_to_license_issue Q96C10 19278996 1 ~ 8 QFPVEHVQLLCINCMVAVGHGSDLRKVEGTHHVNVNPNFSNYYNVSRDPVVINKVFKDWKPGGVISCRNCGEVWGLQMIYKSVKLPVLKVRSMLLETPQGRIQAKKWSRVPFSVPDFDFLQHCAENL 3eqt A 2.0 BS02 rna D 0 E573 H576 K599 F601 W604 R636 E28 H31 K54 F56 W59 R91 3.6.4.13 remove_due_to_license_issue Q96C10 19278996 1 ~ 8 QFPVEHVQLLCINCMVAVGHGSDLRKVEGTHHVNVNPNFSNYYNVSRDPVVINKVFKDWKPGGVISCRNCGEVWGLQMIYKSVKLPVLKVRSMLLETPQGRIQAKKWSRVPFSVPDFDFLQHCAENL 3eqt B 2.0 BS01 rna C 0 E573 H576 K599 F601 W604 E30 H33 K56 F58 W61 3.6.4.13 remove_due_to_license_issue Q96C10 19278996 1 ~ 8 RQQFPVEHVQLLCINCMVAVGHGSDLRKVEGTHHVNVNPNFSNYYNVSRDPVVINKVFKDWKPGGVISCRNCGEVWGLQMIYKSVKLPVLKVRSMLLETPQGRIQAKKWSRVPFSVPDFDFLQHCAENLSDLSLDLEHHHHH 3eqt B 2.0 BS02 rna D 0 T575 H576 V595 I597 G620 L621 K634 V635 K651 W652 S653 T32 H33 V52 I54 G77 L78 K91 V92 K108 W109 S110 3.6.4.13 remove_due_to_license_issue Q96C10 19278996 1 ~ 8 RQQFPVEHVQLLCINCMVAVGHGSDLRKVEGTHHVNVNPNFSNYYNVSRDPVVINKVFKDWKPGGVISCRNCGEVWGLQMIYKSVKLPVLKVRSMLLETPQGRIQAKKWSRVPFSVPDFDFLQHCAENLSDLSLDLEHHHHH 3er3 E 2.0 BS01 0EL E 1 D30 D32 G34 Y75 G76 D114 D215 G217 T218 T219 Y222 D33 D35 G37 Y79 G80 D119 D219 G221 T222 T223 Y226 3.4.23.22 0004190,0006508 Ki=81nM remove_due_to_license_issue P11838 6381096 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 3erd A 2.03 BS02 DES A 1 M343 E353 L387 M421 H524 L525 M39 E49 L83 M117 H220 L221 ? remove_due_to_license_issue Ki=0.128000nM, IC50=0.330000nM, EC50=0.110000nM P03372 9875847 600 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRL 3erk A 2.1 BS01 SB4 A 1 V37 A50 K52 I101 Q103 D104 M106 D109 L154 V32 A45 K47 I96 Q98 D99 M101 D104 L149 D147 K149 S151 N152 D165 T188 D142 K144 S146 N147 D160 T183 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 ic50=18uM remove_due_to_license_issue IC50=18000nM P63086 9753691 800 AAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 3ern A 2.1 BS02 CAR A 1 A100 K104 M105 L106 A131 T132 T133 A101 K105 M106 L107 A132 T133 T134 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=18.91mM remove_due_to_license_issue Kd=18910000nM P62617 19320487 900 EMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 3ern C 2.1 BS02 CAR C 1 K104 M105 L106 A131 T132 T133 K99 M100 L101 A126 T127 T128 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 Kd=18.91mM remove_due_to_license_issue Kd=18910000nM P62617 19320487 900 EMRIGHGFDVHAFGGEGPIIIGGVRIPYESDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIK 3ert A 1.9 BS01 OHT A 1 M343 L346 A350 E353 W383 M421 G521 L525 H550 A551 M38 L41 A45 E48 W78 M116 G216 L220 H245 A246 ? remove_due_to_license_issue IC50=0.790000nM, EC50=10.3nM, Ki=5.7nM P03372 9875847 600 LALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAHRLHA 3esj A 2.7 BS02 CC7 A 1 A100 K104 M105 L106 A131 T133 A103 K107 M108 L109 A134 T136 4.6.1.12 0005515,0006744,0008270,0008299,0008685,0016114,0016829,0019288,0030145,0042802,0046872 remove_due_to_license_issue P62617 19320487 901 MLEMRIGHGFDVHAFGGEGPIIIGGVRIPYEKGLLAHSDGDVALHALTDALLGAAALGDIGKLFPDTDPAFKGADSRELLREAWRRIQAKGYTLGNVDVTIIAQAPKMLPHIPQMRVFIAEDLGCHMDDVNVKATTTEKLGFTGRGEGIACEAVALLIKATK 3ess A 1.191 BS01 18N A 1 H460 G461 Y493 A501 Y504 E581 H35 G36 Y59 A67 Y70 E147 E581 E147 2.4.2.36 0047286 ic50=411nM remove_due_to_license_issue Q5EK40 19793133 1 MAVITPQGVTNWTYQELEATHQALTREGYVFVGYHGTNHVAAQTIVNRIAPVEKWGGLYVATHAEVAHGYARIKEGTGEYGLPTRAERDARGVMLRVYIPRASLERFYRTNTPLENAEEHITQVIGHSLPLRNEAFTGPESAGGEDETVIGWDMAIHAVAIPSTIPGNAYEELAIDEEAVAKEQSISTKPPYKERKDEL 3et7 A 2.7 BS01 349 A 1 L431 E503 L504 Y505 G508 E509 L556 L13 E85 L86 Y87 G90 E91 L138 D549 A551 R553 N554 D567 L587 D131 A133 R135 N136 D149 L157 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q14289 18951788 999 GIAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSRTRLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIAM 3eta A 2.6 BS01 351 A 1 L1002 A1028 K1030 E1047 M1051 E1077 M1079 G1082 F1128 M1139 G1149 D1150 L13 A39 K41 E58 M62 E88 M90 G93 F139 M150 G160 D161 D1132 A1134 R1136 N1137 D1150 E1159 L1171 P1172 D143 A145 R147 N148 D161 E170 L181 P182 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue P06213 19394223 2001 EVSREKITLLRELGQGSFGMVYEGNARDIIKGEAETRVAVKTVNESASLRERIEFLNEASVMKGFTCHHVVRLLGVVSKGQPTLVVMELMAHGDLKSYLRSLRPEAENNPGRPPPTLQEMIQMAAEIADGMAYLNAKKFVHRDLAARNCMVAHDFTVKIGDFGMTRDIYETDYYRKGKGLLPVRWMAPESLKDGVFTTSSDMWSFGVVLWEITSLAEQPYQGLSNEQVLKFVMDGGYLDQPDNCPERVTDLMRMCWQFNPKMRPTFLEIVNLLKDDLHPSFPEVSFFHSEENK 3eu5 A 2.8 BS01 GBO B 1 K164 Y166 K110 Y112 K164 K110 2.5.1.58,2.5.1.59 0004659,0004660,0004661,0004662,0004663,0005515,0005737,0005875,0005953,0005965,0007167,0007323,0008017,0008270,0008284,0008318,0014070,0018342,0018343,0018344,0030971,0034097,0035022,0036094,0042277,0043014,0043066,0045787,0051770,0051771,0060090,0090044,1901363,1904395 remove_due_to_license_issue Q04631 19219049 429 FLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSEKFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVWHFRRVLLRSLQKDLQEEMNYIIAIIEEQPKNYQVWHHRRVLVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFRLWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRAVLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPNLLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDILNKALELCEILAKEKDTIRKEYWRYIGRSLQSKHSR 3eu5 B 2.8 BS02 GBO B 1 W102 H248 G250 Y251 R291 K294 Y300 W303 W78 H224 G226 Y227 R267 K270 Y276 W279 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H224 R267 K270 D273 C275 Y276 D328 D335 H338 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 19219049 429 PLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGFEE 3evc A 1.6 BS02 GTP A 1 K13 L16 N17 F24 S151 S152 S215 K8 L11 N12 F19 S146 S147 S210 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P03314 19101564 902 KTLGEVWKRELNLLDKRQFELYKRTDIVEVDRDTARRHLAEGKVDTGVAVSRGTAKLRWFHERGYVKLEGRVIDLGCGRGGWCYYAAAQKEVSGVKGFTLGRDGHEKPMNVQSLGWNIITFKDKTDIHRLEPVKCDTLLCDIGESSSSSVTEGERTVRVLDTVEKWLACGVDNFCVKVLAPYMPDVLEKLELLQRRFGGTVIRNPLSRNSTHEMYYVSGARSNVTFTVNQTSRLLMRRMRRPTGKVTLEADVILPIGTRSV 3evd A 1.5 BS01 GTP A 1 K13 N17 L19 F24 K28 S150 S151 S215 K8 N12 L14 F19 K23 S145 S146 S210 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P03314 19101564 901 KTLGEVWKRELNLLDKRQFELYKRTDIVEVDRDTARRHLAEGKVDTGVAVSRGTAKLRWFHERGYVKLEGRVIDLGCGRGGWCYYAAAQKEVSGVKGFTLGRDGHEKPMNVQSLGWNIITFKDKTDIHRLEPVKCDTLLCDIGESSSSSVTEGERTVRVLDTVEKWLACGVDNFCVKVLAPYMPDVLEKLELLQRRFGGTVIRNPLSRNSTHEMYYVSGARSNVTFTVNQTSRLLMRRMRRPTGKVTLEADVILPIGTRSV 3evd A 1.5 BS02 GTP A 2 R37 R41 S56 R57 R84 R32 R36 S51 R52 R79 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P03314 19101564 902 KTLGEVWKRELNLLDKRQFELYKRTDIVEVDRDTARRHLAEGKVDTGVAVSRGTAKLRWFHERGYVKLEGRVIDLGCGRGGWCYYAAAQKEVSGVKGFTLGRDGHEKPMNVQSLGWNIITFKDKTDIHRLEPVKCDTLLCDIGESSSSSVTEGERTVRVLDTVEKWLACGVDNFCVKVLAPYMPDVLEKLELLQRRFGGTVIRNPLSRNSTHEMYYVSGARSNVTFTVNQTSRLLMRRMRRPTGKVTLEADVILPIGTRSV 3evf A 1.45 BS01 GTA A 1 K13 L16 N17 L19 F24 K28 S150 S151 S152 S215 K8 L11 N12 L14 F19 K23 S145 S146 S147 S210 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P03314 19101564 902 KTLGEVWKRELNLLDKRQFELYKRTDIVEVDRDTARRHLAEGKVDTGVAVSRGTAKLRWFHERGYVKLEGRVIDLGCGRGGWCYYAAAQKEVSGVKGFTLGRDGHEKPMNVQSLGWNIITFKDKTDIHRLEPVKCDTLLCDIGESSSSSVTEGERTVRVLDTVEKWLACGVDNFCVKVLAPYMPDVLEKLELLQRRFGGTVIRNPLSRNSTHEMYYVSGARSNVTFTVNQTSRLLMRRMRRPTGKVTLEADVILPIGTRSV 3evf A 1.45 BS02 GTA A 2 R37 R41 S56 R57 R84 R32 R36 S51 R52 R79 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P03314 19101564 903 KTLGEVWKRELNLLDKRQFELYKRTDIVEVDRDTARRHLAEGKVDTGVAVSRGTAKLRWFHERGYVKLEGRVIDLGCGRGGWCYYAAAQKEVSGVKGFTLGRDGHEKPMNVQSLGWNIITFKDKTDIHRLEPVKCDTLLCDIGESSSSSVTEGERTVRVLDTVEKWLACGVDNFCVKVLAPYMPDVLEKLELLQRRFGGTVIRNPLSRNSTHEMYYVSGARSNVTFTVNQTSRLLMRRMRRPTGKVTLEADVILPIGTRSV 3ew2 A 2.3 BS01 BTN A 1 S25 Y41 N43 G49 W72 S81 T83 W85 W102 D119 S11 Y27 N29 G35 W58 S67 T69 W71 W88 D105 ? 0005576,0009374 remove_due_to_license_issue Q8KKW2 19111749 400 ASSSWQNQSGSTMIIQVDSFGNVSGQYVNRAQGTGCQNSPYPLTGRVNGTFIAFSVGWNNSTENCNSATGWTGYAQVNGNNTEIVTSWNLAYEGGSGPAIEQGQDTFQYVPTTE 3ew2 B 2.3 BS01 BTN B 1 S225 Y241 N243 T248 G249 W272 T283 W285 W302 D319 S18 Y34 N36 T41 G42 W65 T76 W78 W95 D112 ? 0005576,0009374 remove_due_to_license_issue Q8KKW2 19111749 500 DFSSIASASSSWQNQSGSTMIIQVDSFGNVSGQYVNRAQGTGCQNSPYPLTGRVNGTFIAFSVGWNNSTENCNSATGWTGYAQVNGNNTEIVTSWNLAYEGGSGPAIEQGQDTFQYVPTTE 3ewc A 2.11 BS02 MCF A 1 H44 L85 F88 D172 T173 G174 H175 G201 H226 E229 H253 D310 D311 H38 L79 F82 D166 T167 G168 H169 G195 H220 E223 H247 D304 D305 H42 H44 H226 E229 H253 D310 H36 H38 H220 E223 H247 D304 3.5.4.31,3.5.4.4 0004000,0005829,0006154,0006166,0009168,0009897,0016787,0019239,0043103,0046103,0046872,0046936,0060169,0090614 Ki=20nM remove_due_to_license_issue A5KE01 19728741 373 PIDFLKKEELKNIDLSQMSKKERYKIWKRIPKCELHCHLDLCFSADFFVSCIRKYNLQPNLSDEEVLDYYLFAKGGKSLGEFVEKAIKVADIFHDYEVIEDLAKHAVFNKYKEGVVLMEFRYSPTFVAFKYNLDIELIHQAIVKGIKEVVELLDHKIHVALMCIGDTGHEAANIKASADFCLKHKADFVGFDHGGHEVDLKEYKEIFDYVRESGVPLSVHAGEDVTLPNLNTLYSAIQVLKVERIGHGIRVAESQELIDMVKEKNILLEVCPISNVLLKNAKSMDTHPIRQLYDAGVKVSVNSDDPGMFLTNINDDYEELYTHLNFTLEDFMKMNEWALEKSFMDSNIKDKIKNLYF 3ewh A 1.6 BS01 K11 A 1 L840 V848 A866 K868 E885 T916 F918 C919 L1019 L1035 C1045 D1046 F1047 L26 V34 A49 K51 E68 T99 F101 C102 L152 L168 C178 D179 F180 D1028 A1030 R1032 N1033 D1046 D161 A163 R165 N166 D179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=69nM remove_due_to_license_issue IC50=70nM P35968 19062275 1 EHAERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDTCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDPDYVRLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHH 3ewu A 1.6 BS01 UEP A 1 S257 D259 N312 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 N90 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ewu A 1.6 BS02 UEP B 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ewu B 1.6 BS01 UEP A 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ewu B 1.6 BS02 UEP B 1 S257 D259 K281 N312 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 K59 N90 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ewz A 1.4 BS01 CNU B 1 S257 D259 K281 H283 I368 M371 S372 I401 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 I146 M149 S150 I179 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLGV 3ewz A 1.4 BS02 CNU B 2 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLGV 3ewz B 1.4 BS01 CNU B 1 D317 T321 D95 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=79uM remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLGV 3ewz B 1.4 BS02 CNU B 2 S257 D259 K281 H283 D312 I368 M371 S372 I401 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 D90 I146 M149 S150 I179 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=79uM remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLGV 3ex2 A 1.55 BS01 6CN A 1 S257 D259 K281 H283 D312 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 D90 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50~200uM remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex2 A 1.55 BS02 6CN B 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50~200uM remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex2 B 1.55 BS01 6CN A 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50~200uM remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex2 B 1.55 BS02 6CN B 1 S257 D259 K281 H283 D312 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 D90 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50~200uM remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex3 A 1.45 BS01 U5P A 1 S257 D259 H283 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex3 A 1.45 BS02 U5P B 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex3 B 1.45 BS01 U5P A 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex3 B 1.45 BS02 U5P B 1 S257 D259 K281 H283 K314 M371 S372 P417 Q430 Y432 G450 R451 S35 D37 K59 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 481 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex6 A 1.3 BS01 U5P B 1 D317 I318 T321 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3ex6 B 1.3 BS01 U5P B 1 H283 K314 M371 S372 P417 Q430 Y432 G450 R451 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue P11172 19472232 482 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFENRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3exf A 2.998 BS02 TPP A 1 Y89 R90 V138 G166 D167 G168 A169 N196 Y198 G199 M200 H263 Y90 R91 V139 G167 D168 G169 A170 N197 Y199 G200 M201 H264 Q51 G136 R259 H263 S264 Y272 Q52 G137 R260 H264 S265 Y273 1.2.4.1 0004738,0004739,0005515,0005634,0005730,0005739,0005759,0006006,0006086,0006090,0006099,0016491,0016624,0034604,0043231,0045254,0046872,1902494 remove_due_to_license_issue P08559 19081061 1003 MFANDATFEIKKCDLHRLEEGPPVTTVLTREDGLKYYRMMQTVRRMELKADQLYKQKIIRGFCHLCDGQEACCVGLEAGINPTDHLITAYRAHGFTFTRGLSVREILAELTGRKGGCAKGKGGSMHMYAKNFYGGNGIVGAQVPLGAGIALACKYNGKDEVCLTLYGDGAANQGQIFEAYNMAALWKLPCIFICENNRYGMGTAVERAAASTDYYKRGDFIPGLRVDGMDILCVREATRFAAAYCRSGKGPILMELQTYRYHGHSMSDPGVAYRTREEIQEVRSKSDPIMLLKDRMVNSNLASVEELKEIDVEVRKEIEDAAQFATADPEPPLEELGYHIYSSDPPFEVRGANQWIKFKSVS 3exf B 2.998 BS01 TPP C 1 E28 I57 E59 F85 Q88 E28 I57 E59 F85 Q88 E59 H128 E59 H128 1.2.4.1 0003824,0004739,0005515,0005634,0005654,0005739,0005759,0006006,0006086,0006099,0016491,0034604,0045254,0046872 remove_due_to_license_issue P11177 19081061 1006 LQVTVRDAINQGMDEELERDEKVFLLGEEVAQYDGAYKVSRGLWKKYGDKRIIDTPISEMGFAGIAVGAAMAGLRPICEFMTFNFSMQAIDQVINSAAKTYYMSGGLQPVPIVFRGPNGASAGVAAQHSQCFAAWYGHCPGLKVVSPWNSEDAKGLIKSAIRDNNPVVVLENELMYGVPFEFPPEAQSKDFLIPIGKAKIERQGTHITVVSHSRPVGHCLEAAAVLSKEGVECEVINMRTIRPMDMETIEASVMKTNHLVTVEGGWPQFGVGAEICARIMEGPAFNFLDAPAVRVTGADVPMPYAKILEDNSIPQVKDIIFAIKKTLNI 3exf D 2.998 BS01 TPP A 1 E28 I57 E59 F85 Q88 E28 I57 E59 F85 Q88 E59 H128 E59 H128 1.2.4.1 0003824,0004739,0005515,0005634,0005654,0005739,0005759,0006006,0006086,0006099,0016491,0034604,0045254,0046872 remove_due_to_license_issue P11177 19081061 1003 LQVTVRDAINQGMDEELERDEKVFLLGEEVAQYDGAYKVSRGLWKKYGDKRIIDTPISEMGFAGIAVGAAMAGLRPICEFMTFNFSMQAIDQVINSAAKTYYMSGGLQPVPIVFRGPNGASAGVAAQHSQCFAAWYGHCPGLKVVSPWNSEDAKGLIKSAIRDNNPVVVLENELMYGVPFEFPPEAQSKDFLIPIGKAKIERQGTHITVVSHSRPVGHCLEAAAVLSKEGVECEVINMRTIRPMDMETIEASVMKTNHLVTVEGGWPQFGVGAEICARIMEGPAFNFLDAPAVRVTGADVPMPYAKILEDNSIPQVKDIIFAIKKTLNI 3exh A 2.444 BS02 TPP A 1 Y89 R90 V138 G166 D167 G168 N196 Y198 G199 R259 Y90 R91 V139 G167 D168 G169 N197 Y199 G200 R257 Q51 G136 R259 H263 S264 Y272 Q52 G137 R257 H261 S262 Y270 1.2.4.1 0004738,0004739,0005515,0005634,0005730,0005739,0005759,0006006,0006086,0006090,0006099,0016491,0016624,0034604,0043231,0045254,0046872,1902494 remove_due_to_license_issue P08559 19081061 1502 MFANDATFEIKKCDLHRLEEGPPVTTVLTREDGLKYYRMMQTVRRMELKADQLYKQKIIRGFCHLCDGQEACCVGLEAGINPTDHLITAYRAHGFTFTRGLSVREILAELTGRKGGCAKGKGGSMHMYAKNFYGGNGIVGAQVPLGAGIALACKYNGKDEVCLTLYGDGAANQGQIFEAYNMAALWKLPCIFICENNRYGMGERAAASTDYYKRGDFIPGLRVDGMDILCVREATRFAAAYCRSGKGPILMELQTYRYHGHSMSDPGVAYRTREEIQEVRSKSDPIMLLKDRMVNSNLASVEELKEIDVEVRKEIEDAAQFATADPEPPLEELGYHIYSSDPPFEVRGANQWIKFKSVS 3exh B 2.444 BS01 TPP C 1 I57 E59 F85 Q88 I57 E59 F85 Q88 E59 H128 E59 H128 1.2.4.1 0003824,0004739,0005515,0005634,0005654,0005739,0005759,0006006,0006086,0006099,0016491,0034604,0045254,0046872 remove_due_to_license_issue P11177 19081061 1502 LQVTVRDAINQGMDEELERDEKVFLLGEEVAQYDGAYKVSRGLWKKYGDKRIIDTPISEMGFAGIAVGAAMAGLRPICEFMTFNFSMQAIDQVINSAAKTYYMSGGLQPVPIVFRGPNGASAGVAAQHSQCFAAWYGHCPGLKVVSPWNSEDAKGLIKSAIRDNNPVVVLENELMYGVPFEFPPEAQSKDFLIPIGKAKIERQGTHITVVSHSRPVGHCLEAAAVLSKEGVECEVINMRTIRPMDMETIEASVMKTNHLVTVEGGWPQFGVGAEICARIMEGPAFNFLDAPAVRVTGADVPMPYAKILEDNSIPQVKDIIFAIKKTLNI 3exh D 2.444 BS01 TPP A 1 E28 I57 E59 F85 Q88 E28 I57 E59 F85 Q88 E59 H128 E59 H128 1.2.4.1 0003824,0004739,0005515,0005634,0005654,0005739,0005759,0006006,0006086,0006099,0016491,0034604,0045254,0046872 remove_due_to_license_issue P11177 19081061 1502 LQVTVRDAINQGMDEELERDEKVFLLGEEVAQYDGAYKVSRGLWKKYGDKRIIDTPISEMGFAGIAVGAAMAGLRPICEFMTFNFSMQAIDQVINSAAKTYYMSGGLQPVPIVFRGPNGASAGVAAQHSQCFAAWYGHCPGLKVVSPWNSEDAKGLIKSAIRDNNPVVVLENELMYGVPFEFPPEAQSKDFLIPIGKAKIERQGTHITVVSHSRPVGHCLEAAAVLSKEGVECEVINMRTIRPMDMETIEASVMKTNHLVTVEGGWPQFGVGAEICARIMEGPAFNFLDAPAVRVTGADVPMPYAKILEDNSIPQVKDIIFAIKKTLNI 3exo A 2.1 BS01 5MS A 1 Q12 G13 L30 Y71 K107 F108 F109 I110 W115 G230 Q16 G17 L34 Y75 K111 F112 F113 I114 W119 G223 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=24uM remove_due_to_license_issue IC50=24000nM P56817 19036583 453 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3eyd A 2.3 BS04 BE8 A 1 H57 R123 G137 S139 F154 R155 A156 A157 V158 C159 H57 R123 G137 S139 F154 R155 A156 A157 V158 C159 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P26664 19022670 401 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 3eyg A 1.9 BS01 MI1 A 1 L881 G882 E883 G884 G887 V889 A906 K908 M956 F958 L959 L1010 G1020 D1021 L17 G18 E19 G20 G23 V25 A42 K44 M84 F86 L87 L138 G148 D149 D1003 A1005 R1007 N1008 D1021 D1040 D131 A133 R135 N136 D149 D168 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.6nM remove_due_to_license_issue IC50=15nM, EC50=53nM, Kd=>10000nM, Ki=0.700000nM P23458 19361440 1 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 3eyh A 2.0 BS01 IZA A 1 L881 E883 V889 A906 M956 E957 F958 L959 G962 L1010 L17 E19 V25 A42 M89 E90 F91 L92 G95 L143 D1003 A1005 R1007 N1008 D1021 D1040 D136 A138 R140 N141 D154 D173 2.7.10.2 0004672,0004713,0005524,0006468 ic50=20nM remove_due_to_license_issue IC50=5.2nM P23458 19361440 2001 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPENHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 3eyl A 3.0 BS02 SMK A 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 K44 G53 L54 T55 D56 W57 E61 Q66 W70 2.3.2.27 remove_due_to_license_issue IC50=86nM P98170 18992220 600 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 3ezr A 1.9 BS01 EZR A 1 I10 A31 V64 F80 E81 F82 L83 H84 D86 K89 Q131 L134 A144 D145 F146 I10 A31 V57 F73 E74 F75 L76 H77 D79 K82 Q124 L127 A137 D138 F139 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T140 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=10000nM P24941 19097791 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ezr A 1.9 BS02 EZR A 2 T26 E28 T26 E28 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T140 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=10000nM P24941 19097791 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ezv A 1.99 BS01 EZV A 1 I10 A31 F80 E81 F82 L83 H84 D86 L134 D145 I10 A31 F73 E74 F75 L76 H77 D79 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 19097791 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3f07 A 3.3 BS03 AGE A 1 D101 H142 H143 D178 H180 G206 F208 Y306 D89 H130 H131 D166 H168 G194 F196 Y294 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue Q9BY41 19053282 500 SLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 3f0r A 2.54 BS02 TSN A 1 I34 P35 R37 W141 P273 Y306 I20 P21 R23 W127 P259 Y292 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue IC50=90nM, Ki=45nM, Kd=3.9e+2nM Q9BY41 19053282 800 SLVPVYIYSPEYVSMCDSLIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 3f0r A 2.54 BS03 TSN A 2 Y100 H143 F152 D178 H180 Y306 Y86 H129 F138 D164 H166 Y292 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue IC50=90nM, Ki=45nM, Kd=3.9e+2nM Q9BY41 19053282 801 SLVPVYIYSPEYVSMCDSLIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 3f15 A 1.7 BS06 HS1 A 1 I180 L181 A182 H218 E219 H222 H228 P238 Y240 I75 L76 A77 H113 E114 H117 H123 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=7.88nM remove_due_to_license_issue P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3f16 A 1.16 BS06 HS3 A 1 I180 L181 A182 T215 H218 E219 H222 H228 P238 Y240 I75 L76 A77 T110 H113 E114 H117 H123 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=5.91nM remove_due_to_license_issue P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3f17 A 1.1 BS06 HS4 A 1 I180 A182 L214 T215 H218 E219 H222 H228 V235 P238 Y240 I75 A77 L109 T110 H113 E114 H117 H123 V130 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=2.36nM remove_due_to_license_issue Ki=2.0nM P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3f18 A 1.13 BS06 HS5 A 1 I180 L181 A182 H218 E219 H222 H228 P238 Y240 I75 L76 A77 H113 E114 H117 H123 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=39.5nM remove_due_to_license_issue P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3f19 A 1.13 BS06 HS6 A 1 L181 A182 H218 E219 H222 H228 T239 Y240 L76 A77 H113 E114 H117 H123 T134 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=65.1nM remove_due_to_license_issue P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3f1a A 1.25 BS06 HS7 A 1 L181 A182 H218 E219 H222 H228 P238 Y240 L76 A77 H113 E114 H117 H123 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=61.1nM remove_due_to_license_issue P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3f27 D 2.75 BS01 dna A 0 R70 N73 F75 S99 W106 Y137 R141 R3 N6 F8 S32 W39 Y70 R74 ? remove_due_to_license_issue Q61473 19328208 1 ~ 16 IRRPMNAFMVWAKDERKRLAQQNPDLHNAELSKMLGKSWKALTLAEKRPFVEEAERLRVQHMQDHPNYKYRPRR 3f27 D 2.75 BS02 dna B 0 R69 R70 M72 M76 K80 R83 H94 N95 Y137 R2 R3 M5 M9 K13 R16 H27 N28 Y70 ? remove_due_to_license_issue Q61473 19328208 1 ~ 16 IRRPMNAFMVWAKDERKRLAQQNPDLHNAELSKMLGKSWKALTLAEKRPFVEEAERLRVQHMQDHPNYKYRPRR 3f2a A 1.9 BS01 985 A 1 L44 F49 A65 K67 L120 E121 L174 I185 D186 L13 F18 A34 K36 L89 E90 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=57nM remove_due_to_license_issue IC50=57nM P11309 19256503 1 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLS 3f33 A 1.7 BS01 PFL A 1 S27 Y28 R59 S26 Y27 R58 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 Kd=0.46mM remove_due_to_license_issue P02791 19605349 2001 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3f34 A 1.68 BS01 DIE A 1 S27 Y28 S26 Y27 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 Kd=0.69mM remove_due_to_license_issue P02791 19605349 2001 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3f35 A 1.92 BS01 DIE A 1 S27 R59 S26 R58 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 Kd=0.69mM remove_due_to_license_issue P02791 19605349 2001 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3f36 A 1.7 BS01 IP0 A 1 Y28 R59 Y27 R58 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 Kd=1.3mM remove_due_to_license_issue P02791 19605349 2001 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3f37 A 1.54 BS01 2MY A 1 S27 Y28 L81 S26 Y27 L80 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 Kd=2.4mM remove_due_to_license_issue P02791 19605349 2001 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3f38 A 1.75 BS01 2MY A 1 S27 Y28 R59 S26 Y27 R58 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 Kd=2.4mM remove_due_to_license_issue P02791 19605349 2001 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3f3a A 2.0 BS01 TRP A 1 A22 G24 L25 G26 Y108 F253 T254 S256 F259 S355 I359 A18 G20 L21 G22 Y104 F246 T247 S249 F252 S348 I352 ? 0005886,0016020,0035725 Ki=64800nM remove_due_to_license_issue O67854 19074341 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3f3a A 2.0 BS02 TRP A 2 R30 G249 F253 D404 G408 T409 R26 G242 F246 D397 G401 T402 ? 0005886,0016020,0035725 Ki=64800nM remove_due_to_license_issue O67854 19074341 602 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3f3a A 2.0 BS03 TRP A 3 R11 D272 Q273 D274 G439 R7 D265 Q266 D267 G432 ? 0005886,0016020,0035725 Ki=64800nM remove_due_to_license_issue O67854 19074341 603 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3f3a A 2.0 BS04 TRP A 4 F306 N310 A313 I314 A317 N321 F299 N303 A306 I307 A310 N314 ? 0005886,0016020,0035725 Ki=64800nM remove_due_to_license_issue O67854 19074341 604 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3f3c A 2.1 BS01 PFF A 1 N21 A22 G24 G26 Y108 F253 T254 S256 F259 S355 I359 N17 A18 G20 G22 Y104 F247 T248 S250 F253 S349 I353 ? 0005886,0016020,0035725 Ki=950nM remove_due_to_license_issue O67854 19074341 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3f3d A 2.3 BS03 MET A 1 N21 A22 G24 G26 Y108 F253 T254 S256 S355 I359 N17 A18 G20 G22 Y104 F247 T248 S250 S349 I353 ? 0005886,0016020,0035725 Kd=69nM remove_due_to_license_issue O67854 19074341 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3f3e A 1.8 BS01 LEU A 1 N21 A22 G24 L25 G26 Y108 F253 T254 S256 F259 S355 N17 A18 G20 L21 G22 Y104 F247 T248 S250 F253 S349 ? 0005886,0016020,0035725 Kd=20nM remove_due_to_license_issue O67854 19074341 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3f3t A 2.5 BS01 1AU A 1 K295 E310 M314 I336 T338 D404 F405 K39 E54 M58 I80 T82 D148 F149 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 Kd=26uM remove_due_to_license_issue IC50=6.41e+4nM P00523 19396179 1 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f3t A 2.5 BS02 1AU A 2 L273 G274 Q275 G276 Y340 M341 G344 C345 F405 L17 G18 Q19 G20 Y84 M85 G88 C89 F149 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 Kd=26uM remove_due_to_license_issue IC50=6.41e+4nM P00523 19396179 534 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f3u A 2.5 BS01 1AW A 1 E310 M314 A403 D404 F405 E54 M58 A147 D148 F149 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 Kd=18uM remove_due_to_license_issue P00523 19396179 1 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f3u A 2.5 BS02 1AW A 2 L273 G274 Q275 G276 E280 V281 Y340 M341 C345 F405 L17 G18 Q19 G20 E24 V25 Y84 M85 C89 F149 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 Kd=18uM remove_due_to_license_issue P00523 19396179 534 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f3v A 2.6 BS01 1BU A 1 L273 E310 M314 M341 L393 A403 D404 L17 E54 M58 M85 L137 A147 D148 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=21nM, Kd=73nM P00523 19462975 1 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f3w A 2.6 BS01 1BU A 1 A293 E310 M314 M341 L393 A403 D404 F405 A37 E54 M58 M85 L137 A147 D148 F149 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=21nM, Kd=73nM P00523 19462975 1 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f48 A 1.9 BS03 ALA A 1 A22 G24 G26 Y108 F253 T254 S256 A18 G20 G22 Y104 F247 T248 S250 ? 0005886,0016020,0035725 Kd=512nM remove_due_to_license_issue O67854 19074341 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3f5p A 2.9 BS01 741 A 1 L1005 A1031 K1033 F1047 E1050 M1079 M1082 T1083 M1142 L26 A52 K54 F68 E71 M100 M103 T104 M158 D1135 R1139 N1140 D1153 E1162 D151 R155 N156 D169 E178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=140nM P08069 19041240 1 SFSAADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3f66 A 1.4 BS01 IHX A 1 I1084 A1108 L1157 Y1159 M1160 M1211 I33 A52 L101 Y103 M104 M155 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A182 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.9uM remove_due_to_license_issue IC50=900nM P08581 19059779 1 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHY 3f68 H 1.75 BS03 91U H 1 H57 N98 A190 S195 V213 S214 W215 G216 E217 F227 H43 N95 A191 S196 V216 S217 W218 G219 E220 F230 3.4.21.5 0004252,0005509,0006508,0007596 Ki=8.7uM remove_due_to_license_issue P00734 19520086 901 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3f69 A 2.8 BS01 XDR A 1 L17 V25 A38 V95 A142 L145 D156 L15 V23 A36 V93 A140 L143 D154 D138 K140 A142 N143 D156 T179 D136 K138 A140 N141 D154 T162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P9WI81 19008858 309 TPSHLSDRYELGEILGFGGMSEVHLARDLRDHRDVAVKVLRADLARDPSFYLRFRREAQNAAALNHPAIVAVYDTGEAETPAGPLPYIVMEYVDGVTLRDIVHTEGPMTPKRAIEVIADACQALNFSHQNGIIHRDVKPANILISATNAVKVVDFGIARAITAQYLSPEQARGDSVDARSDVYSLGCVLYEVLTGEPPFTGDSPVSVAYQHVREDPIPPSARHEGLSADLDAVVLKALAKNPENRYQTAAEMRADLVRVHNGEPPEAPKV 3f69 B 2.8 BS01 XDR B 1 V25 A38 K40 M92 V95 A142 L145 V155 D156 V24 A37 K39 M91 V94 A141 L144 V154 D155 D138 K140 A142 N143 D156 T179 D137 K139 A141 N142 D155 T175 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P9WI81 19008858 309 TTPSHLSDRYELGEILGFGGMSEVHLARDLRDHRDVAVKVLRADLARDPSFYLRFRREAQNAAALNHPAIVAVYDTGEAETPAGPLPYIVMEYVDGVTLRDIVHTEGPMTPKRAIEVIADACQALNFSHQNGIIHRDVKPANILISATNAVKVVDFGIARAIADSGNSVTQTIGTAQYLSPEQARGDSVDARSDVYSLGCVLYEVLTGEPPFTGDSPVSVAYQHVREDPIPPSARHEGLSADLDAVVLKALAKNPENRYQTAAEMRADLVRVHNGEPPEAPKV 3f6e X 1.34 BS01 8PA X 1 N23 P24 G25 S26 E47 H70 N22 P23 G24 S25 E46 H69 G25 E47 L109 L110 T111 N112 G401 D428 N455 T457 Y458 A460 L461 S525 G24 E46 L108 L109 T110 N111 G400 D427 N454 T456 Y457 A459 L460 S524 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 19140682 602 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTVSP 3f6g A 2.0 BS01 ILE B 1 G428 Y430 D431 G39 Y41 D42 2.3.3.21 0003852,0009098 remove_due_to_license_issue Q8F3Q1 19351325 1 KVLTIKSCNIHSGIGIRPHAQIELEYQGKIHKEISEGDGGYDAFMNALTKITNRLGISIPKLIDYEVRIPPGGKTDALVETRITWNKSLEEDQTFKTMGVHPDQTVAAVHATEKMLNQILQ 3f6g A 2.0 BS02 ILE A 1 T464 A466 P493 D494 Q495 T75 A77 P102 D103 Q104 2.3.3.21 0003852,0009098 remove_due_to_license_issue Q8F3Q1 19351325 1 KVLTIKSCNIHSGIGIRPHAQIELEYQGKIHKEISEGDGGYDAFMNALTKITNRLGISIPKLIDYEVRIPPGGKTDALVETRITWNKSLEEDQTFKTMGVHPDQTVAAVHATEKMLNQILQ 3f6g B 2.0 BS01 ILE B 1 I458 T464 A466 P493 D494 Q495 I69 T75 A77 P96 D97 Q98 2.3.3.21 0003852,0009098 remove_due_to_license_issue Q8F3Q1 19351325 1 KVLTIKSCNIHSGIGIRPHAQIELEYQGKIHKEISEGDGGYDAFMNALTKITNRLGISIPKLIDYEVRIPPGGKTDALVETRITWNKTFKTMGVHPDQTVAAVHATEKMLNQILQ 3f6g B 2.0 BS02 ILE A 1 G428 Y430 D431 Y454 G39 Y41 D42 Y65 2.3.3.21 0003852,0009098 remove_due_to_license_issue Q8F3Q1 19351325 1 KVLTIKSCNIHSGIGIRPHAQIELEYQGKIHKEISEGDGGYDAFMNALTKITNRLGISIPKLIDYEVRIPPGGKTDALVETRITWNKTFKTMGVHPDQTVAAVHATEKMLNQILQ 3f6h A 2.7 BS01 ILE A 1 G428 Y430 D431 Y454 G39 Y41 D42 Y65 2.3.3.21 0003852,0009098 remove_due_to_license_issue Q8F3Q1 19351325 1 KVLTIKSCNIHSGIGIRPHAQIELEYQGKIHKEISEGDGGYDAFMNALTKITNRLGISIPKLIDYEVRIPPGGKTDALVETRITWNDQTFKTMGVHPDQTVAAVHATEKMLNQILQPWQ 3f70 A 2.1 BS01 MLZ A 1 D546 F570 W573 E608 D329 F353 W356 E391 ? 0005634,0006355 Kd=14uM remove_due_to_license_issue Q969R5 19233876 20 QDALVLGFDWGKFLKDHSYKAAPVSCFKHVPLYDQWEDVMKGMKVEVLNSDAVLRVYWIASVIQTAGYRVLLRYEGFENDASHDFWCNLGTVDVHPIGWCAINSKILVPPRTIHAKFTDWKGYLMKRLVGSRTLPVDFHIKMVESMKYPFRQGMRLEVVDKSQVSRTRMAVVDTVIGGRLRLLYEDDDFWCHMWSPLIHPVGWSRRVGHRAVYTEGGWFEEGMKLEAIDPLNLGNICVATVCKVLLDGYLMICVDDWFCYHASSHAIFPATFCQKNDIELTPPKGYEAQTFNWENYLEKTKSKAAPSRLFNMDCPNHGFKVGMKLEAVDLMEPRLICVATVKRVVHRLLSIHFDGWDSEYDQWVDCESPDIYPVGWCELTGYQLQPPVAAEP 3f78 A 1.6 BS01 ICF A 1 I235 Y257 K287 E301 L302 K305 Y307 I108 Y130 K160 E174 L175 K178 Y180 ? remove_due_to_license_issue P20701 19332643 1 GNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKWKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIY 3f7b A 2.05 BS02 AG5 A 1 N62 H64 S65 K91 Q92 H94 H96 H119 V121 I141 L198 T199 T200 N67 H69 S70 K93 Q94 H96 H98 H121 V123 I136 L197 T198 T199 H64 H94 H96 E106 H119 T199 H69 H96 H98 E108 H121 T198 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 ic50=64nM remove_due_to_license_issue IC50=64nM P22748 20363633 302 ESHWCYEVQAESSNYPCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKGTSPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 3f7g E 2.3 BS01 389 E 1 K121 G130 L131 Q132 S133 W134 D138 E143 W147 K44 G53 L54 Q55 S56 W57 D61 E66 W70 F81 F4 2.3.2.27 remove_due_to_license_issue Q96CA5 19228017 1 GPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQDKVRCFFCYGGLQSWKRGDDPWTEHAKWFPSCQFLLRSKGRDFVHSVQETHS 3f7h A 1.8 BS02 419 A 1 K121 V122 R123 G130 L131 Q132 S133 W134 D138 E143 W147 K44 V45 R46 G53 L54 Q55 S56 W57 D61 E66 W70 F81 F4 2.3.2.27 remove_due_to_license_issue Q96CA5 19228017 1 GPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQDKVRCFFCYGGLQSWKRGDDPWTEHAKWFPGCQFLLRSKGQEYINNIH 3f7i A 1.9 BS02 G13 A 1 K121 G130 L131 Q132 S133 W134 D138 E143 W147 K44 G53 L54 Q55 S56 W57 D61 E66 W70 F81 F4 2.3.2.27 remove_due_to_license_issue Q96CA5 19228017 1 GPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQDKVRCFFCYGGLQSWKRGDDPWTEHAKWFPGCQFLLRSKGQEYINNIH 3f7u A 2.0 BS02 AG4 A 1 H64 Q92 H94 H119 V121 L198 T199 T200 H62 Q87 H89 H114 V116 L187 T188 T189 H64 H94 H96 E106 H119 T199 H62 H89 H91 E101 H114 T188 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 ic50=246nM remove_due_to_license_issue IC50=246nM P22748 20363633 265 WCYEVQAESCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 3f7z A 2.4 BS01 34O A 1 F67 A83 K85 D133 Y134 V135 L188 C199 D200 F34 A50 K52 D97 Y98 V99 L152 C163 D164 D181 K183 N186 D200 S219 D145 K147 N150 D164 S183 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=65nM remove_due_to_license_issue IC50=65nM P49841 19200745 3000 LSKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 3f80 A 1.6 BS03 6HN A 1 D124 H126 D128 S137 H141 D183 D232 D119 H121 D123 S132 H136 D178 D227 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=60uM remove_due_to_license_issue P05089 19032027 551 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 3f81 A 1.9 BS01 STT A 1 M69 D92 C124 R125 E126 Y128 S129 R130 M63 D86 C118 R119 E120 Y122 S123 R124 3.1.3.16,3.1.3.48 0001772,0004721,0004722,0004725,0004726,0005515,0005634,0005654,0005737,0005829,0005856,0006338,0006357,0006470,0008092,0008138,0016311,0016791,0017018,0019901,0030336,0030946,0030971,0031514,0033192,0033549,0035335,0042059,0043409,0045931,0046329,0050860,0050868,0050922,0051893,0070373,0071364,0120183,0140791,0140793,0180004,0180005,0180006,0180007,0180008,1990264,1990439,1990782 ic50=0.074uM remove_due_to_license_issue P51452 19888758 1 LSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVLNAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRVLVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKEGKLKP 3f82 A 2.5 BS01 353 A 1 V1092 A1108 K1110 F1124 E1127 M1131 F1134 L1157 M1160 F1200 H1202 M1211 A1221 D1222 F1223 V38 A49 K51 F61 E64 M68 F71 L94 M97 F137 H139 M148 A158 D159 F160 D1204 A1206 R1208 N1209 D1222 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 Ki=4.6nM remove_due_to_license_issue IC50=3.9nM P08581 19260711 2001 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3f88 A 2.6 BS01 3HT A 1 I62 F67 V70 A83 K85 Y134 V135 L188 C199 D200 I28 F33 V36 A49 K51 Y94 V95 L148 C159 D160 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=2.3nM P49841 19200745 999 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 3f8c A 2.2 BS01 HT1 A 1 M8 V15 A92 W96 M6 V13 A87 W91 ? Kd=21nM remove_due_to_license_issue A2RI36 19096365 127 EIPKEMLRAQTNVILLNVLKQGDNYVYGIIKQVKEASNGEMELNEATLYTIFKRLEKDGIISSYWGDEGRRKYYRLTEIGHENMRLAFESWSRVDKIIENLEA 3f8e A 2.0 BS02 TE1 A 1 N62 H64 N67 I91 Q92 F131 N59 H61 N64 I88 Q89 F127 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=59nM remove_due_to_license_issue IC50=59nM P00918 19206230 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3f8f A 2.2 BS01 DM1 A 1 M8 V15 M89 F93 W96 M8 V15 M87 F91 W94 ? Kd=236nM remove_due_to_license_issue A2RI36 19096365 127 MAEIPKEMLRAQTNVILLNVLKQGDNYVYGIIKQVKEASNGEMELNEATLYTIFKRLEKDGIISSYWGDEGGRRKYYRLTEIGHENMRLAFESWSRVDKIIENLEANKKSEAIK 3f8f B 2.2 BS01 DM1 A 1 V15 W96 V11 W92 ? remove_due_to_license_issue A2RI36 19096365 127 PKEMLRAQTNVILLNVLKQGDNYVYGIIKQVKEASNGEMELNEATLYTIFKRLEKDGIISSYWGDESQGGRRKYYRLTEIGHENMRLAFESWSRVDKIIENLEANKKSEAI 3f8s A 2.43 BS01 PF2 A 1 E205 E206 F357 S630 Y631 Y662 Y666 N710 E167 E168 F319 S592 Y593 Y624 Y628 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=12.9nM remove_due_to_license_issue IC50=13nM P27487 19275964 900 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3f8w A 2.3 BS01 ADN A 1 Y90 A118 G120 Y202 E203 G220 M221 T244 N245 H259 V262 Y84 A112 G114 Y196 E197 G214 M215 T238 N239 H253 V256 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 H259 S32 H60 H82 Y84 E85 A112 M215 S216 N239 S241 H253 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 remove_due_to_license_issue Q9BMI9 20057051 300 SVTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESDLKPNHEEVLATGAQRAELMQSWFEKIIEKLPK 3f8w B 2.3 BS01 ADN B 1 Y90 A118 G120 Y202 E203 G220 M221 T244 N245 H259 V262 Y87 A115 G117 Y199 E200 G217 M218 T241 N242 H256 V259 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 H259 S32 H63 H85 Y87 E88 A115 M218 S219 N242 S244 H256 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 remove_due_to_license_issue Q9BMI9 20057051 301 SVTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSVVGHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESDLKPNHEEVLATGAQRAELMQSWFEKIIEKLPKD 3f9n A 1.9 BS01 38M A 1 F93 D99 E205 L206 P207 F76 D82 E188 L189 P190 D130 K132 E134 N135 D148 T170 D113 K115 E117 N118 D131 T153 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.3uM remove_due_to_license_issue O14757 19155174 324 EDWDLVQTLGGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 3fa3 A 2.6 BS01 OAF A 1 Y44 T46 G47 A48 C124 G125 R161 E191 N214 P240 Y43 T45 G46 A47 C123 G124 R160 E190 N213 P239 Y44 T46 G47 A48 D59 D87 D89 H114 E116 K122 C124 G125 H126 R161 E191 N214 T221 S223 Y43 T45 G46 A47 D58 D86 D88 H113 E115 K121 C123 G124 H125 R160 E190 N213 T220 S222 4.1.3.30 0003824,0016787,0046872 remove_due_to_license_issue Q2L887 19133276 501 PMVTAATSLRRALENPDSFIVAPGVYDGLSARVALSAGFDALYMTGAGTAASVHGQADLGICTLNDMRANAEMISNISPSTPVIADADTGYGGPIMVARTTEQYSRSGVAAFHIEDQVQTKRCGHLAGKILVDTDTYVTRIRAAVQARQRIGSDIVVIARTDSLQTHGYEESVARLRAARDAGADVGFLEGITSREMARQVIQDLAGWPLLLNMVEHGATPSISAAEAKEMGFRIIIFPFAALGPAVAAMREAMEKLKRDGIPGLDKEMTPQMLFRVCGLDESMKVDAQAGGAAFDGGVDL 3fa3 B 2.6 BS01 OAF B 1 Y44 T46 G47 A48 D87 G125 R161 E191 N214 P240 Y43 T45 G46 A47 D86 G124 R160 E190 N213 P239 Y44 T46 G47 A48 D59 D87 D89 H114 E116 K122 C124 G125 H126 R161 E191 N214 T221 S223 Y43 T45 G46 A47 D58 D86 D88 H113 E115 K121 C123 G124 H125 R160 E190 N213 T220 S222 4.1.3.30 0003824,0016787,0046872 remove_due_to_license_issue Q2L887 19133276 501 PMVTAATSLRRALENPDSFIVAPGVYDGLSARVALSAGFDALYMTGAGTAASVHGQADLGICTLNDMRANAEMISNISPSTPVIADADTGYGGPIMVARTTEQYSRSGVAAFHIEDQVQTKRCGHLAGKILVDTDTYVTRIRAAVQARQRIGSDIVVIARTDSLQTHGYEESVARLRAARDAGADVGFLEGITSREMARQVIQDLAGWPLLLNMVEHGATPSISAAEAKEMGFRIIIFPFAALGPAVAAMREAMEKLKRDGIPGLDKEMTPQMLFRVCGLDESMKVDAQAGGAAFDGGVDLK 3faa A 3.35 BS01 55F A 1 I211 A230 K232 Y249 L278 V279 S280 Y282 H283 L340 D351 I41 A60 K62 Y79 L108 V109 S110 Y112 H113 L170 D181 D333 K335 N338 D351 T375 D163 K165 N168 D181 T203 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue Ki=7.1nM, EC50=14800nM P36897 19135364 601 ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDINHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG 3fal B 2.36 BS01 LO2 B 1 L258 A259 S262 M296 T300 F313 F324 I337 H419 L426 W441 L53 A54 S57 M91 T95 F108 F119 I132 H214 L221 W236 ? 0003677,0004879,0006629 ic50=165nM remove_due_to_license_issue Q9Z0Y9 18800767 1 PQLSPEQLGMIEKLVAAQQQCNRRSFSDRLRVTPWPPQSREARQQRFAHFTELAIVSVQEIVDFAKQLPGFLQLSREDQIALLKTSAIEVMLLETSRRYNPGSESITFLKDFSYNREDFAKAGLQVEFINPIFEFSRAMNELQLNDAEFALLIAISIFSADRPNVQDQLQVERLQHTYVEALHAYVSINHPHDPLMFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 3fas A 1.4 BS01 GLU A 1 Y59 L88 T89 R94 G139 S140 T141 E191 Y59 L88 T89 R94 G139 S140 T141 E191 ? 0015276,0016020 Ki=171nM remove_due_to_license_issue P19493 19022251 270 GRTVVVTTIMESPYVMYKKNHEMFEGNDKYEGYCVDLASEIAKHIGIKYKIAIVPDGKYGARDADTKIWNGMVGELVYGKAEIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWTYMRSAEPSVFTRTTAEGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSSLRTPVNLAVLKLSEAGVLDKLKNKWWYDKGECG 3fat A 1.9 BS01 AMQ A 1 Y59 T89 R94 L136 G139 S140 T141 E191 Y59 T89 R94 L136 G139 S140 T141 E191 ? 0015276,0016020 Kd=22.8nM remove_due_to_license_issue Ki=40nM P19493 19022251 427 GRTVVVTTIMESPYVMYKKNHEMFEGNDKYEGYCVDLASEIAKHIGIKYKIAIVPDGKYGARDADTKIWNGMVGELVYGKAEIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWTYMRSAEPSVFTRTTAEGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSSLRTPVNLAVLKLSEAGVLDKLKNKWWYDKGEC 3fc1 X 2.4 BS01 52P X 1 A51 K53 L104 V105 T106 H107 M109 G110 A111 D112 L167 A38 K40 L91 V92 T93 H94 M96 G97 A98 D99 L154 N155 D168 N142 D155 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Kd=2.8nM, IC50=70nM, Ki=0.800000nM Q16539 16302819 362 RPTFYRQELIWEVPERYQNLSPVSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3fc2 A 2.45 BS01 IBI A 1 L59 C67 V114 E131 C133 R134 R136 F183 L23 C31 V78 E95 C97 R98 R100 F147 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=0.87nM remove_due_to_license_issue IC50=0.870000nM P53350 19383823 10 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAP 3fc8 A 1.85 BS01 IFA A 1 K15 S52 A108 L110 K6 S43 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=4.1uM remove_due_to_license_issue P02766 19125186 3000 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3fc8 B 1.85 BS01 IFA B 1 K15 A108 L110 K6 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=4.1uM remove_due_to_license_issue P02766 19125186 2000 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3fcb A 1.8 BS01 IFB A 1 K15 L17 A108 L110 K6 L8 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=4.9uM remove_due_to_license_issue P02766 19125186 3000 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3fcb B 1.8 BS01 IFB B 1 K15 L17 A108 L110 K6 L8 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=4.9uM remove_due_to_license_issue P02766 19125186 2000 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3fcf A 1.84 BS01 FCF A 1 G143 Q144 D145 Y147 C157 F158 S169 N204 G246 S247 H268 S270 S273 G62 Q63 D64 Y66 C76 F77 S88 N123 G165 S166 H187 S189 S192 D145 Y147 F158 H268 D64 Y66 F77 H187 3.2.2.27 0004844,0006281,0006284,0016799 ic50=40uM remove_due_to_license_issue IC50=4.0e+4nM P13051 19396178 1 MEFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPLSVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 3fci A 1.27 BS01 3FI A 1 G143 D145 Y147 C157 F158 N204 G246 S247 H268 S273 G62 D64 Y66 C76 F77 N123 G165 S166 H187 S192 D145 Y147 F158 H268 D64 Y66 F77 H187 3.2.2.27 0004844,0006281,0006284,0016799 ic50=1.3uM remove_due_to_license_issue IC50=1.3e+3nM P13051 19396178 1 MEFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPLSVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 3fck B 1.64 BS01 FCK B 1 G143 Q144 D145 Y147 F158 P168 S169 N204 H268 S270 P271 L272 G61 Q62 D63 Y65 F76 P86 S87 N122 H186 S188 P189 L190 3.2.2.27 0004844,0006281,0006284,0016799 remove_due_to_license_issue IC50=1.00e+5nM P13051 19396178 1 EFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPLSVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 3fcl A 1.7 BS01 3FL A 1 G143 Q144 D145 Y147 C157 F158 N204 H268 S270 S273 G61 Q62 D63 Y65 C75 F76 N122 H186 S188 S191 D145 Y147 F158 H268 D63 Y65 F76 H186 3.2.2.27 0004844,0006281,0006284,0016799 ic50=315uM remove_due_to_license_issue IC50=3.15e+5nM P13051 19396178 1 EFFGESWKKHLSGEFGKPYFIKLMGFVAEERKHYTVYPPPHQVFTWTQMCDIKDVKVVILGQDPYHGPNQAHGLCFSVQRPVPPPPSLENIYKELSTDIEDFVHPGHGDLSGWAKQGVLLLNAVLTVRAHQANSHKERGWEQFTDAVVSWLNQNSNGLVFLLWGSYAQKKGSAIDRKRHHVLQTAHPSPLSVYRGFFGCRHFSKTNELLQKSGKKPIDWKEL 3fcq A 1.75 BS06 M3S A 1 N112 A113 H142 E143 E166 H231 N112 A113 H142 E143 E166 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=1.7mM remove_due_to_license_issue P00800 20394106 600 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 3fd2 A 2.69 BS01 dna B 0 D22 G23 S24 Y26 K28 I30 I49 Q50 R51 R75 I79 Q139 N142 R235 D237 Y238 K239 Q244 N273 R275 R278 G289 R347 D18 G19 S20 Y22 K24 I26 I45 Q46 R47 R71 I75 Q135 N138 R203 D205 Y206 K207 Q212 N241 R243 R246 G257 R315 G21 D22 G17 D18 3.1.-.- 0004519,0009507,0046872 remove_due_to_license_issue C0JWR6 19153140 501 ~ 524 NTLQPTEAAYIAGFLDGDGSIYAKLIPRPDYKDIKYQVSLAISFIQRKDKFPYLQDIYDQLGKRGNLRKDRGDGIADYTIIGSTHLSIILPDLVPYLRIKKKQANRILHIINLYPQAQKNPSKFLDLVKIVDDVQNLNKRADELKSTNYDRLLEEFLKAGKIESSPTGSGSGSKKNTLQPTEAAYIAGFLDGDGSIYAKLIPRPDYKDIKYQVSLAISFIQRKDKFPYLQDIYDQLGKRGNLRKDRGDGIADYTIIGSTHLSIILPDLVPYLRIKKKQANRILHIINLYPQAQKNPSKFLDLVKIVDDVQNLNKRADELKSTNYDRLLEEFLKAGKIE 3fd2 A 2.69 BS02 dna C 0 R32 D34 Y35 K36 Q41 N70 R72 R75 I85 G86 Q122 R144 D225 S227 Y229 K231 I233 I252 Q253 R254 Q342 N345 R28 D30 Y31 K32 Q37 N66 R68 R71 I81 G82 Q118 R140 D193 S195 Y197 K199 I201 I220 Q221 R222 Q310 N313 G21 D22 G17 D18 3.1.-.- 0004519,0009507,0046872 remove_due_to_license_issue C0JWR6 19153140 551 ~ 574 NTLQPTEAAYIAGFLDGDGSIYAKLIPRPDYKDIKYQVSLAISFIQRKDKFPYLQDIYDQLGKRGNLRKDRGDGIADYTIIGSTHLSIILPDLVPYLRIKKKQANRILHIINLYPQAQKNPSKFLDLVKIVDDVQNLNKRADELKSTNYDRLLEEFLKAGKIESSPTGSGSGSKKNTLQPTEAAYIAGFLDGDGSIYAKLIPRPDYKDIKYQVSLAISFIQRKDKFPYLQDIYDQLGKRGNLRKDRGDGIADYTIIGSTHLSIILPDLVPYLRIKKKQANRILHIINLYPQAQKNPSKFLDLVKIVDDVQNLNKRADELKSTNYDRLLEEFLKAGKIE 3fdn A 1.9 BS01 MMH A 1 R137 L139 G140 A160 E211 Y212 A213 G216 T217 R220 L263 R12 L14 G15 A35 E86 Y87 A88 G91 T92 R95 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T159 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=0.033uM remove_due_to_license_issue O14965 19140666 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHACGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPSNCQ 3fed A 1.29 BS04 BIX A 1 R200 N247 D377 E414 E415 G508 R524 R526 Y542 H543 K689 Y690 R152 N199 D328 E365 E366 G459 R475 R477 Y493 H494 K640 Y641 H367 D377 E414 E415 H318 D328 E365 E366 3.4.17.21 0004180,0004181,0005515,0005886,0006508,0008236,0008237,0008239,0016020,0016805,0046872 Ki=34.6nM remove_due_to_license_issue Q9Y3Q0 19678840 1 SIRWKLVSEMKAENIKSFLRSFTKLPHLAGTEQNFLLAKKIQTQWKKFGLDSAKLVHYDVLLSYPNETNANYISIVDEHETEIFKTSPPPDGYENVTNIVPPYNAFSAQGMPEGDLVYVNYARTEDFFKLEREMGINCTGKIVIARYGKIFRGNKVKNAMLAGAIGIILYSDPADYFAPEVQPYPKGWNLPGTAAQRGNVLNLNGAGDPLTPGYPAKEYTFRLDVEEGVGIPRIPVHPIGYNDAEILLRYLGGIAPPDKSWKGALNVSYSIGPGFTGSSFRKVRMHVYNINKITRIYNVVGTIRGSVEPDRYVILGGHRDSWVFGAIDPTSGVAVLQEIARSFGKLMSKGWRPRRTIIFASWDAEEFGLLGSTEWAEENVKILQERSIAYINSDSSIEGNYTLRVDCTPLLYQLVYKLTKEIPSPDDGFESKSLYESWLEKDPSPENKNLPRINKLGSGSDFEAYFQRLGIASGRARYTKNKKTDKYSSYPVYHTIYETFELVEKFYDPTFKKQLSVAQLRGALVYELVDSKIIPFNIQDYAEALKNYAASIYNLSKKHDQQLTDHGVSFDSLFSAVKNFSEAASDFHKRLIQVDLNNPIAVRMMNDQLMLLERAFIDPLGLPGKLFYRHIIFAPSSHNKYAGESFPGIYDAIFDIENKANSRLAWKEVKKHISIAAFTIQAAAGTLKEV 3fee A 1.56 BS04 QUS A 1 R200 N247 E414 G508 Y542 K689 Y690 R154 N201 E367 G461 Y492 K639 Y640 H367 D377 E414 E415 H320 D330 E367 E368 3.4.17.21 0004180,0004181,0005515,0005886,0006508,0008236,0008237,0008239,0016020,0016805,0046872 Ki=230nM remove_due_to_license_issue Q9Y3Q0 19678840 741 SIRWKLVSEMKAENIKSFLRSFTKLPHLAGTEQNFLLAKKIQTQWKKFGLDSAKLVHYDVLLSYPNETNANYISIVDEHETEIFKTSLEPPPDGYENVTNIVPPYNAFSAQGMPEGDLVYVNYARTEDFFKLEREMGINCTGKIVIARYGKIFRGNKVKNAMLAGAIGIILYSDPADYFAPEVQPYPKGWNLPGTAAQRGNVLNLNGAGDPLTPGYPAKEYTFRLDVEEGVGIPRIPVHPIGYNDAEILLRYLGGIAPPDKSWKGALNVSYSIGPGFTGSSFRKVRMHVYNINKITRIYNVVGTIRGSVEPDRYVILGGHRDSWVFGAIDPTSGVAVLQEIARSFGKLMSKGWRPRRTIIFASWDAEEFGLLGSTEWAEENVKILQERSIAYINSDSSIEGNYTLRVDCTPLLYQLVYKLTKEIPSPDDGFESKSLYESWLEKDPSPENKNLPRINKLGSGSDFEAYFQRLGIASGRARYTKNDKYSSYPVYHTIYETFELVEKFYDPTFKKQLSVAQLRGALVYELVDSKIIPFNIQDYAEALKNYAASIYNLSKKHDQQLTDHGVSFDSLFSAVKNFSEAASDFHKRLIQVDLNNPIAVRMMNDQLMLLERAFIDPLGLPGKLFYRHIIFAPSSHNKYAGESFPGIYDAIFDIENKANSRLAWKEVKKHISIAAFTIQAAAGTLKEV 3feg A 1.302 BS01 HC7 A 1 D242 Y267 E283 Y288 F295 W353 W356 E367 F368 Y370 Y373 D193 Y215 E231 Y236 F243 W301 W304 E315 F316 Y318 Y321 2.7.1.32,2.7.1.82 0004103,0004305,0005524,0005737,0005829,0006646,0006656,0006657,0007517,0008654,0016301 remove_due_to_license_issue Q9Y259 20299452 1 SRDAERRAYQWCREYLGGAWRRVQPEELRVYPVNLLFRCSLPDHLPSVGEEPREVLLRLYGQGVDSLVLESVMFAILAERSLGPQLYGVFPEGRLEQYIPSRPLKTQELREPVLSAAIATKMAQFHGMEMPFTKEPHWLFGTMERYLKQIQDLPPTGLPEMNLLEMYSLKDEMGNLRKLLESTPSPVVFCHNDIQEGNILLLSEPDSLMLVDFEYSSYNYRGFDIGNHFCEWVYDYTHEEWPFYKARPTDYPTQEQQLHFIRHYLAEAKKGETLSQEEQRKLEEDLLVEVSRYALASHFFWGLWSILQASMSTIEFGYLDYAQSRFQFYFQQKGQL 3fei A 2.4 BS02 CTM A 1 F273 C275 C276 S280 Y314 F318 M330 V332 M355 H440 Y464 F51 C53 C54 S58 Y92 F96 M108 V110 M133 H218 Y242 ? 0003677,0004879,0005634,0006355 ic50=0.02uM remove_due_to_license_issue Q07869 19326383 1 DLKSLAKRIYEAYLKNFNMNKVKARVILSPFVIHDMETLCMAEKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANLDLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFDFAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDIFLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDMY 3fej A 2.01 BS02 CTM A 1 F282 C285 R288 S289 H323 Y327 L330 M348 M364 H449 Y473 F63 C66 R69 S70 H104 Y108 L111 M129 M145 H230 Y254 ? 0003677,0004879,0005634,0006355 ic50=0.74uM remove_due_to_license_issue P37231 19326383 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3ff3 A 1.37 BS04 GLU A 1 R200 N247 E414 G508 Y542 H543 K689 Y690 R151 N198 E364 G458 Y492 H493 K639 Y640 H367 D377 E414 E415 H317 D327 E364 E365 3.4.17.21 0004180,0004181,0005515,0005886,0006508,0008236,0008237,0008239,0016020,0016805,0046872 remove_due_to_license_issue Q9Y3Q0 19678840 1 SIRWKLVSEMKAENIKSFLRSFTKLPHLAGTEQNFLLAKKIQTQWKKFGLDSAKLVHYDVLLSYPNETNANYISIVDEHETEIFKTSPPDGYENVTNIVPPYNAFSAQGMPEGDLVYVNYARTEDFFKLEREMGINCTGKIVIARYGKIFRGNKVKNAMLAGAIGIILYSDPADYFAPEVQPYPKGWNLPGTAAQRGNVLNLNGAGDPLTPGYPAKEYTFRLDVEEGVGIPRIPVHPIGYNDAEILLRYLGGIAPPDKSWKGALNVSYSIGPGFTGSSFRKVRMHVYNINKITRIYNVVGTIRGSVEPDRYVILGGHRDSWVFGAIDPTSGVAVLQEIARSFGKLMSKGWRPRRTIIFASWDAEEFGLLGSTEWAEENVKILQERSIAYINSDSSIEGNYTLRVDCTPLLYQLVYKLTKEIPSPDDGFESKSLYESWLEKDPSPENKNLPRINKLGSGSDFEAYFQRLGIASGRARYTKNKKTDKYSSYPVYHTIYETFELVEKFYDPTFKKQLSVAQLRGALVYELVDSKIIPFNIQDYAEALKNYAASIYNLSKKHDQQLTDHGVSFDSLFSAVKNFSEAASDFHKRLIQVDLNNPIAVRMMNDQLMLLERAFIDPLGLPGKLFYRHIIFAPSSHNKYAGESFPGIYDAIFDIENKANSRLAWKEVKKHISIAAFTIQAAAGTLKEV 3ff6 A 3.19 BS01 RCP A 1 G2159 F2160 L2229 E2230 E2232 G2233 E2236 G465 F466 L535 E536 E538 G539 E542 6.4.1.2 0003989,0016874 remove_due_to_license_issue IC50=38nM O00763 19390150 1 PYVTKDLLQAKRFQAQTLGTTYIYDFPEMFRQALFKLWGSPDKYPKDILTYTELVLDSQGQLVEMNRLPGGNEVGMVAFKMRFKTQEYPEGRDVIVIGNDITFRIGSFGPGEDLLYLRASEMARAEGIPKIYVAANSGARIGMAEEIKHMFHVAWVDPEDPHKGFKYLYLTPQDYTRISSLNSVHCKHIEEGGESRYMITDIIGKDDGLGVENLRGSGMIAGESSLAYEEIVTISLVTCRAIGIGAYLVRLGQRVIQVENSHIILTGASALNKVLGREVYTSNNQLGGVQIMHYNGVSHITVPDDFEGVYTILEWLSYMPKDNHSPVPIITPTDPIDREIEFLPSRAPYDPRWMLAGRPHPTLKGTWQSGFFDHGSFKEIMAPWAQTVVTGRARLGGIPVGVIAVETRTVEVAVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRQYKQPILIYIPPYAELRGGSWVVIDATINPLCIEMYADKESRGGVLEPEGTVEIKFRKKDLIKSMRRIDPAYKKLMEQLGEPDLSDKDRKDLEGRLKAREDLLLPIYHQVAVQFADFHDTPGRMLEKGVISDILEWKTARTFLYWRLRRLLLEDQVKQEILQASGELSHVHIQSMLRRWFVETEGAVKAYLWDNNQVVVQWLEQHWQRSTIRENITYLKHDSVLKTIRGLVEENPEVAVDCVIYLSQHISPAERAQVVHLL 3ff6 A 3.19 BS02 RCP B 1 T1960 L1965 V1968 T266 L271 V274 6.4.1.2 0003989,0016874 remove_due_to_license_issue IC50=38nM O00763 19390150 2 PYVTKDLLQAKRFQAQTLGTTYIYDFPEMFRQALFKLWGSPDKYPKDILTYTELVLDSQGQLVEMNRLPGGNEVGMVAFKMRFKTQEYPEGRDVIVIGNDITFRIGSFGPGEDLLYLRASEMARAEGIPKIYVAANSGARIGMAEEIKHMFHVAWVDPEDPHKGFKYLYLTPQDYTRISSLNSVHCKHIEEGGESRYMITDIIGKDDGLGVENLRGSGMIAGESSLAYEEIVTISLVTCRAIGIGAYLVRLGQRVIQVENSHIILTGASALNKVLGREVYTSNNQLGGVQIMHYNGVSHITVPDDFEGVYTILEWLSYMPKDNHSPVPIITPTDPIDREIEFLPSRAPYDPRWMLAGRPHPTLKGTWQSGFFDHGSFKEIMAPWAQTVVTGRARLGGIPVGVIAVETRTVEVAVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRQYKQPILIYIPPYAELRGGSWVVIDATINPLCIEMYADKESRGGVLEPEGTVEIKFRKKDLIKSMRRIDPAYKKLMEQLGEPDLSDKDRKDLEGRLKAREDLLLPIYHQVAVQFADFHDTPGRMLEKGVISDILEWKTARTFLYWRLRRLLLEDQVKQEILQASGELSHVHIQSMLRRWFVETEGAVKAYLWDNNQVVVQWLEQHWQRSTIRENITYLKHDSVLKTIRGLVEENPEVAVDCVIYLSQHISPAERAQVVHLL 3ff6 B 3.19 BS01 RCP A 1 L1965 V1968 L269 V272 6.4.1.2 0003989,0016874 remove_due_to_license_issue IC50=38nM O00763 19390150 1 VTKDLLQAKRFQAQTLGTTYIYDFPEMFRQALFKLWGSPDKYPKDILTYTELVLDSQGQLVEMNRLPGGNEVGMVAFKMRFKTQEYPEGRDVIVIGNDITFRIGSFGPGEDLLYLRASEMARAEGIPKIYVAANSGARIGMAEEIKHMFHVAWVDPEDPHKGFKYLYLTPQDYTRISSLNSVHCKHIEEGGESRYMITDIIGKDDGLGVENLRGSGMIAGESSLAYEEIVTISLVTCRAIGIGAYLVRLGQRVIQVENSHIILTGASALNKVLGREVYTSNNQLGGVQIMHYNGVSHITVPDDFEGVYTILEWLSYMPKDNHSPVPIITPTDPIDREIEFLPSRAPYDPRWMLAGRPHPTLKGTWQSGFFDHGSFKEIMAPWAQTVVTGRARLGGIPVGVIAVETRTVEVAVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRQYKQPILIYIPPYAELRGGSWVVIDATINPLCIEMYADKESRGGVLEPEGTVEIKFRKKDLIKSMRRIDPAYKKLMEQLGEPDLSDKDRKDLEGRLKAREDLLLPIYHQVAVQFADFHDTPGRMLEKGVISDILEWKTARTFLYWRLRRLLLEDQVKQEILQASGELSHVHIQSMLRRWFVETEGAVKAYLWDNNQVVVQWLEQHWQATIRENITYLKHDSVLKTIRGLVEENPEVAVDCVIYLSQHISPAERAQVVHLLS 3ff6 B 3.19 BS02 RCP B 1 R2158 G2159 F2160 E2230 E2232 G2233 E2236 R462 G463 F464 E534 E536 G537 E540 6.4.1.2 0003989,0016874 remove_due_to_license_issue IC50=38nM O00763 19390150 2 VTKDLLQAKRFQAQTLGTTYIYDFPEMFRQALFKLWGSPDKYPKDILTYTELVLDSQGQLVEMNRLPGGNEVGMVAFKMRFKTQEYPEGRDVIVIGNDITFRIGSFGPGEDLLYLRASEMARAEGIPKIYVAANSGARIGMAEEIKHMFHVAWVDPEDPHKGFKYLYLTPQDYTRISSLNSVHCKHIEEGGESRYMITDIIGKDDGLGVENLRGSGMIAGESSLAYEEIVTISLVTCRAIGIGAYLVRLGQRVIQVENSHIILTGASALNKVLGREVYTSNNQLGGVQIMHYNGVSHITVPDDFEGVYTILEWLSYMPKDNHSPVPIITPTDPIDREIEFLPSRAPYDPRWMLAGRPHPTLKGTWQSGFFDHGSFKEIMAPWAQTVVTGRARLGGIPVGVIAVETRTVEVAVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRQYKQPILIYIPPYAELRGGSWVVIDATINPLCIEMYADKESRGGVLEPEGTVEIKFRKKDLIKSMRRIDPAYKKLMEQLGEPDLSDKDRKDLEGRLKAREDLLLPIYHQVAVQFADFHDTPGRMLEKGVISDILEWKTARTFLYWRLRRLLLEDQVKQEILQASGELSHVHIQSMLRRWFVETEGAVKAYLWDNNQVVVQWLEQHWQATIRENITYLKHDSVLKTIRGLVEENPEVAVDCVIYLSQHISPAERAQVVHLLS 3ffg A 1.54 BS01 FFG A 1 T98 Y99 R143 F174 D189 A190 Q192 S195 W215 G216 G218 C220 G226 T84 Y85 R132 F162 D179 A180 Q182 S185 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.84nM remove_due_to_license_issue Ki=0.84nM P00742 20100660 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3ffp X 1.81 BS02 LC1 X 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=72.5nM remove_due_to_license_issue Ki=72.5nM P00918 19186056 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3ffu A 2.8 BS01 GTP A 1 V24 R40 E51 F52 G54 G55 K56 E70 I97 P133 N136 V6 R22 E33 F34 G36 G37 K38 E52 I79 P115 N118 3.6.1.55 0005525,0006260,0006281,0008413,0016787,0035539,0042802,0044715,0044716,0046872 remove_due_to_license_issue Q6MPX4 19278661 4033 GHWIPVVAGFLRKDGKILVGQRPENNSLAGQWEFPGGKIENGETPEEALARELNEELGIEAEVGELKLACTHSYGDVGILILFYEILYWKGEPRAKHHMMLEWIHPEELKHRNIPEANRKILHKIYKALGLEW 3fh5 A 1.63 BS02 24P A 1 Q134 Q136 Y267 G269 M270 W311 F314 P374 A377 Y378 Q131 Q133 Y264 G266 M267 W308 F311 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=87nM remove_due_to_license_issue IC50=449nM P09960 19950900 611 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fh7 A 2.05 BS02 25P A 1 Q134 Q136 A137 Y267 G269 M270 E271 H295 E296 H299 W311 F314 E318 V367 L369 P374 Y378 Y383 Q131 Q133 A134 Y264 G266 M267 E268 H292 E293 H296 W308 F311 E315 V364 L366 P371 Y375 Y380 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 Kd=25nM remove_due_to_license_issue P09960 19950900 612 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fh8 A 1.67 BS02 27P A 1 Q134 Q136 Y267 M270 W311 F314 V367 P374 A377 Y378 P382 Q131 Q133 Y264 M267 W308 F311 V364 P371 A374 Y375 P379 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=180nM remove_due_to_license_issue IC50=120nM P09960 19950900 611 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fhb A 2.3 BS01 GAB A 1 H384 G385 Y414 F415 A416 S422 Y425 E514 H209 G210 Y239 F240 A241 S247 Y250 E339 S422 Y425 E514 S247 Y250 E339 2.4.2.- 0003950 Kd>2uM remove_due_to_license_issue Q9Y6F1 19354255 601 SMKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKGPTDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 3fhe A 2.16 BS02 28P A 1 Q136 A137 Y267 G269 M270 E271 H295 E296 H299 W311 F314 E318 V367 P374 A377 Y378 Y383 Q133 A134 Y264 G266 M267 E268 H292 E293 H296 W308 F311 E315 V364 P371 A374 Y375 Y380 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=6.0nM, Kd=350nM, Ki=3.0nM P09960 19950900 612 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fhr A 1.9 BS01 P4O A 1 L50 L52 G53 V58 A71 K73 M121 E122 L173 T186 D187 L18 L20 G21 V26 A39 K41 M89 E90 L140 T153 D154 D166 K168 N171 D187 D133 K135 N138 D154 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=210nM Q16644 19937655 1 EPKKYAVTDDYQLSKQVLGLGVNGKVLECFHRRTGQKCALKLLYDSPKARQEVDHHWQASGGPHIVCILDVYENMHHGKRCLLIIMECMEGGELFSRIQERDQAFTEREAAEIMRDIGTAIQFLHSHNIAHRDVKPENLLYTSKEKDAVLKLTDFGFAKETEKYDKSCDMWSLGVIMYILLCGFPPFGFPNPEWSEVSEDAKQLIRLLLKTDPTERLTITQFMNHPWINQSMVVPQTPLHTARVLQEDKDHWDEVKEEMTSALATMRVDYDQV 3fi2 A 2.28 BS01 JK1 A 1 V78 K93 I124 L144 M146 L148 M149 D150 A151 V196 L206 V29 K44 I75 L95 M97 L99 M100 D101 A102 V147 L157 D189 K191 N194 D207 T226 D140 K142 N145 D158 T165 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.025uM remove_due_to_license_issue IC50=25nM P53779 19261605 600 DNQFYSVEVGDSTFTVLKRYQNLKPIGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYAAAAAADEREHTIEEWKELIYKEVMN 3fi3 A 2.2 BS01 JK2 A 1 I70 A91 K93 I124 M146 L148 M149 D150 A151 L206 I26 A42 K44 I75 M97 L99 M100 D101 A102 L157 D189 K191 N194 D207 T226 D140 K142 N145 D158 T165 2.7.11.24 0004672,0004707,0005524,0006468 ic50=12nM remove_due_to_license_issue IC50=9.0nM P53779 19261605 600 DNQFYSVEVGDSTFTVLKRYQNLKPIGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYPPQIYDKQLDEREHTIEEWKELIYKEVMNS 3fj7 A 1.7 BS01 PEQ A 1 P27 G28 G54 P55 T138 S139 N170 S171 G172 P7 G8 G34 P35 T118 S119 N150 S151 G152 ? 0042597,0140104,1902358 remove_due_to_license_issue Q0PBL7 19236052 301 DVNLYGPGGPHTALKDIANKYSEKTGVKVNVNFGPQATWFEKAKKDADILFGASDQSALAIASDFGKDFNVSKIKPLYFREAIILTQKGNPLKIKGLKDLANKKVRIVVPEGAGKSNTSGTGVWEDMIGRTQDIKTIQNFRNNIVAFVPNSGSARKLFAQDQADAWITWIDWSKSNPDIGTAVAIEKDLVVYRTFNVIAKEGASKETQDFIAYLSSKEAKEIFKKYGWREH 3fjz A 1.7 BS02 GPF A 1 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 Ki=90uM remove_due_to_license_issue Ki=160nM, Kd=160nM, koff=0.120000s-1, IC50=2000nM, kon=0.000001M-1-s-1 P0A6D3 19211556 429 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGIAMRPLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 3fk1 A 1.7 BS02 GPF A 1 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 G96 R124 Q171 D313 E341 R344 H385 R386 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 K22 S23 D49 N94 P119 R124 D313 E341 H385 R386 K411 2.5.1.19 0003824,0003866,0005737,0005829,0008652,0009073,0009423,0016740,0016765 Ki=2420uM remove_due_to_license_issue Ki=160nM, Kd=160nM, koff=0.120000s-1, IC50=2000nM, kon=0.000001M-1-s-1 P0A6D3 19211556 429 MESLTLQPIARVDGTINLPGSKSVSNRALLLAALAHGKTVLTNLLDSDDVRHMLNALTALGVSYTLSADRTRCEIIGNGGPLHAEGALELFLGNAGIAMRSLAAALCLGSNDIVLTGEPRMKERPIGHLVDALRLGGAKITYLEQENYPPLRLQGGFTGGNVDVDGSVSSQFLTALLMTAPLAPEDTVIRIKGDLVSKPYIDITLNLMKTFGVEIENQHYQQFVVKGGQSYQSPGTYLVEGDASSASYFLAAAAIKGGTVKVTGIGRNSMQGDIRFADVLEKMGATICWGDDYISCTRGELNAIDMDMNHIPDAAMTIATAALFAKGTTTLRNIYNWRVKETDRLFAMATELRKVGAEVEEGHDYIRITPPEKLNFAEIATYNDHRMAMCFSLVALSDTPVTILDPKCTAKTFPDYFEQLARISQAA 3fkt A 1.9 BS01 SII A 1 L50 Y91 T92 Q93 G94 F128 I130 Y218 G250 T349 L34 Y75 T76 Q77 G78 F112 I114 Y190 G222 T316 D52 S55 N57 A59 Y91 D248 T251 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=2.8uM remove_due_to_license_issue IC50=2800nM P56817 18811140 406 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHDEFRTAAVEGPFVTLDMEDCG 3fkv A 1.847 BS01 BZB A 1 S64 R67 Y150 N152 Y221 A318 S61 R64 Y147 N149 Y218 A313 S64 R67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 R64 Y109 A111 V118 Y147 G153 E269 K310 A313 3.5.2.6 0008800,0016787,0017001,0042597,0046677 remove_due_to_license_issue IC50=200nM, Ki=27nM P00811 19241376 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSRTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3fl5 A 2.3 BS01 TXQ A 1 V45 R47 V53 K68 V95 F113 V116 H160 M163 I174 D175 V39 R41 V47 K62 V89 F107 V110 H154 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue P28523 19432557 338 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 3fl8 A 2.2881 BS02 RAR A 1 M6 V7 A8 L21 E28 L29 V32 I51 L55 R58 F96 M6 V7 A8 L21 E28 L29 V32 I51 L55 R58 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 ic50=54nM remove_due_to_license_issue IC50=54nM Q81R22 19364848 200 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 3fl9 A 2.4 BS02 TOP A 1 M6 V7 A8 V32 I51 L55 F96 M6 V7 A8 V32 I51 L55 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 ic50=77.2mM remove_due_to_license_issue Ki=24100nM, IC50=71000nM Q81R22 19364848 200 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 3fmq A 2.5 BS03 FUG A 1 F97 H109 D206 L207 I217 H218 Y324 F95 H107 D204 L205 I215 H216 Y322 D130 D141 H210 H218 E243 E339 D128 D139 H208 H216 E241 E337 3.4.11.18 0004177,0004239,0005737,0006508,0008235,0046872,0070006 remove_due_to_license_issue Q8SR45 19660503 481 CILLNQAEELPIEFLPKDGVYGKGKLFDSRNMEIENFTESDILQDARRAAEAHRRARYRVQSIVRPGITLLEIVRSIEDSTRTLLKGERNNGIGFPAGMSMNSCAAHYTVNPGEQDIVLKEDDVLKIDFGTHSDGRIMDSAFTVAFKENLEPLLVAAREGTETGIKSLGVDVRVCDIGRDINEVISSYEVEIGGRMWPIRPISDLHGHSISQFRIHGGISIPAVNNRDTTRIKGDSFYAVETFATTGKGSIDDRPPCSHFVLNTYKSRKLFNKDLIKVYEFVKDSLGTLPFSPRHLDYYGLVKGGSLKSVNLLTMMGLLTPYPPLNDIDGCKVAQFEHTVYLSEHGKEVLTRGDDY 3fmr A 2.89 BS03 TN4 A 1 F97 H109 D206 L207 H208 H218 Y324 F95 H107 D204 L205 H206 H216 Y322 D130 D141 H210 H218 E243 E339 D128 D139 H208 H216 E241 E337 3.4.11.18 0004177,0004239,0005737,0006508,0008235,0046872,0070006 remove_due_to_license_issue Q8SR45 19660503 451 CILLNQAEELPIEFLPKDGVYGKGKLFDSRNMEIENFTESDILQDARRAAEAHRRARYRVQSIVRPGITLLEIVRSIEDSTRTLLKGERNNGIGFPAGMSMNSCAAHYTVNPGEQDIVLKEDDVLKIDFGTHSDGRIMDSAFTVAFKENLEPLLVAAREGTETGIKSLGVDVRVCDIGRDINEVISSYEVEIGGRMWPIRPISDLHGHSISQFRIHGGISIPAVNNRDTTRIKGDSFYAVETFATTGKGSIDDRPPCSHFVLNTYKSRKLFNKDLIKVYEFVKDSLGTLPFSPRHLDYYGLVKGGSLKSVNLLTMMGLLTPYPPLNDIDGCKVAQFEHTVYLSEHGKEVLTRGDDY 3fmz A 2.9 BS01 2T1 A 1 L35 F36 L37 A57 M73 G75 M88 Y90 Q98 H104 R121 L35 F36 L37 A57 M73 G75 M88 Y90 Q98 H104 R121 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 remove_due_to_license_issue IC50=15nM P02753 19147488 184 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYC 3fnm B 1.7 BS01 AVN B 1 T380 N400 D422 S451 S452 G473 I476 T1 N21 D43 S72 S73 G94 I97 2.3.2.2,3.4.19.13 remove_due_to_license_issue O25743 19256527 1 TTHYSVADRWGNAVSVTYTINASYGSAASIDGAGFLLNNEMDDFSIKPGNPNLYGLVGGDANAIEANKRPLSSMSPTIVLKNNKVFLVVGSPGGSRIITTVLQVISNVIDYNMNISEAVSAPRFHMQWLPDELRIEKFGMPADVKDNLTKMGYQIVTKPVMGDVNAIQVLPKTKGSVFYGSTDPRKEF 3fnu A 3.0 BS01 006 A 1 W39 F109A F111 Y112 V120 W40 F110 F113 Y114 V122 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0006508 remove_due_to_license_issue Q8IM15 19285084 329 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFKVPFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKN 3fnu B 3.0 BS01 006 B 1 V12 S35 W39 M104 F109A F111 V120 V13 S36 W40 M104 F110 F113 V122 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0006508 remove_due_to_license_issue Q8IM15 19285084 329 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFKVPFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKN 3fpd A 2.4 BS02 Q4A A 1 D1131 A1134 D1135 R1137 D1140 L1143 D1145 R1214 F1215 D157 A160 D161 R163 D166 L169 D171 R240 F241 Y1124 Y1211 Y150 Y237 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 ic50=0.7uM remove_due_to_license_issue IC50=700nM Q9H9B1 19219047 1 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 3fpm A 3.3 BS01 793 A 1 L72 N75 V78 A91 K93 M138 E139 L141 E190 D207 L29 N32 V35 A48 K50 M95 E96 L98 E147 D164 D186 K188 E190 N191 D207 S216 T226 D143 K145 E147 N148 D164 S173 T174 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=8900nM P49137 19364658 1 PQFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKED 3fq7 A 2.15 BS01 PXG A 1 S1029 V1031 W1067 G1123 T1124 Y1150 H1151 E1212 N1217 D1245 V1247 M1248 K1273 E1406 S23 V25 W61 G117 T118 Y144 H145 E206 N211 D239 V241 M242 K267 E400 V1027 Y1150 D1245 M1248 K1273 A1407 V21 Y144 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 remove_due_to_license_issue P24630 19786580 1434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fq7 A 2.15 BS02 PXG B 1 G1304 T1305 G298 T299 V1027 Y1150 D1245 M1248 K1273 A1407 V21 Y144 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 remove_due_to_license_issue P24630 19786580 2434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fq7 B 2.15 BS01 PXG A 1 A2303 G2304 T2305 A297 G298 T299 V2027 Y2150 E2212 D2245 M2248 K2273 A2407 V21 Y144 E206 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 remove_due_to_license_issue P24630 19786580 1434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fq7 B 2.15 BS02 PXG B 1 S2029 V2031 W2067 S2122 G2123 T2124 Y2150 H2151 E2212 N2217 D2245 V2247 M2248 K2273 E2406 S23 V25 W61 S116 G117 T118 Y144 H145 E206 N211 D239 V241 M242 K267 E400 V2027 Y2150 E2212 D2245 M2248 K2273 A2407 V21 Y144 E206 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 remove_due_to_license_issue P24630 19786580 2434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fqa A 2.35 BS02 GAB A 1 S1029 R1032 W1067 S22 R25 W60 V1027 Y1150 D1245 I1248 K1273 A1407 V20 Y143 D238 I241 K266 A400 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 remove_due_to_license_issue P24630 19786580 2000 KTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRLMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVITGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fqa B 2.35 BS02 GAB A 1 A2303 G2304 T2305 A296 G297 T298 V2027 Y2150 E2212 D2245 I2248 K2273 A2407 V20 Y143 E205 D238 I241 K266 A400 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 remove_due_to_license_issue P24630 19786580 2000 KTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRLMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVITGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fqe A 2.5 BS01 P5C A 1 L377 S379 V385 A400 M448 G454 P455 R498 L501 S511 D512 L15 S17 V23 A38 M81 G87 P88 R131 L134 S144 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K163 2.7.10.2 0004672,0004713,0005524,0006468 Ki~0.0125uM remove_due_to_license_issue IC50=4nM, EC50=2500nM P43405 19220318 1 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 3fqh A 2.26 BS01 057 A 1 L377 G378 A400 A451 G454 P455 K458 L501 L15 G16 A33 A79 G82 P83 K86 L129 D494 A496 R498 N499 D512 K533 D122 A124 R126 N127 D140 K161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.57uM remove_due_to_license_issue IC50=570nM P43405 19220318 1 VYLDRKLLTLEDKELGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV 3fqk A 2.2 BS01 79Z A 1 F193 R200 L204 L314 N316 I363 S365 C366 S368 L384 M414 Y415 Y448 F188 R195 L199 L309 N311 I358 S360 C361 S363 L379 M409 Y410 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.081uM remove_due_to_license_issue P26663 19246450 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3fql A 1.8 BS01 79Z A 1 F193 R200 L204 L314 C316 I363 S365 C366 S368 M414 Y415 Y448 F188 R195 L199 L309 C311 I358 S360 C361 S363 M409 Y410 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.071uM remove_due_to_license_issue Q9WMX2 19246450 571 HHMSYTWTGALITPCAAEETKLPINALSNSLLRHHNLVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSLS 3fqs A 2.1 BS01 585 A 1 L377 S379 V385 A400 A451 G454 P455 L501 L15 S17 V23 A38 A84 G87 P88 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.041uM remove_due_to_license_issue EC50=10nM, IC50=41nM, Kd=19nM, Ki=30nM P43405 19220318 1 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 3fr2 A 2.2 BS01 8CA A 1 F16 P38 A75 D76 R126 Y128 F16 P38 A75 D76 R126 Y128 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 ic50=0.59uM remove_due_to_license_issue IC50=590nM P15090 19217286 501 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 3fr4 A 2.16 BS01 F8A A 1 F16 A33 A36 P38 S53 S55 F57 K58 A75 D76 I104 C117 R126 Y128 F16 A33 A36 P38 S53 S55 F57 K58 A75 D76 I104 C117 R126 Y128 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 ic50=0.049uM remove_due_to_license_issue P15090 19217286 501 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 3fr5 A 2.2 BS01 I4A A 1 F16 P38 S53 S55 A75 D76 C117 R126 Y128 F16 P38 S53 S55 A75 D76 C117 R126 Y128 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 ic50=0.069uM remove_due_to_license_issue IC50=69nM P15090 19217286 132 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 3frg A 1.7 BS01 SK4 A 1 M347 N395 F414 M431 Q443 F446 M195 N243 F262 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=3.98nM remove_due_to_license_issue IC50=3.98nM Q07343 19195882 1 ISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIPQA 3frz A 1.86 BS01 AG0 A 1 L419 R422 M423 H475 I482 R501 W528 L419 R422 M423 H475 I482 R501 W528 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 19209845 577 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQDLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3fsj X 1.37 BS01 D7K X 1 H281 T377 S378 F397 G401 L403 G427 D428 G429 S430 Y433 T457 Y458 G459 A460 L461 F464 V524 S525 H280 T376 S377 F396 G400 L402 G426 D427 G428 S429 Y432 T456 Y457 G458 A459 L460 F463 V523 S524 G25 S26 E28 E47 H70 L109 L110 T111 N112 H281 G401 D428 N455 T457 Y458 A460 L461 S525 G24 S25 E27 E46 H69 L108 L109 T110 N111 H280 G400 D427 N454 T456 Y457 A459 L460 S524 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 Kd=0.113mM remove_due_to_license_issue P20906 19320438 601 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTVS 3fsm A 1.6 BS01 2NC A 1 D25 G27 A28 D29 D30 I47 G48 I50 D129 G131 A132 D133 G152 D25 G27 A28 D29 D30 I47 G48 I50 D129 G131 A132 D133 G152 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=100nM remove_due_to_license_issue P03369 22158985 204 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNFCGGGGPQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3ft5 A 1.9 BS01 MO8 A 1 A55 M98 L107 T109 A40 M83 L92 T94 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=15uM remove_due_to_license_issue P07900 19301319 237 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3ft8 A 2.0 BS01 MOJ A 1 A55 G97 M98 L107 F138 Y139 W162 A40 G82 M83 L92 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.03uM remove_due_to_license_issue P07900 19301319 237 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3ftq A 2.9 BS02 GNP A 1 S46 G49 K50 S51 T52 T78 G104 K183 D185 V240 G241 R256 S13 G16 K17 S18 T19 T30 G56 K134 D136 V189 G190 R205 ? 0005525,0051301 remove_due_to_license_issue P42208 19805342 372 KGFEFTLMVVGESGLGKSTLINSLFKIERTVQIEASTVEIEERGVKLRLTVVDTPGYGDAINCRDCFKTIISYIDEQFERYLHDESGNRRHIIDNRVHCCFYFISPFGHGLKPLDVAFMKAIHNKVNIVPVIAKADTLTLKERERLKKRILDEIEEHSIKIYHLPDAEEDEDFKEQTRLLKASIPFSVVGSNQLIEAKGKKVRGRLYPWGVVEVENPEHNDFLKLRTMLITHMQDLQEVTQDLHYENFRSERLK 3fts A 2.33 BS02 STL A 1 Q136 A137 W311 D312 F314 V367 P374 A377 Y378 Q133 A134 W308 D309 F311 V364 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=212uM remove_due_to_license_issue IC50=366000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3ftu A 1.9 BS02 RE2 A 1 Q136 A137 W311 D312 F314 V367 P374 A377 Y378 P382 Q133 A134 W308 D309 F311 V364 P371 A374 Y375 P379 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=247uM remove_due_to_license_issue IC50=145000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3ftv A 1.7 BS02 11X A 1 Q136 F314 P374 A377 Y378 Q133 F311 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=1667uM remove_due_to_license_issue IC50=1667000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3ftw A 1.85 BS02 11X A 1 Q136 A137 F314 P374 D375 A377 Y378 Q133 A134 F311 P371 D372 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=1667000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fty A 2.15 BS02 3IP A 1 Q136 A137 W311 F314 V367 P374 A377 Y378 Q133 A134 W308 F311 V364 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=619uM remove_due_to_license_issue IC50=619000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3ftz A 2.0 BS02 848 A 1 Q136 A137 F314 V367 P374 A377 Y378 Q133 A134 F311 V364 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=>2000000nM P09960 19950900 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fu0 A 1.8 BS02 22F A 1 W311 F314 L369 P374 A377 Y378 W308 F311 L366 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=5308uM remove_due_to_license_issue IC50=5308000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fu3 A 2.0 BS02 92G A 1 L343 G347 K457 M462 E501 Q505 L340 G344 K454 M459 E498 Q502 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=1443uM remove_due_to_license_issue IC50=1443000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fu3 A 2.0 BS03 92G A 2 W311 F314 F362 K364 L365 V367 L369 P374 A377 Y378 P382 W308 F311 F359 K361 L362 V364 L366 P371 A374 Y375 P379 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=1443uM remove_due_to_license_issue IC50=1443000nM P09960 19618939 720 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fu5 A 2.3 BS02 492 A 1 Q136 A137 Y267 M270 E271 F314 P374 Y378 Q133 A134 Y264 M267 E268 F311 P371 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=75.2uM remove_due_to_license_issue IC50=75200nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fu6 A 2.05 BS02 80G A 1 Q136 A137 W311 F314 V367 P374 Y378 Q133 A134 W308 F311 V364 P371 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=106uM remove_due_to_license_issue IC50=106000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fuc A 1.45 BS01 9D9 A 1 S33 R84 H86 N115 A116 A117 G118 F200 E201 V217 M219 S220 T242 N243 S31 R74 H76 N105 A106 A107 G108 F190 E191 V207 M209 S210 T232 N233 S33 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S31 H76 Y78 E79 A106 M209 S210 N233 V235 H247 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Kd=190pM remove_due_to_license_issue IC50=10.2nM, Ki=1nM, Kd=0.1nM P55859 19944078 301 NGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGENPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESQGKANHEEVLEAGKQAAQKLEQFVSLLMASIPV 3fuc B 1.45 BS01 9D9 B 1 S33 R84 H86 N115 A116 A117 G118 F200 E201 V217 M219 S220 T242 N243 S31 R74 H76 N105 A106 A107 G108 F190 E191 V207 M209 S210 T232 N233 S33 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S31 H76 Y78 E79 A106 M209 S210 N233 V235 H247 2.4.2.1 0003824,0004731,0005737,0006139,0006166,0009116,0016757,0016763,0047975 Kd=190pM remove_due_to_license_issue IC50=10.2nM, Ki=1nM, Kd=0.1nM P55859 19944078 301 NGYTYEDYQDTAKWLLSHTEQRPQVAVICGSGLGGLVNKLTQAQTFDYSEIPNFPGRLVFGILNGRACVMMQGRFHMYEGYPFWKVTFPVRVFRLLGVETLVVTNAAGGLNPNFEVGDIMLIRDHINLPGFSGENPLRGPNEERFGVRFPAMSDAYDRDMRQKAHSTWKQMGEQRELQEGTYVMLGGPNFETVAECRLLRNLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESQGKANHEEVLEAGKQAAQKLEQFVSLLMASIPV 3fud A 2.2 BS02 692 A 1 R24 C25 T35 G36 E182 I188 R21 C22 T32 G33 E179 I185 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50>2000uM remove_due_to_license_issue IC50=1077000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fue A 2.38 BS02 11S A 1 W311 F314 V367 W308 F311 V364 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=1510uM remove_due_to_license_issue IC50=1510000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fuf A 2.6 BS02 14O A 1 W311 F314 P374 W308 F311 P371 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=>2000000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fuh A 1.8 BS02 5H1 A 1 W311 F314 P374 A377 Y378 W308 F311 P371 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 remove_due_to_license_issue IC50=>2000000nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fui A 2.2 BS02 812 A 1 Q134 Q136 Y267 G269 M270 F314 V367 P374 A377 Y378 P382 Q130 Q132 Y263 G265 M266 F310 V363 P370 A373 Y374 P378 E271 H295 E296 H299 E318 D375 Y383 E267 H291 E292 H295 E314 D371 Y379 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=0.157uM remove_due_to_license_issue IC50=157nM P09960 19618939 710 DTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3fuj A 1.9 BS02 00G A 1 Q136 A137 Y267 M270 W311 F314 P374 Y378 Q133 A134 Y264 M267 W308 F311 P371 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=234uM remove_due_to_license_issue P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fuk A 1.95 BS02 58Z A 1 Q136 A137 Y267 G269 M270 H295 E296 H299 W311 F314 E318 P374 Y378 Y383 Q134 A135 Y265 G267 M268 H293 E294 H297 W309 F312 E316 P372 Y376 Y381 E271 H295 E296 H299 E318 D375 Y383 E269 H293 E294 H297 E316 D373 Y381 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=966uM remove_due_to_license_issue IC50=966000nM P09960 19618939 710 IVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 3ful A 2.39 BS02 52D A 1 Q136 A137 Y267 M270 W311 F314 P374 A377 Y378 Q132 A133 Y263 M266 W307 F310 P370 A373 Y374 E271 H295 E296 H299 E318 D375 Y383 E267 H291 E292 H295 E314 D371 Y379 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=199uM remove_due_to_license_issue IC50=199000nM P09960 19950900 710 DTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fum A 2.15 BS02 80A A 1 Q136 A137 Y267 G269 M270 W311 F314 V367 L369 P374 A377 Y378 Y383 Q132 A133 Y263 G265 M266 W307 F310 V363 L365 P370 A373 Y374 Y379 E271 H295 E296 H299 E318 D375 Y383 E267 H291 E292 H295 E314 D371 Y379 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=170uM remove_due_to_license_issue IC50=202000nM P09960 19618939 710 DTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fun A 1.58 BS02 798 A 1 Q134 Q136 A137 Y267 G269 M270 W311 F314 K364 L365 V367 P374 A377 Y378 P382 Q131 Q133 A134 Y264 G266 M267 W308 F311 K361 L362 V364 P371 A374 Y375 P379 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=0.189uM remove_due_to_license_issue IC50=81nM P09960 19618939 710 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 3fup A 2.4 BS01 MI1 A 1 L855 G856 K857 G858 G861 V863 A880 Y931 L932 L983 G993 D994 L13 G14 K15 G16 G19 V21 A38 Y85 L86 L137 G147 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=21.7nM remove_due_to_license_issue IC50=77nM, EC50=93nM, Kd=5nM, Ki=0.700000nM O60674 19361440 1 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG 3fur A 2.3 BS02 Z12 A 1 F282 G284 C285 R288 Y327 L330 I341 F360 F363 M364 K367 H449 F61 G63 C64 R67 Y106 L109 I120 F139 F142 M143 K146 H228 ? 0003677,0004879,0005634,0006355 Ki=10nM remove_due_to_license_issue Ki=10.0nM, EC50=>500nM, IC50=17nM P37231 19452630 1 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3fuz A 1.65 BS01 GLU A 1 Y474 T503 R508 G673 S674 T675 E723 Y60 T89 R94 G139 S140 T141 E189 ? 0015276,0016020 remove_due_to_license_issue P39086 21893069 301 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3fv1 A 1.5 BS01 DYH A 1 E426 Y474 P501 L502 T503 R508 V670 G673 S674 T675 S706 M722 E723 S726 E12 Y60 P87 L88 T89 R94 V136 G139 S140 T141 S172 M188 E189 S192 ? 0015276,0016020 Ki=0.5nM remove_due_to_license_issue Ki=0.740000nM P39086 21893069 1 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3fv2 A 1.5 BS01 NDZ A 1 E426 Y474 P501 L502 T503 R508 V670 G673 S674 T675 M722 E723 S726 E12 Y60 P87 L88 T89 R94 V136 G139 S140 T141 M188 E189 S192 ? 0015276,0016020 Ki=7.7nM remove_due_to_license_issue P39086 21893069 791 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3fv7 A 2.0 BS01 MXS A 1 S81 Y112 W115 S128 V130 S219 G220 W221 R261 S50 Y81 W84 S97 V99 S188 G189 W190 R230 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 20822105 300 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 3fv8 A 2.28 BS01 JK3 A 1 I70 V78 M146 M149 D150 A151 N152 S193 N194 V196 L206 I25 V33 M101 M104 D105 A106 N107 S148 N149 V151 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T169 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 19433357 500 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAAAAAADEREHTIEEWKELIYKEVMN 3fvg A 1.5 BS01 MS8 A 1 E426 Y474 L502 T503 R508 G673 S674 T675 E723 S726 E12 Y60 L88 T89 R94 G139 S140 T141 E189 S192 ? 0015276,0016020 Ki=128nM remove_due_to_license_issue P39086 21893069 901 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3fvk A 1.5 BS01 8DX A 1 E426 Y474 L502 T503 R508 V670 G673 S674 T675 M722 E723 S726 E12 Y60 L88 T89 R94 V136 G139 S140 T141 M188 E189 S192 ? 0015276,0016020 Ki=1.5nM remove_due_to_license_issue P39086 21893069 1 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3fvl A 1.85 BS02 BHK A 1 E72 N144 R145 H196 Y248 A250 G253 E270 E72 N144 R145 H196 Y248 A250 G253 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 remove_due_to_license_issue P00730 311 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVEALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 3fvn A 1.5 BS01 9DX A 1 Y474 P501 L502 T503 R508 V670 G673 S674 T675 S706 M722 E723 Y60 P87 L88 T89 R94 V136 G139 S140 T141 S172 M188 E189 ? 0015276,0016020 Ki=169nM remove_due_to_license_issue P39086 21893069 1 ANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTALVRNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3fw3 A 1.72 BS02 ETS A 1 Q92 H94 H119 V121 L198 T199 T200 Q89 H91 H116 V118 L189 T190 T191 H64 H94 H96 E106 H119 T199 H64 H91 H93 E103 H116 T190 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 ic50=43nM remove_due_to_license_issue Ki=8500nM, IC50=32.0nM P22748 20363633 302 WCYEVQAESSNCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 3fw4 A 2.3 BS01 CAQ A 1 F123 K125 Y132 F133 K134 F119 K121 Y128 F129 K130 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 Kd=0.4nM remove_due_to_license_issue P80188 20581821 180 SDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 3fx6 A 1.851 BS02 BPX A 1 H69 R71 E72 R127 N144 R145 I243 Y248 E270 F279 H69 R71 E72 R127 N144 R145 I243 Y248 E270 F279 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=0.16uM remove_due_to_license_issue P00730 19646864 311 ARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVEALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 3fxb A 2.9 BS01 4CS A 1 E9 F66 R144 N184 P185 F188 F209 E9 F66 R144 N184 P185 F188 F209 ? 0042597,0055085 remove_due_to_license_issue Q5LUA7 19362561 401 DTWRYAFEEAMTDVQGVYAQKFKEEIEANSDHEIQLFPYGTLGESADIMEQTQDGILQFVDQSPGFTGSLIPEAQVFFVPYLLPTDQDHLARFFKESKAINDMFKPLYADQGLELLNMFPEGEVAMTTKTPVTTCSDLDEVKFRVMTNPLLVESYKAFGATPTPLPWGEVYGGLQTNVIQGQENPTFFLYSTKIYEVTDYITYAGHNNFTTAVMANKDFYDGLSAEDQQLVQNAALAAYDHTVVYQQQAADTELAKIMEAKPEMQVTVLTDEQRSCFKEAAAEVEAKFIEMTGDSGAAILKQMKADLAAT 3fxv A 2.26 BS02 643 A 1 M269 F288 L291 M294 A295 F333 R335 S336 I339 M369 Y373 M23 F42 L45 M48 A49 F87 R89 S90 I93 M118 Y122 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=94nM Q96RI1 19328688 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVHKFTPLLCEIWDV 3fxw A 2.0 BS01 F10 A 1 L50 L52 V58 A71 K73 C120 M121 E122 L173 T186 D187 L18 L20 V25 A38 K40 C87 M88 E89 L139 T152 D153 D166 K168 N171 D187 D132 K134 N137 D153 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1100nM Q16644 1 EPKKYAVTDDYQLSKQVLGLGVGKVLECFHRRTGQKCALKLLYDSPKARQEVDHHWQASGGPHIVCILDVYENMHHGKRCLLIIMECMEGGELFSRIQERDQAFTEREAAEIMRDIGTAIQFLHSHNIAHRDVKPENLLYTSKEKDAVLKLTDFGFAKEEKYDKSCDMWSLGVIMYILLCGFPPFGFPNPEWSEVSEDAKQLIRLLLKTDPTERLTITQFMNHPWINQSMVVPQTPLHTARVLQEDKDHWDEVKEEMTSALATMRVDYDQV 3fxz A 1.64 BS01 FLL A 1 I276 G277 Q278 V284 A297 R299 M344 E345 Y346 L347 A348 G350 D393 L396 I28 G29 Q30 V36 A49 R51 M96 E97 Y98 L99 A100 G102 D145 L148 D389 K391 D393 N394 D407 P416 T427 D141 K143 D145 N146 D159 P168 T179 2.7.11.1 0004672,0005524,0006468 ic50=130nM remove_due_to_license_issue Q13153 18973295 1 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT 3fy0 A 2.35 BS01 DW1 A 1 I276 G277 V284 A297 M344 E345 Y346 L347 G350 L396 I28 G29 V36 A49 M96 E97 Y98 L99 G102 L148 D389 K391 D393 N394 D407 P416 T427 D141 K143 D145 N146 D159 P168 T179 2.7.11.1 0004672,0005524,0006468 ic50=1090nM remove_due_to_license_issue Q13153 18973295 200 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT 3fyj X 3.8 BS01 B97 X 1 L70 G71 V78 C140 L141 D142 N191 T206 D207 L26 G27 V34 C96 L97 D98 N147 T162 D163 N191 D207 N147 D163 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=201nM, Ki=5.0nM P49137 19616942 372 QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSKYDKSCDMWSLGVIMYILLCGYPPFYSGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR 3fyk X 3.5 BS01 B98 X 1 G71 G73 A91 K93 M138 L141 T206 D207 G27 G29 A47 K49 M94 L97 T162 D163 N191 D207 N147 D163 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=5nM P49137 19616942 372 QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSKYDKSCDMWSLGVIMYILLCGYPPFYSGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR 3fyl A 1.63 BS01 dna C 0 C450 H451 Y452 K461 K465 K490 R510 C14 H15 Y16 K25 K29 K54 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3fyl A 1.63 BS02 dna D 0 S459 R466 R489 K490 R496 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3fyl B 1.63 BS01 dna C 0 S459 R466 R489 K490 R496 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKT 3fyl B 1.63 BS02 dna D 0 C450 H451 Y452 K461 K465 K490 R510 C14 H15 Y16 K25 K29 K54 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKT 3fyz A 2.1 BS01 MXC A 1 S81 Y112 S128 V130 S219 G220 W221 M223 R261 S50 Y81 S97 V99 S188 G189 W190 M192 R230 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 20822105 300 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 3fz1 A 1.9 BS01 B98 A 1 V18 A31 K33 F80 L83 N132 L134 D145 V18 A31 K33 F73 L76 N125 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T151 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 19616942 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3fzc A 2.0 BS01 MXF A 1 S81 Y112 M114 S128 V130 S219 G220 W221 R261 S50 Y81 M83 S97 V99 S188 G189 W190 R230 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 20822105 300 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 3fzn A 1.62 BS01 D7K A 1 H281 T377 S378 G401 L403 G427 D428 G429 S430 Y433 N455 T457 Y458 G459 A460 H280 T376 S377 G400 L402 G426 D427 G428 S429 Y432 N454 T456 Y457 G458 A459 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 19182954 601 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTV 3fzn A 1.62 BS04 D7K B 1 N23 P24 G25 S26 E47 H70 N22 P23 G24 S25 E46 H69 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 19182954 602 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTV 3fzn B 1.62 BS01 D7K A 1 N23 P24 G25 S26 E47 H70 N22 P23 G24 S25 E46 H69 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 19182954 601 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTV 3fzn B 1.62 BS02 D7K B 1 H281 T377 S378 G401 L403 G427 D428 G429 S430 Y433 N455 T457 Y458 G459 A460 L461 F464 H280 T376 S377 G400 L402 G426 D427 G428 S429 Y432 N454 T456 Y457 G458 A459 L460 F463 N23 G25 S26 N27 E28 E47 H70 L109 L110 T111 N112 Y160 P254 H281 S376 G401 L403 D428 N455 T457 Y458 A460 L461 F464 N22 G24 S25 N26 E27 E46 H69 L108 L109 T110 N111 Y159 P253 H280 S375 G400 L402 D427 N454 T456 Y457 A459 L460 F463 4.1.1.7 0000287,0003824,0003984,0009056,0016831,0018924,0019596,0019752,0030976,0046872,0050660,0050695 remove_due_to_license_issue P20906 19182954 602 ASVHGTTYELLRRQGIDTVFGNPGSNELPFLKDFPEDFRYILALQEACVVGIADGYAQASRKPAFINLHSAAGTGNAMGALSNAWNSHSPLIVTAGQQTRAMIGVEALLTNVDAANLPRPLVKWSYEPASAAEVPHAMSRAIHMASMAPQGPVYLSVPYDDWDKDADPQSHHLFDRHVSSSVRLNDQDLDILVKALNSASNPAIVLGPDVDAANANADCVMLAERLKAPVWVAPSAPRCPFPTRHPCFRGLMPAGIAAISQLLEGHDVVLVIGAPVFRYHQYDPGQYLKPGTRLISVTCDPLEAARAPMGDAIVADIGAMASALANLVEESSRQLPTAAPEPAKVDQDAGRLHPETVFDTLNDMAPENAIYLNESTSTTAQMWQRLNMRNPGSYYFCAAGGLGFALPAAIGVQLAEPERQVIAVIGDGSANYSISALWTAAQYNIPTIFVIMNNGTYGALRWFAGVLEAENVPGLDVPGIDFRALAKGYGVQALKADNLEQLKGSLQEALSAKGPVLIEVSTV 3fzr A 2.7 BS01 3JZ A 1 L431 G432 V439 M502 E503 L504 Y505 G508 E509 L556 L13 G14 V21 M84 E85 L86 Y87 G90 E91 L138 D549 A551 R553 N554 D567 L587 D131 A133 R135 N136 D149 L157 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=31nM Q14289 19244237 999 GIAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSRTRLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIAM 3fzs A 1.75 BS01 B96 A 1 E474 M478 V487 M502 L504 E509 L556 G566 D567 F568 E55 M59 V68 M83 L85 E90 L137 G147 D148 F149 D549 A551 R553 N554 D567 L587 D130 A132 R134 N135 D148 L151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.5uM remove_due_to_license_issue Kd=990nM, IC50=400nM Q14289 19244237 999 IAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA 3fzt A 1.95 BS01 4JZ A 1 K457 E474 M478 V487 L504 Y505 L556 G566 D567 F568 R572 K38 E55 M59 V68 L85 Y86 L137 G147 D148 F149 R153 D549 A551 R553 N554 D567 D576 L587 D130 A132 R134 N135 D148 D154 L156 2.7.10.2 0004672,0004713,0005524,0006468 ic50=637nM remove_due_to_license_issue Q14289 19244237 999 IAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSRDELPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA 3fzy A 1.95 BS01 IHP A 1 E3455 T3456 R3457 K3482 H3483 R3513 S3564 S3597 R3599 R3610 K3611 K3623 K3628 E37 T38 R39 K64 H65 R95 S146 S179 R181 R192 K193 K205 K210 2.3.1.-,3.4.22.-,6.3.2.- remove_due_to_license_issue Q9KS12 19620709 8000 ENLYFQSNALADGKILHNQNVNSWGPITVTPTTDGGETRFDGQIIVQMENDPVVAKAAANLAGKHAESSVVVQLDSDGNYRVVYGDPSKLDGKLRWQLVGHGRDHSETNNTRLSGYSADELAVKLAKFQQSFNQAENINNKPDHISIVGSSLVSDDKQKGFGHQFINAMDANGLRVDVSVRSSELAVDEAGRKHTKDANGDWVQKAENNKVSLSWD 3g08 A 1.6 BS01 FEE A 1 F10 C12 F70 Y73 S76 D80 W133 D153 T156 C168 F171 F4 C6 F64 Y67 S70 D74 W121 D141 T144 C156 F159 ? Kd=6.843nM remove_due_to_license_issue P11609 19949076 286 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMEDYPIEIQLSAGCEMYASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 3g0b A 2.25 BS01 T22 A 1 E205 E206 Y547 S630 Y631 V656 Y662 Y666 V711 E166 E167 Y508 S591 Y592 V617 Y623 Y627 V672 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.007uM remove_due_to_license_issue IC50=3.4nM, Kd=29nM P27487 21186796 800 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3g0c A 2.69 BS01 RUF A 1 E205 E206 Y547 S630 Y631 Y662 Y666 V711 H740 E162 E163 Y504 S587 Y588 Y619 Y623 V668 H697 Y547 S630 Y631 D708 H740 Y504 S587 Y588 D665 H697 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 21186796 800 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3g0d A 2.39 BS01 XIH A 1 R125 E205 E206 Y547 S630 Y631 Y662 Y666 V711 R82 E162 E163 Y504 S587 Y588 Y619 Y623 V668 Y547 S630 Y631 D708 H740 Y504 S587 Y588 D665 H697 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50~5nM remove_due_to_license_issue Ki=2nM P27487 21186796 800 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3g0e A 1.6 BS01 B49 A 1 L595 V603 A621 Y672 C673 C674 G676 L799 C809 F811 L54 V62 A80 Y131 C132 C133 G135 L200 C210 F212 D792 R796 N797 D810 D193 R197 N198 D211 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 Kd=20nM remove_due_to_license_issue Kd=0.370000nM, IC50=48nM, Ki=210nM P10721 19164557 9000 GPTYKYLQKPMYEVQWKVVEEINGNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFICSKTSPAIMEDDELALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISES 3g0f A 2.6 BS01 B49 A 1 L595 A621 Y672 C673 C674 G676 L799 C809 F811 L30 A56 Y107 C108 C109 G111 L160 C170 F172 D792 R796 N797 D810 D153 R157 N158 D171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue Kd=0.370000nM, IC50=48nM, Ki=210nM P10721 19164557 9001 NNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFLDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARHIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISE 3g0f B 2.6 BS01 B49 B 1 L595 V603 A621 Y672 C673 G676 L799 C809 F811 L32 V40 A58 Y109 C110 G113 L162 C172 F174 D792 R796 N797 D810 D155 R159 N160 D173 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue Kd=0.370000nM, IC50=48nM, Ki=210nM P10721 19164557 9001 NGNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFLDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARHIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISE 3g0g A 2.45 BS01 RUM A 1 R125 E205 E206 Y547 S630 Y631 Y662 Y666 R83 E163 E164 Y505 S588 Y589 Y620 Y624 Y547 S630 Y631 D708 H740 Y505 S588 Y589 D666 H698 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.005uM remove_due_to_license_issue IC50=5nM P27487 21186796 800 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3g0i A 2.1 BS01 VPR A 1 D192 L215 F244 Y251 Y314 T317 D190 L213 F242 Y249 Y312 T315 3.3.2.3 0003824,0004301,0016787,0016803,0097176 remove_due_to_license_issue Q9UR30 19469578 1 KAFAKFPSSASISPNPFTVSIPDEQLDDLKTLVRLSKIAPPTYESLQADGRFGITSEWLTTMREKWLSEFDWRPFEARLNSFPQFTTEIEGLTIHFAALFSEREDAVPIALLHGWPGSFVEFYPILQLFREEYTPETLPFHLVVPSLPGYTFSSGPPLDKDFGLMDNARVVDQLMKDLGFGSGYIIQGGDIGSFVGRLLGVGFDACKAVHLNLCAMRAPPEGPSIESLSAAEKEGIARMEKFMTDGLAYAMEHSTRPSTIGHVLSSSPIALLAWIGEKYLQWVDKPLPSETILEMVSLYWLTESFPRAIHTYRETTPMLQKELYIHKPFGFSFFPKDLCPVPRSWIATTGNLVFFRDHAEGGHFAALERPRELKTDLTAFVEQVW 3g0w A 1.95 BS01 LGB A 1 L701 L704 N705 L707 W741 M742 M745 M749 F764 M780 F876 T877 L32 L35 N36 L38 W72 M73 M76 M80 F95 M111 F207 T208 ? Ki=0.3nM remove_due_to_license_issue P15207 19351168 1 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 3g15 A 1.7 BS03 HC6 A 1 D306 Y333 Y354 F361 W420 W423 E434 F435 Y440 D203 Y230 Y251 F258 W317 W320 E331 F332 Y337 2.7.1.32,2.7.1.82 remove_due_to_license_issue P35790 20299452 603 EQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 3g1d A 1.5 BS01 U A 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D13 K35 D63 K65 M119 S120 P173 Q178 G195 R196 K42 D70 K72 D75 K35 D63 K65 D68 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue O26232 19435314 229 VMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1d A 1.5 BS02 U B 1 D75 I76 T79 D68 I69 T72 K42 D70 K72 D75 K35 D63 K65 D68 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue O26232 19435314 229 VMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1d B 1.5 BS01 U A 1 D75 I76 T79 D67 I68 T71 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1d B 1.5 BS02 U B 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D12 K34 D62 K64 M118 S119 P172 Q177 G194 R195 K42 D70 K72 D75 K34 D62 K64 D67 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue O26232 19435314 229 MDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3g1m A 1.7 BS01 RF3 A 1 L87 M102 G106 F110 M142 Y148 T149 N176 N179 E180 L66 M81 G85 F89 M121 Y127 T128 N155 N158 E159 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.522uM remove_due_to_license_issue IC50=500nM P9WMC1 19412174 217 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGEN 3g1v A 1.3 BS01 5FU A 1 D20 K42 L123 M126 S127 P180 Q185 G202 R203 D10 K32 L113 M116 S117 P170 Q175 G192 R193 K42 G70 K72 D75 K32 G60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=645000nM O26232 19435314 501 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIAGFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIK 3g1v A 1.3 BS02 5FU B 1 D75 I76 T79 D65 I66 T69 K42 G70 K72 D75 K32 G60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=645000nM O26232 19435314 502 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIAGFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIK 3g1v B 1.3 BS01 5FU A 1 D75 I76 T79 D65 I66 T69 K42 G70 K72 D75 K32 G60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=645000nM O26232 19435314 501 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIAGFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIK 3g1v B 1.3 BS02 5FU B 1 D20 K42 L123 M126 S127 P180 Q185 G202 R203 D10 K32 L113 M116 S117 P170 Q175 G192 R193 K42 G70 K72 D75 K32 G60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 remove_due_to_license_issue Ki=645000nM O26232 19435314 502 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIAGFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIK 3g2h A 2.03 BS01 KOT A 1 G135 L136 D339 H377 T378 N484 E672 S674 G675 G124 L125 D310 H348 T349 N455 E643 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=151.3uM remove_due_to_license_issue Ki=151000nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3g2i A 2.0 BS01 RUG A 1 G135 N284 D339 H377 T378 N484 E672 S674 G675 G124 N267 D313 H351 T352 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=13.7uM remove_due_to_license_issue Ki=26000nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3g2j A 2.14 BS01 9GP A 1 G135 L136 N284 H377 T378 N484 E672 S674 G675 G124 L125 N267 H351 T352 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=18000nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3g2k A 2.0 BS01 SKY A 1 G135 L136 N284 F285 H341 H377 T378 N484 E672 A673 S674 G675 G124 L125 N267 F268 H315 H351 T352 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=16.1uM remove_due_to_license_issue Ki=16000nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3g2l A 2.3 BS01 LEW A 1 G135 L136 D283 N284 H377 A383 N484 E672 A673 S674 G675 G124 L125 D266 N267 H351 A357 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=135.9uM remove_due_to_license_issue Ki=136000nM, IC50=625000nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3g2n A 2.1 BS01 OAK A 1 G135 L136 N284 H377 N484 E672 S674 G675 G124 L125 N270 H357 N464 E652 S654 G655 H377 K568 R569 K574 T676 K680 H357 K548 R549 K554 T656 K660 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=81000nM P00489 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3g2y A 1.31 BS01 GF4 A 1 N104 Y105 S130 T235 G236 S237 N79 Y80 S105 T210 G211 S212 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9L5C8 19305397 1 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g2z A 1.5 BS01 GZ2 A 1 Y105 S130 T235 G236 S237 Y79 S104 T209 G210 S211 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=4.4mM remove_due_to_license_issue Q9L5C8 19305397 1 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g30 A 1.8 BS01 G30 A 1 S70 S130 N132 N170 S237 G238 D240 S44 S104 N106 N144 S211 G212 D213 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3.1mM remove_due_to_license_issue Q9L5C8 19305397 1 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g30 A 1.8 BS02 G30 A 2 T149 A150 R153 T123 A124 R127 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3.1mM remove_due_to_license_issue Q9L5C8 19305397 2 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g31 A 1.7 BS01 GF1 A 1 E37 K38 G42 R61 E12 K13 G17 R35 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.3mM remove_due_to_license_issue Q9L5C8 19305397 2 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g31 A 1.7 BS02 GF1 A 2 S70 N104 Y105 S130 N132 G236 S237 S44 N78 Y79 S104 N106 G210 S211 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.3mM remove_due_to_license_issue Q9L5C8 19305397 4 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g32 A 1.31 BS01 3G3 A 1 Y105 S130 T235 G236 S237 Y79 S104 T209 G210 S211 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.194mM remove_due_to_license_issue Q9L5C8 19305397 1 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g34 A 1.31 BS01 1CE A 1 Y105 S130 T235 G236 S237 S274 Y79 S104 T209 G210 S211 S246 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.1mM remove_due_to_license_issue Q9L5C8 19305397 1 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g35 A 1.41 BS01 F13 A 1 N104 Y105 S130 N132 P167 N170 T235 G236 S237 D240 N76 Y77 S102 N104 P139 N142 T207 G208 S209 D211 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.021mM remove_due_to_license_issue Q9L5C8 19305397 1 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g35 A 1.41 BS02 F13 A 2 K82 L142 G147 A154 K54 L114 G119 A126 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.021mM remove_due_to_license_issue Q9L5C8 19305397 3 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 3g3d A 1.7 BS01 5FU A 1 S68 D70 H94 K125 M182 S183 P228 Q241 Y243 G261 R262 S34 D36 H60 K91 M148 S149 P194 Q207 Y209 G227 R228 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue Ki=98000nM P11172 19260677 3000 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3g3d A 1.7 BS02 5FU B 1 D128 I129 T132 D94 I95 T98 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue Ki=98000nM P11172 19260677 3000 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3g3d B 1.7 BS01 5FU A 1 D128 I129 T132 D97 I98 T101 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue Ki=98000nM P11172 19260677 3000 APKELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3g3d B 1.7 BS02 5FU B 1 S68 D70 H94 K125 M182 S183 P228 Q241 Y243 G261 R262 S37 D39 H63 K94 M151 S152 P197 Q210 Y212 G230 R231 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue Ki=98000nM P11172 19260677 3000 APKELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3g3m A 1.4 BS01 5FU A 1 S68 D70 H94 K125 M182 S183 P228 Q241 Y243 G261 R262 S35 D37 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 remove_due_to_license_issue Ki=98000nM P11172 19260677 1000 KELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3g3n A 2.4 BS01 TC8 A 1 I323 I363 V380 F384 L401 F416 I185 I225 V242 F246 L263 F278 3.1.4.53 0004114,0007165,0008081 ic50=0.51uM remove_due_to_license_issue IC50=510nM Q13946 19350606 3 DYNGQAKCMLEKVGNWNFDIFLFDRLTNGNSLVSLTFHLFSLHGLIEYFHLDMMKLRRFLVMIQEDYHSQNPYHNAVHAADVTQAMHCYLKEPKLANSVTPWDILLSLIAAATHDLDHPGVNQPFLIKTNHYLATLYKNTSVLENHHWRSAVGLLRESGLFSHLPLESRQQMETQIGALILATDISRQNEYLSLFRSHLDRGDLCLEDTRHRHLVLQMALKCADICNPCRTWELSKQWSEKVTEEFFHQGDIEKKYHLGVSPLCDRHTESIANIQIGFMTYLVEPLFTEWARFSNTRLSQTMLGHVGLNKASWKGLQR 3g3r A 2.0 BS01 ANP A 1 R264 R266 K281 K294 Y359 R361 E426 S457 K458 R70 R72 K87 K100 Y165 R167 E232 S263 K264 2.7.4.1 Kd=0.33uM remove_due_to_license_issue P47075 19390046 1000 VRQTTKYWVHPDNITELKLIILKHLPVLVFNTNKEFEREDSAITSIYFDNENLDLYYGRLRKDEGAEAHRLRWYGGMSTDTIFVERKTHREDWTGEKSVKARFALKERHVNDFLKGKYTVDQVFAKMRKEGKKPMNEIENLEALASEIQYVMLKKKLRPVVRSFYNRTAFQLPGDARVRISLDTELTMVREDNFDGVDRTHKNWRRTDIGVDWPFKQLDDKDICRFPYAVLEVKLQTQLGQEPPEWVRELVGSHLVEPVPKFSKFIHGVATLLNDKVDSIPFWLPQ 3g42 A 2.1 BS01 792 A 1 T347 G349 H405 E406 H409 H415 A439 V440 T127 G129 H185 E186 H189 H195 A219 V220 3.4.24.86 0004222,0006508,0008237 ic50=0.14uM remove_due_to_license_issue IC50=140nM P78536 19410464 1 MKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYVGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3g45 A 2.63 BS02 988 A 1 Y274 H406 I582 M603 Q615 F618 Y28 H119 I295 M316 Q328 F331 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=70nM Q07343 20037581 901 SNKFKRMLNRELTHLSEMSRSGNQVSEYISNTFLDTSISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPQ 3g4f A 2.651 BS01 FPF A 1 D307 R448 D451 E455 Y527 Y535 V536 D279 R420 D423 E427 Y493 Y496 V497 R270 W279 I300 D307 D311 T407 C408 G409 R448 D451 E455 Y527 R242 W251 I272 D279 D283 T379 C380 G381 R420 D423 E427 Y493 4.2.3.13 0000287,0010333,0016102,0016114,0016829,0046872,0047461 remove_due_to_license_issue Q39761 19489610 801 ADFQPSIWGDLFLNCPDDAETEKRHQQLKEEVRKMIVAPMANSTQKLAFIDSVQRLGVSYHFTKEIEDELENIYHNNNDAENDLYTTSIRFRLLREHGYNVSCDVFNKFKDEQGNFKSSVTSDVRGLLELYQASYLRVHGEDILDEAISFTTHHLSLAVASLDHPLSEEVSHALKQSIRRGLPRVEARHYLSVYQDESHNKALLEFAKIDFNMLQFLHRKELSEICRWWKDLDFQRKLPYARDRVVEGYFWISGVYFEPQYSLGRKMLTKVIAMASIVDDTYDSYATYEELIPYTNAIERWDIKCIDEIPEYMKPSYKALLDVYEEMVQLVAEHGRQYRVEYAKNAMIRLAQSYLVEAKWTLQNYKPSFEEFKANALPTCGYAMLAITSFVGMGDIVTPETFKWAASDPKIIQASTIICRFMDDVAEHKFDCSAIECYMEEYGVTAQEAYDVFNKHVESAWKDLNQEFLKPTEMPTEVLNRSLNLARVMDVLYREYVGKAAKGGITSLLIEPIAL 3g4g A 2.3 BS02 D71 A 1 F196 H326 T499 I502 F506 M523 S534 Q535 F538 F6 H85 T258 I261 F265 M282 S293 Q294 F297 3.1.4.53 0004114,0007165,0008081 ic50=19nM remove_due_to_license_issue Q08499 20037581 901 NQVSEFISNTFLDEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQA 3g4i A 1.9 BS02 D71 A 1 H326 T499 I502 M503 M523 S534 Q535 F538 H79 T252 I255 M256 M276 S287 Q288 F291 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 20037581 901 FGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 3g4k A 1.95 BS02 ROL A 1 Y325 H326 T499 I502 M503 F506 Q535 F538 Y78 H79 T252 I255 M256 F259 Q288 F291 3.1.4.53 0004114,0007165,0008081 ic50=288nM remove_due_to_license_issue Q08499 20037581 901 FGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 3g4l A 2.5 BS02 ROF A 1 T437 M439 D484 L485 N487 Y495 W498 T499 I502 M523 S534 Q535 F538 T189 M191 D234 L235 N237 Y245 W248 T249 I252 M273 S284 Q285 F288 3.1.4.53 0004114,0007165,0008081 ic50=5.8nM remove_due_to_license_issue IC50=0.400000nM Q08499 20037581 901 GVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 3g58 A 2.05 BS02 988 A 1 I502 F506 M523 S534 Q535 F538 I259 F263 M280 S291 Q292 F295 3.1.4.53 0004114,0007165,0008081 ic50=5nM remove_due_to_license_issue Q08499 20037581 901 SIPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 3g5d A 2.2 BS01 1N1 A 1 L273 V281 A293 K295 E310 M314 I336 T338 Y340 M341 S342 G344 L393 L17 V22 A34 K36 E46 M50 I72 T74 Y76 M77 S78 G80 L129 D386 R388 A390 N391 D404 F424 D122 R124 A126 N127 D140 F147 2.7.10.2 0004672,0004713,0005524,0006468 Kd=11nM remove_due_to_license_issue Kd=11nM, IC50=0.4nM P00523 19462975 1 KDAWEIPRESLRLEVKLGQGEVWMGTWNGTTRVAIKTLSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3g5k A 1.7 BS01 BB2 A 1 C50 V51 G52 Q57 P111 E112 G113 C114 E115 W149 R152 H156 E157 H160 C48 V49 G50 Q55 P109 E110 G111 C112 E113 W147 R150 H154 E155 H158 G52 Q57 C114 E115 H156 E157 H160 G50 Q55 C112 E113 H154 E155 H158 3.5.1.88 0042586 remove_due_to_license_issue IC50=1.5nM, Ki=0.300000nM Q9HBH1 19236878 1001 HMSFSHVCQVGDPVLRGVAAPVERAQLGGPELQRLTQRLVQVMRRRRCVGLSAPQLGVPRQVLALELPEALCRECPPRQRALRQMEPFPLRVFVNPSLRVLDSRLVTFPEGCESVAGFLACVPRFQAVQISGLDPNGEQVVWQASGWAARIIQHEMDHLQGCLFIDKMDSRTFTNVYWMKVND 3g6g A 2.31 BS01 G6G A 1 V281 A293 E310 M314 T338 Y340 M341 G344 V383 H384 L393 A403 D404 F405 V26 A38 E55 M59 T83 Y85 M86 G89 V128 H129 L138 A148 D149 F150 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F155 2.7.10.2 0004672,0004713,0005524,0006468 ic50=2.8nM remove_due_to_license_issue P00523 19276351 1 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3g6h B 2.35 BS01 G6H B 1 L273 V281 A293 K295 E310 M314 I338 Y340 M341 G344 H384 L393 A403 D404 F405 L16 V24 A36 K38 E53 M57 I81 Y83 M84 G87 H127 L136 A146 D147 F148 D386 R388 A390 N391 D404 D129 R131 A133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4.6nM remove_due_to_license_issue P00523 19276351 1 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVIEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3g6m A 1.65 BS01 CFF A 1 F74 W134 D172 E174 M240 Y242 W381 F36 W96 D134 E136 M202 Y204 W343 D170 D172 E174 Y242 D132 D134 E136 Y204 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0008843,0016798 Ki=19.7mM remove_due_to_license_issue A9LI60 20829286 1 TGSINAVYFTNWGIYGRNFQPADLQASKILHVLYSFMNLRVDGTVYSGDTYADLEKHYSDDSWNDIGTNAYGCVKQLYKLKKANRSLKIMLSIGGWTWSTNFPAAASTEATRATFAKTAVEFMKDWGFDGIDVDWEYPASETDANNMVLLLQRVRQELDSYSATYANGYHFQLSIAAPAGPSHYNVLKLAQLGSVLDNINLMAYDYAGSWDSVSGHQTNLYPSTSNPSSTPFSTKAAVDAYIAAGVPASKIILGMPIYGRAFVGTDGPGKPYSTIGEGSWESGIWDYKVLPKAGATVITDSAAGATYSYDSSSRTMISYDTPDMVRTKVSYAKGLGLGGSMFWEASADKTGSDSLIGTALSSMGSHDSTQNCLSYPNSKFDNIKNSLS 3g6m A 1.65 BS02 CFF A 2 W134 D243 W248 W96 D205 W210 D170 D172 E174 Y242 D132 D134 E136 Y204 3.2.1.14 0000272,0004553,0004568,0005576,0005975,0006032,0008061,0008843,0016798 Ki=19.7mM remove_due_to_license_issue A9LI60 20829286 427 TGSINAVYFTNWGIYGRNFQPADLQASKILHVLYSFMNLRVDGTVYSGDTYADLEKHYSDDSWNDIGTNAYGCVKQLYKLKKANRSLKIMLSIGGWTWSTNFPAAASTEATRATFAKTAVEFMKDWGFDGIDVDWEYPASETDANNMVLLLQRVRQELDSYSATYANGYHFQLSIAAPAGPSHYNVLKLAQLGSVLDNINLMAYDYAGSWDSVSGHQTNLYPSTSNPSSTPFSTKAAVDAYIAAGVPASKIILGMPIYGRAFVGTDGPGKPYSTIGEGSWESGIWDYKVLPKAGATVITDSAAGATYSYDSSSRTMISYDTPDMVRTKVSYAKGLGLGGSMFWEASADKTGSDSLIGTALSSMGSHDSTQNCLSYPNSKFDNIKNSLS 3g6p A 1.985 BS01 dna C 0 C450 H451 Y452 K461 K465 R510 C14 H15 Y16 K25 K29 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 18 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3g6p A 1.985 BS02 dna D 0 S459 R466 R489 R496 S23 R30 R53 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 18 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3g6p B 1.985 BS01 dna C 0 S459 V462 R466 R489 K490 R496 S23 V26 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 18 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKKIK 3g6p B 1.985 BS02 dna D 0 C450 H451 Y452 K461 K465 R510 C14 H15 Y16 K25 K29 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 18 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKKIK 3g6z A 2.0 BS01 A7T A 1 D38 W45 V46 H61 L81 V111 M114 F119 F124 D125 D226 D38 W45 V46 H61 L81 V111 M114 F119 F124 D125 D222 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D222 A225 3.4.23.15 0004190,0006508 ic50=0.2nM remove_due_to_license_issue IC50=19nM P00797 19358611 342 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALARH 3g70 A 2.0 BS01 A5T A 1 D38 G40 L81 M114 F119 A122 F124 D125 V127 D226 G228 D35 G37 L78 M111 F116 A119 F121 D122 V124 D219 G221 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=0.4nM remove_due_to_license_issue IC50=36nM P00797 19358611 342 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALARH 3g72 A 1.9 BS01 A6T A 1 D38 G40 W45 P47 H61 L81 Y83 M114 P118 F119 A122 F124 D125 V127 D226 G228 D35 G37 W42 P44 H58 L78 Y80 M111 P115 F116 A119 F121 D122 V124 D219 G221 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=0.8nM remove_due_to_license_issue IC50=88nM P00797 19358611 343 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3g73 A 2.21 BS01 dna C 0 R236 S240 Y241 K278 N283 S284 H287 R5 S9 Y10 K47 N52 S53 H56 ? 0000086,0003677,0003700,0006355,0043565 remove_due_to_license_issue Q08050 20360045 1 ~ 21 SVSERPPYSYMAMIQFAINSTERKRMTLKDIYTWIEDHFPYFKHIAKPGWKNSIRHNLSLHDMFVRETSANGKVSFWTIHPSANRYLTLD 3g73 A 2.21 BS02 dna D 0 L259 K260 R286 H287 S290 R297 W308 L28 K29 R55 H56 S59 R66 W77 ? 0000086,0003677,0003700,0006355,0043565 remove_due_to_license_issue Q08050 20360045 1 ~ 21 SVSERPPYSYMAMIQFAINSTERKRMTLKDIYTWIEDHFPYFKHIAKPGWKNSIRHNLSLHDMFVRETSANGKVSFWTIHPSANRYLTLD 3g73 B 2.21 BS01 dna C 0 L259 R286 H287 S290 S306 W308 L26 R53 H54 S57 S73 W75 ? 0000086,0003677,0003700,0006355,0043565 remove_due_to_license_issue Q08050 20360045 1 ~ 21 SERPPYSYMAMIQFAINSTERKRMTLKDIYTWIEDHFPYFKHIAKPGWKNSIRHNLSLHDMFVRETSANGKVSFWTIHPSANRYLTLDQVFKPLD 3g73 B 2.21 BS02 dna D 0 R236 S240 Y241 K278 H287 R3 S7 Y8 K45 H54 ? 0000086,0003677,0003700,0006355,0043565 remove_due_to_license_issue Q08050 20360045 1 ~ 21 SERPPYSYMAMIQFAINSTERKRMTLKDIYTWIEDHFPYFKHIAKPGWKNSIRHNLSLHDMFVRETSANGKVSFWTIHPSANRYLTLDQVFKPLD 3g76 A 3.0 BS02 CZ3 A 1 L292 V298 G306 L307 T308 W310 E314 Q319 W323 L41 V47 G55 L56 T57 W59 E63 Q68 W72 2.3.2.27 remove_due_to_license_issue P98170 19393243 600 NSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSL 3g86 A 2.2 BS01 T18 A 1 F193 P197 S288 N291 D318 C366 S368 G410 N411 M414 Y415 I447 Y448 G449 S556 F188 P192 S283 N286 D313 C361 S363 G405 N406 M409 Y410 I442 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.005uM remove_due_to_license_issue P26663 19457662 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3g8e A 3.0 BS01 IS1 A 1 F193 R196 V242 I309 R311 R349 I351 G353 E376 S379 F173 R176 V222 I289 R291 R329 I331 G333 E356 S359 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 19533035 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 3g8e B 3.0 BS01 IS1 A 1 D16 Y18 D8 Y10 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 19533035 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 3g8e B 3.0 BS02 IS1 B 1 Y188 F193 D219 V242 A244 S275 I309 R311 D313 R349 E376 N377 S379 Y168 F173 D199 V222 A224 S255 I289 R291 D293 R329 E356 N357 S359 2.4.2.12 0000166,0001774,0005125,0005576,0005615,0005634,0005737,0007165,0007565,0007623,0008286,0009435,0010507,0014070,0014916,0016757,0019363,0032922,0042802,0045944,0047280,0048511,0048661,0051770,0060612,0071456,0071479,1901363,1904646,1905377,2000773 remove_due_to_license_issue Q80Z29 19533035 502 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKEVYREHFQDDVFNERGWNYILEKYDGHLPIEVKAVPEGSVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGIALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTEAPLIIRPDSGNPLDTVLKVLDILGKKFPVSENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKKWSIENVSFGSGGALLQKLTRDLLNCSFKCSYVVTNGLGVNVFKDPVADPNKRSKKGRLSLHRTPAGTFVTLEEGKGDLEEYGHDLLHTVFKNGKVTKSYSFDEVRKNAQLN 3g8i A 2.2 BS02 RO7 A 1 V255 F273 C276 S280 Y314 L321 M330 V332 M355 K358 H440 Y464 V48 F59 C62 S66 Y100 L107 M116 V118 M141 K144 H226 Y250 ? 0003677,0004879,0005634,0006355 ic50=0.038uM remove_due_to_license_issue IC50=38nM, EC50=103nM Q07869 19349176 1 DLKSLAKRIYEAYLKNFNMNKVKARVILSPPFVIHDMETLCMAEKTLVAKLKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANLDLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFDFAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDIFLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDMY 3g8o A 1.9 BS01 30X A 1 L718 N719 L721 M756 M759 V760 L763 L797 L887 Y890 C891 T894 L36 N37 L39 M74 M77 V78 L81 L115 L205 Y208 C209 T212 ? ic50=125nM remove_due_to_license_issue IC50=125nM, EC50=1300nM P06401 19595590 1 QLIPPLINLLMSIEPDVIYAGHDNTKDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 3g8u A 1.9 BS01 dna D 0 G458 S459 R466 R489 R496 G22 S23 R30 R53 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKK 3g8u A 1.9 BS02 dna C 0 C450 H451 Y452 K465 R510 C14 H15 Y16 K29 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKK 3g8u B 1.9 BS01 dna D 0 C450 H451 Y452 K461 K465 C12 H13 Y14 K23 K27 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 MCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3g8u B 1.9 BS02 dna C 0 S459 R466 R489 K490 S21 R28 R51 K52 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 MCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3g90 X 2.4 BS01 J72 X 1 I70 V78 E147 M149 D150 A151 N152 V196 L206 I25 V31 E100 M102 D103 A104 N105 V149 L159 N194 D207 N147 D160 2.7.11.24 0004672,0004707,0005524,0006468 Ki=0.44uM remove_due_to_license_issue P53779 19361991 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIQLDEREHTIEEWKELIYKEVMN 3g99 A 1.81 BS01 dna D 0 S459 R466 R489 K490 R496 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKK 3g99 A 1.81 BS02 dna C 0 C450 H451 Y452 K461 K465 K490 R510 C14 H15 Y16 K25 K29 K54 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKK 3g99 B 1.81 BS01 dna D 0 C450 Y452 K461 C13 Y15 K24 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 HMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3g99 B 1.81 BS02 dna C 0 G458 S459 R466 R489 R496 G21 S22 R29 R52 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 HMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 3g9e A 2.3 BS02 RO7 A 1 G284 C285 S289 H323 L330 I341 K367 H449 Y473 G65 C66 S70 H104 L111 I122 K148 H230 Y254 ? 0003677,0004879,0005634,0006355 ic50=0.019uM remove_due_to_license_issue IC50=19nM, EC50=21nM P37231 19349176 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3g9l X 2.2 BS01 J67 X 1 I70 V78 K93 I124 M146 E147 L148 M149 D150 A151 N152 V196 I25 V28 K43 I74 M96 E97 L98 M99 D100 A101 N102 V146 N194 D207 N144 D157 2.7.11.24 0004672,0004707,0005524,0006468 Ki=0.74uM remove_due_to_license_issue Ki=740nM P53779 19361991 1 NQFYSVEVGDSTFTVLKRYQNLKPIGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLSFMMTVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIDEREHTIEEWKELIYKEVMN 3g9m A 1.61 BS01 dna D 0 S459 R466 R489 K490 R496 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKK 3g9m A 1.61 BS02 dna C 0 C450 H451 Y452 K461 K465 K490 R510 C14 H15 Y16 K25 K29 K54 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 SHMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKK 3g9m B 1.61 BS01 dna D 0 C450 H451 Y452 K461 K465 K490 C13 H14 Y15 K24 K28 K53 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 HMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKK 3g9m B 1.61 BS02 dna C 0 S459 R466 R489 K490 R496 S22 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06536 19372434 1 ~ 16 HMCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKK 3g9n A 2.8 BS01 J88 A 1 Q31 V34 A47 M102 L104 M105 D106 A107 N108 Q111 V152 L162 Q30 V33 A46 M101 L103 M104 D105 A106 N107 Q110 V151 L161 D145 K147 N150 D163 T182 D144 K146 N149 D162 T176 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue Ki=1800nM P53779 19361991 359 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPKQLDEREHTIEEWKELIYKEVMN 3ga5 A 1.87 BS01 RGG A 1 D14 F16 N91 K92 T110 H152 D154 R158 W183 N211 D236 N256 Q261 D12 F14 N89 K90 T108 H150 D152 R156 W181 N209 D234 N254 Q259 ? 0006935,0030246,0030288,0042597,0046872 Kd=3.2uM remove_due_to_license_issue P23905 19292879 400 TRIGVTIYKYDDNFMSVVRKAIEKDGKSAPDVQLLMNDSQNDQSKQNDQIDVLLAKGVKALAINLVDPAAAGTVIEKARGQNVPVVFFNKEPSRKALDSYDKAYYVGTDSKESGVIQGDLIAKHWQANQGWDLNKDGKIQYVLLKGEPGHPDAEARTTYVVKELNDKGIQTEQLALDTAMWDTAQAKDKMDAWLSGPNANKIEVVIANNDAMAMGAVEALKAHNKSSIPVFGVDALPEALALVKSGAMAGTVLNDANNQAKATFDLAKNLAEGKGAADGTSWKIENKIVRVPYVGVDKDNLSEFT 3gb2 A 2.4 BS01 G3B A 1 I62 F67 A83 K85 D133 Y134 V135 R141 L188 D200 I28 F33 A49 K51 D94 Y95 V96 R102 L149 D161 D181 K183 N186 D200 S219 D142 K144 N147 D161 S180 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=34nM remove_due_to_license_issue P49841 19775160 999 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 3gba A 1.35 BS01 DYH A 1 E13 Y61 P88 L89 T90 R95 V137 G140 S141 T142 S173 M189 E190 S193 E13 Y61 P88 L89 T90 R95 V137 G140 S141 T142 S173 M189 E190 S193 ? 0015276,0016020 Ki=0.848nM remove_due_to_license_issue P22756 19297335 258 GANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3gbb A 2.1 BS01 MS8 A 1 E13 Y61 P88 L89 T90 R95 G140 S141 T142 E190 S193 E11 Y59 P86 L87 T88 R93 G138 S139 T140 E188 S191 ? 0015276,0016020 Ki=126nM remove_due_to_license_issue P22756 19297335 258 NRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3gbe A 1.7 BS01 NOJ A 1 D75 Y78 H118 F178 R212 D214 H341 D342 R429 D60 Y63 H103 F163 R197 D199 H326 D327 R414 D113 R212 D214 E268 H341 D342 D98 R197 D199 E253 H326 D327 5.4.99.11 0004556,0005975,0009313,0050006 Ki=10uM remove_due_to_license_issue D0VX20 19427862 8000 TIPKWWKEAVFYQVYPRSFKDTNGDGIGDINGIIEKLDYLKALGIDAIWINPHYDSPNTDNGYDIRDYRKIMKEYGTMEDFDRLISEMKKRNMRLMIDVVINHTSDQNEWFVKSKSSKDNPYRGYYFWKDAKEGQAPNNYPSFFGGSAWQKDEKTNQYYLHYFAKQQPDLNWDNPKVRQDLYAMLRFWLDKGVSGLRFDTVATYSKIPDFPNLTQQQLKNFAAEYTKGPNIHRYVNEMNKEVLSHYDIATAGEIFGVPLDQSIKFFDRRRDELNIAFTFDLIRLDRDSDQRWRRKDWKLSQFRQIIDNVDRTAGEYGWNAFFLDNHDNPRAVSHFGDDRPQWREPSAKALATLTLTQRATPFIYQGSELGMTNYPFKAIDEFDDIEVKGFWHDYVETGKVKADEFLQNVRLTSRDNSRTPFQWDGSKNAGFTSGKPWFKVNPNYQEINAVSQVTQPDSVFNYYRQLIKIRHDIPALTYGTYTDLDPANDSVYAYTRSLGAEKYLVVVNFKEQMMRYKLPDNLSIEKVIIDSNSKNVVKKNDSLLELKPWQSGVYKLNQ 3gc4 A 1.8 BS01 AAQ A 1 N70 D102 Y106 D156 C158 G229 G230 A232 M260 G261 D280 N60 D92 Y96 D127 C129 G200 G201 A203 M231 G232 D251 D102 D280 C318 C320 C323 H349 D92 D251 C289 C291 C294 H320 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=25nM remove_due_to_license_issue P28720 19894214 395 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQSEEGVTFMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 3gc5 A 1.4 BS02 2MQ A 1 D102 Y106 D156 C158 G229 G230 L231 A232 M260 G261 D280 D92 Y96 D141 C143 G214 G215 L216 A217 M245 G246 D265 D102 D280 C318 C320 C323 H349 D92 D265 C303 C305 C308 H334 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=55nM remove_due_to_license_issue P28720 19894214 400 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSLTKQSEEGVTFKSSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 3gc7 A 1.8 BS01 B45 A 1 Y35 A51 V52 K53 L104 T106 L108 M109 G110 A111 L167 D168 Y32 A48 V49 K50 L101 T103 L105 M106 G107 A108 L164 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.4nM remove_due_to_license_issue IC50=5.6nM Q16539 19622861 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3gcp A 2.25 BS01 SB2 A 1 Y35 A51 K53 L104 V105 T106 L108 M109 F169 L171 Y32 A48 K50 L101 V102 T103 L105 M106 F166 L168 D150 K152 N155 D168 T185 D147 K149 N152 D165 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=15nM remove_due_to_license_issue Q16539 19572644 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLCTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPP 3gcq A 2.0 BS01 1BU A 1 V30 A51 R70 E71 M78 I84 T106 L108 M109 H148 L167 D168 V27 A45 R64 E65 M72 I78 T100 L102 M103 H142 L161 D162 D150 K152 N155 D168 T185 D144 K146 N149 D162 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=342nM remove_due_to_license_issue IC50=800nM Q16539 19572644 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPPLDQ 3gcs A 2.1 BS01 BAX A 1 A51 E71 L74 I84 L108 M109 I141 I166 L167 D168 F169 A44 E64 L67 I77 L101 M102 I134 I159 L160 D161 F162 D150 K152 N155 D168 T185 D143 K145 N148 D161 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=56nM remove_due_to_license_issue Kd=370nM, IC50=400nM Q16539 19572644 401 RPTFYRQELNKTIWEVPERYQNLSPVGYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPP 3gcu A 2.1 BS01 R48 A 1 A51 K53 E71 L75 T106 M109 L167 D168 F169 A48 K50 E68 L72 T103 M106 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T172 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=370nM Q16539 19572644 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3gcv A 2.3 BS01 SS6 A 1 A51 K53 E71 I84 T106 L108 M109 H148 L167 D168 F169 C172 A46 K48 E66 I79 T101 L103 M104 H143 L162 D163 F164 C167 D150 K152 N155 D168 T185 D145 K147 N150 D163 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=74nM remove_due_to_license_issue IC50=420nM Q16539 19572644 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLCVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPPL 3gdt A 1.6 BS01 UP6 A 1 K59 H61 K93 S154 P202 Y217 R235 K57 H59 K91 S152 P200 Y215 R233 4.1.1.23 0004590,0005829,0006207,0006221,0006222,0016831,0044205,0055086,0072528 remove_due_to_license_issue Ki=64nM P03962 19435314 301 KATYKERAATHPSPVAAKLFNIMHEKQTNLCASLDVRTTKELLELVEALGPKICLLKTHVDILTDFSMEGTVKPLKALSAKYNFLLFENRKFADIGNTVKLQYSAGVYRIAEWADITNAHGVVGPGIVSGLKQAAEEVTKEPRGLLMLAELSCKGSLATGEYTKGTVDIAKSDKDFVIGFIAQRDMGGRDEGYDWLIMTPGVGLDDKGDALGQQYRTVDDVVSTGSDIIIVGRGLFAKGRDAKVEGERYRKAGWEAYLRR 3gdt D 1.6 BS01 UP6 D 1 K59 K93 S154 G203 G234 R235 K57 K91 S152 G201 G220 R221 4.1.1.23 0004590,0005829,0006207,0006221,0006222,0016831,0044205,0055086,0072528 remove_due_to_license_issue Ki=64nM P03962 19435314 301 KATYKERAATHPSPVAAKLFNIMHEKQTNLCASLDVRTTKELLELVEALGPKICLLKTHVDILTDFSMEGTVKPLKALSAKYNFLLFENRKFADIGNTVKLQYSAGVYRIAEWADITNAHGVVGPGIVSGLKQAAEEVTKEPRGLLMLAELSCKGSLATGEYTKGTVDIAKSDKDFVIGFIAQRDMGGRDEGYDWLIMTPGVGRTVDDVVSTGSDIIIVGRGLFAKGRDAKVEGERYRKAGWEAYLRRCGQQ 3ge7 A 1.5 BS02 AFQ A 1 L68 N70 D102 Y106 D156 C158 G229 G230 A232 M260 G261 D280 L58 N60 D92 Y96 D132 C134 G205 G206 A208 M236 G237 D256 D102 D280 C318 C320 C323 H349 D92 D256 C294 C296 C299 H325 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=2nM remove_due_to_license_issue P28720 19894214 390 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMTKQSEEGVTFMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 3gen A 1.6 BS01 B43 A 1 L408 V416 A428 K430 M449 T474 Y476 M477 L528 S538 D539 F540 L17 V22 A34 K36 M55 T80 Y82 M83 L134 S144 D145 F146 D521 A523 R525 N526 D539 F559 D127 A129 R131 N132 D145 F165 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=310nM Q06187 20052711 1 YGSWEIDPKDLTFLKELGFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 3gep A 2.6 BS01 24H A 1 K68 D107 T110 I135 D137 T138 G139 T141 K165 F186 V187 K66 D102 T105 I130 D132 T133 G134 T136 K160 F181 V182 E133 D134 D137 F186 R199 E128 D129 D132 F181 R194 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 19527031 218 RSPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSDQSTGDIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 3gfe A 2.1 BS01 P37 A 1 A51 K53 E71 T106 M109 G110 L167 D168 F169 L171 A51 K53 E71 T106 M109 G110 L167 D168 F169 L171 D150 K152 N155 D168 T185 D150 K152 N155 D168 T185 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=3.2nM remove_due_to_license_issue IC50=3.2nM Q16539 19574047 361 MSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3gfw A 2.74 BS01 S22 A 1 I531 G532 A551 E603 G605 D608 S611 A651 L654 I663 I17 G18 A37 E89 G91 D94 S97 A137 L140 I149 D647 K649 N652 D664 T686 D133 K135 N138 D150 T156 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=367nM P33981 20383151 1 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIAGTVNYMPPEAIKDSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 3ggc B 2.78 BS01 H26 B 1 I135 D137 T138 G139 T141 K165 F186 V187 I131 D133 T134 G135 T137 K161 F182 V183 E133 D134 D137 F186 R199 E129 D130 D133 F182 R195 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 19527031 218 RSPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSYCNDQSTGDIKVIGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 3ggj A 2.6 BS01 25H A 1 D137 T138 G139 T141 K165 F186 V187 D134 T135 G136 T138 K162 F183 V184 E133 D134 D137 F186 R199 E130 D131 D134 F183 R196 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 19527031 218 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSYCNDQSTGDIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 3ggu A 1.8 BS01 017 B 1 D25 G27 A28 D30 P81 T82 D25 G27 A28 D30 P81 T82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 19535439 201 PQITLWQRPIVTVKIEGQLKEALLDTGADDTVFEELTLSGRWKPRLIGGIGGFVRVRQYDQVPIEICGHKVIDTVLVGPTPTNVIGRNVMTQLGCTLNF 3ggu B 1.8 BS01 017 B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=170pM remove_due_to_license_issue P03367 19535439 201 PQITLWQRPIVTVKIEGQLKEALLDTGADDTVFEELTLSGRWKPRLIGGIGGFVRVRQYDQVPIEICGHKVIDTVLVGPTPTNVIGRNVMTQLGCTLNF 3ggv A 3.09 BS01 GGV B 1 R8 D25 G27 A28 D29 G49 P81 R8 D25 G27 A28 D29 G49 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 19323562 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ggv B 3.09 BS01 GGV B 1 R8 D25 G27 A28 D29 P81 V82 I84 R8 D25 G27 A28 D29 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 19323562 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gi4 A 1.85 BS01 K60 A 1 D25 G27 D29 G48 I50 D25 G27 D29 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.016nM remove_due_to_license_issue P03369 20237088 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gi4 B 1.85 BS01 K60 A 1 R8 D25 A28 D30 P81 V82 R8 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 20237088 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gi5 A 1.8 BS01 K62 A 1 D25 G27 D29 I50 D25 G27 D29 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.006nM remove_due_to_license_issue P03369 20237088 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gi5 B 1.8 BS01 K62 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 20237088 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gi6 A 1.84 BS01 D78 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.006nM remove_due_to_license_issue P03369 20237088 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gi6 B 1.84 BS01 D78 A 1 D25 A28 D30 I84 D25 A28 D30 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 20237088 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3gib A 2.4 BS01 rna H 0 Y25 G29 I30 K31 L32 Q33 N48 Q52 T61 Y20 G24 I25 K26 L27 Q28 N43 Q47 T56 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 19889981 1 ~ 9 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPSRPVS 3gib B 2.4 BS01 rna H 0 Y25 G29 I30 K31 L32 Q33 N48 Q52 T61 Y22 G26 I27 K28 L29 Q30 N45 Q49 T58 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 19889981 1 ~ 9 GQSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPSRPV 3gib C 2.4 BS01 rna H 0 Y25 G29 I30 K31 L32 Q33 Q52 T61 Y20 G24 I25 K26 L27 Q28 Q47 T56 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 19889981 1 ~ 9 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPSRP 3gjd A 2.0 BS03 LEU A 1 A22 G24 L25 G26 Y108 F253 S256 F259 S355 A18 G20 L21 G22 Y104 F247 S250 F253 S349 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 19307590 519 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3gjw A 2.3 BS01 GJW A 1 H201 G202 Y235 S243 Y246 H201 G202 Y235 S243 Y246 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 Ki=0.005uM remove_due_to_license_issue EC50=6nM, Ki=5nM P09874 19553114 351 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 3gk1 A 2.1 BS03 32A A 1 A83 F87 A83 F87 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=80uM remove_due_to_license_issue P02638 19469484 94 SELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFF 3gk2 A 1.984 BS03 27A A 1 H42 F43 H42 F43 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=2mM remove_due_to_license_issue P02638 19469484 94 SELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFF 3gk4 X 1.9 BS03 53A X 1 H42 F43 L44 E45 H43 F44 L45 E46 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=120uM remove_due_to_license_issue P02638 19469484 94 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 3gkz A 1.9 BS01 B40 A 1 Y41 Y55 Y58 F106 E114 Y175 Y177 H230 W232 F237 Y33 Y47 Y50 F98 E106 Y158 Y160 H213 W215 F220 Kd=10nM remove_due_to_license_issue 19760665 500 EVQLQESGPSLVKPSQTLSLTCSVTGDSVTSGYWSWIRQFPGNKLDYMGYISYRGSTYYNPSLKSRISITRDTSKNQVYLQLKSVSSEDTATYYCSYFDSDDYAMEYWGQGTSVTVSSGGGGSQIVLTQSPAIMSASPGEKVTLTCSASSSVSSSHLYWYQQKPGSSPKLWIYSTSNLASGVPARFSGSGSGTSYSLTISSMEAEDAASYFCHQWSSFPFTFGSGTKLEIKRA 3glf A 3.388 BS01 dna K 0 F215 V244 R248 R252 K313 F215 V244 R248 R252 K313 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28630 19450514 2 ~ 15 MIRLYPEQLRAQLNEGLRAAYLLLGNDPLLLQESQDAVRQVAAAQGFEEHHTFSIDPNTDWNAIFSLCQAMSLFASRQTLLLLLPENGPNAAINEQLLTLTGLLHDDLLLIVRGNKLSKAQENAAWFTALANRSVQVTCQTPEQAQLPRWVAARAKQLNLELDDAANQVLCYCYEGNLLALAQALERLSLLWPDGKLTLPRVEQAVNDAAHFTPFHWVDALLMGKSKRALHILQQLRLEGSEPVILLRTLQRELLLLVNLKRQSAHTPLRALFDKHRVWQNRRGMMGEALNRLSQTQLRQAVQLLTRTELTLKQDYGQSVWAELEGLSLLLCH 3glf B 3.388 BS01 dna K 0 T99 K100 V101 S132 H134 T95 K96 V97 S128 H130 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 VLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 3glf C 3.388 BS01 dna K 0 T99 K100 V101 S132 H134 T96 K97 V98 S129 H131 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 QVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 3glf D 3.388 BS01 dna K 0 K100 V101 S132 H134 K99 V100 S131 H133 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 SYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRM 3glf E 3.388 BS01 dna K 0 G89 V90 R94 T121 G89 V90 R94 T121 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0008408,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28631 19450514 2 ~ 15 MRWYPWLRPDFEKLVASYQAGRGHHALLIQALPGMGDDALIYALSRYLLCQQPQGHKSCGHCRGCQLMQAGTHPDYYTLAPEKGKNTLGVDAVREVTEKLNEHARLGGAKVVWVTDAALLTDAAANALLKTLEEPPAETWFFLATREPERLLATLRSRCRLHYLAPPPEQYAVTWLSREVTMSQDALLAALRLSAGSPGAALALFQGDNWQARETLCQALAYSVPSGDWYSLLAALNHEQAPARLHWLATLLMDALKRHHGAAQVTNVDVPGLVAELANHLSPSRLQAILGDVCHIREQLMSVTGINRELLITDLLLRIEHYLQPGVVLPVPHL 3glf F 3.388 BS01 dna M 0 F215 V244 I245 R248 R252 K313 F215 V244 I245 R248 R252 K313 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28630 19450514 2 ~ 15 MIRLYPEQLRAQLNEGLRAAYLLLGNDPLLLQESQDAVRQVAAAQGFEEHHTFSIDPNTDWNAIFSLCQAMSLFASRQTLLLLLPENGPNAAINEQLLTLTGLLHDDLLLIVRGNKLSKAQENAAWFTALANRSVQVTCQTPEQAQLPRWVAARAKQLNLELDDAANQVLCYCYEGNLLALAQALERLSLLWPDGKLTLPRVEQAVNDAAHFTPFHWVDALLMGKSKRALHILQQLRLEGSEPVILLRTLQRELLLLVNLKRQSAHTPLRALFDKHRVWQNRRGMMGEALNRLSQTQLRQAVQLLTRTELTLKQDYGQSVWAELEGLSLLLCH 3glf G 3.388 BS01 dna M 0 T99 K100 V101 S132 H134 T109 K110 V111 S142 H144 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 GLEVLFQGPHMSYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 3glf H 3.388 BS01 dna M 0 T99 K100 V101 S132 H134 T96 K97 V98 S129 H131 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 QVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 3glf I 3.388 BS01 dna M 0 T99 K100 V101 R105 S132 H134 T98 K99 V100 R104 S131 H133 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 SYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRM 3glf J 3.388 BS01 dna M 0 G89 V90 R94 T121 G89 V90 R94 T121 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0008408,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28631 19450514 2 ~ 15 MRWYPWLRPDFEKLVASYQAGRGHHALLIQALPGMGDDALIYALSRYLLCQQPQGHKSCGHCRGCQLMQAGTHPDYYTLAPEKGKNTLGVDAVREVTEKLNEHARLGGAKVVWVTDAALLTDAAANALLKTLEEPPAETWFFLATREPERLLATLRSRCRLHYLAPPPEQYAVTWLSREVTMSQDALLAALRLSAGSPGAALALFQGDNWQARETLCQALAYSVPSGDWYSLLAALNHEQAPARLHWLATLLMDALKRHHGAAQVTNVDVPGLVAELANHLSPSRLQAILGDVCHIREQLMSVTGINRELLITDLLLRIEHYLQPGVVLPVPHL 3gli A 3.5 BS01 dna K 0 F215 V244 I245 R248 R252 F215 V244 I245 R248 R252 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28630 19450514 2 ~ 15 MIRLYPEQLRAQLNEGLRAAYLLLGNDPLLLQESQDAVRQVAAAQGFEEHHTFSIDPNTDWNAIFSLCQAMSLFASRQTLLLLLPENGPNAAINEQLLTLTGLLHDDLLLIVRGNKLSKAQENAAWFTALANRSVQVTCQTPEQAQLPRWVAARAKQLNLELDDAANQVLCYCYEGNLLALAQALERLSLLWPDGKLTLPRVEQAVNDAAHFTPFHWVDALLMGKSKRALHILQQLRLEGSEPVILLRTLQRELLLLVNLKRQSAHTPLRALFDKHRVWQNRRGMMGEALNRLSQTQLRQAVQLLTRTELTLKQDYGQSVWAELEGLSLLLCH 3gli B 3.5 BS01 dna K 0 K100 V101 S132 H134 K96 V97 S128 H130 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 VLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRM 3gli C 3.5 BS01 dna K 0 T99 K100 V101 S132 H134 T96 K97 V98 S129 H131 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 QVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 3gli D 3.5 BS01 dna K 0 K100 V101 S132 H134 K99 V100 S131 H133 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 SYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRM 3gli E 3.5 BS01 dna K 0 K85 G89 V90 R94 T121 K85 G89 V90 R94 T121 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0008408,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28631 19450514 2 ~ 15 MRWYPWLRPDFEKLVASYQAGRGHHALLIQALPGMGDDALIYALSRYLLCQQPQGHKSCGHCRGCQLMQAGTHPDYYTLAPEKGKNTLGVDAVREVTEKLNEHARLGGAKVVWVTDAALLTDAAANALLKTLEEPPAETWFFLATREPERLLATLRSRCRLHYLAPPPEQYAVTWLSREVTMSQDALLAALRLSAGSPGAALALFQGDNWQARETLCQALAYSVPSGDWYSLLAALNHEQAPARLHWLATLLMDALKRHHGAAQVTNVDVPGLVAELANHLSPSRLQAILGDVCHIREQLMSVTGINRELLITDLLLRIEHYLQPGVVLPVPHL 3gli F 3.5 BS01 dna M 0 F215 E242 V244 I245 R248 R252 K313 F215 E242 V244 I245 R248 R252 K313 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28630 19450514 2 ~ 15 MIRLYPEQLRAQLNEGLRAAYLLLGNDPLLLQESQDAVRQVAAAQGFEEHHTFSIDPNTDWNAIFSLCQAMSLFASRQTLLLLLPENGPNAAINEQLLTLTGLLHDDLLLIVRGNKLSKAQENAAWFTALANRSVQVTCQTPEQAQLPRWVAARAKQLNLELDDAANQVLCYCYEGNLLALAQALERLSLLWPDGKLTLPRVEQAVNDAAHFTPFHWVDALLMGKSKRALHILQQLRLEGSEPVILLRTLQRELLLLVNLKRQSAHTPLRALFDKHRVWQNRRGMMGEALNRLSQTQLRQAVQLLTRTELTLKQDYGQSVWAELEGLSLLLCHK 3gli G 3.5 BS01 dna M 0 T99 K100 V101 S132 H134 T109 K110 V111 S142 H144 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 GLEVLFQGPHMSYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRM 3gli H 3.5 BS01 dna M 0 T99 K100 V101 S132 H134 T96 K97 V98 S129 H131 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 QVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRMPLPEP 3gli I 3.5 BS01 dna M 0 K100 V101 S132 H134 K99 V100 S131 H133 2.7.7.7 0003677,0003887,0005524,0006260,0009360,0016887 remove_due_to_license_issue P06710 19450514 2 ~ 15 SYQVLARKWRPQTFADVVGQEHVLTALANGLSLGRIHHAYLFSGTRGVGKTSIARLLAKGLNCETGITATPCGVCDNCREIEQGRFVDLIEIDAASRTKVEDTRDLLDNVQYAPARGRFKVYLIDEVHMLSRHSFNALLKTLEEPPEHVKFLLATTDPQKLPVTILSRCLQFHLKALDVEQIRHQLEHILNEEHIAHEPRALQLLARAAEGSLRDALSLTDQAIASGDGQVSTQAVSAMLGTLDDDQALSLVEAMVEANGERVMALINEAAARGIEWEALLVEMLGLLHRIAMVQLSPAALGNDMAAIELRMRELARTIPPTDIQLYYQTLLIGRKELPYAPDRRMGVEMTLLRALAFHPRM 3gli J 3.5 BS01 dna M 0 K85 V90 R94 T121 K85 V90 R94 T121 2.7.7.7 0003677,0003689,0003887,0005515,0006260,0006261,0008408,0009360,0030894,0034061,0043846,0071897 remove_due_to_license_issue P28631 19450514 2 ~ 15 MRWYPWLRPDFEKLVASYQAGRGHHALLIQALPGMGDDALIYALSRYLLCQQPQGHKSCGHCRGCQLMQAGTHPDYYTLAPEKGKNTLGVDAVREVTEKLNEHARLGGAKVVWVTDAALLTDAAANALLKTLEEPPAETWFFLATREPERLLATLRSRCRLHYLAPPPEQYAVTWLSREVTMSQDALLAALRLSAGSPGAALALFQGDNWQARETLCQALAYSVPSGDWYSLLAALNHEQAPARLHWLATLLMDALKRHHGAAQVTNVDVPGLVAELANHLSPSRLQAILGDVCHIREQLMSVTGINRELLITDLLLRIEHYLQPGVVLPVPHL 3gm0 A 2.4 BS01 B41 A 1 Y41 Y55 Y58 F106 E114 Y175 H230 W232 F237 Y33 Y47 Y50 F98 E106 Y162 H217 W219 F224 Kd=17nM remove_due_to_license_issue 19760665 600 EVQLQESGPSLVKPSQTLSLTCSVTGDSVTSGYWSWIRQFPGNKLDYMGYISYRGSTYYNPSLKSRISITRDTSKNQVYLQLKSVSSEDTATYYCSYFDSDDYAMEYWGQGTSVTVSGGGGSGGGGSQIVLTQSPAIMSASPGEKVTLTCSASSSVSSSHLYWYQQKPGSSPKLWIYSTSNLASGVPARFSGSGSGTSYSLTISSMEAEDAASYFCHQWSSFPFTFGSGTKLEIKRA 3gn7 A 2.5 BS01 3GN A 1 H201 G202 Y235 F236 S243 Y246 E327 H201 G202 Y235 F236 S243 Y246 E327 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Ki=4nM P09874 900 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 3gnv A 2.75 BS01 XNZ A 1 P197 R200 C366 S367 S368 L384 N411 M414 Y415 Y448 P197 R200 C366 S367 S368 L384 N411 M414 Y415 Y448 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 19507864 579 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3gnw A 2.39 BS01 XNC A 1 P197 R200 C366 S367 S368 N411 M414 Y415 I447 Y448 G449 S556 P194 R197 C363 S364 S365 N408 M411 Y412 I444 Y445 G446 S553 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.79nM remove_due_to_license_issue O92972 19507864 579 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3gol A 2.85 BS01 XND A 1 R200 C366 S367 N411 M414 Y415 Y448 R197 C363 S364 N408 M411 Y412 Y445 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 19342234 579 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASLSGWFVAGYSGGDIYHS 3gp0 A 1.9 BS01 NIL A 1 A51 K53 R67 E71 L75 T106 L108 M109 L167 D168 F169 A43 K45 R59 E63 L67 T98 L100 M101 L159 D160 F161 D150 K152 N155 D168 T185 D142 K144 N147 D160 T170 2.7.11.24 0000165,0001649,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005829,0006468,0007254,0010628,0031098,0032735,0033554,0035556,0038066,0045648,0051149,0051403,0060038,0060043,0060044,0060348,0071347,0071493,0090398,0098586,0106310 remove_due_to_license_issue Kd=36nM Q15759 1 MRAGFYRQELNKTVWEVPQRLQGLRPVGSVCSAYDARLRQKVAVKKLSRPFQSLIHARRTYRELRLLKHLKHENVIGLLDVFTPATSIEDFSEVYLVTTLMGADLNNIVKCQALSDEHVQFLVYQLLRGLKYIHSAGIIHRDLKPSNVAVNEDCELRILDFGEEMGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLQGKALFPGSDYIDQLKRIMEVVGTPSPEVLAKISSEHARTYIQSLPPMPQKDLSSIFRGANPLAIDLLGRMLVLDSDQRVSAAEALAHAYFSQYHDPEDEPEAEPYDESVEAKERTLEEWKELTYQEVLSF 3gpe A 2.0 BS05 PT5 A 1 Y195 K197 K209 K211 N253 Y40 K42 K54 K56 N98 2.7.11.13 remove_due_to_license_issue P05696 19346474 600 TEKRGRIYLKAEVTDEKLHVTVRDAKNLIPMDPNGLSDPYVKLKLIPDPKNESKQKTKTIRSTLNPQWNESFTFKLKPSDKDRRLSVEIWDWDRTTRNDFMGSLSFGVSELMKMPASGWYKLLNQEEGEYYNVPIPE 3gpj H 2.7 BS01 SY2 H 1 T1 T21 Q22 K33 G47 A49 T1 T21 Q22 K33 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 19359491 7710 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 3gpj I 2.7 BS01 SY2 H 1 D114 I116 C118 D124 I126 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 19359491 7710 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 3gpo A 1.9 BS01 APR A 1 D10 I11 N24 G30 D31 G32 V33 C34 L108 S110 T111 G112 V113 Y114 R144 D12 I13 N26 G32 D33 G34 V35 C36 L110 S112 T113 G114 V115 Y116 R146 2.1.1.-,2.7.7.-,2.7.7.19,2.7.7.48,3.1.3.84,3.4.22.-,3.6.1.15,3.6.1.74,3.6.4.13 Kd=5uM remove_due_to_license_issue Q8JUX6 19386706 161 HHAPSYRVKRMDIAKNDEECVVNAANPRGLPGDGVCKAVYKKWPESFKNSATPVGTAKTVMCGTYPVIHAVGPNFSNYSESEGDRELAAAYREVAKEVTRLGVNSVAIPLLSTGVYSGGKDRLTQSLNHLFTAMDSTDADVVIYCRDKEWEKKISEAIQMRT 3gqo A 2.6 BS01 APR A 1 G9 D10 I11 A22 A23 N24 G30 G31 G32 V33 C34 L108 S110 T111 G112 I113 F114 R144 G10 D11 I12 A23 A24 N25 G31 G32 G33 V34 C35 L109 S111 T112 G113 I114 F115 R145 2.1.1.-,2.7.7.-,2.7.7.19,2.7.7.48,3.1.3.84,3.4.22.-,3.6.1.15,3.6.1.74,3.6.4.13 remove_due_to_license_issue P36328 19386706 167 KAPSYHVVRGDIATATEGVIINAANSKGQPGGGVCGALYKKFPESFDLQPIEVGKARLVKGAAKHIIHAVGPNFNKVSEVEGDKQLAEAYESIAKIVNDNNYKSVAIPLLSTGIFSGNKDRLTQSLNHLLTALDTTDADVAIYCRDKKWEMTLKEAVARRE 3gqz A 1.8 BS01 GF7 A 1 L119 Y150 K290 A292 L293 L116 Y147 K287 A289 L290 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=6.7mM remove_due_to_license_issue P00811 19416920 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gr2 A 1.8 BS01 GF4 A 1 N152 V211 S212 Y221 T319 G320 N149 V208 S209 Y218 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=3mM remove_due_to_license_issue P00811 19416920 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3grj A 2.49 BS01 G14 A 1 S166 G167 L168 S163 G164 L165 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K309 A312 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1mM remove_due_to_license_issue P00811 19416920 365 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNLAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gs6 A 2.3 BS01 NP6 A 1 I30 D62 R130 K160 H161 H165 M204 M246 I30 D62 R130 K160 H161 H165 M201 M243 3.2.1.52 0004553,0004563,0005737,0005975,0008360,0009252,0009254,0016231,0016798,0046677,0051301,0071555 remove_due_to_license_issue Q9KU37 19499593 341 MGPLWLDVAGYELSAEDRAILAHPTVGGVILFGRNYHDNQQLLALNKAIRQAAARPILIGVDQEGGRVQRFREGFSRIPPAQYYARAENGVELAEQGGWLMAAELIAHDVDLSFAPVLDMGFACKAIGNRAFGEDVQTVLKHSSAFLRGMKAVGMATTGKHFPGHGAVIHLETPYDERETIAQDMAIFRAQIEAGVLDAMMPAHVVYPHYDAQPASGSSYWLKQVLREELGFKGIVFSDDLSMVMGGPVERSHQALVAGCDMILICNKREAAVEVLDNLPIMEVPQAEALLKKQQFSYSELKRLERWQQASANMQRLIEQFS 3gs7 A 1.8 BS01 8BD A 1 K15 A108 A109 K6 A99 A100 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 19621084 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3gs7 B 1.8 BS01 8BD B 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 19621084 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVT 3gsg A 2.1 BS01 GF1 A 1 S64 N152 Y221 G317 A318 S61 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=2mM remove_due_to_license_issue P00811 19416920 366 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gsm A 2.4 BS01 VPU A 1 D62 R130 K160 H161 M204 D62 R130 K160 H161 M203 3.2.1.52 0004553,0004563,0005737,0005975,0008360,0009252,0009254,0016231,0016798,0046677,0051301,0071555 remove_due_to_license_issue Q9KU37 19499593 341 MGPLWLDVAGYELSAEDRAILAHPTVGGVILFGRNYHDNQQLLALNKAIRQAAARPILIGVDQEGGRVQRFREGFSRIPPAQYYARAENGVELAEQGGWLMAAELIAHDVDLSFAPVLDMGFACKAIGNRAFGEDVQTVLKHSSAFLRGMKAVGMATTGKHFPGHGAVIADHLETPYDERETIAQDMAIFRAQIEAGVLDAMMPAHVVYPHYDAQPASGSSYWLKQVLREELGFKGIVFSDDLSMVMGGPVERSHQALVAGCDMILICNKREAAVEVLDNLPIMEVPQAEALLKKQQFSYSELKRLERWQQASANMQRLIEQFS 3gss A 1.9 BS01 GSH A 1 F8 R13 W38 K44 Q51 L52 Q64 S65 F7 R12 W37 K43 Q50 L51 Q63 S64 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 9012673 211 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3gss A 1.9 BS02 EAA A 1 F8 V10 Y108 F7 V9 Y107 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue IC50=2.6e+4nM P09211 9012673 212 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3gss B 1.9 BS01 GSH B 1 F8 R13 W38 K44 Q51 L52 Q64 S65 F7 R12 W37 K43 Q50 L51 Q63 S64 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 9012673 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3gss B 1.9 BS02 EAA B 1 F8 V10 Y108 F7 V9 Y107 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue IC50=2.6e+4nM P09211 9012673 211 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3gst A 1.9 BS01 GPR A 1 Y6 W7 L12 R42 W45 K49 N58 L59 Q71 S72 R107 I111 S209 Y6 W7 L12 R42 W45 K49 N58 L59 Q71 S72 R107 I111 S209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005496,0005576,0005737,0005829,0006629,0006693,0006749,0007608,0009410,0010038,0010288,0016151,0016740,0018916,0019899,0019901,0032991,0042178,0042802,0042803,0043200,0043295,0045471,0048678,0051122,0070458,0071466,1901687 Ki=0.19uM remove_due_to_license_issue P04905 8110735 223 PMILGYWNVRGLTHPIRLLLEYTDSSYEEKRYAMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGSRKITQSNAIMRYLARKHHLCGETEEERIRADIVENQVMDNRMQLIMLCYNPDFEKQKPEFLKTIPEKMKLYSEFLGKRPWFAGDKVTYVDFLAYDILDQYHIFEPKCLDAFPNLKDFLARFEGLKKISAYMKSSRYLSTPIFSKLAQWSNK 3gst B 1.9 BS01 GPR B 1 Y6 W7 G11 L12 R42 W45 K49 N58 L59 Q71 S72 I111 Y6 W7 G11 L12 R42 W45 K49 N58 L59 Q71 S72 I111 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005496,0005576,0005737,0005829,0006629,0006693,0006749,0007608,0009410,0010038,0010288,0016151,0016740,0018916,0019899,0019901,0032991,0042178,0042802,0042803,0043200,0043295,0045471,0048678,0051122,0070458,0071466,1901687 Ki=0.19uM remove_due_to_license_issue P04905 8110735 220 PMILGYWNVRGLTHPIRLLLEYTDSSYEEKRYAMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGSRKITQSNAIMRYLARKHHLCGETEEERIRADIVENQVMDNRMQLIMLCYNPDFEKQKPEFLKTIPEKMKLYSEFLGKRPWFAGDKVTYVDFLAYDILDQYHIFEPKCLDAFPNLKDFLARFEGLKKISAYMKSSRYLSTPIFSKLAQWSNK 3gt9 A 1.7 BS02 516 A 1 K121 R123 G130 L131 Q132 W134 D138 E143 W147 K44 R46 G53 L54 Q55 W57 D61 E66 W70 F81 F4 2.3.2.27 remove_due_to_license_issue Ki=110000nM Q96CA5 20189383 1 GPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQDKVRCFFCYGGLQSWKRGDDPWTEHAKWFPGCQFLLRSKGQEYINNIH 3gta A 1.7 BS02 851 A 1 K121 R123 G130 L131 Q132 W134 D138 E143 W147 K44 R46 G53 L54 Q55 W57 D61 E66 W70 F81 F4 2.3.2.27 remove_due_to_license_issue Ki=53000nM Q96CA5 20189383 1 GPAFPGMGSEELRLASFYDWPLTAEVPPELLAAAGFFHTGHQDKVRCFFCYGGLQSWKRGDDPWTEHAKWFPGCQFLLRSKGQEYINNIH 3gtc A 1.9 BS01 GTC A 1 H210 V211 S212 Y221 T319 G320 H207 V208 S209 Y218 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=4.5mM remove_due_to_license_issue P00811 19416920 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gtc A 1.9 BS02 GTC A 2 S64 A318 T319 S61 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=4.5mM remove_due_to_license_issue P00811 19416920 364 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gur A 2.5 BS01 BYG A 1 Y6 W7 G11 L12 W45 K49 N58 L59 Q71 S72 R107 A111 Y115 F208 T209 Y6 W7 G11 L12 W45 K49 N58 L59 Q71 S72 R107 A111 Y115 F208 T209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0004602,0005102,0005504,0005515,0005737,0005829,0006629,0006749,0010880,0010881,0014809,0016529,0016740,0018916,0019899,0042178,0042802,0042803,0043295,0043651,0045171,0051122,0055119,0060315,0060316,0070062,0070458,0071313,0098869 remove_due_to_license_issue P28161 19808963 218 PMTLGYWNIRGLAHSIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGTHKITQSNAILRYIARKHNLCGESEKEQIREDILENQFMDSRMQLAKLCYDPDFEKLKPEYLQALPEMLKLYSQFLGKQPWFLGDKITFVDFIAYDVLERNQVFEPSCLDAFPNLKDFISRFEGLEKISAYMKSSRFLPRPVFTKMAVWGNK 3gus A 1.53 BS02 N11 A 1 F8 Q39 I104 Y108 F8 Q39 I104 Y108 Y7 R13 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Kd=0.9uM remove_due_to_license_issue IC50=800nM P09211 19808963 211 PPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3gut A 3.59 BS01 dna X 0 Y36 C38 E39 K122 R187 Y18 C20 E21 K104 R169 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut A 3.59 BS02 dna Y 0 R33 R35 R41 R15 R17 R23 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut B 3.59 BS01 dna X 0 R356 H364 G365 K541 R18 H26 G27 K203 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut B 3.59 BS02 dna Y 0 Y357 C359 E360 T443 K444 K541 K572 Q574 K575 Q606 Y19 C21 E22 T105 K106 K203 K234 Q236 K237 Q268 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut C 3.59 BS01 dna X 0 Y36 C38 E39 K122 K123 R246 Q247 Y18 C20 E21 K104 K105 R228 Q229 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut C 3.59 BS02 dna Y 0 R33 R35 A43 R15 R17 A25 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut D 3.59 BS01 dna X 0 R356 S363 H364 G365 R18 S25 H26 G27 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut D 3.59 BS02 dna Y 0 Y357 C359 E360 K444 K541 Q574 Q606 Y19 C21 E22 K106 K203 Q236 Q268 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut E 3.59 BS01 dna I 0 Y36 C38 E39 K122 R187 Y18 C20 E21 K104 R169 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut E 3.59 BS02 dna J 0 M32 R35 A43 M14 R17 A25 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut F 3.59 BS01 dna I 0 R356 H364 G365 K541 R18 H26 G27 K203 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut F 3.59 BS02 dna J 0 Y357 C359 E360 T443 K444 P543 K572 Q574 K575 Q606 Y19 C21 E22 T105 K106 P205 K234 Q236 K237 Q268 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut G 3.59 BS01 dna I 0 Y36 C38 E39 K122 K123 R187 R246 Q247 Y18 C20 E21 K104 K105 R169 R228 Q229 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut G 3.59 BS02 dna J 0 R33 A43 R15 A25 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue Q04206 19683540 1 ~ 26 AYVEIIEQPKQRGMRFRYKCEGRSAGSIPGERSTDTTKTHPTIKINGYTGPGTVRISLVTKDPPHRPHPHELVGKDCRDGYYEADLCPDRSIHSFQNLGIQCVKKRDLEQAISQRIQTNNNPFHVPIEEQRGDYDLNAVRLCFQVTVRDPAGRPLLLTPVLSHPIFDNRAPNTAELKICRVNRNSGSCLGGDEIFLLCDKVQKEDIEVYFTGPGWEARGSFSQADVHRQVAIVFRTPPYADPSLQAPVRVSMQLRRPSDRELSEPMEFQYLPD 3gut H 3.59 BS01 dna I 0 R356 S363 H364 R18 S25 H26 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3gut H 3.59 BS02 dna J 0 Y357 C359 E360 K444 K541 Q574 Q606 Y19 C21 E22 K106 K203 Q236 Q268 ? 0003677,0003700,0005737,0006355 remove_due_to_license_issue P19838 19683540 1 ~ 26 GPYLQILEQPKQRGFRFRYVCEGPSHGGLPGASSEKNKKSYPQVKICNYVGPAKVIVQLVTNGKNIHLHAHSLVGKHCEDGVCTVTAGPKDMVVGFANLGILHVTKKKVFETLEARMTEACIRGYNPGLLVHSDLAYLQAEGGGDRQLTDREKEIIRQAAVQQTKEMDLSVVRLMFTAFLPDSTGSFTRRLEPVVSDAIYDSKAPNASNLKIVRMDRTAGCVTGGEEIYLLCDKVQKDDIQIRFYEEEENGGVWEGFGDFSPTDVHRQFAIVFKTPKYKDVNITKPASVFVQLRRKSDLETSEPKPFLYYPE 3guz A 1.67 BS01 PAF A 1 P28 T29 M30 Q61 I133 Q155 P28 T29 M30 Q61 I122 Q144 M30 H34 H37 E77 D78 K81 K151 M30 H34 H37 E77 D78 K81 K140 6.3.2.1 0003824,0004592,0009058,0015940 remove_due_to_license_issue P31663 20059543 177 MLIIETLPLLRQQIRRLRMEGKRVALVPTMGNLHDGHMKLVDEAKARADVVAVSIFVNPMQFDRPEDLARYPRTLQEDCEKLNKRKVDLVFAPSVKEIYPNGTETHTYVDVPGGHFRGVSTIVSKLFNLVQPDIACFGEKDFQQLALIRKMVADMGFDIEIVGVP 3gv9 A 1.8 BS01 GV9 A 1 S64 Y221 L293 G317 A318 S61 Y218 L290 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=7.5mM remove_due_to_license_issue P00811 19416920 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gv9 A 1.8 BS02 GV9 A 2 Y92 K164 Y89 K161 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=7.5mM remove_due_to_license_issue P00811 19416920 363 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gv9 A 1.8 BS03 GV9 A 3 V125 K126 S127 A215 L216 V122 K123 S124 A212 L213 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=7.5mM remove_due_to_license_issue P00811 19416920 364 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gvb A 1.8 BS01 3GV A 1 G63 S64 Y150 Y221 I291 T316 G317 A318 G60 S61 Y147 Y218 I288 T313 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=2.6mM remove_due_to_license_issue P00811 19416920 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3gvu A 2.05 BS01 STI A 1 Y299 V302 A315 K317 E332 M336 I359 T361 Y363 M364 I406 H407 A426 D427 F428 Y31 V34 A47 K49 E64 M68 I91 T93 Y95 M96 I138 H139 A158 D159 F160 D409 A411 R413 N414 D427 P448 D141 A143 R145 N146 D159 P173 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=10nM, IC50=272nM P42684 1001 GTENLYFQSMDKWEMERTDITMKHKLGGGQYGEVYVGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTLEPPFYIVTEYMPYGNLLDYLRECNREEVTAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHVVKVADFGLSRGDTYTAKFPIKWTAPESLAYNTFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYDLLEKGYRMEQPEGCPPKVYELMRACWKWSPADRPSFAETHQAFETMFHDS 3gvu A 2.05 BS02 STI A 2 A383 V384 L386 L387 A479 G509 P511 V514 A115 V116 L118 L119 A204 G234 P236 V239 D409 A411 R413 N414 D427 P448 D141 A143 R145 N146 D159 P173 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=10nM, IC50=272nM P42684 1002 GTENLYFQSMDKWEMERTDITMKHKLGGGQYGEVYVGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTLEPPFYIVTEYMPYGNLLDYLRECNREEVTAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHVVKVADFGLSRGDTYTAKFPIKWTAPESLAYNTFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYDLLEKGYRMEQPEGCPPKVYELMRACWKWSPADRPSFAETHQAFETMFHDS 3gw5 A 2.0 BS01 72X A 1 Q19 V36 D38 Y83 P118 F119 L121 A122 F124 D226 G228 A229 S230 M303 Q16 V33 D35 Y80 P115 F116 L118 A119 F121 D223 G225 A226 S227 M300 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 ic50=0.47nM remove_due_to_license_issue IC50=0.47nM P00797 19457666 400 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3gws X 2.2 BS01 T3 X 1 F272 I276 A279 R282 M310 M313 R316 L330 N331 L346 H435 F455 F59 I63 A66 R69 M97 M100 R103 L117 N118 L133 H221 F241 ? 0003677,0004879,0006355 remove_due_to_license_issue P10828 16781732 500 EELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 3gwt A 1.75 BS01 066 A 1 S282 M347 N395 I410 F414 M431 S442 Q443 F446 S131 M196 N244 I259 F263 M280 S291 Q292 F295 3.1.4.53 0004114,0007165,0008081 ic50=7.94pM remove_due_to_license_issue IC50=0.00794nM Q07343 19656678 1 SISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIPQA 3gwu A 2.14 BS02 SRE A 1 L29 R30 Y108 F253 A319 D401 D404 L25 R26 Y104 F247 A313 D395 D398 ? 0005886,0016020,0035725 ic50=19.7uM remove_due_to_license_issue O67854 19430461 801 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3gwv A 2.35 BS02 RFX A 1 L25 R30 A319 F320 L400 D401 D404 L21 R26 A313 F314 L394 D395 D398 ? 0005886,0016020,0035725 ic50=2.54mM remove_due_to_license_issue O67854 19430461 801 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYITHWTVWITRFYIIGLFLFLTFLVFLAERRRNH 3gww A 2.46 BS02 SFX A 1 L25 G26 R30 Y108 A319 F320 D401 D404 L21 G22 R26 Y104 A310 F311 D392 D395 ? 0005886,0016020,0035725 ic50=355mM remove_due_to_license_issue O67854 19430461 801 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNH 3gwx A 2.4 BS01 EPA A 1 C285 T288 T289 H323 I326 M329 I364 H449 Y473 C79 T82 T83 H117 I120 M123 I158 H243 Y267 ? 0003677,0004879,0005634,0006355 ic50=4uM remove_due_to_license_issue IC50=4000nM Q03181 10198642 1 QVADLKAFSKHIYNAYLKNFNMTKKKARSILTGKASHTAPFVIHDIETLWQAEKGLVWKQLVNGLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKDM 3gx0 A 2.3 BS01 GDS A 1 T9 N11 Q38 K51 I52 E71 S72 G109 P110 W169 T9 N11 Q38 K51 I52 E71 S72 G109 P110 W169 T9 T9 1.11.1.-,1.8.4.- 0004364,0004601,0005737,0006979,0015036,0042803,0098869 Kd=2.4uM remove_due_to_license_issue P77526 19537707 301 MIDLYFAPTPNGHKITLFLEEAELDYRLIKVDLGKGGQFRPEFLRISPNNKIPAIVDHSPADGGEPLSLFESGAILLYLAEKTGLFLSHETRERAATLQWLFWQVGGLGPMLGQNHHFNHAAPQTIPYAIERYQVETQRLYHVLNKRLENSPWLGGENYSIADIACWPWVNAWTRQRIDLAMYPAVKNWHERIRSRPATGQALL 3gx4 X 2.7 BS01 dna Y 0 Y25 G26 R39 M45 K46 W56 S62 S67 R69 D70 Y25 G26 R39 M45 K46 W56 S62 S67 R69 D70 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 19516334 201 ~ 213 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 3gx4 X 2.7 BS02 dna Z 0 M3 S36 Y37 R39 Q40 M3 S36 Y37 R39 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 19516334 214 ~ 226 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 3gxl A 1.8 BS01 QIG A 1 I11 G14 A30 K32 L78 S80 Y82 H83 L140 D151 I11 G14 A27 K29 L75 S77 Y79 H80 L137 D148 D133 K135 N138 D151 T175 D130 K132 N135 D148 T167 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.025uM remove_due_to_license_issue IC50=>10000nM P36897 19285388 999 IARTIVLQESIGKGRFGEVWRGKWEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQ 3gxq A 2.35 BS01 dna C 0 K15 K16 N42 V43 S44 R48 K9 K10 N36 V37 S38 R42 ? 0006355 remove_due_to_license_issue A0A0H2XIU6 19759211 2 ~ 11 NSVFFGKKKKVSLHLLVDPDMKDEIIKYAQEKDFDNVSQAGREILKKGLEQIA 3gxq A 2.35 BS02 dna D 0 H20 L22 H14 L16 ? 0006355 remove_due_to_license_issue A0A0H2XIU6 19759211 2 ~ 12 NSVFFGKKKKVSLHLLVDPDMKDEIIKYAQEKDFDNVSQAGREILKKGLEQIA 3gxq B 2.35 BS01 dna C 0 H20 L22 H15 L17 ? 0006355 remove_due_to_license_issue A0A0H2XIU6 19759211 2 ~ 11 ENSVFFGKKKKVSLHLLVDPDMKDEIIKYAQEKDFDNVSQAGREILKKGLEQIA 3gxq B 2.35 BS02 dna D 0 K16 N42 V43 S44 R48 K11 N37 V38 S39 R43 ? 0006355 remove_due_to_license_issue A0A0H2XIU6 19759211 2 ~ 12 ENSVFFGKKKKVSLHLLVDPDMKDEIIKYAQEKDFDNVSQAGREILKKGLEQIA 3gxt A 2.7 BS01 NOJ A 1 D92 D93 Y134 C142 K168 D170 E203 R227 D231 D61 D62 Y103 C111 K137 D139 E172 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue P06280 19374450 430 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTM 3gxt B 2.7 BS01 NOJ B 1 W47 D92 D93 Y134 C142 K168 D170 E203 R227 D231 W16 D61 D62 Y103 C111 K137 D139 E172 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue P06280 19374450 1 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTMQ 3gxy A 2.4 BS01 MAN C 1 E23 R24 T25 E23 R24 T25 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 2 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy A 2.4 BS02 MAN C 2 G2 K3 F4 Q6 T7 G2 K3 F4 Q6 T7 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 3 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy A 2.4 BS03 MAN D 1 N93 D95 N93 D95 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 2 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy A 2.4 BS04 MAN D 2 A92 N93 A92 N93 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 3 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy B 2.4 BS01 MAN C 1 N93 I94 D95 N93 I94 D95 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 2 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy B 2.4 BS02 MAN C 2 A92 N93 A92 N93 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 3 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy B 2.4 BS03 OPM D 1 E23 T25 E23 T25 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 1 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy B 2.4 BS04 MAN D 1 T7 E23 T25 T7 E23 T25 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 2 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gxy B 2.4 BS05 MAN D 2 K3 F4 T7 K3 F4 T7 ? 0030246,0050688 remove_due_to_license_issue P81180 12110688 3 LGKFSQTCYNSAIQGSVLTSTCERTNGGYNTSSIDLNSVIENVDGSLKWQPSNFIETCRNTQLAGSSELAAECKTRAQQFVSTKINLDDHIANIDGTLKYE 3gy2 A 1.57 BS02 BRN A 1 H57 D189 S190 C191 Q192 S195 V213 W215 G216 G219 H40 D171 S172 C173 Q174 S177 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=1.8uM remove_due_to_license_issue P00760 20356563 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3gy3 A 1.7 BS02 PNT A 1 H57 T98 L99 D189 S190 S214 W215 G216 G219 H40 T80 L81 D171 S172 S192 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=2.36uM remove_due_to_license_issue P00760 20356563 246 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3gy4 A 1.55 BS02 PBZ A 1 D189 S190 W215 G216 G219 D171 S172 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=8uM remove_due_to_license_issue P00760 20356563 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3gy7 A 1.55 BS02 BEN A 1 D189 S190 Q192 S195 V213 G219 D171 S172 Q174 S177 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=30uM remove_due_to_license_issue P00760 20356563 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3gyh X 2.8 BS01 dna Y 0 Y25 G26 A38 R39 M45 K46 W56 S62 S67 R69 D70 Y25 G26 A38 R39 M45 K46 W56 S62 S67 R69 D70 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 19516334 201 ~ 213 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 3gyh X 2.8 BS02 dna Z 0 M3 S36 Y37 R39 Q40 M3 S36 Y37 R39 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 19516334 214 ~ 226 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 3gyn A 2.15 BS01 B42 A 1 F193 N291 D318 C366 L384 G410 N411 M414 Y415 Y448 S556 F188 N286 D313 C361 L379 G405 N406 M409 Y410 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.047uM remove_due_to_license_issue P26663 19796938 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3gz9 A 2.0 BS02 D32 A 1 F282 R284 C285 T289 H323 L330 L339 V341 V348 I364 K367 H449 M453 L469 Y473 F69 R71 C72 T76 H110 L117 L126 V128 V135 I151 K154 H236 M240 L256 Y260 ? 0003677,0004879,0005634,0006355 Ki=0.004uM remove_due_to_license_issue EC50=54nM, Ki=4nM Q03181 19464171 1 QVADLKAFSKHIYNAYLKNFNMTKKKARSILTGKAAPFVIHDIETLWQAEKGLVWKGLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFGSLFLNDQVTLLKYGVHEAIFAMLASLVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKD 3gzn B 3.0 BS02 B39 I 1 G78 G79 D100 M101 D102 K147 I148 Q149 L166 D167 A171 W174 G46 G47 D68 M69 D70 K115 I116 Q117 L134 D135 A139 W142 K42 D167 C237 T238 A240 K10 D135 C205 T206 A208 6.2.1.64 0000278,0005515,0005524,0005634,0005737,0005829,0006508,0007113,0008641,0016874,0019781,0019788,0032991,0036211,0042802,0043687,0045116,0046982,0051726 remove_due_to_license_issue IC50=5.0nM Q8TBC4 20129059 464 DWEGRWNHVKKFLERSGPFTHPDFEPSTESLQFLLDTCKVLVIGAGGLGCELLKNLALSGFRQIHVIDMDTIDVSNLNRQFLFRPKDIGRPKAEVAAEFLNDRVPNCNVVPHFNKIQDFNDTFYRQFHIIVCGLDSIIARRWINGMLISLLNYEDGVLDPSSIVPLIDGGTEGFKGNARVILPGMTACIECTLELYPPQVNFPMCTIASMPRLPEHCIEYVRMLQWPKEQPFGEGVPLDGDDPEHIQWIFQKSLERASQYNIRGVTYRLTQGVVKRIIPAVASTNAVIAAVCATEVFKIATSAYIPLNNYLVFNDVDGLYTYTFEAERKENCPACSQLPQNIQFSPSAKLQEVLDYLTNSASLQMKSPAITATLEGKNRTLYLQSVTSIEERTRPNLSKLKELGLVDGQELAVADVTTPQTVLFKLHFT 3h03 A 1.9 BS01 UBP A 1 Y61 P89 L90 T91 R96 T174 Y190 L192 E193 M196 Y220 Y57 P85 L86 T87 R92 T170 Y186 L188 E189 M192 Y216 ? 0015276,0016020 ic50=135uM remove_due_to_license_issue P19491 19284741 801 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 G 2.8 BS01 VBP G 1 Y61 P89 T91 R96 L138 T143 E193 Y220 Y57 P85 T87 R92 L134 T139 E189 Y216 ? 0015276,0016020 remove_due_to_license_issue IC50=290000nM P19491 19284741 803 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h0a D 2.1 BS02 D30 D 1 L255 E259 R280 I281 G284 C285 R288 L330 L333 L340 I341 E343 L353 M364 L50 E54 R68 I69 G72 C73 R76 L118 L121 L128 I129 E131 L141 M152 ? 0003677,0004879,0005634,0006355 Ki=0.033uM remove_due_to_license_issue EC50=160nM, Ki=33nM P37231 19464171 500 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3h0b A 2.7 BS01 B35 A 1 Q12 L30 D32 S35 Y71 W76 F108 W115 I118 D228 G230 Q15 L33 D35 S38 Y74 W79 F111 W118 I121 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 19409780 449 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3h0d A 2.4 BS01 dna C 0 K27 R28 S29 S40 N43 S60 K61 R62 G63 Y67 K26 R27 S28 S39 N42 S59 K60 R61 G62 Y66 ? 0003677,0006355 remove_due_to_license_issue C3W947 19498169 1 ~ 26 PNISDIIEQYLKQVLNMSDQDIVEIKRSEIANKFRCVPSQINYVINTRFTLERGYIVESKRGGGGYIRIMKVKTKSEAQLIDQLLELIDHRISQSSAEDVIKRLMEEKVISEREAKMMLSVMDRSVLYIDLPERDELRARMLKAMLTSLKYKLEI 3h0d A 2.4 BS02 dna D 0 N3 I4 S5 V38 S40 Q41 Y44 R49 K61 R62 G64 N2 I3 S4 V37 S39 Q40 Y43 R48 K60 R61 G63 ? 0003677,0006355 remove_due_to_license_issue C3W947 19498169 1 ~ 26 PNISDIIEQYLKQVLNMSDQDIVEIKRSEIANKFRCVPSQINYVINTRFTLERGYIVESKRGGGGYIRIMKVKTKSEAQLIDQLLELIDHRISQSSAEDVIKRLMEEKVISEREAKMMLSVMDRSVLYIDLPERDELRARMLKAMLTSLKYKLEI 3h0d B 2.4 BS01 dna C 0 K27 R28 S29 S40 N43 S60 K61 R62 G63 G66 Y67 K25 R26 S27 S38 N41 S58 K59 R60 G61 G64 Y65 ? 0003677,0006355 remove_due_to_license_issue C3W947 19498169 1 ~ 26 NISDIIEQYLKQVLNMSDQDIVEIKRSEIANKFRCVPSQINYVINTRFTLERGYIVESKRGGGGYIRIMKVKTKSEAQLIDQLLELIDHRISQSSAEDVIKRLMEEKVISEREAKMMLSVMDRSVLYIDLPERDELRARMLKAMLTSLKYK 3h0d B 2.4 BS02 dna D 0 N3 I4 S5 V38 S40 Q41 Y44 R49 R62 N1 I2 S3 V36 S38 Q39 Y42 R47 R60 ? 0003677,0006355 remove_due_to_license_issue C3W947 19498169 1 ~ 26 NISDIIEQYLKQVLNMSDQDIVEIKRSEIANKFRCVPSQINYVINTRFTLERGYIVESKRGGGGYIRIMKVKTKSEAQLIDQLLELIDHRISQSSAEDVIKRLMEEKVISEREAKMMLSVMDRSVLYIDLPERDELRARMLKAMLTSLKYK 3h0e A 1.997 BS01 H0E A 1 H121 G122 C163 Y204 S205 W206 R207 S251 F256 H88 G89 C130 Y165 S166 W167 R168 S212 F217 T62 S63 H121 G122 C163 R164 T29 S30 H88 G89 C130 R131 3.4.22.56 0001554,0001666,0001782,0001818,0002020,0004175,0004190,0004197,0004861,0005123,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0006974,0007413,0007507,0007605,0007611,0008047,0008233,0008234,0008627,0009410,0009411,0009611,0009749,0010038,0010165,0014069,0014070,0016005,0016241,0016485,0021766,0030163,0030182,0030216,0030218,0030220,0030889,0031264,0031647,0032025,0032355,0032496,0034349,0034612,0035094,0035556,0042542,0043025,0043029,0043065,0043200,0043525,0044346,0044877,0045165,0045786,0046007,0048011,0051146,0051384,0051402,0051604,0061713,0070269,0071407,0071887,0072734,0097153,0097190,0097193,0097194,0097200,0098693,0098978,0140639,1902004,1904019 remove_due_to_license_issue P42574 19836248 1 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIEDDMACHKIPVEADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFY 3h0j A 2.8 BS01 B36 A 1 V1923 R1954 S1957 G1958 L2025 E2026 Q2028 G2029 V442 R473 S476 G477 L544 E545 Q547 G548 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 1 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 3h0j B 2.8 BS01 B36 B 1 V1923 R1954 S1957 G1958 G1959 L2025 E2026 Q2028 G2029 V442 R473 S476 G477 G478 L544 E545 Q547 G548 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 1 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3h0j B 2.8 BS02 B36 C 1 A1761 M1765 A280 M284 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 1 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3h0q A 2.5 BS01 B37 A 1 V1923 R1954 F1956 S1957 G1958 L2025 E2026 Q2028 G2029 I2033 V442 R473 F475 S476 G477 L544 E545 Q547 G548 I552 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 1 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 3h0q B 2.5 BS01 B37 B 1 V1923 R1954 S1957 G1958 L2025 E2026 Q2028 G2029 V442 R473 S476 G477 L544 E545 Q547 G548 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 1 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3h0q B 2.5 BS02 B37 C 1 P1760 A1761 I1762 M1765 P279 A280 I281 M284 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 1 PIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3h0s A 2.43 BS01 B38 A 1 V1923 R1954 F1956 L2025 E2026 Q2028 G2029 V444 R475 F477 L546 E547 Q549 G550 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 101 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLDDKYRELRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 3h0s B 2.43 BS01 B38 B 1 V1923 R1954 F1956 G1958 E2026 Q2028 G2029 V444 R475 F477 G479 E547 Q549 G550 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 20219367 102 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGAPAINKMLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQEPGQVWHPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPQGMVGIKFRREKLLDTMNRLELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3h0v A 2.24 BS01 M2T A 1 F223 C226 G227 Y228 S229 I244 T245 E247 F147 C150 G151 Y152 S153 I168 T169 E171 S229 H243 S153 H167 4.1.1.50 0004014,0006597,0008295 ic50=15uM remove_due_to_license_issue P17707 19527050 368 SMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAAYCMGRMNSDCWYLYTLDFPDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQKIEGFKRLDCQSAMFNDYNFVFTSFAK 3h0v B 2.24 BS01 M2T A 1 F7 S66 E67 F3 S57 E58 E67 E58 4.1.1.50 0004014,0008295 remove_due_to_license_issue P17707 19527050 368 HFFEGTEKLLEVWFSRQQGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 3h0w A 1.81 BS01 N8M A 1 F223 C226 G227 Y228 I244 T245 E247 F146 C149 G150 Y151 I167 T168 E170 S229 H243 S152 H166 4.1.1.50 0004014,0006597,0008295 ic50=600nM remove_due_to_license_issue IC50=600nM P17707 19527050 368 SMFVSKRRFILKTCGTTLLLKALVPLLKLARDYSGFDSIQSFFYSRKNFMKPSHQGYPHRNFQEEIEFLNAIFPNGAAYCMGRMNSDCWYLYTLDFDQTLEILMSELDPAVMDQFYMKDGVTAKDVTRESGIRDLIPGSVIDATMFNPCGYSMNGMKSDGTYWTIHITPEPEFSYVSFETNLSQTSYDDLIRKVVEVFKPGKFVTTLFVNQKIEGFKRLDCQSAMFNDYNFVFTSFAK 3h0w B 1.81 BS01 N8M A 1 F7 S66 E67 F4 S60 E61 E67 E61 4.1.1.50 0004014,0008295 remove_due_to_license_issue IC50=600nM P17707 19527050 368 AHFFEGTEKLLEVWFSRQQPQGSGDLRTIPRSEWDILLKDVQCSIISVTKTDKQEAYVLSE 3h0y A 2.5 BS01 48B A 1 L139 V147 A160 A213 G216 T217 Y219 E260 L263 L14 V22 A35 A88 G91 T92 Y94 E135 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T154 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=0.006uM remove_due_to_license_issue IC50=6nM O14965 19402633 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3h0z A 2.92 BS01 45B A 1 V147 L194 A213 G216 T217 Y219 K224 E260 L263 V20 L67 A86 G89 T90 Y92 K97 E133 L136 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T152 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=4.3nM O14965 19402633 1 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3h1x A 1.4 BS01 IMN A 1 D49 Y52 P56 K69 D48 Y51 P55 K60 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 Kd=0.000000064M remove_due_to_license_issue P59071 19462410 301 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 3h21 A 2.32 BS01 B52 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D90 N109 I111 M134 D173 F178 G205 K209 R243 V28 D54 K220 R254 V27 D53 K209 R243 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=19.8uM remove_due_to_license_issue IC50=19800nM Q81VW8 19899766 278 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h22 A 2.4 BS01 B53 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D88 N107 I109 M132 D171 F176 G203 K207 R241 V28 D54 K220 R254 V27 D51 K207 R241 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=8uM remove_due_to_license_issue IC50=8000nM Q81VW8 19899766 901 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFGGSYNEVDAAVRHAKEMRDEGAHIIDIGGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h23 A 2.2 BS01 B54 A 1 T67 P69 D101 N120 I122 M145 D184 G216 K220 R254 H256 T66 P68 D100 N119 I121 M144 D183 G215 K219 R253 H255 V28 D54 K220 R254 V27 D53 K219 R253 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=19.3uM remove_due_to_license_issue IC50=19300nM Q81VW8 19899766 511 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGESTRPGFAKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGKG 3h26 A 2.5 BS01 B56 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D90 N109 I111 M134 D173 F178 G205 K209 R243 V28 D54 K220 R254 V27 D53 K209 R243 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=32.4uM remove_due_to_license_issue Kd=5260nM, IC50=32400nM Q81VW8 19899766 901 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h2a A 2.4 BS01 B57 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D88 N107 I109 M132 D171 F176 G203 K207 R241 V28 D54 K220 R254 V27 D51 K207 R241 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=108.9uM remove_due_to_license_issue IC50=108900nM Q81VW8 19899766 901 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSGSYNEVDAAVRHAKEMRDEGAHIIDIGGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h2c A 2.6 BS01 B58 A 1 D101 N120 I122 D184 G216 K220 R254 D84 N103 I105 D167 G199 K203 R237 D54 K220 R254 D44 K203 R237 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue IC50=>500000nM Q81VW8 19899766 901 KWDYDLRCGEYTLNLNEKTLIMGILNGSYNEVDAAVRHAKEMRDEGAHIIDIGESTRSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h2f A 2.2 BS01 B60 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D96 N115 I117 M140 D179 F184 G211 K215 R249 V28 D54 K220 R254 V28 D54 K215 R249 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=86.7uM remove_due_to_license_issue IC50=86700nM Q81VW8 19899766 901 MKWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGEFAKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h2m A 2.31 BS01 B61 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D97 N116 I118 M141 D180 F185 G212 K216 R250 V28 D54 K220 R254 V28 D54 K216 R250 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=215uM remove_due_to_license_issue IC50=215000nM Q81VW8 19899766 901 MKWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGESFAKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h2n A 2.4 BS01 B62 A 1 N120 I122 M145 D184 F189 G216 K220 R254 N111 I113 M136 D175 F180 G207 K211 R245 V28 D54 K220 R254 V27 D50 K211 R245 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=212.6uM remove_due_to_license_issue Q81VW8 19899766 901 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFGSYNEVDAAVRHAKEMRDEGAHIIDIGGESTRVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h2o A 2.7 BS01 B63 A 1 N120 I122 M145 D184 G188 G216 K220 S221 R254 N110 I112 M135 D174 G178 G206 K210 S211 R244 V28 D54 K220 R254 V27 D53 K210 R244 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue IC50=25900nM Q81VW8 19899766 501 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h30 A 1.56 BS01 RFZ A 1 V53 N118 M163 I174 V52 N117 M162 I173 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Ki=29.2uM remove_due_to_license_issue Ki=4500nM, IC50=13000nM P68400 18291315 336 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARM 3h30 A 1.56 BS02 RFZ A 2 Q40 I69 P104 Q39 I68 P103 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Ki=29.2uM remove_due_to_license_issue Ki=4500nM, IC50=13000nM P68400 18291315 337 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARM 3h3c A 2.0 BS01 P1E A 1 L431 L504 Y505 G508 E509 L556 L16 L89 Y90 G93 E94 L141 D549 A551 R553 N554 D567 L587 D134 A136 R138 N139 D152 L158 2.7.10.2 0004672,0004713,0005524,0006468 ic50=140nM remove_due_to_license_issue IC50=88nM Q14289 19428251 999 PQYGIAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLTRLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIAME 3h59 A 2.1 BS01 H59 A 1 F193 P197 N291 D318 C366 G410 M414 Y415 Q446 I447 Y448 G449 S556 F188 P192 N286 D313 C361 G405 M409 Y410 Q441 I442 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 19700319 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3h5b A 1.29 BS01 031 B 1 D25 G27 A28 D29 G48 G49 I50 V82 I84 D25 G27 A28 D29 G48 G49 I50 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 19473017 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3h5b B 1.29 BS01 031 B 1 D125 G127 A128 D130 P181 I184 D25 G27 A28 D30 P81 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.099nM remove_due_to_license_issue P03367 19473017 404 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3h5s A 2.0 BS01 H5S A 1 F193 P197 S288 N291 D318 M414 Y415 I447 Y448 G449 S556 F188 P192 S283 N286 D313 M409 Y410 I442 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.005uM remove_due_to_license_issue P26663 19709881 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3h5u A 1.95 BS01 H5U A 1 P197 S288 N291 N316 G317 D318 C366 M414 Y415 I447 Y448 G449 S556 P193 S284 N287 N312 G313 D314 C362 M410 Y411 I443 Y444 G445 S552 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.003uM remove_due_to_license_issue P26663 19709881 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYHS 3h78 A 1.7 BS01 BE2 A 1 A112 L193 F218 N287 A289 G316 S317 A112 L193 F218 N287 A289 G316 S317 2.3.1.262 0004315,0005737,0006633,0016746,0044550 remove_due_to_license_issue P20582 19694421 350 GNPILAGLGFSLPKRQVSNHDLVGRINTSDEFIVERTGVRTRYHVEPEQAVSALMVPAARQAIEAAGLLPEDIDLLLVNTLSPDHHDPSQACLIQPLLGLRHIPVLDIRAQASGLLYGLQMARGQILAGLARHVLVVCGEVLSKRMDCSDRGRNLSILLGDGAGAVVVSAGESLEDGLLDLRLGADGNYFDLLMTAAPGSASPTFLDENVLREGGGEFLMRGRPMFEHASQTLVRIAGEMLAAHELTLDDIDHVICHQPNLRILDAVQEQLGIPQHKFAVTVDRLGNMASASTPVTLAMFWPDIQPGQRVLVLTYGSGATWGAALYRKP 3h78 B 1.7 BS01 BE2 B 1 A112 L193 F218 N287 A289 S317 A119 L200 F225 N294 A296 S324 2.3.1.262 0004315,0005737,0006633,0016746,0044550 remove_due_to_license_issue P20582 19694421 350 SENLYFQGNPILAGLGFSLPKRQVSNHDLVGRINTSDEFIVERTGVRTRYHVEPEQAVSALMVPAARQAIEAAGLLPEDIDLLLVNTLSPDHHDPSQACLIQPLLGLRHIPVLDIRAQASGLLYGLQMARGQILAGLARHVLVVCGEVLSKRMDCSDRGRNLSILLGDGAGAVVVSAGESLEDGLLDLRLGADGNYFDLLMTAAPGSASPTFLDENVLREGGGEFLMRGRPMFEHASQTLVRIAGEMLAAHELTLDDIDHVICHQPNLRILDAVQEQLGIPQHKFAVTVDRLGNMASASTPVTLAMFWPDIQPGQRVLVLTYGSGATWGAALYRKP 3h78 B 1.7 BS02 BE2 B 2 M220 M225 P259 I263 M227 M232 P266 I270 2.3.1.262 0004315,0005737,0006633,0016746,0044550 remove_due_to_license_issue P20582 19694421 351 SENLYFQGNPILAGLGFSLPKRQVSNHDLVGRINTSDEFIVERTGVRTRYHVEPEQAVSALMVPAARQAIEAAGLLPEDIDLLLVNTLSPDHHDPSQACLIQPLLGLRHIPVLDIRAQASGLLYGLQMARGQILAGLARHVLVVCGEVLSKRMDCSDRGRNLSILLGDGAGAVVVSAGESLEDGLLDLRLGADGNYFDLLMTAAPGSASPTFLDENVLREGGGEFLMRGRPMFEHASQTLVRIAGEMLAAHELTLDDIDHVICHQPNLRILDAVQEQLGIPQHKFAVTVDRLGNMASASTPVTLAMFWPDIQPGQRVLVLTYGSGATWGAALYRKP 3h89 A 2.5 BS01 NSX A 1 Q19 C25 E63 G67 G68 L69 M70 A135 A138 G139 H140 E141 L144 F145 D162 H163 A214 Q19 C25 E63 G67 G68 L69 M70 A135 A138 G139 H140 E141 L144 F145 D162 H163 A209 Q19 C25 H163 N187 Q19 C25 H163 N182 3.4.22.15 0006508,0008234 Ki=0.023uM remove_due_to_license_issue P07711 19761244 400 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3h8b A 1.8 BS01 NSY A 1 Q19 Q21 C22 G23 C25 G61 E63 G67 G68 L69 M70 A135 A138 G139 E141 L144 F145 D162 H163 W189 Q19 Q21 C22 G23 C25 G61 E63 G67 G68 L69 M70 A135 A138 G139 E141 L144 F145 D162 H163 W184 Q19 C25 H163 N187 Q19 C25 H163 N182 3.4.22.15 0006508,0008234 Ki=0.511uM remove_due_to_license_issue P07711 19761244 300 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3h8b A 1.8 BS02 NSY E 1 R8 E9 G11 R8 E9 G11 Q19 C25 H163 N187 Q19 C25 H163 N182 3.4.22.15 0006508,0008234 Ki=0.511uM remove_due_to_license_issue P07711 19761244 700 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3h8c A 2.5 BS01 NSZ A 1 Q19 G20 C22 A25 G61 E63 N66 G67 G68 L69 M70 A135 A138 D162 Q19 G20 C22 A25 G61 E63 N66 G67 G68 L69 M70 A135 A138 D162 Q19 C25 H163 N187 Q19 C25 H163 N182 3.4.22.15 0006508,0008234 Ki=0.019uM remove_due_to_license_issue P07711 19761244 300 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3h98 A 1.9 BS01 B5P A 1 N291 D318 C366 S368 L384 M414 Y415 Y448 N288 D315 C363 S365 L381 M411 Y412 Y445 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50<0.005uM remove_due_to_license_issue P26663 19500983 571 HHMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPISGWFVAGYSGGDIYH 3h9f A 2.6 BS02 92M A 1 I531 A551 I586 C604 G605 N606 I607 D608 S611 L654 D664 I17 A37 I72 C90 G91 N92 I93 D94 S97 L140 D150 D647 K649 N652 D664 T686 D133 K135 N138 D150 T165 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=342.2nM P33981 20383151 809 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTTSGTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 3h9k A 2.65 BS01 UFP A 1 R50 C195 R215 S216 N226 H256 R25 C170 R190 S191 N201 H231 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue Ki=14nM P04818 21206062 400 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 3h9k A 2.65 BS02 UFP B 1 R175 R176 R150 R151 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue Ki=14nM P04818 21206062 400 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 3h9k B 2.65 BS01 UFP A 1 R175 R176 R150 R151 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue Ki=14nM P04818 21206062 400 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 3h9k B 2.65 BS02 UFP B 1 R50 C195 R215 S216 N226 R25 C170 R190 S191 N201 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue Ki=14nM P04818 21206062 400 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 3h9o A 2.3 BS01 9BD A 1 L88 A109 K111 L159 S160 Y161 A162 K163 E166 L212 T222 D223 L14 A35 K37 L85 S86 Y87 A88 K89 E92 L138 T148 D149 D205 K207 E209 N210 D223 T245 D131 K133 E135 N136 D149 T162 2.7.11.1 0004672,0004674,0005524,0006468 ic50=70nM remove_due_to_license_issue O15530 19628388 1 RKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3ha6 A 2.36 BS01 2JZ A 1 L139 K141 G142 V147 A160 K162 A213 L263 L16 K18 G19 V24 A37 K39 A90 L140 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=2.1uM remove_due_to_license_issue O14965 19648931 1 GKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3hab A 2.1 BS01 677 A 1 E205 E206 F357 Y547 S630 Y662 Y666 V711 E167 E168 F319 Y509 S592 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.0042uM remove_due_to_license_issue IC50=42nM P27487 19539471 803 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3hac A 2.0 BS01 361 A 1 E205 E206 F357 S630 Y662 Y666 V711 E167 E168 F319 S592 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.0083uM remove_due_to_license_issue EC50=112nM, IC50=67nM P27487 19539471 803 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3hau A 1.3 BS01 2NC A 1 D25 G27 A28 D29 D30 I47 G48 D25 G27 A28 D29 D30 I47 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.42uM remove_due_to_license_issue P03369 22158985 0 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3hav A 2.45 BS02 SRY A 1 D192 S194 D213 C225 D232 W265 Y272 D192 S194 D213 C225 D232 W265 Y272 ? 0005524,0016740,0046872 remove_due_to_license_issue Q9EVD7 19429619 403 MVNLDAEIYEHLNKQIKINELRYLSSGDDSDTFLCNEQYVVKVPKRDSVRISQKREFELYRFLENCKLSYQIPAVVYQSDRFNIMKYIKGERITYEQYHKLSEKEKDALAYDEATFLKELHSIEIDCSVSLFSDALVNKKDKFLQDKKLLISILEKEQLLTDEMLEHIETIYENILNNAVLFKYTPCLVHNDFSANNMIFRNNRLFGVIDFGDFNVGDPDNDFLCLLDCSTDDFGKEFGRKVLKYYQHKAPEVAERKAELNDVYWSIDQIIYGYDREMLIKGVSELLQTQAEMFIF 3haw B 1.3 BS01 2NC B 1 D25 G27 A28 D29 D30 I47 G48 G49 P81 D25 G27 A28 D29 D30 I47 G48 G49 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=1.01uM remove_due_to_license_issue P03369 22158985 0 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3hb4 X 2.21 BS01 E2B X 1 S142 G144 L149 Y155 F192 H221 S142 G144 L149 Y155 F192 H221 1.1.1.51,1.1.1.62 0003824,0004303,0005496,0005515,0005737,0005829,0006629,0006694,0006703,0007040,0007519,0008210,0010467,0016491,0030283,0036094,0042803,0047035,0047045,0050661,0060348,0060612,0061370,0070401,0071248,0072582,1903924 remove_due_to_license_issue IC50=27nM P14061 19929851 700 ARTVVLITGCSSGIGLHLAVRLASDPSQSFKVYATLRDLKTQGRLWEAARALACPPGSLETLQLDVRDSKSVAAARERVTEGRVDVLVCNAGLGLLGPLEALGEDAVASVLDVNVVGTVRMLQAFLPDMKRRGSGRVLVTGSVGGLMGLPFNDVYCASKFALEGLCESLAVLLLPFGVHLSLIECGPVHTAFMEKVLGSPEEVLDRTDIHTFHRFYQYLAHSKQVFREAAQNPEEVAEVFLTALRAPKPTLRYFTTERFLPLLRMRLDDPSGSNYVTAMHREVF 3hb8 A 2.74 BS01 UMP A 1 R50 C195 R215 S216 D218 N226 H256 R25 C170 R190 S191 D193 N201 H231 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 21206062 314 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 3hb8 B 2.74 BS01 UMP A 1 R175 R176 R150 R151 E87 W109 Y135 C195 R215 D218 E62 W84 Y110 C170 R190 D193 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 21206062 314 PPHGELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQKVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPT 3hbo A 1.71 BS01 2NC A 1 R8 L23 D25 G27 A28 D29 G48 I50 V82 R8 L23 D25 G27 A28 D29 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=8.2uM remove_due_to_license_issue P03369 22158985 0 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3hc8 A 1.79 BS01 PD4 A 1 A767 I768 Q775 V782 L804 M816 Q817 F820 A233 I234 Q241 V248 L270 M282 Q283 F286 3.1.4.35,3.1.4.53 0004114,0007165,0008081 ic50=2.9nM remove_due_to_license_issue O76074,P27815 19539468 901 ETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHPGVSNQFLINTNSELALMYNDESVLEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHEKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 3hcm A 2.0 BS03 S45 A 1 F76 M79 A83 F77 M80 A84 ? 0001726,0005509,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0007155,0007409,0007417,0007611,0007613,0008270,0008284,0042802,0042803,0043025,0043123,0043231,0044548,0045666,0046872,0048156,0048168,0048306,0048471,0050786,0097490,1990138,1990845 remove_due_to_license_issue P04271 20077460 94 MSELEKAMVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDNDGDGECDFQEFMAFVAMVTTACHEFFE 3hcm B 2.0 BS03 S45 B 1 E45 V56 F76 M79 E46 V57 F77 M80 ? 0001726,0005509,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0007155,0007409,0007417,0007611,0007613,0008270,0008284,0042802,0042803,0043025,0043123,0043231,0044548,0045666,0046872,0048156,0048168,0048306,0048471,0050786,0097490,1990138,1990845 remove_due_to_license_issue P04271 20077460 94 MSELEKAMVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDNDGDGECDFQEFMAFVAMVTTACHEFFEH 3hd3 A 1.75 BS01 25B A 1 Q19 G23 C25 S61 G65 G66 D161 H162 Q19 G23 C25 S61 G65 G66 D161 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 19773167 216 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLAEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDGAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 3hdk B 1.8 BS01 2NC B 1 D25 G27 A28 D29 D30 I47 G48 D25 G27 A28 D29 D30 I47 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=17.5uM remove_due_to_license_issue P03369 22158985 0 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3hdm A 2.6 BS01 MMG A 1 I104 G107 V112 A125 L176 I179 E183 L229 T239 I24 G27 V32 A45 L83 I86 E90 L136 T146 D222 K224 N227 D240 T260 D129 K131 N134 D147 T167 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=1300nM O00141 19497745 500 QQINLGPSSNPHAKPSDFHFLKVIGKGSFGKVLLARHKAEEVFYAVKVLQKKAILVLLKNVKHPFLVGLHFSFQTADKLYFVLDYINGGELFYHLQRERCFLEPRARFYAAEIASALGYLHSLNIVYRDLKPENILLDSQGHIVLTDFGLCKENIEHNSTTSTFCGTPEYLAPEVLHKQPYDRTVDWWCLGAVLYEMLYGLPPFYSRNTAEMYDNILNKPLQLKPNITNSARHLLEGLLQKDRTKRLGAKDDFMEIKSHVFFSLINWDDLINKKITPPFNPNVSG 3hdn A 3.1 BS01 GMG A 1 I104 G107 V112 A125 K127 I179 L229 T239 I23 G26 V31 A44 K46 I85 L135 T145 D222 K224 N227 D240 T260 D128 K130 N133 D146 T166 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=880nM O00141 19497745 1 QINLGPSSNPHAKPSDFHFLKVIGKGSFGKVLLARHKAEEVFYAVKVLQKKAILVLLKNVKHPFLVGLHFSFQTADKLYFVLDYINGGELFYHLQRERCFLEPRARFYAAEIASALGYLHSLNIVYRDLKPENILLDSQGHIVLTDFGLCKENIEHNSTTSTFCGTPEYLAPEVLHKQPYDRTVDWWCLGAVLYEMLYGLPPFYSRNTAEMYDNILNKPLQLKPNITNSARHLLEGLLQKDRTKRLGAKDDFMEIKSHVFFSLINWDDLINKKITPPFNP 3hdz A 1.8 BS01 PD6 A 1 A767 I768 L804 M816 Q817 F820 A232 I233 L269 M281 Q282 F285 3.1.4.35,3.1.4.53 0004114,0007165,0008081 ic50=51nM remove_due_to_license_issue O76074,P27815 19540112 400 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHPGVSNQFLINTNSELALMYNDESVLEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHEKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 3hec A 2.5 BS01 STI A 1 V30 A51 K53 E71 L75 I84 T106 L108 M109 I147 H148 L167 D168 F169 V26 A42 K44 E62 L66 I75 T97 L99 M100 I138 H139 L158 D159 F160 D150 K152 N155 D168 T185 D141 K143 N146 D159 T162 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=34uM remove_due_to_license_issue Kd=>10000nM, IC50=100000nM Q16539 20337484 1 RPTFYRQELNKTIWEVPERYQNLSPVGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3heg A 2.2 BS01 BAX A 1 V30 V38 A51 E71 L74 L75 I84 T106 M109 H148 I166 L167 D168 F169 V26 V30 A43 E63 L66 L67 I76 T98 M101 H140 I158 L159 D160 F161 D150 K152 N155 D168 T185 D142 K144 N147 D160 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=0.18uM remove_due_to_license_issue Kd=370nM, IC50=400nM Q16539 20337484 1 RPTFYRQELNKTIWEVPERYQNLSPVYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hek A 1.95 BS01 BD0 A 1 N51 D93 M98 N106 L107 V136 F138 Y139 T184 N42 D84 M89 N97 L98 V127 F129 Y130 T175 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=5.4nM remove_due_to_license_issue P07900 19583220 901 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKELEHH 3hf6 A 1.8 BS02 LX0 A 1 G234 Y235 R257 Y264 T265 P266 E267 P268 H272 F313 E317 S336 S337 G121 Y122 R144 Y151 T152 P153 E154 P155 H159 F200 E204 S223 S224 H272 H277 E317 S336 H159 H164 E204 S223 1.14.16.4 0004497,0005506,0009072,0016714 ic50=0.026uM remove_due_to_license_issue IC50=26nM P17752 19631532 401 SVPWFPKKISDLDHCLDADHPGFKDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFRELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTI 3hf8 A 1.85 BS02 ML0 A 1 Y235 L236 S237 P238 R257 Y264 T265 P266 E267 P268 H272 F313 E317 S336 S337 C364 I366 Y116 L117 S118 P119 R138 Y145 T146 P147 E148 P149 H153 F194 E198 S217 S218 C245 I247 H272 H277 E317 S336 H153 H158 E198 S217 1.14.16.4 0004497,0005506,0009072,0016714 Ki=0.31uM remove_due_to_license_issue P17752 20556201 401 SVPWFPKKISDLDHCANRDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFRELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTI 3hfb A 1.92 BS02 ML4 A 1 P238 R257 Y264 T265 P266 H272 Q306 A309 F313 E317 S336 S337 C364 P119 R138 Y145 T146 P147 H153 Q187 A190 F194 E198 S217 S218 C245 H272 H277 E317 S336 H153 H158 E198 S217 1.14.16.4 0004497,0005506,0009072,0016714 Ki=0.03uM remove_due_to_license_issue IC50=40nM P17752 20556201 401 SVPWFPKKISDLDHCANRDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFRELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTI 3hfj A 2.02 BS01 DZ9 A 1 M109 Y112 W116 M109 Y112 W116 0003824,0009058,0009435,0016779 ic50=36uM remove_due_to_license_issue 19716475 202 MRKIGIIGGTFDPPHYGHLLIANEVYHALNLEEVWFLPNQIPPHKQGRNITSVESRLQMLELATEAEEHFSICLEELSRKGPSYTYDTMLQLTKKYPDVQFHFIIGGDMVEYLPKWYNIEALLDLVTFVGVARPGYKLRTPYPITTVEIPEFAVSSSLLRERYKEKKTCKYLLPEKVQVYIERNGLYES 3hfj B 2.02 BS01 DZ9 A 1 F103 M109 Y112 K115 W116 F103 M109 Y112 K115 W116 0003824,0009058,0009435,0016779 remove_due_to_license_issue 19716475 202 MRKIGIIGGTFDPPHYGHLLIANEVYHALNLEEVWFLPNQIPPHKQGRNITSVESRLQMLELATEAEEHFSICLEELSRKGPSYTYDTMLQLTKKYPDVQFHFIIGGDMVEYLPKWYNIEALLDLVTFVGVARPGYKLRTPYPITTVEIPEFAVSSSLLRERYKEKKTCKYLLPEKVQVYIERNGLYES 3hfv A 2.6 BS01 MTY A 1 H119 S121 E159 F232 F234 G254 C255 F276 G277 H109 S111 E149 F222 F224 G244 C245 F266 G267 G105 H119 R143 Q157 T235 A275 G95 H109 R133 Q147 T225 A265 6.1.1.20 0000049,0000166,0004812,0004826,0005515,0005524,0005737,0005739,0005759,0006412,0006418,0006432,0008033,0043039 remove_due_to_license_issue O95363 19549855 416 PGSVVELLGKSYPQDDHSNLTRKVLTRVGRNLHNQQHHPLWLIKERVKEHFYKQYVGRFGTPLFSVYDNLSPVVTTWQNFDSLLIPADHPSRKKGDNYYLNRTHMLRAHTSAHQWDLLHAGLDAFLVVGDVYRRDQIDSQHYPIFHQLEAVRLFSKHELFAGIKDGESLQLFEQSSRSAHKQETHTMEAVKLVEFDLKQTLTRLMAHLFGDELEIRWVDCYFPFTHPSFEMEINFHGEWLEVLGCGVMEQQLVNSAGAQDRIGWAFGLGLERLAMILYDIPDIRLFWCEDERFLKQFCVSNINQKVKFQPLSKYPAVINDISFWLPSENYAENDFYDLVRTIGGDLVEKVDLIDKFVHPKTHKTSHCYRITYRHMERTLSQREVRHIHQALQEAAVQLLGVEGRF 3hfz A 2.9 BS01 MTY A 1 H178 E220 F258 F260 G282 A283 A314 F315 G316 H94 E136 F174 F176 G198 A199 A230 F231 G232 W149 H178 R204 Q218 V261 A314 W65 H94 R120 Q134 V177 A230 6.1.1.20 0000049,0000166,0000287,0004812,0004826,0005524,0005737,0006412,0006432,0043039,0046872 remove_due_to_license_issue Q5SGX2 19549855 351 RVDVSLPGASLFSGGLHPITLMERELVEIFRALGYQAVEGPEVESEFFNFDALNIPEHHPARDMWDTFWLTGEGFRLEGPLGEEVEGRLLLRTHTSPMQVRYMVAHTPPFRIVVPGRVFRFEQTDATHEAVFHQLEGLVVGEGIAMAHLKGAIYELAQALFGPDSKVRFQPVYFPFVEPGAQFAVWWPEGGKWLELGGAGMVHPKVFQAVDAYRERLGLPPAYRGVTGFAFGLGVERLAMLRYGIPDIRYFFGGRLKFLEQFKGVL 3hha A 1.27 BS01 NOW A 1 G23 C25 G67 G68 L69 M70 A135 M161 D162 G23 C25 G67 G68 L69 M70 A135 M161 D162 Q19 C25 H163 N187 Q19 C25 H163 N187 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 19515558 301 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDAGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3hhk A 1.7 BS01 77Z A 1 F193 N291 N316 D318 C366 L384 M414 Y415 Y448 S556 F193 N291 N316 D318 C366 L384 M414 Y415 Y448 S556 3.4.21.98,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=6nM remove_due_to_license_issue Q99AU2 19515564 564 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3hhm A 2.8 BS01 KWT A 1 M772 K776 I800 K802 Y836 E849 V850 V851 I932 D933 M754 K758 I782 K784 Y818 E831 V832 V833 I914 D915 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue IC50=12nM, Kd=5.4nM, Ki=120nM P42336 19805105 1833 SYYHHHHHHDYPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRETSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREAGFSYSHAGLSNRRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGGLKGALQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDARHGGWTTKMDWIFHTI 3hhu A 1.59 BS01 819 A 1 N51 A55 D93 G97 M98 L107 G108 T109 G135 F138 N36 A40 D78 G82 M83 L92 G93 T94 G120 F123 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=41nM remove_due_to_license_issue P07900 19519743 500 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3hig A 2.09 BS04 BRN A 1 Y148 D186 Y371 D373 W376 Y459 Y122 D160 Y335 D337 W340 Y423 Y359 D373 Y461 H510 H512 H675 Y323 D337 Y425 H474 H476 H639 1.4.3.22 0005507,0005509,0005515,0005576,0005615,0005777,0005886,0005923,0008131,0008201,0009308,0009445,0016491,0016641,0035580,0042803,0046872,0048038,0050232,0052597,0052598,0070062 Ki=13nM remove_due_to_license_issue Ki=13nM P19801 19764817 901 PRKAGVFSDLSNQELKAVHSFLWSKKELRLQPSSTTTMAKNTVFLIEMLLPKKYHVLRFLDKGERHPVREARAVIFFGDQEHPNVTEFAVGPLPGPCYMRALSPRPGYQSSWASRPISTAEYALLYHTLQEATKPLHQFFLNTTGFSFQDCHDRCLAFTDVAPRGVASGQRRSWLIIQRYVEGYFLHPTGLELLVDHGSTDAGHWAVEQVWYNGKFYGSPEELARKYADGEVDVVVLEDPLEPPLFSSHKPRGDFPSPIHVSGPRLVQPHGPRFRLEGNAVLYGGWSFAFRLRSSSGLQVLNVHFGGERIAYEVSVQEAVALYGGHTPAGMQTKYLDVGWGLGSVTHELAPGIDCPETATFLDTFHYYDADDPVHYPRALCLFEMPTGVPLRRHFNSNFKGGFNFYAGLKGQVLVLRTTSTVYNYDYIWDFIFYPNGVMEAKMHATGYVHATFYTPEGLRHGTRLHTHLIGNIHTHLVHYRVDLDVAGTKNSFQTLQMKLENITNPWSPRHRVVQPTLEQTQYSWERQAAFRFKRKLPKYLLFTSPQENPWGHKRSYRLQIHSMADQVLPPGWQEEQAITWARYPLAVTKYRESELCSSSIYHQNDPWDPPVVFEQFLHNNENIENEDLVAWVTVGFLHIPHSEDIPNTATPGNSVGFLLRPFNFFPEDPSLASRDTVIVWPRDNGPNYVQRWIPEDRDCSMPPPFSYNGTYRPV 3hig B 2.09 BS04 BRN B 1 Y148 D186 Y371 D373 W376 V458 Y459 Y121 D159 Y330 D332 W335 V417 Y418 Y359 D373 Y461 H510 H512 H675 Y318 D332 Y420 H469 H471 H634 1.4.3.22 0005507,0005509,0005515,0005576,0005615,0005777,0005886,0005923,0008131,0008201,0009308,0009445,0016491,0016641,0035580,0042803,0046872,0048038,0050232,0052597,0052598,0070062 Ki=13nM remove_due_to_license_issue Ki=13nM P19801 19764817 901 RKAGVFSDLSNQELKAVHSFLWSKKELRLQPSSTTTMAKNTVFLIEMLLPKKYHVLRFLDKGERHPVREARAVIFFGDQEHPNVTEFAVGPLPGPCYMRALSPRPGYQSSWASRPISTAEYALLYHTLQEATKPLHQFFLNTTGFSFQDCHDRCLAFTDVAPRGVASGQRRSWLIIQRYVEGYFLHPTGLELLVDHGSTDAGHWAVEQVWYNGKFYGSPEELARKYADGEVDVVVLEPPLFSSHKPRGDFPSPIHVSGPRLVQPHGPRFRLEGNAVLYGGWSFAFRLRSSSGLQVLNVHFGGERIAYEVSVQEAVALYGGHTPAGMQTKYLDVGWGLGSVTHELAPGIDCPETATFLDTFHYYDADDPVHYPRALCLFEMPTGVPLRRHFNSNFKGGFNFYAGLKGQVLVLRTTSTVYNYDYIWDFIFYPNGVMEAKMHATGYVHATFYTPEGLRHGTRLHTHLIGNIHTHLVHYRVDLDVAGTKNSFQTLQMKLENITNPWSPRHRVVQPTLEQTQYSWERQAAFRFKRKLPKYLLFTSPQENPWGHKRSYRLQIHSMADQVLPPGWQEEQAITWARYPLAVTKYRESELCSSSIYHQNDPWDPPVVFEQFLHNNENIENEDLVAWVTVGFLHIPHSEDIPNTATPGNSVGFLLRPFNFFPEDPSLASRDTVIVWPRDNGPNYVQRWIPEDRDCSMPPPFSYNGTYRPV 3hii A 2.149 BS04 PNT A 1 Y148 Y371 D373 W376 V381 Y404 V458 Y459 N460 Y122 Y335 D337 W340 V345 Y368 V422 Y423 N424 Y359 D373 Y461 H510 H512 H675 Y323 D337 Y425 H474 H476 H639 1.4.3.22 0005507,0005509,0005515,0005576,0005615,0005777,0005886,0005923,0008131,0008201,0009308,0009445,0016491,0016641,0035580,0042803,0046872,0048038,0050232,0052597,0052598,0070062 Ki=290nM remove_due_to_license_issue Ki=290nM P19801 19764817 901 PRKAGVFSDLSNQELKAVHSFLWSKKELRLQPSSTTTMAKNTVFLIEMLLPKKYHVLRFLDKGERHPVREARAVIFFGDQEHPNVTEFAVGPLPGPCYMRALSPRPGYQSSWASRPISTAEYALLYHTLQEATKPLHQFFLNTTGFSFQDCHDRCLAFTDVAPRGVASGQRRSWLIIQRYVEGYFLHPTGLELLVDHGSTDAGHWAVEQVWYNGKFYGSPEELARKYADGEVDVVVLEDPLEPPLFSSHKPRGDFPSPIHVSGPRLVQPHGPRFRLEGNAVLYGGWSFAFRLRSSSGLQVLNVHFGGERIAYEVSVQEAVALYGGHTPAGMQTKYLDVGWGLGSVTHELAPGIDCPETATFLDTFHYYDADDPVHYPRALCLFEMPTGVPLRRHFNSNFKGGFNFYAGLKGQVLVLRTTSTVYNYDYIWDFIFYPNGVMEAKMHATGYVHATFYTPEGLRHGTRLHTHLIGNIHTHLVHYRVDLDVAGTKNSFQTLQMKLENITNPWSPRHRVVQPTLEQTQYSWERQAAFRFKRKLPKYLLFTSPQENPWGHKRSYRLQIHSMADQVLPPGWQEEQAITWARYPLAVTKYRESELCSSSIYHQNDPWDPPVVFEQFLHNNENIENEDLVAWVTVGFLHIPHSEDIPNTATPGNSVGFLLRPFNFFPEDPSLASRDTVIVWPRDNGPNYVQRWIPEDRDCSMPPPFSYNGTYRPV 3hii B 2.149 BS04 PNT B 1 Y148 D186 Y371 D373 W376 G377 V381 Y404 Y459 N460 Y121 D159 Y330 D332 W335 G336 V340 Y363 Y418 N419 Y359 D373 Y461 H510 H512 H675 Y318 D332 Y420 H469 H471 H634 1.4.3.22 0005507,0005509,0005515,0005576,0005615,0005777,0005886,0005923,0008131,0008201,0009308,0009445,0016491,0016641,0035580,0042803,0046872,0048038,0050232,0052597,0052598,0070062 Ki=290nM remove_due_to_license_issue Ki=290nM P19801 19764817 901 RKAGVFSDLSNQELKAVHSFLWSKKELRLQPSSTTTMAKNTVFLIEMLLPKKYHVLRFLDKGERHPVREARAVIFFGDQEHPNVTEFAVGPLPGPCYMRALSPRPGYQSSWASRPISTAEYALLYHTLQEATKPLHQFFLNTTGFSFQDCHDRCLAFTDVAPRGVASGQRRSWLIIQRYVEGYFLHPTGLELLVDHGSTDAGHWAVEQVWYNGKFYGSPEELARKYADGEVDVVVLEPPLFSSHKPRGDFPSPIHVSGPRLVQPHGPRFRLEGNAVLYGGWSFAFRLRSSSGLQVLNVHFGGERIAYEVSVQEAVALYGGHTPAGMQTKYLDVGWGLGSVTHELAPGIDCPETATFLDTFHYYDADDPVHYPRALCLFEMPTGVPLRRHFNSNFKGGFNFYAGLKGQVLVLRTTSTVYNYDYIWDFIFYPNGVMEAKMHATGYVHATFYTPEGLRHGTRLHTHLIGNIHTHLVHYRVDLDVAGTKNSFQTLQMKLENITNPWSPRHRVVQPTLEQTQYSWERQAAFRFKRKLPKYLLFTSPQENPWGHKRSYRLQIHSMADQVLPPGWQEEQAITWARYPLAVTKYRESELCSSSIYHQNDPWDPPVVFEQFLHNNENIENEDLVAWVTVGFLHIPHSEDIPNTATPGNSVGFLLRPFNFFPEDPSLASRDTVIVWPRDNGPNYVQRWIPEDRDCSMPPPFSYNGTYRPV 3hio A 2.0 BS01 C2X A 1 D75 N78 Y80 V81 D96 D100 G121 Y123 I172 R180 W211 G212 R213 R258 D71 N74 Y76 V77 D92 D96 G117 Y119 I168 R176 W207 G208 R209 R254 V81 E177 R180 V77 E173 R176 3.2.2.22 0017148,0030598 remove_due_to_license_issue P02879 19920175 268 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPP 3hit A 2.29 BS01 DYN A 1 Y73 V74 E121 Y123 V169 E174 R177 E206 N207 W209 G210 R214 Y233 L254 Y73 V74 E121 Y123 V169 E174 R177 E206 N207 W209 G210 R214 Y233 L254 V74 E174 R177 V74 E174 R177 3.2.2.22 0006952,0016787,0017148,0030598,0035821,0090729 Ki=6.4nM remove_due_to_license_issue Q2QEH4 19920175 260 VIIYELNLQGTTKAQYSTFLKQLRDDIKDPNLHYGGTNLPVIKRPVGPPKFLRVNLKASTGTVSLAVQRSNLYVAAYLAKNNNKQFRAYYFKGFQITTNQLNNLFPEATGVSNQQELGYGESYPQIQNAAGVTRQQAGLGIKKLAESMTKVNGVARVEKDEALFLLIVVQMVGEAARFKYIENLVLNNFDTAKEVEPVPDRVIILENNWGLLSRAAKTANNGVFQTPLVLTSYAVPGVEWRVTTVAEVEIGIFLNVD 3hiv A 2.14 BS01 TXN A 1 N71 Y73 V74 E121 Y123 E174 R177 E206 N207 W209 G210 R214 L254 N71 Y73 V74 E121 Y123 E174 R177 E206 N207 W209 G210 R214 L254 V74 E174 R177 V74 E174 R177 3.2.2.22 0006952,0016787,0017148,0030598,0035821,0090729 Ki=7.5nM remove_due_to_license_issue Q2QEH4 19920175 260 VIIYELNLQGTTKAQYSTFLKQLRDDIKDPNLHYGGTNLPVIKRPVGPPKFLRVNLKASTGTVSLAVQRSNLYVAAYLAKNNNKQFRAYYFKGFQITTNQLNNLFPEATGVSNQQELGYGESYPQIQNAAGVTRQQAGLGIKKLAESMTKVNGVARVEKDEALFLLIVVQMVGEAARFKYIENLVLNNFDTAKEVEPVPDRVIILENNWGLLSRAAKTANNGVFQTPLVLTSYAVPGVEWRVTTVAEVEIGIFLNVD 3hiw A 1.8 BS01 C2X A 1 N71 Y73 V74 E121 S122 Y123 V169 E174 R177 E206 N207 G210 R214 Y233 L254 N71 Y73 V74 E121 S122 Y123 V169 E174 R177 E206 N207 G210 R214 Y233 L254 V74 E174 R177 V74 E174 R177 3.2.2.22 0006952,0016787,0017148,0030598,0035821,0090729 Ki=3.9nM remove_due_to_license_issue Q2QEH4 19920175 260 VIIYELNLQGTTKAQYSTFLKQLRDDIKDPNLHYGGTNLPVIKRPVGPPKFLRVNLKASTGTVSLAVQRSNLYVAAYLAKNNNKQFRAYYFKGFQITTNQLNNLFPEATGVSNQQELGYGESYPQIQNAAGVTRQQAGLGIKKLAESMTKVNGVARVEKDEALFLLIVVQMVGEAARFKYIENLVLNNFDTAKEVEPVPDRVIILENNWGLLSRAAKTANNGVFQTPLVLTSYAVPGVEWRVTTVAEVEIGIFLNVD 3hj0 A 1.34 BS01 A93 A 1 K15 L17 L110 S117 K6 L8 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=1960nM P02766 20081815 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3hj0 B 1.34 BS01 A93 B 1 K15 L17 L110 S117 T118 K6 L8 L101 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=1960nM P02766 20081815 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3hjo A 1.95 BS02 EAA A 1 F8 V10 I104 G205 F8 V10 I104 G205 Y7 R13 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue IC50=2.6e+4nM P09211 19780048 211 PPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIVTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3hjw A 2.35 BS01 rna D 0 G59 T61 H63 E64 K70 K77 A78 G79 H80 T100 R101 V103 Q104 K259 S261 A265 H268 G269 A270 A273 P275 G276 K317 G318 I319 K325 V326 R330 K335 L336 W337 G49 T51 H53 E54 K60 K67 A68 G69 H70 T90 R91 V93 Q94 K249 S251 A255 H258 G259 A260 A263 P265 G266 K307 G308 I309 K315 V316 R320 K325 L326 W327 D85 Y113 R184 D75 Y103 R174 5.4.99.25 0000495,0001522,0003723,0005515,0006396,0008033,0009451,0009982,0016853,0031118,0031119,0031120,0160148,1990481 remove_due_to_license_issue Q7LWY0 19478803 1 ~ 58 RILPADIKREVLIKDENAETNPDWGFPPEKRPIEMHIQFGVINLDKPPGPTSHEVVAWIKKILNLEKAGHGGTLDPKVSGVLPVALEKATRVVQALLPAGKEYVALMHLHGDVPEDKIIQVMKEFEGEIIQRPPLRSAVKRRLRTRKVYYIEVLEIEGRDVLFRVGVEAGTYIRSLIHHIGLALGVGAHMSELRRTRSGPFKEDETLITLHDLVDYYYFWKEDGIEEYFRKAIQPMEKAVEHLPKVWIKDSAVAAVTHGADLAVPGIAKLHAGIKRGDLVAIMTLKDELVALGKAMMTSQEMLEKTKGIAVDVEKVFMPRDWYPKLW 3hjw A 2.35 BS02 rna E 0 H63 H80 G82 T83 D85 P86 L107 K111 R146 A148 V149 K150 R154 A179 G180 Y182 I183 R184 L203 R205 H53 H70 G72 T73 D75 P76 L97 K101 R136 A138 V139 K140 R144 A169 G170 Y172 I173 R174 L193 R195 D85 Y113 R184 D75 Y103 R174 5.4.99.25 0000495,0001522,0003723,0005515,0006396,0008033,0009451,0009982,0016853,0031118,0031119,0031120,0160148,1990481 remove_due_to_license_issue Q7LWY0 19478803 5 ~ 17 RILPADIKREVLIKDENAETNPDWGFPPEKRPIEMHIQFGVINLDKPPGPTSHEVVAWIKKILNLEKAGHGGTLDPKVSGVLPVALEKATRVVQALLPAGKEYVALMHLHGDVPEDKIIQVMKEFEGEIIQRPPLRSAVKRRLRTRKVYYIEVLEIEGRDVLFRVGVEAGTYIRSLIHHIGLALGVGAHMSELRRTRSGPFKEDETLITLHDLVDYYYFWKEDGIEEYFRKAIQPMEKAVEHLPKVWIKDSAVAAVTHGADLAVPGIAKLHAGIKRGDLVAIMTLKDELVALGKAMMTSQEMLEKTKGIAVDVEKVFMPRDWYPKLW 3hjw B 2.35 BS01 rna D 0 R34 S36 E38 R32 S34 E36 ? 0001522,0030515,0042254 remove_due_to_license_issue Q8U1R4 19478803 1 ~ 58 FRIRKCPKCGRYTLKEVCPVCGEKTKVAHPPRFSPEDPYGEYRRRWKREVLGI 3hjw C 2.35 BS01 rna D 0 R34 K35 G36 T37 N38 E39 K42 R46 V58 D59 I93 E94 V95 A96 A97 A98 R31 K32 G33 T34 N35 E36 K39 R43 V55 D56 I90 E91 V92 A93 A94 A95 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006364,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue Q8U160 19478803 1 ~ 58 KPSYVKFEVPKELAEKALQAVEIARDTGKIRKGTNETTKAVERGQAKLVIIAEDVDPEEIVAHLPPLCEEKEIPYIYVPSKKELGAAAGIEVAAASVAIIEPGKARDLVEEIAMKVKELM 3hk1 A 1.7 BS01 B64 A 1 F16 V23 V25 A33 K58 A75 D76 C117 R126 Y128 F16 V23 V25 A33 K58 A75 D76 C117 R126 Y128 ? 0005324,0005634,0005654,0005737,0008289,0009617,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0071285,0071356,0120162 Ki=0.67uM remove_due_to_license_issue P04117 19754198 132 CDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDLVTIRSESTFKNTEISFKLGVEFDEITADDRKVKSIITLDGGALVQVQKWDGKSTTIKRKRDGDKLVVECVMKGVTSTRVYERA 3hkq A 1.7 BS02 1SD A 1 Q92 H94 H96 F130 L197 T198 T199 Q89 H91 H93 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=4550nM P00918 19827837 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3hku A 1.8 BS02 TOR A 1 N62 A65 N67 Q92 H94 F130 L197 T198 T199 N59 A62 N64 Q89 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=10nM, Kd=290nM, IC50=5nM P00918 19827837 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3hkw A 1.55 BS01 IX6 A 1 R200 C366 S367 M414 F415 E446 I447 Y448 G449 S556 R198 C364 S365 M412 F413 E444 I445 Y446 G447 S554 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=80nM remove_due_to_license_issue P26664 20071590 579 SMSYSWTGALVTPCAAEEQKLPINALSNSLLRHHNMVYSTTSRSACQRQKKVTFDRLQVLDSHYQDVLKEVKAAASKVKANLLSVEEACSLTPPHSARSKFGYGAKDVRCHARKAVTHINSVWKDLLEDSVTPIDTTIMAKNEVFCVQPGGRKPARLIVFPDLGVRVCEKMALYDVVSKLPQAVMGSSYGFQYSPGQRVEFLVQAWKSKKSPMGFSYDTRCFDSTVTESDIRTEEAIYQCCDLDPQARVAIKSLTERLYVGGPLTNSKGENCGYRRCRASGVLTTSCGNTLTCYIKARAACRAAGLQDCTMLVCGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDGAGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMFAPTLWARMILMTHFFSVLIARDQLEQALDCEIYGACYSIEPLDLPPIIQRLHGLSAFSLHSYSPGEINRVAACLRKLGVPPLRAWRHRARSVRAKLLSRGGRAAICGKYLFNWAVRTKLKLTPIAAAGQLDLSGWFTAGYSGGDIYHS 3hky A 1.9 BS01 IX6 A 1 R200 C366 S367 L384 N411 Y448 S556 R201 C367 S368 L385 N412 Y449 S557 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=2.3nM remove_due_to_license_issue O92972 20071590 579 SSMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3hl5 A 1.8 BS02 9JZ A 1 L307 T308 D309 E314 Q319 W323 L55 T56 D57 E62 Q67 W71 2.3.2.27 remove_due_to_license_issue Kd=16nM P98170 19492850 1 SHMLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTH 3hl5 A 1.8 BS03 9JZ B 1 P325 H343 H346 P73 H91 H94 2.3.2.27 remove_due_to_license_issue Kd=16nM P98170 19492850 1 SHMLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTH 3hl7 A 1.88 BS01 I47 A 1 A50 L103 V104 T105 M108 A46 L99 V100 T101 M104 D149 K151 N154 D167 T184 D145 K147 N150 D163 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=0.023uM remove_due_to_license_issue Q16539 19496616 401 PTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hl8 A 1.55 BS01 BBP A 1 P228 W245 A312 N313 R327 L331 P220 W237 A298 N299 R313 L317 3.1.11.1 0000175,0000287,0003676,0003677,0003697,0004527,0004529,0005515,0006259,0006274,0006281,0006308,0008310,0046872,0051575 Ki=32uM remove_due_to_license_issue P04995 20018747 501 KQQSTFLFHDYETFGTHPALDRPAQFAAIRTDSEFNVIGEPEVFYCKPADDYLPQPGAVLITGITPQEARAKGENEAAFAARIHSLFTVPKTCILGYNNVRFDDEVTRNIFYRNFYDPYAWSWQHDNSRWDLLDVMRACYALRPEGINWPENDDGLPSFRLEHLTKANGIEHSDAMADVYATIAMAKLVKTRQPRLFDYLFTHRNKHKLMALIDVPQMKPLVHVSGMFGAWRGNTSWVAPLAWHPENRNAVIMVDLAGDISPLLELDSDTLRERLYTANAAVPVKLVHINKCPVLAQANTLRPEDADRLGINRQHCLDNLKILRENPQVREKVVAIFAEPSDNVDAQLYNGFFSDADRAAMKIVLETEPRNLPALDITFVDKRIEKLLFNYRARNFPGTLDYAEQQRWLEHRRQVFTPEFLQGYADELQMLVQQYADDKEKVALLKALWQYADEIV 3hll A 1.95 BS01 I45 A 1 A51 K53 I84 L104 T106 L108 M109 G110 A111 A47 K49 I80 L100 T102 L104 M105 G106 A107 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=0.0058uM remove_due_to_license_issue IC50=247nM, Kd=2.8nM, Ki=2.9nM Q16539 19496616 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hlo A 1.6 BS01 2NC A 1 D25 G27 A28 D29 D30 I47 G48 R112 D129 G131 A132 D133 D134 G152 D25 G27 A28 D29 D30 I47 G48 R112 D129 G131 A132 D133 D134 G152 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.61uM remove_due_to_license_issue P03369 22158985 204 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNFCGGGGPQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3hmm A 1.7 BS01 855 A 1 A30 K32 L60 L78 S80 Y82 H83 L140 D151 A30 K32 L60 L78 S80 Y82 H83 L140 D151 D133 K135 N138 D151 T175 D133 K135 N138 D151 T170 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.025uM remove_due_to_license_issue IC50=25nM P36897 19285388 857 IARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQ 3hmo A 2.4 BS01 STU A 1 I531 G532 V539 A551 K553 C604 G605 N606 D608 L654 I18 G19 V26 A38 K40 C91 G92 N93 D95 L141 N556 L565 D647 K649 N652 D664 T686 N43 L52 D134 K136 N139 D151 T161 2.7.12.1 0004672,0005524,0005975,0006468 Kd=30.5nM remove_due_to_license_issue P33981 20099905 1 ANECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMVGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 3hmp A 2.3 BS01 CX4 A 1 I531 C604 N606 L654 I16 C89 N91 L139 N556 L565 D647 K649 N652 D664 T686 N41 L50 D132 K134 N137 D149 T161 2.7.12.1 0004672,0005524,0005975,0006468 Kd=3.24uM remove_due_to_license_issue P33981 20099905 1 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMSQVGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 3hmv A 2.23 BS02 HBT A 1 M347 D392 N395 Y403 I410 M411 F414 Q443 F446 M196 D241 N244 Y252 I259 M260 F263 Q292 F295 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=50nM Q07343 19525117 530 SISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIPQNRDCQGLMEKFQFELT 3hnb M 1.15 BS01 768 M 1 K2258 Q2311 S2312 W2313 H2315 K86 Q139 S140 W141 H143 ? remove_due_to_license_issue IC50=7800nM P00451 20089867 1 SCSMPLGMESKAISDAQITASSYFTNMFATWSPSKARLHLQGRSNAWRPQVNNPKEWLQVDFQKTMKVTGVTTQGVKSLLTSMYVKEFLISSSQDGHQWTLFFQNGKVKVFQGNQDSFTPVVNSLDPPLLTRYLRIHPQSWVHQIALRMEVLGCEA 3hng A 2.7 BS01 8ST A 1 K861 E878 V909 Y911 C912 L1029 C1039 D1040 F1041 K58 E75 V106 Y108 C109 L161 C171 D172 F173 D1022 A1024 R1026 N1027 D1040 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=180nM P17948 2001 EVPLDEQCERPYDASKWEFARERLKLGKSLGRGAFGKVVQASAFGIKKSPTCRTVAVKMLKEGATASEYKALMTELKILTHIGHHLNVVNLLGACTKQGGPLMVIVEYCKYGNLSNYLKSKRKEPITMEDLISYSFQVARGMEFLSSRKCIHRDLAARNILLSENNVVKICDFGLARDIYKNPDYVRKTRLPLKWMAPESIFDKIYSTKSDVWSYGVLLWEIFSLGGSPYPGVQMDEDFCSRLREGMRMRAPEYSTPEIYQIMLDCWHRDPKERPRFAELVEKLGDLL 3hnz A 2.75 BS01 PMN A 1 A205 T270 S271 H303 T307 P308 A309 G310 H340 F398 G399 F400 A204 T269 S270 H302 T306 P307 A308 G309 H339 F397 G398 F399 A163 H303 E314 K335 H340 F398 F400 A162 H302 E313 K334 H339 F397 F399 2.3.1.179 0004315,0005515,0005829,0006633,0009409,0016746,0016747,0019367,0042803,0044281,1903966 remove_due_to_license_issue P0AAI5 19581087 413 KRRVVVTGLGMLSPVGNTVESTWKALLAGQSGISLIDHFDTSAYATKFAGLVKDFNCEDIISRKEQRKMDAFIQYGIVAGVQAMQDSGLEITEENATRIGAAIGSGIGGLGLIEENHTSLMNGGPRKISPFFVPSTIVNMVAGHLTIMYGLRGPSISIATAATSGVHNIGHAARIIAYGDADVMVAGGAEKASTPLGVGGFGAARALSTRNDNPQAASRPWDKERDGFVLGDGAGMLVLEEYEHAKKRGAKIYAELVGFGMSSDAYHMTSPPENGAGAALAMANALRDAGIEASQIGYVNAHGTSTPAGDKAEAQAVKTIFGEAASRVLVSSTKSMTGHLLGAAGAVESIYSILALRDQAVPPTINLDNPDEGCDLDFVPHEARQVSGMEYTLCNSFGFGGTNGSLIFKKI 3ho2 A 2.0 BS01 N32 A 1 T270 S271 P272 H303 T307 P308 A309 H340 F398 G399 F400 T269 S270 P271 H302 T306 P307 A308 H339 F397 G398 F399 A163 H303 E314 K335 H340 F398 F400 A162 H302 E313 K334 H339 F397 F399 2.3.1.179 0004315,0005515,0005829,0006633,0009409,0016746,0016747,0019367,0042803,0044281,1903966 ic50=113nM remove_due_to_license_issue P0AAI5 19581087 413 KRRVVVTGLGMLSPVGNTVESTWKALLAGQSGISLIDHFDTSAYATKFAGLVKDFNCEDIISRKEQRKMDAFIQYGIVAGVQAMQDSGLEITEENATRIGAAIGSGIGGLGLIEENHTSLMNGGPRKISPFFVPSTIVNMVAGHLTIMYGLRGPSISIATAATSGVHNIGHAARIIAYGDADVMVAGGAEKASTPLGVGGFGAARALSTRNDNPQAASRPWDKERDGFVLGDGAGMLVLEEYEHAKKRGAKIYAELVGFGMSSDAYHMTSPPENGAGAALAMANALRDAGIEASQIGYVNAHGTSTPAGDKAEAQAVKTIFGEAASRVLVSSTKSMTGHLLGAAGAVESIYSILALRDQAVPPTINLDNPDEGCDLDFVPHEARQVSGMEYTLCNSFGFGGTNGSLIFKKI 3ho9 A 1.9 BS01 N3A A 1 R206 T270 S271 P272 H303 T307 P308 A309 H340 F398 G399 F400 R205 T269 S270 P271 H302 T306 P307 A308 H339 F397 G398 F399 A163 H303 E314 K335 H340 F398 F400 A162 H302 E313 K334 H339 F397 F399 2.3.1.179 0004315,0005515,0005829,0006633,0009409,0016746,0016747,0019367,0042803,0044281,1903966 ic50=789nM remove_due_to_license_issue P0AAI5 19581087 413 KRRVVVTGLGMLSPVGNTVESTWKALLAGQSGISLIDHFDTSAYATKFAGLVKDFNCEDIISRKEQRKMDAFIQYGIVAGVQAMQDSGLEITEENATRIGAAIGSGIGGLGLIEENHTSLMNGGPRKISPFFVPSTIVNMVAGHLTIMYGLRGPSISIATAATSGVHNIGHAARIIAYGDADVMVAGGAEKASTPLGVGGFGAARALSTRNDNPQAASRPWDKERDGFVLGDGAGMLVLEEYEHAKKRGAKIYAELVGFGMSSDAYHMTSPPENGAGAALAMANALRDAGIEASQIGYVNAHGTSTPAGDKAEAQAVKTIFGEAASRVLVSSTKSMTGHLLGAAGAVESIYSILALRDQAVPPTINLDNPDEGCDLDFVPHEARQVSGMEYTLCNSFGFGGTNGSLIFKKI 3hp2 A 2.15 BS01 P36 A 1 V30 A51 K53 L104 T106 H107 M109 G110 A111 L167 L171 V27 A48 K50 L101 T103 H104 M106 G107 A108 L164 L168 D150 K152 N155 D168 T185 D147 K149 N152 D165 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=680nM Q16539 19751974 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQ 3hp5 A 2.3 BS01 52P A 1 A51 K53 L104 V105 T106 M109 G110 A111 D112 A41 K43 L94 V95 T96 M99 G100 A101 D102 D150 K152 N155 D168 T185 D140 K142 N145 D158 T163 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Kd=2.8nM, IC50=70nM, Ki=0.800000nM Q16539 19751974 401 PTFYRQELNKTIWEVPERYQNLSPVGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hp9 A 1.6 BS01 CF1 A 1 P228 W245 A312 N313 R327 C330 L331 R338 P219 W236 A295 N296 R310 C313 L314 R321 3.1.11.1 0000175,0000287,0003676,0003677,0003697,0004527,0004529,0005515,0006259,0006274,0006281,0006308,0008310,0046872,0051575 Ki=26uM remove_due_to_license_issue P04995 20018747 501 QQSTFLFHDYETFGTHPALDRPAQFAAIRTDSEFNVIGEPEVFYCKPADDYLPQPGAVLITGITPQEARAKGENEAAFAARIHSLFTVPKTCILGYNNVRFDDEVTRNIFYRNFYDPYAWSWQHDNSRWDLLDVMRACYALRPEGINWPENDDGLPSFRLEHLTKANGIEHSDAMADVYATIAMAKLVKTRQPRLFDYLFTHRNKHKLMALIDVPQMKPLVHVSGMFGAWRGNTSWVAPLAWHPENRNAVIMVDLAGDISPLLELDSDTLRERLYNAAVPVKLVHINKCPVLAQANTLRPEDADRLGINRQHCLDNLKILRENPQVREKVVAIFAESDNVDAQLYNGFFSDADRAAMKIVLETEPRNLPALDITFVDKRIEKLLFNYRARNFPGTLDYAEQQRWLEHRRQVFTPEFLQGYADELQMLVQQYADDKEKVALLKALWQYADEIV 3hpt B 2.19 BS01 YET B 1 T98 Y99 F174 A190 Q192 V213 W215 G216 G218 C220 G226 Y228 T84 Y85 F162 A180 Q182 V203 W205 G206 G208 C209 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=6.5nM remove_due_to_license_issue IC50=12nM, Ki=6.5nM P00742 19541481 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTRGLP 3hq5 A 2.1 BS01 GKK A 1 L718 N719 M756 M759 L763 F778 F794 M801 L887 Y890 C891 F905 L34 N35 M72 M75 L79 F94 F109 M116 L201 Y204 C205 F219 ? ic50=16nM remove_due_to_license_issue IC50=16nM, EC50=9nM P06401 19595590 934 QLIPPLINLLMSIEPDVIYAGHDNDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 3hqw A 1.7 BS02 PF4 A 1 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 V723 I228 Y229 F232 P248 M249 E257 V258 G261 Q262 F265 V269 3.1.4.17 0004114,0007165,0008081 ic50=35nM remove_due_to_license_issue IC50=35nM Q9QYJ6 19630403 999 PARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3hqy A 2.0 BS02 PF6 A 1 Y514 H515 L665 S667 I682 Y683 F686 P702 M703 G715 Q716 F719 Y62 H63 L213 S215 I230 Y231 F234 P250 M251 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=11.5nM remove_due_to_license_issue IC50=11.5nM Q9QYJ6 19630403 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3hqz A 1.7 BS02 PF8 A 1 Y514 L665 Y683 F686 P702 M703 K708 E711 V712 G715 Q716 F719 Y62 L213 Y231 F234 P250 M251 K256 E259 V260 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=0.42nM remove_due_to_license_issue IC50=0.42nM Q9QYJ6 19630403 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3hr1 A 1.53 BS01 PF9 A 1 L665 Y683 F686 P702 M703 K708 E711 V712 G715 Q716 F719 L213 Y231 F234 P250 M251 K256 E259 V260 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=0.37nM remove_due_to_license_issue IC50=0.5nM, Ki=0.17nM Q9QYJ6 19630403 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3hrb A 2.2 BS01 I39 A 1 V30 A51 K53 L104 T106 M109 G110 A111 V27 A43 K45 L96 T98 M101 G102 A103 D150 K152 N155 D168 T185 D142 K144 N147 D160 T177 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=21nM remove_due_to_license_issue IC50=21nM Q16539 19678708 1 ERPTFYRQELNKTIWEVPERYQNLSPVGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hrf A 1.9 BS02 P47 A 1 K76 K115 I119 R131 T148 L155 F157 K2 K41 I45 R57 T74 L81 F83 D205 K207 E209 N210 D223 T245 D131 K133 E135 N136 D149 T171 2.7.11.1 0004672,0004674,0005524,0006468 Kd=10.3uM remove_due_to_license_issue Kd=10300nM, IC50=9.7e+4nM O15530 19718043 1374 RKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3hs4 A 1.1 BS03 AZM A 1 Q92 H94 H119 V121 F131 L198 T199 T200 Q89 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 19851004 701 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3hs4 A 1.1 BS04 AZM A 2 Y114 K213 E214 P215 Y111 K209 E210 P211 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 19851004 702 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3hs4 A 1.1 BS05 AZM A 3 H4 H15 D19 H1 H12 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10nM remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 19851004 703 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ht3 A 1.7 BS01 dna B 0 T550 T552 T556 A558 R578 Y587 R615 Q624 N625 I626 P627 I628 R629 H829 D830 T253 T255 T259 A261 R281 Y290 R318 Q327 N328 I329 P330 I331 R332 H532 D533 2.7.7.7 0000166,0003676,0003677,0003887,0004527,0006139,0006259,0006260,0006261,0006281,0006302,0008408,0034061,0046872,0071897 remove_due_to_license_issue D9N168 21454515 21 ~ 29 KMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNFGIPYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 3ht3 A 1.7 BS02 dna C 0 N527 N529 S530 S585 L610 T611 Q612 T613 R615 S617 S618 T619 E620 N622 Y714 I716 S717 Y719 G720 R771 F786 R789 M790 N793 Q797 N230 N232 S233 S288 L313 T314 Q315 T316 R318 S320 S321 T322 E323 N325 Y417 I419 S420 Y422 G423 R474 F489 R492 M493 N496 Q500 2.7.7.7 0000166,0003676,0003677,0003887,0004527,0006139,0006259,0006260,0006261,0006281,0006302,0008408,0034061,0046872,0071897 remove_due_to_license_issue D9N168 21454515 1 ~ 12 KMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNFGIPYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 3ht3 D 1.7 BS01 dna E 0 T550 K551 T552 T556 A558 R578 K582 Y587 R615 Q624 N625 I626 P627 I628 R629 H829 T253 K254 T255 T259 A261 R281 K285 Y290 R318 Q327 N328 I329 P330 I331 R332 H532 2.7.7.7 0000166,0003676,0003677,0003887,0004527,0006139,0006259,0006260,0006261,0006281,0006302,0008408,0034061,0046872,0071897 remove_due_to_license_issue D9N168 21454515 21 ~ 29 KMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNFGIPYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 3ht3 D 1.7 BS02 dna F 0 N527 S530 K582 S585 T586 L610 T611 Q612 T613 R615 S617 S618 T619 E620 N622 Y714 I716 S717 Y719 R771 N782 F786 R789 M790 N793 Q797 N230 S233 K285 S288 T289 L313 T314 Q315 T316 R318 S320 S321 T322 E323 N325 Y417 I419 S420 Y422 R474 N485 F489 R492 M493 N496 Q500 2.7.7.7 0000166,0003676,0003677,0003887,0004527,0006139,0006259,0006260,0006261,0006281,0006302,0008408,0034061,0046872,0071897 remove_due_to_license_issue D9N168 21454515 1 ~ 12 KMAFTLADRVTEEMLADKAALVVEVVEENYHDAPIVGIAVVNEHGRFFLRPETALADPQFVAWLGDETKKKSMFDSKRAAVALKWKGIELCGVSFDLLLAAYLLDPAQGVDDVAAAAKMKQYEAVRPDEAVYGKGAKRAVPDEPVLAEHLVRKAAAIWELERPFLDELRRNEQDRLLVELEQPLSSILAEMEFAGVKVDTKRLEQMGKELAEQLGTVEQRIYELAGQEFNINSPKQLGVILFEKLQLPVLKKTKTGYSTSADVLEKLAPYHEIVENILHYRQLGKLQSTYIEGLLKVVRPATKKVHTIFNQALTQTGRLSSTEPNLQNIPIRLEEGRKIRQAFVPSESDWLIFAADYSQIELRVLAHIAEDDNLMEAFRRDLDIHTKTAMDIFQVSEDEVTPNMRRQAKAVNFGIPYGISDYGLAQNLNISRKEAAEFIERYFESFPGVKRYMENIVQEAKQKGYVTTLLHRRRYLPDITSRNFNVRSFAERMAMNTPIQGSAADIIKKAMIDLNARLKEERLQAHLLLQVHDELILEAPKEEMERLCRLVPEVMEQAVTLRVPLKVDYHYGSTWYDAK 3hu1 A 2.81 BS01 AGS A 1 I206 G207 P247 G248 T249 G250 K251 T252 L253 N348 I380 H384 G408 A409 I195 G196 P236 G237 T238 G239 K240 T241 L242 N337 I369 H373 G397 A398 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVGLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 3hu1 A 2.81 BS02 AGS F 1 R359 F360 R348 F349 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVGLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 3hu1 B 2.81 BS01 AGS A 1 R359 F360 R348 F349 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVGLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 3hu1 B 2.81 BS02 AGS B 1 I206 G207 P247 G248 T249 G250 K251 T252 L253 N348 I380 H384 G408 A409 I195 G196 P236 G237 T238 G239 K240 T241 L242 N337 I369 H373 G397 A398 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVGLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 3hu2 A 2.85 BS01 AGS A 1 I206 G207 P247 G248 T249 G250 K251 T252 L253 N348 I380 H384 G408 A409 I195 G196 P236 G237 T238 G239 K240 T241 L242 N337 I369 H373 G397 A398 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNAVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSA 3hu2 A 2.85 BS02 AGS F 1 R359 F360 R348 F349 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNAVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSA 3hu2 B 2.85 BS01 AGS A 1 R359 F360 R348 F349 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNAVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSA 3hu2 B 2.85 BS02 AGS B 1 I206 G207 P247 G248 T249 G250 K251 T252 L253 N348 H384 G408 A409 I195 G196 P236 G237 T238 G239 K240 T241 L242 N337 H373 G397 A398 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 20512113 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNAVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSA 3hu3 A 2.2 BS01 AGS A 1 G207 P247 G248 T249 G250 K251 T252 L253 N348 H384 G408 A409 G191 P231 G232 T233 G234 K235 T236 L237 N332 H368 G392 A393 3.6.4.6 0005524,0016887 Kd=0.13uM remove_due_to_license_issue P55072 20512113 800 LKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSALRETVV 3hu3 B 2.2 BS01 AGS B 1 G207 P247 G248 T249 G250 K251 T252 L253 N348 I380 H384 G408 A409 G191 P231 G232 T233 G234 K235 T236 L237 N332 I364 H368 G392 A393 3.6.4.6 0005524,0016887 Kd=0.13uM remove_due_to_license_issue P55072 20512113 800 LKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 3hub A 2.25 BS01 469 A 1 V30 Y35 A51 K53 L104 T106 M109 G110 A111 N115 V27 Y32 A48 K50 L101 T103 M106 G107 A108 N112 D150 K152 N155 D168 T185 D147 K149 N152 D165 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=8.2nM remove_due_to_license_issue IC50=9nM, Kd=0.480000nM Q16539 20201574 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPP 3huc A 1.8 BS01 G97 A 1 Y35 V38 K53 L104 T106 F169 Y32 V35 K50 L101 T103 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=1030nM remove_due_to_license_issue Q16539 20201574 362 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hv3 A 2.0 BS01 R49 A 1 V30 A51 K53 E71 M78 I84 T106 M109 L167 D168 F169 G170 V27 A45 K47 E65 M72 I78 T100 M103 L161 D162 F163 G164 D150 K152 N155 D168 T185 D144 K146 N149 D162 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=900nM remove_due_to_license_issue IC50=900nM Q16539 19928858 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPPL 3hv4 A 2.6 BS01 L51 A 1 V30 K53 R67 E71 M109 L167 D168 F169 V27 K50 R64 E68 M106 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T172 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=290nM Q16539 19928858 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hv5 A 2.25 BS01 R24 A 1 V30 A51 K53 E71 T106 M109 H148 L167 D168 F169 V27 A48 K50 E68 T103 M106 H145 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T172 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=150nM remove_due_to_license_issue IC50=95nM Q16539 19928858 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hv6 A 1.95 BS01 R39 A 1 E71 M78 I84 L108 M109 H148 L167 D168 F169 E64 M71 I77 L101 M102 H139 L158 D159 F160 D150 K152 N155 D168 T185 D141 K143 N146 D159 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=5500nM remove_due_to_license_issue IC50=5500nM, koff=0.003900s-1, kon=13000M-1-s-1, Kd=300nM Q16539 19928858 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hv7 A 2.4 BS01 1AU A 1 K53 E71 L75 M78 I84 L104 T106 H148 L167 D168 F169 K46 E64 L68 M71 I77 L97 T99 H137 L156 D157 F158 D150 K152 N155 D168 T185 D139 K141 N144 D157 T163 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd~12nM remove_due_to_license_issue Kd=12nM, IC50=170nM Q16539 19928858 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hv8 A 1.445 BS01 C2E A 1 Q461 L477 L478 R479 P490 L494 H533 F652 E654 G672 Y673 Q21 L37 L38 R39 P50 L54 H88 F207 E209 G227 Y228 3.1.4.52 0071111 Kd=104.2nM remove_due_to_license_issue Q9HUK6 19679088 900 GDVIAILQQALETNSFRLLFQPVISLRGDSHENYEVLLRLLNPQGQEVPPAEFLHAAKEAGLAEKIDRWVILNSIKLLAEHQTKLFVHLSSASLQDPGLLPWLGVALKAARLPPESLVFQISEADATSYLKQAKQLTQGLATLHCQAAISQFGCSLNPFNALKHLTVQFIKIDGSFVQDLNQVENQEILKGLIAELHEQQKLSIVPFVESASVLATLWQAGATYIQGYYLQGPSQAMDYDFS 3hvc A 2.1 BS01 GG5 A 1 V38 A51 K53 L104 V105 T106 L108 M109 L167 V31 A44 K46 L97 V98 T99 L101 M102 L156 D150 K152 N155 D168 T185 D139 K141 N144 D157 T160 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=600nM remove_due_to_license_issue Ki=600nM, IC50=67nM Q16539 19501598 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hvc A 2.1 BS02 GG5 A 2 P191 E192 L195 W197 P242 L246 I259 L291 S293 P166 E167 L170 W172 P217 L221 I234 L266 S268 D150 K152 N155 D168 T185 D139 K141 N144 D157 T160 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=600nM remove_due_to_license_issue Ki=600nM, IC50=67nM Q16539 19501598 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3hvg A 2.26 BS01 EV0 A 1 D32 Y71 T72 Q73 W115 D228 D37 Y76 T77 Q78 W120 D222 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50~2mM remove_due_to_license_issue Kd=4450000nM P56817 19799414 441 TGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3hvh A 1.3 BS01 542 A 1 M83 Y111 E133 M134 A161 S162 Q163 D184 H185 W186 K187 R189 N213 P217 L241 E242 M38 Y66 E88 M89 A116 S117 Q118 D139 H140 W141 K142 R144 N168 P172 L196 E197 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=3nM remove_due_to_license_issue P22734 19882607 1 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3hvi A 1.2 BS02 619 A 1 W81 M83 Y111 E133 M134 S162 Q163 D184 H185 W186 K187 N213 P217 L241 E242 W36 M38 Y66 E88 M89 S117 Q118 D139 H140 W141 K142 N168 P172 L196 E197 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=5nM remove_due_to_license_issue P22734 19882607 267 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3hvj A 1.79 BS01 705 A 1 W81 M83 Y111 E133 M134 A161 S162 Q163 D184 H185 W186 K187 R189 N213 P217 E242 W36 M38 Y66 E88 M89 A116 S117 Q118 D139 H140 W141 K142 R144 N168 P172 E197 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=2nM remove_due_to_license_issue P22734 19882607 1 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3hvk A 1.3 BS02 719 A 1 W81 M83 E133 M134 S162 Q163 D184 H185 W186 K187 N213 V216 P217 L241 E242 W36 M38 E88 M89 S117 Q118 D139 H140 W141 K142 N168 V171 P172 L196 E197 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=3nM remove_due_to_license_issue P22734 19882607 267 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3hw1 A 2.48 BS01 EV2 A 1 D32 G34 Y71 D228 D36 G38 Y75 D219 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.87mM remove_due_to_license_issue P56817 19799414 393 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3hwn A 2.33 BS01 BD3 A 1 C25 E63 G68 L69 M70 D71 A135 M161 D162 C25 E63 G68 L69 M70 D71 A135 M161 D162 Q19 C25 H163 N187 Q19 C25 H163 N180 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 19616430 221 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDAGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3hww A 1.95 BS01 AKG A 1 S391 L392 G441 D442 L443 S444 S391 L392 G441 D442 L443 S444 2.2.1.9 0000287,0003824,0009234,0016740,0030145,0030976,0042803,0044281,0046872,0070204 Kd=75nM remove_due_to_license_issue P17109 19703421 557 MSVSAFNRRWAAVILEALTRHGVRHICIAPGSRSTLLTLAAAENSAFIHHTHFDERGLGHLALGLAKVSKQPVAVIVTSGTAVANLYPALIEAGLTGEKLILLTADRPPELIDCGANQAIRQPGMFASHPTHSISLPRPTQDIPARWLVSTIDHALGTLHAGGVHINCPFAEPLYGEMDDTGLSWQQRLGDWWQDDKPWLREAPRLESEKQRDWFFWRQKRGVVVAGRMSAEEGKKVALWAQTLGWPLIGDVLSQTGQPLPCADLWLGNAKATSELQQAQIVVQLGSSLTGKRLLQWQASCEPEEYWIVDDIEGRLDPAHHRGRRLIANIADWLELHPAEKRQPWCVEIPRLAEQAMQAVIARRDAFGEAQLAHRICDYLPEQGQLFVGNSLVVRLIDALSQLPAGYPVYSNRGASGIDGLLSTAAGVQRASGKPTLAIVGDLSALYDLNALALLRQVSAPLVLIVVNNNGYLMPQNVHFEHAAAMFELKYHRPQNWQELETAFADAWRTPTTTVIEMVVNDTDGAQTLQQLLAQVSHL 3hww D 1.95 BS01 AKG D 1 E369 S391 L392 V393 L443 N469 E366 S388 L389 V390 L440 N466 2.2.1.9 0000287,0003824,0009234,0016740,0030145,0030976,0042803,0044281,0046872,0070204 Kd=75nM remove_due_to_license_issue P17109 19703421 557 SVSAFNRRWAAVILEALTRHGVRHICIAPGSRSTLLTLAAAENSAFIHHTHFDERGLGHLALGLAKVSKQPVAVIVTSGTAVANLYPALIEAGLTGEKLILLTADRPPELIDCGANQAIRQPGMFASHPTHSISLPRPTQDIPARWLVSTIDHALGTLHAGGVHINCPFAEPLEMDDTGLSWQQRLGDWWQDDKPWLREAPRLESEKQRDWFFWRQKRGVVVAGRMSAEEGKKVALWAQTLGWPLIGDVLSQTGQPLPCADLWLGNAKATSELQQAQIVVQLGSSLTGKRLLQWQASCEPEEYWIVDDIEGRLDPAHHRGRRLIANIADWLELHPAEKRQPWCVEIPRLAEQAMQAVIARRDAFGEAQLAHRICDYLPEQGQLFVGNSLVVRLIDALSQLPAGYPVYSNRGASGIDGLLSTAAGVQRASGKPTLAIVGDLSALYDLNALALLRQVSAPLVLIVVNNNGQNVHFEHAAAMFELKYHRPQNWQELETAFADAWRTPTTTVIEMVVNDTDGAQTLQQLLAQVSHL 3hwx A 2.6 BS01 TPP A 1 S391 L392 I418 D419 G441 D442 L443 S444 N469 G471 G472 Q473 S390 L391 I417 D418 G440 D441 L442 S443 N468 G470 G471 Q472 2.2.1.9 0000287,0003824,0009234,0016740,0030145,0030976,0042803,0044281,0046872,0070204 remove_due_to_license_issue P17109 19703421 601 MSVSAFNRRWAAVILEALTRHGVRHICIAPGSRSTLLTLAAAENSAFIHHTHFDERGLGHLALGLAKVSKQPVAVIVTSGTAVANLYPALIEAGLTGEKLILLTADRPPELIDCGANQAIRQPGMFASHPTHSISLPRPTQDIPARWLVSTIDHALGTLHAGGVHINCPFAEPLYGMDDTGLSWQQRLGDWWQDDKPWLREAPRLESEKQRDWFFWRQKRGVVVAGRMSAEEGKKVALWAQTLGWPLIGDVLSQTGQPLPCADLWLGNAKATSELQQAQIVVQLGSSLTGKRLLQWQASCEPEEYWIVDDIEGRLDPAHHRGRRLIANIADWLELHPAEKRQPWCVEIPRLAEQAMQAVIARRDAFGEAQLAHRICDYLPEQGQLFVGNSLVVRLIDALSQLPAGYPVYSNRGASGIDGLLSTAAGVQRASGKPTLAIVGDLSALYDLNALALLRQVSAPLVLIVVNNNGGQIFSLLPTPQSERERFYLMPQNVHFEHAAAMFELKYHRPQNWQELETAFADAWRTPTTTVIEMVVNDTDGAQTLQQLLAQVSHL 3hwx A 2.6 BS03 TPP B 1 E55 A82 E55 A82 2.2.1.9 0000287,0003824,0009234,0016740,0030145,0030976,0042803,0044281,0046872,0070204 remove_due_to_license_issue P17109 19703421 601 MSVSAFNRRWAAVILEALTRHGVRHICIAPGSRSTLLTLAAAENSAFIHHTHFDERGLGHLALGLAKVSKQPVAVIVTSGTAVANLYPALIEAGLTGEKLILLTADRPPELIDCGANQAIRQPGMFASHPTHSISLPRPTQDIPARWLVSTIDHALGTLHAGGVHINCPFAEPLYGMDDTGLSWQQRLGDWWQDDKPWLREAPRLESEKQRDWFFWRQKRGVVVAGRMSAEEGKKVALWAQTLGWPLIGDVLSQTGQPLPCADLWLGNAKATSELQQAQIVVQLGSSLTGKRLLQWQASCEPEEYWIVDDIEGRLDPAHHRGRRLIANIADWLELHPAEKRQPWCVEIPRLAEQAMQAVIARRDAFGEAQLAHRICDYLPEQGQLFVGNSLVVRLIDALSQLPAGYPVYSNRGASGIDGLLSTAAGVQRASGKPTLAIVGDLSALYDLNALALLRQVSAPLVLIVVNNNGGQIFSLLPTPQSERERFYLMPQNVHFEHAAAMFELKYHRPQNWQELETAFADAWRTPTTTVIEMVVNDTDGAQTLQQLLAQVSHL 3hwx B 2.6 BS01 TPP A 1 P30 E55 A82 P30 E55 A82 2.2.1.9 0000287,0003824,0009234,0016740,0030145,0030976,0042803,0044281,0046872,0070204 remove_due_to_license_issue P17109 19703421 601 MSVSAFNRRWAAVILEALTRHGVRHICIAPGSRSTLLTLAAAENSAFIHHTHFDERGLGHLALGLAKVSKQPVAVIVTSGTAVANLYPALIEAGLTGEKLILLTADRPPELIDCGANQAIRQPGMFASHPTHSISLPRPTQDIPARWLVSTIDHALGTLHAGGVHINCPFAEPLYGEMDDTGLSWQQRLGDWWQDDKPWLREAPRLESEKQRDWFFWRQKRGVVVAGRMSAEEGKKVALWAQTLGWPLIGDVLSQTGQPLPCADLWLGNAKATSELQQAQIVVQLGSSLTGKRLLQWQASCEPEEYWIVDDIEGRLDPAHHRGRRLIANIADWLELHPAEKRQPWCVEIPRLAEQAMQAVIARRDAFGEAQLAHRICDYLPEQGQLFVGNSLVVRLIDALSQLPAGYPVYSNRGASGIDGLLSTAAGVQRASGKPTLAIVGDLSALYDLNALALLRQVSAPLVLIVVNNNGGQIFSLLPTPQSERERFYLMPQNVHFEHAAAMFELKYHRPQNWQELETAFADAWRTPTTTVIEMVVNDTDGAQTLQQLLAQVSHL 3hwx B 2.6 BS02 TPP B 1 S391 L392 G417 I418 D419 G441 D442 L443 S444 N469 G471 G472 Q473 I474 S391 L392 G417 I418 D419 G441 D442 L443 S444 N469 G471 G472 Q473 I474 2.2.1.9 0000287,0003824,0009234,0016740,0030145,0030976,0042803,0044281,0046872,0070204 remove_due_to_license_issue P17109 19703421 601 MSVSAFNRRWAAVILEALTRHGVRHICIAPGSRSTLLTLAAAENSAFIHHTHFDERGLGHLALGLAKVSKQPVAVIVTSGTAVANLYPALIEAGLTGEKLILLTADRPPELIDCGANQAIRQPGMFASHPTHSISLPRPTQDIPARWLVSTIDHALGTLHAGGVHINCPFAEPLYGEMDDTGLSWQQRLGDWWQDDKPWLREAPRLESEKQRDWFFWRQKRGVVVAGRMSAEEGKKVALWAQTLGWPLIGDVLSQTGQPLPCADLWLGNAKATSELQQAQIVVQLGSSLTGKRLLQWQASCEPEEYWIVDDIEGRLDPAHHRGRRLIANIADWLELHPAEKRQPWCVEIPRLAEQAMQAVIARRDAFGEAQLAHRICDYLPEQGQLFVGNSLVVRLIDALSQLPAGYPVYSNRGASGIDGLLSTAAGVQRASGKPTLAIVGDLSALYDLNALALLRQVSAPLVLIVVNNNGGQIFSLLPTPQSERERFYLMPQNVHFEHAAAMFELKYHRPQNWQELETAFADAWRTPTTTVIEMVVNDTDGAQTLQQLLAQVSHL 3hx3 A 1.69 BS01 RET A 1 F161 F173 Y180 E202 F204 L220 M223 F240 F105 F117 Y124 E146 F148 L164 M167 F184 ? 0005502,0005515,0005654,0005737,0005813,0005829,0006776,0007601,0019841,0044297,1902936 Kd~10nM remove_due_to_license_issue P12271 19846785 400 ETREEAVRELQEMVQAQAASGEELAVAVAERVQEKDSGFFLRFIRARKFNVGRAYELLRGYVNFRLQYPELFDSLSPEAVRCTIEAGYPGVLSSRDKYGRVVMLFNIENWQSQEITFDEILQAYCFILEKLLENEETQINGFCIIENFKGFTMQQAASLRTSDLRKMVDMLQDSFPAWFKAIHFIHQPWYFTTTYNVVKPFLKSKLLERVFVHGDDLSGFYQEIDENILPSDFGGTLPKYDGKAVAEQLF 3hxb B 2.25 BS01 BD5 B 1 S48 L96 R144 F147 G192 Q193 Y195 W244 S41 L89 R137 F140 G185 Q186 Y188 W237 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 remove_due_to_license_issue Q08603 19894725 332 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3hxc B 1.95 BS03 BD6 B 1 W52 R144 F147 G192 Q193 D238 C240 W244 F289 W44 R136 F139 G184 Q185 D230 C232 W236 F281 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H182 R224 K227 D230 C232 Y233 D272 D279 H282 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 remove_due_to_license_issue Q08603 19894725 334 QKDVTIKSDAPDTLLLEKHADYIASYGSYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3hxd B 1.95 BS03 BD7 B 1 W52 L96 R144 C148 G192 Q193 C196 D238 C240 W244 F289 W45 L89 R137 C141 G185 Q186 C189 D231 C233 W237 F282 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 remove_due_to_license_issue Q08603 19894725 334 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3hxe B 1.95 BS03 BD8 B 1 G49 W52 L96 R144 G192 Q193 D238 C240 W244 P288 F289 H290 F293 C314 G42 W45 L89 R137 G185 Q186 D231 C233 W237 P281 F282 H283 F286 C307 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 remove_due_to_license_issue Q08603 19894725 334 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3hxf B 1.9 BS03 BD9 B 1 Y44 L45 S48 Y51 W52 Y97 F147 G192 C240 Y241 W244 F289 H290 F293 Y36 L37 S40 Y43 W44 Y89 F139 G184 C232 Y233 W236 F281 H282 F285 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H182 R224 K227 D230 C232 Y233 D272 D279 H282 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 remove_due_to_license_issue Q08603 19894725 334 QKDVTIKSDAPDTLLLEKHADYIASYGSYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELV 3hxi A 1.8 BS02 GTG A 1 F37 W43 G75 K88 W89 E90 Q141 R143 K148 W152 R192 F17 W23 G55 K68 W69 E70 Q121 R123 K128 W132 R172 0003723,0003743,0005737,0006413 remove_due_to_license_issue 19710013 501 EFPHPLQDSWSYYLFQFRKALDWDECLEKVATFSTIEDFWSVLTHTVRPREITYGKDLYMFKSDIMPKWEDPKNENGGRWLINVTARQDVDFLWDELLMLLIGSDWDTDEEDRQICGAVFQPRSRGSKLSVWLTSDNEEETILSIGRRIKERLELEDTIYFQPVSDQRSQTRGSDCTGKYEI 3hxo A 2.4 BS01 dna B 0 K599 F603 Q625 E626 Q628 R629 S631 R632 N633 Y637 A657 L659 K660 K93 F97 Q119 E120 Q122 R123 S125 R126 N127 Y131 A151 L153 K154 ? remove_due_to_license_issue P04275 19913482 1 ~ 40 FYCSRLLDLVFLLDGSSRLSEAEFEVLKAFVVDMMERLRISQKWVRVAVVEYHDGSHAYIGLKDRKRPSELRRIASQVKYAGSQVASTSEVLKYTLFQIFSKIDRPEASRIALLLMASQEPQRMSRNFVRYVQGLKKKKVIVIPVGIGPHANLKQIRLIEKQAPENKAFVLSSVDELEQQRDEIVSYLCDLAPEAPPPT 3hxq A 2.694 BS01 dna B 0 R524 F603 Q625 E626 P627 Q628 R629 S631 R632 N633 R636 Y637 L659 K660 R23 F102 Q124 E125 P126 Q127 R128 S130 R131 N132 R135 Y136 L158 K159 ? remove_due_to_license_issue P04275 19913482 1 ~ 41 PPLHDFYCSRLLDLVFLLDGSSRLSEAEFEVLKAFVVDMMERLRISQKWVRVAVVEYHDGSHAYIGLKDRKRPSELRRIASQVKYAGSQVASTSEVLKYTLFQIFSKIDRPEASRIALLLMASQEPQRMSRNFVRYVQGLKKKKVIVIPVGIGPHANLKQIRLIEKQAPENKAFVLSSVDELEQQRDEIVSYLCDLAPEAP 3hy5 A 3.04 BS01 RET A 1 F161 F173 Y180 E202 F204 M223 F240 F247 V266 F139 F151 Y158 E180 F182 M201 F218 F225 V244 ? 0005502,0005515,0005654,0005737,0005813,0005829,0006776,0007601,0019841,0044297,1902936 remove_due_to_license_issue P12271 19846785 400 EQLTTKDHGPVFGPCSQLPRHTLQKAKDELNEREETREEAVRELQEMVQAQAASGEELAVAVAERVQEKDSGFFLRFIRARKFNVGRAYELLRGYVNFRLQYPELFDSLSPEAVRCTIEAGYPGVLSSRDKYGRVVMLFNIENWQSQEITFDEILQAYCFILEKLLENEETQINGFCIIENFKGFTMQQAASLRTSDLRKMVDMLQDSFPARFKAIHFIHQPWYFTTTYNVVKPFLKSKLLERVFVHGDDLSGFYQEIDENILPSDFGGTLPKYDGKAVAEQLF 3hy7 A 1.69 BS01 097 A 1 D377 T378 L379 G380 H410 E411 H414 H420 S441 I442 L443 D114 T115 L116 G117 H147 E148 H151 H157 S178 I179 L180 3.4.24.- 0004222,0006508,0008237 ic50=106nM remove_due_to_license_issue IC50=10000nM Q9UNA0 19586907 801 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hy9 A 2.02 BS05 098 A 1 H373 D377 T378 L379 G380 T407 H410 E411 H414 H420 S440 S441 L443 H110 D114 T115 L116 G117 T144 H147 E148 H151 H157 S177 S178 L180 3.4.24.- 0004222,0006508,0008237 ic50=17nM remove_due_to_license_issue IC50=12nM Q9UNA0 19586907 801 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyf A 1.7 BS03 ON1 A 1 D443 D498 H539 D18 D73 H122 D443 G444 E478 D498 H539 D549 D18 G19 E53 D73 H122 D132 3.1.26.13,3.1.26.4 0003676,0004523 ic50=1.2uM remove_due_to_license_issue P0A7Y4,Q72547 19791799 701 MYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIITQWIHNWKKRGWPVKNVDLVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRKVL 3hyg A 1.4 BS05 099 A 1 D377 T378 L379 T407 H410 E411 H414 H420 S440 S441 I442 L443 D114 T115 L116 T144 H147 E148 H151 H157 S177 S178 I179 L180 3.4.24.- 0004222,0006508,0008237 ic50=93nM remove_due_to_license_issue Q9UNA0 19586907 801 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hzi B 2.98 BS01 dna T 0 T27 Q28 Q39 S43 T24 Q25 Q36 S40 ? 0000976,0001046,0001217,0003677,0005515,0006351,0006355,0032993,0040008,0042803,0043565,0045892,0110001 remove_due_to_license_issue P23873 19150849 699 ~ 719 FQKIYSPTQLANAMKLVRQQNGWTQSELAKKIGIKQATISNFENNPDNTTLTTFFKILQSLELSMTLCDAK 3hzy A 2.1 BS01 KDA C 1 N27D R27F N31 R33 remove_due_to_license_issue 20000757 1 DIVMTQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTISSVQAEDLAVYYCKQSYNLRTFGGGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDIAVKWKIDGSERNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 3i06 A 1.1 BS01 QL2 A 1 G23 C25 S64 G66 L67 D161 H162 G163 G23 C25 S64 G66 L67 D161 H162 G163 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue IC50=10nM P25779 19908842 220 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 3i0r A 2.98 BS01 RT3 A 1 L100 K102 K103 K104 S105 V106 Y181 Y188 W229 L234 H235 P236 Y318 L101 K103 K104 K105 S106 V107 Y182 Y189 W230 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 19631528 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGG 3i0s A 2.7 BS01 RT7 A 1 L100 K102 K103 K104 V106 V179 Y181 Y188 F227 W229 L234 H235 P236 Y318 L101 K103 K104 K105 V107 V180 Y182 Y189 F228 W230 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 19631528 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3i1y A 2.469 BS01 33N A 1 D335 W336 Y383 Q384 L408 M419 Y466 V498 H524 W525 D332 W333 Y380 Q381 L405 M416 Y463 V495 H521 W522 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F264 H331 D332 W333 N356 N375 Y380 Y463 D493 H521 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=7nM remove_due_to_license_issue IC50=7nM P34913 19746975 999 RAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 3i25 A 2.1 BS01 MV7 A 1 G11 Q12 G13 L30 D32 G34 S35 P70 Y71 T72 Q73 G74 F108 I110 Y198 I226 D228 G230 T231 T232 N233 R235 T329 A335 G14 Q15 G16 L33 D35 G37 S38 P73 Y74 T75 Q76 G77 F111 I113 Y190 I218 D220 G222 T223 T224 N225 R227 T317 A323 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 Ki=3.1nM remove_due_to_license_issue Ki=3.1nM P56817 20122837 531 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3i28 A 1.95 BS01 34N A 1 F267 D335 W336 M339 Y383 L408 M419 Y466 F497 V498 H524 F264 D332 W333 M336 Y380 L405 M416 Y463 F494 V495 H521 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F264 H331 D332 W333 N356 N375 Y380 Y463 D493 H521 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=6nM remove_due_to_license_issue IC50=8nM, EC50=0.14nM P34913 19746975 999 RAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 3i3b A 2.2 BS01 149 A 1 D201 H391 N460 E461 M502 Y503 E537 H540 W568 F601 N604 D189 H379 N448 E449 M490 Y491 E525 H528 W556 F589 N592 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5.9mM remove_due_to_license_issue P00722 20921997 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAAGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3i3b D 2.2 BS01 149 D 1 D201 H391 E461 M502 Y503 E537 H540 W568 F601 D189 H379 E449 M490 Y491 E525 H528 W556 F589 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=5.9mM remove_due_to_license_issue P00722 20921997 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAAGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3i3d A 2.2 BS01 IPT A 1 N102 D201 E461 E537 H540 N604 W999 N90 D189 E449 E525 H528 N592 W987 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=10.3mM remove_due_to_license_issue Ki=7.6e+4nM P00722 20921997 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAAGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3i3d A 2.2 BS02 IPT A 2 E304 R645 D648 Q702 W708 E292 R633 D636 Q690 W696 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=10.3mM remove_due_to_license_issue Ki=7.6e+4nM P00722 20921997 2002 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAAGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3i3d D 2.2 BS01 IPT D 1 N102 D201 E461 E537 H540 N604 W999 N90 D189 E449 E525 H528 N592 W987 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=10.3mM remove_due_to_license_issue Ki=7.6e+4nM P00722 20921997 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAAGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3i3d D 2.2 BS02 IPT D 2 E304 P306 R645 D648 W708 E292 P294 R633 D636 W696 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=10.3mM remove_due_to_license_issue Ki=7.6e+4nM P00722 20921997 2002 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAAGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3i4a A 1.898 BS01 LN5 A 1 L30 D73 F76 D79 R98 G129 R145 H173 V268 D269 C274 L23 D66 F69 D72 R91 G122 R138 H166 V261 D262 C267 3.5.3.18 0000052,0003073,0003824,0005829,0006525,0006527,0007263,0008285,0016403,0016597,0016787,0043116,0045429,0045766,0046209,0046872,0070062,1900038 remove_due_to_license_issue Ki=5.2e+4nM, IC50=300000nM O94760 19663506 500 AAFGRATHAVVRALPESLGQHALRSAKGEEVDVARAERQHQLYVGVLGSKLGLQVVELPADESLPDCVFVEDVAVVCEETALITRPGAPSRRKEVDMMKEALEKLQLNIVEMKDENATLDGGDVLFTGREFFVGLSKRTNQRGAEILADTFKDYAVSTVPVADGLHLKSFCSMAGPNLIAIGSSESAQKALKIMQQMSDHRYDKLTVPDDIAANCIYLNIPNKGHVLLHRTPEEYPESAKVYEKLKDHMLIPVSMSELEKVDGLLTCCSVLINKK 3i4b A 2.3 BS01 Z48 A 1 N64 G65 S66 G68 V70 A83 K85 V135 P136 L188 C199 D200 N38 G39 S40 G42 V44 A57 K59 V109 P110 L162 C173 D174 D181 K183 N186 D200 S219 D155 K157 N160 D174 S193 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 Ki=7nM remove_due_to_license_issue Ki=7nM P49841 19827834 501 SMKVSRDGSKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQ 3i4b B 2.3 BS01 Z48 B 1 N64 G65 S66 G68 V70 A83 K85 Y134 V135 P136 L188 C199 D200 N29 G30 S31 G33 V35 A48 K50 Y99 V100 P101 L153 C164 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 Ki=7nM remove_due_to_license_issue Ki=7nM P49841 19827834 501 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 3i4y A 1.85 BS02 35C A 1 L77 V81 I102 P105 Y106 Y162 Y196 R217 H222 L53 V57 I78 P81 Y82 Y138 Y172 R193 H198 Y162 Y196 R217 H220 H222 Y138 Y172 R193 H196 H198 1.13.11.1 0003824,0005506,0008199,0009056,0009712,0016702,0018576,0046872,0051213 Ki=0.09uM remove_due_to_license_issue P95607 20040374 1 ATADTSPERLAAIAKDALGALNDVILKHGVTYPEYRVFKQWLIDVGEGGEWPLFLDVFIEHSVEEVLARSRKGTMGSIEGPYYIENSPELPSKCTLPMREEDEKITPLVFSGQVTDLDGNGLAGAKVELWHADNDGYYSQFAPHLPEWNLRGTIIADEEGRYEITTIQPAPYQIPTDGPTGQFIEAQNGHPWRPAHLHLIVSAPGKESVTTQLYFKGGEWIDSDVASATKPELILDPKTGDDGKNYVTYNFVLDPA 3i51 A 1.8 BS02 45C A 1 D80 V81 P105 Y106 Y162 Y196 R217 H220 H222 D56 V57 P81 Y82 Y138 Y172 R193 H196 H198 Y162 Y196 R217 H220 H222 Y138 Y172 R193 H196 H198 1.13.11.1 0003824,0005506,0008199,0009056,0009712,0016702,0018576,0046872,0051213 Ki=0.02uM remove_due_to_license_issue P95607 20040374 1 ATADTSPERLAAIAKDALGALNDVILKHGVTYPEYRVFKQWLIDVGEGGEWPLFLDVFIEHSVEEVLARSRKGTMGSIEGPYYIENSPELPSKCTLPMREEDEKITPLVFSGQVTDLDGNGLAGAKVELWHADNDGYYSQFAPHLPEWNLRGTIIADEEGRYEITTIQPAPYQIPTDGPTGQFIEAQNGHPWRPAHLHLIVSAPGKESVTTQLYFKGGEWIDSDVASATKPELILDPKTGDDGKNYVTYNFVLDPA 3i5n A 2.0 BS01 B2D A 1 I1084 A1108 Y1159 M1160 D1164 R1208 M1211 D1222 Y1230 I33 A57 Y98 M99 D103 R147 M150 D161 Y169 D1204 A1206 R1208 N1209 D1222 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0005524,0006468 ic50=17nM remove_due_to_license_issue IC50=17nM P08581 19819693 1 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNREVSQFLTEGIIMKDFSHPNVLSLLGICLPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 3i5x A 1.9 BS01 rna B 0 P188 T189 R190 G220 G221 D223 F224 T242 G244 R245 D248 K252 F277 T382 V383 K384 H407 G408 R415 T433 D528 S532 S535 S536 S539 F576 P101 T102 R103 G133 G134 D136 F137 T155 G157 R158 D161 K165 F190 T295 V296 K297 H320 G321 R328 T346 D441 S445 S448 S449 S452 F489 3.6.4.13 0003676,0005524 remove_due_to_license_issue P15424 19748356 1 ~ 10 SKLIHVPKEDNSKEVTLDSLLEEGVLDKEIHKAITRMEFPGLTPVQQKTIKPILSSEDHDVIARAKTGTGKTFAFLIPIFQHLINTKFDSQYMVKAVIVAPTRDLALQIEAEVKKIHDMNYGLKKYACVSLVGGTDFRAAMNKMNKLRPNIVIATPGRLIDVLEKYSNKFFRFVDYKVLDEADRLLEIGFRDDLETISGILNEKNSKSADNIKTLLFSATLDDKVQKLANNIMNKKECLFLDTVDKNEPEAHERIDQSVVISEKFANSIFAAVEHIKKQIKERDSNYKAIIFAPTVKFTSFLCSILKNEFKKDLPILEFHGKITQNKRTSLVKRFKKDESGILVCTDVGARGMDFPNVHEVLQIGVPSELANYIHRIGRTARSGKEGSSVLFICKDELPFVRELEDAKNIVIAKQEKYEPSEEIKSEVLEAVTEEPEDISDIVISLISSYRSCIKEYRFSERRILPEIASTYGVLLNDPQLKIPVSRRFLDKLGLSRSPIGKAMFEIRD 3i5z A 2.2 BS01 Z48 A 1 G32 G35 A50 K52 M106 E107 L154 D165 G27 G30 A45 K47 M101 E102 L149 D160 D147 K149 S151 N152 D165 T188 D142 K144 S146 N147 D160 T169 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Ki=2nM remove_due_to_license_issue Ki=4nM P28482 19827834 401 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVVATRWYRAPEIMLTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 3i60 A 2.5 BS01 E86 A 1 I29 G32 G35 A50 K52 I54 M106 T108 D109 L154 D165 I24 G27 G30 A45 K47 I49 M101 T103 D104 L149 D160 D147 K149 S151 N152 D165 T188 D142 K144 S146 N147 D160 T170 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Ki<2nM remove_due_to_license_issue Ki=<2nM P28482 19827834 401 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADATRWYRAPEIMLNYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 3i6c A 1.3 BS01 GIA A 1 H59 Q131 F134 S154 H157 H9 Q81 F84 S104 H107 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 Ki=12uM remove_due_to_license_issue Ki=12000nM, IC50=12000nM Q13526 20207139 301 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3i6c A 1.3 BS02 GIA A 2 R74 Q75 R80 F110 R24 Q25 R30 F60 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 Ki=12uM remove_due_to_license_issue Ki=12000nM, IC50=12000nM Q13526 20207139 303 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3i6m A 2.26 BS01 G3X A 1 W84 G117 G118 G119 Y121 E199 S200 F290 F330 F331 Y334 H440 W83 G116 G117 G118 Y120 E198 S199 F289 F329 F330 Y333 H439 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G117 G118 G150 S199 A200 A238 F289 F291 E326 H439 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 20025280 1 DHSELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 3i6o A 1.17 BS01 GR6 B 1 D25 G27 A28 D29 D30 G49 I50 V82 D25 G27 A28 D29 D30 G49 I50 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 19746963 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3i6o B 1.17 BS01 GR6 B 1 D125 G127 A128 D129 D130 G148 P181 V182 I184 D25 G27 A28 D29 D30 G48 P81 V82 I84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=45pM remove_due_to_license_issue P03367 19746963 301 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3i6z A 2.19 BS01 G6X A 1 Y70 W84 G117 G118 G119 Y121 E199 S200 W279 F290 F330 F331 Y334 H440 Y67 W81 G114 G115 G116 Y118 E196 S197 W276 F287 F327 F328 Y331 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 20025280 1 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 3i73 A 2.4 BS01 ADP A 1 K240 T241 V242 T243 L417 D418 A419 A422 F427 P428 A429 Q505 D506 A507 F508 K178 T179 V180 T181 L341 D342 A343 A346 F351 P352 A353 Q429 D430 A431 F432 K240 E263 R264 L438 K178 E201 R202 L362 3.1.-.-,7.1.2.2 0005524,0015986,0016887,0033178,0046034,0046961,1902600 Kd=3.23uM remove_due_to_license_issue O57728 19944110 589 EPVVGTGASLSVELGPRLLTSIYDGIQRPLEVIREKTGDFIARGVTAPALPRDKKWHFIPKAKVGDKVVGGDIIGEVPETSIIVHKIMVPPGIEGEIVEIAEEGDYTIEEVIAKVKTPSGEIKELKMYQRWPVRVKRPYKEKLPPEVPLITGQRVIDTFFPQAKGGTAAIPGPFGSGKTVTQHQLAKWSDAQVVIYIGCGERGNEMTDVLEEFPKLKDPKTGKPLMERTVLIANTSNMPVAAREASIYTGITIAEYFRDMGYDVALMADSTSRWAEAEGYPAYLASKLAEFYERAGRVVTLGSDYRVGSVSVIGAVSPPGGDFSEPVVQNTLRVVKVFWALDADLARRRHFPAINWLTSYSLYVDAVKDWWHKNIDPEWKAMRDKAMALLQKESELQEIVRIVGPDALPERERAILLVARMLREDYLQQDAFDEVDTYCPPEKQVTMMRVLLNFYDKTMEAINRGVPLEEIAKLPVREEIGRMKFERDVSKIRSLIDKTNEQFEELFKKYGA 3i7b A 1.988 BS01 BK1 A 1 V65 A78 K80 M112 L126 V130 Y131 L181 I194 D195 V20 A33 K35 M67 L81 V85 Y86 L136 I149 D150 D174 K176 E178 N179 D195 T214 D129 K131 E133 N134 D150 T169 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 ic50=0.066uM remove_due_to_license_issue IC50=128nM Q9BJF5 20436472 701 IFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMSAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3i7c A 1.98 BS01 BK2 A 1 L57 V65 A78 K80 M112 L126 Y131 L181 I194 L15 V23 A36 K38 M70 L84 Y89 L139 I152 D174 K176 E178 N179 D195 T214 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 ic50=0.018uM remove_due_to_license_issue IC50=15.0nM Q9BJF5 20436472 701 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3i7e A 1.7 BS01 DJR A 1 D25 G27 A28 D29 D30 G48 I50 I84 D25 G27 A28 D29 D30 G48 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=14pM remove_due_to_license_issue P03369 19746963 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3i7e B 1.7 BS01 DJR A 1 D25 G27 A28 D30 P81 V82 D25 G27 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 19746963 100 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3i7g A 1.95 BS06 732 A 1 G183 L185 H222 E223 L239 F241 I243 G80 L82 H119 E120 L136 F138 I140 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=430nM remove_due_to_license_issue IC50=430nM P45452 19692239 999 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTFMLPDDDVQGIQSLYGPGDED 3i7i A 2.208 BS06 518 A 1 G183 L185 H222 E223 L239 F241 P242 I243 Y244 T245 T247 F252 P255 G80 L82 H119 E120 L136 F138 P139 I140 Y141 T142 T144 F145 P148 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=620nM remove_due_to_license_issue IC50=620nM P45452 19692239 999 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTFMLPDDDVQGIQSLYGPGDED 3i81 A 2.08 BS01 EBI A 1 L975 V983 A1001 M1049 E1050 M1052 T1053 G1055 N1110 M1112 G1122 D1123 M1126 L21 V29 A47 M95 E96 M98 T99 G101 N155 M157 G167 D168 M171 D1105 R1109 N1110 D1123 E1132 D150 R154 N155 D168 E177 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=13nM remove_due_to_license_issue IC50=2nM P08069 19778024 201 DVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3i97 A 2.9 BS01 8DR A 1 Y25 T44 D48 S74 E76 T77 Y81 I143 Y24 T43 D47 S73 E75 T76 Y80 I142 ? remove_due_to_license_issue O14786 20151671 156 KCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 3i9g H 1.9 BS01 S1P L 1 T33 I56 Y98 G99 S100 W100C T33 I57 Y102 G103 S104 W107 remove_due_to_license_issue 19815502 401 EVQLVQSGAEVKKPGESLKISCQSFGYIFIDHTIHWMRQMPGQGLEWMGAISPRHDITKYNEMFRGQVTISADKSSSTAYLQWSSLKASDTAMYFCARGGFYGSTIWFDFWGQGTMVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKRVEPK 3i9g L 1.9 BS03 S1P L 1 D30 D32 E50 S91 D92 L94 D30 D32 E50 S91 D92 L94 Kd=1.1nM remove_due_to_license_issue 19815502 401 ETTVTQSPSFLSASVGDRVTITCITTTDIDDDMNWFQQEPGKAPKLLISEGNILRPGVPSRFSSSGYGTDFTLTISKLQPEDFATYYCLQSDNLPFTFGQGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGE 3ia6 A 2.31 BS01 UNT A 1 F282 G284 C285 Q286 S289 H323 L330 I341 H449 L469 Y473 F62 G64 C65 Q66 S69 H103 L110 I121 H229 L249 Y253 ? 0003677,0004879,0005634,0006355 ic50=0.003uM remove_due_to_license_issue IC50=3nM, EC50=13nM P37231 19783444 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 3iad A 2.65 BS01 15X A 1 S374 F506 S534 Q535 F538 F599 S126 F258 S286 Q287 F290 F333 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 20037581 901 GVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTNQVSEFISNTFLD 3iae A 2.3 BS01 D7K A 1 G393 A394 L395 T396 Y397 S420 M421 G447 D448 G449 S450 Y453 N475 S477 W478 G479 A480 T481 G392 A393 L394 T395 Y396 S419 M420 G446 D447 G448 S449 Y452 N474 S476 W477 G478 A479 T480 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iae A 2.3 BS03 D7K B 1 H26 G27 S28 E50 T73 Q113 H25 G26 S27 E49 T72 Q112 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iae B 2.3 BS01 D7K A 1 H26 G27 S28 E50 T73 G76 Q113 H25 G26 S27 E49 T72 G75 Q112 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iae B 2.3 BS02 D7K B 1 G393 A394 L395 T396 Y397 S420 M421 G447 D448 G449 S450 Y453 N475 S477 W478 G479 A480 T481 G392 A393 L394 T395 Y396 S419 M420 G446 D447 G448 S449 Y452 N474 S476 W477 G478 A479 T480 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iaf A 2.8 BS01 TPP A 1 A394 L395 T396 M421 G447 G449 S450 Y453 N475 S477 W478 G479 T481 A393 L394 T395 M420 G446 G448 S449 Y452 N474 S476 W477 G478 T480 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iaf A 2.8 BS03 TPP B 1 L25 H26 S28 E50 T73 G76 L24 H25 S27 E49 T72 G75 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iaf B 2.8 BS01 TPP A 1 H26 E50 T73 G76 G77 H25 E49 T72 G75 G76 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iaf B 2.8 BS02 TPP B 1 L395 T396 G419 S420 M421 G447 D448 G449 S450 N475 S477 W478 G479 T481 L394 T395 G418 S419 M420 G446 D447 G448 S449 N474 S476 W477 G478 T480 L25 G27 S28 H29 I30 E50 T73 L112 Q113 A114 G115 W163 L256 T284 G393 G419 M421 D448 N475 S477 W478 A480 T481 F484 L546 L24 G26 S27 H28 I29 E49 T72 L111 Q112 A113 G114 W162 L255 T283 G392 G418 M420 D447 N474 S476 W477 A479 T480 F483 L545 4.1.2.38 0000287,0003824,0003984,0005948,0009097,0009099,0016829,0019752,0030976,0046872,0050660 remove_due_to_license_issue Q9F4L3 20030408 571 AMITGGELVVRTLIKAGVEHLFGLHGSHIDTIFQACLDHDVPIIDTRHEAAAGHAAEGYARAGAKLGVALVTAGGGFTNAVTPIANAWLDRTPVLFLTGSGALRDDETNTLQAGIDQVAMAAPITKWAHRVMATEHIPRLVMQAIRAALSAPRGPVLLDLPWDILMNQIDEDSVIIPDLVLSAHGARPDPADLDQALALLRKAERPVIVLGSEASRTARKTALSAFVAATGVPVFADYEGLSMLSGLPDAMRGGLVQNLYSFAKADAAPDLVLMLGARFGLNTGHGSGQLIPHSAQVIQVDPDACELGRLQGIALGIVADVGGTIEALAQATAQDAAWPDRGDWCAKVTDLAQERYASIAAKSSSEHALHPFHASQVIAKHVDAGVTVVADGALTYLWLSEVMSRVKPGGFLCHGYLGSMGVGFGTALGAQVADLEAGRRTILVTGDGSVGYSIGEFDTLVRKQLPLIVIIMNNQSWGATLHFQQLAVGPNRVTGTRLENGSYHGVAAAFGADGYHVDSVESFSAALAQALAHNRPACINVAVALDPIPPEELI 3iag C 2.0 BS01 dna A 0 K84 Y86 S191 K192 S194 K196 R220 Q222 K32 Y34 S139 K140 S142 K144 R168 Q170 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 19866488 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMERDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKQSLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDESEGEEFTVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTPEP 3iag C 2.0 BS02 dna B 0 K90 R91 F92 K192 R218 S221 T223 K38 R39 F40 K140 R166 S169 T171 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 19866488 16 ~ 30 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMERDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKQSLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDESEGEEFTVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTPEP 3iaw A 1.61 BS01 2NC A 1 D25 G27 D29 G48 G49 I50 P81 L127 D129 G131 A132 D133 D134 I151 G152 I154 P185 D25 G27 D29 G48 G49 I50 P81 L127 D129 G131 A132 D133 D134 I151 G152 I154 P185 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=1.57uM remove_due_to_license_issue P03369 22158985 204 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNFCGGGGPQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3ibi A 1.93 BS02 BOW A 1 H94 L198 T199 H92 L195 T196 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.6nM remove_due_to_license_issue Ki=2.6nM P00918 19731956 300 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3ibl A 1.55 BS02 O59 A 1 H94 F131 L198 T199 T200 P202 H92 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=14.6nM remove_due_to_license_issue Ki=14.6nM P00918 19731956 300 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ibn A 2.2 BS02 O60 A 1 H94 H119 F131 L198 T199 P202 H92 H117 F128 L195 T196 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=24.5nM remove_due_to_license_issue Ki=24.5nM P00918 19731956 300 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ibu A 1.41 BS02 O48 A 1 H94 F131 L198 T199 P202 H92 F128 L195 T196 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.7nM remove_due_to_license_issue Ki=0.7nM P00918 19731956 300 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3idp B 2.7 BS01 L1E B 1 V471 A481 K483 E501 L505 L514 T529 W531 C532 F583 G593 D594 F595 V23 A33 K35 E53 L57 L66 T81 W83 C84 F135 G145 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=1nM, IC50=2nM P15056 19764794 1 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 3ie3 A 1.8 BS02 N11 A 1 F8 R13 Y108 F8 R13 Y108 Y7 R13 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Kd=0.21uM remove_due_to_license_issue IC50=800nM P09211 19808963 211 PPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYASLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 3iej A 2.18 BS01 599 A 1 G23 G68 F70 M71 N161 V162 N163 G165 F211 G25 G70 F72 M73 N163 V164 N165 G167 F213 Q19 S25 H164 N184 Q21 S27 H166 N186 3.4.22.27 0006508,0008234 ic50=0.22uM remove_due_to_license_issue IC50=220nM P25774 19773165 221 AALPDSVDWREKGCVTEVKYQGSCGASWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEILQ 3ieo A 2.0 BS02 AMJ A 1 Q92 V121 F131 Q89 V118 F127 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=331nM remove_due_to_license_issue P00918 20028100 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3ies A 2.0 BS01 M24 A 1 H245 F247 G315 G316 A317 P318 G339 Y340 G341 L342 T343 S347 A348 V362 D422 H238 F240 G308 G309 A310 P311 G332 Y333 G334 L335 T336 S340 A341 V355 D415 S198 R218 H245 T343 E344 S196 R211 H238 T336 E337 1.13.12.7 0004497,0005524,0005777,0008218,0016405,0046872,0047077,0051087 Kd~120pM remove_due_to_license_issue P08659 20194791 552 DAKNIKKGPAPFYPLEDGTAGEQLHKAMKRYALVPGTIAFTDAHIEVNITYAEYFEMSVRLAEAMKRYGLNTNHRIVVCSENSLQFFMPVLGALFIGVAVAPANDIYNERELLNSMNISQPTVVFVSKKGLQKILNVQKKLPIIQKIIIMDSKTDYQGFQSMYTFVTSHLPPGFNEYDFVPESFDRDKTIALIMNSLPKGVALPHRTACVRFSHARDPIFGNQIIPDTAILSVVPFHHGFGMFTTLGYLICGFRVVLMYRFEEELFLRSLQDYKIQSALLVPTLFSFFAKSTLIDKYDLSNLHEIASGGAPLSKEVGEAVAKRFHLPGIRQGYGLTETTSAILITPEGDDKPGAVGKVVPFFEAKVVDLDTGKTLGVNQRGELCVRGPMIMSGYVNNPEATNALIDKDGWLHSGDIAYWDEDEHFFIVDRL 3if7 A 1.6 BS05 SPU A 1 E11 M76 A88 F92 E123 M124 E127 F141 M144 M145 E9 M74 A84 F88 E119 M120 E123 F137 M140 M141 V35 V33 ? 0000922,0002027,0005509,0005513,0005515,0005737,0005813,0005819,0005829,0005856,0005876,0008179,0010856,0010880,0019901,0019904,0030017,0031432,0032465,0032991,0034704,0043209,0043539,0044325,0046872,0051592,0055117,0060315,0060316,0072542,0097720,0098901,1902494 Kd=61nM remove_due_to_license_issue P62157 20522785 153 QLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMT 3if7 A 1.6 BS06 SPU A 2 M109 M124 M105 M120 V35 V33 ? 0000922,0002027,0005509,0005513,0005515,0005737,0005813,0005819,0005829,0005856,0005876,0008179,0010856,0010880,0019901,0019904,0030017,0031432,0032465,0032991,0034704,0043209,0043539,0044325,0046872,0051592,0055117,0060315,0060316,0072542,0097720,0098901,1902494 Kd=61nM remove_due_to_license_issue P62157 20522785 154 QLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMT 3if7 A 1.6 BS07 SPU A 3 F12 L32 M51 E54 V55 M71 M72 F10 L30 M49 E52 V53 M69 M70 V35 V33 ? 0000922,0002027,0005509,0005513,0005515,0005737,0005813,0005819,0005829,0005856,0005876,0008179,0010856,0010880,0019901,0019904,0030017,0031432,0032465,0032991,0034704,0043209,0043539,0044325,0046872,0051592,0055117,0060315,0060316,0072542,0097720,0098901,1902494 Kd=61nM remove_due_to_license_issue P62157 20522785 155 QLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMT 3if7 A 1.6 BS08 SPU A 4 M72 M145 M70 M141 V35 V33 ? 0000922,0002027,0005509,0005513,0005515,0005737,0005813,0005819,0005829,0005856,0005876,0008179,0010856,0010880,0019901,0019904,0030017,0031432,0032465,0032991,0034704,0043209,0043539,0044325,0046872,0051592,0055117,0060315,0060316,0072542,0097720,0098901,1902494 Kd=61nM remove_due_to_license_issue P62157 20522785 156 QLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMT 3ig6 B 1.83 BS02 438 B 1 V41 C42 H57 L97B A98 H99 D189 S190 C191 Q192 G193 S195 V213 W215 G216 G218 V30 C31 H46 L92 A93 H94 D192 S193 C194 Q195 G196 S198 V216 W218 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=0.025uM remove_due_to_license_issue IC50=25nM P00749 19703768 400 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 3ig6 B 1.83 BS03 438 D 1 Y149 L150 Y148 L149 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 ic50=0.025uM remove_due_to_license_issue IC50=25nM P00749 19703768 401 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 3ig7 A 1.8 BS01 EFP A 1 E8 I10 A31 K33 F82 L83 H84 Q85 L134 D145 E8 I10 A31 K33 F74 L75 H76 Q77 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=9nM remove_due_to_license_issue P24941 19700321 999 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3igb A 2.238 BS01 454 A 1 L92 D94 F170 W177 I180 D290 L33 D35 F108 W115 I118 D222 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=38uM remove_due_to_license_issue IC50=38000nM, EC50=16000nM P56817 19757823 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLEDCGYN 3igg A 1.8 BS01 EFQ A 1 E8 I10 A31 F80 F82 L83 H84 Q85 L134 D145 E8 I10 A31 F72 F74 L75 H76 Q77 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=95nM remove_due_to_license_issue P24941 19700321 999 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3igm A 2.2 BS01 dna C 0 M75 F81 R88 R89 S90 R91 T92 H94 M14 F20 R27 R28 S29 R30 T31 H33 ? 0003700,0006355 remove_due_to_license_issue Q8IKH2 19913037 1 ~ 8 MSSGYPGVSWNKRMCAWLAFFYDGASRRSRTFHPKHFNMDKEKARLAAVEFMKTVE 3igm A 2.2 BS02 dna D 0 S63 G68 S70 N72 K73 R74 F81 R88 S2 G7 S9 N11 K12 R13 F20 R27 ? 0003700,0006355 remove_due_to_license_issue Q8IKH2 19913037 1 ~ 7 MSSGYPGVSWNKRMCAWLAFFYDGASRRSRTFHPKHFNMDKEKARLAAVEFMKTVE 3igm B 2.2 BS01 dna W 0 M75 F81 R88 R89 S90 R91 T92 H94 M14 F20 R27 R28 S29 R30 T31 H33 ? 0003700,0006355 remove_due_to_license_issue Q8IKH2 19913037 1 ~ 8 MSSGYPGVSWNKRMCAWLAFFYDGASRRSRTFHPKHFNMDKEKARLAAVEFMKTVENNGRKK 3igm B 2.2 BS02 dna X 0 M62 S63 P67 G68 S70 N72 K73 R74 F81 R88 M1 S2 P6 G7 S9 N11 K12 R13 F20 R27 ? 0003700,0006355 remove_due_to_license_issue Q8IKH2 19913037 1 ~ 8 MSSGYPGVSWNKRMCAWLAFFYDGASRRSRTFHPKHFNMDKEKARLAAVEFMKTVENNGRKK 3igp A 1.65 BS02 DT7 A 1 H94 H119 V121 L198 T199 T200 H93 H118 V120 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=32.8nM remove_due_to_license_issue P00918 20170095 263 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3igp A 1.65 BS03 DT7 A 2 H4 H10 H15 D19 H3 H9 H14 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=32.8nM remove_due_to_license_issue P00918 20170095 264 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3igv A 2.6 BS01 B80 A 1 P197 R200 N291 D318 C366 S368 L384 M414 Y415 Y448 S556 P192 R195 N286 D313 C361 S363 L379 M409 Y410 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 19796938 579 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 3ihz A 1.67 BS01 FK5 A 1 Y43 D55 F64 V73 I74 W77 Y100 F117 Y40 D52 F61 V70 I71 W74 Y97 F114 Y43 F54 D55 I74 Y100 F117 Y40 F51 D52 I71 Y97 F114 5.2.1.8 0003755 ic50=160nM remove_due_to_license_issue A5K8X6 20572013 501 ETLEQVHLTEDGGVVKTILRKGEGGEENAPKKGNEVTVHYVGKLESSGKVFDSSRERNVPFKFHLGQGEVIKGWDICVASMTKNEKCSVRLDSKYGYGEEGCGESIPGNSVLIFEIELISFRE 3ihz B 1.67 BS01 FK5 A 1 D55 F64 W77 C105 G106 S108 D50 F59 W72 C100 G101 S103 Y43 F54 D55 I74 Y100 F117 Y38 F49 D50 I69 Y95 F112 5.2.1.8 0003755 remove_due_to_license_issue A5K8X6 20572013 501 LEQVHLTEDGGVVKTILRKGEGGEENAPKKGNEVTVHYVGKLESSGKVFDSSRERNVPFKFHLGQGEVIKGWDICVASMTKNEKCSVRLDSKYGYGEEGCGESIPGNSVLIFEIELISFRE 3ii5 A 2.79 BS01 831 A 1 I462 A480 K482 E500 L504 L513 T528 G592 D593 F594 I16 A34 K36 E54 L58 L67 T82 G146 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S158 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=24nM P15056 19864136 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVQLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 3iit A 1.8 BS03 D14 A 1 T98 F174 D189 A190 C191 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 T84 F162 D179 A180 C181 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=9.5nM remove_due_to_license_issue IC50=9.5nM P00742 19900814 700 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 3ijg C 1.7 BS01 AVR C 1 Q35 Y36 W108 F113 Q35 Y36 W108 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=54uM remove_due_to_license_issue P14174 20534506 200 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3ijh A 2.1 BS01 KO2 B 1 S91 N92 R95 S96 N97 R100 remove_due_to_license_issue 19767317 214 IVMTQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTISSVQAEDLAVYYCKQSNNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 3ijh B 2.1 BS01 KO2 B 1 Y33 R52 K53 I96 P98 E100E Y33 R52 K56 I102 P104 E111 Kd=100uM remove_due_to_license_issue 19767317 214 EVMLVESGGGLVQPGNSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKAKGYTTEYSASVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDISPSYGVYYEGFAYWGQGTLVTVSAATTTAPSVYPLVPGGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKTELIKRIEPR 3ijy A 2.85 BS01 KDO E 1 S91 N92 R95 S96 N97 R100 remove_due_to_license_issue 19767317 2 IVMTQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTISSVQAEDLAVYYCKQSNNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNR 3ijy B 2.85 BS01 KDO E 1 Y33 R52 I96 E100E Y33 R52 I102 E111 remove_due_to_license_issue 19767317 2 EVMLVESGGGLVQPGNSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKAKGYTTEYSASVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDISPSYGVYYEGFAYWGQGTLVTVSAATTTAPSVYPLVPGGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKTELIKRIEPR 3ijz A 2.21 BS01 15C A 1 E60 I81 W82 W85 L195 E60 I81 W82 W85 L195 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue Ki=6000nM P00469 21696158 468 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIKA 3ik1 A 2.25 BS01 20C A 1 E60 I81 W82 W85 L195 E60 I81 W82 W85 L195 E60 W82 Y146 C198 R218 D221 E60 W82 Y146 C198 R218 D221 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue Ki=14000nM P00469 21696158 490 MLEQPYLDLAKKVLDEGHFKPDRTHTGTYSIFGHQMRFDLSKGFPLLTTKKVPFGLIKSELLWFLHGDTNIRFLLQHRNHIWDEWAFEKWVKSDEYHGPDMTDFGHRSQKDPEFAAVYHEEMAKFDDRVLHDDAFAAKYGDLGLVYGSQWRAWHTSKGDTIDQLGDVIEQIKTHPYSRRLIVSAWNPEDVPTMALPPCHTLYQFYVNDGKLSLQLYQRSADIFLGVPFNIASYALLTHLVAHECGLEVGEFIHTFGDAHLYVNHLDQIKEQLSRTPRPAPTLQLNPDKHDIFDFDMKDIKLLNYDPYPAIK 3ik3 A 1.9 BS01 0LI A 1 L248 Y253 A269 K271 E286 M290 I293 V299 I313 I315 F317 M318 I360 H361 L370 V379 A380 D381 F382 L21 Y26 A42 K44 E59 M63 I66 V72 I86 I88 F90 M91 I133 H134 L143 V152 A153 D154 F155 D363 A365 R367 N368 D381 P402 D136 A138 R140 N141 D154 P169 2.7.10.2 0004672,0004713,0005524,0006468 ic50=2nM remove_due_to_license_issue P00520 19878872 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELGKR 3ika A 2.9 BS01 0UN A 1 L718 G719 V726 A743 M790 L792 M793 G796 C797 D800 L844 L23 G24 V31 A48 M95 L97 M98 G101 C102 D105 L149 D837 A839 R841 N842 D855 G874 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=<1nM, Kd=1.2nM, EC50=68nM P00533 20033049 1797 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHEEDMDDVVDADEYLIPQ 3ikc A 2.6 BS01 KDO E 1 Y32 S91 N92 R95 Y37 S96 N97 R100 remove_due_to_license_issue 19767317 2 IVMTQSPSSLAVSAGEKVTMSCKSSQSLLNSRTRKNYLAWYQQKPGQSPKLLIYWASTRESGVPDRFTGSGSGTDFTLTISSVQAEDLAVYYCKQSNNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 3ikc B 2.6 BS01 KME E 1 K53 Y100C K56 Y109 remove_due_to_license_issue 19767317 1 EVMLVESGGGLVQPGNSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKAKGYTTEYSASVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDISPSYGVYYEGFAYWGQGTLVTVSAATTTAPSVYPLVPGGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKTELIKRIEPR 3ikc B 2.6 BS02 KDO E 1 Y33 R52 I96 E100E Y33 R52 I102 E111 remove_due_to_license_issue 19767317 2 EVMLVESGGGLVQPGNSLRLSCATSGFTFTDYYMSWVRQPPGKALEWLGFIRNKAKGYTTEYSASVKGRFTISRDNSQSILYLQMNTLRAEDSATYYCARDISPSYGVYYEGFAYWGQGTLVTVSAATTTAPSVYPLVPGGSSVTLGCLVKGYFPEPVTVKWNYGALSSGVRTVSSVLQSGFYSLSSLVTVPSSTWPSQTVICNVAHPASKTELIKRIEPR 3ikd A 2.0 BS01 J9Z A 1 H59 K63 R68 R69 C113 L122 F134 S154 H157 H9 K13 R18 R19 C63 L72 F84 S104 H107 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 remove_due_to_license_issue IC50=180nM, Ki=179nM Q13526 19729306 501 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3ikg A 1.86 BS01 J8Z A 1 H59 K63 R68 R69 C113 S115 L122 M130 F134 S154 H157 H9 K13 R18 R19 C63 S65 L72 M80 F84 S104 H107 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 remove_due_to_license_issue Q13526 19729306 1 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3il5 A 2.6 BS01 B82 A 1 R42 G220 I223 F224 H250 A252 N253 I256 N280 F312 G313 R37 G215 I218 F219 H245 A247 N248 I251 N275 F307 G308 2.3.1.180 0004315,0005737,0006633,0016746,0033818 remove_due_to_license_issue IC50=1600nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTSDEWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWAALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL 3il5 B 2.6 BS01 B82 B 1 R42 G220 I223 F224 A252 N253 I256 N280 F312 R36 G214 I217 F218 A246 N247 I250 N274 F306 2.3.1.180 0004315,0005737,0006633,0016746,0033818 remove_due_to_license_issue IC50=1600nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTDEWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWAALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL 3il6 A 2.5 BS01 B83 A 1 R42 C117 S157 L161 M218 G220 R221 I223 F224 H250 A252 I256 N280 F312 R37 C112 S152 L156 M213 G215 R216 I218 F219 H245 A247 I251 N275 F307 2.3.1.180 0004315,0005737,0006633,0016746,0033818 ic50=0.27uM remove_due_to_license_issue IC50=270nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTSAAWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWTALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL 3ilq C 2.05 BS01 1O2 C 1 F70 Y73 S76 F77 R79 D80 L84 I98 F120 W142 T156 F64 Y67 S70 F71 R73 D74 L78 I92 F111 W133 T147 ? Kd=6.2uM remove_due_to_license_issue P11609 20080535 286 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 3imc A 1.6 BS01 BZ3 A 1 H44 G46 H47 K160 P185 V187 H41 G43 H44 K157 P182 V184 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D85 D86 Q89 K157 S193 S194 R195 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1100uM remove_due_to_license_issue Kd=1100000nM P9WIL5 19780086 702 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3ime A 2.39 BS01 BZ2 A 1 P38 T39 M40 H47 Q164 P35 T36 M37 H44 Q161 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D85 D86 Q89 K157 S193 S194 R195 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1000uM remove_due_to_license_issue Kd=1000000nM P9WIL5 19780086 301 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGNGSGRLLVAARLGTTRLLDNIAIEIGT 3img A 1.8 BS02 BZ3 A 1 H44 G46 H47 K160 P185 T186 V187 H42 G44 H45 K158 P183 T184 V185 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 remove_due_to_license_issue Kd=1100000nM P9WIL5 19780086 401 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3imy A 2.55 BS01 B72 A 1 A279 R282 M310 M313 L330 N331 L346 H435 F455 A69 R72 M100 M103 L120 N121 L136 H225 F245 ? 0003677,0004879,0006355 remove_due_to_license_issue Kd=0.1nM, Ki=0.32nM, EC50=2.82nM P10828 18237438 462 MEELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGQKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 3in3 A 2.0 BS01 472 A 1 G73 G75 D94 S97 F170 I172 I180 D290 G292 G14 G16 D35 S38 F111 I113 I121 D225 G227 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D225 T228 3.4.23.46 0004190,0006508,0016020 ic50=0.06uM remove_due_to_license_issue IC50=60nM P56817 20045648 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGY 3in4 A 2.3 BS01 BX2 A 1 G73 Q74 D94 G96 S97 W138 F170 I172 W177 I180 D290 G292 G14 Q15 D35 G37 S38 W79 F111 I113 W118 I121 D225 G227 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D225 T228 3.4.23.46 0004190,0006508,0016020 ic50=0.04uM remove_due_to_license_issue P56817 20045648 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGY 3ind A 2.246 BS01 593 A 1 L92 D94 S97 Y133 F170 I180 D290 G292 L33 D35 S38 Y74 F111 I121 D225 G227 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D225 T228 3.4.23.46 0004190,0006508,0016020 ic50=1.53uM remove_due_to_license_issue IC50=1530nM, EC50=930nM P56817 19968289 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGYNI 3ine A 1.996 BS01 X17 A 1 L92 D94 S97 Y133 W138 F170 W177 D290 L33 D35 S38 Y74 W77 F109 W116 D222 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.17uM remove_due_to_license_issue EC50=130nM, IC50=170nM P56817 19968289 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTMEDCGYN 3inf A 1.852 BS01 X45 A 1 G73 G75 D94 S97 Y133 W138 F170 I172 W177 I180 D290 G292 G14 G16 D35 S38 Y74 W76 F108 I110 W115 I118 D223 G225 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=0.04uM remove_due_to_license_issue IC50=40nM, EC50=120nM P56817 19968289 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACDEFRTAAVEGPFVTEDCGYNI 3inh A 1.8 BS01 569 A 1 G73 Q74 G75 D94 S97 V131 W138 F170 I172 W177 I180 R190 D290 G292 G14 Q15 G16 D35 S38 V72 W76 F108 I110 W115 I118 R128 D221 G223 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.02uM remove_due_to_license_issue IC50=20nM, EC50=270nM P56817 19968289 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGYNI 3iny A 2.75 BS01 7DG A 1 A116 A117 G118 F200 E201 V217 T242 N243 A115 A116 G117 F199 E200 V216 T241 N242 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S32 H63 H85 Y87 E88 A115 M218 S219 N242 V244 H256 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue P00491 19932753 293 ENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS 3io7 A 2.6 BS01 1P5 A 1 L855 K857 G858 V863 M929 L932 R980 N981 L983 D994 L14 K16 G17 V20 M83 L86 R134 N135 L137 D148 M865 D976 A978 R980 N981 D994 S1016 M22 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=7nM, IC50=>20000nM O60674 19857967 1 TQFEERHLKFLQQLGKGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 3iob A 1.8 BS01 A4D A 1 H44 G46 H47 F157 G158 K160 D161 T186 V187 M195 H42 G44 H45 F155 G156 K158 D159 T184 V185 M193 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=380uM remove_due_to_license_issue Kd=3.80e+5nM P9WIL5 19827080 301 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 3ioc A 2.5 BS01 A5D A 1 P38 H44 G46 H47 L50 V142 F157 G158 K160 D161 Q164 T186 V187 M195 P35 H41 G43 H44 L47 V127 F142 G143 K145 D146 Q149 T171 V172 M180 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D73 D74 Q77 K145 S181 S182 R183 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=210uM remove_due_to_license_issue Kd=210000nM P9WIL5 19827080 301 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIG 3iod A 1.75 BS01 A6D A 1 P38 T39 M40 H44 G46 H47 F67 Q72 F157 G158 D161 Q164 T186 V187 M195 P35 T36 M37 H41 G43 H44 F64 Q69 F149 G150 D153 Q156 T178 V179 M187 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D80 D81 Q84 K152 S188 S189 R190 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=80uM remove_due_to_license_issue Kd=80000nM P9WIL5 19827080 302 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGNGSGRLLVAARLGTTRLLDNIAIEIG 3ioe A 1.95 BS01 A7D A 1 T39 H44 G46 H47 L50 Q72 V142 F157 G158 K160 D161 Q164 T186 V187 M195 T36 H41 G43 H44 L47 Q69 V139 F154 G155 K157 D158 Q161 T183 V184 M192 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D85 D86 Q89 K157 S193 S194 R195 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=540uM remove_due_to_license_issue P9WIL5 19827080 901 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 3iof A 1.44 BS02 IFS A 1 V67 W87 T119 D120 I153 F156 T157 L161 N233 H263 V21 W41 T71 D72 I104 F107 T108 L112 N174 H204 N116 H118 D120 H196 C221 K224 N233 H263 N68 H70 D72 H147 C166 K169 N174 H204 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=6uM remove_due_to_license_issue Ki=2000nM P26918 20527888 308 AGMSLTQVSGPVYVVEDNYYVQENSMVYFGAKGVTVVGATWTPDTARELHKLIKRVSRKPVLEVINTNYHTDRAGGNAYWKSIGAKVVSTRQTRDLMKSDWAEIVAFTRKGLPEYPDLPLVLPNVVHDGDFTLQEGKVRAFYAGPAHTPDGIFVYFPDEQVLYGGCILKEKLGNLSFADVKAYPQTLERLKAMKLPIKTVIGGHDSPLHGPELIDHYEALIKAAPQS 3iog A 1.41 BS02 SDF A 1 V67 W87 H196 K224 N233 H263 V21 W41 H147 K169 N174 H204 N116 H118 D120 H196 C221 K224 N233 H263 N68 H70 D72 H147 C166 K169 N174 H204 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=3uM remove_due_to_license_issue Ki=5000nM P26918 20527888 311 AGMSLTQVSGPVYVVEDNYYVQENSMVYFGAKGVTVVGATWTPDTARELHKLIKRVSRKPVLEVINTNYHTDRAGGNAYWKSIGAKVVSTRQTRDLMKSDWAEIVAFTRKGLPEYPDLPLVLPNVVHDGDFTLQEGKVRAFYAGPAHTPDGIFVYFPDEQVLYGGCILKEKLGNLSFADVKAYPQTLERLKAMKLPIKTVIGGHDSPLHGPELIDHYEALIKAAPQS 3ioi A 1.45 BS02 1GW A 1 F121 A122 I123 Y126 R188 D211 V212 D213 G267 A268 H301 D302 E303 F57 A58 I59 Y62 R116 D139 V140 D141 G195 A196 H229 D230 E231 H233 G266 W300 E303 A343 H161 G194 W228 E231 A271 2.4.1.37,2.4.1.40 0005975,0016020,0016758 Ki=0.53uM remove_due_to_license_issue P16442 20364127 355 SLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPK 3iok A 2.1 BS01 1P6 A 1 L855 G856 K857 V863 A880 M929 L932 R980 N981 L983 G993 D994 L14 G15 K16 V20 A37 M86 L89 R137 N138 L140 G150 D151 M865 D976 A978 R980 N981 D994 S1016 M22 D133 A135 R137 N138 D151 S173 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.0002uM remove_due_to_license_issue O60674 19857967 1201 TQFEERHLKFLQQLGKGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 3ion A 2.4 BS01 8H1 A 1 G89 E90 G91 S94 A109 K111 L159 S160 A162 G165 E166 N210 L212 T222 D223 G15 E16 G17 S20 A35 K37 L85 S86 A88 G91 E92 N136 L138 T148 D149 D205 K207 E209 N210 D223 T245 D131 K133 E135 N136 D149 T160 2.7.11.1 0004672,0004674,0005524,0006468 ic50=8nM remove_due_to_license_issue IC50=8nM O15530 20074837 1 RKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3iop A 2.2 BS01 8I1 A 1 G89 E90 G91 S94 V96 A109 K111 L159 S160 Y161 A162 G165 E209 L212 T222 D223 G15 E16 G17 S20 V22 A35 K37 L85 S86 Y87 A88 G91 E135 L138 T148 D149 D205 K207 E209 N210 D223 T245 D131 K133 E135 N136 D149 T162 2.7.11.1 0004672,0004674,0005524,0006468 ic50=17nM remove_due_to_license_issue IC50=17nM O15530 20074837 1 RKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3ip5 A 1.35 BS01 ALA A 1 F77 N78 S79 A100 A101 T102 Y150 D226 F77 N78 S79 A100 A101 T102 Y150 D226 ? 0006865,0046872 Kd=0.6uM remove_due_to_license_issue Q7CX36 20630861 500 MDVVIAVGAPLTGPNAAFGAQIQKGAEQAAKDINAAGGINGEQIKIVLGDDVSDPKQGISVANKFVADGVKFVVGHFNSGVSIPASEVYAENGILEITPAATNPVFTERGLWNTFRTCGRDDQQGGIAGKYLADHFKDAKVAIIHDKTPYGQGLADETKKAANAAGVTEVMYEGVNVGDKDFSALISKMKEAGVSIIYWGGLHTEAGLIIRQAADQGLKAKLVSGDGIVSNELASIAGDAVEGTLNTFGPDPTLRPENKELVEKFKAAGFNPEAYTLYSYAAMQAIAGAAKAAGSVEPEKVAEALKKGSFPTALGEISFDEKGDPKLPGYVMYEWKKGPDGKFTYIQQ 3ip6 A 1.4 BS01 PRO A 1 F77 N78 S79 A100 A101 T102 Y150 D226 Y275 F77 N78 S79 A100 A101 T102 Y150 D226 Y275 ? 0006865,0046872 Kd=0.25uM remove_due_to_license_issue Q7CX36 20630861 500 MDVVIAVGAPLTGPNAAFGAQIQKGAEQAAKDINAAGGINGEQIKIVLGDDVSDPKQGISVANKFVADGVKFVVGHFNSGVSIPASEVYAENGILEITPAATNPVFTERGLWNTFRTCGRDDQQGGIAGKYLADHFKDAKVAIIHDKTPYGQGLADETKKAANAAGVTEVMYEGVNVGDKDFSALISKMKEAGVSIIYWGGLHTEAGLIIRQAADQGLKAKLVSGDGIVSNELASIAGDAVEGTLNTFGPDPTLRPENKELVEKFKAAGFNPEAYTLYSYAAMQAIAGAAKAAGSVEPEKVAEALKKGSFPTALGEISFDEKGDPKLPGYVMYEWKKGPDGKFTYIQQ 3ip8 A 1.498 BS01 B85 A 1 P14 P15 G74 T75 S76 Y126 V156 C188 G189 G190 P8 P9 G68 T69 S70 Y120 V150 C182 G183 G184 4.1.1.76 0016831,0047436 Ki=5.2mM remove_due_to_license_issue Q05115 19739187 249 PTIGMIVPPAAGLVPADGARLYPDLPFIASGLGLGSVTPEGYDAVIESVVDHARRLQKQGAAVVSLMGTSLSFYRGAAFNAALTVAMREATGLPCTTMSTAVLNGLRALGVRRVALATAYIDDVNERLAAFLAEESLVPTGCRSLGITGVEAMARVDTATLVDLCVRAFEAAPDSDGILLSCGGLLTLDAIPEVERRLGVPVVSSSPAGFWDAVRLAGGGAKARPGYGRLFD 3ip9 A 1.8 BS01 ABU A 1 N78 S79 A100 A101 T102 Y150 D226 Y275 N78 S79 A100 A101 T102 Y150 D226 Y275 ? 0006865,0046872 Kd=2.4uM remove_due_to_license_issue Q7CX36 20630861 357 MDVVIAVGAPLTGPNAAFGAQIQKGAEQAAKDINAAGGINGEQIKIVLGDDVSDPKQGISVANKFVADGVKFVVGHFNSGVSIPASEVYAENGILEITPAATNPVFTERGLWNTFRTCGRDDQQGGIAGKYLADHFKDAKVAIIHDKTPYGQGLADETKKAANAAGVTEVMYEGVNVGDKDFSALISKMKEAGVSIIYWGGLHTEAGLIIRQAADQGLKAKLVSGDGIVSNELASIAGDAVEGTLNTFGPDPTLRPENKELVEKFKAAGFNPEAYTLYSYAAMQAIAGAAKAAGSVEPEKVAEALKKGSFPTALGEISFDEKGDPKLPGYVMYEWKKGPDGKFTYIQQ 3ipa A 1.55 BS01 ALA A 1 F77 N78 S79 A100 A101 T102 Y150 D226 F77 N78 S79 A100 A101 T102 Y150 D226 ? 0006865,0046872 remove_due_to_license_issue Q7CX36 20630861 500 MDVVIAVGAPLTGPNAAFGAQIQKGAEQAAKDINAAGGINGEQIKIVLGDDVSDPKQGISVANKFVADGVKFVVGHFNSGVSIPASEVYAENGILEITPAATNPVFTERGLWNTFRTCGRDDQQGGIAGKYLADHFKDAKVAIIHDKTPYGQGLADETKKAANAAGVTEVMYEGVNVGDKDFSALISKMKEAGVSIIYWGGLHTEAGLIIRQAADQGLKAKLVSGDGIVSNELASIAGDAVEGTLNTFGPDPTLRPENKELVEKFKAAGFNPEAYTLYSYAAMQAIAGAAKAAGSVEPEKVAEALKKGSFPTALGEISFDEKGDPKLPGYVMYEWKKGPDGKFTYIQQ 3ipb A 1.9 BS01 JZD A 1 L17 A108 S117 T119 L8 A99 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.2uM remove_due_to_license_issue P02766 21059958 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3ipb A 1.9 BS02 JZD B 1 K15 S117 K6 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.2uM remove_due_to_license_issue P02766 21059958 129 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3ipb B 1.9 BS01 JZD A 1 K15 L17 L110 S117 K6 L8 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.2uM remove_due_to_license_issue P02766 21059958 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3ipb B 1.9 BS02 JZD B 1 K15 A108 S117 T118 T119 V121 K6 A99 S108 T109 T110 V112 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.2uM remove_due_to_license_issue P02766 21059958 129 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3ipe A 1.4 BS01 JZE B 1 L17 S117 L8 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 21059958 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3ipe B 1.4 BS01 JZE B 1 L17 A108 S117 L8 A99 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.15uM remove_due_to_license_issue P02766 21059958 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3iph A 2.1 BS01 G11 A 1 A51 K53 E71 I84 T106 H107 M109 A111 L167 D168 F169 A48 K50 E68 I81 T103 H104 M106 A108 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T180 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=0.0000251mM remove_due_to_license_issue IC50=316.23nM, Ki=25.12nM Q16539 19772287 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3ipq A 2.0 BS02 965 A 1 F257 L260 S264 I295 M298 L299 T302 R305 F315 L316 F326 F335 I336 I339 F340 W443 F32 L35 S39 I70 M73 L74 T77 R80 F90 L91 F101 F110 I111 I114 F115 W218 ? 0003677,0004879,0006629 Ki=27nM remove_due_to_license_issue EC50=200nM, IC50=235nM Q13133 20382159 801 QLSPEQLGMIEKLVAAQQTPWPEARQQRFAHFTELAIVSVQEIVDFAKQLPGFLQLSREDQIALLKTSAIEVMLLETSRRYNPGSESITFLKDFSYNREDFAKAGLQVEFINPIFEFSRAMNELQLNDAEFALLIAISIFSADRPNVQDQLQVERLQHTYVEALHAYVSIHHPHDRLMFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 3ips A 2.26 BS02 O90 A 1 F257 L260 S264 M298 E301 T302 R305 F315 F335 W443 F35 L38 S42 M76 E79 T80 R83 F93 F113 W221 ? 0003677,0004879,0006629 Ki=64nM remove_due_to_license_issue EC50=35nM, IC50=32nM Q13133 20382159 1 QLSPEQLGMIEKLVAAQQVTPWPSREARQQRFAHFTELAIVSVQEIVDFAKQLPGFLQLSREDQIALLKTSAIEVMLLETSRRYNPGSESITFLKDFSYNREDFAKAGLQVEFINPIFEFSRAMNELQLNDAEFALLIAISIFSADRPNVQDQLQVERLQHTYVEALHAYVSIHHPHDRLMFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVH 3ipu A 2.4 BS02 O40 A 1 R232 F257 L260 A261 R305 F315 H421 R29 F50 L53 A54 R98 F108 H214 ? 0003677,0004879,0006629 Ki=48nM remove_due_to_license_issue Q13133 20382159 801 PQLSPEQLGMIEKLVAAQQQCNRRSFSDRLRVTPWPPHSREARQQRFAHFTELAIVSVQEIVDFAKQLPGFLQLSREDQIALLKTSAIEVMLLETSRRYNPGSESITFLKDFSYNREDFAKAGLQVEFINPIFEFSRAMNELQLNDAEFALLIAISIFSADRPNVQDQLQVERLQHTYVEALHAYVSIHHPHDRLMFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 3ipx A 2.0 BS02 B86 A 1 I30 E53 L82 Y86 F96 Q97 D133 F137 E197 I11 E34 L51 Y55 F65 Q66 D102 F106 E166 E53 R128 E34 R97 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 ic50=120nM remove_due_to_license_issue IC50=>4000nM P27707 19836232 262 RIKKISIEGNIAAGKSTFVNILKQLCEDWEVVPEPVARWCNVQSTNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESECMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 3irw P 2.7 BS01 rna R 0 Y13 N15 N16 E19 K20 S48 L49 K50 M51 R52 G53 Q54 F56 Q85 Y86 K88 D90 S91 D92 Y7 N9 N10 E13 K14 S42 L43 K44 M45 R46 G47 Q48 F50 Q79 Y80 K82 D84 S85 D86 ? 0003676,0003723 remove_due_to_license_issue P09012 19898477 8 RPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAK 3irx A 2.8 BS01 UDR A 1 P95 L100 V106 V108 Y181 Y188 G190 F227 W229 L234 P96 L101 V107 V109 Y182 Y189 G191 F228 W230 L235 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 19775161 556 VPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 3is9 A 2.55 BS01 AC7 A 1 L100 V106 Y181 Y188 K223 F227 L228 W229 L234 H235 Y318 L100 V106 Y181 Y188 K223 F227 L228 W229 L234 H235 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 19775161 556 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 3isj A 2.2 BS01 A8D A 1 H44 G46 H47 K160 V187 M195 H42 G44 H45 K158 V185 M193 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=210uM remove_due_to_license_issue P9WIL5 19780086 308 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 3iss A 2.5 BS01 EPU A 1 K22 N23 P121 V122 D123 L124 K160 S162 V163 G164 D305 K22 N23 P121 V122 D123 L124 K160 S162 V163 G164 D305 K22 N23 D49 A92 C115 R120 H299 D305 E325 L370 R371 R397 K22 N23 D49 A92 C115 R120 H299 D305 E325 L370 R371 R397 2.5.1.7 0003824,0005737,0005829,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P0A749 19899805 601 MDKFRVQGPTKLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDVDTSMKLLSQLGAKVERDGSVHIDARDVNVFCAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCTIGARPVDLHISGLEQLGATIKLEEGYVKASVDGRLKGAHIVMDKVSVGATVTIMCAATLAEGTTIIENAAREPEIVDTANFLITLGAKISGQGTDRIVIEGVERLGGGVYRVLPDRIETGTFLVAAAISRGKIICRNAQPDTLDAVLAKLRDAGADIEVGEDWISLDMHGKRPKAVNVRTAPHPAFPTDMQAQFTLLNLVAEGTGFITETVFENRFMHVPELSRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKG 3itz A 2.25 BS01 P66 A 1 Y35 A51 K53 E71 T106 M109 G110 A111 D168 F169 L171 Y39 A55 K57 E75 T110 M113 G114 A115 D172 F173 L175 D150 K152 N155 D168 T185 D154 K156 N159 D172 T189 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=1.4nM remove_due_to_license_issue IC50=1.4nM, Ki=1.000000nM Q16539 20138761 401 HMLEMSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3iu7 A 1.4 BS03 FCD A 1 Y97 H114 D131 D142 H205 H212 W255 E269 Y96 H113 D130 D141 H204 H211 W254 E268 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=16uM remove_due_to_license_issue P9WK19 20038112 288 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3iu7 A 1.4 BS04 FCD A 2 N144 R164 M168 F268 E269 H270 N143 R163 M167 F267 E268 H269 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=16uM remove_due_to_license_issue P9WK19 20038112 289 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3iu8 A 1.85 BS01 T03 A 1 Y97 C105 H114 D131 D142 H205 E238 W255 E269 Y96 C104 H113 D130 D141 H204 E237 W254 E268 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=0.58uM remove_due_to_license_issue P9WK19 20038112 289 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3iu9 A 1.75 BS01 T07 A 1 Y27 S93 T94 Y97 C105 H114 D131 T133 D142 H205 F211 H212 E238 E269 Y26 S92 T93 Y96 C104 H113 D130 T132 D141 H204 F210 H211 E237 E268 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=0.24uM remove_due_to_license_issue P9WK19 20038112 288 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3iub A 1.5 BS01 FG2 A 1 T39 H44 G46 H47 Y82 D161 Q164 V184 P185 V187 T36 H41 G43 H44 Y79 D158 Q161 V181 P182 V184 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D85 D86 Q89 K157 S193 S194 R195 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=29uM remove_due_to_license_issue Kd=29000nM P9WIL5 19780086 302 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 3iub A 1.5 BS02 FG2 A 2 M71 L114 P133 T134 G138 M68 L111 P130 T131 G135 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D85 D86 Q89 K157 S193 S194 R195 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=29uM remove_due_to_license_issue Kd=29000nM P9WIL5 19780086 303 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 3iuc A 2.4 BS01 ADP A 1 T37 T38 Y39 G226 G227 G255 E293 K296 R297 S300 G364 S365 R367 T10 T11 Y12 G199 G200 G228 E266 K269 R270 S273 G337 S338 R340 D34 S40 F68 T69 K96 E201 D224 D7 S13 F41 T42 K69 E174 D197 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11021 20072699 1 GTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQLTSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDIGGGQTKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLS 3iue A 1.73 BS01 FG3 A 1 T39 M40 H44 G46 H47 Y82 K160 D161 Q164 V187 M195 S196 S197 T37 M38 H42 G44 H45 Y80 K158 D159 Q162 V185 M193 S194 S195 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1.5uM remove_due_to_license_issue Kd=1500nM P9WIL5 19780086 302 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3iue A 1.73 BS02 FG3 A 2 L114 P133 T134 A137 G138 L112 P131 T132 A135 G136 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1.5uM remove_due_to_license_issue Kd=1500nM P9WIL5 19780086 303 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3iut A 1.2 BS01 KB2 A 1 G23 C25 S61 S64 G65 G66 L67 D161 H162 G23 C25 S61 S64 G65 G66 L67 D161 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 20088534 300 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLAEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDGAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 3iv5 A 2.9 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3iv5 A 2.9 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3iv5 B 2.9 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3iv5 B 2.9 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3ivc A 2.13 BS01 FG4 A 1 P38 T39 M40 H44 G46 H47 K160 Q164 V187 S196 S197 P38 T39 M40 H44 G46 H47 K160 Q164 V187 S196 S197 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=75uM remove_due_to_license_issue P9WIL5 19780086 302 MAIPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFAGTDRPDG 3ivg B 1.95 BS01 FG5 B 1 P38 T39 M40 H44 G46 H47 Q72 V142 K160 V187 S196 P37 T38 M39 H43 G45 H46 Q71 V129 K147 V174 S183 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M39 H43 H46 D75 D76 Q79 K147 S183 S184 R185 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=50uM remove_due_to_license_issue P9WIL5 19780086 305 AIPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIG 3ivh A 1.8 BS01 1LI A 1 D93 G95 S96 Y132 T133 F169 Y259 I287 D289 G291 D35 G37 S38 Y74 T75 F111 Y197 I225 D227 G229 D93 S96 N98 A100 Y132 D289 T292 D35 S38 N40 A42 Y74 D227 T230 3.4.23.46 0004190,0006508,0016020 ic50=47nM remove_due_to_license_issue IC50=47nM P56817 19811916 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3ivi A 2.2 BS01 2LI A 1 D93 G95 S96 P131 Y132 T133 F169 Y259 I287 D289 G291 T292 T390 V393 D35 G37 S38 P73 Y74 T75 F111 Y197 I225 D227 G229 T230 T323 V326 D93 S96 N98 A100 Y132 D289 T292 D35 S38 N40 A42 Y74 D227 T230 3.4.23.46 0004190,0006508,0016020 ic50=12nM remove_due_to_license_issue P56817 19811916 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3ivx A 1.73 BS01 FG6 A 1 P38 T39 M40 H44 G46 H47 V143 F157 K160 Q164 V187 M195 S196 S197 P36 T37 M38 H42 G44 H45 V141 F155 K158 Q162 V185 M193 S194 S195 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1.8uM remove_due_to_license_issue Kd=1800nM P9WIL5 19780086 302 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3ivx A 1.73 BS02 FG6 A 2 M71 L114 P133 T134 G138 M69 L112 P131 T132 G136 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1.8uM remove_due_to_license_issue Kd=1800nM P9WIL5 19780086 303 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3iw4 A 2.8 BS01 LW4 A 1 L345 F350 V353 A366 T401 M417 E418 Y419 V420 D467 M470 A480 D481 L15 F20 V23 A36 T71 M87 E88 Y89 V90 D137 M140 A150 D151 D463 K465 N468 D481 T501 D133 K135 N138 D151 T171 2.7.11.13 0004672,0004674,0004697,0005524,0006468 remove_due_to_license_issue IC50=2.1nM P17252 19827831 901 LDRVKLTDFNFLMVLGKGSFGKVMLADRKGTEELYAIKILKKDVVIQDDDVECTMVEKRVLALLDKPPFLTQLHSCFQTVDRLYFVMEYVNGGDLMYHIQQVGKFKEPQAVFYAAEISIGLFFLHKRGIIYRDLKLDNVMLDSEGHIKIADFGMCKEHMMDGVTTREFCGTPDYIAPEIIAYQPYGKSVDWWAYGVLLYEMLAGQPPFDGEDEDELFQSIMEHNVSYPKSLSKEAVSICKGLMTKHPAKRLGCGPEGERDVREHAFFRRIDWEKLENREIQPPFKPKVFDKFFTRGQPVLTPPDQLVIANIDQSDFEGFSYVNPQFVHPILQ 3iw5 A 2.5 BS01 DF3 A 1 V30 V38 A51 K53 L75 L104 T106 L108 M109 G110 A111 L167 L171 V27 V33 A46 K48 L70 L99 T101 L103 M104 G105 A106 L162 L166 D150 K152 N155 D168 T185 D145 K147 N150 D163 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=0.839uM remove_due_to_license_issue Q16539 19950957 362 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPPL 3iw6 A 2.1 BS01 PP0 A 1 V30 K53 L75 L104 T106 M109 G110 A111 D112 N115 L171 V27 K48 L70 L99 T101 M104 G105 A106 D107 N110 L166 D150 K152 N155 D168 T185 D145 K147 N150 D163 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=3.29uM remove_due_to_license_issue Q16539 19950957 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPPL 3iw7 A 2.4 BS01 IPK A 1 V38 K53 T106 M109 G110 A111 L171 V33 K48 T101 M104 G105 A106 L166 D150 K152 N155 D168 T185 D145 K147 N150 D163 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 19950957 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPP 3iw8 A 2.0 BS01 HIZ A 1 K53 E71 L74 L104 T106 D168 F169 K48 E66 L69 L99 T101 D163 F164 D150 K152 N155 D168 T185 D145 K147 N150 D163 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=13.4uM remove_due_to_license_issue Q16539 19950957 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPP 3iwn C 3.2 BS01 rna A 0 Y808 N810 N811 E814 K817 S843 L844 K845 M846 R847 G848 Q849 F851 Q880 K883 T884 S886 D887 Y8 N10 N11 E14 K17 S43 L44 K45 M46 R47 G48 Q49 F51 Q80 K83 T84 S86 D87 ? 0003676,0003723 remove_due_to_license_issue P09012 19898478 1 ~ 93 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAK 3iwn D 3.2 BS01 rna A 0 T901 R965 Q968 G969 R978 Y981 T1 R65 Q68 G69 R78 Y81 ? 0003676,0003723 remove_due_to_license_issue P09012 19898478 1 ~ 93 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAK 3iwn D 3.2 BS02 rna B 0 Y908 K917 R942 L944 K945 M946 R947 G948 Q949 F951 K983 S986 D987 Y8 K17 R42 L44 K45 M46 R47 G48 Q49 F51 K83 S86 D87 ? 0003676,0003723 remove_due_to_license_issue P09012 19898478 101 ~ 193 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAK 3iww A 2.3 BS04 YZE A 1 R210 N257 E424 L428 R463 D465 G518 N519 R534 R536 Y552 H553 Y700 R156 N203 E370 L374 R409 D411 G464 N465 R480 R482 Y498 H499 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=11nM remove_due_to_license_issue Ki=11nM Q04609 19897367 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3ixg B 2.14 BS01 BZB B 1 S64 L119 Q120 Y150 N152 Y221 A318 S61 L116 Q117 Y147 N149 Y218 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue IC50=200nM, Ki=27nM P00811 19913034 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFIGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3ixj A 2.2 BS01 586 A 1 G59 Q60 G61 L78 D80 G82 P118 Y119 T120 Q121 G122 F156 I158 Y246 D276 G278 T279 T280 N281 R283 G14 Q15 G16 L33 D35 G37 P73 Y74 T75 Q76 G77 F111 I113 Y190 D220 G222 T223 T224 N225 R227 D80 S83 N85 A87 Y119 D276 T279 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.32nM remove_due_to_license_issue Ki=<1nM, IC50=0.320000nM P56817 20128595 500 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3ixk A 2.5 BS01 929 A 1 G59 Q60 G61 D80 G82 S83 P118 Y119 T120 Q121 G122 F156 I158 Y246 D276 G278 T279 T280 N281 R283 G14 Q15 G16 D35 G37 S38 P73 Y74 T75 Q76 G77 F111 I113 Y190 D220 G222 T223 T224 N225 R227 D80 S83 N85 A87 Y119 D276 T279 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=6.6nM remove_due_to_license_issue IC50=4500nM P56817 20036448 500 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3jdw A 2.4 BS01 ORN A 1 M302 H303 A306 R322 S354 S355 C407 M239 H240 A243 R259 S291 S292 C344 E71 D170 D254 H303 D305 N361 H406 C407 E8 D107 D191 H240 D242 N298 H343 C344 2.1.4.1 0005515,0005737,0005739,0005743,0005758,0006600,0006601,0007611,0014889,0015067,0015068,0016740,0070062,0120162 Ki=253uM remove_due_to_license_issue P50440 9218780 500 CPVSSYNEWDPLEEVIVGRAENACVPPFTIEVKANTYEKYWPFYQKQGGHYFPKDHLKKAVAEIEEMCNILKTEGVTVRRPDPIDWSLKYKTPDFESTGLYSAMPRDILIVVGNEIIEAPMAWRSRFFEYRAYRSIIKDYFHRGAKWTTAPKPTMADELYNQDYPIHSVEDRHKLAAQGKFVTTEFEPCFDAADFIRAGRDIFAQRSQVTNYLGIEWMRRHLAPDYRVHIISFKDPNPMHIDATFNIIGPGIVLSNPDRPCHQIDLFKKAGWTIITPPTPIIPDDHPLWMSSKWLSMNVLMLDEKRVMVDANEVPIQKMFEKLGITTIKVNIRNANSLGGGFHCWTCDVRRRGTLQSYLD 3jpv A 2.35 BS02 1DR A 1 L44 F49 V52 K67 L174 I185 D186 L12 F17 V20 K35 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.12uM remove_due_to_license_issue IC50=120nM P11309 19788246 313 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3jq7 A 1.8 BS02 DX2 A 1 R14 S95 F97 Y174 V206 L209 P210 R13 S94 F96 Y155 V187 L190 P191 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki=1.2uM remove_due_to_license_issue Q581W1 19916554 271 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jq8 A 1.95 BS02 DX3 A 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki>35uM remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jq9 A 2.3 BS02 AX1 A 1 S95 F97 D161 M163 C168 Y174 P210 S94 F96 D142 M144 C149 Y155 P191 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki=0.4uM remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jq9 D 2.3 BS02 AX1 D 1 S95 F97 M163 C168 Y174 G205 S94 F96 M144 C149 Y155 G186 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki=0.4uM remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jqa A 1.9 BS02 DX4 A 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jqb A 2.4 BS02 DX6 A 1 S95 F97 Y174 M213 W221 S94 F96 Y155 M194 W202 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki=0.96uM remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jqf A 1.6 BS02 AX2 A 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jqg A 1.9 BS02 AX6 A 1 R14 S95 F97 Y174 P210 W221 R13 S94 F96 Y155 P191 W202 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki=18uM remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jqg D 1.9 BS02 AX6 D 1 S95 F97 Y174 P210 M213 S94 F96 Y155 P191 M194 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0016491 Ki=18uM remove_due_to_license_issue Q581W1 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3jr9 A 2.9 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jr9 A 2.9 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jr9 B 2.9 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jr9 B 2.9 BS02 dna D 0 I83 N84 T87 K90 I83 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jra A 3.11 BS01 dna C 0 I83 N84 T87 K90 I76 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jra A 3.11 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jra B 3.11 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jra B 3.11 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrb A 3.1 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrb A 3.1 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrb B 3.1 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrb B 3.1 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrc A 3.08 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrc A 3.08 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrc B 3.08 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrc B 3.08 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrd A 3.1 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrd A 3.1 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrd B 3.1 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrd B 3.1 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jre A 3.17 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jre A 3.17 BS02 dna D 0 Q74 T75 R85 R89 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jre B 3.17 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jre B 3.17 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrf A 3.05 BS01 dna C 0 N84 T87 N77 T80 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrf A 3.05 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrf B 3.05 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrf B 3.05 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrg A 3.11 BS01 dna C 0 I83 N84 T87 K90 I76 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrg A 3.11 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrg B 3.11 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrg B 3.11 BS02 dna D 0 N84 T87 N84 T87 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrh A 2.88 BS01 dna C 0 N84 T87 N77 T80 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrh A 2.88 BS02 dna D 0 Q74 T75 R85 R89 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrh B 2.88 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrh B 2.88 BS02 dna D 0 N84 T87 N84 T87 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jri A 3.11 BS01 dna C 0 I83 N84 T87 K90 I76 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jri A 3.11 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jri B 3.11 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jri B 3.11 BS02 dna D 0 N84 T87 N84 T87 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 20395367 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 3jrs A 2.05 BS01 A8S A 1 K86 A116 F135 L144 F189 V193 K56 A86 F105 L114 F154 V158 ? 0004864,0005515,0005634,0005737,0005886,0006952,0009536,0009738,0010427,0038023,0042802,0042803,0062049,0080163 Kd=52uM remove_due_to_license_issue Q8VZS8 19855379 1 DLTQDEFTQLSQSIAEFHTYQLGNGRCSSLLAQRIHAPPETVWSVVRRFDRPQIYKHFIKSCNVSEDFEMRVGCTRDVNVISGLPANTSRERLDLLDDDRRVTGFSITGGEHRLRNYKSVTTVHRFEKRIWTVVLESYVVDVPEGNSEEDTRLFADTVIRLNLQKLASITEAMN 3jrx A 2.5 BS01 S1A A 1 K274 R277 S278 P590 E593 M594 V598 N599 W681 F704 K38 R41 S42 P348 E351 M352 V356 N357 W429 F442 E567 E580 N582 E588 R652 E325 E338 N340 E346 R410 6.4.1.2 0003989,0005524,0046872 Kd~1nM remove_due_to_license_issue O00763 19900410 1000 DLHRDFTVASPAEFVTRFGGDRVIEKVLIANNGIAAVKCMRSIRRWAYEMFRNERAIRFVVMVTPEDLKANAEYIKMADHYVPVPGGPNNNNYANVELIVDIAKRIPVQAVWAGWGHASENPKLPELLCKNGVAFLGPPSEAMWALGDKIASTVVAQTLQVPTLPWSGSGLTVEWQGKRISVPEDVYDKGCVKDVDEGLEAAERIGFPLMIKASEGGGGKGIRKAESAEDFPILFRQVQSEIPGSPIFLMKLAQHARHLEVQILADQYGNAVSLFGRDCSIQRRHQKIVEEAPATIAPLAIFEFMEQCAIRLAKTVGYVSAGTVEYLYSQDGSFHFLELNPRLQVEHPCTEMIADVNLPAAQLQIAMGVPLHRLKDIRLLYGESPWGVTPISFETPSNPPLARGHVIAARITSSGTVQELNFRSSKNVWGYFSVASQFGHCFSWGENREEAISNMVVALKELSIRGDFRTTVEYLINLLETESFQNNDIDTGWLDY 3jsi A 2.72 BS02 WTC A 1 M365 L420 Y424 A452 Q453 F456 M188 L243 Y247 A275 Q276 F279 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue IC50=2.1nM O76083 19919087 903 GSHMTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 3jso A 2.29 BS01 dna C 0 T5 R7 F37 R38 S39 N41 A42 E45 H46 G61 A62 S63 T4 R6 F36 R37 S38 N40 A41 E44 H45 G60 A61 S62 M118 S119 E152 A156 M107 S108 E141 A145 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLGLPLVGRVAAGEPLIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNG 3jso A 2.29 BS02 dna D 0 T27 R28 N41 S60 G61 S63 R64 T26 R27 N40 S59 G60 S62 R63 M118 S119 E152 A156 M107 S108 E141 A145 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLGLPLVGRVAAGEPLIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNG 3jso B 2.29 BS01 dna C 0 T27 R28 N41 K48 S60 R64 T26 R27 N40 K47 S59 R63 M118 S119 E152 A156 M105 S106 E139 A143 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLGLPLVGRVAAGEIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNGDWL 3jso B 2.29 BS02 dna D 0 T5 R7 F37 R38 S39 N41 A42 E45 H46 R52 G61 S63 T4 R6 F36 R37 S38 N40 A41 E44 H45 R51 G60 S62 M118 S119 E152 A156 M105 S106 E139 A143 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLGLPLVGRVAAGEIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNGDWL 3jsp A 2.9 BS01 dna C 0 T5 R7 Q8 F37 R38 S39 N41 A42 E45 H46 S63 T4 R6 Q7 F36 R37 S38 N40 A41 E44 H45 S62 M118 S119 E152 A156 M113 S114 E147 A151 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLQGLPLVGRVAAGEPLLAQQHIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNG 3jsp A 2.9 BS02 dna D 0 T27 R28 N41 E44 K48 S60 S63 R64 T26 R27 N40 E43 K47 S59 S62 R63 M118 S119 E152 A156 M113 S114 E147 A151 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLQGLPLVGRVAAGEPLLAQQHIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNG 3jsp B 2.9 BS01 dna C 0 T27 R28 N41 E44 K48 S63 R64 T26 R27 N40 E43 K47 S62 R63 M118 S119 E152 A156 M108 S109 E142 A146 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLQEGLPLVGRVLAQQHIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNGDWL 3jsp B 2.9 BS02 dna D 0 T5 R7 Q8 F37 R38 S39 N41 A42 E45 H46 R52 S63 T4 R6 Q7 F36 R37 S38 N40 A41 E44 H45 R51 S62 M118 S119 E152 A156 M108 S109 E142 A146 3.4.21.88 0000976,0001217,0003677,0004252,0005515,0005829,0006260,0006281,0006351,0006355,0006508,0006974,0009432,0016787,0032993,0042802,0045892 remove_due_to_license_issue P0A7C2 20703307 1 ~ 22 KALTARQQEVFDLIRDHISQTGMPPTRAEIAQRLGFRSPNAAEEHLKALARKGVIEIVSGASRGIRLLQEGLPLVGRVLAQQHIEGHYQVDPSLFKPNADFLLRVSGMSMKDIGIMDGDLLAVHKTQDVRNGQVVVARIDDEVTVARLKKQGNKVELLPENSEFKPIVVDLRQQSFTIEGLAVGVIRNGDWL 3jsw A 2.3 BS02 JAR A 1 L420 Y424 Q453 F456 V460 L243 Y247 Q276 F279 V283 3.1.4.35 0004114,0007165,0008081 ic50=66nM remove_due_to_license_issue IC50=66nM O76083 19919087 900 GSHMTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 3juk A 2.3 BS01 UPG A 1 A10 G11 E26 Q102 M105 G107 L108 A111 D131 Y170 G171 E190 K191 V203 A10 G11 E26 Q94 M97 G99 L100 A103 D123 Y162 G163 E182 K183 V195 2.7.7.9 0003983,0006011,0009058,0016779,0046872 remove_due_to_license_issue O25363 20238176 282 MIKKCLFPAAGYGTRFLPITKTIPKEMLPIVDKPLIQYAVEEAMEAGCEVMAIVTGRNKRSLEDYFDTSYTNKENALKSIRNIIEKCCFSYVRQKQMKGLGHAILTGEALIGNEPFAVILADDLCISHDHPSVLKQMTSLYQKYQCSIVAIEEVALEEVSKYGVIRGEWLEEGVYEIKDMVEKPNQEDAPSNLAVIGRYILTPDIFEILSETKPGKNNEIQITDALRTQAKRKRIIAYQFKGKRYDCGSVEGYIEASNAYYKKRL 3juo A 2.2 BS01 AJD A 1 R38 R41 H73 A74 S77 F81 W84 E140 R29 R32 H64 A65 S68 F72 W75 E131 ? 0017000 Kd=8.55uM remove_due_to_license_issue Q396C9 19876985 500 TSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLPS 3juo B 2.2 BS01 AJD B 1 R38 R41 H73 A74 S77 F81 W84 E140 R31 R34 H66 A67 S70 F74 W77 E133 ? 0017000 Kd=8.55uM remove_due_to_license_issue Q396C9 19876985 500 ENTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLP 3jup A 1.9 BS01 AKD A 1 I62 H73 F81 W84 E140 Q147 I54 H65 F73 W76 E132 Q139 ? 0017000 Kd=2.63uM remove_due_to_license_issue Q396C9 19876985 500 NTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLPS 3jup B 1.9 BS01 AKD B 1 I62 H73 F81 W84 E140 Q147 I54 H65 F73 W76 E132 Q139 ? 0017000 Kd=2.63uM remove_due_to_license_issue Q396C9 19876985 500 NTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLPS 3juq A 1.75 BS01 AJD A 1 R38 R41 H73 A74 S77 F81 W84 E140 R30 R33 H65 A66 S69 F73 W76 E132 ? 0017000 Kd=8.55uM remove_due_to_license_issue Q396C9 19876985 500 NTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGLP 3juq B 1.75 BS01 AJD B 1 R38 R41 H73 A74 S77 W84 E140 R31 R34 H66 A67 S70 W77 E133 ? 0017000 Kd=8.55uM remove_due_to_license_issue Q396C9 19876985 500 ENTSENRAQVAARQHNRKIVEQYMHTRGEARLKRHLLFTEDGVGGLWTTDSGQPIAIRGREKLGEHAVWSLQCFPDWVWTDIQIFETQDPNWFWVECRGEGAIVFPGYPRGQYRNHFLHSFRFENGLIKEQREFMNPCEQFRSLGIEVPEVRRDGL 3jvr A 1.76 BS01 AGX A 1 F93 D94 I96 E97 P98 G204 E205 L206 F79 D80 I82 E83 P84 G190 E191 L192 D130 K132 E134 N135 D148 T170 D116 K118 E120 N121 D134 T156 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=1.89uM remove_due_to_license_issue Ki=1.89e+3nM O14757 19743875 901 AVPFVEDWDLVQTLGEEVQLAVNRVTEEAVAVKIVDMENIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKG 3jvs A 1.9 BS01 AGY A 1 F93 D94 I96 E97 P98 P133 G204 E205 L206 F77 D78 I80 E81 P82 P117 G188 E189 L190 D130 K132 E134 N135 D148 T170 D114 K116 E118 N119 D132 T154 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Kd=0.29uM remove_due_to_license_issue Ki=146nM O14757 19743875 900 AVPFVEDWDLVQTLGEEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKG 3jwq A 2.87 BS02 VIA A 1 M804 Q817 F820 M269 Q282 F285 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76074,P51160 19798052 901 ETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFWEQGDLERTVLQQQPIPMMDRNKRDELPKLQVGFIDFVCTQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQ 3jwr A 2.994 BS04 IBM A 1 H613 F786 Q817 F820 H77 F250 Q281 F284 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76074,P51160 19798052 901 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFWEQGDLERTVLQQQPIPMMDRNKRDELPKLQVGFIDFVCTQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQ 3jwr A 2.994 BS05 IBM A 2 L701 S702 L704 Y709 L165 S166 L168 Y173 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76074,P51160 19798052 902 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFWEQGDLERTVLQQQPIPMMDRNKRDELPKLQVGFIDFVCTQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQ 3jwr A 2.994 BS06 IBM A 3 D687 L690 D151 L154 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76074,P51160 19798052 903 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFWEQGDLERTVLQQQPIPMMDRNKRDELPKLQVGFIDFVCTQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQ 3jxw A 2.8 BS01 LXG A 1 F49 V52 A65 K67 L174 I185 D186 F17 V20 A33 K35 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue Ki=1nM P11309 1000 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 3jy0 A 2.4 BS01 LYG A 1 V52 A65 K67 E121 N172 L174 I185 D186 V20 A33 K35 E89 N140 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue Ki=5nM P11309 1000 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSL 3jy9 A 2.1 BS01 JZH A 1 L855 G856 V863 A880 E898 V911 M929 Y931 L932 L983 D994 F995 L14 G15 V20 A37 E55 V68 M83 Y85 L86 L137 D148 F149 M865 D976 A978 R980 N981 D994 S1016 M22 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.001uM remove_due_to_license_issue IC50=2.7E2nM, Ki=1nM O60674 20014869 1 TQFEERHLKFLQQLGKGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 3jya A 2.1 BS01 LWG A 1 L44 F49 V52 A65 R122 L174 I185 L12 F17 V20 A33 R90 L142 I153 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue Ki=130.1nM P11309 1000 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 3jyj A 1.87 BS01 JZI A 1 H59 L61 K63 C113 S114 L122 F134 S154 H157 H9 L11 K13 C63 S64 L72 F84 S104 H107 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 Ki=1.8uM remove_due_to_license_issue IC50=>50000nM, Ki=1800nM Q13526 20207139 301 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3jzb A 2.007 BS01 4HY A 1 F215 F218 I222 M256 M259 A263 R266 L276 S277 L292 H381 F72 F75 I79 M113 M116 A120 R123 L133 S134 L149 H238 ? 0003677,0004879,0006355 ic50~0.1nM remove_due_to_license_issue IC50=0.14nM P10827 19926848 1 GSHMEEMIRSLQQRPEPTPEEWDLIHIATEAHRSTNAQGSHWKQRRKFLPDDIGQSPIVSMPDGDKVDLEAFSEFTKIITPAITRVVDFAKKLPMFSELPCEDQIILLKGCCMEIMSLRAAVRYDPESDTLTLSGEMAVKREQLKNGGLGVVSDAIFELGKSLSAFNLDDTEVALLQAVLLMSTDRSGLLCVDKIEKSQEAYLLAFEHYVNHRKHNIPHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 3jzc A 2.5 BS01 4HY A 1 F269 F272 I276 A279 M313 L330 N331 L346 H435 F455 F57 F60 I64 A67 M101 L118 N119 L134 H223 F243 ? 0003677,0004879,0006355 ic50~1nM remove_due_to_license_issue IC50=0.0407nM P10828 19926848 1 EELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGQVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFE 3jzf B 2.13 BS01 JZK B 1 K116 K159 A160 G164 G166 R167 G168 M169 Y199 E201 K202 Y203 H209 H236 L278 I287 E288 K118 K161 A162 G166 G168 R169 G170 M171 Y201 E203 K204 Y205 H211 H238 L280 I289 E290 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K118 K161 D198 H211 R237 T276 E278 E290 N292 R294 E298 R340 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=5uM remove_due_to_license_issue P24182 19875284 466 RHMLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLG 3jzi A 2.31 BS01 JZL A 1 K116 K159 A160 G164 G165 M169 Y199 E201 K202 Y203 H209 Q233 H236 L278 I287 E288 K116 K159 A160 G164 G165 M169 Y199 E201 K202 Y203 H209 Q233 H236 L278 I287 E288 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=5uM remove_due_to_license_issue P24182 19875284 466 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLG 3jzk A 2.1 BS01 YIN A 1 L54 G58 I61 M62 F86 F91 V93 H96 I99 Y100 L37 G41 I44 M45 F69 F74 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 ic50=1.23uM remove_due_to_license_issue Q00987 19856920 1 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 3k02 A 1.55 BS01 TXT A 1 T27 E32 F59 E83 W86 D133 D180 Y182 W183 W254 W290 R358 N365 T11 E16 F43 E67 W70 D117 D164 Y166 W167 W238 W274 R342 N349 ? 0015768,0042956,0055052,1901982 Kd=10uM remove_due_to_license_issue B0B0V1 20132828 405 ELSGTVTFWDTSNEAEKATYQALAEGFEKEHPKVDVKYVNVPFGEANAKFKNAAGGNSGAPDVMRTEVAWVADFASIGYLAPLDGTPALDDGSDHLPQAAASTRYEGKTYAVPQVIDTLALFYNKELLTKAGVEVPGSVAELKTAAAEITEKTGATGLYLRGDDPYWFLPYLYGEGGDLVDEKNKTVTVDDEAGVRAYRVIKDLVDSKAAITDASDGWNNMQNAFKSGKVAMMVNGPWAIEDVKAGARFKDAGNLGVAPVPAGSAGQGSPQGGWNLSVYAGSKNLDASYAFVKYMSSAKVQQQTTEKLSLLPTRTSVYEVPSVADNEMVKFFKPAVDKAVERPWIAEGNALFEPIRLQMANVLSGETSPDEAAANTGDAYRKLLKDYK 3k0j A 3.1 BS01 rna E 0 Y213 N215 N216 E219 K222 D224 K227 K228 I243 R247 S248 L249 K250 M251 R252 Q254 F256 K280 R283 Q285 Y286 A287 K288 T289 D290 S291 D292 Y8 N10 N11 E14 K17 D19 K22 K23 I38 R42 S43 L44 K45 M46 R47 Q49 F51 K75 R78 Q80 Y81 A82 K83 T84 D85 S86 D87 ? 0003676,0003723 remove_due_to_license_issue P09012 19948769 4 ~ 90 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAKM 3k0j B 3.1 BS01 rna F 0 Y313 N315 N316 E319 K328 H331 I343 R347 S348 L349 K350 M351 R352 Q354 F356 R383 K388 D390 S391 D392 Y8 N10 N11 E14 K23 H26 I38 R42 S43 L44 K45 M46 R47 Q49 F51 R78 K83 D85 S86 D87 ? 0003676,0003723 remove_due_to_license_issue P09012 19948769 104 ~ 190 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKTDSDIIAKM 3k0j C 3.1 BS01 rna F 0 E425 K428 E22 K25 ? 0003676,0003723 remove_due_to_license_issue P09012 19948769 104 ~ 190 PETRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSLKMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKT 3k0j D 3.1 BS01 rna E 0 E525 K528 E20 K23 ? 0003676,0003723 remove_due_to_license_issue P09012 19948769 4 ~ 90 TRPNHTIYINNLNEKIKKDELKKSLHAIFSRFGQILDILVSRSMRGQAFVIFKEVSSATNALRSMQGFPFYDKPMRIQYAKT 3k1j A 2.0 BS01 ADP A 1 V43 I44 G70 T71 G72 K73 S74 M75 E342 R345 L378 R379 V26 I27 G53 T54 G55 K56 S57 M58 E273 R276 L309 R310 ? 0000166,0004176,0004252,0005524,0005886,0006355,0006508,0008134,0008236,0016887,0030163 remove_due_to_license_issue B6YU74 20834233 642 GESLELGIEFTTTEEIEVPEKLIDQVIGQEHAVEVIKTAANQKRHVLLIGEPGTGKSMLGQAMAELLPTETLEDILVFPNPEDENMPRIKTVPACQGRRIVEKYREKAKSQESVLVPKLLVDNCGRTKAPFIDATGAHAGALLGDVRHDPFLGTPAHERVEPGMIHRAHKGVLFIDEIATLSLKMQQSLLTAMQEKKFPITGQSEMSSGAMVRTEPVPCDFVLVAAGNLDTVDKMHPALRSRIRGYGYEVYMRTTMPDTIENRRKLVQFVAQEVKRDGKIPHFTKEAVEEIVREAQKRAGRKGHLTLRLRDLGGIVRAAGDIAVKKGKKYVEREDVIEAVKMAKPLEKQLADWYIERKKEYQVIKTEGSEIGRVNGLAVIGEQSGIVLPIEAVVAPAASKEEGKIIVTGKLGEIAKEAVQNVSAIIKRYKGEDISRYDIHVQFLQTYEGVEGDAASISVATAVISALEGIPIRQDVAMTGSLSVRGEVLPIGGATPAIEAAIEAGIKMVIIPKSNEKDVFLSKDKAEKIQIFPVETIDEVLEIALEESEKKRELLRRIRETLPLSL 3k22 A 2.1 BS02 JZS A 1 L563 N564 L566 G567 Q570 A574 M601 M604 A607 F623 F749 L38 N39 L41 G42 Q45 A49 M76 M79 A82 F97 F223 ? remove_due_to_license_issue P04150 19822747 1 PQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k23 A 3.0 BS03 JZN A 1 P541 M560 L563 N564 L566 Q570 M601 L603 M604 A605 A607 L608 F623 C736 P17 M35 L38 N39 L41 Q45 M76 L78 M79 A80 A82 L83 F98 C206 ? remove_due_to_license_issue IC50=6.3nM P04150 19822747 1 LPQLTPTLVSLLEVIEPEVLYAGYDSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k2f A 1.98 BS02 NKX A 1 W5 N62 H64 N67 Q92 H94 H119 V121 F131 L198 T199 T200 W209 W2 N59 H61 N64 Q89 H91 H116 V118 F127 L194 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=63nM remove_due_to_license_issue P00918 19854054 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3k37 A 2.0 BS02 BCZ A 1 R116 E117 D149 R150 E275 R292 R374 Y409 R39 E40 D72 R73 E198 R215 R297 Y332 D149 E276 R292 R374 Y409 D72 E199 R215 R297 Y332 3.2.1.18 0004308,0005975,0016020,0033644,0055036 Ki=1.2nM remove_due_to_license_issue Q3S340 20695427 468 PEWTYPRLSCPGSTFQKALLISPHRFGETKGNSAPLIIREPFIACGPKECKHFALTHYAAQPGGYYNGTRGDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGKEWTYIGVDGPDNNALLKIKYGEAYTDTYHSYANNILRTQESACNCIGGNCYLMITDGSASGISECRFLKIREGRIIKEIFPTGRVKHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTETYLDTPRPDDGSITGPCESNGDKGSGGIKGGFVHQRMASKIGRWYSRTMSKTKRMGMGLYVKYDGDPWTDSDALALSGVMVSMEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKETWHSAATAIYCLMGSGQLLWDTVTGVDMAL 3k39 A 2.54 BS02 BCZ A 1 R116 E117 D149 R223 E226 E275 R292 R374 Y409 R39 E40 D72 R146 E149 E198 R215 R297 Y332 D149 E276 R292 R374 Y409 D72 E199 R215 R297 Y332 3.2.1.18 0004308,0005975,0016020,0033644,0055036 remove_due_to_license_issue Q3S340 20695427 1001 PEWTYPRLSCPGSTFQKALLISPHRFGETKGNSAPLIIREPFIACGPKECKHFALTHYAAQPGGYYNGTRGDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGKEWTYIGVDGPENNALLKIKYGEAYTDTYHSYANNILRTQESACNCIGGNCYLMITDGSASGISECRFLKIREGRIIKEIFPTGRVKHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTETYLDTPRPDDGSITGPCESNGDKGSGGIKGGFVHQRMASKIGRWYSRTMSKTKRMGMGLYVKYDGDPWTDSDALALSGVMVSMEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKETWHSAATAIYCLMGSGQLLWDTVTGVDMAL 3k3a A 2.59 BS02 G39 A 1 R116 E117 D149 R150 R223 E275 R292 R374 Y409 R39 E40 D72 R73 R146 E198 R215 R297 Y332 D149 E276 R292 R374 Y409 D72 E199 R215 R297 Y332 3.2.1.18 0004308,0005975,0016020,0033644,0055036 remove_due_to_license_issue Q3S340 20695427 1 PEWTYPRLSCPGSTFQKALLISPHRFGETKGNSAPLIIREPFIACGPKECKHFALTHYAAQPGGYYNGTRGDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGKEWTYIGVDGPENNALLKIKYGEAYTDTYHSYANNILRTQESACNCIGGNCYLMITDGSASGISECRFLKIREGRIIKEIFPTGRVKHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTETYLDTPRPDDGSITGPCESNGDKGSGGIKGGFVHQRMASKIGRWYSRTMSKTKRMGMGLYVKYDGDPWTDSDALALSGVMVSMEEPGWYSFGFEIKDKKCDVPCIGIEMVHDGGKETWHSAATAIYCLMGSGQLLWDTVTGVDMAL 3k3b A 2.4 BS02 L31 A 1 E116 E118 R119 W127 D130 A133 I136 P137 Y211 L214 E101 E103 R104 W112 D115 A118 I121 P122 Y196 L199 ? 0003777,0005524,0007018,0008017 ic50=0.2uM remove_due_to_license_issue IC50=200nM P52732 19945875 371 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSEAGNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 3k3e A 2.7 BS02 PDB A 1 H252 I403 L420 Y424 Q453 F456 H66 I217 L234 Y238 Q267 F270 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76083 20121115 600 LLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 3k3g A 2.4 BS01 MMU A 1 E187 F190 F243 E184 F187 F240 ? 0005886,0015204,0015265,0016020,0033219,0042802,0070207,0071918 ic50=1.4mM remove_due_to_license_issue Q72CX3 19865084 347 RAFGEQLLKNPLIEFCDSVCRGCGQVMFQNNTVTGLLFFAGIFYNSTTLGVCAVLGTAASTLTAQLLGVDKPLVRAGLFGFNGTLAGIALPFFFNYEPAMLGYVALNGAFTTIIMASLLNFLGKWGVPALTAPFVLATWLLMFGVYKLSLFHPGALIAPALPSVDMGTVTGRTFMEGLFKGVGEVMFQDNIVTGVIFVVAILVNSRISALFAVIGSLVGLCTALIMHSPETPVRLGLYGFNSVLCGIAMGGIFFYLNIRTFLYALGCMVLGAIATGAFSVLLSPIGMPALTWPFIVVTWLFLFAGSMFRNIAQVPTEKAGTPEDNLRSLAI 3k3g A 2.4 BS02 MMU A 2 Q24 V25 F27 F80 Q25 V26 F28 F81 ? 0005886,0015204,0015265,0016020,0033219,0042802,0070207,0071918 ic50=1.4mM remove_due_to_license_issue Q72CX3 19865084 348 RAFGEQLLKNPLIEFCDSVCRGCGQVMFQNNTVTGLLFFAGIFYNSTTLGVCAVLGTAASTLTAQLLGVDKPLVRAGLFGFNGTLAGIALPFFFNYEPAMLGYVALNGAFTTIIMASLLNFLGKWGVPALTAPFVLATWLLMFGVYKLSLFHPGALIAPALPSVDMGTVTGRTFMEGLFKGVGEVMFQDNIVTGVIFVVAILVNSRISALFAVIGSLVGLCTALIMHSPETPVRLGLYGFNSVLCGIAMGGIFFYLNIRTFLYALGCMVLGAIATGAFSVLLSPIGMPALTWPFIVVTWLFLFAGSMFRNIAQVPTEKAGTPEDNLRSLAI 3k3h A 2.5 BS02 BYE A 1 H252 L420 Y424 F441 Q453 F456 H67 L235 Y239 F256 Q268 F271 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76083 20121115 600 YLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 3k3i A 1.7 BS01 JZJ A 1 K53 E71 L74 L75 I84 T106 I141 H148 L167 D168 K49 E67 L70 L71 I80 T102 I133 H140 L159 D160 D150 K152 N155 D168 T185 D142 K144 N147 D160 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=1900nM Q16539 19843080 1 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3k3j A 1.995 BS01 F4C A 1 K53 R70 E71 L74 I84 L104 T106 H148 D168 F169 K47 R64 E65 L68 I78 L98 T100 H138 D158 F159 D150 K152 N155 D168 T185 D140 K142 N145 D158 T162 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=2.4e+3nM Q16539 19843080 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3k41 A 1.9 BS01 M6D A 1 Y45 Q66 Y102 D103 N104 H105 R111 E133 R135 Y143 Y36 Q57 Y93 D94 N95 H96 R102 E124 R126 Y134 ? 0005768,0005794,0006622,0019904 Kd=150mM remove_due_to_license_issue P11456 19928875 500 KTCDLVSEKQLALLKRLTPLFQKSFESTVGQSPDMYSYVFRVCREAGQHSSGAGLVQIQKSNGKETVVGRFNETQIFQGSNWIMLIYKGGDEYDNHCGREQRRAVVMISCNRHTLADNFNPVSEERGMVQDCFYLFEMDSSLACS 3k49 A 2.5 BS01 rna B 0 Q550 R554 Q557 F587 N589 Y590 Y623 R626 Q629 Q658 N661 H662 Q665 C697 R698 Q701 N733 Y734 Q737 K772 S775 N776 E779 N824 Y825 L864 A865 S866 K869 Q30 R34 Q37 F67 N69 Y70 Y103 R106 Q109 Q138 N141 H142 Q145 C177 R178 Q181 N213 Y214 Q217 K252 S255 N256 E259 N304 Y305 L342 A343 S344 K347 ? 0003723 remove_due_to_license_issue Q07807 19918084 1 ~ 10 SPLLEQLRNSSSNMSLKDIFGHSLEFCKDQHGSRFIQRELATSPASEKEVIFNEIRDDAIELSNDVFGNYVIQKFFEFGSKIQKNTLVDQFKGNMKQLSLQMYACRVIQKALEYIDSNQRIELVLELSDSVLQMIKDQNGNHVIQKAIETIPIEKLPFILSSLTGHIYHLSTHSYGCRVIQRLLEFGSSEDQESILNELKDFIPYLIQDQYGNYVIQYVLQQDQFTNKEMVDIKQEIIETVANNVVEYSKHKFASNVVEKSILYGSKNQKDLIISKILPRDKNHALNLEDDSPMILMIKDQFANYVIQKLVNVSEGEGKKLIVIAIRAYLDKLNKSNGNRHLASVEKLAALVE 3k49 C 2.5 BS01 rna D 0 Q550 R554 Q557 N589 Y590 Y623 R626 Q629 Q658 N661 H662 Q665 C697 R698 Q701 N733 Y734 Q737 K772 S775 N776 E779 N824 Y825 L864 A865 S866 K869 Q30 R34 Q37 N69 Y70 Y103 R106 Q109 Q138 N141 H142 Q145 C177 R178 Q181 N213 Y214 Q217 K252 S255 N256 E259 N304 Y305 L342 A343 S344 K347 ? 0003723 remove_due_to_license_issue Q07807 19918084 1 ~ 10 SPLLEQLRNSSSNMSLKDIFGHSLEFCKDQHGSRFIQRELATSPASEKEVIFNEIRDDAIELSNDVFGNYVIQKFFEFGSKIQKNTLVDQFKGNMKQLSLQMYACRVIQKALEYIDSNQRIELVLELSDSVLQMIKDQNGNHVIQKAIETIPIEKLPFILSSLTGHIYHLSTHSYGCRVIQRLLEFGSSEDQESILNELKDFIPYLIQDQYGNYVIQYVLQQDQFTNKEMVDIKQEIIETVANNVVEYSKHKFASNVVEKSILYGSKNQKDLIISKILPRDKNHALNLEDDSPMILMIKDQFANYVIQKLVNVSEGEGKKLIVIAIRAYLDKLNKSNGNRHLASVEKLAALVE 3k49 E 2.5 BS01 rna F 0 Q550 R554 Q557 F587 N589 Y590 Q593 Y623 R626 Q629 Q658 N661 H662 Q665 C697 R698 Q701 N733 Y734 Q737 K772 S775 N776 E779 N824 Y825 L864 A865 S866 K869 Q30 R34 Q37 F67 N69 Y70 Q73 Y103 R106 Q109 Q138 N141 H142 Q145 C177 R178 Q181 N213 Y214 Q217 K252 S255 N256 E259 N304 Y305 L342 A343 S344 K347 ? 0003723 remove_due_to_license_issue Q07807 19918084 1 ~ 10 SPLLEQLRNSSSNMSLKDIFGHSLEFCKDQHGSRFIQRELATSPASEKEVIFNEIRDDAIELSNDVFGNYVIQKFFEFGSKIQKNTLVDQFKGNMKQLSLQMYACRVIQKALEYIDSNQRIELVLELSDSVLQMIKDQNGNHVIQKAIETIPIEKLPFILSSLTGHIYHLSTHSYGCRVIQRLLEFGSSEDQESILNELKDFIPYLIQDQYGNYVIQYVLQQDQFTNKEMVDIKQEIIETVANNVVEYSKHKFASNVVEKSILYGSKNQKDLIISKILPRDKNHALNLEDDSPMILMIKDQFANYVIQKLVNVSEGEGKKLIVIAIRAYLDKLNKSNGNRHLASVEKLAALVE 3k4d A 2.393 BS01 EVA A 1 D163 H330 E413 Y468 Y472 E504 W549 K568 D165 H332 E408 Y463 Y467 E499 W544 K563 D163 H296 H330 V355 F357 E413 Y468 E504 K568 D165 H298 H332 V357 F359 E408 Y463 E499 K563 3.2.1.31 0004553,0004566,0005829,0005975,0016798,0030246,0032991,0042802 Ki=7750nM remove_due_to_license_issue Ki=232nM P05804 21051639 604 SHMLRPVETPTREIKKLDGLWAFSLDRENCGIDQRWWESALQESRAIAVPGSFNDQFADADIRNYAGNVWYQREVFIPKGWAGQRIVLRFDAVTHYGKVWVNNQEVMEHQGGYTPFEADVTPYVIAGKSVRITVCVNNELNWQTIPPGMVITDENGKKKQSYFHDFFNYAGIHRSVMLYTTPNTWVDDITVVTHVAQDCNHASVDWQVVANGDVSVELRDADQQVVATGQGTSGTLQVVNPHLWQPGEGYLYELCVTAKSQTECDIYPLRVGIRSVAVKGEQFLINHKPFYFTGFGRHEDADLRGKGFDNVLMVHDHALMDWIGANSYRTSHYPYAEEMLDWADEHGIVVIDETAAVGFNLSLGKPKELYSEEAVNGETQQAHLQAIKELIARDKNHPSVVMWSIANEPDTRPQGAREYFAPLAEATRKLDPTRPITCVNVMFCDAHTDTISDLFDVLCLNRYYGWYVQSGDLETAEKVLEKELLAWQEKLHQPIIITEYGVDTLAGLHSMYTDMWSEEYQCAWLDMYHRVFDRVSAVVGEQVWNFADFATSQGILRVGGNKKGIFTRDRKPKSAAFLLQKRWTGMNFGEKPQQGG 3k4e A 3.2 BS01 rna B 0 Q550 R554 Q557 F587 N589 Y590 Y623 R626 Q629 H662 C697 R698 Y731 N733 Y734 Q737 K772 S775 N776 E779 N824 Y825 L864 A865 S866 Q28 R32 Q35 F65 N67 Y68 Y101 R104 Q107 H140 C175 R176 Y209 N211 Y212 Q215 K250 S253 N254 E257 N302 Y303 L332 A333 S334 ? 0003723 remove_due_to_license_issue Q07807 19918084 1 ~ 10 SPLLEQLRNSNMSLKDIFGHSLEFCKDQHGSRFIQRELATSPASEKEVIFNEIRDDAIELSNDVFGNYVIQKFFEFGSKIQKNTLVDQFKGNMKQLSLQMYACRVIQKALEYIDSNQRIELVLELSDSVLQMIKDQNGNHVIQKAIETIPIEKLPFILSSLTGHIYHLSTHSYGCRVIQRLLEFGSSEDQESILNELKDFIPYLIQDQYGNYVIQYVLQQDQFTNKEMVDIKQEIIETVANNVVEYSKHKFASNVVEKSILYGSKNQKDLIISKILPRDKNHALNLEDDSPMILMIKDQFANYVIQKLVNVSEGEGKKLIVIAIRAYLDKLLASVEKLAALVE 3k4e C 3.2 BS01 rna D 0 Q550 R554 Q557 F587 N589 Y590 Y623 R626 Q629 H662 C697 R698 Y731 N733 Y734 Q737 K772 S775 N776 E779 F822 N824 Y825 L864 A865 S866 Q28 R32 Q35 F65 N67 Y68 Y101 R104 Q107 H140 C175 R176 Y209 N211 Y212 Q215 K250 S253 N254 E257 F300 N302 Y303 L332 A333 S334 ? 0003723 remove_due_to_license_issue Q07807 19918084 1 ~ 10 SPLLEQLRNSNMSLKDIFGHSLEFCKDQHGSRFIQRELATSPASEKEVIFNEIRDDAIELSNDVFGNYVIQKFFEFGSKIQKNTLVDQFKGNMKQLSLQMYACRVIQKALEYIDSNQRIELVLELSDSVLQMIKDQNGNHVIQKAIETIPIEKLPFILSSLTGHIYHLSTHSYGCRVIQRLLEFGSSEDQESILNELKDFIPYLIQDQYGNYVIQYVLQQDQFTNKEMVDIKQEIIETVANNVVEYSKHKFASNVVEKSILYGSKNQKDLIISKILPRDKNHALNLEDDSPMILMIKDQFANYVIQKLVNVSEGEGKKLIVIAIRAYLDKLLASVEKLAALVE 3k4e E 3.2 BS01 rna F 0 Q550 R554 Q557 F587 N589 Y590 Y623 R626 Q629 H662 C697 R698 Y731 N733 Y734 Q737 K772 S775 N776 E779 F822 N824 Y825 L864 A865 S866 Q28 R32 Q35 F65 N67 Y68 Y101 R104 Q107 H140 C175 R176 Y209 N211 Y212 Q215 K250 S253 N254 E257 F300 N302 Y303 L332 A333 S334 ? 0003723 remove_due_to_license_issue Q07807 19918084 1 ~ 10 SPLLEQLRNSNMSLKDIFGHSLEFCKDQHGSRFIQRELATSPASEKEVIFNEIRDDAIELSNDVFGNYVIQKFFEFGSKIQKNTLVDQFKGNMKQLSLQMYACRVIQKALEYIDSNQRIELVLELSDSVLQMIKDQNGNHVIQKAIETIPIEKLPFILSSLTGHIYHLSTHSYGCRVIQRLLEFGSSEDQESILNELKDFIPYLIQDQYGNYVIQYVLQQDQFTNKEMVDIKQEIIETVANNVVEYSKHKFASNVVEKSILYGSKNQKDLIISKILPRDKNHALNLEDDSPMILMIKDQFANYVIQKLVNVSEGEGKKLIVIAIRAYLDKLLASVEKLAALVE 3k4q A 2.2 BS01 IHS A 1 Q27 Y28 R58 H59 R62 K68 R142 K278 H338 D339 Q21 Y22 R52 H53 R56 K62 R136 K272 H332 D333 3.1.3.-,3.1.3.8 0003993,0005576,0016158,0016787,0016791 Ki=4.6uM remove_due_to_license_issue P34752 20541524 500 SCDTVDQGYQCFSETSHLWGQYAPFFSLANESVISPEVPAGCRVTFAQVLSRHGARYPTDSKGKKYSALIEEIQQNATTFDGKYAFLKTYNYSLGADDLTPFGEQELVNSGIKFYQRYESLTRNIVPFIRSSGSSRVIASGKKFIEGFQSTKLKDPRAQPGQSSPKIDVVISEASSSNNTLDPGTCTVFEDSELADTVEANFTATFVPSIRQRLENDLSGVTLTDTEVTYLMDMCSFDTISTSTVDTKLSPFCDLFTHDEWINYDYLQSLKKYYGHGAGNPLGPTQGVGYANELIARLTHSPVHDDTSSNHTLDSSPATFPLNSTLYADFSHDNGIISILFALGLYNGTKPLSTTTVENITQTDGFSSAWTVPFASRLYVEMMQCQAEQEPLVRVLVNDRVVPLHGCPVDALGRCTRDSFVRGLSFARSGGDWAECFA 3k54 A 1.94 BS01 1N1 A 1 A428 K430 E445 I472 T474 M477 A478 G480 L528 A37 K39 E47 I74 T76 M79 A80 G82 L130 D521 A523 R525 N526 D539 F559 D123 A125 R127 N128 D141 F144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=1.4nM, IC50=3.0nM Q06187 20052711 1 YGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 3k5c A 2.12 BS01 0BI A 1 G11 Q12 D32 G34 Y71 T72 Q73 F108 I110 I126 Y198 D228 G230 T231 T232 R235 G14 Q15 D35 G37 Y74 T75 Q76 F111 I113 I129 Y190 D220 G222 T223 T224 R227 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=17nM remove_due_to_license_issue IC50=20nM P56817 19963375 387 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3k5d A 2.9 BS01 XLI A 1 G11 Q12 D32 G34 Y71 T72 Q73 F108 D228 G230 T231 T232 G14 Q15 D35 G37 Y74 T75 Q76 F111 D218 G220 T221 T222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D218 T221 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=53nM P56817 20172717 393 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3k5f A 2.25 BS01 AYH A 1 G13 D32 G34 Y71 T72 Q73 F108 Y198 D228 G230 T232 G16 D35 G37 Y74 T75 Q76 F111 Y190 D220 G222 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=3.7uM remove_due_to_license_issue IC50=3700nM P56817 20172717 387 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVRTAAVEGPFVTLDMEDCGYN 3k5g A 2.0 BS01 BJC A 1 G11 Q12 G13 D32 G34 S35 Y71 T72 Q73 F108 I126 Y198 D228 G230 T231 T232 G14 Q15 G16 D35 G37 S38 Y74 T75 Q76 F111 I129 Y190 D220 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.0025uM remove_due_to_license_issue P56817 20172717 387 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3k5i B 2.0 BS03 AIR B 1 G13 Q14 L15 E73 R271 K345 R352 G13 Q14 L15 E73 R266 K340 R347 E254 E267 N274 S275 K353 E249 E262 N269 S270 K348 4.1.1.21 0004638,0005524,0006189,0046872 remove_due_to_license_issue A1CII2 20050602 402 MWNSRKVGVLGGGQLGRMLVESANRLNIQVNVLDADNSPAKQISAHDGHVTGSFKEREAVRQLAKTCDVVTAEIEHVDTYALEEVASEVKIEPSWQAIRTIQNKFNQKEHLRKYGIPMAEHRELVENTPAELAKVGEQLGYPLMLKSKTRGNFRVNSQDDIPEALEALKDRPLYAEKWAYFKMELAVIVVKTKDEVLSYPTVETVQEDSICKLVYAPARNVSDAINQKAQELARKAVAAFDGKGVFGVEMFLLEDDSIMLCEIASRIHNSGHYTIEGCALSQFDAHLRAILDLPIPAQSLEIRQPSIMLNIIGGAAPDTHLQAAECALSIPNASIHLYSKGAAKPGRKMGHITVTAPTMHEAETHIQPLIDVVDRI 3k5k A 1.7 BS06 DXQ A 1 D1074 A1077 D1078 D1083 L1086 D1088 F1152 Y1154 R1157 F1158 D158 A161 D162 D167 L170 D172 F234 Y236 R239 F240 Y1067 Y1154 Y151 Y236 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 Kd=23nM remove_due_to_license_issue IC50=15nM, Ki=2.6nM, Kd=23nM Q96KQ7 19891491 2000 RTEKIICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLDNKEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKSKYFTCQCGSEKCKHSAEAIALEQSRLA 3k5q A 2.2 BS01 rna B 0 K201 C204 E208 N244 Y245 R288 Q291 Q322 N323 H326 K360 Y361 R364 Y413 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S554 K557 K34 C37 E41 N77 Y78 R121 Q124 Q155 N156 H159 K193 Y194 R197 Y246 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 Q337 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 19901328 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3k5u A 2.35 BS01 PFQ A 1 L139 G140 V147 A213 G216 T217 L263 L14 G15 V22 A88 G91 T92 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=309nM remove_due_to_license_issue IC50=309nM O14965 20039358 1001 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPSNCQ 3k5v A 1.74 BS01 STJ A 1 A356 L359 L360 L448 A452 E481 C483 P484 I521 L529 A113 L116 L117 L205 A209 E238 C240 P241 I278 L286 D382 A384 R386 N387 D400 P421 D139 A141 R143 N144 D157 P178 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 20072125 1 AMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKEL 3k5x A 1.4 BS01 P8D A 1 H20 D22 Y68 E123 H150 H191 H212 R223 F248 D320 G323 T324 H20 D22 Y68 E123 H150 H191 H212 R223 F248 D320 G323 T324 H20 D22 E123 H150 H191 H212 D320 H20 D22 E123 H150 H191 H212 D320 ? 0006508,0046872,0070573 Ki=390nM remove_due_to_license_issue Q93J45 20000809 401 MTSLEKARELLREFPVVDGHNDLPWALREQVRYDLDARDIAADQSAHLHTDLARLRSGGVGAQYWSVYVRSDLPGAVTATLEQIDCVRRLIDRHPGELRAALTAADMEAARAEGRIASLMGAEGGHSIDNSLATLRALYALGVRYMTLTHNDNNAWADSATDEPGVGGLSAFGREVVREMNREGMLVDLSHVAATTMRDALDTSTAPVIFSHSSSRAVCDHPRNIPDDVLERLSANGGMAMVTFVPKFVLQAAVDWTAEADDNMRAHGFHHLDSSPEAMKVHAAFEERVPRPVATVSTVADHLDHMREVAGVDHLGIGGDYDGTPFTPDGLGDVSGYPNLIAELLDRGWSQSDLAKLTWKNAVRVLDAAEDVSRGLRAARGPSNATIEQLD 3k5y A 2.3 BS01 rna B 0 K201 F242 N244 Y245 R288 Q291 H326 K360 Y361 R364 Y413 N415 Y416 Q419 K450 S453 H454 E457 F498 N500 Y501 Q504 S554 K557 K34 F75 N77 Y78 R121 Q124 H159 K193 Y194 R197 Y246 N248 Y249 Q252 K283 S286 H287 E290 F331 N333 Y334 Q337 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 19901328 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3k5z A 2.4 BS01 rna B 0 K201 N244 Y245 R288 Q291 N323 H326 K360 Y361 R364 Y413 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 K557 K28 N71 Y72 R115 Q118 N150 H153 K187 Y188 R191 Y240 N242 Y243 Q246 K277 S280 H281 E284 N327 Y328 Q331 K384 ? 0003723 remove_due_to_license_issue Q09312 19901328 1 ~ 9 LPTWSLRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3k61 A 2.21 BS01 rna B 0 K201 N244 Y245 K284 R288 Q291 Q322 N323 H326 K360 Y361 R364 Y413 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S554 K557 K27 N70 Y71 K110 R114 Q117 Q148 N149 H152 K186 Y187 R190 Y239 N241 Y242 Q245 K276 S279 H280 E283 N326 Y327 Q330 S380 K383 ? 0003723 remove_due_to_license_issue Q09312 19901328 1 ~ 9 LPTWSRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3k62 A 1.9 BS01 rna B 0 K201 F242 N244 Y245 Q248 F285 R288 Q291 H326 K360 Y361 R364 Y413 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S554 K557 K34 F75 N77 Y78 Q81 F118 R121 Q124 H159 K193 Y194 R197 Y246 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 Q337 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 19901328 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3k64 A 2.0 BS01 rna B 0 K201 F242 N244 Y245 Q248 R288 Q291 H326 K360 Y361 R364 Y413 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S554 K557 K34 F75 N77 Y78 Q81 R121 Q124 H159 K193 Y194 R197 Y246 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 Q337 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 19901328 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3k7f A 1.95 BS01 F2C A 1 M191 F192 S193 S217 D237 I238 G239 S241 G268 C269 V270 F381 M495 M160 F161 S162 S186 D206 I207 G208 S210 G237 C238 V239 F350 M464 K142 S217 S218 T236 I238 G239 G240 S241 F244 K111 S186 S187 T205 I207 G208 G209 S210 F213 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue IC50=100nM, Ki=10.3nM P97612 19924997 1 TGRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTP 3k83 A 2.251 BS01 F27 A 1 M191 F192 S193 S217 D237 I238 G239 S241 G268 C269 V270 L278 T488 M159 F160 S161 S185 D205 I206 G207 S209 G236 C237 V238 L246 T456 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 Ki=22nM remove_due_to_license_issue Ki=22nM, IC50=6nM P97612 19924997 1 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQP 3k84 A 2.25 BS01 K84 A 1 M191 F192 S193 S217 T236 I238 G239 S241 T377 T488 W531 M159 F160 S161 S185 T204 I206 G207 S209 T345 T456 W499 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue Ki=3nM P97612 19924997 1 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQP 3k8c A 2.1 BS01 RES A 1 D10 H11 C69 G70 S71 G74 D10 H11 C69 G70 S71 G74 D10 C69 S71 H102 H138 D10 C69 S71 H102 H138 5.3.1.6 0005975,0016853,0042802 remove_due_to_license_issue Q4CQE2 21205211 160 MTRRVAIGTDHPAFAIHENLILYVKEAGDEFVPVYCGPKTAESVDYPDFASRVAEMVARKEVEFGVLACGSGIGMSIAANKVPGVRAALCHDHYTAAMSRIHNDANIVCVGERTTGVEVIREIIITFLQTPFSGEERHVRRIEKIRAIEASH 3k8c A 2.1 BS02 RES B 1 H102 N103 R137 R141 H102 N103 R137 R141 D10 C69 S71 H102 H138 D10 C69 S71 H102 H138 5.3.1.6 0005975,0016853,0042802 remove_due_to_license_issue Q4CQE2 21205211 160 MTRRVAIGTDHPAFAIHENLILYVKEAGDEFVPVYCGPKTAESVDYPDFASRVAEMVARKEVEFGVLACGSGIGMSIAANKVPGVRAALCHDHYTAAMSRIHNDANIVCVGERTTGVEVIREIIITFLQTPFSGEERHVRRIEKIRAIEASH 3k8c B 2.1 BS01 RES A 1 H102 N103 R137 R141 H101 N102 R136 R140 D10 C69 S71 H102 H138 D9 C68 S70 H101 H137 5.3.1.6 0005975,0016853,0042802 remove_due_to_license_issue Q4CQE2 21205211 160 TRRVAIGTDHPAFAIHENLILYVKEAGDEFVPVYCGPKTAESVDYPDFASRVAEMVARKEVEFGVLACGSGIGMSIAANKVPGVRAALCHDHYTAAMSRIHNDANIVCVGERTTGVEVIREIIITFLQTPFSGEERHVRRIEKIRAIEASH 3k8c B 2.1 BS02 RES B 1 D10 H11 C69 G70 S71 G74 R113 D9 H10 C68 G69 S70 G73 R112 D10 C69 S71 H102 H138 D9 C68 S70 H101 H137 5.3.1.6 0005975,0016853,0042802 remove_due_to_license_issue Q4CQE2 21205211 160 TRRVAIGTDHPAFAIHENLILYVKEAGDEFVPVYCGPKTAESVDYPDFASRVAEMVARKEVEFGVLACGSGIGMSIAANKVPGVRAALCHDHYTAAMSRIHNDANIVCVGERTTGVEVIREIIITFLQTPFSGEERHVRRIEKIRAIEASH 3k8o E 2.4 BS01 229 E 1 A116 A117 G118 F200 E201 G218 M219 N243 H257 A114 A115 G116 F198 E199 G216 M217 N241 H255 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S31 H62 H84 Y86 E87 A114 M217 S218 N241 V243 H255 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=780nM, Kd=0.0086nM P00491 9006 NGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLP 3k8o Y 2.4 BS01 229 Y 1 A116 A117 G118 F200 E201 M219 N243 H257 A114 A115 G116 F198 E199 M217 N241 H255 S33 H64 H86 Y88 E89 A116 M219 S220 N243 H257 S31 H62 H84 Y86 E87 A114 M217 S218 N241 H255 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=780nM, Kd=0.0086nM P00491 9001 NGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLP 3k8q A 2.5 BS01 22A A 1 A116 A117 G118 F200 E201 V217 M219 N243 A116 A117 G118 F200 E201 V217 M219 N243 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=0.11nM P00491 290 MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPD 3k97 A 1.95 BS01 4CD A 1 N51 A55 D93 I96 G97 M98 F138 T184 N36 A40 D78 I81 G82 M83 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=10nM remove_due_to_license_issue P07900 19908836 901 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3k98 A 2.4 BS01 1RC A 1 N51 A55 K58 D93 I96 G97 M98 L107 T184 N43 A47 K50 D85 I88 G89 M90 L99 T172 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki<1nM remove_due_to_license_issue P07900 19908836 901 DQPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEAADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKELE 3k99 A 2.1 BS01 PFT A 1 N51 A55 D93 I96 M98 T184 N43 A47 D85 I88 M90 T176 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=60nM remove_due_to_license_issue P07900 19908836 901 DQPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKEL 3k9x B 1.9 BS01 MBM B 1 T98 Y99 E147 F174 A190 C191 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 T84 Y85 E135 F162 A180 C181 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=4nM remove_due_to_license_issue IC50=4nM P00742 19896847 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTRGLP 3ka2 A 1.4 BS01 2NC A 1 G27 D29 G48 G49 I50 P81 V82 D129 G131 A132 D133 D134 I151 G152 I154 P185 G27 D29 G48 G49 I50 P81 V82 D129 G131 A132 D133 D134 I151 G152 I154 P185 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.24uM remove_due_to_license_issue P03369 22158985 204 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIAGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNFCGGGGPQITLWKRPLVTIRIGGQLKEALLDTGADDTVIEELNLPGCWKPKLIGGIGGFIKVRQYDQIPVEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3kab A 2.19 BS01 4BL A 1 L61 C113 M130 Q131 F134 S154 L43 C95 M112 Q113 F116 S136 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=630uM remove_due_to_license_issue IC50=630000nM Q13526 19969456 166 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kac A 2.0 BS01 4BX A 1 H59 K63 R69 C113 F134 S154 H157 H9 K13 R19 C63 F84 S104 H107 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 ic50=740uM remove_due_to_license_issue IC50=>10000nM Q13526 19969456 1 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kad A 1.95 BS01 4C0 A 1 H59 L61 K63 R69 C113 S115 L122 F134 S154 H157 H41 L43 K45 R51 C95 S97 L104 F116 S136 H139 H59 C113 A131 S154 H157 H41 C95 A113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=7.5uM remove_due_to_license_issue IC50=7500nM Q13526 19969456 164 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMAKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kaf A 2.3 BS01 4D9 A 1 H59 K63 C113 S114 L122 M130 F134 S154 H157 H41 K45 C95 S96 L104 M112 F116 S136 H139 H59 C113 A131 S154 H157 H41 C95 A113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=0.83uM remove_due_to_license_issue IC50=830nM, Kd=10000nM Q13526 19969456 164 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMAKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kag A 1.9 BS01 4D7 A 1 H59 L61 K63 C113 S114 F134 S154 H157 H41 L43 K45 C95 S96 F116 S136 H139 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=6.6uM remove_due_to_license_issue IC50=6600nM Q13526 19969456 164 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kah A 2.3 BS01 4DH A 1 H59 L61 K63 C113 S114 S115 Q131 F134 S154 H41 L43 K45 C95 S96 S97 Q113 F116 S136 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=0.26uM remove_due_to_license_issue Q13526 19969456 165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kai A 1.9 BS01 4FI A 1 H59 C113 S114 S115 Q131 F134 S154 H41 C95 S96 S97 Q113 F116 S136 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=3.9uM remove_due_to_license_issue IC50=4200nM Q13526 19969456 165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kb3 A 1.95 BS01 A8S A 1 K64 A93 S96 F112 H119 Y124 F165 V169 K52 A81 S84 F100 H107 Y112 F153 V157 ? 0004864,0005515,0005634,0005737,0005886,0009738,0010427,0038023,0042802,0042803,0062049 remove_due_to_license_issue O80992 189 SEQKTLEPVIKTYHQFEPDPTTCTSLITQRIHAPASVVWPLIRRFDNPERYKHFVKRCRLISGDGDVGSVREVTVISGLPASTSTERLEFVDDDHRVLSFRVVGGEHRLKNYKSVTSVNEFLNQDSGKVYTVVLESYTVDIPEGNTEEDTKMFVDTVVKLNLQKLGVAATSAPMHD 3kb7 A 2.5 BS01 071 A 1 L59 C67 A80 K82 C133 R136 S137 E140 F183 D194 L21 C29 A42 K44 C95 R98 S99 E102 F145 D156 D176 K178 G180 N181 D194 T214 D138 K140 G142 N143 D156 T176 2.7.11.21 0004672,0005524,0006468 ic50=0.007uM remove_due_to_license_issue IC50=7nM P53350 20397705 1 EIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKTLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 3kba A 2.0 BS01 WOW A 1 L715 L718 N719 L721 M759 V760 F778 F794 M801 L887 Y890 C891 F905 L29 L32 N33 L35 M73 V74 F92 F106 M113 L198 Y201 C202 F216 ? ic50=16nM remove_due_to_license_issue IC50=16nM, EC50=25nM P06401 19926282 1 QLIPPLINLLMSIEPDVIYAGHDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKEFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILAGMVKPLLFHK 3kbz A 2.45 BS01 2T4 A 1 V17 E20 G21 A24 G26 T27 G28 E29 L30 T31 K112 Y113 V9 E12 G13 A16 G18 T19 G20 E21 L22 T23 K96 Y97 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=124nM remove_due_to_license_issue IC50=124nM P09467 20045638 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3kbz C 2.45 BS01 2T4 C 1 V17 G21 A24 G26 T27 G28 E29 L30 T31 K112 Y113 M177 V9 G13 A16 G18 T19 G20 E21 L22 T23 K95 Y96 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=124nM remove_due_to_license_issue IC50=124nM P09467 20045638 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3kc0 A 2.8 BS01 2T5 A 1 V17 G21 A24 G26 T27 G28 E29 L30 T31 K112 Y113 M177 V9 G13 A16 G18 T19 G20 E21 L22 T23 K96 Y97 M161 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=12nM P09467 20045638 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3kc0 C 2.8 BS01 2T5 C 1 V17 G21 A24 G26 T27 G28 L30 T31 K112 Y113 M177 V9 G13 A16 G18 T19 G20 L22 T23 K95 Y96 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 remove_due_to_license_issue IC50=12nM P09467 20045638 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3kc1 A 2.25 BS01 2T6 A 1 V17 G21 A24 G26 T27 G28 E29 L30 K112 Y113 M177 V9 G13 A16 G18 T19 G20 E21 L22 K96 Y97 M161 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=1nM remove_due_to_license_issue IC50=1nM P09467 20045638 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3kc1 C 2.25 BS01 2T6 C 1 V17 G21 A24 G26 T27 G28 E29 L30 K112 Y113 M177 V9 G13 A16 G18 T19 G20 E21 L22 K95 Y96 M160 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=1nM remove_due_to_license_issue IC50=1nM P09467 20045638 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 3kc3 A 2.9 BS01 MK2 A 1 L70 V78 K93 L141 D142 L193 T206 D207 L28 V36 K51 L99 D100 L148 T161 D162 D186 K188 E190 N191 D207 D141 K143 E145 N146 D162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1300nM P49137 19919896 500 FPQFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHISPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKE 3kce A 1.9 BS01 4BY A 1 H59 K63 C113 Q131 F134 S154 H157 H42 K46 C96 Q114 F117 S137 H140 H59 C113 Q131 S154 H157 H42 C96 Q114 S137 H140 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 remove_due_to_license_issue Kd=200000nM, IC50=16000nM Q13526 19969456 165 KLPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3kcf A 2.8 BS01 JZO A 1 I211 A230 K232 L260 S280 Y282 H283 K337 L340 D351 I41 A60 K62 L90 S110 Y112 H113 K167 L170 D181 D333 K335 N338 D351 T375 D163 K165 N168 D181 T203 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=3690nM, Ki=35nM P36897 19914068 1 ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDINHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG 3kck A 2.2 BS01 3KC A 1 L855 V863 A880 E898 V911 M929 E930 Y931 L932 L983 G993 D994 L14 V20 A37 E55 V68 M86 E87 Y88 L89 L140 G150 D151 M865 D976 A978 R980 N981 D994 S1016 M22 D133 A135 R137 N138 D151 S173 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.0008uM remove_due_to_license_issue O60674 19945871 1 TQFEERHLKFLQQLGKGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 3kdb A 1.66 BS01 006 B 1 D25 G27 A28 D29 V32 I47 G48 I50 P81 V82 D25 G27 A28 D29 V32 I47 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 20028396 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kdb B 1.66 BS01 006 B 1 D25 G27 A28 D29 D30 I47 G49 I50 I84 D25 G27 A28 D29 D30 I47 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.14nM remove_due_to_license_issue P03367 20028396 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kdc A 2.2 BS01 JZP A 1 D25 G27 A28 D29 D30 V32 G48 I50 P81 V82 D25 G27 A28 D29 D30 V32 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.52nM remove_due_to_license_issue P03367 20028396 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kdc B 2.2 BS01 JZP A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 20028396 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kdd A 1.8 BS01 JZQ A 1 R8 D25 G27 A28 D29 G49 I50 I84 R8 D25 G27 A28 D29 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=3.45nM remove_due_to_license_issue P03367 20028396 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kdd B 1.8 BS01 JZQ A 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 V82 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 20028396 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kde C 1.74 BS01 dna A 0 M1 I17 H18 K21 Q42 R65 R66 R67 M1 I17 H18 K21 Q42 R63 R64 R65 2.7.7.- remove_due_to_license_issue Q7M3K2 20010837 1 ~ 10 MKYCKFCCKAVTGVKLIHVPKCAIKRKLWEQSLGCSLGENSQICDTHFNDSQWKAAKGQTFKRRRLNADAVPSK 3kde C 1.74 BS02 dna B 0 M1 Y3 K5 N40 K54 F63 K64 R65 M1 Y3 K5 N40 K54 F61 K62 R63 2.7.7.- remove_due_to_license_issue Q7M3K2 20010837 11 ~ 20 MKYCKFCCKAVTGVKLIHVPKCAIKRKLWEQSLGCSLGENSQICDTHFNDSQWKAAKGQTFKRRRLNADAVPSK 3kdm H 1.5 BS01 TES H 1 W47 Y59 D99 Y105 Y107 W47 Y59 D99 Y105 Y107 Kd=0.1uM remove_due_to_license_issue 21360611 226 QVQLVESGGGLVQPGGSLRLSCAASGFTFSSYAMSWVRQAPGKGLEWVSAISGSGGSTYYADSVKGRFTISRDNSKNTLYLQMNSLRAEDTAVYYCARDPGLWDYYYGMDVWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSSVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKAEPK 3kdm L 1.5 BS01 TES H 1 P99 Y100 P97 Y98 remove_due_to_license_issue 21360611 226 ALTQPASVSGSPGQSITISCTGTSSDVGGYNYVSWYQQHPGKAPKLMIYGVTNRPSGVSNRFSGSKSGNTASLTISGLQAGDEADYYCSSYTSTRTPYVFGTGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 3kdt A 2.7 BS01 7HA A 1 C275 C276 S280 Y314 I317 F318 V332 M355 H440 C72 C73 S77 Y111 I114 F115 V129 M152 H237 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=10nM, IC50=260nM Q07869 20218621 501 SETADLKSLAKRIYEAYLKNFNMNKVKARVILSGKASNNPPFVIHDMETLCMAEKTLVAIQNKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANLDLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFDFAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDIFLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDM 3kdu A 2.07 BS01 NKS A 1 F273 C276 S280 Y314 L321 M330 V332 I354 M355 H440 F70 C73 S77 Y111 L118 M127 V129 I151 M152 H237 ? 0003677,0004879,0005634,0006355 ic50=347nM remove_due_to_license_issue IC50=347nM, EC50=8nM Q07869 20218621 501 SETADLKSLAKRIYEAYLKNFNMNKVKARVILSGKASNNPPFVIHDMETLCMAEKTLVAIQNKEAEVRIFHCCQCTSVETVTELTEFAKAIPGFANLDLNDQVTLLKYGVYEAIFAMLSSVMNKDGMLVAYGNGFITREFLKSLRKPFCDIMEPKFDFAMKFNALELDDSDISLFVAAIICCGDRPGLLNVGHIEKMQEGIVHVLRLHLQSNHPDDIFLFPKLLQKMADLRQLVTEHAQLVQIIKKTESDAALHPLLQEIYRDM 3kec A 2.05 BS06 3KE A 1 K140 N215 F217 L218 V219 H222 L239 F241 P242 I243 Y244 T245 T247 K249 F252 K37 N112 F114 L115 V116 H119 L136 F138 P139 I140 Y141 T142 T144 K146 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=58nM remove_due_to_license_issue IC50=130nM P45452 20005097 271 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGD 3ked A 2.3 BS02 DAB A 1 E121 M260 A262 M263 E264 H297 E298 E320 Y381 E117 M256 A258 M259 E260 H293 E294 E316 Y377 E264 H297 E298 H301 E320 N373 Y381 E260 H293 E294 H297 E316 N369 Y377 3.4.11.2 0004177,0005515,0005886,0006508,0008237,0008270,0042802,0046872 ic50=3.6mM remove_due_to_license_issue P04825 22025387 880 PQAKYRHDYRAPDYQITDIDLTFDLDAQKTVVTAVSQAVRHGASDAPLRLNGEDLKLVSVHINDEPWTAWKEEEGALVISNLPERFTLKIINEISPAANTALEGLYQSGDALCTQCEAEGFRHITYYLDRPDVLARFTTKIIADKIKYPFLLSNGNRVAQGELENGRHWVQWQDPFPKPCYLFALVAGDFDVLRDTFTTRSGREVALELYVDRGNLDRAPWAMTSLKNSMKWDEERFGLEYDLDIYMIVAVDFFNMGAMENKGLNIFNSKYVLARTDTATDKDYLDIERVIGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSSDLGSRAVNRINNVRTMRGLQFAEDASPMAHPIRPDMVIEMNNFYTLTVYEKGAEVIRMIHTLLGEENFQKGMQLYFERHDGSAATCDDFVQAMEDASNVDLSHFRRWYSQSGTPIVTVKDDYNPETEQYTLTISQRTPATPDQAEKQPLHIPFAIELYDNEGKVIPLQKGGHPVNSVLNVTQAEQTFVFDNVYFQPVPALLCEFSAPVKLEYKWSDQQLTFLMRHARNDFSRWDAAQSLLATYIKLNVARHQQGQPLSLPVHVADAFRAVLLDEKIDPALAAEILTLPSVNEMAELFDIIDPIAIAEVREALTRTLATELADELLAIYNANYQSEYRVEHEDIAKRTLRNACLRFLAFGETHLADVLVSKQFHEANNMTDALAALSAAVAAQLPCRDALMQEYDDKWHQNGLVMDKWFILQATSPAANVLETVRGLLQHRSFTMSNPNRIRSLIGAFAGSNPAAFHAEDGSGYLFLVEMLTDLNSRNPQVASRLIEPLIRLKRYDAKRQEKMRAALEQLKGLENLSGDLYEKITKALA 3kej A 2.3 BS06 3EJ A 1 F217 L218 H222 L239 F241 I243 Y244 T245 Y246 T247 K249 F114 L115 H119 L136 F138 I140 Y141 T142 Y143 T144 K146 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=75.9nM remove_due_to_license_issue Ki=76nM P45452 20005097 801 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLY 3kek A 1.97 BS06 3EK A 1 K140 F217 L218 V219 H222 A238 L239 F241 I243 Y244 T245 Y246 T247 F252 P255 K37 F114 L115 V116 H119 A135 L136 F138 I140 Y141 T142 Y143 T144 F149 P152 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=4.4nM remove_due_to_license_issue P45452 20005097 801 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYG 3ken A 2.5 BS02 ZZD A 1 E116 G117 E118 R119 A133 P137 Y211 L214 E215 E99 G100 E101 R102 A116 P120 Y194 L197 E198 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=1000nM, EC50=1720nM, Ki=143.8nM P52732 20299460 370 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 3kf4 A 1.9 BS01 B90 A 1 L248 Y253 A269 V270 K271 E286 M290 I313 T315 F317 M318 T319 G321 L370 A380 D381 L20 Y25 A41 V42 K43 E53 M57 I80 T82 F84 M85 T86 G88 L137 A147 D148 D363 A365 R367 N368 D381 P402 D130 A132 R134 N135 D148 P169 2.7.10.2 0004672,0004713,0005524,0006468 ic50<0.5nM remove_due_to_license_issue P00520 19895503 1 SPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELGKRG 3kf7 A 2.0 BS01 L9G A 1 V30 V38 A51 K53 I84 L104 V105 T106 M109 G110 A111 L167 V26 V34 A47 K49 I80 L100 V101 T102 M105 G106 A107 L163 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=40nM remove_due_to_license_issue Q16539 19969459 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3kfa A 1.22 BS01 B91 A 1 L248 A269 V270 E282 E286 V289 M290 I293 I313 T315 F317 M318 G321 F359 H361 L370 A380 D381 F382 L21 A42 V43 E55 E59 V62 M63 I66 I86 T88 F90 M91 G94 F132 H134 L143 A153 D154 F155 D363 A365 R367 N368 D381 P402 D136 A138 R140 N141 D154 P175 2.7.10.2 0004672,0004713,0005524,0006468 ic50=25nM remove_due_to_license_issue P00520 19895503 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG 3kfc A 2.4 BS01 61X A 1 F271 L274 A275 S278 M312 R319 F329 L330 H435 W457 F46 L49 A50 S53 M87 R94 F104 L105 H210 W232 ? 0003677,0004879,0006629 ic50=2.8nM remove_due_to_license_issue IC50=40nM P55055 19932617 1 LTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWD 3kfn A 1.77 BS01 3TL A 1 R8 D25 G27 A28 D29 G48 G49 F53 P81 V82 I84 R8 D25 G27 A28 D29 G48 G49 F53 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 20659109 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kfn B 1.77 BS01 3TL A 1 D25 G27 A28 D29 G48 G49 F53 P81 V82 D25 G27 A28 D29 G48 G49 F53 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12499 20659109 200 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3kga A 2.55 BS02 LX9 A 1 L70 Q80 I81 F82 K89 F90 A91 K93 M138 C140 L141 D207 L24 Q34 I35 F36 K43 F44 A45 K47 M92 C94 L95 D161 D186 K188 N191 D207 D140 K142 N145 D161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=61nM P49137 20060294 365 HVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTGEKYDKSCDMWSLGVIMYILLCGYPPFYSPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR 3kgp A 2.35 BS01 4AZ A 1 S190 C191 Q192 W215 G226 S187 C188 Q189 W212 G223 H57 D102 Q192 G193 D194 S195 G196 H42 D91 Q189 G190 D191 S192 G193 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 4069 IIGGEFTTIENQPWFAAIYRRHVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 3kgt A 1.95 BS01 GEN A 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.1uM remove_due_to_license_issue P02766 20211733 3071 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3kgt B 1.95 BS01 GEN B 1 K15 L17 A108 L110 S117 K6 L8 A95 L97 S104 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.1uM remove_due_to_license_issue P02766 20211733 3071 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANRRYTIAALLSPYSYSTTAVVTNP 3kgu A 1.85 BS01 GEN A 1 K15 L17 K6 L8 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=1.2uM remove_due_to_license_issue P02766 20211733 3071 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3kgu B 1.85 BS01 GEN B 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=1.2uM remove_due_to_license_issue P02766 20211733 3071 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3khc B 2.2 BS01 dna C 0 T51 G53 Y55 M57 W69 G75 Y76 K127 S129 H131 R161 R210 T43 G45 Y47 M49 W61 G67 Y68 K119 S121 H123 R153 R202 1.14.11.33 0005515,0005737,0005829,0006281,0006307,0008198,0035513,0035515,0035516,0042245,0046872,0051213,0070989,0072702 remove_due_to_license_issue P05050 20084272 2 ~ 9 EPWQEPLAAGAVILRRFAFNAAEQLIRDINDVASQSPFRQMVTPGGYTMSVAMTNCGHLGWTTHRQGYLYSPIDPQTNKPWPAMPQSFHNLCQRAATAAGYPDFQPDACLINRYAPGAKLSLHQDKAEPDLRAPIVSVSLGLPAIFQFGGLKRNDPLKRLLLEHGDVVVWGGESRLFYHGIQPLKAGFHPLTIDCRYNLTFRQAGKK 3khj A 2.8 BS02 C64 B 1 S354 G357 Y358 S277 G280 Y281 1.1.1.205 0003824,0003938,0006164,0016491 remove_due_to_license_issue Q5CPK7 20052976 901 TKNIGKGLTFEDILLVPNYSEVLPREVSLETKLTKNVSLKIPLISSAMDTVTEHLMAVGMARLGGIGIIHKNMDMESQVNEVLKVKNSGGLRVGAAIGVNEIERAKLLVEAGVDVIVLDSAHGHSLNIIRTLKEIKSKMNIDVIVGNVVTEEATKELIENGADGIKVGIGPGSICTTRIVAGVGVPQITAIEKCSSVASKFGIPIIADGGIRYSGDIGKALAVGASSVMIGSILAGTEESPGEKELIGDTVYKYYGRVKYKGEMEGVVYQLVGGLRSCMGYLGSASIEELWKKSSYVEITTS 3khj B 2.8 BS02 C64 B 1 A165 H166 M302 G303 M308 E329 A121 H122 M258 G259 M264 E269 1.1.1.205 0003824,0003938,0006164,0016491 remove_due_to_license_issue Q5CPK7 20052976 901 TKNIGKGLTFEDILLVPNYSEVLPREVSLETKLTKNVSLKIPLISSAMDTVTEHLMAVGMARLGGIGIIHKNMDMESQVNEVLKVKNSGGLRVGAAIGVNEIERAKLLVEAGVDVIVLDSAHGHSLNIIRTLKEIKSKMNIDVIVGNVVTEEATKELIENGADGIKVGIGPGSICTTRIVAGVGVPQITAIEKCSSVASKFGIPIIADGGIRYSGDIGKALAVGASSVMIGSILAGTEESPGEKELIGDTVYKYYRGMGSVGAMKMVPEGIEGRVKYKGEMEGVVYQLVGGLRSCMGYLGSASIEELWKKSSYVEITT 3khv A 2.35 BS01 4AL A 1 D189 S190 C191 D185 S186 C187 H57 D102 Q192 G193 D194 S195 G196 H42 D90 Q188 G189 D190 S191 G192 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 4069 IIGGEFTTIENQPWFAAIYRRSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSAAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 3kid U 2.71 BS01 2BS U 1 S190 Q192 S195 V213 G219 S185 Q187 S190 V208 G213 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 1 IIGGEFTTIENQPWFAAIYRRVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSAAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 3kig A 1.39 BS03 DA4 A 1 Q92 H94 H119 F130 L197 T198 T199 Q90 H92 H117 F128 L195 T196 T197 C64 H94 H96 E106 H119 T198 C62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=245nM remove_due_to_license_issue Ki=66nM P00918 21506176 504 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGCAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3kiv A 1.8 BS01 ACA A 1 R35 D55 W62 F64 R71 W72 R36 D55 W61 F63 R70 W71 3.4.21.- Kd=20uM remove_due_to_license_issue P08519 10026282 100 QCYHGNGQSYRGTFSTTVTGRTCQSWSSMTPHRHQRTPENYPNDGLTMNYCRNPDADTGPWCFTTDPSIRWEYCNLTRC 3kjd A 1.95 BS01 78P A 1 H428 G429 Y462 S470 Y473 H199 G200 Y233 S241 Y244 K264 A265 I289 F305 T307 S470 Y473 E558 K39 A40 I64 F80 T82 S241 Y244 E329 2.4.2.-,2.4.2.30 0003950 Kd=2.9nM remove_due_to_license_issue IC50=1.3nM, Kd=5.8nM Q9UGN5 20092359 1 TENLYFQSMDLRVQELIKLICNVQAMEEMMMEMKYNTKKAPLGKLTVAQIKAGYQSLKKIEDCIRAGQHGRALMEACNEFYTRIPHDFGLRTPPLIRTQKELSEKIQLLEALGDIEIAIKLVKSPEHPLDQHYRNLHCALRPLDHESYEFKVISQYLQSTHAPTHSDYTMTLLDLFEVEKDGEKEAFREDLHNRMLLWHGSRMSNWVGILSHGLRIAHPEAPITGYMFGKGIYFADMSSKSANYCFASRLKNTGLLLLSEVALGQCNELLEANPKAEGLLQGKHSTKGLGKMAPSSAHFVTLNGSTVPLGPASDTGILNPDGYTLNYNEYIVYNPNQVRMRYLLKVQFNF 3kjf A 2.0 BS01 B92 B 1 R64 H121 C163 R31 H88 C130 T62 S63 H121 G122 C163 R164 T29 S30 H88 G89 C130 R131 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue P42574 20580860 285 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIE 3kjf B 2.0 BS01 B92 B 1 Y204 S205 W206 R207 N208 S209 W214 Y29 S30 W31 R32 N33 S34 W39 3.4.22.56 0004197,0006508,0008234 remove_due_to_license_issue P42574 20580860 285 SGVDDDMACHKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH 3kjn A 1.8 BS01 B93 A 1 R260 H317 C360 R38 H95 C138 R258 D259 H317 G318 C360 Q361 R36 D37 H95 G96 C138 Q139 3.4.22.61 0004197,0006508,0008234 remove_due_to_license_issue Q14790 20580860 950 DKVYQMKSKPRGYCLIINNHNFAKAREKVPKLHSIRDRNGTHLDAGALTTTFEELHFEIKPHDDCTVEQIYEILKIYQLMDHSNMDCFICCILSHGDKGIIYGTDGQEAPIYELTSQFTGLKCPSLAGKPKVFFIQACQGDNYQKGIPVETD 3kjn B 1.8 BS01 B93 A 1 S411 R413 N414 P415 W420 S22 R24 N25 P26 W31 3.4.22.61 0004197,0006508,0008234 remove_due_to_license_issue Q14790 20580860 950 TRYIPDEADFLLGMATVNNCVSYRNPAEGTWYIQSLCQSLRERCPRGDDILTILTEVNYEVSNKDDKKNMGKQMPQPTFTLRKKLVFPSD 3kjo A 1.8 BS01 dna B 0 F31 K33 Y36 S38 K39 G40 T41 D42 T48 L60 F62 Y89 Y161 Y223 D224 S243 H245 H266 S270 Y271 R273 F26 K28 Y31 S33 K34 G35 T36 D37 T43 L55 F57 Y84 Y155 Y215 D216 S235 H237 H258 S262 Y263 R265 ? 0000723,0000781,0003677,0043047 remove_due_to_license_issue Q9NUX5 20080730 3 ~ 12 ATNYIYTPLNQLKGGTIVNVYGVVKFFKPPYLSKGTDYCSVVTIVDQTNVKLTCLLFSGNYEALPIIYKNGDIVRFHRLKIQVYKKETQGITSSGFASLTFEGTLGAPIIPRTSSKYFNFTTEDHKMVEALRVWASTHMSPSTLLKLCDVQPMQYFDLTCQLLGKAEVDGASFLLKVWDGTRTPFPSWRVLIQVLEGDLSHIHRLQNLTIDILVYDNHVHVARSLKVGSFLRIYSLHTKLQSMNSENQTMLSLEFHLHGGTSYGRGIRVLPESNSDVDQLKKDLESANLTA 3kjp A 1.8 BS01 dna B 0 F31 K33 Y36 S38 K39 G40 T41 D42 T48 L60 F62 Y89 Q94 Y161 Y223 D224 S243 H266 S270 Y271 R273 F26 K28 Y31 S33 K34 G35 T36 D37 T43 L55 F57 Y84 Q89 Y155 Y217 D218 S237 H260 S264 Y265 R267 ? 0000723,0000781,0003677,0043047 remove_due_to_license_issue Q9NUX5 20080730 2 ~ 12 ATNYIYTPLNQLKGGTIVNVYGVVKFFKPPYLSKGTDYCSVVTIVDQTNVKLTCLLFSGNYEALPIIYKNGDIVRFHRLKIQVYKKETQGITSSGFASLTFEGTLGAPIIPRTSSKYFNFTTEDHKMVEALRVWASTHMSPSTLLKLCDVQPMQYFDLTCQLLGKAEVDGASFLLKVWDGTRTPFPSWRVLIQDLVLEGDLSHIHRLQNLTIDILVYDNHVHVARSLKVGSFLRIYSLHTKLQSMNSENQTMLSLEFHLHGGTSYGRGIRVLPESNSDVDQLKKDLESANLTA 3kjq A 1.8 BS01 B94 A 1 R258 R260 H317 C360 R36 R38 H95 C138 R258 D259 H317 G318 C360 Q361 R36 D37 H95 G96 C138 Q139 3.4.22.61 0004197,0006508,0008234 Ki=1.32uM remove_due_to_license_issue Q14790 20580860 480 DKVYQMKSKPRGYCLIINNHNFAKAREKVPKLHSIRDRNGTHLDAGALTTTFEELHFEIKPHDDCTVEQIYEILKIYQLMDHSNMDCFICCILSHGDKGIIYGTDGQEAPIYELTSQFTGLKCPSLAGKPKVFFIQACQGDNYQKGIPVETD 3kjq A 1.8 BS02 B94 A 2 Y334 T337 S338 Y112 T115 S116 R258 D259 H317 G318 C360 Q361 R36 D37 H95 G96 C138 Q139 3.4.22.61 0004197,0006508,0008234 Ki=1.32uM remove_due_to_license_issue Q14790 20580860 481 DKVYQMKSKPRGYCLIINNHNFAKAREKVPKLHSIRDRNGTHLDAGALTTTFEELHFEIKPHDDCTVEQIYEILKIYQLMDHSNMDCFICCILSHGDKGIIYGTDGQEAPIYELTSQFTGLKCPSLAGKPKVFFIQACQGDNYQKGIPVETD 3kjq B 1.8 BS01 B94 A 1 S411 Y412 R413 P415 S22 Y23 R24 P26 3.4.22.61 0004197,0006508,0008234 remove_due_to_license_issue Q14790 20580860 480 TRYIPDEADFLLGMATVNNCVSYRNPAEGTWYIQSLCQSLRERCPRGDDILTILTEVNYEVSNKDDKKNMGKQMPQPTFTLRKKLVFPSD 3kjq B 1.8 BS02 B94 A 2 E396 F399 T467 E7 F10 T78 3.4.22.61 0004197,0006508,0008234 remove_due_to_license_issue Q14790 20580860 481 TRYIPDEADFLLGMATVNNCVSYRNPAEGTWYIQSLCQSLRERCPRGDDILTILTEVNYEVSNKDDKKNMGKQMPQPTFTLRKKLVFPSD 3kku A 1.28 BS01 B95 A 1 C25 W26 G65 G66 L67 M68 A138 Q159 L160 D161 H162 C25 W26 G65 G66 L67 M68 A138 Q159 L160 D161 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 Ki=2uM remove_due_to_license_issue IC50=800nM, Ki=2000nM P25779 20540517 216 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 3kl6 A 1.45 BS01 443 A 1 E97 T98 F174 D189 A190 Q192 S195 V213 S214 W215 G216 G219 C220 G226 I227 Y228 E83 T84 F162 D179 A180 Q182 S185 V203 S204 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=3.5nM remove_due_to_license_issue IC50=3.5nM, Ki=1.8nM P00742 20355714 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSM 3km4 A 1.9 BS01 22X A 1 Q19 Y20 V36 D38 G40 P118 F119 L121 A122 F124 D226 G228 S230 Q16 Y17 V33 D35 G37 P115 F116 L118 A119 F121 D223 G225 S227 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P00797 19959358 400 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3km4 A 1.9 BS02 22X A 2 T18 A229 S230 Y231 F253 D254 F286 T297 H301 T15 A226 S227 Y228 F250 D251 F283 T294 H298 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P00797 19959358 341 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3km4 A 1.9 BS03 22X B 2 L117 F253 L114 F250 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P00797 19959358 341 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3km4 B 1.9 BS01 22X A 2 L117 F253 L114 F246 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P00797 19959358 341 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3km4 B 1.9 BS02 22X B 1 T18 Q19 Y20 V36 D38 G40 Y83 P118 F119 L121 A122 F124 V127 D226 G228 S230 M303 T15 Q16 Y17 V33 D35 G37 Y80 P115 F116 L118 A119 F121 V124 D219 G221 S223 M296 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P00797 19959358 400 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3km4 B 1.9 BS03 22X B 2 S230 Y231 D254 F286 T297 S223 Y224 D247 F279 T290 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM P00797 19959358 341 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3kmm A 2.8 BS01 LHL A 1 V259 A271 V272 K273 E288 T316 Y318 M319 G322 L371 D382 V29 A41 V42 K43 E58 T86 Y88 M89 G92 L141 D152 D364 R366 A368 N369 D382 A400 F402 D134 R136 A138 N139 D152 A170 F172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=0.2nM P06239 1 KPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 3kmp A 2.7 BS01 dna C 0 S70 L71 Q76 K81 S62 L63 Q68 K73 ? 0005667,0006355 remove_due_to_license_issue P70340 20147459 1 ~ 15 FTSPAVKRLLGWKQGDEEEKWAEKAVDALVKKLKKKKGAMEELEKALSCPGQPSNCVTIPRSLDGRLQVSHRKGLPHVIYCRVWRWPDLQSHHELKPLECCEFPFGSKQKEVCINPYHYKRVES 3kmp A 2.7 BS02 dna D 0 R74 K81 R66 K73 ? 0005667,0006355 remove_due_to_license_issue P70340 20147459 2 ~ 16 FTSPAVKRLLGWKQGDEEEKWAEKAVDALVKKLKKKKGAMEELEKALSCPGQPSNCVTIPRSLDGRLQVSHRKGLPHVIYCRVWRWPDLQSHHELKPLECCEFPFGSKQKEVCINPYHYKRVES 3kmp B 2.7 BS01 dna C 0 R74 H101 R65 H92 ? 0005667,0006355 remove_due_to_license_issue P70340 20147459 1 ~ 15 TSPAVKRLLGWKQGDEEEKWAEKAVDALVKKLKKKKGAMEELEKALSCPGQPSNCVTIPRSLDGRLQVSHRKGLPHVIYCRVWRWPDLQSHHELKPLECCEFPFGSKQKEVCINPYHYKRVES 3kmp B 2.7 BS02 dna D 0 L71 L75 Q76 K81 L62 L66 Q67 K72 ? 0005667,0006355 remove_due_to_license_issue P70340 20147459 2 ~ 16 TSPAVKRLLGWKQGDEEEKWAEKAVDALVKKLKKKKGAMEELEKALSCPGQPSNCVTIPRSLDGRLQVSHRKGLPHVIYCRVWRWPDLQSHHELKPLECCEFPFGSKQKEVCINPYHYKRVES 3kmx A 1.7 BS01 G00 A 1 D93 G95 Y132 Q134 D289 G291 D41 G43 Y80 Q82 D237 G239 D93 S96 N98 A100 Y132 D289 T292 D41 S44 N46 A48 Y80 D237 T240 3.4.23.46 0004190,0006508,0016020 Kd=15uM remove_due_to_license_issue Kd=15nM, IC50=200nM P56817 20043700 501 EPGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3kmy A 1.9 BS01 D8Y A 1 D93 Y132 G135 K136 F169 D289 D41 Y80 G83 K84 F117 D237 D93 S96 N98 A100 Y132 D289 T292 D41 S44 N46 A48 Y80 D237 T240 3.4.23.46 0004190,0006508,0016020 Kd=32uM remove_due_to_license_issue Kd=32nM P56817 20043700 501 EPGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3kn0 A 1.9 BS01 3TO A 1 S71 Q73 G74 D93 Y132 F169 D289 G291 T292 T293 S14 Q16 G17 D36 Y75 F109 D229 G231 T232 T233 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D229 T232 3.4.23.46 0004190,0006508,0016020 Kd~100uM remove_due_to_license_issue IC50=250nM P56817 20043700 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3koo A 2.791 BS01 24D A 1 F267 D335 W336 M339 Y383 Q384 Y466 F497 V498 L499 M503 H524 F264 D332 W333 M336 Y380 Q381 Y463 F494 V495 L496 M500 H521 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F264 H331 D332 W333 N356 N375 Y380 Y463 D493 H521 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=15nM P34913 19969453 556 RAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 3kpu A 2.4 BS02 ES1 A 1 Y35 R44 K57 F182 M258 V269 Y12 R21 K34 F159 M235 V246 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=690uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kpv A 2.4 BS02 ADE A 1 Y35 N39 R44 F182 E219 Y222 D267 Y12 N16 R21 F159 E196 Y199 D244 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=180uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kpw A 2.4 BS02 1SQ A 1 Y35 N39 Y40 K57 F182 V269 Y12 N16 Y17 K34 F159 V246 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=14uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqa A 2.25 BS01 TR9 A 1 C115 A116 L138 C115 A116 L138 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 20392080 500 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 3kqb A 2.25 BS01 LGJ A 1 E97 T98 Y99 R143 F174 D189 A190 C191 Q192 S195 W215 G216 G218 C220 G226 E83 T84 Y85 R132 F162 D179 A180 C181 Q182 S185 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.5nM remove_due_to_license_issue Ki=0.5nM P00742 20100660 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3kqc A 2.2 BS01 LGK A 1 E97 T98 Y99 R143 E146 F174 D189 A190 Q192 W215 G216 G218 C220 G226 E83 T84 Y85 R132 E135 F162 D179 A180 Q182 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=2.2nM remove_due_to_license_issue Ki=2.2nM P00742 20100660 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3kqd A 2.75 BS01 LGL A 1 K96 T98 Y99 F174 D189 A190 C191 Q192 W215 G216 G218 C220 K82 T84 Y85 F162 D179 A180 C181 Q182 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=0.4nM P00742 20100660 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3kqe A 2.35 BS01 LGM A 1 E97 T98 Y99 F174 D189 A190 C191 Q192 W215 G216 G218 C220 G226 E83 T84 Y85 F162 D179 A180 C181 Q182 W205 G206 G208 C209 G216 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=8.1nM remove_due_to_license_issue Ki=8.1nM P00742 20100660 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3kqm A 2.4 BS02 ES3 A 1 Y35 F182 Y12 F159 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=170uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqo A 2.4 BS02 ES4 A 1 Y35 N39 R44 V53 F182 V269 Y12 N16 R21 V30 F159 V246 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=140uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqp A 2.4 BS02 ES5 A 1 Y35 N39 V53 F182 Y12 N16 V30 F159 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=380uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqr A 1.5 BS01 OPE A 1 N59 Y64 Y74 E136 D138 Q148 N59 Y64 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 remove_due_to_license_issue P02743 21360619 700 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 3kqs A 2.005 BS02 AX7 A 1 Y35 N39 Y40 V53 F182 Y12 N16 Y17 V30 F159 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=6.3uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqt A 2.399 BS02 ES7 A 1 Y35 N39 Y40 V53 K57 F182 Y12 N16 Y17 V30 K34 F159 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=4.6uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqw A 2.486 BS02 ES9 A 1 Y35 R44 K57 F182 M258 Y12 R21 K34 F159 M235 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=97uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kqy A 2.2 BS02 ES0 A 1 Y35 R44 K57 F182 M258 Y12 R21 K34 F159 M235 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=15uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kr0 A 2.6 BS02 172 A 1 R44 V53 K57 F182 R21 V30 K34 F159 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 remove_due_to_license_issue P11086 20642456 1001 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kr1 A 2.3 BS02 VGD A 1 Y35 N39 R44 V53 F182 M258 Y12 N16 R21 V30 F159 M235 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=1.8uM remove_due_to_license_issue P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kr2 A 2.3 BS02 ET2 A 1 Y35 N39 Y40 R44 V53 F182 M258 Y12 N16 Y17 R21 V30 F159 M235 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=7.2uM remove_due_to_license_issue P11086 20642456 1001 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kr4 A 2.0 BS03 BES A 1 K374 M392 M396 F398 D399 N457 D459 E461 L487 T488 G489 K289 M307 M311 F313 D314 N372 D374 E376 L402 T403 G404 K386 R463 K301 R378 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=25nM remove_due_to_license_issue Q8IL11 20133789 1003 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3kr4 F 2.0 BS03 BES F 1 K374 D379 M396 F398 D399 N457 D459 E461 R463 T486 L487 G489 K281 D286 M303 F305 D306 N364 D366 E368 R370 T393 L394 G396 K386 R463 K293 R370 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=25nM remove_due_to_license_issue Q8IL11 20133789 1003 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3kr5 A 2.56 BS04 BEY A 1 K374 D379 K386 M396 F398 D399 N457 D459 E461 L487 T488 G489 A577 K289 D294 K301 M311 F313 D314 N372 D374 E376 L402 T403 G404 A492 K386 R463 K301 R378 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue Q8IL11 20133789 1003 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3kr5 F 2.56 BS04 BEY F 1 K374 D379 K386 M396 F398 D399 N457 D459 A460 E461 L487 T488 G489 L492 A577 K281 D286 K293 M303 F305 D306 N364 D366 A367 E368 L394 T395 G396 L399 A484 K386 R463 K293 R370 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue Q8IL11 20133789 1003 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3kr8 A 2.1 BS02 XAV A 1 H1031 G1032 F1035 Y1050 Y1060 F1061 A1062 S1068 Y1071 I1075 E1138 H80 G81 F84 Y99 Y109 F110 A111 S117 Y120 I124 E183 2.4.2.-,2.4.2.30 0003950 Kd=8nM remove_due_to_license_issue IC50=4nM, Kd=10nM Q9H2K2 20565110 1163 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 3krd C 2.5 BS01 FEB C 1 T301 S320 T321 Q322 S327 G347 T348 A349 T1 S20 T21 Q22 S27 G47 T48 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 20558127 300 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 3krd C 2.5 BS02 FEB J 1 D424 A425 D124 A125 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 20558127 300 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 3krd E 2.5 BS01 FEB E 1 T301 S320 T321 Q322 G347 T348 A349 T1 S20 T21 Q22 G47 T48 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 20558127 300 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 3krd H 2.5 BS01 FEB H 1 T301 S320 T321 Q322 S327 G347 T348 A349 T1 S20 T21 Q22 S27 G47 T48 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 20558127 300 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 3krj A 2.1 BS01 KRJ A 1 A614 Y665 C666 G669 D670 L785 F797 R801 A71 Y122 C123 G126 D127 L176 F188 R192 D778 A780 R782 N783 D796 N805 D169 A171 R173 N174 D187 N196 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=1.1nM remove_due_to_license_issue P07333,P11362 22039836 923 PKYQVRWKIIESYEGNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKRPPGQLSSRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQA 3krl A 2.4 BS01 KRL A 1 L588 K616 T663 Y665 C666 G669 L785 F797 L28 K56 T102 Y104 C105 G108 L155 F167 D778 A780 R782 N783 D796 N805 D148 A150 R152 N153 D166 N175 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=0.8nM remove_due_to_license_issue P07333,P11362 22039836 1 KYQVRWKIIPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKRQLSSRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQE 3krr A 1.8 BS01 DQX A 1 L855 G856 G858 V863 A880 M929 Y931 L932 P933 G935 N981 L983 G993 D994 L17 G18 G20 V25 A42 M91 Y93 L94 P95 G97 N143 L145 G155 D156 D976 A978 R980 N981 D994 S1016 D138 A140 R142 N143 D156 S178 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.48nM remove_due_to_license_issue Kd=42000nM, IC50=7.3nM O60674 20587663 1 SDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 3krw A 2.9 BS01 BA1 A 1 G198 R199 G200 G201 F202 G203 V205 A218 K220 E239 D272 L273 A321 L324 S334 D335 G167 R168 G169 G170 F171 G172 V174 A187 K189 E208 D241 L242 A290 L293 S303 D304 D317 K319 N322 D335 K344 T353 D286 K288 N291 D304 K313 T322 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue IC50=42nM P25098 20128603 690 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLAHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPREEDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHGYMSKMWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKPRSP 3krx A 3.1 BS01 BA1 A 1 G198 R199 G200 G201 F202 G203 V205 A218 K220 E239 D272 L273 A321 L324 S334 D335 G167 R168 G169 G170 F171 G172 V174 A187 K189 E208 D241 L242 A290 L293 S303 D304 D317 K319 N322 D335 K344 T353 D286 K288 N291 D304 K313 T322 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue IC50=42nM P25098 20128603 690 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLAHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPREEDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHGYMSKMWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKPRSP 3kry A 1.9 BS05 3KR A 1 L184 L185 A186 H222 E223 H226 H232 L239 F241 P242 I243 Y244 T245 L81 L82 A83 H119 E120 H123 H129 L136 F138 P139 I140 Y141 T142 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.1nM remove_due_to_license_issue P45452 20726512 1800 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYG 3ksl A 2.05 BS01 SZH B 1 K164 Y200 K111 Y147 K164 K111 2.5.1.58,2.5.1.59 0004659,0004660,0004661,0004662,0004663,0005515,0005737,0005875,0005953,0005965,0007167,0007323,0008017,0008270,0008284,0008318,0014070,0018342,0018343,0018344,0030971,0034097,0035022,0036094,0042277,0043014,0043066,0045787,0051770,0051771,0060090,0090044,1901363,1904395 remove_due_to_license_issue Q04631 19954434 438 GFLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSEKFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVWHFRRVLLRSLQKDLQEEMNYITAIIEEQPKNYQVWHHRRVLVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFRLWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRAVLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPNLLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDILNKALELCEILAKEKDTIRKEYWRYIGRSLQSKHS 3ksl B 2.05 BS02 SZH B 1 W102 H248 Y251 C254 R291 K294 Y300 W303 W82 H228 Y231 C234 R271 K274 Y280 W283 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H228 R271 K274 D277 C279 Y280 D332 D339 H342 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 19954434 438 EPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 3ksq B 2.1 BS04 Z96 B 1 Y93 C95 L96 W106 D297 C299 Y300 D359 Y361 H362 Y73 C75 L76 W86 D277 C279 Y280 D339 Y341 H342 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H228 R271 K274 D277 C279 Y280 D332 D339 H342 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=0.38nM remove_due_to_license_issue Q02293 20056542 439 EPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 3kv2 A 1.55 BS03 NNH A 1 D124 H126 D128 S137 H141 D183 T246 D119 H121 D123 S132 H136 D178 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=47.51nM remove_due_to_license_issue Kd=47nM, IC50=1360nM P05089 20153713 901 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 3kvw A 2.28 BS01 IRB A 1 I155 A176 K178 F228 L230 L231 S232 I294 D295 I100 A121 K123 F173 L175 L176 S177 I239 D240 D275 K277 N280 D295 S312 D220 K222 N225 D240 S257 2.7.12.1 0004672,0004712,0005524,0006468 remove_due_to_license_issue Q92630 1 HHSSGVDLGTENLYFQSMGKVKATPMTPEQAMKQYMQKLTAFEHHEIFSYPEIYFLGLNAKKRQGMTGGPNNGGYDDDQGSYVQVPHDHVAYRYEVLKVIGKGSFGQVVKAYDHKVHQHVALKMVRNEKRFHRQAAEEIRILEHLRKQDKDNTMNVIHMLENFTFRNHICMTFELLSMNLYELIKKNKFQGFSLPLVRKFAHSILQCLDALHKNRIIHCDLKPENILLKQQGRSGIKVIDFGSSCYEHQRVYTYIQSRFYRAPEVILGARYGMPIDMWSLGCILAELLTGYPLLPGEDEGDQLACMIELLGMPSQKLLDASKRAKNFVSSKGYPRYCTVTTLSDVVLNGGRSRRGKLRGPPESREWGNALKGCDDPLFLDFLKQCLEWDPAVRMTPGQALRHPWLR 3kvx A 2.4 BS01 FMY A 1 I70 G73 A74 Q75 V78 A91 K93 M146 E147 L148 M149 N152 S193 V196 L206 I25 G28 A29 Q30 V33 A46 K48 M101 E102 L103 M104 N107 S148 V151 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T169 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.148uM remove_due_to_license_issue P53779 19947601 403 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEEREHTIEEWKELIYKEVMNS 3kw9 A 1.8 BS01 ORG A 1 Q19 G23 C25 G65 G66 Y67 A134 L160 N161 H162 L209 Q19 G23 C25 G65 G66 Y67 A134 L160 N161 H162 L209 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=1nM P43235 20149657 216 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3kwa A 2.0 BS02 SPM A 1 Q92 H94 V121 L198 T199 T200 P201 P202 Q89 H91 V118 L194 T195 T196 P197 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=84000nM P00918 20590092 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3kwb X 2.02 BS01 ORH X 1 G1023 C1025 Y1067 A1134 A1137 S1138 L1160 N1161 L1209 G23 C25 Y67 A134 A137 S138 L160 N161 L209 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=17nM P43235 20153187 1216 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3kwf A 2.4 BS01 B1Q A 1 E205 E206 F357 Y662 Y666 N710 E167 E168 F319 Y624 Y628 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=6.8nM remove_due_to_license_issue IC50=6.8nM P27487 20031405 1 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3kwj A 2.8 BS01 23Q A 1 E205 E206 F357 Y547 S630 Y631 V656 Y662 Y666 V711 E167 E168 F319 Y509 S592 Y593 V618 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=0.500000nM P27487 20031408 1 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3kwz A 1.49 BS01 KWZ A 1 G23 C25 G64 G65 A134 L160 N161 H162 A163 G23 C25 G64 G65 A134 L160 N161 H162 A163 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=4nM P43235 20149657 222 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3kx1 A 1.51 BS01 KX1 A 1 G23 C25 G64 G65 G66 N161 H162 G21 C23 G62 G63 G64 N159 H160 Q19 C25 H162 N182 Q17 C23 H160 N180 3.4.22.38 0006508,0008234 ic50=100nM remove_due_to_license_issue IC50=100nM P43235 20149657 216 DSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3kxz A 2.37 BS02 925 A 1 E249 L251 A271 K273 E288 T316 M319 E320 L371 D382 E12 L14 A34 K36 E51 T79 M82 E83 L134 D145 D364 R366 A368 N369 D382 A400 F402 D127 R129 A131 N132 D145 A163 F165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.035uM remove_due_to_license_issue P06239 20038108 1 WEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTAT 3kyf A 2.1 BS01 5GP A 1 R127 H201 R120 H194 ? 0000166,0009288,0009425,0035438,0071945,0071973 remove_due_to_license_issue Q88EQ6 20226196 501 PQPPKVLSTPLEIAANLRQLQESHDPLIITFHDRSHRFQSYVVHVDRESNTLALDEMIPRDGEKFIENGEHFRVEGFHDGVRIAWECDHALKISEVDGHRCYSGPLPQEVTYHQRRNAFRAALKLSQLVDIILDGAHLKGNGAMRGKLLDISATGCKLRFEGNVEDRLQLGQVYERFKAGNPLGLVDTMVELRHLHYEERINTTFAGVRFHNLSGQAQRKIESFVYQLQRE 3kyf A 2.1 BS02 5GP A 2 F84 G87 Q121 R122 R123 F77 G80 Q114 R115 R116 ? 0000166,0009288,0009425,0035438,0071945,0071973 remove_due_to_license_issue Q88EQ6 20226196 502 PQPPKVLSTPLEIAANLRQLQESHDPLIITFHDRSHRFQSYVVHVDRESNTLALDEMIPRDGEKFIENGEHFRVEGFHDGVRIAWECDHALKISEVDGHRCYSGPLPQEVTYHQRRNAFRAALKLSQLVDIILDGAHLKGNGAMRGKLLDISATGCKLRFEGNVEDRLQLGQVYERFKAGNPLGLVDTMVELRHLHYEERINTTFAGVRFHNLSGQAQRKIESFVYQLQRE 3kyf A 2.1 BS03 5GP A 3 R127 D157 T161 G162 C163 K164 R200 H201 G214 V215 R216 R120 D150 T154 G155 C156 K157 R193 H194 G207 V208 R209 ? 0000166,0009288,0009425,0035438,0071945,0071973 remove_due_to_license_issue Q88EQ6 20226196 503 PQPPKVLSTPLEIAANLRQLQESHDPLIITFHDRSHRFQSYVVHVDRESNTLALDEMIPRDGEKFIENGEHFRVEGFHDGVRIAWECDHALKISEVDGHRCYSGPLPQEVTYHQRRNAFRAALKLSQLVDIILDGAHLKGNGAMRGKLLDISATGCKLRFEGNVEDRLQLGQVYERFKAGNPLGLVDTMVELRHLHYEERINTTFAGVRFHNLSGQAQRKIESFVYQLQRE 3kyf A 2.1 BS04 5GP A 4 R122 R123 N124 R127 R115 R116 N117 R120 ? 0000166,0009288,0009425,0035438,0071945,0071973 remove_due_to_license_issue Q88EQ6 20226196 504 PQPPKVLSTPLEIAANLRQLQESHDPLIITFHDRSHRFQSYVVHVDRESNTLALDEMIPRDGEKFIENGEHFRVEGFHDGVRIAWECDHALKISEVDGHRCYSGPLPQEVTYHQRRNAFRAALKLSQLVDIILDGAHLKGNGAMRGKLLDISATGCKLRFEGNVEDRLQLGQVYERFKAGNPLGLVDTMVELRHLHYEERINTTFAGVRFHNLSGQAQRKIESFVYQLQRE 3kyg A 2.1 BS01 5GP A 1 R136 R140 R169 N208 Q210 R116 R120 R149 N188 Q190 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 501 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg A 2.1 BS02 5GP A 2 R99 G100 Q134 R136 R79 G80 Q114 R116 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 502 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg A 2.1 BS03 5GP A 3 R140 D162 S164 G167 C168 R169 C207 N208 G219 L220 R120 D142 S144 G147 C148 R149 C187 N188 G199 L200 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 503 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg A 2.1 BS04 5GP A 4 E101 R135 R136 K137 R140 E81 R115 R116 K117 R120 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 504 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg B 2.1 BS01 5GP B 1 R136 R140 R169 N208 Q210 R116 R120 R149 N188 Q190 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 501 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg B 2.1 BS02 5GP B 2 R99 G100 Q134 R136 R79 G80 Q114 R116 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 502 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg B 2.1 BS03 5GP B 3 R140 D162 S164 G167 C168 R169 C207 N208 G219 E221 R120 D142 S144 G147 C148 R149 C187 N188 G199 E201 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 503 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyg B 2.1 BS04 5GP B 4 E101 R135 R136 K137 E81 R115 R116 K117 ? 0000166,0003674,0005515,0005575,0008150,0009288,0009425,0035438 remove_due_to_license_issue Q9KNC3 20226196 504 SKTVSTINSTDALAMVEHSSELTLSITTPVGTKFVCRTPFIGTHTDKFLLVEMPKISADDLQYFFQEGFWMNIRAISPRGEGALIHFRSQLMHILQEPVPMAFLSIPNTMQVSQRRKEPRFELNLAGKVLFDEHRGDCELRDLSRSGCRFITPPLGKTYQVGDLVALEIFSDLRGTKTFPPLTGKICNLQRSLHHARYGLEFNEEGRNNAKNLLAQLKFNGTKLTLN 3kyq A 2.443 BS01 DPV A 1 S27 F28 Q32 T43 Y64 S28 F29 Q33 T44 Y65 2.3.1.- 0000139,0005484,0005737,0005739,0005768,0005783,0005794,0005829,0005886,0006888,0006903,0006904,0008150,0015031,0016020,0016192,0016740,0019706,0030659,0031201,0031410,0042147,0043025,0061025,0097440,0097441 Kd=61uM remove_due_to_license_issue Q5EGY4 20159557 201 LMKLYSLSVFYKGEPKAVLLKAAYDVSSFSFFQRSSVQEFMTFTSQLIVERSAKGSRASVKEQEYLCHVYVRSDSLAGVVIADSEYPSRVAFTLLEKVLDEFSKQVDRIDWPVGSPATIHYTALDGHLSRYQNPREADPMSKVQAELDETKIILHNTMESLLERGEKLDDLVSKSEVLGTQSKAFYKTARKQN 3kyr A 2.6 BS01 038 A 1 G34 Y68 P70 Y71 T72 K75 R128 Y198 K224 I226 D228 R235 T329 G37 Y71 P73 Y74 T75 K78 R131 Y190 K216 I218 D220 R227 T310 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=190nM P56817 500 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 3l08 A 2.7 BS01 ZIG A 1 M804 I831 K833 I879 I881 V882 N951 M953 D964 M558 I585 K587 I633 I635 V636 N700 M702 D713 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=0.600000nM P48736 24900173 1109 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGSFNADKLTSATNPDKENSMSISILLIALPKHQRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLDVSSQVISQLKQKLENLQNLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGRVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 3l0e A 2.3 BS02 G58 A 1 F268 F271 T272 L274 A275 S278 M312 T316 R319 F329 L330 G344 L345 H435 F50 F53 T54 L56 A57 S60 M94 T98 R101 F111 L112 G126 L127 H217 ? 0003677,0004879,0006629 ic50=10nM remove_due_to_license_issue P55055 20345102 1 QLTAAQELMIQQLVAAQLQSNKRSFSDQPKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETESITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMSSLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLADAALPPLLSEIWDVHE 3l0k A 1.34 BS01 6AU A 1 S33 D35 K57 H59 D88 K90 M147 S148 P193 Q206 Y208 G226 R227 S35 D37 K59 H61 D90 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=24uM remove_due_to_license_issue P11172 19472232 257 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3l0k A 1.34 BS02 6AU B 1 D93 I94 T97 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=24uM remove_due_to_license_issue P11172 19472232 257 MELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3l0k B 1.34 BS01 6AU A 1 D93 I94 T97 D94 I95 T98 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=24uM remove_due_to_license_issue P11172 19472232 257 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3l0k B 1.34 BS02 6AU B 1 S33 D35 K57 H59 D88 K90 M147 S148 P193 Q206 Y208 G226 R227 S34 D36 K58 H60 D89 K91 M148 S149 P194 Q207 Y209 G227 R228 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=24uM remove_due_to_license_issue P11172 19472232 257 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3l0n A 1.74 BS01 S5P A 1 S33 D35 K57 H59 D88 K90 M147 S148 P193 Q206 Y208 G226 R227 S34 D36 K58 H60 D89 K91 M148 S149 P194 Q207 Y209 G227 R228 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=1680uM remove_due_to_license_issue P11172 19472232 257 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 3l0n A 1.74 BS02 S5P B 1 D93 I94 T97 D94 I95 T98 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=1680uM remove_due_to_license_issue P11172 19472232 257 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 3l0n B 1.74 BS01 S5P A 1 D93 I94 T97 D94 I95 T98 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=1680uM remove_due_to_license_issue P11172 19472232 257 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 3l0n B 1.74 BS02 S5P B 1 S33 D35 K57 H59 D88 K90 M147 S148 P193 Q206 Y208 G226 R227 S34 D36 K58 H60 D89 K91 M148 S149 P194 Q207 Y209 G227 R228 2.4.2.10,4.1.1.23 0004590,0006207,0044205 ic50=1680uM remove_due_to_license_issue P11172 19472232 257 ELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRL 3l0v A 1.75 BS02 724 A 1 T347 L348 G349 L401 V402 H405 E406 H409 H415 P437 A439 T132 L133 G134 L182 V183 H186 E187 H190 H196 P218 A220 3.4.24.86 0004222,0006508,0008237 Ki=23nM remove_due_to_license_issue Ki=23nM P78536 20172725 485 ADPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3l13 A 3.0 BS01 JZW A 1 K802 M804 A805 I831 D841 Y867 I879 E880 I881 V882 M953 I963 D964 K565 M567 A568 I594 D604 Y630 I642 E643 I644 V645 M716 I726 D727 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=15nM P48736 20050669 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3l16 A 2.9 BS01 JZX A 1 M804 I831 I879 E880 I881 V882 M953 I963 D964 M567 I594 I642 E643 I644 V645 M716 I726 D727 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=33nM P48736 20050669 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3l17 A 3.0 BS01 JZY A 1 M804 I831 K833 I879 E880 I881 V882 M953 I963 D964 M567 I594 K596 I642 E643 I644 V645 M716 I726 D727 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=5.2nM P48736 20050669 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3l1n A 1.3 BS01 PLM A 1 L96 S127 L91 S122 ? Kd=6.34uM remove_due_to_license_issue O42721 20053994 161 EATKVQRDISAFKKVMQNISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQIMLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAF 3l1s A 2.9 BS01 Z92 A 1 I62 V70 A83 K85 V110 L132 D133 Y134 V135 R141 L188 C199 D200 I35 V43 A56 K58 V83 L98 D99 Y100 V101 R107 L154 C165 D166 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 20138514 421 SMKVSRDSKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 3l25 A 2.0 BS01 rna C 0 F239 S272 Q274 I340 F22 S55 Q57 I123 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 A 2.0 BS02 rna F 0 G234 A306 K309 G17 A89 K92 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 B 2.0 BS01 rna C 0 I278 Q279 K282 R312 R322 I61 Q62 K65 R95 R105 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 B 2.0 BS02 rna F 0 F239 I340 F22 I123 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 D 2.0 BS01 rna C 0 G234 A306 K309 G17 A89 K92 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 D 2.0 BS02 rna F 0 F239 S272 Q274 C275 I340 F22 S55 Q57 C58 I123 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 E 2.0 BS01 rna C 0 F239 Q274 I340 F22 Q57 I123 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l25 E 2.0 BS02 rna F 0 I278 Q279 K282 R312 R322 I61 Q62 K65 R95 R105 ? remove_due_to_license_issue Q05127 20081868 1 ~ 8 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 3l2c A 1.868 BS01 dna B 0 R94 N95 S101 Y102 N148 H152 R2 N3 S9 Y10 N56 H60 ? 0003700,0006355,0043565 remove_due_to_license_issue P98177 21123876 1 ~ 13 RRNAWGNQSYAELISQAIESAPEKRLTLAQIYEWMVRTVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIKVHNEATGKSSWWMLN 3l2c A 1.868 BS02 dna C 0 L120 N141 S142 R151 H152 S155 K162 S171 S172 W174 L28 N49 S50 R59 H60 S63 K70 S79 S80 W82 ? 0003700,0006355,0043565 remove_due_to_license_issue P98177 21123876 25 ~ 37 RRNAWGNQSYAELISQAIESAPEKRLTLAQIYEWMVRTVPYFKDKGDSNSSAGWKNSIRHNLSLHSKFIKVHNEATGKSSWWMLN 3l2y A 2.7 BS03 OPE A 1 N61 L64 F66 E138 N61 L64 F66 E138 ? 0001849,0005509,0005515,0005576,0005615,0006953,0006954,0008228,0010628,0010745,0010888,0030169,0032677,0032930,0032945,0033265,0042310,0042802,0045087,0046790,0046872,0050750,0050830 remove_due_to_license_issue P02741 21360619 550 QTDMSRKAFVFPKESDTSYVSLKAPLTKPLKAFTVCLHFYTELSSTRGYSIFSYATKRQDNEILIFWSKDIGYSFTVGGSEILFEVPEVTVAPVHICTSWESASGIVEFWVDGKPRVRKSLKKGYTVGAEASIILGQEQDSFGGNFEGSQSLVGDIGNVNMWDFVLSPDEINTIYLGGPFSPNVLNWRALKYEVQGEVFTKPQLWP 3l38 A 2.1 BS01 879 A 1 Q74 G75 L92 D94 G96 V131 Y133 W138 F170 I172 W177 I180 D290 G292 Q15 G16 L33 D35 G37 V72 Y74 W76 F108 I110 W115 I118 D222 G224 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.1uM remove_due_to_license_issue IC50=100nM P56817 20223661 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCG 3l3a A 2.362 BS01 625 A 1 G73 Q74 G75 L92 D94 V131 Y133 W138 F170 I172 W177 I180 R190 D290 G292 T294 G14 Q15 G16 L33 D35 V72 Y74 W79 F111 I113 W118 I121 R131 D224 G226 T228 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.42uM remove_due_to_license_issue IC50=420nM P56817 20223661 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGY 3l3l A 2.5 BS01 L3L A 1 H201 G202 G227 Y228 Y235 K242 S243 Y246 E327 H201 G202 G227 Y228 Y235 K242 S243 Y246 E327 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 Ki=33nM remove_due_to_license_issue EC50=51nM, Ki=33nM P09874 20045315 351 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 3l3m A 2.5 BS01 A92 A 1 E102 D105 H201 G202 Y228 Y235 F236 S243 Y246 E101 D104 H200 G201 Y227 Y234 F235 S242 Y245 S243 Y246 E327 S242 Y245 E326 2.4.2.-,2.4.2.30 0003950 Ki=0.006uM remove_due_to_license_issue P09874 20337371 351 SKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 3l3n A 2.3 BS03 LSW A 1 Q281 H353 A354 V380 H383 E384 H387 E411 K511 H513 V518 Y520 Y523 F527 Q242 H314 A315 V341 H344 E345 H348 E372 K469 H471 V476 Y478 Y481 F485 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H471 Y481 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=7000nM P12821 20233165 1 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWP 3l4t A 1.9 BS01 BJ1 A 1 D203 Y299 D327 W406 D443 M444 F450 R526 D542 F575 H600 D190 Y286 D314 W393 D430 M431 F437 R513 D529 F562 H587 3.2.1.20 0003824,0004553,0005975,0030246 Ki=3.8uM remove_due_to_license_issue O43451 20039683 1001 NELERINCIPDQPPTKATCDQRGCCWNPQAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l4u A 1.9 BS01 DSK A 1 D203 Y299 D327 W406 D443 R526 D542 F575 H600 D197 Y293 D321 W400 D437 R520 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=0.03uM remove_due_to_license_issue O43451 20039683 4001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSQTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l4v A 2.1 BS01 KTL A 1 D203 Y299 D327 W406 D443 R526 D542 F575 H600 D197 Y293 D321 W400 D437 R520 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=0.19uM remove_due_to_license_issue O43451 20039683 1001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l4w A 2.0 BS01 MIG A 1 Y299 D327 W406 D443 M444 R526 W539 D542 F575 H600 Y293 D321 W400 D437 M438 R520 W533 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=1uM remove_due_to_license_issue IC50=6000nM, Ki=1000nM O43451 20039683 1001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l4x A 1.9 BS01 NR3 A 1 D203 Y299 D327 W406 D443 R526 D542 F575 H600 D197 Y293 D321 W400 D437 R520 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=0.13uM remove_due_to_license_issue O43451 20039683 1001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l4y A 1.8 BS01 NR4 A 1 D203 T205 Y299 D327 W406 D443 R526 D542 F575 H600 D197 T199 Y293 D321 W400 D437 R520 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=0.1uM remove_due_to_license_issue O43451 20039683 1001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l4z A 2.0 BS01 SSD A 1 D203 Y299 D327 W406 D443 R526 D542 F575 H600 D197 Y293 D321 W400 D437 R520 D536 F569 H594 3.2.1.20 0003824,0004553,0005975,0030246 Ki=0.19uM remove_due_to_license_issue O43451 20039683 1001 VNELERINCIPDQPPTKATCDQRGCCWNPQGAVSVPWCYYSKNHSYHVEGNLVNTNAGFTARLKNLPSSPVFGSNVDNVLLTAEYQTSNRFHFKLTDQTNNRFEVPHEHVQSFSGNAAASLTYQVEISRQPFSIKVTRRSNNRVLFDSSIGPLLFADQFLQLSTRLPSTNVYGLGEHVHQQYRHDMNWKTWPIFNRDTTPNGNGTNLYGAQTFFLCLEDASGLSFGVFLMNSNAMEVVLQPAPAITYRTIGGILDFYVFLGNTPEQVVQEYLELIGRPALPSYWALGFHLSRYEYGTLDNMREVVERNRAAQLPYDVQHADIDYMDERRDFTYDSVDFKGFPEFVNELHNNGQKLVIIVDPAISNNSSSSKPYGPYDRGSDMKIWVNSSDGVTPLIGEVWPGQTVFPDYTNPNCAVWWTKEFELFHNQVEFDGIWIDMNEVSNFVDGSVSGCSTNNLNNPPFTPRILDGYLFCKTLCMDAVQHWGKQYDIHNLYGYSMAVATAEAAKTVFPNKRSFILTRSTFAGSGKFAAHWLGDNTATWDDLRWSIPGVLEFNLFGIPMVGPDICGFALDTPEELCRRWMQLGAFYPFSRNHNGQGYKDQDPASFGADSLLLNSSRHYLNIRYTLLPYLYTLFFRAHSRGDTVARPLLHEFYEDNSTWDVHQQFLWGPGLLITPVLDEGAEKVMAYVPDAVWYDYETGSQVRWRKQKVEMELPGDKIGLHLRGGYIFPTQQPNTTTLASRKNPLGLIIALDENKEAKGELFWDDGETKDTVANKVYLLCEFSVTQNRLEVNISQSTYKDPNNLAFNEIKILGTEEPSNVTVKHNGVPSTSPTVTYDSNLKVAIITDIDLLLGEAYTVEWAH 3l54 A 2.3 BS01 LXX A 1 M804 I831 K833 Y867 I879 E880 I881 V882 M953 I963 D964 M556 I583 K585 Y619 I631 E632 I633 V634 M705 I715 D716 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 24900173 1 MSQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTDFVLRVCGRDEYLVGETPIKNFQWVRQCLKNGEEIHVVLDTPPDPALDEVRKESLWDCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGQLLYYVNLLLIDHRFLLRRGEYVLHMWQIFNADKLTSATNPDKENSMSISILLDIALPKAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLDVSSQVISQLKQKLENLQNLNLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYRVPFVLTPDFLFVMGTSGKKTSPHFQKFQDVCVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLGI 3l58 A 1.8 BS01 CS5 A 1 G72 L91 D93 G95 Y132 T133 Q134 F169 Y259 D289 G291 T292 T293 R296 G20 L39 D41 G43 Y80 T81 Q82 F117 Y207 D237 G239 T240 T241 R244 D93 S96 N98 A100 Y132 D289 T292 D41 S44 N46 A48 Y80 D237 T240 3.4.23.46 0004190,0006508,0016020 ic50=8nM remove_due_to_license_issue IC50=20nM P56817 20043696 1 EPGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l59 A 2.0 BS01 BDJ A 1 D93 Y132 D289 G291 D36 Y75 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Kd=200uM remove_due_to_license_issue P56817 20043696 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l5b A 1.8 BS01 BDO A 1 D93 D289 G291 D36 D229 G231 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D229 T232 3.4.23.46 0004190,0006508,0016020 Kd=123uM remove_due_to_license_issue P56817 20043696 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l5c A 1.8 BS01 BDQ A 1 D93 Y132 K168 F169 Y259 D289 D36 Y75 K108 F109 Y199 D229 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D229 T232 3.4.23.46 0004190,0006508,0016020 ic50=7000nM remove_due_to_license_issue P56817 20043696 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l5d A 1.75 BS01 BDV A 1 D93 D289 G291 T292 T293 D36 D228 G230 T231 T232 D93 S96 N98 A100 D289 T292 D36 S39 N41 A43 D228 T231 3.4.23.46 0004190,0006508,0016020 ic50~78000nM remove_due_to_license_issue P56817 20043696 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l5e A 1.53 BS01 BDW A 1 Q73 D93 S96 V130 Y132 I187 R189 D289 G291 T292 T293 Q16 D36 S39 V73 Y75 I130 R132 D232 G234 T235 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=27nM remove_due_to_license_issue Ki=27nM P56817 20043696 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l5f A 1.7 BS01 BDX A 1 L91 D93 G95 Y132 R189 D289 G291 L34 D36 G38 Y75 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=605nM remove_due_to_license_issue P56817 20043696 1 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3l5r A 1.94 BS01 47X A 1 P1 K32 Y36 H62 S63 I64 V106 F113 P1 K32 Y36 H62 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=38nM remove_due_to_license_issue IC50=38nM, Ki=38nM P14174 20185308 123 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3l5r C 1.94 BS01 47X A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue IC50=38nM, Ki=38nM P14174 20185308 123 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFALEHH 3l79 A 1.86 BS01 DKX A 1 G135 L136 N284 H377 N484 E672 S674 G675 G124 L125 N267 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=3.46mM remove_due_to_license_issue P00489 20430629 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3l7a A 1.9 BS01 DKY A 1 G135 L136 N282 N284 F285 H377 A383 N484 E672 A673 S674 G675 G124 L125 N265 N267 F268 H352 A358 N459 E647 A648 S649 G650 H377 K568 R569 K574 T676 K680 H352 K543 R544 K549 T651 K655 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=46.42uM remove_due_to_license_issue P00489 20430629 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3l7b A 2.0 BS01 DKZ A 1 G135 L136 N284 H377 N484 E672 S674 G675 G124 L125 N267 H350 N457 E645 S647 G648 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.01mM remove_due_to_license_issue P00489 20430629 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3l7c A 1.93 BS01 DK4 A 1 G135 L136 D283 N284 H377 T378 N484 E672 A673 S674 G675 G124 L125 D266 N267 H353 T354 N460 E648 A649 S650 G651 H377 K568 R569 K574 T676 K680 H353 K544 R545 K550 T652 K656 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=3.67mM remove_due_to_license_issue P00489 20430629 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3l7d A 2.0 BS01 DK5 A 1 G135 L136 N282 N284 F285 F286 H341 H377 A383 N484 E672 A673 S674 G675 G124 L125 N265 N267 F268 F269 H314 H350 A356 N457 E645 A646 S647 G648 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=6.55mM remove_due_to_license_issue P00489 20430629 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3l7g A 2.7 BS01 M44 A 1 Y212 D244 D255 H332 H343 E381 R418 E420 Y212 D244 D255 H332 H343 E366 R403 E405 D45 H226 D244 D255 H332 H336 H343 E381 Y385 R418 E420 D45 H226 D244 D255 H332 H336 H343 E366 Y370 R403 E405 3.1.8.1,3.4.13.9,3.8.2.2 0004063,0004177,0005829,0006508,0008235,0008237,0009636,0016795,0016805,0046872,0047862,0102009 remove_due_to_license_issue Q44238 20000741 518 MNKLAVLYAEHIATLQKRTREIIERENLDGVVFHSGQAKRQFLDDMYYPFKVNPQFKAWLPVIDNPHCWIVANGTDKPKLIFYRPVDFWHKVPDEPNEYWADYFDIELLVKPDQVEKLLPYDKARFAYIGEYLEVAQALGFELMNPEPVMNFYHYHRAYKTQYELACMREANKIAVQGHKAARDAFFQGKSEFEIQQAYLLATQHSENDNPYGNIVALNENCAILHYTHFDRVAPATHRSFLIDAGANFNGYAADITRTYDFTGEGEFAELVATMKQHQIALMNQLAPGKLYGELHLDCHQRVAQTLSDFNIVDLSADEIVAKGITSTFFPHGLGHHIGLQVHDVGGFMALRCTRKIEANQVFTIEPGLYFIDSLLGDLAATDNNQHINWDKVAELKPFGGIRIEDNIIVHEDSLENMTRELRLR 3l8s A 2.35 BS01 BFF A 1 A51 K53 I84 T106 L108 M109 G110 A111 D112 A45 K47 I78 T100 L102 M103 G104 A105 D106 D150 K152 N155 D168 T185 D144 K146 N149 D162 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=99nM remove_due_to_license_issue Q16539 20201574 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSLESRDLLIDEWKSLTYDEVISFVPPPL 3l8v A 2.4 BS01 L8V A 1 I1084 V1092 A1108 K1110 E1127 M1131 F1134 L1157 M1160 H1202 M1211 V1220 A1221 D1222 F1223 I31 V39 A55 K57 E74 M78 F81 L104 M107 H149 M158 V167 A168 D169 F170 D1204 A1206 R1208 N1209 D1222 A1243 D151 A153 R155 N156 D169 A176 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.008uM remove_due_to_license_issue IC50=8nM P08581 20382527 1 DLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3l9h A 2.0 BS02 EMQ A 1 E116 E118 R119 W127 A133 P137 L160 L214 A218 R221 E101 E103 R104 W112 A118 P122 L145 L199 A203 R206 ? 0003777,0005524,0007018,0008017 ic50=8nM remove_due_to_license_issue IC50=8nM P52732 20149654 601 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNK 3l9l A 2.0 BS02 L9L A 1 F54 V57 A70 K72 Y122 V123 E127 E170 N171 L173 T183 D184 F327 F44 V47 A60 K62 Y112 V113 E117 E160 N161 L163 T173 D174 F317 D166 K168 E170 N171 D184 T201 D156 K158 E160 N161 D174 T191 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 ic50=167nM remove_due_to_license_issue P17612 20137943 351 EQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3l9m A 1.9 BS02 L9M A 1 L49 F54 A70 K72 M120 E121 E170 N171 M173 T183 D184 F327 L39 F44 A60 K62 M110 E111 E160 N161 M163 T173 D174 F317 D166 K168 E170 N171 D184 T201 D156 K158 E160 N161 D174 T191 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 20137943 351 EQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3l9n A 2.0 BS02 L9N A 1 L49 F54 A70 K72 M120 E121 A123 E170 N171 M173 T183 D184 L36 F41 A57 K59 M107 E108 A110 E157 N158 M160 T170 D171 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 20137943 351 SVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3lau A 2.1 BS01 OFI A 1 L139 V147 E211 Y212 A213 L263 L16 V24 E88 Y89 A90 L140 D256 K258 E260 N261 D274 D133 K135 E137 N138 D151 2.7.11.1 0004672,0005524,0006468 ic50=0.044uM remove_due_to_license_issue O14965 20167481 1 MKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 3lbj E 1.5 BS01 WW8 E 1 M53 L56 G57 I60 M61 Y66 Q71 V92 L98 M29 L32 G33 I36 M37 Y42 Q47 V68 L74 ? 0005634,0043066,0051726 remove_due_to_license_issue EC50=20000nM O15151 20237429 1 NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV 3lbj E 1.5 BS02 WW8 E 2 V27 V49 Y99 R103 V3 V25 Y75 R79 ? 0005634,0043066,0051726 remove_due_to_license_issue EC50=20000nM O15151 20237429 112 NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV 3lbk A 2.3 BS01 K23 A 1 L54 L57 G58 I61 M62 F86 V93 H96 I99 Y100 L29 L32 G33 I36 M37 F61 V68 H71 I74 Y75 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=920nM Q00987 20237429 1 TLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 3lbl A 1.6 BS01 MI6 A 1 L54 I61 M62 F86 H96 I99 L38 I45 M46 F70 H80 I83 2.3.2.27 0005634,0043066,0051726 Ki=36nM remove_due_to_license_issue Ki=3.0nM Q00987 20237429 1 MQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 3lbz A 2.3 BS02 Z89 A 1 N21 R24 L25 R28 N15 R18 L19 R22 ? Kd=138uM remove_due_to_license_issue P41182 20385364 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 3lbz A 2.3 BS03 Z89 A 2 M51 G55 Y58 M45 G49 Y52 ? Kd=138uM remove_due_to_license_issue P41182 20385364 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 3lbz B 2.3 BS01 Z89 A 1 M51 Y58 M45 Y52 ? Kd=138uM remove_due_to_license_issue P41182 20385364 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 3lbz B 2.3 BS02 Z89 A 2 N21 R24 L25 R28 N15 R18 L19 R22 ? Kd=138uM remove_due_to_license_issue P41182 20385364 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 3lbz B 2.3 BS04 Z89 B 1 I60 K66 N73 D75 P76 Y111 I54 K60 N67 D69 P70 Y105 ? Kd=138uM remove_due_to_license_issue P41182 20385364 203 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 3lc3 A 1.9 BS01 IYX A 1 D189 S190 C191 Q192 S195 W215 G216 E217 C220 D179 S180 C181 Q182 S185 W205 G206 E207 C209 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 Ki=5.9uM remove_due_to_license_issue P00740 20121198 1 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGRSALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKLT 3lc3 A 1.9 BS02 IYX A 2 K98 Y99 H147 W215 G216 E217 K85 Y86 H135 W205 G206 E207 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 Ki=5.9uM remove_due_to_license_issue P00740 20121198 2 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGRSALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKLT 3lc5 A 2.62 BS02 IZX A 1 R143 H147 F174 D189 S190 Q192 S195 W215 G216 E219 C220 R132 H135 F162 D179 S180 Q182 S185 W205 G206 E208 C209 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 remove_due_to_license_issue P00740 20121197 1 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGRSALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKLT 3lcd A 2.5 BS01 BDY A 1 L588 G589 A614 Y665 C666 G669 L785 L31 G32 A57 Y108 C109 G112 L164 D778 A780 R782 N783 D796 N814 D157 A159 R161 N162 D175 N191 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=40nM remove_due_to_license_issue P07333 20137931 923 GNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKAEADLDPLELRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMSNYIVKGNARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQ 3lce A 2.0 BS01 LCE A 1 S67 K70 S115 V117 T206 G207 F208 R250 S47 K50 S95 V97 T186 G187 F188 R230 S67 K70 S115 F120 W154 F208 S47 K50 S95 F100 W134 F188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0042597,0046677,0071555 remove_due_to_license_issue P14489 20141132 269 SITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNDLARASKEYLPASTFKIPNAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLTLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLYLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKETEVYFFAFNMDIDNESKLPLRKSIPTKIMESEGIIG 3lco A 3.4 BS01 LC0 A 1 L588 A614 K616 V647 E664 C666 L785 G795 D796 F797 L30 A56 K58 V89 E106 C108 L167 G177 D178 F179 D778 R782 N783 D796 D160 R164 N165 D178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=143nM P07333 20137931 999 KIIEFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKAEAMLGPSGRPLELRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVRLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQAQ 3lcu A 2.1 BS01 SAH A 1 I60 F64 H102 S104 T105 R108 A133 C134 D156 I157 D182 L183 L198 Q207 I53 F57 H95 S97 T98 R101 A126 C127 D149 I150 D175 L176 L191 Q200 2.1.1.179 0006364,0008168,0008649,0031167,0032259,0046677 Kd=300uM remove_due_to_license_issue Q7M0R2 20194115 6732 DRIDEIERAITKSRRYQTVAPATVRRLARAALVAARGDVPDAVKRTKRGLHEIYGAFLPPSPPNYAALLRHLDSAVDAGDDEAVRAALLRAMSVHISTRERLPHLDEFYRELFRHLPRPNTLRDLACGLNPLAAPWMGLPAETVYIASDIDARLVGFVDEALTRLNVPHRTNVADLLEDRLDEPADVTLLLKTLPCLETQQRGSGWEVIDIVNSPNIVVTFPTKGMFQNYSQSFESQARERSCRIQRLEIGNELIYVIQK 3lcv B 2.0 BS01 SAM B 1 I60 F64 S104 T105 R108 A133 C134 D156 I157 D182 L183 L198 K199 Q207 I53 F57 S97 T98 R101 A126 C127 D149 I150 D175 L176 L191 K192 Q200 2.1.1.179 0006364,0008168,0008649,0031167,0032259,0046677 Kd=18uM remove_due_to_license_issue Q7M0R2 20194115 301 DRIDEIERAITKSRRYQTVAPATVRRLARAALVAARGDVPDAVKRTKRGLHEIYGAFLPPSPPNYAALLRHLDSAVDAGDDEAVRAALLRAMSVHISTRERLPHLDEFYRELFRHLPRPNTLRDLACGLNPLAAPWMGLPAETVYIASDIDARLVGFVDEALTRLNVPHRTNVADLLEDRLDEPADVTLLLKTLPCLETQQRGSGWEVIDIVNSPNIVVTFPTKGMFQNYSQSFESQARERSCRIQRLEIGNELIYVIQ 3ldp A 2.2 BS01 3P1 A 1 Y39 G227 G255 E293 K296 R297 S300 G364 R367 D391 Y14 G202 G230 E268 K271 R272 S275 G339 R342 D366 D34 K96 E201 D224 D9 K71 E176 D199 3.6.4.10 0005524,0140662 Kd=2.41uM remove_due_to_license_issue koff=0.4s-1, Kd=2.41e+3nM P11021 21526763 408 DVGTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQLTSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDIGGGQTKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLS 3ldq A 1.9 BS01 3P1 A 1 G202 E268 K271 R272 S275 G339 R342 G198 E264 K267 R268 S271 G335 R338 D10 K71 E175 D199 D6 K67 E171 D195 3.6.4.10 0005524,0140662 Kd=2.41uM remove_due_to_license_issue P11142 21526763 401 PAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 3ldw A 2.47 BS01 ZOL A 1 D126 R135 Q195 K243 T244 D287 K301 D92 R101 Q161 K205 T206 D249 K263 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 Ki=10.7nM remove_due_to_license_issue A5K4U6 21084289 397 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3le6 A 2.0 BS01 2BZ A 1 I10 G11 E12 G13 V18 A31 F80 E81 F82 L83 H84 D86 L134 I10 G11 E12 G13 V18 A31 F69 E70 F71 L72 H73 D75 L123 D127 K129 Q131 N132 D145 T158 T165 D116 K118 Q120 N121 D134 T147 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.035uM remove_due_to_license_issue P24941 20832307 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVP 3le8 A 1.7 BS01 2B5 A 1 P38 T39 M40 H44 G46 H47 F157 K160 Q164 V187 S196 S197 P36 T37 M38 H42 G44 H45 F155 K158 Q162 V185 S194 S195 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=860nM remove_due_to_license_issue Kd=860nM P9WIL5 20232910 301 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 3le9 A 1.85 BS02 727 A 1 T347 L348 G349 L350 L401 V402 H405 E406 H415 P437 T130 L131 G132 L133 L178 V179 H182 E183 H192 P214 3.4.24.86 0004222,0006508,0008237 Ki=6nM remove_due_to_license_issue Ki=6nM P78536 20663669 485 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3lea A 2.0 BS01 Z93 A 1 T347 L348 G349 L350 L401 V402 H405 E406 H409 H415 A439 T131 L132 G133 L134 L185 V186 H189 E190 H193 H199 A223 3.4.24.86 0004222,0006508,0008237 Ki=0.8nM remove_due_to_license_issue P78536 20663669 1 DPDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3lf0 A 2.4 BS01 ATP A 1 G35 Y36 G37 R38 G87 G89 K90 G37 Y38 G39 R40 G74 G76 K77 ? 0000166,0005524,0005829,0005886,0006808,0030234,0043531,0051701 Kd=1.93uM remove_due_to_license_issue P9WN31 20521335 701 SHMKLITAIVKPFTLDDVKTSLEDAGVLGMTVSEIQGYGRDFVPKVRIEVVVDDSIVDKVVDSIVRAARTGKIGDGKVWVSPVDTIVRVRTGERGHDAL 3lf0 A 2.4 BS02 ATP C 1 G27 V63 V64 R101 R103 G29 V50 V51 R88 R90 ? 0000166,0005524,0005829,0005886,0006808,0030234,0043531,0051701 Kd=1.93uM remove_due_to_license_issue P9WN31 20521335 701 SHMKLITAIVKPFTLDDVKTSLEDAGVLGMTVSEIQGYGRDFVPKVRIEVVVDDSIVDKVVDSIVRAARTGKIGDGKVWVSPVDTIVRVRTGERGHDAL 3lf0 B 2.4 BS01 ATP A 1 G27 M28 T29 V63 V64 R101 R103 G28 M29 T30 V63 V64 R101 R103 ? 0000166,0005524,0005829,0005886,0006808,0030234,0043531,0051701 Kd=1.93uM remove_due_to_license_issue P9WN31 20521335 701 HMKLITAIVKPFTLDDVKTSLEDAGVLGMTVSEIQGYGRQGHTEVYRGAEYSVDFVPKVRIEVVVDDSIVDKVVDSIVRAARTGKIGDGKVWVSPVDTIVRVRTGERGHDAL 3lf0 B 2.4 BS02 ATP B 1 G35 Y36 G37 R38 I86 G87 G89 K90 G36 Y37 G38 R39 I86 G87 G89 K90 ? 0000166,0005524,0005829,0005886,0006808,0030234,0043531,0051701 Kd=1.93uM remove_due_to_license_issue P9WN31 20521335 701 HMKLITAIVKPFTLDDVKTSLEDAGVLGMTVSEIQGYGRQGHTEVYRGAEYSVDFVPKVRIEVVVDDSIVDKVVDSIVRAARTGKIGDGKVWVSPVDTIVRVRTGERGHDAL 3lfn A 2.28 BS01 A27 A 1 I10 V18 A31 K33 F80 F82 L83 H84 L134 A144 D145 L148 I10 V18 A31 K33 F76 F78 L79 H80 L130 A140 D141 L144 D127 K129 Q131 N132 D145 T165 D123 K125 Q127 N128 D141 T152 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=3160nM remove_due_to_license_issue P24941 20167481 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3lfs A 2.4 BS01 A07 A 1 I10 A31 K33 F80 L83 H84 Q85 D86 K89 N132 L134 D145 I10 A31 K33 F72 L75 H76 Q77 D78 K81 N124 L126 D137 D127 K129 Q131 N132 D145 T158 T165 D119 K121 Q123 N124 D137 T150 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=2.5uM remove_due_to_license_issue IC50=2500nM P24941 20167481 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3lgp A 1.9 BS02 50X A 1 T347 G349 L350 E398 L401 H405 E406 H409 H415 V434 Y436 P437 I438 A439 V440 S441 N447 T130 G132 L133 E175 L178 H182 E183 H186 H192 V211 Y213 P214 I215 A216 V217 S218 N224 3.4.24.86 0004222,0006508,0008237 Ki=2nM remove_due_to_license_issue Ki=2nM P78536 20638281 485 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3lgs A 2.2 BS01 SAH A 1 T116 C117 G118 L181 K199 D200 M201 D225 F237 T95 C96 G97 L160 K178 D179 M180 D204 F216 3.2.2.16 0000003,0003824,0005829,0005886,0008930,0009086,0009116,0010087,0016787,0019509 Kd=24.8uM remove_due_to_license_issue Q9T0I8 20554051 268 ILRPISSVVFVIAMQAEALPLVNKFGLSETTDSPLGKGLPWVLYHGVHKDLRINVVCPGRDAALGIDSVGTVPASLITFASIQALKPDIIINAGTCGGFKVKGANIGDVFLVSDVVFHDRRIPIPMFDLYGVGLRQAFSTPNLLKELNLKIGRLSTGDSLDMSTQDETLIIANDATLKDMEGAAVAYVADLLKIPVVFLKAVTDLVDGDKPTAEEFLQNLTVVTAALEGTATKVINFINGRNLSDL 3lgs B 2.2 BS01 SAH B 1 T116 C117 G118 L181 K199 D200 M201 T224 D225 F237 T94 C95 G96 L159 K177 D178 M179 T202 D203 F215 3.2.2.16 0000003,0003824,0005829,0005886,0008930,0009086,0009116,0010087,0016787,0019509 Kd=24.8uM remove_due_to_license_issue Q9T0I8 20554051 268 LRPISSVVFVIAMQAEALPLVNKFGLSETTDSPLGKGLPWVLYHGVHKDLRINVVCPGRDAALGIDSVGTVPASLITFASIQALKPDIIINAGTCGGFKVKGANIGDVFLVSDVVFHDRRIPIPMFDLYGVGLRQAFSTPNLLKELNLKIGRLSTGDSLDMSTQDETLIIANDATLKDMEGAAVAYVADLLKIPVVFLKAVTDLVDGDKPTAEEFLQNLTVVTAALEGTATKVINFINGRNLSDL 3lhg A 2.1 BS01 Z81 A 1 G73 G75 D94 S97 F170 I172 W177 I180 D290 G292 G14 G16 D35 S38 F111 I113 W118 I121 D224 G226 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.02uM remove_due_to_license_issue IC50=20nM P56817 20202842 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTDCGYN 3lhj A 3.31 BS01 LHJ A 1 K53 E71 L75 T106 A111 L167 D168 F169 K49 E67 L71 T102 A107 L163 D164 F165 D150 K152 N155 D168 T185 D146 K148 N151 D164 T174 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Ki=2.3nM, Kd=0.31nM Q16539 20218619 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3lhs A 1.3 BS01 SF8 A 1 R104 R126 H209 Y244 R299 R304 R306 R69 R91 H174 Y209 R264 R269 R271 ? remove_due_to_license_issue A0A0H3K9U6 20147287 501 ASTISVKDENGTVKVPKDAKRIVVLEYSFADALAALDVKPVGIADDGKKKRIIKPVREKIGDYTSVGTRKQPNLEEISKLKPDLIIADSSRHKGINKELNKIAPTLSLKSFDGDYKQNINSFKTIAKALNKEKEGEKRLAEHDKLINKYKDEIKFDRNQKVLPAVVAKAGLLAHPNYSYVGQFLNELGFKNALSDDVTKGLSKYLKGPYLQLDTEHLADLNPERMIIMTDHAKKDSAEFKKLQEDATWKKLNAVKNNRVDIVDRDVWARSRGLISSEEMAKELVELSKKEQ 3li2 A 2.2 BS01 SF8 A 1 R104 R126 V200 A202 K203 H209 Y239 Y244 R299 R304 R306 R69 R91 V165 A167 K168 H174 Y204 Y209 R264 R269 R271 ? remove_due_to_license_issue A0A0H3K9U6 20147287 501 ASTISVKDENGTVKVPKDAKRIVVLEYSFADALAALDVKPVGIADDGKKKRIIKPVREKIGDYTSVGTRKQPNLEEISKLKPDLIIADSSRHKGINKELNKIAPTLSLKSFDGDYKQNINSFKTIAKALNKEKEGEKRLAEHDKLINKYKDEIKFDRNQKVLPAVVAKAGLLAHPNYSYVGQFLNELGFKNALSDDVTKGLSKYLKGPYLQLDTEHLADLNPERMIIMTDHAKKDSAEFKKLQEDATWKKLNAVKNNRVDIVDRDVWARSRGLISSEEMAKELVELSK 3lik A 1.8 BS06 EEG A 1 G178 G179 L181 T215 H218 K233 A234 V235 P238 T239 Y240 K241 G74 G75 L77 T111 H114 K129 A130 V131 P134 T135 Y136 K137 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=1.92nM remove_due_to_license_issue Ki=1.92nM P39900 20817735 301 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3lil A 1.8 BS06 EEA A 1 G178 G179 L181 T215 H218 K233 A234 V235 P238 T239 Y240 K241 V243 G74 G75 L77 T111 H114 K129 A130 V131 P134 T135 Y136 K137 V139 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=8.3nM remove_due_to_license_issue Ki=8.3nM P39900 20817735 301 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3lir A 1.9 BS06 EEC A 1 G178 G179 L181 T215 H218 V235 F237 P238 T239 Y240 G74 G75 L77 T111 H114 V131 F133 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=119nM remove_due_to_license_issue Ki=119nM P39900 20817735 1 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3liw A 2.22 BS03 RUP A 1 Y99 R143 E146 F174 D189 A190 C191 Q192 W215 G216 G218 C220 Y85 R132 E135 F162 D179 A180 C181 Q182 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.025uM remove_due_to_license_issue P00742 12437104 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3lj3 A 2.43 BS01 WYE A 1 W812 I831 K833 D841 Y867 I879 E880 V882 M953 D964 W563 I582 K584 D592 Y618 I630 E631 V633 M703 D714 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=43nM remove_due_to_license_issue P48736 20188552 1109 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMSEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVRLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 3lj7 A 2.3 BS01 OHO A 1 F192 I238 G239 S241 F160 I206 G207 S209 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 20493882 1 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQ 3ljg A 1.313 BS06 EEF A 1 G179 L181 T215 H218 V235 F237 P238 T239 Y240 G75 L77 T111 H114 V131 F133 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=18.6nM remove_due_to_license_issue P39900 20817735 302 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3ljj A 1.55 BS01 10U A 1 D189 S190 C191 Q192 S214 W215 G216 S217 G219 D171 S172 C173 Q174 S192 W193 G194 S195 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=300nM remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3ljo A 1.5 BS01 11U A 1 L99 D189 S190 C191 V213 W215 G216 S217 G219 L81 D171 S172 C173 V191 W193 G194 S195 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=239nM remove_due_to_license_issue P00760 21111747 501 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3ljt A 1.6 BS01 LA3 A 1 D377 L379 F406 T407 H410 E411 H414 H420 L438 S441 I442 L443 I446 D115 L117 F144 T145 H148 E149 H152 H158 L176 S179 I180 L181 I184 3.4.24.- 0004222,0006508,0008237 ic50=129nM remove_due_to_license_issue Q9UNA0 21370305 801 ASRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3ljz A 2.0 BS05 LA3 A 1 L185 A186 L218 H222 E223 H226 H232 L239 P242 I243 Y244 L82 A83 L115 H119 E120 H123 H129 L136 P139 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=7.3nM remove_due_to_license_issue P45452 21370305 801 ANVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTHFMLPDDDVQGIQSLYG 3lk0 B 2.04 BS03 Z80 B 1 H42 F87 H43 F88 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=696.9uM remove_due_to_license_issue P02638 21132089 92 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFF 3lk8 A 1.8 BS06 Z79 A 1 I180 L181 A182 T215 H218 E219 H222 H228 P238 Y240 I75 L76 A77 T110 H113 E114 H117 H123 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=19.7nM remove_due_to_license_issue Ki=20nM P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3lka A 1.8 BS06 M4S A 1 T215 H218 E219 P238 Y240 T110 H113 E114 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=1.5mM remove_due_to_license_issue P39900 20415416 1 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3lkh A 2.05 BS01 LT6 A 1 F193 Q194 Y195 S196 P197 S368 L384 M414 Y415 Y448 Y452 L466 W550 F551 G554 F188 Q189 Y190 S191 P192 S363 L379 M409 Y410 Y443 Y447 L461 W541 F542 G545 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.8uM remove_due_to_license_issue O92972 20219368 577 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPLDLSGWFVAGYSGGDIYHS 3lkj A 2.5 BS01 LKJ C 1 L168 Y170 V228 E230 L259 L261 L48 Y50 V100 E102 L131 L133 ? 0005164,0006955,0016020 remove_due_to_license_issue P29965 21417339 1 QIAAHVISEASSKTTSVLQWAEKGYYTMSNNLVTLENGKQLTVKRQGLYYIYAQVTFCASSQAPFIASLCLKSPGRFERILLRAANTKPCGQQSIHLGGVFELQPGASVFVNVTDPSQVSHGTGFTSFGLLKL 3lkj B 2.5 BS01 LKJ C 1 Y170 A173 H224 L225 Y47 A50 H95 L96 ? 0005164,0006955,0016020 remove_due_to_license_issue P29965 21417339 1 QIAAHVISEASTSVLQWAEKGYYTMSNNLVTLENGKQLTVKRQGLYYIYAQVTFCSNAPFIASLCLKSPGRFERILLRAANTHSSAKPCGQQSIHLGGVFELQPGASVFVNVTDPSQVSHGTGFTSFGLLKL 3lkj C 2.5 BS01 LKJ C 1 Q121 H125 Y145 Y146 Y170 Y172 H224 L259 Q1 H5 Y25 Y26 Y50 Y52 H92 L127 ? 0005164,0006955,0016020 ic50=25uM remove_due_to_license_issue P29965 21417339 1 QIAAHVISEASSKTTSVLQWAEKGYYTMSNNLVTLENGKQLTVKRQGLYYIYAQVTFCSNPFIASLCLKSPGRFERILLRAANTPCGQQSIHLGGVFELQPGASVFVNVTDPSQVSHGTGFTSFGLLKL 3lkz A 2.0 BS01 SFG A 1 S56 G58 G81 G86 W87 K105 H110 E111 D131 V132 F133 D146 I147 S52 G54 G77 G82 W83 K101 H106 E107 D127 V128 F129 D142 I143 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0004482,0004483,0005524,0008168,0032259 remove_due_to_license_issue Q9Q6P4 20685660 301 GRTLGEVWKERLNQMTKEEFTRYRKEAIIEVDRSAAKHARKEGNVTGGHPVSRGTAKLRWLVERRFLEPVGKVIDLGCGRGGWCYYMATQKRVQEVRGYTKGGPGHEEPQLVQSYGWNIVTMKSGVDVFYRPSECCDTLLCDIGESSSSAEVEEHRTIRVLEMVEDWLHRGPREFCVKVLCPYMPKVIEKMELLQRRYGGGLVRNPLSRNSTHEMYWVSRASGNVVHSVNMTSQVLLGRMEKRTWKGPQYEEDVNLGSGTRA 3lle A 1.85 BS03 SGE A 1 F43 C84 F87 F88 F44 C85 F88 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 remove_due_to_license_issue P02638 21132089 94 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 3lle B 1.85 BS03 SGE B 1 F43 C84 F87 F88 F44 C85 F88 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 remove_due_to_license_issue P02638 21132089 94 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 3llm A 2.8 BS02 ADP A 1 T413 G414 C415 G416 K417 T418 T419 R456 T85 G86 C87 G88 K89 T90 T91 R128 3.6.4.13 0003676,0005524,0033679 remove_due_to_license_issue Q08211 20510246 565 VVPWSPPQSNWNPWTSSNIDEGPLAFATPEQISMDLKNELMYQLEQDHDLQAILQERELLPVKKFESEILEAISQNSVVIIRGATGCGKTTQVPQFILDDFIQNDRAAECNIVVTQPRRISAVSVAERVAFERGEEPGKSCGYSVRFESILPRPHASIMFCTVGVLLRKLEAGIRGISHVIVDEIHERDINTDFLLVVLRDVVQAYPEVRIVLMSATIDTSMFCEYFFNCPIIEV 3lm1 A 2.1 BS04 LEC A 1 G1 E76 Y78 G121 Y122 W123 D125 G1 E76 Y78 G121 Y122 W123 D125 ? 0030246 Kd=20uM remove_due_to_license_issue P18674 20826825 134 GVTFDDGAYTGIREINFEYNSETAIGGLRVTYDLNGMPFVAEDHKSFITGFKPVKISLEFPSEYIVEVSGYVGKVEGYTVIRSLTFKTNKQTYGPYGVTNGTPFSLPIENGLIVGFKGSIGYWLDYFSIYLSL 3lmk A 2.44 BS01 GLU A 1 Y64 W100 S151 S152 S173 A174 T175 Y223 D305 K396 Y40 W76 S102 S103 S124 A125 T126 Y174 D256 K339 ? 0004930,0007186,0016020 remove_due_to_license_issue P41594 506 RRVVAHMPGDIIIGALFSVHHQPTVDKVHERKCGAVREQYGIQRVEAMLHTLERINSDPTLLPNITLGCEIRDSCWHSAVALEQSIEFIRDKPIVGVIGPGSSSVAIQVQNLLQLFNIPQIAYSATSMDLSDKTLFKYFMRVVPSDAQQARAMVDIVKRYNWTYVSAVHTEGNYGESGMEAFKDMSAKEGISIAHSYKIYSNAGEQSFDKLLKKLTSHLPKARVVACFCEGMTVRGLLMAMRRLGLAGEFLLLGSDGWADRYDVTDGYQREAVGGITIKLQSPDVKWFDDYYLKLRPETNHRNPWFQEFWQHRFQCRLEGNKTCNSSLTLKTHHVQDSKMGFVINAIYSMAYGLHNMQMSLCPGYAGLCDAMKPIDGRKLLESLMKTNFTGVSGDTILFDENGDSPGRYEIMNFKEMGKDYFDYINVGSWDNGELKMD 3lmp A 1.9 BS02 CEK A 1 I262 K263 G284 C285 F287 R288 S289 L330 I341 L353 M364 K367 I56 K57 G71 C72 F74 R75 S76 L117 I128 L140 M151 K154 ? 0003677,0004879,0005634,0006355 Ki=14nM remove_due_to_license_issue P37231 20219371 23 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3lnk A 1.8 BS01 74A A 1 G72 D93 G95 Y132 T133 F169 I171 W176 Y259 D289 G291 T293 T390 G16 D37 G39 Y76 T77 F113 I115 W120 Y203 D233 G235 T237 T331 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 ic50=1150nM remove_due_to_license_issue IC50=1150nM P56817 20347593 1 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3lnq A 2.25 BS01 dna B 0 R87 R89 T90 F92 N135 K139 R1 R3 T4 F6 N49 K53 ? 0000981,0003677,0006355 remove_due_to_license_issue Q06453 20389279 1 ~ 14 RYRTTFTSFQLEELEKAFSRTHYPDVFTREELAMKIGLTEARIQVWFQNRRAKWRKQE 3lnq A 2.25 BS02 dna C 0 R87 R89 T91 Y109 Q134 R137 R141 R1 R3 T5 Y23 Q48 R51 R55 ? 0000981,0003677,0006355 remove_due_to_license_issue Q06453 20389279 1 ~ 14 RYRTTFTSFQLEELEKAFSRTHYPDVFTREELAMKIGLTEARIQVWFQNRRAKWRKQE 3lok A 2.48 BS01 DJK A 1 A293 I294 M338 C345 A390 L393 D404 A34 I35 M67 C74 A119 L122 D133 D386 R388 A390 N391 D404 D115 R117 A119 N120 D133 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>27000nM P00523 21080395 1345 KDAWEIPRESLRLEVKLGFGEVWMGTWNGTTRVAIKTLEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3loo A 2.0 BS01 B4P A 1 N14 L16 D18 G64 C122 A135 F168 T263 G265 S266 V284 L287 N296 G297 A298 G299 D300 A327 I331 N11 L13 D15 G61 C119 A132 F165 T260 G262 S263 V281 L284 N287 G288 A289 G290 D291 A318 I322 0004001,0006166,0016301 Ki=860nM remove_due_to_license_issue 21247194 349 LRDGMLVGLGNPLLDISAVVEKDLLNKYDMQPNNAILAEEKHMPMYQELIEKYQAEYIAGGSVQNSLRVAQWILQRPRTAIFFGCVGQDEYARILEERATSNGVNVQYQRSATSPTGTCAVLVTGTQRSLCANLAAANDFTPEHLRSDGNRAYLQGAQFFYVSGFFFTVSFESALSVAKEAAATGRMFMMNLSAPFVPQFYKNNLEEIFPYVDVLFGNETEAIALAKEFNYGTEDLREIGKRIAALPKENGKRKRIVIITQGSDPVLLIEAGTDNVREFPVQKLATNGAGDAFVGGFLAQLLQSRTVDVCIKCGIWAAREIIQRSGCTFEGEPSF 3lox A 2.65 BS04 MCX A 1 H57 R123 I132 L135 G137 S139 F154 R155 A156 A157 D168 H57 R123 I132 L135 G137 S139 F154 R155 A156 A157 D168 H57 D81 G137 S139 H57 D81 G137 S139 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue Q9ELS8 20303756 999 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 3lp0 A 2.79 BS03 LP7 A 1 D498 A538 H539 D496 A536 H537 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 20484498 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3lp1 A 2.23 BS01 LP8 A 1 D443 E478 D498 H539 D440 E475 D495 H536 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 20484498 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3lp2 A 2.8 BS01 LP9 A 1 V108 Y181 Q182 Y188 K223 F227 L228 W229 L234 V105 Y178 Q179 Y185 K220 F224 L225 W226 L231 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 20484498 601 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3lp4 A 1.9 BS03 LYS A 1 S137 H141 D183 T246 S132 H136 D178 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=13100nM remove_due_to_license_issue P05089 20153713 401 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 3lp7 A 2.04 BS03 HAR A 1 D124 H126 D128 N130 S137 H141 D183 T246 D119 H121 D123 N125 S132 H136 D178 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Kd=3600nM remove_due_to_license_issue P05089 20153713 906 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 3lpb A 2.0 BS01 NVB A 1 L855 G856 K857 V863 A880 M929 Y931 L932 P933 G935 L983 G993 L14 G15 K16 V22 A39 M83 Y85 L86 P87 G89 L137 G147 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=42nM remove_due_to_license_issue IC50=42nM O60674 20231096 1133 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 3lpf A 2.26 BS01 Z77 A 1 H162 D163 L361 G362 I363 E413 F448 Y472 H164 D165 L363 G364 I365 E415 F450 Y474 D163 H296 H330 V355 F357 E413 Y468 E504 K568 D165 H298 H332 V357 F359 E415 Y470 E506 K570 3.2.1.31 0004553,0004566,0005829,0005975,0016798,0030246,0032991,0042802 Ki=208nM remove_due_to_license_issue Ki=2.1e+2nM P05804 21051639 604 SHMLRPVETPTREIKKLDGLWAFSLDRENCGIDQRWWESALQESRAIAVPGSFNDQFADADIRNYAGNVWYQREVFIPKGWAGQRIVLRFDAVTHYGKVWVNNQEVMEHQGGYTPFEADVTPYVIAGKSVRITVCVNNELNWQTIPPGMVITDENGKKKQSYFHDFFNYAGIHRSVMLYTTPNTWVDDITVVTHVAQDCNHASVDWQVVANGDVSVELRDADQQVVATGQGTSGTLQVVNPHLWQPGEGYLYELCVTAKSQTECDIYPLRVGIRSVAVKGEQFLINHKPFYFTGFGRHEDADLRGKGFDNVLMVHDHALMDWIGANSYRTSHYPYAEEMLDWADEHGIVVIDETAAVGFNLSLGIGFEAGNKPKELYSEEAVNGETQQAHLQAIKELIARDKNHPSVVMWSIANEPDTRPQGAREYFAPLAEATRKLDPTRPITCVNVMFCDAHTDTISDLFDVLCLNRYYGWYVQSGDLETAEKVLEKELLAWQEKLHQPIIITEYGVDTLAGLHSMYTDMWSEEYQCAWLDMYHRVFDRVSAVVGEQVWNFADFATSQGILRVGGNKKGIFTRDRKPKSAAFLLQKRWTGMNFGEKPQQGG 3lpg A 2.425 BS01 Z78 A 1 L361 I363 M447 F448 Y472 L561 L363 I365 M449 F450 Y474 L563 D163 H296 H330 V355 F357 E413 Y468 E504 K568 D165 H298 H332 V357 F359 E415 Y470 E506 K570 3.2.1.31 0004553,0004566,0005829,0005975,0016798,0030246,0032991,0042802 remove_due_to_license_issue P05804 21051639 604 SHMLRPVETPTREIKKLDGLWAFSLDRENCGIDQRWWESALQESRAIAVPGSFNDQFADADIRNYAGNVWYQREVFIPKGWAGQRIVLRFDAVTHYGKVWVNNQEVMEHQGGYTPFEADVTPYVIAGKSVRITVCVNNELNWQTIPPGMVITDENGKKKQSYFHDFFNYAGIHRSVMLYTTPNTWVDDITVVTHVAQDCNHASVDWQVVANGDVSVELRDADQQVVATGQGTSGTLQVVNPHLWQPGEGYLYELCVTAKSQTECDIYPLRVGIRSVAVKGEQFLINHKPFYFTGFGRHEDADLRGKGFDNVLMVHDHALMDWIGANSYRTSHYPYAEEMLDWADEHGIVVIDETAAVGFNLSLGIGFEAGNKPKELYSEEAVNGETQQAHLQAIKELIARDKNHPSVVMWSIANEPDTRPQGAREYFAPLAEATRKLDPTRPITCVNVMFCDAHTDTISDLFDVLCLNRYYGWYVQSGDLETAEKVLEKELLAWQEKLHQPIIITEYGVDTLAGLHSMYTDMWSEEYQCAWLDMYHRVFDRVSAVVGEQVWNFADFATSQGILRVGGNKKGIFTRDRKPKSAAFLLQKRWTGMNFGEKPQQGG 3lpi A 2.05 BS01 Z74 A 1 G72 D93 G95 Y132 T133 Q134 F169 R189 Y259 D289 G291 T293 G15 D36 G38 Y75 T76 Q77 F112 R132 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=3nM remove_due_to_license_issue IC50=120nM, Ki=3nM P56817 20347593 456 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3lpj A 1.79 BS01 Z75 A 1 G72 D93 G95 Y132 T133 Q134 F169 Y259 D289 G291 T293 G15 D36 G38 Y75 T76 Q77 F112 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=120nM remove_due_to_license_issue IC50=120nM P56817 20347593 456 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3lpk A 1.93 BS01 Z76 A 1 G72 D93 G95 Y132 T133 Q134 G135 F169 I171 R189 Y259 D289 G291 T293 G15 D36 G38 Y75 T76 Q77 G78 F112 I114 R132 Y202 D232 G234 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=0.8nM remove_due_to_license_issue IC50=7nM, Ki=0.800000nM P56817 20347593 456 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3lpp B 2.15 BS01 KTL B 1 D231 W327 D355 W435 W470 D472 M473 K509 R555 D571 F604 H629 D202 W298 D326 W406 W441 D443 M444 K480 R526 D542 F575 H600 3.2.1.10,3.2.1.48 0003824,0004553,0005975,0030246 Ki=0.6uM remove_due_to_license_issue P14410 20356844 5001 CPNVLNDPVNVRINCIPEQFPTEGICAQRGCCWRPWNDSLIPWCFFVDNHGYNVQDMTTTSIGVEAKLNRIPSPTLFGNDINSVLFTTQNQTPNRFRFKITDPNNRRYEVPHQYVKEFTGPTVSDTLYDVKVAQNPFSIQVIRKSNGKTLFDTSIGPLVYSDQYLQISARLPSDYIYGIGEQVHKRFRHDLSWKTWPIFTRDQLPGDNNNNLYGHQTFFMCIEDTSGKSFGVFLMNSNAMEIFIQPTPIVTYRVTGGILDFYILLGDTPEQVVQQYQQLVGLPAMPAYWNLGFQLSRWNYKSLDVVKEVVRRNREAGIPFDTQVTDIDYMEDKKDFTYDQVAFNGLPQFVQDLHDHGQKYVIILDPAISIGRRANGTTYATYERGNTQHVWINESDGSTPIIGEVWPGLTVYPDFTNPNCIDWWANECSIFHQEVQYDGLWIDMNEVSSFIQGSTKGCNVNKLNYPPFTPDILDKLMYSKTICMDAVQNWGKQYDVHSLYGYSMAIATEQAVQKVFPNKRSFILTRSTFAGSGRHAAHWLGDNTASWEQMEWSITGMLEFSLFGIPLVGADICGFVAETTEELCRRWMQLGAFYPFSRNHNSDGYEHQDPAFFGQNSLLVKSSRQYLTIRYTLLPFLYTLFYKAHVFGETVARPVLHEFYEDTNSWIEDTEFLWGPALLITPVLKQGADTVSAYIPDAIWYDYESGAKRPWRKQRVDMYLPADKIGLHLRGGYIIPIQEPDVTTTASRKNPLGLIVALGENNTAKGDFFWDDGETKDTIQNGNYILYTFSVSNNTLDIVCTHSSYQEGTTLAFQTVKILGLTDSVTEVRVAENNQPMNAHSNFTYDASNQVLLIADLKLNLGRNFSVQW 3lpt A 2.0 BS01 723 A 1 T124 T125 A128 A129 T70 T71 A74 A75 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 20473303 1 DCSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGIPYNESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGYSAGERIVDIIATDIQ 3lpu A 1.95 BS01 976 A 1 T125 A128 A129 T71 A74 A75 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 20473303 1 DCSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGIPYNPSMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGYSAGERIVDIIATDIQ 3lq5 A 3.0 BS01 SLQ A 1 I25 A46 F105 C106 H108 L156 D167 I20 A39 F90 C91 H93 L141 D152 D149 K151 A153 N154 D167 T191 D134 K136 A138 N139 D152 T172 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=110nM P50750 21779453 331 DSVECPFCDEVSKYEKLAKIGQFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKGM 3lq8 A 2.02 BS01 88Z A 1 I1084 V1092 A1108 K1110 E1127 M1131 F1134 L1157 Y1159 M1160 G1163 H1202 M1211 A1221 D1222 F1223 I32 V40 A56 K58 E72 M76 F79 L98 Y100 M101 G104 H143 M152 A162 D163 F164 D1204 A1206 R1208 N1209 D1222 A1243 D145 A147 R149 N150 D163 A176 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.4nM remove_due_to_license_issue IC50=0.400000nM P08581 19808973 1 IDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRIGEVSQFLTEGIIMKDFSHPNVLSLLGICLSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDDKEYYSAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 3lrn A 2.6 BS01 rna C 0 S829 H830 H847 F853 K858 K861 I875 K888 W908 S27 H28 H45 F51 K56 K59 I73 K86 W106 3.6.4.13 remove_due_to_license_issue O95786 20637642 0 ~ 13 KENKKLLCRKCKALACYTADVRVIEESHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 3lrn B 2.6 BS01 rna D 0 S829 H830 H847 F853 K858 K861 I875 K888 W908 S27 H28 H45 F51 K56 K59 I73 K86 W106 3.6.4.13 remove_due_to_license_issue O95786 20637642 0 ~ 13 KENKKLLCRKCKALACYTADVRVIEESHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 3ls4 H 2.0 BS01 TCI H 1 V33 V35 S50 Y58 G98 T99 V102 A103 G104 V33 V35 S50 Y58 G98 T99 V102 A103 G104 remove_due_to_license_issue 20630472 220 EVKLVESGGGLVKPGGSLKLSCAASGFTFNNYVMVWLRQTPEKRLEWVASISRGGSTYYPDSVKGRFTISRDNARNILYLQMSSLRSEDTAMYYCVRGTTIVAGDVWGAGTTVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRDC 3ls4 L 2.0 BS01 TCI H 1 Y37 Q90 I95 Y37 Q90 I95 remove_due_to_license_issue 20630472 220 DIVLTQSPTTMAASPGEKITITCSASSSISSNYLHWYQQKPGFSPKLLIYRTSNLASGVPARFSGSGSGTSYSLTIGTMEAEDVATYYCQQGSSIPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 3lsp A 2.66 BS01 dna B 0 R5 S34 L35 R36 R40 Y50 R2 S31 L32 R33 R37 Y47 ? 0000976,0001217,0003677,0032993,0045892,0045922 remove_due_to_license_issue Q9HUS3 20639888 5 ~ 28 PRAEQKQQTRHALMSAARHLMESGRGFGSLSLREVTRAAGIVPAGFYRHFSDMDQLGLALVAEVDETFRATLRAVRRNEFELGGLIDASVRIFLDAVGANRSQFLFLAREQYGGSLPIRQAIASLRQRITDDLAADLALLNKMPHLDGAALDVFADLVVKTVFATLPELIDHLMPAAKITHQLRFIMIGGKHWH 3lsp A 2.66 BS02 dna D 0 R5 S34 L35 R36 R40 Y50 R2 S31 L32 R33 R37 Y47 ? 0000976,0001217,0003677,0032993,0045892,0045922 remove_due_to_license_issue Q9HUS3 20639888 5 ~ 28 PRAEQKQQTRHALMSAARHLMESGRGFGSLSLREVTRAAGIVPAGFYRHFSDMDQLGLALVAEVDETFRATLRAVRRNEFELGGLIDASVRIFLDAVGANRSQFLFLAREQYGGSLPIRQAIASLRQRITDDLAADLALLNKMPHLDGAALDVFADLVVKTVFATLPELIDHLMPAAKITHQLRFIMIGGKHWH 3lvp A 3.0 BS01 PDR A 1 L1005 G1006 Q1007 A1031 K1033 M1079 M1082 G1085 M1142 L17 G18 Q19 A43 K45 M91 M94 G97 M152 D1135 R1139 N1140 D1153 D145 R149 N150 D163 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue P08069 20545947 1 PDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMEPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3lvw A 2.5 BS01 GSH A 1 E52 E96 R196 F197 M262 C266 I317 Y362 W445 E51 E95 R195 F196 M261 C265 I316 Y361 W444 6.3.2.2 0003824,0004357,0005524,0005737,0006750,0016874,0042542,0046686 Ki=2.12mM remove_due_to_license_issue P32477 20220146 693 GLLALGTPLQWFESRTYNEHIRDEGIEQLLYIFQAAGKRDNDPLFWGDELEYMVVDFDDKERNSMLDVCHDKILTELNMEDSSLCEANDVSFHPEYGRYMLEATPASPYLNYVGSYVEVNMQKRRAIAEYKLSEYARQDSKNNLHVGSRSVPLTLTVFPRMGCPDFINIKDPWNHKNAASRSLFLPDEVINRHVRFPNLTASIRTRRGEKVCMNVPMYKDIATPETDDSIYDRDWFLPEDKEAKLASKPGFIYMDSMGFGMGCSCLQVTFQAPNINKARYLYDALVNFAPIMLAFSAAAPAFKGWLADQDVRWNVISGAVDDRTPKERGVAPLLPKYNKNGFGGIAKDVQDKVLEIPKSRYSSVDLFLGGSKFFNRTYNDTNVPINEKVLGRLLENDKAPLDYDLAKHFAHLYIRDPVSTFEELLNQDNKTSSNHFENIQSTNWQTLRFKPPTQQATPDKKDSPGWRVEFRPFEVQLLDFENAAYSVLIYLIVDSILTFSDNINAYIHMSKVWENMKIAHHRDAILFEKFHWKKSFRNDTDVETEDYSISEIFHNPENGIFPQFVTPILCQKGFVTKDWKELKHSSKHERLYYYLKLISDRASGELPTTAKFFRNFVLQHPDYKHDSKISKSINYDLLSTCDRLTHLDDSKGELTSFLGAEIAEYVKKNKPS 3lw0 A 1.79 BS01 CCX A 1 M1054 V1063 M1079 H1133 L1174 M72 V81 M97 H142 L180 D1135 R1139 N1140 D1153 E1162 D144 R148 N149 D162 E171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue P08069 24900194 1 AADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3lw0 A 1.79 BS02 CCX A 2 Y1090 K1111 Q1114 M1115 E1118 F1147 E1271 P1272 Y108 K120 Q123 M124 E127 F156 E277 P278 D1135 R1139 N1140 D1153 E1162 D144 R148 N149 D162 E171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue P08069 24900194 1287 AADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3lw0 A 1.79 BS03 CCX D 2 G1273 V1277 G279 V283 D1135 R1139 N1140 D1153 E1162 D144 R148 N149 D162 E171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue P08069 24900194 1287 AADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3lwl A 2.25 BS01 dna B 0 R487 T506 K508 T509 S513 T514 S515 A516 R536 K540 Y545 R573 N583 I584 P585 R587 V783 H784 D785 R193 T212 K214 T215 S219 T220 S221 A222 R242 K246 Y251 R279 N289 I290 P291 R293 V485 H486 D487 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20400942 101 ~ 112 EEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPRELMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3lwl A 2.25 BS02 dna C 0 N483 N485 S486 S543 T544 T569 A570 T571 S575 S576 S577 D578 N580 Y671 M673 S674 H676 R728 R746 M747 N750 Q754 N189 N191 S192 S249 T250 T275 A276 T277 S281 S282 S283 D284 N286 Y373 M375 S376 H378 R430 R448 M449 N452 Q456 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20400942 203 ~ 216 EEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPRELMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3lwm A 2.186 BS01 dna B 0 R487 T506 K508 T509 S513 T514 S515 A516 R536 K540 Y545 R573 N583 I584 P585 V586 R587 D785 R193 T212 K214 T215 S219 T220 S221 A222 R242 K246 Y251 R279 N289 I290 P291 V292 R293 D491 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20400942 101 ~ 112 EEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPREAVDPLMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3lwm A 2.186 BS02 dna C 0 N483 N485 S486 S543 T544 T569 A570 T571 S575 S576 S577 D578 N580 Y671 R728 R746 M747 N750 Q754 N189 N191 S192 S249 T250 T275 A276 T277 S281 S282 S283 D284 N286 Y377 R434 R452 M453 N456 Q460 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20400942 205 ~ 216 EEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPREAVDPLMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3lxe A 1.9 BS02 TOR A 1 Q92 H94 H96 H119 L198 T199 H200 Q88 H90 H92 H115 L194 T195 H196 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=250nM remove_due_to_license_issue Ki=250nM, IC50=250nM P00915 20505865 262 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 3lxg A 2.3 BS01 Z73 A 1 L665 V668 I682 F686 M703 Q716 F719 L213 V216 I230 F234 M251 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=7.28nM remove_due_to_license_issue Q9QYJ6 20450197 1 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIRGEE 3lxk A 2.0 BS01 MI1 A 1 G829 K830 G831 G834 S835 V836 A853 Y904 L905 R953 L956 D967 G15 K16 G17 G20 S21 V22 A39 Y90 L91 R139 L142 D153 D949 A951 R953 N954 D967 D135 A137 R139 N140 D153 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.2nM remove_due_to_license_issue IC50=55nM, Ki=0.400000nM, Kd=2.2nM P52333 20478313 1125 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 3lxl A 1.74 BS01 IZA A 1 L828 A853 M902 E903 Y904 L905 G908 L956 L15 A40 M89 E90 Y91 L92 G95 L143 D949 A951 R953 N954 D967 D136 A138 R140 N141 D154 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=5nM P52333 20478313 1 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 3lxo A 1.549 BS01 T3P A 1 Q11 H12 T45 H119 F120 Q11 H12 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Kd=15uM remove_due_to_license_issue P61823 20602460 601 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3lxs A 1.5 BS01 4MC A 1 Q19 G23 C25 S64 G65 G66 L67 L160 D161 H162 W184 E208 Q19 G23 C25 S64 G65 G66 L67 L160 D161 H162 W184 E208 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 20856868 216 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 3ly2 A 2.6 BS01 Z72 A 1 M347 D392 L393 N395 M411 M431 S442 Q443 F446 M207 D252 L253 N255 M271 M291 S302 Q303 F306 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=5nM Q07343 20378348 1000 SSGLVPRGSHMSISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 3lzb A 2.7 BS02 ITI A 1 L694 V702 A719 K721 M742 C751 L753 L764 T766 M769 P770 F771 G772 L820 T830 D831 F832 L834 L16 V24 A41 K43 M64 C73 L75 L86 T88 M91 P92 F93 G94 L142 T152 D153 F154 L156 D813 A815 R817 N818 D831 D135 A137 R139 N140 D153 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=32nM P00533 20346655 1 LLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQG 3lzi A 2.3 BS01 dna T 0 K89 R249 K251 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 N572 W574 K705 R707 K800 F803 K844 K874 K89 R249 K251 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 N572 W574 K705 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 20411947 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3lzi A 2.3 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 20411947 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3lzj A 2.05 BS01 dna T 0 K251 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 K878 K251 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 20411947 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3lzj A 2.05 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 20411947 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3lzs A 1.95 BS01 017 A 1 D25 G27 A28 D30 G48 P81 V82 I84 D25 G27 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.0109nM remove_due_to_license_issue P24740 20660190 200 PQITLWKRPLVTVKIGGQLKEALLDTGADDTVLEDINLPGKWKPKMIGGIGGFIKVRQYDQILIEICGKKAIGTVLVGPTPVNIIGRNMLTQIGCTLNF 3lzs B 1.95 BS01 017 A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P24740 20660190 200 PQITLWKRPLVTVKIGGQLKEALLDTGADDTVLEDINLPGKWKPKMIGGIGGFIKVRQYDQILIEICGKKAIGTVLVGPTPVNIIGRNMLTQIGCTLNF 3lzu A 1.76 BS01 017 A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.087nM remove_due_to_license_issue P24740 20660190 200 PQITLWKRPLVTVKIGGQLKEALLDTGADDTVLEDINLPGKWKPKMIGGIGGFIKVRQYDQILIEICGKKAIGTVLVGPTPVNIIGRSMLTQIGCTLNF 3lzu B 1.76 BS01 017 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P24740 20660190 200 PQITLWKRPLVTVKIGGQLKEALLDTGADDTVLEDINLPGKWKPKMIGGIGGFIKVRQYDQILIEICGKKAIGTVLVGPTPVNIIGRSMLTQIGCTLNF 3lzv A 2.15 BS01 017 A 1 D25 G27 A28 D29 N30 I47 G48 I50 D25 G27 A28 D29 N30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=0.026nM remove_due_to_license_issue P03369 20660190 200 PQITLWKRPLVTIRIGGQLKEALLDTGADNTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRDLLTQIGCTLNF 3lzv B 2.15 BS01 017 A 1 D25 A28 N30 P81 V82 D25 A28 N30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 20660190 200 PQITLWKRPLVTIRIGGQLKEALLDTGADNTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPVEICGHKAIGTVLVGPTPVNIIGRDLLTQIGCTLNF 3lzz A 2.5 BS01 GDP A 1 H24 P25 F31 E33 T54 I56 F140 H15 P16 F22 E24 T45 I47 F131 ? remove_due_to_license_issue Q6WRH7 173 EEVKRLIALYELTPHPASGGWFRETYRSDVQVEAEGFDGKRSVLTMIYYLMQAGQPDPFHRVKSDETFVHNLGGSMKIHMIHPDGSYSCSILGNPLEHPEARHQVVVPRRVWFAQEVDGYCLASVLVAPGFDFKDFSLGKREELIKEYPQHRDVIMRCTSS 3m11 A 2.75 BS01 AKI A 1 L139 G140 V147 A160 K162 L164 L178 E181 A213 G216 T217 D274 L14 G15 V22 A35 K37 L39 L53 E56 A88 G91 T92 D149 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=43nM O14965 20550212 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 3m1k A 1.35 BS02 BEW A 1 H94 H96 H119 T199 T200 H91 H93 H116 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=4.1uM remove_due_to_license_issue P00918 20629007 502 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3m1s A 3.134 BS01 DW1 A 1 I62 G63 F67 V70 A83 L132 D133 Y134 V135 P136 T138 R141 Q185 L188 D200 I28 G29 F33 V36 A49 L97 D98 Y99 V100 P101 T103 R106 Q150 L153 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 20821241 421 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTFFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQ 3m2u A 1.4 BS04 TXZ A 1 R270 M324 F330 F443 M480 N481 R269 M323 F329 F442 M479 N480 Q147 Y333 G445 N481 Q146 Y332 G444 N480 2.8.4.1 0005737,0015948,0016740,0046872,0050524 remove_due_to_license_issue P11558 20707311 555 ADKLFINALKKKFEESPEEKKTTFYTLGGWKQSERKTEFVNAGKEVAAKRGIPQYNPDIGTPLGQRVLMPYQVSTTDTYVEGDDLHFVNNAAMQQMWDDIRRTVIVGLNHAHAVIEKRLGKEVTPETITHYLETVNHAMPGAAVVQEHMVETHPALVADSYVKVFTGNDEIADEIDPAFVIDINKQFPEDQAETLKAEVGDGIWQVVRIPTIVSRTCDGATTSRWSAMQIGMSMISAYKQAAGEAATGDFAYAAKHAEVIHMGTYLPVRRARGENEPGGVPFGYLADICQSSRVNYEDPVRVSLDVVATGAMLYDQIWLGSYMSGGVGFTQYATAAYTDNILDDFTYFGKEYVEDKYGLCEAPNNMDTVLDVATEVTFYGLEQYEEYPALLEDQFGGSQRAAVVAAAAGCSTAFATGNAQTGLSGWYLSMYLHKEQHSRLGFYGYDLQDQCGASNVFSIRGDEGLPLELRGPNYPNYAMNVGHQGEYAGISQAPHAARGDAFVFNPLVKIAFADDNLVFDFTNVRGEFAKGALREFEPAGERALITPA 3m2u A 1.4 BS07 TXZ D 1 R225 K256 H257 R224 K255 H256 Q147 Y333 G445 N481 Q146 Y332 G444 N480 2.8.4.1 0005737,0015948,0016740,0046872,0050524 remove_due_to_license_issue P11558 20707311 556 ADKLFINALKKKFEESPEEKKTTFYTLGGWKQSERKTEFVNAGKEVAAKRGIPQYNPDIGTPLGQRVLMPYQVSTTDTYVEGDDLHFVNNAAMQQMWDDIRRTVIVGLNHAHAVIEKRLGKEVTPETITHYLETVNHAMPGAAVVQEHMVETHPALVADSYVKVFTGNDEIADEIDPAFVIDINKQFPEDQAETLKAEVGDGIWQVVRIPTIVSRTCDGATTSRWSAMQIGMSMISAYKQAAGEAATGDFAYAAKHAEVIHMGTYLPVRRARGENEPGGVPFGYLADICQSSRVNYEDPVRVSLDVVATGAMLYDQIWLGSYMSGGVGFTQYATAAYTDNILDDFTYFGKEYVEDKYGLCEAPNNMDTVLDVATEVTFYGLEQYEEYPALLEDQFGGSQRAAVVAAAAGCSTAFATGNAQTGLSGWYLSMYLHKEQHSRLGFYGYDLQDQCGASNVFSIRGDEGLPLELRGPNYPNYAMNVGHQGEYAGISQAPHAARGDAFVFNPLVKIAFADDNLVFDFTNVRGEFAKGALREFEPAGERALITPA 3m2u B 1.4 BS03 TXZ A 1 F361 F362 G369 H379 I380 F360 F361 G368 H378 I379 Y367 Y366 2.8.4.1 0005737,0015948,0016740,0050524 remove_due_to_license_issue P11560 20707311 555 AKFEDKVDLYDDRGNLVEEQVPLEALSPLRNPAIKSIVQGIKRTVAVNLEGIENALKTAKVGGPACKIMGRELDLDIVGNAESIAAAAKEMIQVTEDDDTNVELLGGGKRALVQVPSARFDVAAEYSAAPLVTATAFVQAIINEFDVSMYDANMVKAAVLGRYPQSVEYMGANIATMLDIPQKLEGPGYALRNIMVNHVVAATLKNTLQAAALSTILEQTAMFEMGDAVGAFERMHLLGLAYQGMNADNLVFDLVKANGKEGTVGSVIADLVERALEDGVIKVEKELTDYKVYGTDDLAMWNAYAAAGLMAATMVNQGAARAAQGVSSTLLYYNDLIEFETGLPSVDFGKVEGTAVGFSFFSHSIYGGGGPGIFNGNHIVTRHSKGFAIPCVAAAMALDAGTQMFSPEATSGLIKEVFSQVDEFREPLKYVVEAAAEIKNEI 3m2u D 1.4 BS03 TXZ A 1 R225 K256 H257 R224 K255 H256 Q147 Y333 G445 N481 Q146 Y332 G444 N480 2.8.4.1 0005737,0015948,0016740,0046872,0050524 remove_due_to_license_issue P11558 20707311 555 ADKLFINALKKKFEESPEEKKTTFYTLGGWKQSERKTEFVNAGKEVAAKRGIPQYNPDIGTPLGQRVLMPYQVSTTDTYVEGDDLHFVNNAAMQQMWDDIRRTVIVGLNHAHAVIEKRLGKEVTPETITHYLETVNHAMPGAAVVQEHMVETHPALVADSYVKVFTGNDEIADEIDPAFVIDINKQFPEDQAETLKAEVGDGIWQVVRIPTIVSRTCDGATTSRWSAMQIGMSMISAYKQAAGEAATGDFAYAAKHAEVIHMGTYLPVRRARGENEPGGVPFGYLADICQSSRVNYEDPVRVSLDVVATGAMLYDQIWLGSYMSGGVGFTQYATAAYTDNILDDFTYFGKEYVEDKYGLCEAPNNMDTVLDVATEVTFYGLEQYEEYPALLEDQFGGSQRAAVVAAAAGCSTAFATGNAQTGLSGWYLSMYLHKEQHSRLGFYGYDLQDQCGASNVFSIRGDEGLPLELRGPNYPNYAMNVGHQGEYAGISQAPHAARGDAFVFNPLVKIAFADDNLVFDFTNVRGEFAKGALREFEPAGERALITPA 3m2u D 1.4 BS07 TXZ D 1 R270 M324 F330 F443 M480 N481 R269 M323 F329 F442 M479 N480 Q147 Y333 G445 N481 Q146 Y332 G444 N480 2.8.4.1 0005737,0015948,0016740,0046872,0050524 remove_due_to_license_issue P11558 20707311 556 ADKLFINALKKKFEESPEEKKTTFYTLGGWKQSERKTEFVNAGKEVAAKRGIPQYNPDIGTPLGQRVLMPYQVSTTDTYVEGDDLHFVNNAAMQQMWDDIRRTVIVGLNHAHAVIEKRLGKEVTPETITHYLETVNHAMPGAAVVQEHMVETHPALVADSYVKVFTGNDEIADEIDPAFVIDINKQFPEDQAETLKAEVGDGIWQVVRIPTIVSRTCDGATTSRWSAMQIGMSMISAYKQAAGEAATGDFAYAAKHAEVIHMGTYLPVRRARGENEPGGVPFGYLADICQSSRVNYEDPVRVSLDVVATGAMLYDQIWLGSYMSGGVGFTQYATAAYTDNILDDFTYFGKEYVEDKYGLCEAPNNMDTVLDVATEVTFYGLEQYEEYPALLEDQFGGSQRAAVVAAAAGCSTAFATGNAQTGLSGWYLSMYLHKEQHSRLGFYGYDLQDQCGASNVFSIRGDEGLPLELRGPNYPNYAMNVGHQGEYAGISQAPHAARGDAFVFNPLVKIAFADDNLVFDFTNVRGEFAKGALREFEPAGERALITPA 3m2w A 2.41 BS01 L8I A 1 L70 L72 A91 K93 M138 C140 L141 D142 L193 D207 L24 L26 A45 K47 M92 C94 L95 D96 L147 D161 D186 K188 N191 D207 D140 K142 N145 D161 2.7.11.1 0004672,0005524,0006468 ic50<0.003uM remove_due_to_license_issue IC50=<3nM P49137 20591669 1 HVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTGEKYDKSCDMWSLGVIMYILLCGYPPFYSPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR 3m35 A 2.2 BS01 M35 A 1 N97 T98 D189 S190 C191 Q192 V213 W215 G216 G219 N79 T80 D171 S172 C173 Q174 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue Ki=60nM P00760 14640539 301 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3m36 A 2.15 BS01 M35 A 1 E97 T98 Y99 R143 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G218 C220 E83 T84 Y85 R132 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=0.15nM, IC50=2.4nM P00742 14640539 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3m37 A 1.9 BS01 M37 A 1 K96 E97 T98 Y99 E146 F174 A190 C191 Q192 S195 W215 G216 G218 C220 K82 E83 T84 Y85 E135 F162 A180 C181 Q182 S185 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=0.910nM P00742 14640539 301 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 3m3c A 2.0 BS01 GAL C 1 P42 N43 H59 R63 W80 E83 P43 N44 H60 R64 W81 E84 3.1.21.- 0004518,0004536,0006259,0006915,0030246,0030247,0043065 remove_due_to_license_issue Q6WY08 20530247 2 MQGVNIYNISAGTSVDLAAPVTTGDIVTFFSSALNLNAGAGNPNNTTLNLFAENGAYLLHIAFRLQENVIIFNSRQPDGPWLVEQRVSDVANQFAGIDGKAMVTVFDHGDKYQVVINEKTVIQYTKQISGLTSSLSYNATEETSIFSTVVEAVTYTGLA 3m3e A 2.1 BS01 GAL E 1 N43 H59 R63 N72 W80 E83 N44 H60 R64 N73 W81 E84 3.1.21.- 0004518,0004536,0006259,0006915,0030246,0030247,0043065 remove_due_to_license_issue Q6WY08 20530247 2 MQGVNIYNISAGTSVDLAAPVTTGDIVTFFSSALNLNAGAGNPNNTTLNLFAENGAYLLHIAFRLQANVIIFNSRQPDGPWLVEQRVSDVANQFAGIDGKAMVTVFDHGDKYQVVINEKTVIQYTKQISGLTSSLSYNATEETSIFSTVVEAVTYTGLA 3m3o A 2.1 BS01 GAL B 1 N43 H59 R63 W80 E83 N43 H59 R63 W80 E83 3.1.21.- 0004518,0004536,0006259,0006915,0030246,0030247,0043065 remove_due_to_license_issue Q6WY08 20530247 2 QGVNIYNISAGTSVDLAAPVTTGDIVTFFSSALNLNAGAGNPNNTTLNLFAENGAYLLHIAFRLQENVIIFNSRQPDGPWLVEQAVSDVANQFAGIDGKAMVTVFDHGDKYQVVINEKTVIQYTKQISGLTSSLSYNATEETSIFSTVVEAVTYTGLA 3m3x A 1.68 BS02 JS7 A 1 H94 H96 H119 F131 V135 L198 T199 T200 P202 H92 H94 H117 F128 V132 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.15uM remove_due_to_license_issue Kd=150nM P00918 20889345 264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3m3z A 2.1 BS01 3F5 A 1 Y15 G202 G230 E268 K271 R272 S275 G339 S340 R342 Y11 G198 G226 E264 K267 R268 S271 G335 S336 R338 D10 K71 E175 D199 D6 K67 E171 D195 3.6.4.10 0005524,0140662 Kd=12.36uM remove_due_to_license_issue P11142 21526763 401 PAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 3m40 A 1.6 BS02 J45 A 1 Q92 H94 H96 H119 F131 L198 T199 T200 Q90 H92 H94 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.17uM remove_due_to_license_issue Kd=90nM P00918 20889345 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3m5e A 1.7 BS02 JDR A 1 Q92 H94 H96 H119 F131 L198 T199 T200 Q90 H92 H94 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.043uM remove_due_to_license_issue Kd=24nM P00918 20889345 264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3m67 A 1.8 BS01 E36 A 1 H94 H119 V121 L198 T199 T200 P202 H91 H116 V118 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.18uM remove_due_to_license_issue Kd=20nM P00918 20926301 262 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3m6f A 1.85 BS01 BJZ A 1 V157 Y166 T231 I235 Y257 I259 K287 L302 I306 V30 Y39 T104 I108 Y130 I132 K160 L175 I179 ? remove_due_to_license_issue IC50=60nM P20701 20405922 1 MNVDLVFLFDGSMSLQPDEFQKILDFMKDVMKKLSNTSYQFAAVQFSTSYKTEFDFSDYVKRKDPDALLKHVKHMLLLTNTFGAINYVATEVFREELGARPDATKVLIIITDGEATDSGNIDAAKDIIRYIIGIGKHFQTKESQETLHKFASKPASEFVKILDTFEKLKDLFTELQKKIY 3m6p A 2.0 BS01 BB2 A 1 G41 I42 G43 Q48 F87 D88 G90 C91 L92 Y98 H133 E134 H137 G41 I42 G43 Q48 F87 D88 G90 C91 L92 Y98 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 3.5.1.88 0042586 Ki=0.9nM remove_due_to_license_issue Q9FUZ2 21629676 194 MEIVEYPDPILRAKNKRIDIFDENLKNLVDAMFDVMYKTDGIGLSAPQVGLNVQLMVFNPAGEPGEGKEIVLVNPKIKKYSDKLVPFDEGCLSFPGIYAEVVRPQSVKIDARDITGERFSISLSRLPARIFQHEYDHLEGVLFFDRMTDQVLDSIREELEALEKKYEEKTGLPSPERVEA 3m6q A 2.4 BS01 BB2 A 1 Q41 I42 G43 Q48 D88 G90 C91 L92 I130 H133 E134 H137 Q41 I42 G43 Q48 D88 G90 C91 L92 I130 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 3.5.1.88 0042586 Kd=48nM remove_due_to_license_issue Q9FUZ2 21629676 194 MEIVEYPDPILRAKNKRIDIFDENLKNLVDAMFDVMYKTDQIGLSAPQVGLNVQLMVFNPAGEPGEGKEIVLVNPKIKKYSDKLVPFDEGCLSFPGIYAEVVRPQSVKIDARDITGERFSISLSRLPARIFQHEYDHLEGVLFFDRMTDQVLDSIREELEALEKKYEEKTGLPSPERVEAR 3m6r A 2.4 BS01 BB2 A 1 M41 I42 G43 Q48 D88 E89 G90 C91 H133 E134 H137 M41 I42 G43 Q48 D88 E89 G90 C91 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 3.5.1.88 0042586 Kd=32nM remove_due_to_license_issue Q9FUZ2 21629676 194 MEIVEYPDPILRAKNKRIDIFDENLKNLVDAMFDVMYKTDMIGLSAPQVGLNVQLMVFNPAGEPGEGKEIVLVNPKIKKYSDKLVPFDEGCLSFPGIYAEVVRPQSVKIDARDITGERFSISLSRLPARIFQHEYDHLEGVLFFDRMTDQVLDSIREELEALEKKYEEKTGLPSPERVEA 3m89 A 2.0 BS01 GSP A 1 G31 Q32 K33 G139 G140 V141 E175 N213 K237 N241 G31 Q32 K33 G128 G129 V130 E164 N202 K226 N230 3.6.5.- Kd=0.69uM remove_due_to_license_issue Q8KNP3 20534443 408 MLLNSNELEHIHSTNHSVNDISIRWGVIGAGQKGNKEADLFAGYKFSNGTTCYPTLAVNFAESDMMHLQNIIKEDRIHFVVTDLFDPETNPNANGYLDKLAQELGRKFTNEEGEVIVDQFLICLGAGGGVGTGWGSLVLQLIREQFFPCPVSMLISLPSGDPDEINNALVLLSEIDEFMREQDRLFGNSDIKPLANVIVNDNTQMQRIIESQKGTKDLKNRYVNWKEVANDNVVSTLHEINIIPENYGSDNVTYDPSDLIKLLSIPGRFLTIGKARIAKFDLHSLENSIKRSLDEGFFSAEHQFETATMYGGFVLRPSNADFFKDVNTENRIRNTLGEYKRLDEIAGKFGDPIWDNEYAVCYTIFAGMTMPKRYISLAREGKELAEKQEQLRA 3m8p A 2.67 BS01 65B A 1 L100 K101 K103 V106 V179 Y181 Y188 F227 W229 L234 H235 P236 Y318 L96 K97 K99 V102 V175 Y177 Y184 F223 W225 L230 H231 P232 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 20538456 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAG 3m8q A 2.7 BS01 DJZ A 1 L100 K101 K103 K104 S105 V106 V179 Y181 Y188 F227 W229 L234 H235 Y318 L97 K98 K100 K101 S102 V103 V176 Y178 Y185 F224 W226 L231 H232 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 20538456 562 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3m8r A 2.0 BS01 dna B 0 R487 T506 K508 T509 S513 T514 S515 A516 R536 K540 Y545 R573 N583 I584 P585 R587 R660 V783 H784 R194 T213 K215 T216 S220 T221 S222 A223 R243 K247 Y252 R280 N290 I291 P292 R294 R367 V490 H491 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20572212 101 ~ 112 LEEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPREAVDPLMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3m8r A 2.0 BS02 dna C 0 N483 N485 S486 I503 S513 S515 A517 S543 T544 T569 A570 T571 R573 S575 S576 S577 D578 N580 F667 G668 Y671 G672 M673 S674 H676 R677 Q680 R728 R746 M747 N750 Q754 N190 N192 S193 I210 S220 S222 A224 S250 T251 T276 A277 T278 R280 S282 S283 S284 D285 N287 F374 G375 Y378 G379 M380 S381 H383 R384 Q387 R435 R453 M454 N457 Q461 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20572212 201 ~ 216 LEEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPREAVDPLMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3m8s A 2.2 BS01 dna B 0 R487 T506 K508 T509 S513 T514 S515 A516 R536 K540 Y545 R573 N583 I584 P585 R587 R660 V783 H784 R194 T213 K215 T216 S220 T221 S222 A223 R243 K247 Y252 R280 N290 I291 P292 R294 R367 V490 H491 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20572212 101 ~ 112 LEEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPREAVDPLMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3m8s A 2.2 BS02 dna C 0 N483 N485 S486 I503 S515 A517 S543 T544 T569 A570 T571 R573 S575 S576 S577 D578 N580 F667 G668 Y671 G672 M673 S674 H676 R677 Q680 R728 R746 M747 N750 Q754 N190 N192 S193 I210 S222 A224 S250 T251 T276 A277 T278 R280 S282 S283 S284 D285 N287 F374 G375 Y378 G379 M380 S381 H383 R384 Q387 R435 R453 M454 N457 Q461 2.7.7.7 0001882,0003676,0003677,0003887,0006260,0006261,0006281 remove_due_to_license_issue P19821 20572212 201 ~ 216 LEEAPWPPPEGAFVGFVLSRKEPMWADLLALAAARGGRVHRAPEPYKALRDLKEARGLLAKDLSVLALREGLGLPPGDDPMLLAYLLDPSNTTPEGVARRYGGEWTEEAGERAALSERLFANLWGRLEGEERLLWLYREVERPLSAVLAHMEATGVRLDVAYLRALSLEVAEEIARLEAEVFRLAGHPFNLNSRDQLERVLFDELGLPAIGKTEKTGKRSTSAAVLEALREAHPIVEKILQYRELTKLKSTYIDPLPDLIHPRTGRLHTRFNQTATATGRLSSSDPNLQNIPVRTPLGQRIRRAFIAEEGWLLVALDYSQIELRVLAHLSGDENLIRVFQEGRDIHTETASWMFGVPREAVDPLMRRAAKTINFGVLYGMSAHRLSQELAIPYEEAQAFIERYFQSFPKVRAWIEKTLEEGRRRGYVETLFGRRRYVPDLEARVKSVREAAERMAFNMPVQGTAADLMKLAMVKLFPRLEEMGARMLLQVHDELVLEAPKERAEAVARLAKEVMEGVYPLAVPLEVEVGIGEDWLSAKE 3m8u A 1.85 BS01 GDS A 1 R33 D45 G46 I47 F263 R379 A380 S381 G428 W429 S430 D432 N503 F504 Q516 F519 G520 Y521 R10 D22 G23 I24 F240 R356 A357 S358 G405 W406 S407 D409 N480 F481 Q493 F496 G497 Y498 ? 0030288,0042938,0043190,0055085,1904680 Kd=12.9uM remove_due_to_license_issue B8F653 20628015 1 DKTFINCVSRSPTGFSPALVMDGISYNASSQQVYNRLVEFKRGSTDIEPALAESWTVSDDGLTYTFNLRKGVKFHSNKEFTPSRDFNADDVVFSFQRQLDPNHPYHNVSKATYPYFKAMKFSTLLKSVEKVDMHTVKITLNRQDATFLASLGMDFISIYSAEYADKMLAAGKPETIDTTPIGTGPFLFAGYQVDQKSRYLAHKEYWKGKADIDRLIFEIVPDATARYAKLQAGACDLIDFPNAADLEKMKTDPKVNLHSQSGLNIAYIAFNTEKAPFDNVKVRQALNYAVDKNAIIDAVYRGAGVAAKNPLPPTIWGYNNEITGYEYSPEKAKQLLKEAGFENGFETDIWVQPVVRASNPNPRRMAELVQSDWEKVGVKSKLVSYEWGDYIKRTKAGELTAGTYGWSGDNGDPDNFLSPLFGSENVGNSNYARFKNPELDALLHKAVGLSDKAERAKIYEQAQVLLKEQAPWINVAHSINFAPTSKRVQDYKQSPFGYTYLYGTKLAD 3m93 A 2.9 BS02 M7G A 1 W69 M114 W115 E116 R170 W22 M67 W68 E69 R123 ? 0003723,0003743,0005737,0006413 remove_due_to_license_issue Q6PKX2 21965542 1 MRHPLQCHWALWYLKADRSKDWEDCLKQVAVFDTVEDFWSLYNHIQAASGLTWGSDYYLFKEGIKPMWEDENNVKGGRWLVVVDKQKRAQLLDHYWLELLMAIIGEQFEDNGEYICGAVVNVRQKGDKVSLWTRDSLKDDVNLRIGQILKAKLEIPDTEPIRYEVHTGSMVKPRIVIPSK 3m94 A 2.05 BS02 M7M A 1 W69 M114 W115 E116 N168 R170 K175 W22 M67 W68 E69 N121 R123 K128 ? 0003723,0003743,0005737,0006413 remove_due_to_license_issue Q6PKX2 21965542 1 MRHPLQCHWALWYLKADRSKDWEDCLKQVAVFDTVEDFWSLYNHIQAASGLTWGSDYYLFKEGIKPMWEDENNVKGGRWLVVVDKQKRAQLLDHYWLELLMAIIGEQFEDNGEYICGAVVNVRQKGDKVSLWTRDSLKDDVNLRIGQILKAKLEIPDTEPIRYEVHKTGSMVKPRIVIPS 3m96 A 1.4 BS02 E38 A 1 H94 H96 H119 V121 L198 T199 T200 P202 H91 H93 H116 V118 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.06uM remove_due_to_license_issue P00918 20926301 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3m9e A 2.406 BS01 dna C 0 Y116 H117 Y118 R131 L177 V178 L179 R184 K187 R188 Y13 H14 Y15 R28 L74 V75 L76 R81 K84 R85 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRREELQ 3m9e A 2.406 BS02 dna D 0 E124 R132 R157 N158 Q161 R164 L190 N194 R195 E21 R29 R54 N55 Q58 R61 L87 N91 R92 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRREELQ 3m9e B 2.406 BS01 dna C 0 E124 G125 F129 R132 R157 N158 Q161 R164 I191 N194 R195 E21 G22 F26 R29 R54 N55 Q58 R61 I88 N91 R92 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRREE 3m9e B 2.406 BS02 dna D 0 H117 Y118 K127 R131 L177 V178 L179 R184 K187 R188 H14 Y15 K24 R28 L74 V75 L76 R81 K84 R85 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRREE 3m9e E 2.406 BS01 dna G 0 H117 Y118 R131 L177 V178 L179 R184 K187 H14 Y15 R28 L74 V75 L76 R81 K84 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRREELQK 3m9e E 2.406 BS02 dna H 0 E124 G125 R132 R157 N158 Q161 R164 L190 N194 R195 E21 G22 R29 R54 N55 Q58 R61 L87 N91 R92 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRREELQK 3m9e F 2.406 BS01 dna G 0 E124 G125 F129 R132 R157 N158 Q161 R164 E21 G22 F26 R29 R54 N55 Q58 R61 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRR 3m9e F 2.406 BS02 dna H 0 Y116 H117 Y118 K127 R131 V178 L179 Y13 H14 Y15 K24 R28 V75 L76 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue P18113 20610536 1 ~ 22 ELCVVCGDKATGYHYRCITCEGCKGFFRRTIQKSLHPSYSCKYEGKCIIDKVTRNQCQECRFKKCIYVGMATDLVLDDSKRLAKRKLIEENREKRRR 3m9f A 1.8 BS01 595 A 1 D25 G27 A28 D29 G48 G49 I50 V82 D25 G27 A28 D29 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.007nM remove_due_to_license_issue Q9WFL7 20547452 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3m9f A 1.8 BS02 595 B 1 R8 L23 D25 G27 A28 G48 G49 I50 V82 I84 R8 L23 D25 G27 A28 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.007nM remove_due_to_license_issue Q9WFL7 20547452 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3m9f B 1.8 BS01 595 A 1 D25 G27 A28 G48 G49 I50 P81 I84 D25 G27 A28 G48 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.007nM remove_due_to_license_issue Q9WFL7 20547452 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3m9f B 1.8 BS02 595 B 1 D25 G27 A28 D29 G48 G49 I50 P81 V82 I84 D25 G27 A28 D29 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.007nM remove_due_to_license_issue Q9WFL7 20547452 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3ma3 A 2.3 BS02 01I A 1 A65 K67 V126 L174 I185 D186 A27 K29 V88 L136 I147 D148 D167 K169 N172 D186 L193 T204 D129 K131 N134 D148 L155 T166 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=60nM remove_due_to_license_issue P11309 20400536 313 QYQVGPLLGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3mag A 1.8 BS02 3MA A 1 Y22 F180 Y22 F174 2.1.1.57 0003723,0003746,0004483,0006370,0008168,0031440,0032259,0044423 Kd=86uM remove_due_to_license_issue P07617 10377383 600 MDVVSLDKPFMYFEEIDNELDYEPESANEVAKKLPYQGQLKLLLGELFFLSKLQRHGILDGATVVYIGSAPGTHIRYLRDHFYNLGVIIKWMLIDGRHHDPILNGLRDVTLVTRFVDEEYLRSIKKQLHPSKIILISDVRSPSTADLLSNYALQNVMISILNPVASSLKWRCPFPDQWIKDFYIPHGNKMLQPFAPSYSAEMRLLSIYTGENMRLTRVTKSDAVNYEKKMYYLNKIVRNKVVVNFDYPNQEYDYFHMYFMLRTVYCNKTFPTTKAKVLFLQQSIFRFLNIP 3max A 2.05 BS03 LLX A 1 M35 R39 L144 H145 H146 G154 F155 C156 D181 H183 F210 L276 G305 G306 Y308 M24 R28 L133 H134 H135 G143 F144 C145 D170 H172 F199 L265 G294 G295 Y297 3.5.1.-,3.5.1.98 0004407 ic50=0.027uM remove_due_to_license_issue IC50=900nM Q92769 20392638 400 AKKKVCYYYDGDIGNYYYGQGHPMKPHRIRMTHNLLLNYGLYRKMEIYRPHKATAEEMTKYHSDEYIKFLRSIRPDNMSEYSKQMQRFNVGEDCPVFDGLFEFCQLSTGGSVAGAVKLNRQQTDMAVNWAGGLHHAKKSEASGFCYVNDIVLAILELLKYHQRVLYIDIDIHHGDGVEEAFYTTDRVMTVSFHKYGEYFPGTGDLRDIGAGKGKYYAVNFPMRDGIDDESYGQIFKPIISKVMEMYQPSAVVLQCGADSLSGDRLGCFNLTVKGHAKCVEVVKTFNLPLLMLGGGGYTIRNVARCWTYETAVALDCEIPNELPYNDYFEYFGPDFKLHISPSNMTNQNTPEYMEKIKQRLFENLRML 3mb6 A 1.75 BS01 01I A 1 L45 V66 K68 F113 M163 I174 D175 L43 V64 K66 F111 M161 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 ic50=100nM remove_due_to_license_issue P68400 20400536 332 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 3mb7 A 1.65 BS01 14I A 1 L45 V53 V66 K68 V116 N118 M163 I174 L44 V52 V65 K67 V115 N117 M162 I173 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 ic50=200nM remove_due_to_license_issue P68400 20400536 332 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 3mbl A 2.6 BS03 LSG A 1 N78 K97 V127 I141 M143 D208 F209 G210 V211 S212 L215 I216 N18 K37 V67 I81 M83 D148 F149 G150 V151 S152 L155 I156 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T166 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=18nM Q02750 20621728 7 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL 3mbz A 2.6 BS01 MXC A 1 S81 K84 Y112 S128 V130 S219 W221 R261 S50 K53 Y81 S97 V99 S188 W190 R230 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 20822105 276 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 3mct A 2.0 BS02 3MC A 1 Y22 F180 E233 Y22 F174 E227 2.1.1.57 0003746,0004483,0006370,0031440 Kd=85.5uM remove_due_to_license_issue P07617 10377383 600 MDVVSLDKPFMYFEEIDNELDYEPESANEVAKKLPYQGQLKLLLGELFFLSKLQRHGILDGATVVYIGSAPGTHIRYLRDHFYNLGVIIKWMLIDGRHHDPILNGLRDVTLVTRFVDEEYLRSIKKQLHPSKIILISDVRSPSTADLLSNYALQNVMISILNPVASSLKWRCPFPDQWIKDFYIPHGNKMLQPFAPSYSAEMRLLSIYTGENMRLTRVTKSDAVNYEKKMYYLNKIVRNKVVVNFDYPNQEYDYFHMYFMLRTVYCNKTFPTTKAKVLFLQQSIFRFLNIP 3mdz A 2.32 BS02 EZL A 1 H96 V123 L200 T201 T202 H93 V120 L197 T198 T199 H66 H96 H98 E108 H121 T201 H63 H93 H95 E105 H118 T198 4.2.1.1 0004089,0005737,0005829,0006730,0008270,0016829,0032230,0032849,0046872,0051453,0070050,2001225 remove_due_to_license_issue Ki=0.8nM, Kd=0.710000nM P43166 264 MHGWGYGQDDGPSHWHKLYPIAQGDRQSPINIISSQAVYSPSLQPLELSYEACMSLSITNNGHSVQVDFNDSDDRTVVTGGPLEGPYRLKQFHFHWGKKHDVGSEHTVDGKSFPSELHLVHWNAKKYSTFGEAASAPDGLAVVGVFLETGDEHPSMNRLTDALYMVRFKGTKAQFSCFNPKCLLPASRHYWTYPGSLTTPPLSESVTWIVLREPICISERQMGKFRSLLFTSEDDERIHMVNNFRPPQPLKGRVVKASF 3mf5 A 2.0 BS01 HJZ A 1 L419 R422 M423 S476 Y477 I482 L497 R501 W528 L414 R417 M418 S471 Y472 I477 L492 R496 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.042uM remove_due_to_license_issue P26663 20584604 571 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 3mfv A 1.9 BS03 Z70 A 1 H126 D128 S137 H141 D183 T246 H121 D123 S132 H136 D178 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Ki=3000uM remove_due_to_license_issue Ki=3000000nM P05089 20441173 0 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 3mfw A 1.47 BS01 B3U A 1 H126 D128 N130 S137 H141 G142 D183 T246 H122 D124 N126 S133 H137 G138 D179 T242 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 Ki=300uM remove_due_to_license_issue Ki=300000nM P05089 20441173 600 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 3mg0 H 2.68 BS01 BO2 H 1 T1 S20 T21 Q22 K33 A46 G47 A49 T1 S20 T21 Q22 K33 A46 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 20632995 1400 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 3mg0 I 2.68 BS01 BO2 H 1 D114 C118 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 20632995 1400 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 3mg4 K 3.11 BS02 LXT K 1 A20 T21 V31 M45 G47 G48 A49 A20 T21 V31 M45 G47 G48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20632995 213 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3mg4 L 3.11 BS02 LXT K 1 D114 P115 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20632995 213 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3mg6 K 2.6 BS02 LZT K 1 A20 T21 V31 K33 M45 G47 G48 A49 S96 A20 T21 V31 K33 M45 G47 G48 A49 S96 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20632995 213 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3mg6 L 2.6 BS01 LZT K 1 P94 Y96 D114 P104 Y106 D126 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20632995 213 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3mg7 K 2.78 BS02 L2T K 1 A20 T21 V31 K33 M45 A46 G47 G48 A49 S96 A20 T21 V31 K33 M45 A46 G47 G48 A49 S96 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20632995 213 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3mg7 L 2.78 BS01 L2T K 1 Y-5 P94 Y96 D114 P115 Y5 P104 Y106 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20632995 213 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3mg8 K 2.59 BS02 L3T K 1 A20 T21 V31 K33 M45 A46 G47 A49 A20 T21 V31 K33 M45 A46 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20632995 213 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3mg8 L 2.59 BS01 L3T K 1 Y96 D114 P115 S118 Y119 Y106 D126 P127 S130 Y131 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20632995 213 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3mhc A 1.698 BS02 ARZ A 1 Q92 H94 H119 F131 L198 T199 T200 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11nM remove_due_to_license_issue Ki=10nM P00918 20605094 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mhi A 1.7 BS02 J90 A 1 H94 H119 V121 L198 T199 T200 P202 H91 H116 V118 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.2uM remove_due_to_license_issue Kd=200nM P00918 20889345 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mhi A 1.7 BS03 J90 A 2 H4 W5 H10 N11 H15 W16 D19 H1 W2 H7 N8 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.2uM remove_due_to_license_issue Kd=200nM P00918 20889345 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mhl A 1.9 BS02 J71 A 1 I91 Q92 H94 H119 F131 L198 T199 T200 I88 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.056uM remove_due_to_license_issue Kd=56nM P00918 20889345 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mhm A 1.5 BS02 J75 A 1 I91 Q92 H94 H96 H119 D130 F131 G132 L198 T199 T200 I88 Q89 H91 H93 H116 D126 F127 G128 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.1uM remove_due_to_license_issue Kd=100nM P00918 20889345 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mho A 1.15 BS02 J43 A 1 W5 H94 H96 H119 F131 L198 T199 T200 P202 W2 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.32uM remove_due_to_license_issue Kd=320nM P00918 20889345 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3mhw U 1.45 BS01 ABV U 1 D189 S190 C191 Q192 W215 G219 G226 D191 S192 C193 Q194 W217 G220 G228 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 245 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADLAHHNDIALLKIRSKEGRCAQPSRTIQTISLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 3mi2 A 1.2 BS01 PFU A 1 S68 D70 K92 H94 K125 M182 S183 P228 Q241 Y243 G261 R262 S35 D37 K59 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 Ki=0.00000079M remove_due_to_license_issue Ki=17nM P11172 20452222 1 KELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3mi2 A 1.2 BS02 PFU B 1 D128 I129 T132 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 Ki=0.00000079M remove_due_to_license_issue Ki=17nM P11172 20452222 1 KELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3mi2 B 1.2 BS01 PFU A 1 D128 I129 T132 D95 I96 T99 2.4.2.10,4.1.1.23 0004590,0006207,0044205 Ki=0.00000079M remove_due_to_license_issue Ki=17nM P11172 20452222 1 KELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3mi2 B 1.2 BS02 PFU B 1 S68 D70 K92 H94 K125 M182 S183 P228 Q241 Y243 G261 R262 S35 D37 K59 H61 K92 M149 S150 P195 Q208 Y210 G228 R229 2.4.2.10,4.1.1.23 0004590,0006207,0044205 Ki=0.00000079M remove_due_to_license_issue Ki=17nM P11172 20452222 1 KELSFGARAELPRIHPVASKLLRLMQKKETNLCLSADVSLARELLQLADALGPSICMLKTHVDILNDFTLDVMKELITLAKCHEFLIFEDRKFADIGNTVKKQYEGGIFKIASWADLVNAHVVPGSGVVKGLQEVGLPLHRGCLLIAEMSSTGSLATGDYTRAAVRMAEEHSEFVVGFISGSRVSMKPEFLHLTPGVQLEAGGDNLGQQYNSPQEVIGKRGSDIIIVGRGIISAADRLEAAEMYRKAAWEAYLSRLG 3mi3 A 2.38 BS01 LYS A 1 R43 D123 T197 H224 H226 R20 D100 T163 H190 H192 Q47 Q24 2.3.3.14 0003824,0004410,0005634,0005739,0005759,0005829,0009085,0016740,0019752,0019878,0044283,0046872,0046912 Ki=3.56uM remove_due_to_license_issue Q9Y823 20089861 1000 NPSDFLSRVNNFSIIESTLREGEQFANAFFDTEKKIQIAKALDNFGVDYIELTSPVASEQSRQDCEAICKLGLKCKILTHIRCHMDDARVAVETGVDGVDVVIGTSMTYIIDSATEVINFVKSKGIEVRFSSEDSFRSDLVDLLSLYKAVDKIGVNRVGIADTVGCATPRQVYDLIRTLRGVVSCDIECHFHNDTGMAIANAYCALEAGATHIDTSILGIGERNGITPLGALLARMYVTDREYITHKYKLNQLRELENLVADAVEVQIPFNNYITGMCAFTHKAGIHAKAILANPSTYEILKPEDFGMSRYVHVGSRLTGWNAIKSRAEQLNLHLTDAQAKELTVRIKKLADVRTLAMDDVDRVLREYHA 3mi3 B 2.38 BS01 LYS B 1 R43 D123 T197 H224 H226 R20 D100 T161 H188 H190 Q47 Q24 2.3.3.14 0003824,0004410,0005634,0005739,0005759,0005829,0009085,0016740,0019752,0019878,0044283,0046872,0046912 Ki=3.56uM remove_due_to_license_issue Q9Y823 20089861 1000 NPSDFLSRVNNFSIIESTLREGEQFANAFFDTEKKIQIAKALDNFGVDYIELTSPVASEQSRQDCEAICKLGLKCKILTHIRCHMDDARVAVETGVDGVDVVIGMTYIIDSATEVINFVKSKGIEVRFSSEDSFRSDLVDLLSLYKAVDKIGVNRVGIADTVGCATPRQVYDLIRTLRGVVSCDIECHFHNDTGMAIANAYCALEAGATHIDTSILGIGERNGITPLGALLARMYVTDREYITHKYKLNQLRELENLVADAVEVQIPFNNYITGMCAFTHKAGIHAKAILANPSTYEILKPEDFGMSRYVHVGSRLTGWNAIKSRAEQLNLHLTDAQAKELTVRIKKLADVRTLAMDDVDRVLREYHAD 3miy A 1.67 BS01 B49 A 1 I369 A389 K391 F435 F437 M438 E439 H440 G441 L489 I15 A33 K35 F74 F76 M77 E78 H79 G80 L128 D482 A484 R486 N487 D500 P521 D121 A123 R125 N126 D139 P141 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=21nM remove_due_to_license_issue Kd=13nM Q08881 20545945 1 GSVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTISEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEASVIHRDLAARNCLVGENQVIKVSDFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAAIAASG 3mj1 A 1.72 BS01 614 A 1 I369 S371 A389 E436 F437 M438 E439 H440 G441 C442 L489 I15 S17 A33 E69 F70 M71 E72 H73 G74 C75 L122 D482 A484 R486 N487 D500 P521 D115 A117 R119 N120 D133 P135 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=15nM remove_due_to_license_issue Q08881 20545945 1 GSVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEASVIHRDLAARNCLVGENQVIKVSDFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYERSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAAI 3mj2 A 1.9 BS01 MJG A 1 I369 S371 V377 A389 K391 F435 M438 E439 G441 N487 L489 S499 I13 S15 V21 A33 K35 F79 M82 E83 G85 N131 L133 S143 D482 A484 R486 N487 D500 P521 D126 A128 R130 N131 D144 P165 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=15nM remove_due_to_license_issue IC50=19nM, Ki=16nM Q08881 20545945 1 VIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEASVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAAI 3mj5 A 2.63 BS01 GRM A 1 L163 G164 D165 P248 P249 Y269 Q270 Y274 L160 G161 D162 P245 P246 Y266 Q267 Y271 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0006508,0008234 remove_due_to_license_issue IC50=320nM P0C6U8 20527968 801 KTIKVFTTVDNTNLHTQLVDMSMTYGQQFGPTYLDGADVTKIKPHVNHEGKTFFVLPSDDTLRSEAFEYYHTLDESFLGRYMSALNHTKKWKFPQVGGLTSIKWADNNCYLSSVLLALQQLEVKFNAPALQEAYYRARAGDAANFCALILAYSNKTVGELGDVRETMTHLLQHANLESAKRVLNVVCKHCGQKTTTLTGVEAVMYMGTLSYDNLKTGVSIPCVCGRDATQYLVQQESSFVMMSAPPAEYKLQQGTFLCANEYTGNYQCGHYTHITAKETLYRIDGAHLTKMSEYKGPVTDVFYKETSYTTTI 3mj5 A 2.63 BS03 GRM B 1 M209 G210 P248 Y269 M206 G207 P245 Y266 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0006508,0008234 remove_due_to_license_issue IC50=320nM P0C6U8 20527968 801 KTIKVFTTVDNTNLHTQLVDMSMTYGQQFGPTYLDGADVTKIKPHVNHEGKTFFVLPSDDTLRSEAFEYYHTLDESFLGRYMSALNHTKKWKFPQVGGLTSIKWADNNCYLSSVLLALQQLEVKFNAPALQEAYYRARAGDAANFCALILAYSNKTVGELGDVRETMTHLLQHANLESAKRVLNVVCKHCGQKTTTLTGVEAVMYMGTLSYDNLKTGVSIPCVCGRDATQYLVQQESSFVMMSAPPAEYKLQQGTFLCANEYTGNYQCGHYTHITAKETLYRIDGAHLTKMSEYKGPVTDVFYKETSYTTTI 3mjl A 1.9 BS03 2AI A 1 H126 D128 T246 H121 D123 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue Ki=3600000nM P05089 5001 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 3mke A 1.75 BS03 CB4 A 1 M69 S70 D104 Y105 S130 N132 E166 N170 T235 G236 A237 M44 S45 D79 Y80 S105 N107 E141 N145 T210 G211 A212 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Ki=2200nM P0AD64 21041505 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3mkf A 1.33 BS01 CZ7 A 1 M69 S70 Y105 N132 E166 T167 N170 G236 A237 E240 M44 S45 Y80 N107 E141 T142 N145 G211 A212 E214 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 21041505 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3mkn A 2.0 BS02 DNB A 1 D15 N40 I81 H82 M150 E164 F165 N166 D240 D13 N38 I79 H80 M148 E162 F163 N164 D231 D11 D16 N40 Q75 V124 F165 N166 H239 D240 D9 D14 N38 Q73 V122 F163 N164 H230 D231 3.2.2.8 0005509,0005829,0006139,0006152,0006206,0008477,0016798,0016799,0045437,0046133,0046872,0050263 Ki=76uM remove_due_to_license_issue C3T3U2 21082835 502 KRKIILDCDPGHDDAIAIMMAAKHPAIDLLGITIVAGNQTLDKTLINGLNVCQKLEINVPVYAGMPQPIMRQQIVADNIHGDTGLDGPVFEPLTRQAESTHAVKYIIDTLMASDGDITLVPVGPLSNIAVAMRMQPAILPKIREIVLMGGAYGTGNFTPSAEFNIFADPEAARVVFTSGVPLVMMGLDLTNQTVCTPDVIARMERAGGPAGELFSDIMNFTLKTQFEPVHDATCIGYLINPDGIKTQEMYVEVDVNSGPCYGRTVCDELGVLGKPANTKVGITIDTDWFWGLVEECVRGYIKT 3mkn C 2.0 BS02 DNB C 1 D15 N40 A78 M150 E164 F165 N166 D240 D13 N38 A76 M143 E157 F158 N159 D221 D11 D16 N40 Q75 V124 F165 N166 H239 D240 D9 D14 N38 Q73 V117 F158 N159 H220 D221 3.2.2.8 0005509,0005829,0006139,0006152,0006206,0008477,0016798,0016799,0045437,0046133,0046872,0050263 Ki=76uM remove_due_to_license_issue C3T3U2 21082835 502 KRKIILDCDPGHDDAIAIMMAAKHPAIDLLGITIVAGNQTLDKTLINGLNVCQKLEINVPVYAGMPQPIMRQQIVADTGLDGPVFEPLTRQAESTHAVKYIIDTLMASDGDITLVPVGPLSNIAVAMRMQPAILPKIREIVLMGGAYGTGNFTPSAEFNIFADPEAARVVFTSGVPLVMMGLDLTNQTVCTPDVIARMERAGGPAGELFSDIMNFTGPVHDATCIGYLINPDGIKTQEMYVEVDVNSGPCYGRTVCDELGVLGKPANTKVGITIDTDWFWGLVEECVRGYIK 3mks D 2.6 BS01 C1C D 1 Q629 G630 R655 W657 R664 S667 Q330 G331 R356 W358 R365 S368 ? remove_due_to_license_issue P07834 20581844 1 NLKRDLITSLPFEISLKIFNYLQFEDIINSLGVSQNWNKIIRKSTSLWKKLLISENFVSPKGFNSLNLKLSQKYPKLSQQDRLRLSFLENIFILKNWYNPKFVPQRTTLRGHMTSVITCLQFEDNYVITGADDKMIRVYDSINKKFLLQLSGHDGGVWALKYAHGGILVSGSTDRTVRVWDIKKGCCTHVFEGHNSTVRCLDIVEYKNIKYIVTGSRDNTLHVWKLPKEYPLVFHTPEENPYFVGVLRGHMASVRTVSGHGNIVVSGSYDNTLIVWDVAQMKCLYILSGHTDRIYSTIYDHERKRCISASMDTTIRIWDLENGELMYTLQGHTALVGLLRLSDKFLVSAAADGSIRGWDANDYSRKFSYHHTNLSAITTFYVSDNILVSGSENQFNIYNLRSGKLVHANILKDADQIWSVNFKGKTLVAAVEKDGQSFLEILDFS 3ml2 A 1.8 BS02 SU0 A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=9.1nM remove_due_to_license_issue Ki=9nM P00918 20598552 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ml5 A 2.05 BS02 AZM A 1 H94 V121 F131 L198 T199 T200 H94 V121 F131 L198 T199 T200 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T199 4.2.1.1 0004089,0005737,0005829,0006730,0008270,0016829,0032230,0032849,0046872,0051453,0070050,2001225 remove_due_to_license_issue Ki=2.5nM, Kd=17nM, IC50=3440nM P43166 20688517 264 GHHGWGYGQDDGPSHWHKLYPIAQGDRQSPINIISSQAVYSPSLQPLELSYEACMSLSITNNGHSVQVDFNDSDDRTVVTGGPLEGPYRLKQFHFHWGKKHDVGSEHTVDGKSFPSELHLVHWNAKKYSTFGEAASAPDGLAVVGVFLETGDEHPSMNRLTDALYMVRFKGTKAQFSCFNPKSLLPASRHYWTYPGSLTTPPLSESVTWIVLREPISISERQMGKFRSLLFTSEDDERIHMVNNFRPPQPLKGRVVKASFRA 3mlb A 1.8 BS01 LJZ A 1 F103 I104 I105 G106 M109 Y112 W116 F103 I104 I105 G106 M109 Y112 W116 2.7.7.18 0003824,0004515,0005524,0009058,0009165,0009435,0016779,0019363,0070566 ic50=16uM remove_due_to_license_issue C3L5T6 20578699 192 MRKIGIIGGTFDPPHYGHLLIANEVYHALNLEEVWFLPNQIPPHKQGRNITSVESRLQMLELATEAEEHFSICLEELSRKGPSYTYDTMLQLTKKYPDVQFHFIIGGDMVEYLPKWYNIEALLDLVTFVGVARPGYKLRTPYPITTVEIPEFAVSSSLLRERYKEKKTCKYLLPEKVQVYIERNGLYES 3mlb B 1.8 BS01 LJZ A 1 I21 F103 I105 G106 M109 Y112 W116 I21 F99 I101 G102 M105 Y108 W112 2.7.7.18 0003824,0004515,0005524,0009058,0009165,0009435,0016779,0019363,0070566 remove_due_to_license_issue C3L5T6 20578699 192 MRKIGIIGGTFDPPHYGHLLIANEVYHALNLEEVWFLPNQIPPHNITSVESRLQMLELATEAEEHFSICLEELSRKGPSYTYDTMLQLTKKYPDVQFHFIIGGDMVEYLPKWYNIEALLDLVTFVGVARPGYKLRTPYPITTVEIPEFAVSSSLLRERYKEKKTCKYLLPEKVQVYIERNGLYES 3mle A 2.8 BS03 ADP A 1 N10 A11 G12 K13 T14 T15 N175 N12 A13 G14 K15 T16 T17 N177 T9 N10 K13 T14 K35 T39 D50 E116 T11 N12 K15 T16 K37 T41 D52 E118 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue O24872 22284390 226 GHMLFISATNTNAGKTTCARLLAQYCNACGVKTILLKPIETGVNDAINHSSDAHLFLQDNRLLDRSLTLKDISFYRYHKVSAPLIAQQEEDPNAPIDTDNLTQRLHNFTKTYDLVIVEGAGGLCVPITLEENMLDFALKLKAKMLLISHDNLGLINDCLLNDFLLKSHQLDYKIAINLKGNNTAFHSISLPYIELFNTRSNNPIVIFQQSLKVLMSFALKG 3mmf A 1.5 BS02 D9H A 1 I91 Q92 H94 H119 F131 L198 T199 T200 I88 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=37nM remove_due_to_license_issue Ki=37nM P00918 21515057 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mmr A 2.14 BS03 ABH A 1 D216 H218 D220 S229 H233 G234 D274 D323 E368 D113 H115 D117 S126 H130 G131 D171 D220 E265 H193 D216 H218 D220 H233 D323 D325 E368 H90 D113 H115 D117 H130 D220 D222 E265 3.5.3.1 0000050,0004053,0005737,0005829,0006525,0016787,0019547,0030145,0042802,0046872 Kd=11uM remove_due_to_license_issue Q8I384 20527960 551 KNVSIIGSPLAAGQPLGGVQLACDDLRKLGLHNVIDVLGWKYEDIGNIDNCYYDNIRNIKEIGIFSKNLFDTMSNELRKKNFVLNIGGDHGVAFSSILSSLQMYQNLRVIWIDAHGDINIPETSPSGNYHGMTLAHTLGLFKKKVPYFEWSENLTYLKPENTAIIGIRDIDAYEKIILKKCNINYYTIFDIEKNGIYNTICTALEKIDPNSNCPIHISLDIDSVDNVFAPGTGTVAKGGLNYREINLLMKILAETKRVVSMDLVEYNPSLDEVDKKVHGDSLPILDNATKTGKLCLELIARVLGYDIV 3mn8 A 2.7 BS02 GEM A 1 H101 E104 R165 N174 R175 H217 D228 G279 W282 Y283 L285 E305 H73 E76 R137 N146 R147 H181 D192 G243 W246 Y247 L249 E269 3.4.17.22 0004181,0006508,0008270 remove_due_to_license_issue P42787 20600119 601 KEDESFLQQPHYASQEQLEDLFAGLEKAYPNQAKVHFLGRSLEGRNLLALQISRNTRSRNLLTPPVKYIANMHGDETVGRQLLVYMAQYLLGNHERISDLGQLVNSTDIYLVPTMNPDGYALSQEGNCESLPNYVGRGNAANIDLNRDFPDRLEAQSRQPETAALVNWIVSKPFVLSANFHGGAVVASYPYDNSLAHNECCEESLTPDDRVFKQLAHTYSDNHPIMRKGNNCNDSFSGGITNGAHWYELSGGMQDFNYAFSNCFELTIELSCCKYPAASTLPQEWQRNKASLLQLLRQAHIGIKGLVTDASGFPIADANVYVAGLEEKPMRTSKRGEYWRLLTPGLYSVHASAFGYQTSAPQQVRVTNDNQEALRLDFKLAPV 3mna A 1.5 BS02 DWH A 1 Q92 H94 H119 F131 L198 T199 T200 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=41nM remove_due_to_license_issue Ki=41nM P00918 21515057 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mnu A 1.8 BS02 BON A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=48nM remove_due_to_license_issue Ki=48nM P00918 20472429 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mo0 A 2.78 BS02 E11 A 1 D1131 A1134 D1135 E1138 D1140 L1143 D1145 R1214 F1215 K1219 D148 A151 D152 E155 D157 L160 D162 R231 F232 K236 Y1124 Y1211 Y141 Y228 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 remove_due_to_license_issue Q9H9B1 20434463 2001 RIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRH 3mo0 A 2.78 BS08 E11 A 2 D1131 A1134 R1137 E1138 D1140 L1143 D1145 R1214 F1215 K1219 D148 A151 R154 E155 D157 L160 D162 R231 F232 K236 Y1124 Y1211 Y141 Y228 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 remove_due_to_license_issue Q9H9B1 20434463 2002 RIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRH 3mo2 A 2.49 BS05 E67 A 1 D1131 A1134 D1135 R1137 E1138 D1140 S1141 L1143 D1145 Y1211 R1214 F1215 D154 A157 D158 R160 E161 D163 S164 L166 D168 Y231 R234 F235 Y1124 Y1211 Y147 Y231 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Kd=244nM remove_due_to_license_issue Q9H9B1 20434463 1 IVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 3mo5 A 2.14 BS05 E72 A 1 D1131 A1134 D1135 R1137 D1140 L1143 D1145 Y1211 R1214 F1215 D154 A157 D158 R160 D163 L166 D168 Y231 R234 F235 Y1124 Y1211 Y147 Y231 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Kd=136nM remove_due_to_license_issue IC50=100nM, Kd=136nM Q9H9B1 20434463 1236 IVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 3moe A 1.25 BS03 SPV A 1 R87 G237 K243 K244 H264 S286 R405 R89 G239 K245 K246 H266 S288 R407 R87 Y235 K244 H264 S286 C288 D311 R405 R89 Y237 K246 H266 S288 C290 D313 R407 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 Ki=50uM remove_due_to_license_issue P07379 20476774 1200 GSMPPQLHNGLDFSAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEATGKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 3moh A 2.1 BS03 PGA A 1 R87 G237 K244 D311 F333 R405 R76 G226 K233 D300 F322 R394 R87 Y235 K244 H264 S286 C288 D311 R405 R76 Y224 K233 H253 S275 C277 D300 R394 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 Ki=1460uM remove_due_to_license_issue P07379 20476774 900 SAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEATKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 3moj B 2.902 BS01 rna A 0 K413 R417 D420 V422 G423 T424 A426 K427 A433 I436 G437 I439 T466 V467 K468 G469 K470 K473 K10 R14 D17 V19 G20 T21 A23 K24 A30 I33 G34 I36 T63 V64 K65 G66 K67 K70 3.6.4.13 remove_due_to_license_issue P42305 20673833 2508 ~ 2581 MKLYFNGGKKKKIRAVDFVGTIAKIDGVSADDIGIITIMDNASYVEILNGKGPHVLKVMKNTTVKGKQLKVNKAN 3mpm A 1.95 BS01 5LK A 1 L251 A271 K273 E288 T316 Y318 M319 E320 G322 L371 L14 A34 K36 E51 T79 Y81 M82 E83 G85 L134 N364 R366 A368 N369 D382 F402 N127 R129 A131 N132 D145 F161 2.7.10.2 0004672,0005524,0006468 ic50=30nM remove_due_to_license_issue P06239 20483608 1 WEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRNLRAANILVSDTLSCKIADFGLARLIEDNEYTARFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFF 3mpt A 1.89 BS01 1GK A 1 K53 T106 H107 L108 M109 A111 A157 K50 T103 H104 L105 M106 A108 A154 D150 K152 N155 D168 T185 D147 K149 N152 D165 T180 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.25uM remove_due_to_license_issue Q16539 20570148 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3mq6 A 2.0 BS01 dna L 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 R152 R246 S247 D248 R24 T26 Q29 L30 Q32 Q33 N85 A86 K89 R145 R239 S240 D241 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 A 2.0 BS02 dna K 0 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 A88 K89 G92 R145 S146 K235 R236 S237 R239 R242 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 B 2.0 BS01 dna L 0 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 A94 K95 G98 R151 S152 K241 R242 S243 R245 R248 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 B 2.0 BS02 dna K 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 V97 R246 S247 D248 N286 R30 T32 Q35 L36 Q38 Q39 N91 A92 K95 V96 R245 S246 D247 N285 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 C 2.0 BS01 dna N 0 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 A94 K95 G98 R151 S152 K241 R242 S243 R245 R248 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLASAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 C 2.0 BS02 dna M 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 R246 S247 D248 R30 T32 Q35 L36 Q38 Q39 N91 A92 K95 R245 S246 D247 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLASAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 D 2.0 BS01 dna N 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 R246 S247 D248 N286 R25 T27 Q30 L31 Q33 Q34 N86 A87 K90 R240 S241 D242 N280 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 D 2.0 BS02 dna M 0 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 A89 K90 G93 R146 S147 K236 R237 S238 R240 R243 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 E 2.0 BS01 dna P 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 R152 R246 S247 D248 R25 T27 Q30 L31 Q33 Q34 N86 A87 K90 R146 R240 S241 D242 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 2 ~ 17 PFTYSIEATRNLATTERCIQDIRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 E 2.0 BS02 dna O 0 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 A89 K90 G93 R146 S147 K236 R237 S238 R240 R243 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 F 2.0 BS01 dna P 0 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 A94 K95 G98 R151 S152 K241 R242 S243 R245 R248 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 2 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 F 2.0 BS02 dna O 0 R31 T33 Q36 L37 Q39 Q40 D90 N92 A93 K96 R246 S247 D248 R30 T32 Q35 L36 Q38 Q39 D89 N91 A92 K95 R245 S246 D247 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGRSAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 G 2.0 BS01 dna R 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 R152 R246 S247 D248 R30 T32 Q35 L36 Q38 Q39 N91 A92 K95 R151 R245 S246 D247 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 G 2.0 BS02 dna Q 0 S91 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 S90 A94 K95 G98 R151 S152 K241 R242 S243 R245 R248 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 H 2.0 BS01 dna R 0 R29 A95 K96 G99 R152 S153 K242 R243 S244 R246 R249 R28 A94 K95 G98 R151 S152 K241 R242 S243 R245 R248 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mq6 H 2.0 BS02 dna Q 0 R31 T33 Q36 L37 Q39 Q40 N92 A93 K96 R246 S247 D248 G284 R30 T32 Q35 L36 Q38 Q39 N91 A92 K95 R245 S246 D247 G283 3.1.21.4 0042802,0046872 remove_due_to_license_issue Q9F6L0 21151881 1 ~ 17 PFTYSIEATRNLATTERCIQDIRNAPVRNRSTQFQLAQQNMLAYTFGEVIPGFASAGINGMDYRDVIGRPVENAVTEGTHFFRDDFRVDSNAKAKVAGDIFEIVSSAVMWNCAARWNSLMVGEGWRSQPRYSRPTLSPSPRRQVAVLNLPRSFDWVSLLVPESQEVIEEFRAGLRKDGLGLPTSTPDLAVVVLPEEFQNDEMWREEIAGLTRPNQILLSGAYQRLQGRVQPGEISLAVAFKRSLRSDRLYQPLYEANVMQLLLEGKLGAPKVEFEVHTLAPEGTNAFVTYEAASLYGLAEGAVHRAIRELYVPPTAADLARRFFAFLNERMELVNG 3mqf A 1.951 BS01 20X A 1 E88 G135 L136 N282 D283 N284 H341 H377 N484 E672 S674 G675 E77 G124 L125 N265 D266 N267 H314 H350 N457 E645 S647 G648 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=5.7uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mqf A 1.951 BS02 20X A 2 R60 V64 W67 E190 K191 A192 R49 V53 W56 E179 K180 A181 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=5.7uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mrt A 1.98 BS01 12E A 1 R60 V64 W67 E190 K191 A192 P229 R49 V53 W56 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=200uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mrt A 1.98 BS02 12E A 2 G135 L136 D283 N284 D339 H341 H377 T378 A383 N484 E672 S674 G675 G124 L125 D266 N267 D313 H315 H351 T352 A357 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=200uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mrv A 1.94 BS01 16F A 1 R60 V64 W67 W189 E190 K191 A192 P229 R49 V53 W56 W178 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=180uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mrv A 1.94 BS02 16F A 2 G135 L136 D283 N284 F285 H341 H377 A383 N484 E672 S674 G675 G124 L125 D266 N267 F268 H315 H351 A357 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=180uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mrx A 1.95 BS01 17S A 1 R60 L63 W67 E190 K191 A192 P229 R49 L52 W56 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H352 K543 R544 K549 T651 K655 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=406.5uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mrx A 1.95 BS02 17S A 2 E88 G135 L136 N282 D283 H341 H377 N484 E672 S674 G675 E77 G124 L125 N266 D267 H316 H352 N459 E647 S649 G650 H377 K568 R569 K574 T676 K680 H352 K543 R544 K549 T651 K655 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=406.5uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms2 A 2.1 BS01 18S A 1 R60 V64 W67 E190 K191 A192 P229 R49 V53 W56 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H352 K543 R544 K549 T651 K655 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=192.4uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms2 A 2.1 BS02 18S A 2 E88 G135 L136 Y280 N282 D283 R292 H341 H377 V455 N484 E672 S674 G675 E77 G124 L125 Y264 N266 D267 R276 H316 H352 V430 N459 E647 S649 G650 H377 K568 R569 K574 T676 K680 H352 K543 R544 K549 T651 K655 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=192.4uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms4 A 2.07 BS01 21N A 1 R60 L63 W67 N187 E190 K191 A192 P229 R49 L52 W56 N176 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=524.3uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms4 A 2.07 BS02 21N A 2 E88 G135 L136 Y280 N282 R292 H377 N484 E672 A673 S674 G675 E77 G124 L125 Y263 N265 R275 H351 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=524.3uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms7 A 1.95 BS01 22S A 1 R60 W189 E190 K191 A192 R49 W178 E179 K180 A181 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=370uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms7 A 1.95 BS02 22S A 2 E88 G135 L136 N282 D283 N284 F285 H341 H377 A383 N484 E672 S674 G675 E77 G124 L125 N265 D266 N267 F268 H314 H350 A356 N457 E645 S647 G648 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=370uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3ms9 A 1.8 BS02 MS9 A 1 A337 L340 L341 I432 A433 P465 V468 A106 L109 L110 I199 A200 P232 V235 D363 A365 R367 N368 D381 P402 D132 A134 R136 N137 D150 P169 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 20450175 516 AMDPPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ 3msc A 1.951 BS01 24S A 1 E88 N133 G135 L136 N282 D283 N284 F285 H341 H377 N484 E672 S674 G675 E77 N122 G124 L125 N265 D266 N267 F268 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=484.2uM remove_due_to_license_issue P00489 20947361 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3msc A 1.951 BS02 24S A 2 R60 W189 E190 K191 P229 R49 W178 E179 K180 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=484.2uM remove_due_to_license_issue P00489 20947361 844 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3msj A 1.8 BS01 EV3 A 1 D32 G34 Y71 W76 D228 D36 G38 Y75 W80 D221 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=770uM remove_due_to_license_issue IC50=770000nM P56817 20656487 393 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3msk A 2.0 BS01 EV4 A 1 L30 D32 Y71 W76 F108 D228 G230 L32 D34 Y73 W78 F110 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=26uM remove_due_to_license_issue IC50=26000nM P56817 20656487 396 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3msl A 2.4 BS01 EV5 A 1 D32 Y71 W76 F108 D228 G230 D34 Y73 W78 F110 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=7uM remove_due_to_license_issue IC50=7000nM P56817 20656487 395 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3mss A 1.95 BS02 MS7 A 1 L341 A433 P465 V468 L108 A199 P231 V234 D363 A365 R367 N368 D381 P402 D130 A132 R134 N135 D148 P168 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 20450175 516 MDPSYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ 3mt7 A 2.0 BS01 16O A 1 R60 W67 N187 E190 K191 A192 P229 R49 W56 N176 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=93.2uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mt7 A 2.0 BS02 16O A 2 E88 G135 L136 Y280 N282 D283 R292 H341 H377 N484 E672 S674 G675 E77 G124 L125 Y263 N265 D266 R275 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=93.2uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mt8 A 2.0 BS01 17T A 1 R60 V64 W67 E190 K191 A192 P229 R49 V53 W56 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=28.3uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mt8 A 2.0 BS02 17T A 2 E88 G135 L136 Y280 N282 D283 H377 N484 E672 S674 G675 E77 G124 L125 Y263 N265 D266 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=28.3uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mt9 A 2.05 BS01 18O A 1 R60 L63 W189 E190 K191 A192 P229 R49 L52 W178 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=25.7uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mt9 A 2.05 BS02 18O A 2 E88 G135 L136 Y280 N282 D283 N284 F285 R292 H341 H377 N484 E672 S674 G675 E77 G124 L125 Y263 N265 D266 N267 F268 R275 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=25.7uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mta A 2.23 BS01 22O A 1 R60 V64 N187 W189 E190 K191 A192 P229 R49 V53 N176 W178 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=50.4uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mta A 2.23 BS02 22O A 2 G135 L136 L139 N282 N284 F285 F286 H341 H377 N484 E672 A673 S674 G675 G124 L125 L128 N265 N267 F268 F269 H315 H351 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=50.4uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mtb A 1.95 BS01 23V A 1 R60 V64 W67 W189 E190 K191 A192 P229 R49 V53 W56 W178 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=23.2uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 3mtb A 1.95 BS02 23V A 2 G135 L136 N282 N284 F285 F286 H341 H377 N484 E672 A673 S674 G675 G124 L125 N265 N267 F268 F269 H315 H351 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=23.2uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 3mtd A 2.096 BS01 25E A 1 L136 D283 N284 F285 H341 H377 A383 N484 E672 S674 G675 L125 D266 N267 F268 H315 H351 A357 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=340.5uM remove_due_to_license_issue P00489 20947361 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mtd A 2.096 BS02 25E A 2 R60 V64 W189 E190 K191 A192 R49 V53 W178 E179 K180 A181 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=340.5uM remove_due_to_license_issue P00489 20947361 844 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3mtw A 1.7 BS03 M3R A 1 H171 K211 V218 F219 H252 H272 D294 N297 D318 I321 Q325 D344 H145 K185 V192 F193 H226 H246 D268 N271 D292 I295 Q299 D318 ? 0016787,0016810,0046872 Ki=92nM remove_due_to_license_issue Q9A4Z9 20604542 430 AEIKAVSAARLLDVASGKYVDNPLVIVTDGRITSIGKKGDAVPAGATAVDLPGVTLLPGLIDMHVHLDSLAEVGGYNSLEYSDRFWSVVQTANAKKTLEAGFTTVRNVGAADYDDVGLREAIDAGYVPGPRIVTAAISFGATGGHCDSTFFPPSMDQKNPFNSDSPDEARKAVRTLKKYGAQVIKICATGGVFSRGNEPGQQQLTYEEMKAVVDEAHMAGIKVAAHAHGASGIREAVRAGVDTIEHASLVDDEGIKLAVQKGAYFSMDIYNTDYTQAEGKKNGVLEDNLRKDRDIGELQRENFRKALKAGVKMVYGTDAGIYPHGDNAKQFAVMVRYGATPLQAIQSATLTAAEALGRSKDVGQVAVGRYGDMIAVAGDPLADVTTLEKPVFVMKGGAVVKAP 3muf A 2.3 BS02 S3P A 1 M10 D33 R57 G79 G80 G81 R116 R132 M9 D32 R56 G78 G79 G80 R115 R131 2.7.1.71 0000287,0004765,0005524,0005737,0005829,0008652,0009073,0009423,0016301,0019752,0046872 remove_due_to_license_issue P56073 22438938 201 QHLVLIGFMGSGKSSLAQELGLALKLEVLDTDMIISERVGLSVREIFEELGEDNFRMFEKNLIDELKTLKTPHVISTGGGIVMHENLKGLGTTFYLKMDFETLIKRLNQKEREKRPLLNNLTQAKELFEKRQALYEKNASFIIDARGGLNNSLKQVLQFI 3muz 1 1.9 BS01 IPT 1 1 N102 D201 E461 Y503 E537 H540 N604 W999 N90 D189 E449 Y491 E525 H528 N592 W987 D201 E461 Y503 E537 D189 E449 Y491 E525 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDAQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3muz 1 1.9 BS02 IPT 1 2 E304 P306 R645 D648 Q702 W708 E292 P294 R633 D636 Q690 W696 D201 E461 Y503 E537 D189 E449 Y491 E525 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 2002 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDAQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3muz 4 1.9 BS01 IPT 4 1 N102 D201 E461 E537 H540 N604 W999 N90 D189 E449 E525 H528 N592 W987 D201 E461 Y503 E537 D189 E449 Y491 E525 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDAQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3muz 4 1.9 BS02 IPT 4 2 E304 P306 R645 D648 Q702 W708 E292 P294 R633 D636 Q690 W696 D201 E461 Y503 E537 D189 E449 Y491 E525 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 2002 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDAQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3mv0 1 2.2 BS01 149 1 1 D201 H391 N460 E461 M502 Y503 E537 H540 W568 F601 N604 D189 H379 N448 E449 M490 Y491 E525 H528 W556 F589 N592 D201 E461 Y503 E537 D189 E449 Y491 E525 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue P00722 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDAQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3mv0 4 2.2 BS01 149 4 1 D201 H391 E461 M502 Y503 E537 H540 W568 F601 N604 D189 H379 E449 M490 Y491 E525 H528 W556 F589 N592 D201 E461 Y503 E537 D189 E449 Y491 E525 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue P00722 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDAQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3mv5 A 2.47 BS03 XFE A 1 A177 M227 A230 E234 M281 T291 F438 A34 M84 A87 E91 M138 T148 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 ic50=180nM remove_due_to_license_issue IC50=180nM P31749 20481595 999 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMIRPHFPQFDYSAS 3mvh A 2.01 BS03 WFE A 1 L156 G157 K158 G162 V164 A177 M227 E228 Y229 A230 E234 M281 T291 D292 F438 L12 G13 K14 G18 V20 A33 M83 E84 Y85 A86 E90 M137 T147 D148 F294 D274 K276 N279 D292 T312 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.5nM remove_due_to_license_issue IC50=0.5nM P31749 20481595 999 VTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQRPHFPQFDYSA 3mvj A 2.49 BS03 XFE A 1 L49 V57 A70 V123 L173 T183 F327 L35 V43 A56 V109 L159 T169 F313 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 ic50=3200nM remove_due_to_license_issue P17612 20481595 351 VKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3mvl A 2.8 BS01 38P A 1 A51 K53 E71 I84 T106 L108 M109 G110 A111 L167 D168 F169 L171 A47 K49 E67 I80 T102 L104 M105 G106 A107 L163 D164 F165 L167 D150 K152 N155 D168 T185 D146 K148 N151 D164 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=13nM Q16539 20804198 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3mvm A 2.0 BS01 39P A 1 A51 K53 E71 L75 I84 L104 T106 L108 M109 L167 D168 F169 L171 A43 K45 E63 L67 I76 L96 T98 L100 M101 L159 D160 F161 L163 D150 K152 N155 D168 T185 D142 K144 N147 D160 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=3.9nM remove_due_to_license_issue IC50=3.9nM Q16539 20804198 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3mw1 A 2.8 BS01 MIH A 1 A51 L104 T106 L108 M109 G110 A111 D168 A43 L96 T98 L100 M101 G102 A103 D160 D150 K152 N155 D168 T185 D142 K144 N147 D160 T175 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=0.820000nM Q16539 21999461 1 ERPTFYRQELNKTIWEVPERYQNLSPVGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLATDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3mwu A 1.98 BS05 BK3 A 1 A103 K105 M136 I150 Y155 E159 L205 D219 A38 K40 M71 I85 Y90 E94 L140 D154 D198 K200 E202 N203 D219 T238 D133 K135 E137 N138 D154 T169 2.7.11.17 0004672,0005509,0005524,0006468 remove_due_to_license_issue A3FQ16 21116453 561 LYFQGTFAERYNIVCMLGKGSFGEVLKCKDRITQQEYAVKVINKASAKNKDTSTILREVELLKKLDHPNIMKLFEILEDSSSFYIVGELYTGGELFDEIIKRKRFSEHDAARIIKQVFSGITYMHKHNIVHRDLKPENILLESKEKDCDIKIIDFGLSTCFQQNDRIGTAYYIAPEVLRGTYDEKCDVWSAGVILYILLSGTPPFYGKNEYDILKRVETGKYAFDLPQWRTISDDAKDLIRKMLTFHPSLRITATQCLEHPWIQKYSSETPTISDLPSLESAMTNIRQFQAEKKLAQAALLYMASKLTTLDETKQLTEIFRKLDTNNDGMLDRDELVRGYHEFMRLKGVDSNSLIQNEGSTIEDQIDSLMPLLDMDGSGSIEYSEFIASAIDRTILLSRERMERAFKMFDKDGSGKISTKELEQVDNNKDGEVDFNEFVEMLQNFVR 3mww B 2.8 BS01 BIW B 1 A396 H428 L492 V494 P495 W500 R503 A374 H406 L470 V472 P473 W478 R481 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 20942454 577 SMSYTWTGALITPCAAEMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3mx9 A 2.6 BS01 dna C 0 D20 G21 S22 I24 Q26 Y44 T46 Q47 K48 R51 Q75 N136 D137 S138 R141 K142 R221 S223 N224 K225 Q229 Y257 Y259 S261 E271 I272 K330 D19 G20 S21 I23 Q25 Y43 T45 Q46 K47 R50 Q74 N135 D136 S137 R140 K141 R175 S177 N178 K179 Q183 Y211 Y213 S215 E225 I226 K284 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQINPNQSSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRASNKEFLLYLAGFVDSDGSIIAQIKPRQSNKFKHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 3mx9 A 2.6 BS02 dna D 0 S32 S33 K34 R38 R40 Y66 R68 D137 S210 D211 G212 S213 I215 Q217 K219 T237 Q238 K239 R268 A324 N327 D328 S329 T331 R332 K333 S31 S32 K33 R37 R39 Y65 R67 D136 S164 D165 G166 S167 I169 Q171 K173 T191 Q192 K193 R222 A278 N281 D282 S283 T285 R286 K287 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNKEFLLYLAGFVDGDGSIIAQINPNQSSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRASNKEFLLYLAGFVDSDGSIIAQIKPRQSNKFKHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 3mxb A 2.3 BS01 dna C 0 D20 S22 I24 Q26 Y44 T46 Q47 K48 R51 Q75 N136 D137 S138 T140 K142 D19 S21 I23 Q25 Y43 T45 Q46 K47 R50 Q74 N135 D136 S137 T139 K141 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNKKFLLYLAGFVDGDGSIIAQINPNQSSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 3mxb A 2.3 BS02 dna E 0 S33 R38 R40 R68 E80 K139 S32 R37 R39 R67 E79 K138 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNKKFLLYLAGFVDGDGSIIAQINPNQSSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 3mxb B 2.3 BS01 dna C 0 R30 S32 N33 K34 Q38 Y66 Y68 E80 I81 K116 K139 R29 S31 N32 K33 Q37 Y65 Y67 E79 I80 K115 K138 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNEEFLLYLAGFVDSDGSIIAQIKPRQSNKFKHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 3mxb B 2.3 BS02 dna E 0 S19 D20 G21 S22 I24 Q26 K28 T46 Q47 K48 R51 R77 N136 D137 S138 T140 R141 K142 S18 D19 G20 S21 I23 Q25 K27 T45 Q46 K47 R50 R76 N135 D136 S137 T139 R140 K141 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNEEFLLYLAGFVDSDGSIIAQIKPRQSNKFKHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 3mxb R 2.3 BS01 dna T 0 D20 G21 S22 I24 Q26 Y44 T46 Q47 K48 R51 Q75 N136 D137 S138 T140 R141 K142 D19 G20 S21 I23 Q25 Y43 T45 Q46 K47 R50 Q74 N135 D136 S137 T139 R140 K141 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNKKFLLYLAGFVDGDGSIIAQINPNQSSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDSL 3mxb R 2.3 BS02 dna V 0 S33 R38 R40 R68 E80 K116 S32 R37 R39 R67 E79 K115 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNKKFLLYLAGFVDGDGSIIAQINPNQSSKFKHRLRLTFYVTQKTQRRWFLDKLVDEIGVGYVRDSGSVSQYVLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDSL 3mxb S 2.3 BS01 dna T 0 R30 S32 N33 Q38 Y66 Y68 R77 E80 I81 K139 R29 S31 N32 Q37 Y65 Y67 R76 E79 I80 K138 0004519 remove_due_to_license_issue 20846960 501 ~ 524 NTKYNEEFLLYLAGFVDSDGSIIAQIKPRQSNKFKHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 3mxb S 2.3 BS02 dna V 0 S19 D20 G21 S22 I24 Q26 K28 T46 Q47 K48 R51 N136 D137 S138 T140 R141 K142 S18 D19 G20 S21 I23 Q25 K27 T45 Q46 K47 R50 N135 D136 S137 T139 R140 K141 0004519 remove_due_to_license_issue 20846960 601 ~ 624 NTKYNEEFLLYLAGFVDSDGSIIAQIKPRQSNKFKHQLSLTFAVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSDYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 3mxd A 1.95 BS01 K53 A 1 D25 G27 A28 D29 D30 I47 G48 I50 D25 G27 A28 D29 D30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.47nM remove_due_to_license_issue P03369 20958050 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3mxd B 1.95 BS01 K53 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 20958050 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3mxe A 1.85 BS01 K54 A 1 D25 G27 A28 D29 D30 I47 G48 I50 D25 G27 A28 D29 D30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.097nM remove_due_to_license_issue P03369 20958050 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3mxe B 1.85 BS01 K54 A 1 D25 A28 D30 G48 V82 D25 A28 D30 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 20958050 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3mxf A 1.6 BS01 JQ1 A 1 W81 P82 L92 L94 N140 I146 M149 W40 P41 L51 L53 N99 I105 M108 ? remove_due_to_license_issue O60885 20871596 1 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 3mxr A 1.3 BS01 CZ8 A 1 M69 S70 N132 E166 T167 N170 G236 A237 E240 M44 S45 N107 E141 T142 N145 G211 A212 E214 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 21041505 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3mxs A 1.24 BS01 CZ9 A 1 M69 S70 N132 E166 T167 N170 G236 A237 G238 M44 S45 N107 E141 T142 N145 G211 A212 G213 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 21041505 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3my1 A 2.8 BS01 RFZ A 1 A46 D104 F105 C106 L156 D167 A41 D92 F93 C94 L144 D155 D149 K151 A153 N154 D167 S180 T191 D137 K139 A141 N142 D155 S168 T179 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 20851342 336 DSVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKKGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAKNSQPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKGM 3my5 A 2.1 BS01 RFZ A 1 I10 V18 A31 K33 F80 E81 L83 L134 I12 V20 A33 K35 F79 E80 L82 L133 D127 K129 Q131 N132 D145 T158 T165 D126 K128 Q130 N131 D144 T157 T164 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=65uM remove_due_to_license_issue P24941 20851342 300 GSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3myg A 2.4 BS01 EML A 1 R137 L139 L194 L210 Y212 A213 P214 L215 G216 L263 D274 R12 L14 L69 L85 Y87 A88 P89 L90 G91 L138 D149 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 24900197 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3myq A 1.35 BS02 E27 A 1 Q92 H94 H96 H119 V121 F131 L198 T199 T200 P202 Q89 H91 H93 H116 V118 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.03uM remove_due_to_license_issue P00918 20926301 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3mz3 A 3.2 BS02 B3N A 1 Y100 H142 H143 F152 D178 H180 F208 Y306 Y80 H122 H123 F132 D158 H160 F188 Y286 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue Q9BY41 20545365 390 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 3mz3 A 3.2 BS03 B3N B 1 F152 P273 F132 P253 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue Q9BY41 20545365 390 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 3mz6 A 2.0 BS02 B3N A 1 H143 D178 H180 F208 Y306 H122 D157 H159 F187 Y285 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue Q9BY41 20545365 701 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGEYGLGYLCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 3mzc A 1.498 BS02 S6I A 1 H94 H96 F131 L198 T199 T200 H91 H93 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=226nM remove_due_to_license_issue Ki=226nM P00918 20922253 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3n0h A 1.92 BS01 TOP A 1 V8 A9 E30 F31 F34 I60 L67 V8 A9 E30 F31 F34 I60 L67 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=617nM remove_due_to_license_issue IC50=680000nM, Ki=19070nM P00374 21684339 187 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFSRMTTTSSVEGKQNLVIMGKKTWFSIPEKFRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3n0h A 1.92 BS02 TOP A 2 S59 P61 F64 S59 P61 F64 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=617nM remove_due_to_license_issue IC50=680000nM, Ki=19070nM P00374 21684339 191 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFSRMTTTSSVEGKQNLVIMGKKTWFSIPEKFRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3n0n A 1.5 BS02 P9B A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=50nM remove_due_to_license_issue Ki=50nM P00918 20922253 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3n1c A 2.0 BS01 F6P A 1 D14 G39 N43 R90 G138 S139 D256 D14 G39 N43 R90 G138 S139 D256 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 21147773 400 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3n1c A 2.0 BS02 F6P D 1 K27 R29 K27 R29 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 21147773 403 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3n1c D 2.0 BS01 F6P A 1 K27 R29 K27 R29 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 21147773 400 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3n1c D 2.0 BS02 F6P D 1 D14 G38 G39 N43 R90 N92 G138 S139 D256 D14 G38 G39 N43 R90 N92 G138 S139 D256 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 21147773 403 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3n1i A 2.2 BS01 dna B 0 L82 M96 L115 A117 H139 D140 M143 L144 K153 L28 M42 L61 A63 H85 D86 M89 L90 K99 ? 0003677,0003697,0006355,0006952 remove_due_to_license_issue D9J034 20551348 1 ~ 9 GRVFAPYSVFKGKAALSAEPRLPTFNRLDSGGVKLNRRGVIMLTFWPSVGERKYDWEKRQLFALSATEVGSLISMGTRDSSEFFHDPSMLSSNAGQVRKSLSIKPNADGSGYFISLSVVNNNLKTNDRFTVPVTTAEFAVMRTAFSFALPHIMGWDRFTNR 3n1j A 2.65 BS01 dna B 0 L115 A117 F138 H139 D140 M143 L144 K153 L61 A63 F84 H85 D86 M89 L90 K99 ? 0003677,0003697,0006355,0006952 remove_due_to_license_issue D9J034 20551348 1 ~ 9 GRVFAPYSVFKGKAALSAEPRLPTFNRLDSGGVKLNRRGVIMLTFWPSVGERKYDWEKRQLFALSATEVGSLISMGTRDSSEFFHDPSMLSSNAGQVRKSLSIKPNADGSGYFISLSVVNNNLKTNDRFTVPVTTAEFAVMRTAFSFALPHIMGWDRFTNR 3n1k A 2.702 BS01 dna B 0 L82 F116 A117 F138 H139 D140 M143 L144 K153 L28 F62 A63 F84 H85 D86 M89 L90 K99 ? 0003677,0003697,0006355,0006952 remove_due_to_license_issue D9J034 20551348 1 ~ 9 GRVFAPYSVFKGKAALSAEPRLPTFNRLDSGGVKLNRRGVIMLTFWPSVGERKYDWEKRQLFALSATEVGSLISMGTRDSSEFFHDPSMLSSNAGQVRKSLSIKPNADGSGYFISLSVVNNNLKTNDRFTVPVTTAEFAVMRTAFSFALPHIMGWDRFTNR 3n1l A 2.35 BS01 dna B 0 L115 F116 A117 F138 H139 D140 M143 L144 K153 L61 F62 A63 F84 H85 D86 M89 L90 K99 ? 0003677,0003697,0006355,0006952 remove_due_to_license_issue D9J034 20551348 1 ~ 9 GRVFAPYSVFKGKAALSAEPRLPTFNRLDSGGVKLNRRGVIMLTFWPSVGERKYDWEKRQLFALSATEVGSLISMGTRDSSEFFHDPSMLSSNAGQVRKSLSIKPNADGSGYFISLSVVNNNLKTNDRFTVPVTTAEFAVMRTAFSFALPHIMGWDRFTNR 3n1v F 2.18 BS01 3N1 F 1 K57 N59 R60 S205 F206 F239 K347 K50 N52 R53 S198 F199 F232 K340 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50>500uM remove_due_to_license_issue IC50=>500000000nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n1v F 2.18 BS02 3N1 F 2 E318 Y322 E311 Y315 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50>500uM remove_due_to_license_issue IC50=>500000000nM P14324 20711197 354 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n1w F 2.56 BS01 3N2 F 1 N59 R60 S205 F206 F239 K347 N52 R53 S198 F199 F232 K340 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=>500000000nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n23 A 4.6 BS01 OBN A 1 P118 D121 V322 A323 F783 T797 R880 P94 D97 V298 A299 F759 T773 R856 D369 D710 D714 D345 D686 D690 7.2.2.13 0000166,0002028,0005215,0005391,0005515,0005524,0005886,0005890,0006813,0006814,0006883,0008556,0010248,0016020,0016323,0016887,0030007,0030424,0030955,0031402,0036376,0042383,0042470,0042995,0046872,0051117,0055085,0086009,1902600,1990573 remove_due_to_license_issue P05024 21182963 1 MDELKKEVSMDDHKLSLDELHRKYGTDLSRGLTPARAAEILARDGPNALTPPPTTPEWVKFCRQLFGGFSMLLWIGAILCFLAYGIQAATEEEPQNDNLYLGVVLSAVVIITGCFSYYQEAKSSKIMESFKNMVPQQALVIRNGEKMSINAEEVVVGDLVEVKGGDRIPADLRIISANGCKVDNSSLTGESEPQTRSPDFTNENPLETRNIAFFSTNCVEGTARGIVVYTGDRTVMGRIATLASGLEGGQTPIAAEIEHFIHIITGVAVFLGVSFFILSLILEYTWLEAVIFLIGIIVANVPEGLLATVTVCLTLTAKRMARKNCLVKNLEAVETLGSTSTICSDKTGTLTQNRMTVAHMWSDNQIHEADTTENQSGVSFDKTSATWLALSRIAGLCNRAVFQANQENLPILKRAVAGDASESALLKCIELCCGSVKEMRERYTKIVEIPFNSTNKYQLSIHKNPNTAEPRHLLVMKGAPERILDRCSSILIHGKEQPLDEELKDAFQNAYLELGGLGERVLGFCHLFLPDEQFPEGFQFDTDDVNFPLDNLCFVGLISMIDPPRAAVPDAVGKCRSAGIKVIMVTGDHPITAKAIAKGVGIISEGNETVEDIAARLNIPVSQVNPRDAKACVVHGSDLKDMTSEQLDDILKYHTEIVFARTSPQQKLIIVEGCQRQGAIVAVTGDGVNDSPASKKADIGVAMGIAGSDVSKQAADMILLDDNFASIVTGVEEGRLIFDNLKKSIAYTLTSNIPEITPFLIFIIANIPLPLGTVTILCIDLGTDMVPAISLAYEQAESDIMKRQPRNPKTDKLVNEQLISMAYGQIGMIQALGGFFTYFVILAENGFLPIHLLGLRVNWDDRWINDVEDSYGQQWTYEQRKIVEFTCHTPFFVTIVVVQWADLVICKTRRNSVFQQGMKNKILIFGLFEETALAAFLSYCPGMGVALRMYPLKPTWWFCAFPYSLLIFVYDEVRKLIIRRRPGGWVEKETYY 3n2c A 2.81 BS03 LWY A 1 H65 H140 K188 V195 A196 Y231 H249 D321 H64 H139 K187 V194 A195 Y230 H248 D320 ? 0005737,0016787,0016810,0046872 remove_due_to_license_issue Q393A1 20604542 427 TITVLQGGNVLDLERGVLLEHHHVVIDGERIVEVTDRPVDLPNAQAIDVRGKTVMPGFIDCHVHVLASNANLGVNATQPNILAAIRSLPILDAMLSRGFTSVRDAGGADWSLMQAVETGLVSGPRIFPSGKALSQTGGHGDFRPRGDLLEPCSCCFRTGAIARVVDGVEGVRLAVREEIQKGATQIKIMASGGVASPTDPIANTQYSEDEIRAIVDEAEAANTYVMAHAYTGRAIARAVRCGVRTIEHGNLVDEAAAKLMHEHGAFVVPTLVTYDALAKHGAEFGMPPESVAKVASVQQKGRESLEIYANAGVKMGFGSDLLGEMHAFQSGEFRIRAEVLGNLEALRSATTVAAEIVNMQGQLGVIAVGAIADLVVLDGNPLEDIGVVADEGARVEYVLQRGTLVKRQ 3n2e A 2.53 BS01 OSA A 1 F9 R45 F48 R57 G80 G81 M84 R116 R132 L135 Y136 F9 R45 F48 R57 G80 G81 M84 R116 R132 L135 Y136 2.7.1.71 0000287,0004765,0005524,0005737,0005829,0008652,0009073,0009423,0016301,0019752,0046872 remove_due_to_license_issue P56073 22438938 1001 MQHLVLIGFMGSGKSSLAQELGLALKLEVLDTDMIISERVGLSVREIFEELGEDNFRMFEKNLIDELKTLKTPHVISTGGGIVMHENLKGLGTTFYLKMDFETLIKRLNQKERAKRPLLNNLTQAKELFEKRQALYEKNASFIIDARGGLNNSLKQVLQFIALQPSLS 3n2p A 1.648 BS02 AYX A 1 I91 Q92 H94 H119 F131 L198 T199 T200 I89 Q90 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=15nM remove_due_to_license_issue Ki=15nM P00918 20922253 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3n2u A 1.81 BS06 D3X A 1 I180 L181 A182 H218 E219 H222 H228 Y240 I75 L76 A77 H113 E114 H117 H123 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=14nM P39900 20965620 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3n2v A 1.55 BS06 JT5 A 1 I180 L181 A182 L214 T215 H218 E219 H222 H228 V235 P238 T239 Y240 I75 L76 A77 L109 T110 H113 E114 H117 H123 V130 P133 T134 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=31nM P39900 20965620 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3n3g A 1.6 BS02 93N A 1 Y18 G20 F146 L147 R149 W186 N189 F190 Y18 G20 F146 L147 R149 W186 N189 F190 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue EC50=138nM, IC50=58nM P25774 20580231 221 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 3n3j A 1.5 BS02 WWV A 1 H94 H96 F131 L198 T199 T200 H92 H94 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.3nM remove_due_to_license_issue Ki=3.3nM P00918 20922253 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3n3l F 2.74 BS01 MS0 F 1 N59 R60 T63 F206 F239 L344 K347 N52 R53 T56 F199 F232 L337 K340 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=>500000000nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n3l F 2.74 BS02 MS0 F 2 L315 E318 E319 Y322 L308 E311 E312 Y315 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=>500000000nM P14324 20711197 2 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n45 F 1.88 BS01 3N3 F 1 K57 N59 R60 F206 F239 Q242 L344 I348 K50 N52 R53 F199 F232 Q235 L337 I341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=>500000000nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n46 F 2.35 BS01 3N5 F 1 K57 N59 R60 T63 F239 L344 K347 I348 K50 N52 R53 T56 F232 L337 K340 I341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=5.0e+4nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n49 F 2.5 BS01 3N4 F 1 K57 N59 R60 T63 F206 L344 K347 I348 K50 N52 R53 T56 F199 L337 K340 I341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=7uM remove_due_to_license_issue IC50=7e+3nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n4b A 1.6 BS02 WWZ A 1 H94 H119 L198 T199 T200 P202 H92 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=96nM remove_due_to_license_issue Ki=960nM P00918 20922253 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3n4c A 1.9 BS01 EF3 A 1 G23 C25 G68 G69 F70 N163 G165 G23 C25 G68 G69 F70 N163 G165 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue P25774 20598883 218 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 3n4l A 2.7 BS01 842 A 1 D38 G40 P76 Y77 T78 F114 I132 Y204 I232 D234 G236 D35 G37 P73 Y74 T75 F111 I129 Y189 I217 D219 G221 D38 S41 N43 A45 Y77 D234 T237 D35 S38 N40 A42 Y74 D219 T222 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=59nM P56817 20634069 407 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3n51 A 2.1 BS01 BK3 A 1 V65 A78 V79 K80 M112 L126 V130 Y131 E135 L181 D195 V21 A34 V35 K36 M68 L82 V86 Y87 E91 L137 D151 D174 K176 E178 N179 D195 T214 D130 K132 E134 N135 D151 T170 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue IC50=15.0nM Q9BJF5 21116453 701 AIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3n5h F 2.2 BS01 GO0 F 1 N59 R60 S205 F206 F239 K347 N52 R53 S198 F199 F232 K340 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=2uM remove_due_to_license_issue IC50=2e+3nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n5h F 2.2 BS02 GO0 F 2 S109 L110 T111 T260 D264 K293 S102 L103 T104 T253 D257 K286 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=2uM remove_due_to_license_issue IC50=2e+3nM P14324 20711197 2 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n5j F 2.35 BS01 GO1 F 1 K57 N59 R60 S205 F206 F239 K347 K50 N52 R53 S198 F199 F232 K340 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=6uM remove_due_to_license_issue IC50=6e+3nM P14324 20711197 1 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n5j F 2.35 BS02 GO1 F 2 S109 L110 T111 T260 D264 S102 L103 T104 T253 D257 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=6uM remove_due_to_license_issue IC50=6e+3nM P14324 20711197 2 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n6k F 2.25 BS01 BFH F 1 K57 N59 R60 F206 L344 I348 K48 N50 R51 F197 L335 I339 2.5.1.1,2.5.1.10 0004659,0008299,0016765 Kd=180nM remove_due_to_license_issue IC50=920nM P14324 20711197 1 YAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 3n75 A 2.0 BS01 G4P A 1 R97 R206 K417 G418 R97 R206 K417 G418 H245 D330 K367 H245 D330 K367 4.1.1.18 0003824,0005515,0005737,0006520,0006554,0008923,0016831,0042802,0097216 Kd=12.8nM remove_due_to_license_issue P0A9H3 21278708 716 MNVIAILNHMGVYFKEEPIRELHRALERLNFQIVYPNDRDDLLKLIENNARLCGVIFDWDKYNLELCEEISKMNENLPLYAFANTYSTLDVSLNDLRLQISFFEYALGAAEDIANKIKQTTDEYINTILPPLTKALFKYVREGKYTFCTPGHMGGTAFQKSPVGSLFYDFFGPNTMKSDISISVSELGSLLDHSGPHKEAEQYIARVFNADRSYMVTNGTSTANKIVGMYSAPAGSTILIDRNCHKSLTHLMMMSDVTPIYFRPTRNAYGILGGIPQSEFQHATIAKRVKETPNATWPVHAVITNSTYDGLLYNTDFIKKTLDVKSIHFDSAWVPYTNFSPIYEGKCGMSGGRVEGKVIYETQSTHKLLAAFSQASMIHVKGDVNEETFNEAYMMHTTTSPHYGIVASTETAAAMMKGNAGKRLINGSIERAIKFRKEIKRLRTESDGWFFDVWQPDHIDTTECWPLRSDSTWHGFKNIDNEHMYLDPIKVTLLTPGMEKDGTMSDFGIPASIVAKYLDEHGIVVEKTGPYNLLFLFSIGIDKTKALSLLRALTDFKRAFDLNLRVKNMLPSLYREDPEFYENMRIQELAQNIHKLIVHHNLPDLMYRAFEVLPTMVMTPYAAFQKELHGMTEEVYLDEMVGRINANMILPYPPGVPLVMPGEMITEESRPVLEFLQMLCEIGAHYPGFETDIHGAYRQADGRYTVKVLKE 3n75 A 2.0 BS02 G4P C 1 R558 L564 R565 N568 R585 R558 L564 R565 N568 R585 H245 D330 K367 H245 D330 K367 4.1.1.18 0003824,0005515,0005737,0006520,0006554,0008923,0016831,0042802,0097216 Kd=12.8nM remove_due_to_license_issue P0A9H3 21278708 716 MNVIAILNHMGVYFKEEPIRELHRALERLNFQIVYPNDRDDLLKLIENNARLCGVIFDWDKYNLELCEEISKMNENLPLYAFANTYSTLDVSLNDLRLQISFFEYALGAAEDIANKIKQTTDEYINTILPPLTKALFKYVREGKYTFCTPGHMGGTAFQKSPVGSLFYDFFGPNTMKSDISISVSELGSLLDHSGPHKEAEQYIARVFNADRSYMVTNGTSTANKIVGMYSAPAGSTILIDRNCHKSLTHLMMMSDVTPIYFRPTRNAYGILGGIPQSEFQHATIAKRVKETPNATWPVHAVITNSTYDGLLYNTDFIKKTLDVKSIHFDSAWVPYTNFSPIYEGKCGMSGGRVEGKVIYETQSTHKLLAAFSQASMIHVKGDVNEETFNEAYMMHTTTSPHYGIVASTETAAAMMKGNAGKRLINGSIERAIKFRKEIKRLRTESDGWFFDVWQPDHIDTTECWPLRSDSTWHGFKNIDNEHMYLDPIKVTLLTPGMEKDGTMSDFGIPASIVAKYLDEHGIVVEKTGPYNLLFLFSIGIDKTKALSLLRALTDFKRAFDLNLRVKNMLPSLYREDPEFYENMRIQELAQNIHKLIVHHNLPDLMYRAFEVLPTMVMTPYAAFQKELHGMTEEVYLDEMVGRINANMILPYPPGVPLVMPGEMITEESRPVLEFLQMLCEIGAHYPGFETDIHGAYRQADGRYTVKVLKE 3n75 D 2.0 BS01 G4P A 1 R558 L564 R565 N568 R585 R558 L564 R565 N568 R585 H245 D330 K367 H245 D330 K367 4.1.1.18 0003824,0005515,0005737,0006520,0006554,0008923,0016831,0042802,0097216 Kd=12.8nM remove_due_to_license_issue P0A9H3 21278708 716 MNVIAILNHMGVYFKEEPIRELHRALERLNFQIVYPNDRDDLLKLIENNARLCGVIFDWDKYNLELCEEISKMNENLPLYAFANTYSTLDVSLNDLRLQISFFEYALGAAEDIANKIKQTTDEYINTILPPLTKALFKYVREGKYTFCTPGHMGGTAFQKSPVGSLFYDFFGPNTMKSDISISVSELGSLLDHSGPHKEAEQYIARVFNADRSYMVTNGTSTANKIVGMYSAPAGSTILIDRNCHKSLTHLMMMSDVTPIYFRPTRNAYGILGGIPQSEFQHATIAKRVKETPNATWPVHAVITNSTYDGLLYNTDFIKKTLDVKSIHFDSAWVPYTNFSPIYEGKCGMSGGRVEGKVIYETQSTHKLLAAFSQASMIHVKGDVNEETFNEAYMMHTTTSPHYGIVASTETAAAMMKGNAGKRLINGSIERAIKFRKEIKRLRTESDGWFFDVWQPDHIDTTECWPLRSDSTWHGFKNIDNEHMYLDPIKVTLLTPGMEKDGTMSDFGIPASIVAKYLDEHGIVVEKTGPYNLLFLFSIGIDKTKALSLLRALTDFKRAFDLNLRVKNMLPSLYREDPEFYENMRIQELAQNIHKLIVHHNLPDLMYRAFEVLPTMVMTPYAAFQKELHGMTEEVYLDEMVGRINANMILPYPPGVPLVMPGEMITEESRPVLEFLQMLCEIGAHYPGFETDIHGAYRQADGRYTVKVLKE 3n75 D 2.0 BS02 G4P D 1 R97 R206 K417 G418 R97 R206 K417 G418 H245 D330 K367 H245 D330 K367 4.1.1.18 0003824,0005515,0005737,0006520,0006554,0008923,0016831,0042802,0097216 Kd=12.8nM remove_due_to_license_issue P0A9H3 21278708 716 MNVIAILNHMGVYFKEEPIRELHRALERLNFQIVYPNDRDDLLKLIENNARLCGVIFDWDKYNLELCEEISKMNENLPLYAFANTYSTLDVSLNDLRLQISFFEYALGAAEDIANKIKQTTDEYINTILPPLTKALFKYVREGKYTFCTPGHMGGTAFQKSPVGSLFYDFFGPNTMKSDISISVSELGSLLDHSGPHKEAEQYIARVFNADRSYMVTNGTSTANKIVGMYSAPAGSTILIDRNCHKSLTHLMMMSDVTPIYFRPTRNAYGILGGIPQSEFQHATIAKRVKETPNATWPVHAVITNSTYDGLLYNTDFIKKTLDVKSIHFDSAWVPYTNFSPIYEGKCGMSGGRVEGKVIYETQSTHKLLAAFSQASMIHVKGDVNEETFNEAYMMHTTTSPHYGIVASTETAAAMMKGNAGKRLINGSIERAIKFRKEIKRLRTESDGWFFDVWQPDHIDTTECWPLRSDSTWHGFKNIDNEHMYLDPIKVTLLTPGMEKDGTMSDFGIPASIVAKYLDEHGIVVEKTGPYNLLFLFSIGIDKTKALSLLRALTDFKRAFDLNLRVKNMLPSLYREDPEFYENMRIQELAQNIHKLIVHHNLPDLMYRAFEVLPTMVMTPYAAFQKELHGMTEEVYLDEMVGRINANMILPYPPGVPLVMPGEMITEESRPVLEFLQMLCEIGAHYPGFETDIHGAYRQADGRYTVKVLKE 3n76 A 1.9 BS01 CA2 A 1 N12 R15 R19 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N11 R14 R18 Y23 N74 G76 G77 H80 H100 I101 S102 R111 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P10 N11 R18 Y23 N74 G77 E98 H100 R107 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=0.14uM remove_due_to_license_issue P9WPX7 21410435 147 ELIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEHV 3n7a A 2.0 BS01 FA1 A 1 Y24 N75 G77 G78 H81 H101 I102 S103 R112 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=200uM remove_due_to_license_issue Kd=200000nM, Ki=200000nM P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n7a L 2.0 BS01 FA1 L 1 Y24 N75 G77 G78 H81 H101 I102 S103 R112 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=200uM remove_due_to_license_issue Kd=200000nM, Ki=200000nM P9WPX7 21410435 148 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n7h A 1.6 BS01 DE3 A 1 L76 H77 A88 M89 G92 W114 L76 H77 A88 M89 G92 W114 ? 0005549,0005576 Kd=31.3uM remove_due_to_license_issue Q8T6S0 21671117 129 DTTPRRDAEYPPPELLEALKPLHDICLGKTGVTEEAIKKFSDEEIHEDEKLKCYMNCLFHEAKVVDDNGDVHLEKLHDSLPSSMHDIAMHMGKRCLYPEGETLCDKAFWLHKCWKQSDPKHYFLV 3n7h B 1.6 BS01 DE3 B 1 L76 H77 A88 G92 L96 W114 L76 H77 A88 G92 L96 W114 ? 0005549,0005576 Kd=31.3uM remove_due_to_license_issue Q8T6S0 21671117 132 DTTPRRDAEYPPPELLEALKPLHDICLGKTGVTEEAIKKFSDEEIHEDEKLKCYMNCLFHEAKVVDDNGDVHLEKLHDSLPSSMHDIAMHMGKRCLYPEGETLCDKAFWLHKCWKQSDPKHYFLV 3n7o A 1.8 BS01 N7O A 1 H57 Y94 N95 T96 L99 D102 A190 F191 K192 S195 S214 Y215 G216 H45 Y81 N82 T83 L86 D89 A174 F175 K176 S179 S194 Y195 G196 H57 D102 K192 G193 D194 S195 G196 H45 D89 K176 G177 D178 S179 G180 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 Ki=72nM remove_due_to_license_issue IC50=58nM P23946 20599788 1 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPSFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 3n7s A 2.1 BS01 3N6 A 1 I41 G71 W72 F92 D94 R119 W121 T122 Y124 I10 G37 W38 F58 D60 R85 W87 T88 Y90 ? 0004930,0004948,0007186,0016020 Kd<20nM remove_due_to_license_issue IC50=0.030000nM, Ki=0.010000nM, EC50=0.026000nM Q16602 20826335 1 IQLGVTRNKIMTAQYECYQKIMQDPIEGVYCNRTWDGWLCWNDVAAGTESMQLCPDYFQDFDPSEKVTKICDQDGNWFRHPASNRTWTNYTQCN 3n7s D 2.1 BS01 3N6 A 1 A70 D71 W74 W84 A44 D45 W48 W58 ? 0006886,0008277,0015026,0016020 remove_due_to_license_issue O60894 20826335 1 CQEANYGALLRELCLTQFQVDMEAVGETLWCDWGRTIRSYRELADCTWHMAEKLGCFWPNAEVDRFFLAVHGRYFRSCPISGRA 3n86 A 1.9 BS01 RJP A 1 N12 R15 E20 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N10 R13 E18 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=2.3uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n86 A 1.9 BS02 RJP K 1 D88 E92 D86 E90 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=2.3uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n86 L 1.9 BS01 RJP A 1 D88 E92 D86 E90 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=2.3uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n86 L 1.9 BS02 RJP L 1 N12 E20 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N10 E18 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=2.3uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n87 A 2.4 BS01 N87 A 1 N12 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N10 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=11uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n87 L 2.4 BS01 N87 A 1 D88 E92 D86 E90 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=11uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n87 L 2.4 BS02 N87 L 1 N12 R19 E20 Y24 N75 G77 G78 H101 I102 S103 R112 N10 R17 E18 Y22 N73 G75 G76 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=11uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n8k A 2.25 BS01 D1X A 1 R19 Y24 N75 G77 H81 H101 I102 S103 R112 R17 Y22 N73 G75 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Kd=90uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEHV 3n8k L 2.25 BS01 D1X L 1 R19 Y24 N75 G77 H81 H101 I102 S103 R112 R17 Y22 N73 G75 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Kd=90uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n8n A 2.5 BS01 N88 A 1 N75 G77 G78 H101 I102 S103 R112 N69 G71 G72 H95 I96 S97 R106 P11 N12 N75 G78 E99 H101 R108 P9 N10 N69 G72 E93 H95 R102 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=27uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRREPGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n8n L 2.5 BS01 N88 L 1 N12 N75 G77 G78 H81 H101 I102 S103 R112 N10 N66 G68 G69 H72 H92 I93 S94 R103 P11 N12 N75 G78 E99 H101 R108 P9 N10 N66 G69 E90 H92 R99 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=27uM remove_due_to_license_issue P9WPX7 21410435 147 LIVNVINGPNLGRLGRGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 3n9r A 1.8 BS02 TD3 A 1 H83 H180 G181 K184 H210 G211 S213 N253 D255 T256 H83 H170 G171 K174 H200 G201 S203 N243 D245 T246 C69 E70 G136 H180 A226 N253 C69 E70 G136 H170 A216 N243 0004332,0005975,0006096,0008270,0016832,0030388 Ki=5.5uM remove_due_to_license_issue 20929256 311 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMGIAVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3n9r e 1.8 BS02 TD3 e 1 D82 H83 H180 G181 K184 H210 G211 S213 N253 D255 T256 D82 H83 H170 G171 K174 H200 G201 S203 N243 D245 T246 0004332,0005975,0006096,0008270,0016832,0030388 remove_due_to_license_issue 20929256 311 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMGIAVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3n9s A 1.85 BS01 TD4 A 1 N23 S49 D82 H83 H180 G181 K184 H210 G211 S213 N253 D255 T256 N23 S49 D82 H83 H180 G181 K184 H210 G211 S213 N253 D255 T256 C69 E70 G136 H180 A226 N253 C69 E70 G136 H180 A226 N253 0004332,0005975,0006096,0008270,0016832,0030388 Ki=0.07uM remove_due_to_license_issue 20929256 308 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMGIEDNISVDEKDAVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3n9s B 1.85 BS03 TD4 B 1 N23 S49 D82 H83 H180 G181 K184 H210 G211 S213 N253 D255 T256 N23 S49 D82 H83 H168 G169 K172 H198 G199 S201 N241 D243 T244 C69 E70 G136 H180 A226 N253 C69 E70 G136 H168 A214 N241 0004332,0005975,0006096,0008270,0016832,0030388 Ki=0.07uM remove_due_to_license_issue 20929256 311 MLVKGNEILLKAHKEGYGVGAFNFVNFEMLNAIFEAGNEENSPLFIQASEGAIKYMGIDMAVGMVKIMCERYPHIPVALHLDHGTTFESCEKAVKAGFTSVMIDASHHAFEENLELTSKVVKMAHNAGVSVEAELGRLMAVLVNPKEAEQFVKESQVDYLAPAIGTSHGAFKFKGEPKLDFERLQEVKRLTNIPLVLHGASAIPDNVRKSYLDAGGDLKGSKGVPFEFLQESVKGGINKVNTDTDLRIAFIAEVRKVANEDKSQFDLRKFFSPAQLALKNVVKERMKLLGSANKI 3nae A 2.003 BS01 dna T 0 E219 I253 E254 R260 K279 F359 S360 P361 I362 Y391 P392 G393 A394 S565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 K279 F359 S360 P361 I362 Y391 P392 G393 A394 S565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 20795733 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nae A 2.003 BS02 dna P 0 N284 T622 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 T622 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 20795733 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nal A 2.65 BS01 DBK A 1 L249 L253 E255 F256 Q259 L260 V263 V772 L828 I829 F834 L249 L253 E255 F256 Q259 L260 V263 V772 L828 I829 F834 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005515,0005524,0006816,0016020,0016529,0016887,0033017,0046872,0070588 remove_due_to_license_issue B6CAM1 20551329 997 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 3nam A 3.1 BS02 OTK A 1 E255 F256 L260 V772 F834 Y837 E255 F256 L260 V772 F834 Y837 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005515,0005524,0006816,0016020,0016529,0016887,0033017,0046872,0070588 remove_due_to_license_issue B6CAM1 20551329 997 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 3nan A 3.1 BS01 HZ1 A 1 L253 E255 F256 Q259 L260 V263 I307 P308 E309 P312 I765 V772 V773 L828 I829 F834 L253 E255 F256 Q259 L260 V263 I307 P308 E309 P312 I765 V772 V773 L828 I829 F834 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005515,0005524,0006816,0016020,0016529,0016887,0033017,0046872,0070588 remove_due_to_license_issue B6CAM1 20551329 997 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 3nb5 A 1.8 BS02 R21 A 1 H94 H119 F130 G131 L197 T198 T199 H91 H116 F127 G128 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=18nM remove_due_to_license_issue Ki=18nM P00918 21332115 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3nba A 2.68 BS01 APC A 1 S9 F10 G16 H17 I20 G88 R90 T118 S126 S127 S128 S9 F10 G16 H17 I20 G88 R90 T118 S126 S127 S128 H17 K41 R90 S127 H17 K41 R90 S127 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779,0034214 remove_due_to_license_issue P9WPA5 20851704 200 MTGAVCPGSFDPVTLGHVDIFERAAAQFDEVVVAILVNPAKTGMFDLDERIAMVKESTTHLPNLRVQVGHGLVVDFVRSCGMTAIVKGLRTGTDFEYELQMAQMNKHIAGVDTFFVATAPRYSFVSSSLAKEVAMLGGDVSELLPEPVNRRLRDRL 3nba C 2.68 BS01 APC C 1 S9 F10 G16 H17 I20 G88 R90 T118 V125 S126 S127 S128 S9 F10 G16 H17 I20 G88 R90 T118 V125 S126 S127 S128 H17 K41 R90 S127 H17 K41 R90 S127 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779,0034214 remove_due_to_license_issue P9WPA5 20851704 200 MTGAVCPGSFDPVTLGHVDIFERAAAQFDEVVVAILVNPAKTGMFDLDERIAMVKESTTHLPNLRVQVGHGLVVDFVRSCGMTAIVKGLRTGTDFEYELQMAQMNKHIAGVDTFFVATAPRYSFVSSSLAKEVAMLGGDVSELLPEPVNRRLRDRL 3nc4 A 2.07 BS01 26O A 1 E88 N133 G135 L136 D283 N284 H341 H377 N484 E672 S674 G675 E77 N122 G124 L125 D266 N267 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=26.6uM remove_due_to_license_issue P00489 20947361 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3nc4 A 2.07 BS02 26O A 2 R60 V64 W67 E190 K191 A192 P229 R49 V53 W56 E179 K180 A181 P218 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=26.6uM remove_due_to_license_issue P00489 20947361 920 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3nc9 A 2.4 BS01 TR3 B 1 A226 E227 G229 P246 A256 F260 C282 A285 C289 A224 E225 G227 P244 A254 F258 C280 A283 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=590nM P50053 21033679 299 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3nc9 B 2.4 BS01 TR3 B 2 A226 G229 P246 A256 A229 G232 P249 A259 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=330nM remove_due_to_license_issue IC50=590nM P50053 21033679 300 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3ncg A 2.49 BS04 BK1 A 1 V90 A103 K105 M136 I150 L154 Y155 L205 V25 A38 K40 M71 I85 L89 Y90 L140 D198 K200 E202 N203 D219 T238 D133 K135 E137 N138 D154 T168 2.7.11.17 0004672,0005509,0005524,0006468 remove_due_to_license_issue A3FQ16 21116453 561 LYFQGTFAERYNIVCMLGKGSFGEVLKCKDRITQQEYAVKVINKASAKNKDTSTILREVELLKKLDHPNIMKLFEILEDSSSFYIVGELYTGGELFDEIIKRKRFSEHDAARIIKQVFSGITYMHKHNIVHRDLKPENILLESKEKDCDIKIIDFGLSTCFQQNTIGTAYYIAPEVLRGTYDEKCDVWSAGVILYILLSGTPPFYGKNEYDILKRVETGKYAFDLPQWRTISDDAKDLIRKMLTFHPSLRITATQCLEHPWIQKYSSETPTISDLPSLESAMTNIRQFQAEKKLAQAALLYMASKLTTLDETKQLTEIFRKLDTNNDGMLDRDELVRGYHEFMRLKGVDSNGSTIEDQIDSLMPLLDMDGSGSIEYSEFIASAIDRTILLSRERMERAFKMFDKDGSGKISTKELDFNEFVEMLQN 3nci A 1.79 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 N564 S565 Y567 G568 G571 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 N564 S565 Y567 G568 G571 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21158418 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nci A 1.79 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21158418 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3ncq A 1.24 BS01 ATP A 1 G35 R36 G37 Q38 Q39 P86 G87 G89 K90 G35 R36 G37 Q38 Q39 P86 G87 G89 K90 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 201 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSL 3ncq A 1.24 BS02 ATP C 1 G27 M28 T29 V64 R101 R103 G27 M28 T29 V64 R101 R103 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 200 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSL 3ncq B 1.24 BS01 ATP A 1 G27 M28 T29 V64 R101 R103 G27 M28 T29 V64 R101 R103 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 201 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSL 3ncq B 1.24 BS02 ATP B 1 G35 R36 G37 Q38 Q39 P86 G87 G89 K90 G35 R36 G37 Q38 Q39 P86 G87 G89 K90 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 202 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSL 3ncr A 1.44 BS01 ADP A 1 G35 R36 G37 Q38 Q39 G87 G89 K90 G35 R36 G37 Q38 Q39 G87 G89 K90 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 120 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSLE 3ncr A 1.44 BS04 ADP C 1 G27 M28 T29 V64 E113 G27 M28 T29 V64 E113 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 120 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSLE 3ncr B 1.44 BS01 ADP A 1 G27 M28 T29 V64 G27 M28 T29 V64 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 120 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSL 3ncr B 1.44 BS03 ADP B 1 G35 R36 G37 Q38 Q39 P86 G87 G89 K90 G35 R36 G37 Q38 Q39 P86 G87 G89 K90 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28527 20643148 120 MKKIEAIVRAEKFPEVKAALEERGFYGMTVTDVKGRGQQGGMQIQFRGRTMEVTLLPKVKLEIVVKDDAVEEVIGLIVNSAFTGSPGDGKIFIIPVEDVVRIRTGERGDDSL 3ncu A 2.55 BS01 rna C 0 C829 H830 H847 F853 K858 K861 G874 I875 K888 K907 C26 H27 H44 F50 K55 K58 G71 I72 K85 K104 3.6.4.13 remove_due_to_license_issue O95786 20581823 1 ~ 12 ENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 3ncu A 2.55 BS02 rna D 0 K849 F853 S854 K46 F50 S51 3.6.4.13 remove_due_to_license_issue O95786 20581823 1 ~ 12 ENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 3ncu B 2.55 BS01 rna D 0 C829 H830 H847 K851 F853 K858 K861 G874 I875 K888 K907 W908 C26 H27 H44 K48 F50 K55 K58 G71 I72 K85 K104 W105 3.6.4.13 remove_due_to_license_issue O95786 20581823 1 ~ 12 ENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 3ncz A 3.0 BS01 3NC A 1 I82 A103 D202 N203 L205 A215 D216 I79 A100 D199 N200 L202 A212 D213 D198 K200 N203 D216 T237 D195 K197 N200 D213 T234 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q13464 20678931 900 HMSFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3ndk A 2.0 BS01 dna T 0 E219 I253 E254 R260 F359 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 F359 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3ndk A 2.0 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 K800 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3ndm B 3.3 BS01 3ND B 1 R84 G85 V90 A103 M153 M156 D202 L205 A215 R78 G79 V84 A97 M147 M150 D196 L199 A209 D198 K200 N203 D216 T237 D192 K194 N197 D210 T231 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q13464 20471253 900 FETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3ne6 A 2.001 BS01 dna T 0 E219 I253 E254 N255 R260 F359 S360 P361 I362 Y391 P392 G393 A394 L561 N564 G565 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 E219 I253 E254 N255 R260 F359 S360 P361 I362 Y391 P392 G393 A394 L561 N564 G565 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3ne6 A 2.001 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nef A 2.4 BS01 PYV A 1 I68 V87 A95 S98 E100 H121 L123 Y126 V172 I66 V85 A93 S96 E98 H119 L121 Y124 V165 3.1.3.16 0004864,0005515,0005634,0005737,0005886,0006952,0009536,0009738,0010427,0038023,0042802,0042803,0062049,0080163 remove_due_to_license_issue Q8VZS8 20554531 201 HHQTMPSDLTQDEFTQLSQSIAEFHTYQLGNGRCSSLLAQRIHAPPETVWSVVRRFDRPQIYKHFIKSCNVSEDFEMRVGCTRDVNVISGLPANTSRERLDLLDDDRRVTGFSITGGEHRLRNYKSVTTVHRFEKRIWTVVLESYVVDVPEGNSEEDTRLFADTVIRLNLQKLASITEAMNR 3neg A 2.801 BS01 PYV A 1 K65 I68 V87 A95 S98 E100 H121 Y126 K63 I66 V85 A93 S96 E98 H119 Y124 3.1.3.16 0004864,0005515,0005634,0005737,0005886,0006952,0009536,0009738,0010427,0038023,0042802,0042803,0062049,0080163 remove_due_to_license_issue Q8VZS8 20554531 201 HHQTMPSDLTQDEFTQLSQSIAEFHTYQLGNGRCSSLLAQRIHAPPETVWSVVRRFDRPQIYKHFIKSCNVSEDFEMRVGCTRDVNVISGLPANTSRERLDLLDDDRRVTGFSITGGEHRLRNYKSVTTVHRFEKRIWTVVLESYVVDVPEGNSEEDTRLFADTVIRLNLQKLASITEAMNR 3neo A 2.0 BS01 G24 A 1 M13 K15 E54 A108 L110 M4 K6 E45 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 20937391 1 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3neo B 2.0 BS01 G24 B 1 S117 T118 T119 S106 T107 T108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 20937391 1 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSRRYTIAALLSPYSYSTTAVVTNP 3nes A 1.75 BS01 B72 A 1 K15 L17 E54 A108 A109 L110 K6 L8 E45 A99 A100 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 20937391 1 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3nes B 1.75 BS01 B72 B 1 M13 K15 L17 A108 A109 L110 M4 K6 L8 A99 A100 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 20937391 1 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3new A 2.51 BS01 3NE A 1 E192 L195 W197 K249 I250 S251 S252 I259 L291 E174 L177 W179 K231 I232 S233 S234 I241 L273 D150 K152 N155 D168 T185 D144 K146 N149 D162 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 21090814 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3nex A 1.7 BS01 G24 A 1 M13 K15 L17 E54 A108 L110 M4 K6 L8 E45 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 20937391 126 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3nex B 1.7 BS01 G24 B 1 A108 L110 S117 T119 A99 L101 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 20937391 126 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3nf6 A 1.9 BS01 IMV A 1 A169 E170 H171 T174 M178 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=295uM remove_due_to_license_issue P12497 21602613 215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf6 A 1.9 BS02 IMV A 2 V79 G82 V150 M154 E157 H183 V23 G26 V94 M98 E101 H127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=295uM remove_due_to_license_issue P12497 21602613 230 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf6 A 1.9 BS03 IMV B 1 Q95 L102 A128 A129 W132 Q39 L46 A72 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=295uM remove_due_to_license_issue P12497 21602613 216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf6 B 1.9 BS01 IMV A 1 Q95 T125 A128 A129 W132 Q39 T69 A72 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=295uM remove_due_to_license_issue P12497 21602613 215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf6 B 1.9 BS02 IMV B 1 A169 E170 H171 T174 M178 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=295uM remove_due_to_license_issue P12497 21602613 216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf6 B 1.9 BS03 IMV B 2 G82 V150 M154 E157 H183 G26 V94 M98 E101 H127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=295uM remove_due_to_license_issue P12497 21602613 231 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf7 A 1.8 BS01 CIW A 1 V77 V79 G82 V150 M154 E157 L158 H183 V21 V23 G26 V94 M98 E101 L102 H127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=340uM remove_due_to_license_issue P12497 21602613 221 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 A 1.9 BS01 CDQ A 1 R107 P109 I204 D207 I208 R51 P53 I144 D147 I148 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 225 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 A 1.9 BS02 CDQ A 2 V79 G82 I84 V150 M154 E157 H183 V23 G26 I28 V94 M98 E101 H127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 247 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 A 1.9 BS03 CDQ A 3 E170 H171 T174 M178 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 267 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 A 1.9 BS04 CDQ A 4 H185 S195 G197 E198 H129 S135 G137 E138 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 277 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 A 1.9 BS05 CDQ B 1 Q95 Y99 T125 A129 W132 Q39 Y43 T69 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 235 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 B 1.9 BS01 CDQ A 1 H185 S195 G197 E198 H129 S135 G137 E138 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 225 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 B 1.9 BS02 CDQ A 3 Q95 Y99 T125 A129 W132 Q39 Y43 T69 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 267 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 B 1.9 BS03 CDQ A 4 R107 P109 I204 D207 R51 P53 I144 D147 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 277 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 B 1.9 BS04 CDQ B 1 E170 H171 K173 T174 M178 E114 H115 K117 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 235 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf8 B 1.9 BS05 CDQ B 2 V79 G82 I84 V150 M154 E157 L158 H183 V23 G26 I28 V94 M98 E101 L102 H127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 21602613 257 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nf9 A 1.95 BS01 CD9 A 1 V79 G82 V150 S153 M154 H183 V23 G26 V94 S97 M98 H127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=290uM remove_due_to_license_issue P12497 21602613 220 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3nga A 2.71 BS01 3NG A 1 L45 G46 V53 V66 K68 F113 H115 V116 H160 I174 D175 L44 G45 V52 V65 K67 F112 H114 V115 H159 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=2000nM, Kd=0.562341nM, Ki=0.380000nM P68400 21093442 1000 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 3ngi A 1.886 BS01 dna T 0 E219 I253 E254 R260 F359 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 F359 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3ngi A 1.886 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 K800 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nhg A 2.5 BS01 dna T 0 E219 I253 E254 N255 Y257 R260 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 N572 K705 R707 N786 K800 F803 K844 K874 E219 I253 E254 N255 Y257 R260 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 N572 K705 R707 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nhg A 2.5 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 21216248 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3nhi A 1.43 BS01 EAH A 1 L13 Y16 Y20 W37 W40 L42 Y52 V56 L60 Y117 G134 T135 K152 L12 Y15 Y19 W36 W39 L41 Y51 V55 L59 Y116 G133 T134 K151 ? 0005549,0005576,0005615,0007608,0035821,0042311,0090729 remove_due_to_license_issue Q95NY5 21152418 1 QPWKALDAEQALYVYKRCYEDHLPSGSDRKTYMTLWNAWRLEPNDAITHCYAKCVLTGLQIYDPQENAFKSDRIPVQYQAYKTITQSKQKEVTEYQKALAAANAKSGSCVDLYNAYLPVHNRFVNLSRQLYHGTVEGAAKIYAAMPEIKQKGESFHAYCEKRAWKGNKQSEWKNGRRYKLTGSPELKDAIDCIFRGLRYMDDTGLKVDEIVRDFNLINKSELEPEVRSVLASCKGSEAYDYYVCLVNSRLKQHFKNAFDFHELRSADYAYLLRKVYENPEKVKEEMKKLNTTVHF 3nht A 1.45 BS01 U46 A 1 Y16 Y20 W37 W40 L42 Y52 V56 G134 T135 K152 Y15 Y19 W36 W39 L41 Y51 V55 G133 T134 K151 ? 0005549,0005576,0005615,0007608,0035821,0042311,0090729 Kd=98nM remove_due_to_license_issue Q95NY5 21152418 1 QPWKALDAEQALYVYKRCYEDHLPSGSDRKTYMTLWNAWRLEPNDAITHCYAKCVLTGLQIYDPQENAFKSDRIPVQYQAYKTITQSKQKEVTEYQKALAAANAKSGSCVDLYNAYLPVHNRFVNLSRQLYHGTVEGAAKIYAAMPEIKQKGESFHAYCEKRAWKGNKQSEWKNGRRYKLTGSPELKDAIDCIFRGLRYMDDTGLKVDEIVRDFNLINKSELEPEVRSVLASCKGSEAYDYYVCLVNSRLKQHFKNAFDFHELRSADYAYLLRKVYENPEKVKEEMKKLNTTVHF 3ni5 A 2.1 BS02 C1H A 1 Q92 H94 H119 F131 L198 T199 T200 P202 Q89 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=28nM remove_due_to_license_issue Ki=28nM P00918 21549597 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3nif A 2.4 BS05 NIF A 1 F160 Y190 L192 D224 S225 F231 F160 Y190 L192 D224 S225 F231 ? 0007155,0008305 remove_due_to_license_issue IC50=9700nM P08514 20679525 455 LNLDPVQLTFYAGPNGSQFGFSLDFHKDSHGRVAIVVGAPRTLGPSQEETGGVFLCPWRAEGGQCPSLLFDLRDETRNVGSQTLQTFKARQGLGASVVSWSDVIVACAPWQHWNVLEKTEEAEKTPVGSCFLAQPESGRRAEYSPCRGNTLSRIYVENDFSWDKRYCEAGFSSVVTQAGELVLGAPGGYYFLGLLAQAPVADIFSSYRPGILLWHVSSQSLSFDSSNPEYFDGYWGYSVAVGEFDGDLNTTEYVVGAPTWSWTLGAVEILDSYYQRLHRLRGEQMASYFGHSVAVTDVNGDGRHDLLVGAPLYMESRADRKLAEVGRVYLFLQPRGPHALGAPSLLLTGTQLYGRFGSAIAPLGDLDRDGYNDIAVAAPYGGPSGRGQVLVFLGQSEGLRSRPSQVLDSPFPTGSAFGFSLRGAVDIDDNGYPDLIVGAYGANQVAVYRAQPVV 3njq B 2.0 BS01 NJQ B 1 L79 L83 V89 A90 I105 L106 W109 S191 P192 L193 L76 L80 V86 A87 I102 L103 W106 S184 P185 L186 H46 S114 S116 H134 R142 R143 H43 S111 S113 H127 R135 R136 3.4.21.97 0004252,0006508 Kd=1.7uM remove_due_to_license_issue P88911 21723875 198 GLYVGGFVDVVSCPKLEQELYLDPDQVTDYLPVTEPLPITIEHLPETEVGWTLGLFQVSHGIFCTGAITSPAFLELASRLADTSHVARAPVKNLPKEPLLEILHTWLPGLSLSSIHPREPSGPVFQHVSLCALGRRRGTVAVYGHDAEWVVSRFSSVSKSERAHILQHVSSCRLEDLSTPNFVSPLETL 3njq B 2.0 BS02 NJQ B 2 E45 L140 E42 L133 H46 S114 S116 H134 R142 R143 H43 S111 S113 H127 R135 R136 3.4.21.97 0004252,0006508 Kd=1.7uM remove_due_to_license_issue P88911 21723875 199 GLYVGGFVDVVSCPKLEQELYLDPDQVTDYLPVTEPLPITIEHLPETEVGWTLGLFQVSHGIFCTGAITSPAFLELASRLADTSHVARAPVKNLPKEPLLEILHTWLPGLSLSSIHPREPSGPVFQHVSLCALGRRRGTVAVYGHDAEWVVSRFSSVSKSERAHILQHVSSCRLEDLSTPNFVSPLETL 3njy A 2.6 BS02 8XQ A 1 Y132 Y177 F185 H188 K206 W208 H276 Y125 Y170 F178 H181 K199 W201 H269 G170 Y177 H188 E190 H276 S288 G163 Y170 H181 E183 H269 S281 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=1700nM, EC50=87000nM O75164 21124847 360 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 3nk8 A 1.15 BS02 JKZ A 1 S190 Q192 S195 S214 W215 G219 C220 S172 Q174 S177 S192 W193 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 20886466 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3nkk A 1.12 BS02 JLZ A 1 D189 S190 C191 Q192 S214 W215 G219 D171 S172 C173 Q174 S192 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=20uM remove_due_to_license_issue P00760 20886466 1 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3nlb A 1.9 BS01 5BE A 1 L15 G16 E17 V23 A36 E85 Y86 C87 G90 E91 E134 L137 L10 G11 E12 V18 A31 E75 Y76 C77 G80 E81 E124 L127 D130 K132 E134 N135 D148 T170 D120 K122 E124 N125 D138 T160 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=35nM remove_due_to_license_issue O14757 20976184 298 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3nmq A 2.2 BS01 7PP A 1 N51 A55 I96 G97 M98 L107 F138 W162 N39 A43 I84 G85 M86 L95 F126 W150 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P08238 21131419 1 GEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYLEKER 3nmr A 1.85 BS01 rna B 0 K109 F111 G113 M114 R138 L140 R148 G149 C150 F152 S178 S179 V182 K184 A186 D187 K97 F99 G101 M102 R126 L128 R136 G137 C138 F140 S166 S167 V170 K172 A174 D175 ? 0003676,0003723,1990904 remove_due_to_license_issue Q92879 20947024 1 ~ 6 SDAIKMFVGQVPRTWSEKDLRELFEQYGAVYEINVLRDRSQNPPQSKGCCFVTFYTRKAALEAQNALHNMKVLPGMHHPIQMKPADSEKNNAVEDRKLFIGMISKKCTENDIRVMFSSFGQIEECRILRGPDGLSRGCAFVTFTTRAMAQTAIKAMHQAQTMEGCSSPMVVKFAD 3nnu A 2.4 BS01 EDB A 1 A51 K53 R67 R70 E71 I84 L104 T106 I141 H148 D168 F169 A47 K49 R63 R66 E67 I80 L100 T102 I137 H144 D164 F165 D150 K152 N155 D168 T185 D146 K148 N151 D164 T181 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=48nM remove_due_to_license_issue Q16539 20800479 355 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3nnv A 2.1 BS01 437 A 1 A51 K53 R67 R70 E71 L75 I84 L104 T106 L167 D168 F169 A47 K49 R63 R66 E67 L71 I80 L100 T102 L163 D164 F165 D150 K152 N155 D168 T185 D146 K148 N151 D164 T181 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=27nM remove_due_to_license_issue IC50=27nM Q16539 20800479 355 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3nnw A 1.89 BS01 EDD A 1 A51 K53 R67 R70 E71 I84 L104 T106 D168 F169 A48 K50 R64 R67 E68 I81 L101 T103 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=9nM remove_due_to_license_issue Q16539 20800479 355 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3nnx A 2.28 BS01 EDD A 1 A51 K53 R67 R70 E71 L75 I84 L104 T106 L167 D168 F169 A47 K49 R63 R66 E67 L71 I80 L100 T102 L159 D160 F161 D150 K152 N155 D168 T185 D142 K144 N147 D160 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=11nM remove_due_to_license_issue Q16539 20800479 355 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3nox A 2.338 BS01 6A5 A 1 R125 E205 E206 Y547 S630 Y662 Y666 N710 H740 R86 E166 E167 Y508 S591 Y623 Y627 N671 H701 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=2.2nM remove_due_to_license_issue Ki=2.2nM P27487 20684603 1 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3np7 A 2.05 BS01 Z15 A 1 Q96 L494 C495 P497 K544 Y548 E654 K655 Q85 L471 C472 P474 K521 Y525 E631 K632 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=95uM remove_due_to_license_issue IC50=169900nM P00489 21821421 997 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3np7 A 2.05 BS02 Z15 A 2 G135 L136 D283 N284 D339 H341 H377 T378 N484 E672 S674 G675 G124 L125 D269 N270 D316 H318 H354 T355 N461 E649 S651 G652 H377 K568 R569 K574 T676 K680 H354 K545 R546 K551 T653 K657 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=95uM remove_due_to_license_issue IC50=169900nM P00489 21821421 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3np9 A 1.999 BS01 Z2T A 1 G135 L136 D283 N284 D339 H377 T378 N484 E672 S674 G675 G124 L125 D266 N267 D313 H351 T352 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=39.8uM remove_due_to_license_issue IC50=39800nM P00489 21821421 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3npa A 1.969 BS01 Z57 A 1 G135 L136 D283 N284 D339 H341 H377 T378 N484 E672 S674 G675 G124 L125 D266 N267 D313 H315 H351 T352 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=136.4uM remove_due_to_license_issue IC50=136400nM P00489 21821421 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3npc A 2.35 BS01 B96 A 1 A53 K55 R69 E73 I86 L106 M108 L110 M111 D169 F170 A47 K49 R63 E67 I80 L100 M102 L104 M105 D163 F164 D151 K153 N156 D169 T188 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue Kd=7.3nM, IC50=6nM P45984 20655210 365 DNQFYSVEVADSTFTVLKRYQQLKPIGSGAQGIVCAAFDTVLGINVAVKKLSRPFQNQTHAKRAYRELVLLKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIHMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTACTNFMMTPYVVTRYYRAPEVILGMGYAANVDIWSVGCIMGELVKGCVIFQGTDHIDQWNKVIEQLGTPSAEFMAALQPTVRNYVENRPKYPGIKFEELFPDWIFPSESERDKIKTSQARDLLSKMLVIDPDKRISVDEALRHPYITVWYDPAEAEAPPPQIYDAQLEEREHAIEEWKELIYKEVMDW 3nq9 A 1.9 BS01 OCA A 1 K69 M107 K69 M107 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=92.6uM remove_due_to_license_issue P02754 21360616 1111 LIVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 3nrm A 3.05 BS01 NRM A 1 R137 L139 L194 L210 Y212 A213 P214 G216 L263 A273 D274 R12 L14 L69 L85 Y87 A88 P89 G91 L138 A148 D149 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 20674350 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRAALCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3nrz C 1.8 BS01 HPA C 1 E802 R880 F914 F1009 T1010 A1079 E232 R310 F344 F439 T440 A509 Q767 E802 R880 H884 R912 G1260 E1261 Q197 E232 R310 H314 R342 G690 E691 1.17.1.4,1.17.3.2 0005506,0016491,0043546 remove_due_to_license_issue P80457 20615869 1 DTVGRPLPHLAAAMQASGEAVYCDDIPRYENELFLRLVTSTRAHAKIKSIDVSEAQKVPGFVCFLSADDIPGSNETGLFNDETVFAKDTVTCVGHIIGAVVADTPEHAERAAHVVKVTYEDLPAIITIEDAIKNNSFYGSELKIEKGDLKKGFSEADNVVSGELYIGGQDHFYLETHCTIAIPKGEEGEMELFVSTQNAMKTQSFVAKMLGVPVNRILVRVKRMGGGFGGKETRSTLVSVAVALAAYKTGHPVRCMLDRNEDMLITGGRHPFLARYKVGFMKTGTIVALEVDHYSNAGNSRDLSHSIMERALFHMDNCYKIPNIRGTGRLCKTNLSSNTAFRGFGGPQALFIAENWMSEVAVTCGLPAEEVRWKNMYKEGDLTHFNQRLEGFSVPRCWDECLKSSQYYARKSEVDKFNKENCWKKRGLCIIPTKFGISFTVPFLNQAGALIHVYTDGSVLVSHGGTEMGQGLHTKMVQVASKALKIPISKIYISETSTNTVPNSSPTAASVSTDIYGQAVYEACQTILKRLEPFKKKNPDGSWEDWVMAAYQDRVSLSTTGFYRTPNLGYSFETNSGNAFHYFTYGVACSEVEIDCLTGDHKNLRTDIVMDVGSSLNPAIDIGQVEGAFVQGLGLFTLEELHYSPEGSLHTRGPSTYKIPAFGSIPTEFRVSLLRDCPNKKAIYASKAVGEPPLFLGASVFFAIKDAIRAARAQHTNNNTKELFRLDSPATPEKIRNACVDKFTTLCVTGAPGNCK 3ns7 A 2.6 BS01 3NS B 1 R179 S236 H237 Q283 C285 R44 S101 H102 Q148 C150 P177 R178 H237 G238 C285 R286 P42 R43 H102 G103 C150 R151 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 20656488 1 CSLEEAQRIWKQKSAEIYPIMDKSSRTRLALIICNEEFDSIPRRTGAEVDITGMTMLLQNLGYSVDVKKNLTASDMTTELEAFAHRPEHKTSDSTFLVFMSHGIREGICGKKHSEQVPDILQLNAIFNMLNTKNCPSLKDKPKVIIIQACRGDSPGVVWFKD 3ns7 B 2.6 BS01 3NS B 1 S339 W340 R341 R383 S23 W24 R25 R67 E390 E74 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 20656488 1 AIKKAHIEKDFIAFCSSTPDNVSWRHPTMGSVFIGRLIEHMQEYACSCDVEEIFRKVRFSFEQPDGRAQMPTTERVTLTRCFYLFPGH 3ns9 A 1.78 BS01 NS9 A 1 I10 V18 A31 F80 F82 L83 Q85 L134 I8 V16 A29 F71 F73 L74 Q76 L125 D127 K129 Q131 N132 D145 T158 T165 D118 K120 Q122 N123 D136 T149 T156 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.003uM remove_due_to_license_issue IC50=3nM P24941 21080703 0 NFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3nsh A 2.2 BS01 957 A 1 D38 G40 P76 Y77 T78 F114 R134 D234 D35 G37 P73 Y74 T75 F111 R131 D221 D38 S41 N43 A45 Y77 D234 T237 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=470nM remove_due_to_license_issue IC50=470nM P56817 20822903 407 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3nsn A 2.1 BS01 TMX B 1 R220 D367 E368 W448 D477 W490 W524 E526 R198 D345 E346 W426 D455 W468 W502 E504 D367 E368 D345 E346 3.2.1.52 0000272,0004553,0004563,0005886,0005975,0006032,0016231,0016798,0030203 remove_due_to_license_issue Q06GJ0 21106526 4 EDVVWRWSCDNGKCVKLKNDPRSSEPALSLEACKMFCNEYGLLWPRPTGEADLGNFLSKINLNSIEVKILKKGATDDLMEAAAKRFKEQVSLAIPRGSTPKLTGKAVDVYLVNENPNEKAFSLEMDESYGLRVSPSGADRVNATITANSFFGMRHGLETLSQLFVFDDIRDHLLMVRDVNISDKPVYPYRGILLDTARNYYSIESIKRTIEAMAAVKLNTFHWHITDSQSFPFVTTKRPNLYKFGALSPQKVYTKAAIREVVRFGLERGVRVLPEFDAPAHVGEGWQDTDLTVCFKAEPWKSYCVEPPCGQLNPTKDELYQYLEDIYSDMAEVFDTTDIFHMGGDEVSEACWNSSDSIQNFMMQNRWDLDKESFLKLWNYFQQKAQDKAYKAFGKKLPLILWTSTLTNYKHIDDYLNKDDYIIQVWTTGVDPQIKGLLEKGYRLIMSNYDALYFDCGYGAWVGAGNNWCSPYIGWQKVYDNSPAVIALEHRDQVLGGEAALWSEQSDTSTLDGRLWPRAAALAERLWAEPATSWQDAEYRMLHIRERLVRMGIQAESLQPEWCYQNEGYCYS 3nsq B 2.6 BS01 CHZ B 1 F313 F346 F50 F83 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 21084305 1 PVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQMT 3ntp A 1.762 BS01 RZD A 1 K63 R68 R69 C113 L122 Q129 M130 Q131 F134 S154 K47 R52 R53 C97 L106 Q113 M114 Q115 F118 S138 H59 C113 Q131 S154 H157 H43 C97 Q115 S138 H141 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=12uM remove_due_to_license_issue Q13526 21980916 164 KLPPGWEKAMSRSSGRVYYFNHITNASQWERPSGEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3nu3 A 1.02 BS01 478 B 1 D25 A28 D30 D25 A28 D30 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu3 B 1.02 BS01 478 B 1 D125 G127 A128 D130 G149 I150 D25 G27 A28 D30 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.15nM remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu4 A 1.2 BS01 478 B 1 D25 A28 D30 G48 V82 D25 A28 D30 G48 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu4 B 1.2 BS01 478 B 1 D125 G127 A128 D130 G149 I150 D25 G27 A28 D30 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.5nM remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu5 A 1.29 BS01 478 B 1 D25 G27 A28 D30 G48 V82 I84 D25 G27 A28 D30 G48 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu5 B 1.29 BS01 478 B 1 D125 G127 A128 D130 G149 V150 D25 G27 A28 D30 G49 V50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.5nM remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu6 A 1.16 BS01 478 B 1 D25 G27 A28 D30 G48 I50 V82 I84 D25 G27 A28 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu6 B 1.16 BS01 478 B 1 D25 G27 A28 D30 G49 I50 I84 D25 G27 A28 D30 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.5nM remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nu9 A 1.85 BS01 478 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.9nM remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 3nu9 B 1.85 BS01 478 A 1 D125 G127 A128 D130 G149 I150 D25 G27 A28 D30 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNVIGRNLLTQIGATLNF 3nuj A 1.5 BS01 478 B 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFVKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nuj B 1.5 BS01 478 B 1 D25 G27 A28 D30 G49 I50 D25 G27 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.41nM remove_due_to_license_issue P03366 20695887 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFVKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3nuo A 1.35 BS01 478 B 1 D25 A28 D30 G48 V82 D25 A28 D30 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20695887 478 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 3nuo B 1.35 BS01 478 B 1 D25 G27 A28 D30 G49 I50 D25 G27 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.16nM remove_due_to_license_issue P03366 20695887 478 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 3nus A 2.75 BS01 JNZ A 1 A109 S160 Y161 A162 L212 A37 S88 Y89 A90 L140 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 24900229 374 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3nuu A 1.9803 BS01 JOZ A 1 L88 A109 L159 S160 L212 L16 A37 L87 S88 L140 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=169000nM O15530 24900229 361 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3nuy A 2.1 BS01 JPZ A 1 A109 S160 L212 A37 S88 L140 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 24900229 370 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3nw5 A 2.14 BS01 LGX A 1 G976 Q977 V983 A1001 M1049 E1050 M1052 T1053 G1055 D1056 I1130 G22 Q23 V29 A47 M95 E96 M98 T99 G101 D102 I176 D1105 R1109 N1110 D1123 E1132 D151 R155 N156 D169 E178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=8400nM remove_due_to_license_issue IC50=8400nM P08069 20675137 1 DVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3nw6 A 2.2 BS01 LGW A 1 L975 G976 V983 A1001 K1003 M1049 E1050 M1052 T1053 G1055 R1109 M1112 G1122 M1126 R1128 L20 G21 V28 A46 K48 M94 E95 M97 T98 G100 R154 M157 G167 M171 R173 D1105 R1109 N1110 D1123 E1132 D150 R154 N155 D168 E177 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=7nM remove_due_to_license_issue IC50=162nM P08069 20675137 1 VYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3nw7 A 2.11 BS01 LGV A 1 L975 G976 V983 A1001 K1003 M1049 E1050 M1052 G1055 D1056 N1110 M1112 D1123 M1126 L19 G20 V27 A45 K47 M93 E94 M96 G99 D100 N154 M156 D167 M170 D1105 R1109 N1110 D1123 E1132 D149 R153 N154 D167 E176 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=5.3nM remove_due_to_license_issue IC50=5.3nM P08069 20675137 1 YVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 3nw9 A 1.65 BS02 637 A 1 W38 M40 Y68 E90 M91 A118 S119 D141 H142 W143 K144 N170 P174 L198 E199 W36 M38 Y66 E88 M89 A116 S117 D139 H140 W141 K142 N168 P172 L196 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=1nM remove_due_to_license_issue P22734 21538606 228 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3nwb A 1.3 BS02 659 A 1 W38 M40 E90 M91 Y95 A118 S119 Q120 D141 H142 W143 K144 N170 P174 L198 E199 W36 M38 E88 M89 Y93 A116 S117 Q118 D139 H140 W141 K142 N168 P172 L196 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 ic50=11nM remove_due_to_license_issue P22734 22349227 226 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3nwe A 1.5 BS02 662 A 1 W38 M40 E90 I91 S119 Q120 D141 H142 W143 K144 R146 N170 P174 L198 E199 W36 M38 E88 I89 S117 Q118 D139 H140 W141 K142 R144 N168 P172 L196 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 ic50=25nM remove_due_to_license_issue P22734 22349227 227 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3nww A 2.09 BS01 3NW A 1 G33 A51 K53 E71 L75 L104 T106 M109 G110 A111 L167 D168 F169 G29 A47 K49 E67 L71 L100 T102 M105 G106 A107 L163 D164 F165 D150 K152 N155 D168 T185 D146 K148 N151 D164 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=7nM remove_due_to_license_issue IC50=7nM Q16539 20732813 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3nx7 A 1.8 BS06 NHK A 1 L181 A182 H218 E219 H222 H228 P238 Y240 L76 A77 H113 E114 H117 H123 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Kd=7.88nM remove_due_to_license_issue Ki=7.6nM P39900 17269766 0 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3nxq A 1.99 BS02 RX4 A 1 Q259 H331 A332 S333 A334 H361 E362 H365 Y369 R381 E389 K489 F490 H491 T496 Y498 Y501 Q256 H328 A329 S330 A331 H358 E359 H362 Y366 R378 E386 K486 F487 H488 T493 Y495 Y498 H331 A332 H361 E362 H365 E389 H491 Y501 H328 A329 H358 E359 H362 E386 H488 Y498 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue P12821 20826823 700 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 3nyd A 1.23 BS01 3NY A 1 A21 W44 G82 G83 M84 D127 L236 M237 A20 W43 G81 G82 M83 D126 L235 M236 E131 M172 H209 M237 D239 E130 M171 H208 M236 D238 3.2.1.8 0004553,0005975,0016798,0031176,0045493 remove_due_to_license_issue P23360 22357762 317 AAQSVDQLIKARGKVYFGVATDQNRLTTGKNAAIIQADFGMVWPENSMKWDATEPSQGNFNFAGADYLVNWAQQNGKLIGGGMLVWHSQLPSWVSSITDKNTLTNVMKNHITTLMTRYKGKIRAWDVVGEAFNEDGSLRQTVFLNVIGEDYIPIAFQTARAADPNAKLYIMDYNLDSASYPKTQAIVNRVKQWRAAGVPIDGIGSQTHLSAGQGAGVLQALPLLASAGTPEVSILMLDVAGASPTDYVNVVNACLNVQSCVGISVFGVADPDSWRASTTPLLFDGNFNPKPAYNAIVQDLQQG 3nyn A 2.72 BS01 SGV A 1 L192 V200 A213 M266 D270 L318 L191 V199 A212 M265 D269 L317 D311 K313 E315 N316 D329 E338 T348 D310 K312 E314 N315 D328 E337 T347 2.7.11.16 0004672,0004674,0004703,0005515,0005524,0005737,0005886,0006468,0007165,0007186,0008277,0009966,0016020,0016055,0047696 remove_due_to_license_issue P43250 20729810 577 ELENIVANTVLLKAREGGGGNRKGKSKKWRQMLQFPHISQCEELRLSLERDYHSLCERQPIGRLLFREFCATRPELSRCVAFLDGVAEYEVTPDDKRKACGRQLTQNFLSHTGPDLIPEVPRQLVTNCTQRLEQGPCKDLFQELTRLTHEYLSVAPFADYLDSIYFNRFLQWKWLERQPVTKNTFRQYRVLGKGGFGEVCACQVRATGKMYACKKLEKKRIKKRKGEAMALNEKQILEKVNSRFVVSLAYAYETKDALCLVLTLMNGGDLKFHIYHMGQAGFPEARAVFYAAEICCGLEDLHRERIVYRDLKPENILLDDHGHIRISDLGLAVHVPEGQTIKGRVGTVGYMAPEVVKNERYTFSPDWWALGCLLYEMIAGQSPFQKKIKREEVERLVKEVPEEYSERFSPQARSLCSQLLCKDPAERLGCRGGSAREVKEHPLFKKLNFKRLGAGMLEPPFKPDPQAIYCKDVLDIEQFSTVKGVELEPTDQDFYQKFATGSVPIPWQNEMVETECFQELNVFGLDGSVPPDLDWKGQPPAPPKKGLLQRLFS 3nyx A 2.5 BS01 TZ1 A 1 F908 K930 I960 Y962 L976 M978 V981 L1030 D1041 F1042 G1043 F20 K40 I70 Y72 L85 M87 V90 L139 D150 F151 G152 N1023 A1025 R1027 N1028 D1041 P1064 N132 A134 R136 N137 D150 P173 2.7.10.2 0004672,0005524,0006468 Ki=32nM remove_due_to_license_issue P29597 21117080 1 PTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGEMVAVKALKADCGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDQEKSLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHSQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPCEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYRH 3nzc X 2.0 BS01 D2O X 1 I10 V11 A12 L25 E32 I33 F36 P66 F69 I123 I10 V11 A12 L25 E32 I33 F36 P66 F69 I123 1.5.1.3 0004146,0005739,0006730,0016491,0046452,0046654,0046655,0050661 remove_due_to_license_issue P16184 21206056 207 MNQQKSLTLIVALTTSYGIGRSNSLPWKLKKEISYFKRVTSFVPTFDSFESMNVVLMGRKTWESIPLQFRPLKGRINVVITRNESLDLGNGIHSAKSLDHALELLYRTYGSESSVQINRIFVIGGAQLYKAAMDHPKLDRIMATIIYKDIHCDVFFPLKFRDKEWSSVWKKEKHSDLESWVGTKVPHGKINEDGFDYEFEMWTRDL 3nzk A 1.8 BS01 C90 A 1 E78 T191 F192 I198 G210 S211 V217 H238 D242 H265 E78 T191 F192 I198 G210 S211 V217 H238 D242 H265 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 Ki=0.54nM remove_due_to_license_issue A1JJJ9 21171638 501 MIKQRTLKRIVQATGVGLHTGKKVTLTMRPAPANTGVIYRRTDLNPPVDFPADAKSVRDTMLCTCLVNEHDVRISTVEHLNAALAGLGIDNIIIEVNAPEVPIMDGSASPFVYLLLDAGIEELNSAKKFLRLKETVRVEDGDKWAELSPFNGFRLDFTIDFNHPAIDSSTQRYRLDFSADSFVRQISRARTFGFMRDIEYLQSRGLCLGGSFDCAIVVDDYRVLNEDGLRFEDEFVRHKMLDAIGDLFMCGHNIIGAFTAYKSGHALNNKLLQAVLAKQEAWEFVTFQDEAEMPLAFK 3nzs A 2.75 BS01 NZS A 1 M804 W812 I831 K833 Y867 E880 I881 V882 T887 K890 M953 I963 D964 M553 W561 I580 K582 Y616 E629 I630 V631 T636 K639 M702 I712 D713 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 20822905 1 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKSLWDCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISFNADKLTSATNPDKENSMSISILLDALPKEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIRVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 3nzu A 2.6 BS01 NZU A 1 I831 Y867 I879 E880 V882 T886 T887 K890 M953 D964 I568 Y604 I616 E617 V619 T623 T624 K627 M690 D701 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 20822905 1 QAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISFNADKLTSATNPDKENSMSISILLDEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYRVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLGI 3o0g B 1.95 BS01 3O0 B 1 I10 V18 A31 K33 C83 D84 Q85 L133 N144 I5 V8 A15 K17 C59 D60 Q61 L109 N120 N131 N144 C157 N270 V272 R274 I275 D288 N107 N120 C133 N246 V248 R250 I251 D264 2.7.11.1 0000226,0000307,0001764,0001963,0002039,0004672,0004674,0004676,0004677,0004679,0004693,0004694,0004711,0005176,0005515,0005524,0005634,0005654,0005737,0005829,0005874,0005886,0006338,0006468,0006886,0006915,0007160,0007268,0007399,0007409,0007416,0007519,0008017,0008045,0008306,0008542,0014044,0014069,0016020,0016079,0016241,0016301,0016310,0016477,0016533,0018105,0018107,0019233,0021537,0021549,0021695,0021697,0021766,0021819,0021954,0021987,0022038,0030027,0030036,0030054,0030175,0030182,0030334,0030424,0030425,0030426,0030517,0030549,0030900,0031175,0031397,0031594,0031914,0032801,0035175,0035249,0035402,0035403,0035418,0035979,0042220,0042981,0042995,0043005,0043025,0043113,0043125,0043204,0043525,0044022,0044023,0044024,0044025,0045202,0045786,0045861,0045892,0045956,0046826,0048148,0048156,0048167,0048488,0048489,0048511,0048675,0048709,0048813,0050321,0051301,0051402,0051649,0051726,0051879,0051966,0060078,0060079,0061001,0070509,0072354,0072371,0072518,0090314,0098793,0106310,0140823,0140855,0140857,1901987,1903076,1903421,1904646,1990244 Ki=0.6uM remove_due_to_license_issue Q00535 16039528 293 KLEKIGTVFKAEIVALKRVRPSSALREICLLKELKHKNIVRLHDVLHSDKKLTLVFEFCDQDLKKYFDSCNGDLDPEIVKSFLFQLLKGLGFCHSRNVLHRDLKPQNLLINRNGELKLANFGLARAFGIPVRCYSAEVVTLWYRPPDVLFGAKLYSTSIDMWSAGCIFAELANAGRPLFPGNDVDDQLKRIFRLLGTPTEEQWPSMTKLPDYKPYPMYPATTSLVNVVPKLNATGRDLLQNLLKCNPVQRISAEEALQHPYFSD 3o0j A 1.95 BS02 3OJ A 1 H234 D275 M347 D392 M431 F446 H73 D114 M186 D231 M270 F285 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=240nM Q07343 22841723 485 NEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMI 3o0u A 1.8 BS01 O47 A 1 G23 C25 G65 G66 Y67 A134 N161 G23 C25 G65 G66 Y67 A134 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 20843687 216 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3o1g A 1.65 BS01 O75 A 1 G23 C25 N60 D61 G64 G65 G66 Y67 A134 L160 N161 H162 G23 C25 N60 D61 G64 G65 G66 Y67 A134 L160 N161 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=<1nM P43235 20843687 218 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3o23 A 2.1 BS01 MQY A 1 K1033 M1054 V1062 M1079 M1082 F1131 M1142 D1153 M1156 K43 M64 V72 M89 M92 F141 M152 D163 M166 D1135 R1139 N1140 D1153 E1162 D145 R149 N150 D163 E172 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.5uM remove_due_to_license_issue P08069 21441024 1 EWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSE 3o2m A 2.7 BS02 46A A 1 F180 L198 G199 Y230 Q253 V256 F174 L192 G193 Y224 Q247 V250 D151 K153 N156 D169 T188 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P45983 21090814 701 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPAFMKKLQPTVRNYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 3o2m A 2.7 BS03 46A B 1 P184 V256 P178 V250 D151 K153 N156 D169 T188 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P45983 21090814 701 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPAFMKKLQPTVRNYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 3o3i X 2.801 BS01 rna A 0 Y312 Y317 F332 A335 Y345 Y346 Q349 Y350 M381 Y37 Y42 F57 A60 Y70 Y71 Q74 Y75 M96 3.1.26.- 0003723 remove_due_to_license_issue Q96J94 21193640 1 ~ 14 SETVLDFMFNFYHQTEEHKFQEQVSKELIGLVVLTKYNNKTYRVDDIDWDQNPKSTFKKADGSEVSFLEYYRKQYNQEITDLKQPVLVSQPKGPAMLIPELCYLTGLT 3o3j A 3.0 BS05 BB4 A 1 Q48 E89 G90 C91 L92 R129 H133 E134 H137 Q48 E89 G90 C91 L92 R129 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 3.5.1.88 0042586 remove_due_to_license_issue Q9FUZ2 21629676 300 MEIVEYPDPILRAKNKRIDIFDENLKNLVDAMFDVMYKTDGIGLSAPQVGLNVQLMVFNPAGEPGEGKEIVLVNPKIKKYSDKLVPFDEGCLSFPGIYAEVVRPQSVKIDARDITGERFSISLSRLPARIFQHEYDHLEGVLFFDRMTDQVLDSIREELEALEKKYEEKTGLPSPERVEA 3o4k A 2.11 BS01 LTC C 1 R31 N140 E142 R31 N140 E142 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 21454594 172 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3o4k C 2.11 BS01 LTC C 1 E24 L64 W66 C67 A92 H93 G95 N99 Q150 E24 L64 W66 C67 A92 H93 G95 N99 Q150 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 Kd=24nM remove_due_to_license_issue Q9GK12 21454594 172 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3o4k D 2.11 BS01 LTC C 1 G95 P96 T97 W98 K144 V149 Q150 P151 G95 P96 T97 W98 K144 V149 Q150 P151 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 21454594 172 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3o56 A 2.42 BS02 ZG1 A 1 S282 M347 L393 N395 T407 I410 F414 M431 Q443 F446 S130 M195 L241 N243 T255 I258 F262 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=794pM remove_due_to_license_issue Q07343 20732811 506 ISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIPQA 3o57 A 2.0 BS02 ZG2 A 1 M347 L393 T407 I410 M431 Q443 G445 F446 M196 L242 T256 I259 M280 Q292 G294 F295 3.1.4.53 0004114,0007165,0008081 ic50=79.4pM remove_due_to_license_issue Q07343 20732811 506 SISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIPQA 3o5n E 1.83 BS01 BR0 E 1 F656 G657 F658 V659 L660 V721 I724 R725 F20 G21 F22 V23 L24 V72 I75 R76 ? Ki=17.2uM remove_due_to_license_issue Q4ACU6 21626699 1 SDYVIDDKVAILQKRDHEGFGFVLPTPAFPALQYLESVDVEGVAWRAGLRTGDFLIEVNGVNVVKVGHKQVVGLIRQGGNRLVMKVVSVTRK 3o5x A 2.0 BS01 JZG A 1 R362 K364 R465 Q510 R90 K92 R193 Q238 D425 C459 R465 T466 Q506 D153 C187 R193 T194 Q234 3.1.3.48 0004725,0006470,0016311 ic50=5.5uM remove_due_to_license_issue IC50=5500nM, Ki=5200nM Q06124 20170098 1 LYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPNEPVSDYINANIIMPKKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETLQR 3o64 B 1.88 BS01 786 B 1 T347 L348 G349 L350 V402 H405 E406 H409 H415 Y433 V434 Y436 P437 I438 A439 N447 T127 L128 G129 L130 V182 H185 E186 H189 H195 Y213 V214 Y216 P217 I218 A219 N227 3.4.24.86 0004222,0006508,0008237 Ki=0.4nM remove_due_to_license_issue IC50=720nM, Ki=0.400000nM P78536 21458257 501 MKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQER 3o6e X 2.904 BS01 rna A 0 Y312 Y317 F332 Y345 Y346 Q349 Y350 M381 Y36 Y41 F56 Y69 Y70 Q73 Y74 M95 3.1.26.- 0003723 remove_due_to_license_issue Q96J94 21193640 1 ~ 14 ETVLDFMFNFYHQTEEHKFQEQVSKELIGLVVLTKYNNKTYRVDDIDWDQNPKSTFKKADGSEVSFLEYYRKQYNQEITDLKQPVLVSQPKGPAMLIPELCYLTGLT 3o6t A 2.4 BS01 PX5 A 1 C37 P39 I80 C31 P33 I74 C37 G38 P39 S40 C31 G32 P33 S34 ? 0005576,0005737,0005829,0005886,0009055,0009274,0015035,0015036,0015038,0016491,0045454 remove_due_to_license_issue P9WG67 20981751 117 SATIKVTDASFATDVLSSNKPVLVDFWATWCGPSKMVAPVLEEIATERATDLTVAKLDVDTNPETARNFQVVSIPTLILFKDGQPVKRIVGAKGKAALLRELSDVVPN 3o75 A 2.3 BS01 F1X A 1 S75 Y76 D148 R149 R197 F220 S247 Y248 F273 G274 Q291 R322 S16 Y17 D89 R90 R138 F161 S188 Y189 F214 G215 Q232 R263 ? 0003677,0006355,0009750 Kd=209nM remove_due_to_license_issue Q88PQ6 21239488 1 HTRTLGFILPDLENPSYARIAKQLEQGARARGYQLLIASSDDQPDSERQLQQLFRARRCDALFVASCLPPEDDSYRELQDKGLPVIAIDRRLDPAHFCSVISDDRDASRQLAASLLSSAPRSIALIGARPELSVSQARAGGFDEALQGYTGEVRRYQGEAFSRECGQRLMQQLIDDLGGLPDALVTTSYVLLQGVFDTLQARPVDSRQLQLGTFGDNQLLDFLPLPVNAMAQQHGQIAATALELALAAIEEKRYEPGVHAVGRTFKQRIS 3o7u A 1.708 BS04 O7U A 1 H63 L81 Q156 H214 E217 H246 D313 D314 W319 H60 L78 Q153 H211 E214 H243 D310 D311 W316 H61 H63 Q156 H214 E217 D313 H58 H60 Q153 H211 E214 D310 3.5.4.-,3.5.4.1 0004131,0005829,0006209,0008198,0008270,0016787,0016810,0019858,0035888,0042802,0046872 Ki=52nM remove_due_to_license_issue P25524 21545144 430 ALQTIINARLPGEEGLWQIHLQDGKISAIDAQSGVMPITENSLDAEQGLVIPPFVEPHIHLDTTQTAGQPNWNQSGTLFEGIERWAERKALLTHDDVKQRAWQTLKWQIANGIQHVRTHVDVSDATLTALKAMLEVKQEVAPWIDLQIVAFPQEGILSYPNGEALLEEALRLGADVVGAIPHFEFTREYGVESLHKTFALAQKYDRLIDVHCDEIDDEQSRFVETVAALAHHEGMGARVTASHTTAMHSYNGAYTSRLFRLLKMSGINFVANPLVNIHLQGRFDTYPKRRGITRVKEMLESGINVCFGHDDVFDPWYPLGTANMLQVLHMGLHVCQLMGYGQINDGLNLITHHSARTLNLQDYGIAAGNSANLIILPAENGFDALRRQVPVRYSVRGGKVIASTQPAQTTVYLEQPEAIDYK 3o84 A 2.1 BS01 HTJ A 1 H241 N242 F243 S247 V286 G314 F337 G338 M339 H237 N238 F239 S243 V282 G310 F333 G334 M335 S217 E341 S213 E337 0008668,0019290 Kd=58nM remove_due_to_license_issue 20853905 995 KQLIEFVRWSPERAQHYRNKGYWIDQPLTRILTVGVQSHPHSLAIICGERQLSYIELDRLSTNLATRLAEKGLGKGDTALVQLPNVAEFYIVFFALLKAGVVVLNALYSHRQYELNAFIKQIQPKLLIGSRQHEVFSNNQFIDSLHDVNLSPEIILMLNHQATDFGLLDWIETPAETFVDFSSTPADEVAFFQLSGTGTPKLIPRTHNDYDYSVRASAEICGLNSNTRLLCALPAPHNFMLSSPGALGVLHAGGCVVMAPNPEPLNCFSIIQRHQVNMASLVPSAVIMWLEKAAQYKDQIQSLKLLQVGGASFPESLARQVPEVLNCKLQQVFGMAEGLVNYTRLDDSDEQIFTTQGRPISSDDEIKIVDEQYREVPEGEIGMLATRGPYTFCGYYQSPEHNSQVFDEDNYYYSGDLVQRTPDGNLRVVGRIK 3o86 A 1.6 BS01 BSF A 1 S64 Y150 N152 Y221 A318 S61 Y147 N149 Y218 A308 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K305 A308 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 20945905 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3o87 A 1.78 BS01 BSG A 1 S64 Y150 N152 V211 S212 Y221 A318 T319 G320 S61 Y147 N149 V208 S209 Y218 A308 T309 G310 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K305 A308 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 20945905 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3o88 A 1.64 BS01 BSH A 1 G63 S64 L119 Q120 Y150 N152 Y221 G317 A318 T319 G320 G60 S61 L116 Q117 Y147 N149 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 20945905 1 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3o8g A 1.9 BS01 O8G A 1 M102 G106 F110 Y148 T149 N176 N179 E180 M81 G85 F89 Y127 T128 N155 N158 E159 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=7.4uM remove_due_to_license_issue P9WMC1 20704273 217 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGEN 3o8h A 1.9 BS01 O8H A 1 M102 G106 I107 F110 F114 T121 G124 Q125 W138 Y148 T149 N176 N179 E180 L183 F184 W207 M81 G85 I86 F89 F93 T100 G103 Q104 W117 Y127 T128 N155 N158 E159 L162 F163 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=580nM remove_due_to_license_issue IC50=580nM P9WMC1 20704273 217 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGEN 3o8p A 2.1 BS01 BMU A 1 K53 E71 M78 I84 G168 F169 K49 E67 M74 I80 G164 F165 D150 K152 N155 G168 T185 D146 K148 N151 G164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Kd=1160nM, kon=118000M-1-s-1, koff=0.140000s-1, IC50=21000nM Q16539 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILGFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 3o95 A 2.85 BS01 01T A 1 R125 E205 E206 F357 S630 Y662 Y666 V711 H740 R86 E166 E167 F318 S591 Y623 Y627 V672 H701 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=5.3nM P27487 21218817 1 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3o96 A 2.7 BS01 IQO A 1 W80 I84 S205 L210 L264 K268 Y272 D292 C296 W76 I80 S157 L162 L216 K220 Y224 D244 C248 D274 K276 N279 D292 D226 K228 N231 D244 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue IC50=58nM P31749 20886116 444 SDVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDVEAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFTPEEREEWTTAIQTVADGLKKQVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVANRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQV 3o99 A 1.95 BS01 K13 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o99 B 1.95 BS01 K13 A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9a A 1.9 BS01 K14 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9a B 1.9 BS01 K14 A 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9b A 1.5 BS01 K2A A 1 D25 G27 A28 D29 D30 G48 I50 V82 D25 G27 A28 D29 D30 G48 I50 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9b B 1.5 BS01 K2A A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9c A 1.85 BS01 K20 A 1 D25 G27 A28 D29 G48 I50 V82 D25 G27 A28 D29 G48 I50 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9c B 1.85 BS01 K20 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9d A 1.85 BS01 K19 A 1 D25 G27 A28 D29 G48 I50 D25 G27 A28 D29 G48 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9d B 1.85 BS01 K19 A 1 D25 A28 D30 G48 P81 V82 D25 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9e A 1.5 BS01 A60 A 1 D25 G27 A28 D29 D30 G48 I50 V82 I84 D25 G27 A28 D29 D30 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9e B 1.5 BS01 A60 A 1 D25 G27 A28 D30 V32 P81 V82 I84 D25 G27 A28 D30 V32 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9f A 1.7 BS01 K2D A 1 D25 G27 A28 D29 D30 G48 I50 I84 D25 G27 A28 D29 D30 G48 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9f B 1.7 BS01 K2D A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9g A 1.65 BS01 F53 A 1 D25 G27 A28 D29 D30 G48 I50 I84 D25 G27 A28 D29 D30 G48 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9g B 1.65 BS01 F53 A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9h A 1.7 BS01 K2E B 1 D25 G27 A28 D29 G48 I50 V82 I84 D25 G27 A28 D29 G48 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9h B 1.7 BS01 K2E B 1 D25 G27 A28 D30 P81 D25 G27 A28 D30 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9i A 1.45 BS01 A61 A 1 D25 G27 A28 D29 D30 G48 I50 I84 D25 G27 A28 D29 D30 G48 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9i B 1.45 BS01 A61 A 1 D25 G27 A28 D30 P81 V82 D25 G27 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03369 24012370 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3o9l A 2.4 BS01 LPN A 1 T18 Y20 V36 D38 W45 H61 V88 M114 F119 F124 D125 T15 Y17 V33 D35 W42 H58 V85 M111 F116 F121 D122 D38 S41 N43 W45 Y83 D35 S38 N40 W42 Y80 3.4.23.15 0004190,0006508 ic50=0.22nM remove_due_to_license_issue IC50=0.22nM P00797 20843686 168 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRD 3o9l B 2.4 BS01 LPN A 1 D226 G228 D56 G58 D226 A229 D56 A59 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.22nM P00797 20843686 168 SLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALARH 3o9p A 2.07 BS01 MHI A 1 K20 V32 L34 Q267 R402 R411 S413 W414 V415 D417 Y483 T484 K14 V26 L28 Q261 R396 R405 S407 W408 V409 D411 Y477 T478 ? 0015031,0015833,0015834,0016020,0030288,0035351,0042597,0042938,0042939,0043190,0055052,0055085,0140207,1900750,1904680 Kd=0.3uM remove_due_to_license_issue P77348 21705338 516 TVLAEKQELVRHIKDEPASLDPAKAVGLPEIQVIRDLFEGLVNQNEKGEIVPGVATQWKSNDNRIWTFTLRDNAKWADGTPVTAQDFVYSWQRLVDPKTLSPFAWFAALAGINNAQAIIDGKATPDQLGVTAVDAHTLKIQLDKPLPWFVNLTANFAFFPVQKANVESGKEWTKPGNLIGNGAYVLKERVVNEKLVVVPNTHYWDNAKTVLQKVTFLPINQESAATKRYLAGDIDITESFPKNMYQKLLKDIPGQVYTPPQLGTYYYAFNTQKGPTADQRVRLALSMTIDRRLMTEKVLGTGEKPAWHFTPDVTAGFTPEPSPFEQMSQEELNAQAKTLLSAAGYGPQKPLKLTLLYNTSENHQKIAIAVASMWKKNLGVDVKLQNQEWKTYIDSRNTGNFDVIRASWVGDYNEPSTFLTLLTSTHSGNISRFNNPAYDKVLAQASTENTVKARNADYNAAEKILMEQAPIAPIYQYTNGRLIKPWLKGYPINNPEDVAYSRTMYIVKH 3o9v A 2.75 BS01 10T A 1 R125 E205 E206 Y547 S630 Y662 Y666 V711 R86 E166 E167 Y508 S591 Y623 Y627 V672 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=18nM P27487 21218817 1 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3o9x A 2.0999 BS01 dna F 0 F22 R23 G93 G94 N97 R101 Y102 A107 Q108 F23 R24 G94 G95 N98 R102 Y103 A108 Q109 ? 0003677,0005515,0006355,0042803,0043565,0044010,0046872,0110001 remove_due_to_license_issue Q46864 21068382 1 ~ 26 HMKCPVCHQGEMVSGIKDIPYTFRGRKTVLKGIHGLYCVHCEESIMNKEESDAFMAQVKAFRASVNAETVAPEFIVKVRKKLSLTQKEASEIFGGGVNAFSRYEKGNAQPHPSTIKLLRVLDKHPELLNEIR 3o9x A 2.0999 BS02 dna E 0 T84 Q85 N97 S100 H110 T85 Q86 N98 S101 H111 ? 0003677,0005515,0006355,0042803,0043565,0044010,0046872,0110001 remove_due_to_license_issue Q46864 21068382 1 ~ 26 HMKCPVCHQGEMVSGIKDIPYTFRGRKTVLKGIHGLYCVHCEESIMNKEESDAFMAQVKAFRASVNAETVAPEFIVKVRKKLSLTQKEASEIFGGGVNAFSRYEKGNAQPHPSTIKLLRVLDKHPELLNEIR 3o9x B 2.0999 BS01 dna F 0 Q85 N97 S100 H110 Q86 N98 S101 H111 ? 0003677,0005515,0006355,0042803,0043565,0044010,0046872,0110001 remove_due_to_license_issue Q46864 21068382 1 ~ 26 HMKCPVCHQGEMVSGIKDIPYTFRGRKTVLKGIHGLYCVHCEESIMNKEESDAFMAQVKAFRASVNAETVAPEFIVKVRKKLSLTQKEASEIFGGGVNAFSRYEKGNAQPHPSTIKLLRVLDKHPELLNEIR 3o9x B 2.0999 BS02 dna E 0 F22 R23 G93 G94 N97 R101 Y102 Q108 F23 R24 G94 G95 N98 R102 Y103 Q109 ? 0003677,0005515,0006355,0042803,0043565,0044010,0046872,0110001 remove_due_to_license_issue Q46864 21068382 1 ~ 26 HMKCPVCHQGEMVSGIKDIPYTFRGRKTVLKGIHGLYCVHCEESIMNKEESDAFMAQVKAFRASVNAETVAPEFIVKVRKKLSLTQKEASEIFGGGVNAFSRYEKGNAQPHPSTIKLLRVLDKHPELLNEIR 3oad A 2.17 BS01 LPO A 1 T18 Q19 Y20 V36 D38 G40 W45 V46 H61 Y83 M114 F119 F124 D125 V127 T15 Q16 Y17 V33 D35 G37 W42 V43 H58 Y80 M111 F116 F121 D122 V124 D38 S41 N43 W45 Y83 D35 S38 N40 W42 Y80 3.4.23.15 0004190,0006508 ic50=0.24nM remove_due_to_license_issue IC50=0.12nM P00797 20843686 167 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRD 3oad B 2.17 BS01 LPO A 1 D226 G228 A229 D56 G58 A59 D226 A229 D56 A59 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.12nM P00797 20843686 167 SLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALARH 3oaf A 1.7 BS01 OAG A 1 V8 A9 L22 E30 F31 F34 S59 P61 V8 A9 L22 E30 F31 F34 S59 P61 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 remove_due_to_license_issue Ki=24nM P00374 23545530 187 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFSRMTTTSSVEGKQNLVIMGKKTWFSIPEKFRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3oag A 2.3 BS01 LPQ A 1 D38 G40 W45 V46 H61 L81 Y83 M114 F119 F124 D125 V127 D35 G37 W42 V43 H58 L78 Y80 M111 F116 F121 D122 V124 D38 S41 N43 W45 Y83 D35 S38 N40 W42 Y80 3.4.23.15 0004190,0006508 ic50=0.56nM remove_due_to_license_issue P00797 20843686 167 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRD 3oag B 2.3 BS01 LPQ A 1 D226 G228 S230 D56 G58 S60 D226 A229 D56 A59 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 20843686 167 SLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALARH 3oaw A 2.75 BS01 OAW A 1 I831 Y867 I879 V882 M953 I963 D964 I588 Y624 I636 V639 M710 I720 D721 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 20817449 1 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKESLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNYCHPIALPRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYRVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLG 3oay H 1.95 BS01 BDF H 1 A31 H32 T33 K95 G96 L100 S100A N100C D100D A31 H32 T33 K99 G100 L104 S105 N107 D108 remove_due_to_license_issue 20852065 229 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 3oc0 A 2.7 BS01 B2Q A 1 E205 E206 S209 F357 Y662 E167 E168 S171 F319 Y624 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=710nM P27487 20031405 900 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3ocb A 2.7 BS02 XM1 A 1 G162 K163 V164 A177 K179 M227 E228 A230 E234 E278 M281 T291 D292 F438 G19 K20 V21 A34 K36 M84 E85 A87 E91 E135 M138 T148 D149 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=5nM P31749 20810279 1 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMRPHFPQFDYSASS 3ocg A 2.21 BS01 OCG A 1 A51 K53 E71 L75 T106 M109 A111 L167 D168 A48 K50 E68 L72 T103 M106 A108 L164 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=3nM remove_due_to_license_issue IC50=3nM Q16539 21035336 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3ocp A 2.49 BS01 CMP A 1 L172 F181 G182 E183 L184 A185 R192 T193 A194 L81 F90 G91 E92 L93 A94 R101 T102 A103 2.7.11.12 Kd=27+-3.6nM (21526164) Kd=27nM remove_due_to_license_issue Q13976 21526164 250 SHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMR 3oct A 1.95 BS01 1N1 A 1 A428 K430 M449 I472 T474 Y476 M477 A478 G480 L528 S538 F540 A33 K35 M51 I74 T76 Y78 M79 A80 G82 L130 S140 F142 D521 A523 R525 N526 D539 F559 D123 A125 R127 N128 D141 F147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=1.4nM, IC50=3.0nM Q06187 663 SWEIDPKDLTFLKELGQFGVVKYGKWRGQYDVAIKMIKMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMD 3ocz A 1.35 BS02 SRA A 1 D64 D66 F86 W91 T124 N125 K161 Y221 D56 D58 F78 W83 T116 N117 K153 Y213 3.1.3.2 0009279 Ki=0.035uM remove_due_to_license_issue P26093 21933344 264 EEHANMQLQQQAVLGLNWMQDSGEYKALAYQAYNAAKVAFDHAKVAKGKKKAVVADLDETMLDNSPYAGWQVQNNKPFDGKDWTRWVDARQSRAVPGAVEFNNYVNSHNGKVFYVTNRKDSTEKSGTIDDMKRLGFNGVEESAFYLKKDKSAKAARFAEIEKQGYEIVLYVGDNLDDFGNTVYGKLNADRRAFVDQNQGKFGKTFIMLPNANYGGWEGGLAEGYFKKDTQGQIKARLDAVQAWDGKL 3od0 A 2.9 BS01 PCG A 1 L172 F181 G182 E183 L184 A185 R192 T193 L81 F90 G91 E92 L93 A94 R101 T102 2.7.11.12 Kd=12+-1.6nM (21526164) remove_due_to_license_issue Q13976 21526164 250 SHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMR 3od0 A 2.9 BS02 PCG B 1 L187 N189 L96 N98 2.7.11.12 Kd=12+-1.6nM (21526164) remove_due_to_license_issue Q13976 21526164 250 SHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMR 3od0 B 2.9 BS01 PCG B 1 L172 F181 G182 E183 L184 A185 R192 T193 A194 L81 F90 G91 E92 L93 A94 R101 T102 A103 2.7.11.12 Kd=12+-1.6nM (21526164) remove_due_to_license_issue Q13976 21526164 250 SHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMR 3odh A 2.3 BS01 dna C 0 R134 R143 R148 T188 D189 G190 R191 R134 R143 R148 T188 D189 G190 R191 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRAIR 3odh A 2.3 BS02 dna D 0 V52 K53 K56 G83 T102 N104 R110 K114 T141 D142 R143 K186 G187 D189 R191 A192 V52 K53 K56 G83 T102 N104 R110 K114 T141 D142 R143 K186 G187 D189 R191 A192 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRAIR 3odh B 2.3 BS01 dna C 0 G51 V52 R81 T102 N104 K114 T141 D142 R143 K186 T188 G51 V52 R81 T102 N104 K114 T141 D142 R143 K186 T188 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRA 3odh B 2.3 BS02 dna D 0 N104 R134 R143 N104 R134 R143 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRA 3odh E 2.3 BS01 dna G 0 N104 R143 T188 D189 G190 N104 R143 T188 D189 G190 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRAIR 3odh E 2.3 BS02 dna H 0 V52 K56 G83 T102 R110 K114 T141 D142 R143 K186 G187 D189 G190 R191 A192 V52 K56 G83 T102 R110 K114 T141 D142 R143 K186 G187 D189 G190 R191 A192 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRAIR 3odh F 2.3 BS01 dna G 0 V52 K53 R81 G83 T102 N104 T141 D142 R143 K186 T188 V52 K53 R81 G83 T102 N104 T141 D142 R143 K186 T188 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRAIR 3odh F 2.3 BS02 dna H 0 K53 N104 R143 K53 N104 R143 0000287,0003677,0009036,0009307 remove_due_to_license_issue 20833632 1 ~ 12 MKIKRIEVLINNGSVPGIPMILNEIQDAIKTVSWPEGNNSFVINPVRKGNGVKPIKNSCMRHLHQKGWALEHPVRIKAEMRPGPLDAVKMIGGKAFALEWETGNISSSHRAINKMVMGMLERVIIGGVLILPSRDMYNYLTDRVGNFRELEPYFSVWRQFNLKDAYLAIVEIEHDSVDAQVSLIPKGTDGRAIR 3odk A 2.3 BS01 ODK A 1 L61 K63 C113 Q131 F134 S154 L43 K45 C95 Q113 F116 S136 H59 C113 Q131 S154 H157 H41 C95 Q113 S136 H139 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 ic50=720uM remove_due_to_license_issue IC50=720000nM Q13526 20932746 165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPSEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3odu A 2.5 BS01 ITD A 1 W94 D97 Y116 I185 C186 D187 E288 W68 D71 Y90 I159 C160 D161 E426 E1011 D1020 E215 D224 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0019955,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P61073 20929726 1500 PCFREENANFNKIFLPTIYSIIFLTGIVGNGLVILVMGYQKKLRSMTDKYRLHLSVADLLFVITLPFWAVDAVANWYFGNFLCKAVHVIYTVNLYSSVWILAFISLDRYLAIVHATNSQRPRKLLAEKVVYVGVWIPALLLTIPDFIFANVSEADDRYICDRFYPNDLWVVVFQFQHIMVGLILPGIVILSCYCIIISKLSHSGSNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYGSKGHQKRKALKTTVILILAFFACWLPYYIGISIDSFILLEIIKQGCEFENTVHKWISITEALAFFHCCLNPILYAFLGAKFKTSAQHALTSGRPLEVLFQ 3oe4 A 1.49 BS02 610 A 1 W38 M40 Y68 E90 I91 A118 S119 D141 H142 W143 K144 N170 P174 E199 W36 M38 Y66 E88 I89 A116 S117 D139 H140 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=34nM remove_due_to_license_issue P22734 21538606 223 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3oe5 A 1.52 BS02 611 A 1 W38 M40 Y68 E90 I91 A118 S119 D141 H142 W143 K144 N170 P174 E199 W36 M38 Y66 E88 I89 A116 S117 D139 H140 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=132nM remove_due_to_license_issue P22734 21538606 223 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3oe6 A 3.2 BS01 ITD A 1 W94 D97 Y116 R183 C186 D187 E288 W60 D63 Y82 R149 C152 D153 E394 E1011 D1020 E194 D203 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0019955,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P61073 20929726 1500 NFNKIFLPTIYSIIFLTGIVGNGLVILVMGYQKKLRSMTDKYRLHLSVADLLFVITLPFWAVDAVANWYFGNFLCKAVHVIYTVNLYSSVWILAFISLDRYLAIVHATNSQRPRKLLAEKVVYVGVWIPALLLTIPDFIFANVSEADDRYICDRFYPNDLWVVVFQFQHIMVGLILPGIVILSCYCIIISKLDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDRKALKTTVILILAFFACWLPYYIGISIDSFILLEIIKQGCEFENTVHKWISITEALAFFHCCLNPILYAFLGAKFKTS 3oe9 A 3.1 BS01 ITD A 1 W94 D97 V112 Y116 R183 C186 E288 W63 D66 V81 Y85 R152 C155 E405 E1011 E207 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0019955,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P61073 20929726 1500 CFRNFNKIFLPTIYSIIFLTGIVGNGLVILVMGYQKKLRSMTDKYRLHLSVADLLFVITLPFWAVDAVANWYFGNFLCKAVHVIYTVNLYSSVWILAFISLDRYLAIVHATNSQRPRKLLAEKVVYVGVWIPALLLTIPDFIFANVSEADDRYICDRFYPNDLWVVVFQFQHIMVGLILPGIVILSCYCIIISKLSHNIFEMLRIDEGLRLKIYKGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKALKPTVILILAFFACWLPYYIGISIDSFILLEIIKCEFENTVHKWISITEALAFFHCCLNPILYA 3oeu K 2.6 BS02 OEU K 1 A20 T21 V31 K33 M45 A46 G47 G48 A49 S96 A20 T21 V31 K33 M45 A46 G47 G48 A49 S96 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20875739 213 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3oeu L 2.6 BS01 OEU K 1 P94 D114 P115 P104 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20875739 213 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3oev K 2.85 BS02 3OE K 1 A20 T21 V31 K33 M45 A46 G47 G48 A49 A20 T21 V31 K33 M45 A46 G47 G48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20875739 213 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3oev L 2.85 BS01 3OE K 1 Y-5 P94 Y96 D114 Y5 P104 Y106 D126 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20875739 213 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3of8 A 2.2 BS01 I0Y A 1 Q20 C26 G62 E64 G69 L70 M71 A136 D163 H164 W190 Q20 C26 G62 E64 G69 L70 M71 A136 D163 H164 W190 Q20 C26 H164 N188 Q20 C26 H164 N188 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 20850545 501 EAPRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 3og7 A 2.45 BS01 032 A 1 I463 A481 L505 L514 T529 W531 C532 F583 D594 F595 G596 I15 A33 L57 L66 T81 W83 C84 F132 D143 F144 G145 D576 K578 N580 N581 D594 S616 D125 K127 N129 N130 D143 S147 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=31nM, Kd=51nM, EC50=2290nM P15056 20823850 1 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTAPQLAIVTQWCEGSSLYHHLHASFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 3ogm B 3.34 BS02 OGK B 1 R85 F89 R348 V385 Y386 R409 L469 R496 W519 R74 F78 R337 V374 Y375 R398 L458 R485 W508 ? 0005515,0006952,0009611,0009625,0009641,0009753,0009861,0009867,0009901,0009909,0010118,0010218,0016567,0019005,0031146,0031348,0042742,0048364,0048443,0050832,0106167 remove_due_to_license_issue O04197 20927106 1100 SCVATVDDVIEQVMTYITDPKDRDSASLVCRRWFKIDSETREHVTMALCYTATPDRLSRRFPNLRSLKLKGKPRAAMFNLIPENWGGYVTPWVTEISNNLRQLKSVHFRRMIVSDLDLDRLAKARADDLETLKLDKCSGFTTDGLLSIVTHCRKIKTLLMEESSFSEKDGKWLHELAQHNTSLEVLNFYMTEFAKISPKDLETIARNCRSLVSVKVGDFEILELVGFFKAAANLEEFCGGSLNEDIGMPEKYMNLVFPRKLCRLGLSYMGPNEMPILFPFAAQIRKLDLLYALLETEDHCTLIQKCPNLEVLETRNVIGDRGLEVLAQYCKQLKRLRIERGADEQGMEDEEGLVSQRGLIALAQGCQELEYMAVYVSDITNESLESIGTYLKNLCDFRLVLLDREERITDLPLDNGVRSLLIGCKKLRRFAFYLRQGGLTDLGLSYIGQYSPNVRWMLLGYVGESDEGLMEFSRGCPNLQKLEMRGCCFSERAIAAAVTKLPSLRYLWVQGYRASMTGQDLMQMARPYWNIELIPSRREHPAHILAYYSLAGQRTDCPTTVRVLKEPI 3ogp A 1.7 BS01 017 A 1 D30 G32 A33 D34 I35 G58 I59 D26 G28 A29 D30 I31 G54 I55 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 ic50=36nM remove_due_to_license_issue P16088 21636894 200 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLSVNLLGRDNMIKFNIRLVM 3ogp A 1.7 BS02 017 B 1 D30 I35 M56 G58 I59 L101 D26 I31 M52 G54 I55 L97 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 ic50=36nM remove_due_to_license_issue P16088 21636894 200 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLSVNLLGRDNMIKFNIRLVM 3ogp B 1.7 BS01 017 A 1 D30 G32 A33 I35 L101 D26 G28 A29 I31 L97 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 ic50=36nM remove_due_to_license_issue P16088 21636894 200 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLSVNLLGRDNMIKFNIRLVM 3ogp B 1.7 BS02 017 B 1 D30 G32 A33 D34 I35 I57 I59 D26 G28 A29 D30 I31 I53 I55 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 ic50=36nM remove_due_to_license_issue P16088 21636894 200 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLSVNLLGRDNMIKFNIRLVM 3ogq A 1.8 BS01 AB1 A 1 D30 G32 A33 D34 I35 I59 D26 G28 A29 D30 I31 I55 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 ic50=30nM remove_due_to_license_issue P16088 21636894 200 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLSVNLLGRDNMIKFNIRLVM 3ogq B 1.8 BS01 AB1 A 1 L28 D30 G32 A33 D34 M56 I57 G58 I59 L101 L24 D26 G28 A29 D30 M52 I53 G54 I55 L97 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 remove_due_to_license_issue P16088 21636894 200 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITVLNRRDFQVKNSIENGRQMMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLSVNLLGRDNMIKFNIRLVM 3ogu A 1.845 BS01 dna T 0 S229 K230 G231 T233 K234 S220 K221 G222 T224 K225 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 21107011 1 ~ 6 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINLLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGKTKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGMLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 3ogu A 1.845 BS02 dna P 0 S104 G105 G107 P108 S109 A110 S95 G96 G98 P99 S100 A101 D190 D192 D256 D181 D183 D247 2.7.7.7,4.2.99.-,4.2.99.18 0001701,0003677,0003684,0003887,0003906,0005515,0005634,0005654,0005737,0005874,0005876,0006259,0006260,0006261,0006281,0006284,0006287,0006290,0006297,0006303,0006915,0006954,0006974,0007435,0008017,0008630,0010332,0016445,0016446,0016779,0016829,0019899,0032991,0034061,0045471,0046872,0048535,0048536,0048872,0051402,0051575,0055093,0071707,0071897,0140078 remove_due_to_license_issue P06746 21107011 1 ~ 6 TLNGGITDMLTELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAKKLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINLLTRVSGIGPSAARKFVDEGIKTLEDLRKNEDKLNHHQRIGLKYFGDFEKRIPREEMLQMQDIVLNEVKKVDSEYIATVCGSFRRGAESSGDMDVLLTHPSFTSESTKQPKLLHQVVEQLQKVHFITDTLSKGKTKFMGVCQLPSKNDEKEYPHRRIDIRLIPKDQYYCGMLYFTGSDIFNKNMRAHALEKGFTINEYTIRPLGVTGVAGEPLPVDSEKDIFDYIQWKYREPKDRSE 3ohf A 2.1 BS01 3HF A 1 L78 D80 G82 Y119 T120 Q121 F156 Y246 D276 G278 T279 T280 R283 L32 D34 G36 Y73 T74 Q75 F110 Y200 D230 G232 T233 T234 R237 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 ic50=94nM remove_due_to_license_issue P56817 21078556 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3ohh A 2.01 BS01 3HH A 1 G59 D80 G82 Y119 T120 Q121 F156 I158 Y246 D276 G278 T279 T280 R283 G13 D34 G36 Y73 T74 Q75 F110 I112 Y200 D230 G232 T233 T234 R237 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 ic50=18nM remove_due_to_license_issue P56817 21078556 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3ohi A 2.3 BS02 HDX A 1 S50 D83 H84 H178 G179 K182 G211 S213 N253 D255 S256 R259 S49 D82 H83 H174 G175 K178 G207 S209 N249 D251 S252 R255 4.1.2.13 0004332,0005515,0005975,0006096,0008270,0016829,0016832,0046872 Ki=14uM remove_due_to_license_issue A8B2U2 21333622 341 PLCTLRQMLGEARKHKYGVGAFNVNNMEQIQGIMKAVVQLKSPVILQCSRGALKYSDMIYLKKLCEAALEKHPDIPICIHLDHGDTLESVKMAIDLGFSSVMIDASHHPFDENVRITKEVVAYAHARSVSVEAELGTLGGIEQNTVQLTEPQDAKKFVELTGVDALAVAIGTSHGAYKFKSESDIRLAIDRVKTISDLTGIPLVMHGSSSVPKDVKDMINKYGGKMPDAVGVPIESIVHAIGEGVCKINVDSDSRMAMTGAIRKVFVEHPEKFDPRDYLGPGRDAITEMLIPKIKAFGSAGHAGDYKVVSLEEAKAWYK 3ohi B 2.3 BS02 HDX B 1 N24 S50 D83 H178 G179 G211 S213 D255 S256 R259 N23 S49 D82 H173 G174 G206 S208 D250 S251 R254 4.1.2.13 0004332,0005515,0005975,0006096,0008270,0016829,0016832,0046872 Ki=14uM remove_due_to_license_issue A8B2U2 21333622 343 PLCTLRQMLGEARKHKYGVGAFNVNNMEQIQGIMKAVVQLKSPVILQCSRGALKYSDMIYLKKLCEAALEKHPDIPICIHLDHGDTLESVKMAIDLGFSSVMIDASHHPFDENVRITKEVVAYAHARSVSVEAELGTLGGIENTVQLTEPQDAKKFVELTGVDALAVAIGTSHGAYKFKSESDIRLAIDRVKTISDLTGIPLVMHGSSSVPKDVKDMINKYGGKMPDAVGVPIESIVHAIGEGVCKINVDSDSRMAMTGAIRKVFVEHPEKFDPRDYLGPGRDAITEMLIPKIKAFGSAGHAGDYKVVSLEEAKAWYK 3oik A 1.5 BS02 WZB A 1 H94 V135 L198 T199 T200 P202 H92 V132 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=232nM, IC50=290nM P00918 300 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3oil A 1.5 BS02 VZ5 A 1 N62 Q67 Q92 H94 H96 V121 F131 L198 T199 T200 N59 Q64 Q89 H91 H93 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3oim A 1.45 BS02 VZ5 A 1 H94 H96 V121 F131 L198 T199 T200 P202 H92 H94 V119 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3oj8 A 1.9 BS01 OJ8 A 1 M191 F192 S217 D237 I238 G239 S241 L278 F381 F432 T488 M159 F160 S185 D205 I206 G207 S209 L246 F349 F400 T456 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 21428410 1 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTP 3ok9 A 1.27 BS01 G52 A 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=5.9pM remove_due_to_license_issue P03366 20827746 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3ok9 B 1.27 BS01 G52 A 1 D125 A128 D130 G148 P181 V182 D25 A28 D30 G48 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 20827746 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3oka A 2.2 BS01 GDD A 1 R206 K211 R260 L261 M266 E298 R203 K208 R257 L258 M263 E295 2.4.1.346 0008654,0009247,0016020,0016757,0016758,0033164,0043750,0046488 Kd=19uM remove_due_to_license_issue Q8NNK8 20843801 701 SRKTLVVTNDFPPRIGGIQSYLRDFIATQDPESIVVFASTQNAEEAHAYDKTLDYEVIRWPRSVMLPTPTTAHAMAEIIREREIDNVWFGAAAPLALMAGTAKQAGASKVIASTHGHEVGWSMLPGSRQSLRKIGTEVDVLTYISQYTLRRFKSAFGSHPTFEHLPSGVDVKRFTPATPEDKSATRKKLGFTDTTPVIACNSRLVPRKGQDSLIKAMPQVIAARPDAQLLIVGSGRYESTLRRLATDVSQNVKFLGRLEYQDMINTLAAADIFAMPARTRGGGLDVEGLGIVYLEAQACGVPVIAGTSGGAPETVTPATGLVVEGSDVDKLSELLIELLDDPIRRAAMGAAGRAHVEAEWSWEIMGERLTNILQSEPR 3okc A 2.4 BS01 GDP A 1 K211 R260 L261 M266 I294 V295 E298 K208 R257 L258 M263 I291 V292 E295 2.4.1.346 0008654,0009247,0016020,0016757,0016758,0033164,0043750,0046488 Kd=36.5uM remove_due_to_license_issue Q8NNK8 20843801 601 SRKTLVVTNDFPPRIGGIQSYLRDFIATQDPESIVVFASTQNAEEAHAYDKTLDYEVIRWPRSVMLPTPTTAHAMAEIIREREIDNVWFGAAAPLALMAGTAKQAGASKVIASTHGHEVGWSMLPGSRQSLRKIGTEVDVLTYISQYTLRRFKSAFGSHPTFEHLPSGVDVKRFTPATPEDKSATRKKLGFTDTTPVIACNSRLVPRKGQDSLIKAMPQVIAARPDAQLLIVGSGRYESTLRRLATDVSQNVKFLGRLEYQDMINTLAAADIFAMPARTRGGGLDVEGLGIVYLEAQACGVPVIAGTSGGAPETVTPATGLVVEGSDVDKLSELLIELLDDPIRRAAMGAAGRAHVEAEWSWEIMGERLTNILQSEPR 3okh A 2.5 BS02 OKH A 1 M269 I277 R335 H348 M22 I30 R88 H101 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=5720nM Q96RI1 21134747 1 ELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDV 3okh A 2.5 BS03 OKH A 2 L291 M294 H298 M332 F333 R335 S336 I339 F340 L352 I356 I361 M369 Y373 L44 M47 H51 M85 F86 R88 S89 I92 F93 L105 I109 I114 M122 Y126 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=5720nM Q96RI1 21134747 2 ELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDV 3oki A 2.0 BS02 OKI A 1 I273 I277 M294 H298 M332 S336 I356 M369 Y373 M454 I27 I31 M48 H52 M86 S90 I110 M123 Y127 M208 ? 0003677,0004879,0006355,0032052,0038183 ic50=0.07uM remove_due_to_license_issue IC50=70nM Q96RI1 21134747 2 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3okp A 2.0 BS01 GDD A 1 R206 K211 R260 L261 M266 I294 V295 E298 R203 K208 R257 L258 M263 I291 V292 E295 2.4.1.346 0008654,0009247,0016020,0016757,0016758,0033164,0043750,0046488 Kd=19uM remove_due_to_license_issue Q8NNK8 20843801 601 SRKTLVVTNDFPPRIGGIQSYLRDFIATQDPESIVVFASTQNAEEAHAYDKTLDYEVIRWPRSVMLPTPTTAHAMAEIIREREIDNVWFGAAAPLALMAGTAKQAGASKVIASTHGHEVGWSMLPGSRQSLRKIGTEVDVLTYISQYTLRRFKSAFGSHPTFEHLPSGVDVKRFTPATPEDKSATRKKLGFTDTTPVIACNSRLVPRKGQDSLIKAMPQVIAARPDAQLLIVGSGRYESTLRRLATDVSQNVKFLGRLEYQDMINTLAAADIFAMPARTRGGGLDVEGLGIVYLEAQACGVPVIAGTSGGAPETVTPATGLVVEGSDVDKLSELLIELLDDPIRRAAMGAAGRAHVEAEWSWEIMGERLTNILQSEPR 3oku A 1.45 BS02 VZ4 A 1 H94 H96 V121 F131 L198 T199 P201 P202 H92 H94 V119 F128 L195 T196 P198 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3okv A 1.45 BS02 VZ4 A 1 N62 H64 Q67 H94 H96 L198 T199 T200 N59 H61 Q64 H91 H93 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3okv A 1.45 BS03 VZ4 A 2 I91 Q92 F131 I88 Q89 F127 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3old A 2.0 BS01 GLC B 1 W58 W59 Q63 H305 W57 W58 Q62 H304 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 1 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS02 GLC B 2 G104 T163 G103 T162 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS03 GLC C 1 K200 E240 K199 E239 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS04 G6D C 1 A198 H201 E233 G306 A197 H200 E232 G305 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 3 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS05 GLC D 1 W134 K172 Y174 W133 K171 Y173 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 1 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS06 GLC D 2 S132 W134 D135 Y174 S131 W133 D134 Y173 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS07 GLC E 1 K322 T377 W388 Q390 K321 T376 W387 Q389 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS08 GLC E 2 R387 R389 Q390 R386 R388 Q389 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 3 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3old A 2.0 BS10 ACI A 1 W58 Y62 H101 R195 D197 E233 H299 D300 W57 Y61 H100 R194 D196 E232 H298 D299 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 503 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS01 GLC B 1 W58 W59 Q63 H305 W57 W58 Q62 H304 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 1 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS02 G6D B 1 W59 Q63 T163 W58 Q62 T162 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS03 GLC C 1 Y151 K200 E240 Y150 K199 E239 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS04 G6D C 1 H201 E233 G306 H200 E232 G305 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 3 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS05 GLC D 1 W134 K172 Y174 W133 K171 Y173 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 1 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS06 GLC D 2 S132 W134 D135 Y174 S131 W133 D134 Y173 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS07 GLC E 1 K322 T377 W388 Q390 K321 T376 W387 Q389 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS08 GLC E 2 R387 R389 Q390 R386 R388 Q389 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 3 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3ole A 1.55 BS10 ACI A 1 W58 Y62 H101 D197 E233 H299 D300 W57 Y61 H100 D196 E232 H298 D299 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 504 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olf A 1.9 BS02 OLF A 1 I277 M294 H298 M332 F333 R335 S336 I339 F340 I356 M369 Y373 I31 M48 H52 M86 F87 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=20nM, EC50=500nM Q96RI1 21269824 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3olg A 2.3 BS01 GLC B 1 W58 W59 Q63 H305 W57 W58 Q62 H304 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 1 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS02 G6D B 1 W59 T163 W58 T162 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS03 GLC C 1 Y151 K200 E240 G306 Y150 K199 E239 G305 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS04 G6D C 1 H201 E233 D300 G306 H200 E232 D299 G305 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 3 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS05 GLC D 1 W134 K172 Y174 W133 K171 Y173 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 2 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS06 GLC D 2 S132 W134 D135 Y174 S131 W133 D134 Y173 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 3 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS07 BGC E 1 K140 E171 W203 D206 K139 E170 W202 D205 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 1 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS09 HSD A 1 W58 Y62 H101 D197 E233 H299 D300 W57 Y61 H100 D196 E232 H298 D299 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 503 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3olg A 2.3 BS11 GLC A 1 K322 T377 W388 Q390 K321 T376 W387 Q389 D197 S226 D300 D196 S225 D299 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 21111049 512 YSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFMPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 3omm A 2.1 BS02 OMM A 1 L291 M294 M332 F333 R335 S336 I339 F340 I356 M369 Y373 L45 M48 M86 F87 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue EC50=300nM, IC50=37nM Q96RI1 21269824 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3on0 A 2.874 BS01 dna P 0 S32 L33 S31 L32 ? 0003677,0005737 remove_due_to_license_issue P33788 21565799 1 ~ 24 PKIQTYVNNNVYEQITDLVTIRKQEGIEEASLSNVSSMLLELGLRVYMIQQEKFNQMEYNKLMLENVSRVRAMCTEILKMSVLNQESIASGNFDYAVIKPAIDKFAREQVSIFFPDDEDDQ 3on0 B 2.874 BS01 dna P 0 Q5 Y7 Q4 Y6 ? 0003677,0005737 remove_due_to_license_issue P33788 21565799 1 ~ 24 PKIQTYVNNNVYEQITDLVTIRKQEGIEEASLSNVSSMLLELGLRVYMIQQEKREGGFNQMEYNKLMLENVSRVRAMCTEILKMSVLNQESIASGNFDYAVIKPAIDKFAREQVSIFF 3on0 C 2.874 BS01 dna P 0 S32 L33 S34 N35 S31 L32 S33 N34 ? 0003677,0005737 remove_due_to_license_issue P33788 21565799 1 ~ 24 PKIQTYVNNNVYEQITDLVTIRKQEGIEEASLSNVSSMLLELGLRVYMIQQEKREGGFNQMEYNKLMLENVSRVRAMCTEILKMSVLNQESIASGNFDYAVIKPAIDKFAREQVSIFF 3on0 D 2.874 BS01 dna P 0 K3 Q5 Y7 K2 Q4 Y6 ? 0003677,0005737 remove_due_to_license_issue P33788 21565799 1 ~ 24 PKIQTYVNNNVYEQITDLVTIRKQEGIEEASLSNVSSMLLELGLRVFNQMEYNKLMLENVSRVRAMCTEILKMSVLNQESIASGNFDYAVIKPAIDKFAREQVSIFF 3oof A 2.29 BS02 OOF A 1 I277 L291 M294 M332 F333 R335 S336 F340 I356 S359 M369 Y373 I31 L45 M48 M86 F87 R89 S90 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=50nM, EC50=2500nM Q96RI1 21269824 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3ook A 2.29 BS02 OOK A 1 I277 L291 M294 H298 M332 F333 R335 S336 I339 F340 I356 M369 Y373 I31 L45 M48 H52 M86 F87 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=4nM, EC50=1400nM Q96RI1 21269824 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3ool A 2.3 BS01 dna C 0 G13 N15 K17 D44 Y46 R48 R50 E61 W62 K63 N90 N94 V96 W149 D150 N152 K193 G11 N13 K15 D42 Y44 R46 R48 E59 W60 K61 N88 N92 V94 W147 D148 N150 K191 3.1.-.- 0004519,0005739,0006314,0006397,0008380 remove_due_to_license_issue P03882 21029741 2 ~ 25 NIKKNQVMNLGPNSKLLKEYKSQLIELNIEQFEAGIGLILGDAYIRSRDEGKTYCMQFEWKNKAYMDHVCLLYDQWVLSPPHKKERVNHLGNLVITWGAQTFKHQAFNKLANLFIVNNKKTIPNNLVENYLTPMSLAYWFMDDGGKWDYNKNSTNKSIVLNTQSFTFEEVEYLVKGLRNKFQLNCYVKINKNKPIIYIDSMSYLIFYNLIKPYLIPQMMYKLP 3ool A 2.3 BS02 dna D 0 P14 N15 K23 L80 S81 H84 K86 R88 Q102 F104 K105 Y151 N152 Q165 S166 P12 N13 K21 L78 S79 H82 K84 R86 Q100 F102 K103 Y149 N150 Q163 S164 3.1.-.- 0004519,0005739,0006314,0006397,0008380 remove_due_to_license_issue P03882 21029741 2 ~ 25 NIKKNQVMNLGPNSKLLKEYKSQLIELNIEQFEAGIGLILGDAYIRSRDEGKTYCMQFEWKNKAYMDHVCLLYDQWVLSPPHKKERVNHLGNLVITWGAQTFKHQAFNKLANLFIVNNKKTIPNNLVENYLTPMSLAYWFMDDGGKWDYNKNSTNKSIVLNTQSFTFEEVEYLVKGLRNKFQLNCYVKINKNKPIIYIDSMSYLIFYNLIKPYLIPQMMYKLP 3oor A 2.5 BS01 dna C 0 G13 N15 K17 D44 Y46 R48 R50 E61 W62 K63 N90 N94 W149 D150 N152 K193 G11 N13 K15 D42 Y44 R46 R48 E59 W60 K61 N88 N92 W147 D148 N150 K191 3.1.-.- 0004519,0005739,0006314,0006397,0008380 remove_due_to_license_issue P03882 21029741 2 ~ 25 NIKKNQVMNLGPNSKLLKEYKSQLIELNIEQFEAGIGLILGDAYIRSRDEGKTYCMQFEWKNKAYMDHVCLLYDQWVLSPPHKRERVNHLGNLVITWTAQTFKHQAFNKLANLFIVNNKKTIPNNLVENYLTPMSLAYWFMDDGGKWDYNKNSTNKSIVLNTQSFTFEEVEYLVKGLRNKFQLNCYVKINKNKPIIYIDSMSYLIFYNLIKPYLIPQMMYKLP 3oor A 2.5 BS02 dna D 0 P14 N15 L80 S81 R86 R88 F104 K105 D144 Y151 N152 N163 Q165 S166 K193 K195 Y222 P12 N13 L78 S79 R84 R86 F102 K103 D142 Y149 N150 N161 Q163 S164 K191 K193 Y220 3.1.-.- 0004519,0005739,0006314,0006397,0008380 remove_due_to_license_issue P03882 21029741 2 ~ 25 NIKKNQVMNLGPNSKLLKEYKSQLIELNIEQFEAGIGLILGDAYIRSRDEGKTYCMQFEWKNKAYMDHVCLLYDQWVLSPPHKRERVNHLGNLVITWTAQTFKHQAFNKLANLFIVNNKKTIPNNLVENYLTPMSLAYWFMDDGGKWDYNKNSTNKSIVLNTQSFTFEEVEYLVKGLRNKFQLNCYVKINKNKPIIYIDSMSYLIFYNLIKPYLIPQMMYKLP 3oot A 2.55 BS01 SSR A 1 Q13 D32 Y75 T77 V120 D215 G217 A218 S219 H287 Q16 D35 Y80 T82 V124 D223 G225 A226 S227 H298 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=2nM P00797 20850300 327 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3ooz A 1.8 BS01 ZOO A 1 Q74 G75 D94 S97 N99 Y133 W138 F170 I172 W177 I180 D290 G292 T293 T294 Q14 G15 D34 S37 N39 Y73 W78 F110 I112 W117 I120 D223 G225 T226 T227 D94 S97 N99 A101 Y133 D290 T293 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=0.014uM remove_due_to_license_issue IC50=32nM P56817 20880704 1 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACDEFRTAAVEGPFVTLDMEDCGY 3opm A 2.72 BS01 LUI A 1 E205 E206 F357 Y547 Y662 Y666 E166 E167 F318 Y508 Y623 Y627 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=240nM P27487 21764322 800 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3opp A 1.8 BS01 SA2 A 1 S70 Y105 S130 N132 T235 G236 A237 S45 Y80 S105 N107 T204 G205 A206 S70 K73 S130 K234 A237 S45 K48 S105 K203 A206 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 21357298 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDSWALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3opr A 1.65 BS03 SA2 A 1 S70 Y105 S130 T235 G236 A237 S45 Y80 S105 T203 G204 A205 S70 K73 S130 K234 A237 S45 K48 S105 K202 A205 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 21357298 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDHALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3oqf A 2.78 BS01 S51 A 1 Q13 D32 Y75 T77 P111 V120 D215 G217 S219 M289 Q16 D35 Y80 T82 P115 V124 D223 G225 S227 M300 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=91nM P00797 20850300 328 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3oqk A 2.9 BS01 S52 A 1 Q13 D32 Y75 T77 V120 D215 G217 A218 S219 M289 Q16 D35 Y80 T82 V124 D223 G225 A226 S227 M300 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=420nM P00797 20850300 327 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3oqm A 2.96 BS01 dna E 0 S16 A18 T19 R22 N29 V30 K31 T34 L56 A57 K59 S15 A17 T18 R21 N28 V29 K30 T33 L55 A56 K58 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqm A 2.96 BS02 dna B 0 T5 I6 S21 Y47 N50 A53 R54 A57 T4 I5 S20 Y46 N49 A52 R53 A56 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqm C 2.96 BS01 dna E 0 T5 I6 Y7 M17 S21 Y47 P49 N50 A53 R54 A57 T4 I5 Y6 M16 S20 Y46 P48 N49 A52 R53 A56 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqm C 2.96 BS02 dna B 0 S16 M17 A18 T19 R22 N29 V30 K31 T34 L56 K59 S15 M16 A17 T18 R21 N28 V29 K30 T33 L55 K58 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqn A 3.3 BS01 dna E 0 M2 I6 A18 S21 N25 Y47 P49 N50 A53 R54 A57 M1 I5 A17 S20 N24 Y46 P48 N49 A52 R53 A56 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqn A 3.3 BS02 dna B 0 S16 A18 T19 R22 N29 V30 K31 T34 L56 A57 K59 S15 A17 T18 R21 N28 V29 K30 T33 L55 A56 K58 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqn C 3.3 BS01 dna E 0 S16 A18 T19 R22 N29 V30 K31 T34 L56 A57 K59 S15 A17 T18 R21 N28 V29 K30 T33 L55 A56 K58 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3oqn C 3.3 BS02 dna B 0 T5 I6 Y7 M17 S21 Y47 N50 A53 R54 A57 T4 I5 Y6 M16 S20 Y46 N49 A52 R53 A56 ? 0000976,0001216,0001217,0003677,0003700,0005515,0006355,0032993,0045892,0045893 remove_due_to_license_issue P25144 21106498 700 ~ 715 MNITIYDVAREANVSMATVSRVVNGNPNVKPTTRKKVLEAIERLGYRPNAVARGLASKKTTTVGVIIPDISSIFYSELARGIEDIATMYKYNIILSNSDQNMEKELHLLNTMLGKQVDGIVFMGGNITDEHVAEFKRSPVPIVLAASVEEQEETPSVAIDYEQAIYDAVKLLVDKGHTDIAFVSGPMAEPINRSKKLQGYKRALEEANLPFNEQFVAEGDYTYDSGLEALQHLMSLDKKPTAILSATDEMALGIIHAAQDQGLSIPEDLDIIGFDNTRLSLMVRPQLSTVVQPTYDIGAVAMRLLTKLMNKEPVEEHIVELPHRIELRKSTK 3orn A 2.8 BS03 3OR A 1 G80 K97 L118 V127 I141 R189 D208 F209 G210 V211 L215 I216 N221 G20 K37 L58 V67 I81 R129 D148 F149 G150 V151 L155 I156 N161 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T166 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=8.8nM, Kd=0.24nM Q02750 21316218 400 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIG 3os3 A 2.8 BS02 3OS A 1 G80 K97 L118 I141 R189 D208 F209 V211 L215 I216 M219 G19 K36 L57 I80 R128 D147 F148 V150 L154 I155 M158 D190 K192 S194 N195 D208 D217 T226 D129 K131 S133 N134 D147 D156 T165 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue Q02750 21316218 400 ELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPMAIFELLDYIVNEPPPKLPVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCST 3osf A 2.032 BS01 dna B 0 K49 Q50 K51 R84 Q85 R89 Y93 N139 K2 Q3 K4 R37 Q38 R42 Y46 N92 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 13 KKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osf A 2.032 BS02 dna C 0 K48 K49 W71 R87 K91 R120 W122 A123 K138 K1 K2 W24 R40 K44 R73 W75 A76 K91 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 13 KKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osf D 2.032 BS01 dna E 0 K49 Q50 K51 F52 R84 Q85 R89 Y93 N139 T143 K2 Q3 K4 F5 R37 Q38 R42 Y46 N92 T96 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 13 KKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osf D 2.032 BS02 dna F 0 K48 K49 K72 R87 K91 R120 W122 A123 K138 K1 K2 K25 R40 K44 R73 W75 A76 K91 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 13 KKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osg A 1.997 BS01 dna B 0 K49 Q50 K51 R84 Q85 R89 Y93 N139 V142 T143 N146 K9 Q10 K11 R44 Q45 R49 Y53 N99 V102 T103 N106 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 12 VQVNKAAKKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osg A 1.997 BS02 dna C 0 A47 K48 K49 R87 R120 W122 A123 K138 A7 K8 K9 R47 R80 W82 A83 K98 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 12 VQVNKAAKKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osg D 1.997 BS01 dna E 0 K49 Q50 K51 F52 R84 Q85 R89 Y93 N139 K2 Q3 K4 F5 R37 Q38 R42 Y46 N92 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 12 KKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osg D 1.997 BS02 dna F 0 K48 K49 R87 K91 R120 W122 A123 K138 K1 K2 R40 K44 R73 W75 A76 K91 ? remove_due_to_license_issue Q58HP3 21771861 1 ~ 12 KKQKFTPEEDEMLKRAVAQHGSDWKMIAATFPNRNARQCRDRWKNYLAPSISHTPWTAEEDALLVQKIQEYGRQWAIIAKFFPGRTDIHIKNRWVTISNKLGI 3osi A 2.7 BS01 XDH A 1 C285 R288 S289 L340 I341 S342 E343 C69 R72 S73 L124 I125 S126 E127 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 21561829 1 NPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3osw A 2.55 BS01 XDI A 1 C285 R288 S289 L340 I341 S342 E343 C70 R73 S74 L125 I126 S127 E128 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 21561829 1 NPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKISKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3ot3 A 1.44 BS01 22K A 1 L15 G16 A36 V68 C87 E91 L137 K270 K271 L11 G12 A31 V56 C75 E79 L125 K258 K259 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.005uM remove_due_to_license_issue O14757 21094607 1 FVEDWDLVQTLGEGAGEVQLAVNRVTEEAVAVKIVDMENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3ot8 A 1.6455 BS01 MI5 A 1 G16 A36 V68 Y86 C87 G90 E91 E134 L137 D148 K271 G12 A29 V53 Y66 C67 G70 E71 E114 L117 D128 K251 D130 K132 E134 N135 D148 T170 D110 K112 E114 N115 D128 T150 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.009uM remove_due_to_license_issue IC50=9nM O14757 21094608 1 FVEDWDLVQTLGEGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3otf A 2.4 BS01 CMP A 1 V642 F658 G659 E660 I661 C662 R669 T670 R710 V122 F138 G139 E140 I141 C142 R149 T150 R190 ? Kd=0.83uM remove_due_to_license_issue Q9Y3Q4 20829353 725 DSSRRQYQEKYKQVEQYMSFHKLPPDTRQRIHDYYEHRYQGKMFDEESILGELSEPLREEIINFNCRKLVASMPLFANADPNFVTSMLTKLRFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKETKLADGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVALDRLDRIGKK 3otq A 3.0 BS01 MZL A 1 F267 D335 W336 Y383 S407 L408 R410 S415 M419 L428 Y466 V498 H524 F264 D332 W333 Y380 S404 L405 R407 S412 M416 L425 Y463 V495 H521 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F264 H331 D332 W333 N356 N375 Y380 Y463 D493 H521 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=41nM P34913 20934334 556 RAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 3otx A 1.55 BS01 AP5 A 1 N13 L15 D17 G63 S64 N67 C123 R132 A136 F169 N222 T264 D266 I267 V283 Q288 G296 A297 G298 D299 H323 A326 Q327 I330 N10 L12 D14 G60 S61 N64 C120 R129 A133 F166 N219 T261 D263 I264 V280 Q285 G293 A294 G295 D296 H320 A323 Q324 I327 R132 D299 R129 D296 2.7.1.20 0004001,0005524,0005634,0005654,0005737,0005829,0006144,0006166,0009152,0016301,0020015,0044209,0097014 ic50=29.4uM remove_due_to_license_issue Q584S0 21629723 346 APLRVYVQCNPLLDVSAHVSDEFLVKYGLERGTAILLSERQKGIFDDIEKMPNVRYVPGGSGLNVARVAQWMQQAYKGKFVTYVGCIADDRYGKVLKEAAEHEGIVMAVEHTTKAGSGACAVCITGKERTLVADLGAANHLSSEHMRSPAVVRAMDESRIFYFSGFTLTVDVNHVLQACRKAREVDGLFMINLSAPFIMQFFSAQLGEVLPYTDIIVANRHEAKEFANMMKWDTDCVEEIARRAVSEVPYTGTKGRVVVFTRDIESTVLATKDGVETVPVPQLDQDKVIDMNGAGDAFMGGFLSAYAVGKDLRRCCETGHYTAQEVIQRDPEKPSFSP 3ouh A 2.51 BS02 014 A 1 M299 Y310 H313 D315 Y329 L343 H374 V376 R383 W389 M108 Y119 H122 D124 Y138 L152 H183 V185 R192 W198 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=79.43nM Q9GZT9 24900242 417 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKY 3oui A 1.7 BS02 42Z A 1 R252 M299 Y310 H313 D315 Y329 H374 V376 R383 W389 R54 M101 Y112 H115 D117 Y127 H172 V174 R181 W187 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=12589.25nM Q9GZT9 24900242 393 PALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFD 3oui A 1.7 BS03 42Z A 2 N203 I280 C283 K286 S289 Y290 N15 I82 C85 K88 S91 Y92 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=12589.25nM Q9GZT9 24900242 2 PALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFD 3ouj A 2.3 BS02 AKG A 1 Y310 H313 Y329 L343 H374 V376 R383 Y124 H127 Y143 L157 H188 V190 R197 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue Q9GZT9 24900242 417 GQTKPLPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVGEKGVRVELNK 3ovn A 1.95 BS02 MPV A 1 G197 V201 G133 V137 3.1.13.2,3.1.26.13 0003676,0015074 Kd=2.8mM remove_due_to_license_issue Q72498 21275048 213 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEDGIPESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATD 3ovn A 1.95 BS03 MPV B 1 R107 W108 P109 I204 R52 W53 P54 I140 3.1.13.2,3.1.26.13 0003676,0015074 Kd=2.8mM remove_due_to_license_issue Q72498 21275048 213 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEDGIPESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATD 3ovn B 1.95 BS03 MPV A 1 R107 P109 I208 R51 P53 I140 3.1.13.2,3.1.26.13 0003676,0015074 Kd=2.8mM remove_due_to_license_issue Q72498 21275048 213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEDESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATDIQ 3ovn B 1.95 BS04 MPV B 1 G197 E198 G129 E130 3.1.13.2,3.1.26.13 0003676,0015074 Kd=2.8mM remove_due_to_license_issue Q72498 21275048 213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACDWAGIKQEDESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGIGGYSAGERIVDIIATDIQ 3ovx A 1.49 BS01 O64 A 1 G23 C25 W26 G68 G69 V162 N163 G165 G23 C25 W26 G68 G69 V162 N163 G165 Q19 C25 H164 N184 Q19 C25 H164 N184 3.4.22.27 0006508,0008234 remove_due_to_license_issue IC50=31nM P25774 21030256 218 LPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEI 3ovz A 2.02 BS01 O96 A 1 Q19 G23 C25 G65 G66 Y67 A134 L160 N161 H162 A163 L209 Q17 G21 C23 G63 G64 Y65 A132 L158 N159 H160 A161 L207 Q19 C25 H162 N182 Q17 C23 H160 N180 3.4.22.38 0006508,0008234 remove_due_to_license_issue IC50=8.7nM P43235 21030256 1 DSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 3ow3 A 1.9 BS02 SMY A 1 L49 G50 T51 V57 A70 K72 M120 Y122 V123 E127 L173 T183 D184 F327 L35 G36 T37 V43 A56 K58 M106 Y108 V109 E113 L159 T169 D170 F313 D166 K168 E170 N171 D184 T201 D152 K154 E156 N157 D170 T187 2.7.11.11 0000122,0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,0141156,1904262,1904539,1990044,2000810 ic50=742nM remove_due_to_license_issue P05132 20971641 401 VKEFLAKAKEDFLKKWETPSQNTAQLDQFDRIKTLGTGSFGRVMLVKHKESGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVAGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 3ow4 A 2.6 BS02 SMY A 1 L156 G162 K163 V164 A230 E234 M281 T291 F438 L13 G19 K20 V21 A87 E91 M138 T148 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=22nM P31749 20971641 1 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITRPHFPQFDYSASS 3ow6 A 1.8 BS01 MEX A 1 N51 A55 D93 I96 G97 M98 T184 N35 A39 D77 I80 G81 M82 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=220nM P07900 21106457 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3owb A 2.05 BS01 BSM A 1 N51 S52 A55 K58 D93 I96 G97 M98 D102 L107 G108 F138 T184 N35 S36 A39 K42 D77 I80 G81 M82 D86 L91 G92 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 21106457 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3owd A 1.63 BS01 MEY A 1 N51 A55 D93 I96 G97 M98 N106 F138 T184 N35 A39 D77 I80 G81 M82 N90 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue EC50=190nM, IC50=550nM P07900 21106457 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYETLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3owj A 1.85 BS01 1EL A 1 V53 V66 H160 I174 V51 V64 H158 I172 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.86uM remove_due_to_license_issue P68400 21118972 332 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 3owk A 1.8 BS01 18E A 1 V53 V66 K68 F113 V116 I174 D175 V52 V65 K67 F112 V115 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 ic50=1.5uM remove_due_to_license_issue P68400 21118972 332 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 3owl A 2.1 BS01 19E A 1 V53 V66 K68 F113 M163 I174 D175 V52 V65 K67 F112 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.67uM remove_due_to_license_issue P68400 21118972 332 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 3own A 2.0 BS01 3OX A 1 Q16 D35 G37 Y80 T82 P115 L118 F121 Q132 D223 G225 A226 S227 Y228 S230 M300 Q16 D35 G37 Y80 T82 P115 L118 F121 Q132 D220 G222 A223 S224 Y225 S227 M297 D35 S38 N40 W42 Y80 D223 A226 D35 S38 N40 W42 Y80 D220 A223 3.4.23.15 0004190,0006508 Ki=34nM remove_due_to_license_issue P00797 21112780 500 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3oxc A 1.16 BS01 ROC A 1 D25 G27 D29 D30 G48 I50 I84 D25 G27 D29 D30 G48 I50 I84 3.4.23.16 0004190,0006508,0042802 Ki=3.9nM remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3oxc B 1.16 BS01 ROC A 1 R108 D125 G127 G149 I150 V182 I184 R8 D25 G27 G49 I50 V82 I84 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 17243183 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3oxi A 2.2 BS02 SYY A 1 I70 G71 V78 A91 M146 E147 L148 M149 N152 V196 L206 I25 G26 V33 A46 M101 E102 L103 M104 N107 V151 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T166 2.7.11.24 0004672,0004707,0005524,0006468 ic50=2.2uM remove_due_to_license_issue IC50=2200nM P53779 21071223 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVREHTIEEWKELIYKEVMN 3oxz A 2.2 BS01 0LI A 1 L248 Y253 A269 K271 E286 M290 I293 L298 V299 T315 F317 M318 I360 H361 L370 V379 A380 D381 F382 L21 Y26 A42 K44 E53 M57 I60 L65 V66 T82 F84 M85 I127 H128 L137 V146 A147 D148 F149 D363 A365 R367 N368 D381 P402 D130 A132 R134 N135 D148 P159 2.7.10.2 0004672,0004713,0005524,0006468 ic50=8.6nM remove_due_to_license_issue P00520 21118377 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSYTGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG 3oy0 A 1.6 BS02 OY0 A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10.1nM remove_due_to_license_issue Ki=10.1nM P00918 21506569 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3oy1 A 1.7 BS01 589 A 1 I70 V78 A91 K93 I124 L144 M146 M149 Q155 S193 L206 I25 V30 A43 K45 I76 L96 M98 M101 Q107 S145 L158 D189 K191 N194 D207 T226 D141 K143 N146 D159 T164 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.016uM remove_due_to_license_issue IC50=16nM P53779 21112785 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPEREHTIEEWKELIYKEVMN 3oy3 A 1.95 BS01 XY3 A 1 L248 A269 V270 E286 M290 V299 I315 F317 M318 I360 H361 V379 A380 D381 F382 L21 A42 V43 E59 M63 V72 I88 F90 M91 I133 H134 V152 A153 D154 F155 D363 A365 R367 N368 D381 P402 D136 A138 R140 N141 D154 P175 2.7.10.2 0004672,0004713,0005524,0006468 ic50=35.8nM remove_due_to_license_issue P00520 21118377 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG 3oy8 A 2.19 BS01 GCO C 1 R48 E71 R73 R48 E71 R73 ? 0002317,0003723,0005515,0005576,0005615,0005737,0005788,0005829,0005886,0006915,0007165,0030246,0030395,0031295,0042981,0043065,0043123,0043236,0045445,0046598,0048018,0050729,0062023,0070062,0098609,1990724,2000329,2001200 remove_due_to_license_issue P09382 20826047 1 ACGLVASNLNLKPGECLRVRGEVAPDAKSFVLNLGKDSNNLCLHFNPRFNAHGDANTIVCNSKDGGAWGTEQREAVFPFQPGSVAEVCITFDQANLTVKLPDGYEFKFPNRLNLEAINYMAADGDFKIKCVAFD 3oy8 A 2.19 BS02 GAL C 1 H44 R48 N61 E71 H44 R48 N61 E71 ? 0002317,0003723,0005515,0005576,0005615,0005737,0005788,0005829,0005886,0006915,0007165,0030246,0030395,0031295,0042981,0043065,0043123,0043236,0045445,0046598,0048018,0050729,0062023,0070062,0098609,1990724,2000329,2001200 remove_due_to_license_issue P09382 20826047 2 ACGLVASNLNLKPGECLRVRGEVAPDAKSFVLNLGKDSNNLCLHFNPRFNAHGDANTIVCNSKDGGAWGTEQREAVFPFQPGSVAEVCITFDQANLTVKLPDGYEFKFPNRLNLEAINYMAADGDFKIKCVAFD 3oyl A 2.54 BS06 ZZX A 1 D128 D185 Y212 P214 Q215 E221 D121 D178 Y205 P207 Q208 E214 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0015074 remove_due_to_license_issue P14350 21030679 398 LDAELDQLLQGHYIKGYPKQYTYFLEDGKVKVSRPEGVKIIPPQSDRQKIVLQAHNLAHTGREATLLKIANLYWWPNMRKDVVKQLGRCQQCLITNASNKASGPILRPDRPQKPFDKFFIDYIGPLPPSQGYLYVLVVVDGMTGFTWLYPTKAPSTSATVKSLNVLTSIAIPKVIHSDQGAAFTSSTFAEWAKERGIHLEFSTPYHPQSHGKVERKNSDIKRLLTKLLVGRPTKWYDLLPVVQLALNNTYSPVLKYTPHQLLFGIDSNTPFANQDTLDLTREEELSLLQEIRTSLYHPSTPPASSRSWSPVVGQLVQERVARPASLRPRWHKPSTVLKVLNPRTVVILDHLGNNRTVSIDNLKPTSHQ 3oyn A 2.68 BS06 ZZX A 1 D128 D185 P214 E221 D121 D178 P207 E214 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0015074 remove_due_to_license_issue P14350 21030679 398 LDAELDQLLQGHYIKGYPKQYTYFLEDGKVKVSRPEGVKIIPPQSDRQKIVLQAHNLAHTGREATLLKIANLYWWPNMRKDVVKQLGRCQQCLITNASNKASGPILRPDRPQKPFDKFFIDYIGPLPPSQGYLYVLVVVDGMTGFTWLYPTKAPSTSATVKSLNVLTSIAIPKVIHSDQGAAFTSSTFAEWAKERGIHLEFSTPYHPQSSGKVERKHSDIKRLLTKLLVGRPTKWYDLLPVVQLALNNTYSPVLKYTPHQLLFGIDSNTPFANQDTLDLTREEELSLLQEIRTSLYHPSTPPASSRSWSPVVGQLVQERVARPASLRPRWHKPSTVLKVLNPRTVVILDHLGNNRTVSIDNLKPTSHQ 3oyq A 1.47 BS02 OYQ A 1 H94 H96 H119 F131 L198 T199 T200 P202 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10.3nM remove_due_to_license_issue P00918 21506569 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3oys A 1.538 BS02 OYS A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=9nM remove_due_to_license_issue Ki=107nM P00918 21506569 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3oz1 A 3.0 BS02 BMB A 1 D297 G306 L307 R308 C309 W310 E311 D314 W323 L353 D45 G54 L55 R56 C57 W58 E59 D62 W71 L101 2.3.2.27 remove_due_to_license_issue IC50=<2nM Q13490 20954235 600 FSISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRYPHLLEQLLS 3ozg A 1.993 BS01 SSI A 1 Y116 E144 D145 I146 D148 T149 G150 T152 K176 F197 V198 Y115 E143 D144 I145 D147 T148 G149 T151 K175 F196 V197 E144 D145 D148 F197 R210 E143 D144 D147 F196 R209 2.4.2.22,2.4.2.8 0000166,0000287,0000310,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032265,0046100,0046872,0052657 Ki=0.65nM remove_due_to_license_issue P20035 22726686 232 PIPNNPGAGENAFDPVFVNDDDGYDLDSFMIPAHYKKYLTKVLVPNGVIKNRIEKLAYDIKKVYNNEEFHILCLLKGSRGFFTALLKHLSRIHNYSAVETSKPLFGEHYVRVKSYCNDQSTGTLEIVSEDLSCLKGKHVLIVEDIIDTGKTLVKFCEYLKKFEIKTVAIACLFIKRTPLWNGFKADFVGFSIPDHFVVGYSLDYNEIFRDLDHCCLVNDEGKKKYKA 3ozj A 2.1 BS02 BGV A 1 I268 F313 F346 C432 L436 I25 F70 F103 C189 L193 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 21262235 1 NEDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 3ozp A 2.0 BS01 OAN A 1 R220 D367 E368 W424 W448 Y475 D477 W490 W524 E526 R198 D345 E346 W402 W426 Y453 D455 W468 W502 E504 D367 E368 D345 E346 3.2.1.52 0000272,0004553,0004563,0005886,0005975,0006032,0016231,0016798,0030203 Ki=0.24uM remove_due_to_license_issue Q06GJ0 21692744 1 EDVVWRWSCDNGKCVKLKNDPRSSEPALSLEACKMFCNEYGLLWPRPTGEADLGNFLSKINLNSIEVKILKKGATDDLMEAAAKRFKEQVSLAIPRGSTPKLTGKAVDVYLVNENPNEKAFSLEMDESYGLRVSPSGADRVNATITANSFFGMRHGLETLSQLFVFDDIRDHLLMVRDVNISDKPVYPYRGILLDTARNYYSIESIKRTIEAMAAVKLNTFHWHITDSQSFPFVTTKRPNLYKFGALSPQKVYTKAAIREVVRFGLERGVRVLPEFDAPAHVGEGWQDTDLTVCFKAEPWKSYCVEPPCGQLNPTKDELYQYLEDIYSDMAEVFDTTDIFHMGGDEVSEACWNSSDSIQNFMMQNRWDLDKESFLKLWNYFQQKAQDKAYKAFGKKLPLILWTSTLTNYKHIDDYLNKDDYIIQVWTTGVDPQIKGLLEKGYRLIMSNYDALYFDCGYGAWVGAGNNWCSPYIGWQKVYDNSPAVIALEHRDQVLGGEAALWSEQSDTSTLDGRLWPRAAALAERLWAEPATSWQDAEYRMLHIRERLVRMGIQAESLQPEWCYQNEGYCYS 3ozr A 1.73 BS02 OZR A 1 W38 M40 Y68 E90 C95 H142 K144 N170 E199 W36 M38 Y66 E88 C93 H140 K142 N168 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=7022nM remove_due_to_license_issue P22734 21538606 224 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3ozs A 1.44 BS02 OZS A 1 W38 M40 G66 M89 E90 I91 S119 D141 H142 W143 K144 N170 P174 E199 W36 M38 G64 M87 E88 I89 S117 D139 H140 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=4645nM remove_due_to_license_issue P22734 21538606 223 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3ozt A 1.48 BS02 OZZ A 1 W38 M40 G66 Y68 M89 E90 I91 A118 S119 D141 H142 W143 K144 N170 P174 E199 W36 M38 G64 Y66 M87 E88 I89 A116 S117 D139 H140 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 Ki=74.9uM remove_due_to_license_issue P22734 21538606 223 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3p0g A 3.5 BS01 P0G A 1 W109 D113 V117 C191 F193 A200 S203 S207 F289 F290 N293 Y308 N312 W87 D91 V95 C169 F171 A178 S181 S185 F229 F230 N233 Y248 N252 3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue P00720,P07550 21228869 366 DVTQQRDEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCLRR 3p17 H 1.43 BS03 99P H 1 Y60A W60D E192 S214 W215 G216 G219 Y47 W50 E195 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=33.4uM remove_due_to_license_issue P00734 22366545 1001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3p1d A 1.86 BS01 MB3 A 1 V1115 N1168 V33 N86 2.3.1.-,2.3.1.48 remove_due_to_license_issue IC50=2300000nM Q92793 22464331 1198 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 3p23 A 2.7 BS02 ADP A 1 H579 G580 A597 K599 I642 C645 K690 D711 H17 G18 A35 K37 I80 C83 K128 D149 D688 K690 N693 D711 T734 D126 K128 N131 D149 T160 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue O75460 21317875 1002 VVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCKKLVPGTEGWIAPEMLSEDNPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPAEVRETLGTLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFH 3p2e A 1.68 BS01 SAH A 1 G32 T33 N38 D55 P56 A86 A87 E88 L104 F105 W107 T109 L110 S195 W197 G31 T32 N37 D54 P55 A85 A86 E87 L103 F104 W106 T108 L109 S180 W182 2.1.1.180 0008168,0032259,0046677 Kd=0.6uM remove_due_to_license_issue A8C927 21062819 6732 LILKGTKTVDLSKDELTEIIGQFDRVHIDLGTGDGRNIYKLAINDQNTFYIGIDPVKENLFDISKKIIKKPSKGGLSNVVFVIAAAESLPFELKNIADSISILFPWGTLLEYVIKPNRDILSNVADLAKKEAHFEFVTTYSDLSKAYFLSEQYKAELSNSGFRIDDVKELDNEYVKQFNSLWAKRLAFGRKRSFFRVSGHV 3p2h A 2.0 BS02 NOO A 1 F27 L31 L102 R104 F105 I142 G143 V144 T145 F146 M149 F27 L31 L100 R102 F103 I130 G131 V132 T133 F134 M137 2.3.1.184 0007165,0009372,0016740,0061579 remove_due_to_license_issue Q4VSJ8 21730159 300 MQTFVHEAGRLPAHIAAELGSYRYRVFVEQLGWQLPSEDEKMERDQYDRDDTVYVLGRDANGEICGCARLLPTTRPYLLQEVFPHLLADEAPRSAHVWELSRFAATAWSVRPMLAAAVECAARRGARQLIGVTFCSMERMFRRIGVHAHRAGAPVSIDGRMVVACWIDIDAQTLAALDLDPALC 3p2k A 2.7 BS01 SAM A 1 G32 T33 N38 D55 P56 A87 E88 L104 F105 W107 L110 S195 W197 G31 T32 N37 D54 P55 A86 E87 L103 F104 W106 L109 S176 W178 2.1.1.180 0008168,0032259,0046677 remove_due_to_license_issue A8C927 21062819 6735 LILKGTKTVDLSKDELTEIIGQFDRVHIDLGTGDGRNIYKLAINDQNTFYIGIDPVKENLFDISKKIIKKPSKGGLSNVVFVIAAAESLPFELKNIADSISILFPWGTLLEYVIKPNRDILSNVADLAKKEAHFEFVTTYKAYFLSEQYKAELSNSGFRIDDVKELDNEYVKQFNSLWAKRLAFGRKRSFFRVSGHV 3p3g A 1.65 BS02 3P3 A 1 L62 C63 E78 H79 T191 M195 I198 G210 S211 F212 A215 H238 D242 H265 L62 C63 E78 H79 T191 M195 I198 G210 S211 F212 A215 H238 D242 H265 0009245,0103117 Ki=0.18nM remove_due_to_license_issue 21167751 401 MIKQRTLKRIVQATGVGLHTGKKVTLTLRPAPANTGVIYRRTDLNPPVDFPADAKSVRDTMLCTCLVNEHDVRISTVEHLNAALAGLGIDNIVIEVNAPEIPIMDGSAAPFVYLLLDAGIDELNCAKKFVRIKETVRVEDGDKWAEFKPYNGFSLDFTIDFNHPAIDSSNQRYAMNFSADAFMRQISRARTFGFMRDIEYLQSRGLCLGGSFDCAIVVDDYRVLNEDGLRFEDEFVRHKMLDAIGDLFMCGHNIIGAFTAYKSGHALNNKLLQAVLAKQEAWEYVTFQDDAELPLAFKAP 3p3h A 1.5 BS02 84A A 1 Q92 H94 H119 V121 F130 L197 T198 P200 P201 Q90 H92 H117 V119 F128 L195 T196 P198 P199 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22258283 300 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p3j A 1.6 BS01 498 A 1 H94 H119 V121 F130 L197 T198 P200 P201 H91 H116 V118 F127 L194 T195 P197 P198 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22258283 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p3r A 1.25 BS01 3M1 A 1 K15 L17 A108 A109 L110 S117 K6 L8 A99 A100 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=755nM, Kd=184nM P02766 21865539 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3r B 1.25 BS01 3M1 B 1 K15 L17 A108 L110 K6 L8 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=755nM, Kd=184nM P02766 21865539 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3p3s A 1.6 BS01 3M2 A 1 K15 L17 K5 L7 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 21865539 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3s A 1.6 BS02 3M2 A 2 V65 E66 N98 D99 S100 G101 P102 V55 E56 N88 D89 S90 G91 P92 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 21865539 129 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3s B 1.6 BS01 3M2 B 1 K15 L17 A108 S117 K5 L7 A98 S107 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 21865539 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3s B 1.6 BS02 3M2 B 2 E66 N98 D99 S100 G101 P102 E56 N88 D89 S90 G91 P92 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 21865539 129 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3t A 1.45 BS01 3M3 A 1 A108 L110 S117 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=296nM, Kd=320nM P02766 21865539 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3t B 1.45 BS01 3M3 B 1 K15 A108 L110 S117 K5 A98 L100 S107 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=296nM, Kd=320nM P02766 21865539 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3p3u A 1.5 BS01 3M4 A 1 A108 L110 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=329nM P02766 21865539 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3p3u B 1.5 BS01 3M4 B 1 A108 L110 S117 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue IC50=329nM P02766 21865539 128 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3p44 A 2.2 BS01 067 A 1 H94 F130 V134 L197 T198 T199 H91 F127 V131 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22258283 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p4q A 3.35 BS02 OAA A 1 G50 F116 H232 T244 E245 H355 R390 G51 F117 H233 T245 E246 H356 R391 A47 F116 T203 Q230 H232 L242 E245 R248 R287 H355 Y356 R390 A48 F117 T204 Q231 H233 L243 E246 R249 R288 H356 Y357 R391 1.3.5.1 0000104,0000166,0005515,0005829,0005886,0006113,0006974,0008177,0009055,0009061,0016020,0016491,0016627,0019645,0022900,0044780,0045283,0050660,0071949 remove_due_to_license_issue P00363 21098488 702 MQTFQADLAIVGAGGAGLRAAIAAAQANPNAKIALISKVYPMRSHTVAAEGGSAAVAQDHDSFEYHFHDTVAGGDWLCEQDVVDYFVHHCPTEMTQLELWGCPWSRRPDGSVNVRRFGGMKIERTWFAADKTGFHMLHTLFQTSLQFPQIQRFDEHFVLDILVDDGHVRGLVAMNMMEGTLVQIRANAVVMATGGAGRVYRYNTNGGIVTGDGMGMALSHGVPLRDMEFVQYHPTGLPGSGILMTEGCRGEGGILVNKNGYRYLQDYGMGPETPLGEPKNKYMELGPRDKVSQAFWHEWRKGNTISTPRGDVVYLDLRHLGEKKLHERLPFICELAKAYVGVDPVKEPIPVRPTAHYTMGGIETDQNCETRIKGLFAVGECSSVGLHGANRLGSNSLAELVVFGRLAGEQATERAATAGNGNEAAIEAQAAGVEQRLKDLVNQDGGENWAKIRDEMGLAMEEGCGIYRTPELMQKTIDKLAELQERFKRVRITDTSSVFNTDLLYTIELGHGLNVAECMAHSAMARKESRGAHQRLDEGCTERDDVNFLKHTLAFRDADGTTRLEYSDVKITTLPPA 3p4r A 3.05 BS02 GUA A 1 G50 H232 T244 E245 R390 G392 S393 G51 H233 T245 E246 R391 G393 S394 A47 F116 T203 Q230 H232 L242 E245 R248 R287 H355 Y356 R390 A48 F117 T204 Q231 H233 L243 E246 R249 R288 H356 Y357 R391 1.3.5.1 0000104,0000166,0005515,0005829,0005886,0006113,0006974,0008177,0009055,0009061,0016020,0016491,0016627,0019645,0022900,0044780,0045283,0050660,0071949 remove_due_to_license_issue P00363 21098488 577 MQTFQADLAIVGAGGAGLRAAIAAAQANPNAKIALISKVYPMRSHTVAAEGGSAAVAQDHDSFEYHFHDTVAGGDWLCEQDVVDYFVHHCPTEMTQLELWGCPWSRRPDGSVNVRRFGGMKIERTWFAADKTGFHMLHTLFQTSLQFPQIQRFDEHFVLDILVDDGHVRGLVAMNMMEGTLVQIRANAVVMATGGAGRVYRYNTNGGIVTGDGMGMALSHGVPLRDMEFVQYHPTGLPGSGILMTEGCRGEGGILVNKNGYRYLQDYGMGPETPLGEPKNKYMELGPRDKVSQAFWHEWRKGNTISTPRGDVVYLDLRHLGEKKLHERLPFICELAKAYVGVDPVKEPIPVRPTAHYTMGGIETDQNCETRIKGLFAVGECSSVGLHGANRLGSNSLAELVVFGRLAGEQATERAATAGNGNEAAIEAQAAGVEQRLKDLVNQDGGENWAKIRDEMGLAMEEGCGIYRTPELMQKTIDKLAELQERFKRVRITDTSSVFNTDLLYTIELGHGLNVAECMAHSAMARKESRGAHQRLDEGCTERDDVNFLKHTLAFRDADGTTRLEYSDVKITTLPPA 3p4v A 2.0 BS02 PMX A 1 F130 L197 W208 F127 L194 W205 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8uM remove_due_to_license_issue Ki=8000nM P00918 21332115 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p4w A 3.2 BS01 DSF A 1 P120 I202 T255 I258 P116 I198 T251 I254 ? 0004888,0005216,0005230,0005267,0005272,0005886,0006811,0006814,0016020,0034220,0035725,0042802,0071805,1902495 remove_due_to_license_issue Q7NDN8 21248852 319 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 3p4w B 3.2 BS01 DSF B 1 P120 I201 T255 I258 P116 I197 T251 I254 ? 0004888,0005216,0005230,0005267,0005272,0005886,0006811,0006814,0016020,0034220,0035725,0042802,0071805,1902495 remove_due_to_license_issue Q7NDN8 21248852 319 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 3p50 A 3.3 BS01 PFL A 1 I202 L206 Y254 T255 I258 N307 I198 L202 Y250 T251 I254 N303 ? 0004888,0005216,0005230,0005267,0005272,0005886,0006811,0006814,0016020,0034220,0035725,0042802,0071805,1902495 remove_due_to_license_issue Q7NDN8 21248852 319 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 3p55 A 2.0 BS01 670 A 1 H94 H119 F130 V134 L197 T198 T199 H91 H116 F127 V131 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22258283 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p58 A 1.49 BS02 P58 A 1 N62 H64 N67 Q92 H94 V143 T199 T200 N59 H61 N64 Q89 H91 V139 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=25.4nM remove_due_to_license_issue P00918 22218610 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p5k A 2.09 BS01 P5K A 1 A51 K53 E71 L75 M78 I84 L104 T106 H148 D168 F169 G170 A44 K46 E64 L68 M71 I77 L97 T99 H141 D161 F162 G163 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=0.076uM remove_due_to_license_issue P47811 22014550 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3p5l A 1.498 BS02 IT5 A 1 Q92 H94 H96 F131 L198 T199 T200 P202 Q89 H91 H93 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=40.8nM remove_due_to_license_issue P00918 22218610 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3p5o A 1.6 BS01 EAM A 1 W81 P82 F83 L92 L94 N140 I146 M149 W40 P41 F42 L51 L53 N99 I105 M108 ? Kd=55.2nM remove_due_to_license_issue IC50=190nM, Ki=50nM, Kd=99nM O60885 21068722 1 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 3p76 A 1.93 BS01 P76 A 1 I18 E73 T179 F180 I186 I189 G198 T203 H226 K227 D230 H253 I17 E72 T178 F179 I185 I188 G197 T202 H225 K226 D229 H252 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue O67648 21273067 273 GLEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFAFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQK 3p78 A 2.3 BS01 P78 A 1 A51 K53 E71 L75 I84 L104 T106 H148 L167 D168 F169 A44 K46 E64 L68 I77 L97 T99 H141 L160 D161 F162 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=0.11uM remove_due_to_license_issue P47811 22014550 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3p79 A 2.1 BS01 P79 A 1 A51 K53 R67 R70 E71 L74 M78 I84 L104 T106 H148 L167 D168 A44 K46 R60 R63 E64 L67 M71 I77 L97 T99 H141 L160 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=2.3uM remove_due_to_license_issue P47811 22014550 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3p7a A 2.31 BS01 P7A A 1 A51 K53 R67 E71 I84 L104 T106 L167 D168 F169 A44 K46 R60 E64 I77 L97 T99 L160 D161 F162 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=0.52uM remove_due_to_license_issue P47811 22014550 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3p7b A 1.9 BS01 P7B A 1 K53 R67 R70 E71 L74 L75 M78 I84 L104 T106 L167 D168 F169 K46 R60 R63 E64 L67 L68 M71 I77 L97 T99 L160 D161 F162 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=0.018uM remove_due_to_license_issue P47811 22014550 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3p7c A 2.3 BS01 P7C A 1 A51 K53 R70 E71 M78 I84 L104 H148 L167 D168 A44 K46 R63 E64 M71 I77 L97 H141 L160 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 ic50=0.022uM remove_due_to_license_issue P47811 22014550 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3p7i A 1.71 BS01 P7I A 1 Y47 G65 Y93 S127 T128 S129 H157 D205 Y43 G61 Y89 S123 T124 S125 H153 D201 ? 0015716,0030313,0043190,0055085 Kd=19.9nM remove_due_to_license_issue Q1R3F7 22019591 313 KALNFGIISTESQQNLKPQWTPFLQDMEKKLGVKVNAFFAPDYAGIIQGMRFNKVDIAWYGNLSAMEAVDRANGQVFAQTVAADGSPGYWSVLIVNKDSPINNLNDLLAKRKDLTFGNGDPNSTSGFLVPGYYVFAKNNISASDFKRTVNAGHETNALAVANKQVDVATNNTENLDKLKTSAPEKLKELKVIWKSPLIPGDPIVWRKNLSETTKDKIYDFFMNYGKTPEEKAVLERLGWAPFRASSDLQLVPIRQLALFKEMQSVKDNKGLNEQDKLAKTTAIQAQLDDLDRLNNALSAM 3p8e A 2.4946 BS01 LN7 A 1 L30 D73 F76 D79 R98 G129 R145 H173 V268 D269 C274 L22 D63 F66 D69 R88 G119 R135 H163 V258 D259 C264 3.5.3.18 0000052,0003073,0003824,0005829,0006525,0006527,0007263,0008285,0016403,0016597,0016787,0043116,0045429,0045766,0046209,0046872,0070062,1900038 remove_due_to_license_issue O94760 20979083 286 AFGRATHAVVRALPESLGQHALRSGEEVDVARAERQHQLYVGVLGSKLGLQVVELPADESLPDCVFVEDVAVVCEETALITRPGAPSRRKEVDMMKEALEKLQLNIVEMKDENATLDGGDVLFTGREFFVGLSKRTNQRGAEILADTFKDYAVSTVPVADGLHLKSFCSMAGPNLIAIGSSESAQKALKIMQQMSDHRYDKLTVPDDIAANCIYLNIPNKGHVLLHRTPEEYPESAKVYEKLKDHMLIPVSMSELEKVDGLLTCCSVLINKK 3p8h A 2.55 BS01 P8H A 1 D355 N358 L361 C363 F379 W382 Y386 D150 N153 L156 C158 F174 W177 Y181 ? 0005634,0006355 remove_due_to_license_issue IC50=21000nM Q9Y468 21417280 600 WSWESYLEEQKAITAPVSLFQDSQAVTHNKNGFKLGMKLEGIDPQHPSMYFILTVAEVCGYRLRLHFDGYSECHDFWVNANSPDIHPAGWFEKTGHKLQPPKGYKEEEFSWSQYLRSTRAQAAPKHLFVSQSHSPPPLGFQVGMKLEAVDRMNPSLVCVASVTDVVDSRFLVHFDNWDDTYDYWCDPSSPYIHPVGWCQKQGKPLTPPQDYPDPDNFCWEKYLEETGASAVPTWAFKVRPPHSFLVNMKLEAVDRRNPALIRVASVEDVEDHRIKIHFDGWSHGYDFWIDADHPDIHPAGWCSKTGHPLQPPL 3p8n A 1.9 BS02 L4T A 1 Y56 H57 V78 D79 D81 R123 L135 K136 S139 F154 R155 A156 A157 V158 D168 Y56 H57 V78 D79 D81 R123 L135 K136 S139 F154 R155 A156 A157 V158 D168 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=0.53nM remove_due_to_license_issue P26662 21270126 188 APITAYSQQTRGLLGCIITSLTGRDKNQVDGEVQVLSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWPAPPGARSMTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHVVGIFRAAVCTRGVAKAVDFIPVESMETTMRAS 3p8o A 2.3 BS02 L5T A 1 H57 V78 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 V158 C159 H57 V78 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 V158 C159 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=1.89nM remove_due_to_license_issue P26662 21270126 188 APITAYSQQTRGLLGCIITSLTGRDKNQVDGEVQVLSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWPAPPGARSMTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHVVGIFRAAVCTRGVAKAVDFIPVESMETTMRAS 3p8p A 2.5 BS01 LN6 A 1 L30 D73 F76 D79 R98 R145 H173 K175 V268 D269 S274 L23 D66 F69 D72 R91 R138 H166 K168 V261 D262 S267 3.5.3.18 0000052,0003073,0003824,0005829,0006525,0006527,0007263,0008285,0016403,0016597,0016787,0043116,0045429,0045766,0046209,0046872,0070062,1900038 Kd=28uM remove_due_to_license_issue O94760 20979083 286 AAFGRATHAVVRALPESLGQHALRSAKGEEVDVARAERQHQLYVGVLGSKLGLQVVELPADESLPDCVFVEDVAVVCEETALITRPGAPSRRKEVDMMKEALEKLQLNIVEMKDENATLDGGDVLFTGREFFVGLSKRTNQRGAEILADTFKDYAVSTVPVADGLHLKSFCSMAGPNLIAIGSSESAQKALKIMQQMSDHRYDKLTVPDDIAANCIYLNIPNKGHVLLHRTPEEYPESAKVYEKLKDHMLIPVSMSELEKVDGLLTSCSVLINKK 3p8z A 1.7 BS01 36A A 1 S56 G58 G81 G86 W87 T104 K105 H110 K130 D131 V132 D146 I147 R163 M167 S51 G53 G76 G81 W82 T99 K100 H105 K125 D126 V127 D141 I142 R158 M162 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P27915 21147775 263 GETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 3p9j A 2.8 BS01 P9J A 1 L139 G140 A160 Y212 A213 P214 G216 L263 L14 G15 A35 Y87 A88 P89 G91 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 21128645 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVGTLDYLPPEMIEGDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3p9t A 2.02 BS01 TCL A 1 H67 F70 M93 L114 G132 F133 A136 M140 H167 V170 H62 F65 M88 L109 G127 F128 A131 M135 H162 V165 ? 0000976,0003677,0003700,0006355,0045892 Kd=0.63uM remove_due_to_license_issue Q8KLP4 21738470 221 KEDTQATREGILDAAEACFHEHGVARTTLEMIGARAGYTRGAVYWHFKNKSEVLAAIVERVHLPFMQELERTSTDQRDTPVHDLRAVMIHSFIELSEDERLRKTMEIMLRSDASANTRVLTEMQQAGFRDALDRMERALRRARDLGQLREGADPKIAARMLHATVLGVLHGAMVEPELMDLKRDGMLALDMTLAAYVKDGVFVPGTVPEPLPE 3p9t A 2.02 BS02 TCL A 2 H67 F70 L100 M113 H62 F65 L95 M108 ? 0000976,0003677,0003700,0006355,0045892 Kd=0.63uM remove_due_to_license_issue Q8KLP4 21738470 222 KEDTQATREGILDAAEACFHEHGVARTTLEMIGARAGYTRGAVYWHFKNKSEVLAAIVERVHLPFMQELERTSTDQRDTPVHDLRAVMIHSFIELSEDERLRKTMEIMLRSDASANTRVLTEMQQAGFRDALDRMERALRRARDLGQLREGADPKIAARMLHATVLGVLHGAMVEPELMDLKRDGMLALDMTLAAYVKDGVFVPGTVPEPLPE 3pa3 A 1.4 BS01 C70 A 1 L15 A36 E85 Y86 C87 G90 E134 N135 L137 D148 K271 L11 A32 E73 Y74 C75 G78 E122 N123 L125 D136 K259 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1nM O14757 21074424 1 FVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3pa4 A 1.59 BS01 C72 A 1 L15 E17 A36 E85 Y86 C87 G90 E134 N135 L137 D148 K271 L10 E12 A30 E71 Y72 C73 G76 E120 N121 L123 D134 K257 D130 K132 E134 N135 D148 T170 D116 K118 E120 N121 D134 T156 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=3nM O14757 21074424 1 VEDWDLVQTLGEGAGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3pa5 A 1.7 BS01 C73 A 1 L15 E17 A36 E85 Y86 C87 G90 E134 N135 L137 D148 K271 L13 E15 A32 E69 Y70 C71 G74 E118 N119 L121 D132 K255 D130 K132 E134 N135 D148 T170 D114 K116 E118 N119 D132 T154 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=2nM remove_due_to_license_issue IC50=10nM O14757 21074424 1 VPFVEDWDLVQTLGEGGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3pa8 A 2.0 BS01 621 A 1 I46 H110 C155 V201 R202 I40 H104 C149 V195 R196 2.4.1.- remove_due_to_license_issue Q189K3 21095570 300 DFSQNIVVDKEYLLEKISSLARSSERGYIHYIVQLQGDKISYEAACNLFAKTPYDSVLFQKNIEDSEIAYYYNPGDGEIQEIDKYKIPSIISDRPKIKLTFIGHGKDEFNTDIFAGFDVDSLSTEIEAAIDLAKEDISPKSIEINLLGCNMFSYSINVEETYPGKLLLKVKDKISELMPSISQDSIIVSANQYEVRINSEGRRELLDHSGEWINKEESIIKDISSKEYISFNPKENKITVKSKNL 3pax A 2.4 BS01 3MB A 1 H862 G863 Y896 F897 K903 S904 Y907 E988 H201 G202 Y235 F236 K242 S243 Y246 E327 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 ic50=10uM remove_due_to_license_issue P26446 9521710 1 KSKLAKPIQDLIKMIFDVESMKKAMVEFEIDLQKMPLGKLSKRQIQSAYSILNEVQQAVSDGGSESQILDLSNRFYTLIPHDFGMKKPPLLSNLEYIQAKVQMLDNLLDIEVAYSLLRGGNEDGDKDPIDINYEKLRTDIKVVDKDSEEAKIIKQYVKNTHAATHNAYDLKVVEIFRIEREGESQRYKPFKQLHNRQLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQADPIGLILLGEVALGNMYELKNASHITKLPKGKHSVKGLGKTAPDPTATTTLDGVEVPLGNGISTGINDTCLLYNEYIVYDVAQVNLKYLLKLKFNYKT 3pb3 A 1.9 BS01 SAH A 1 G32 T33 N38 D55 P56 A86 A87 E88 L104 F105 W107 T109 L110 S195 W197 G31 T32 N37 D54 P55 A85 A86 E87 L103 F104 W106 T108 L109 S178 W180 2.1.1.180 0008168,0032259,0046677 remove_due_to_license_issue A8C927 21062819 6732 LILKGTKTVDLSKDELTEIIGQFDRVHIDMGTGDGRNIYKLAINDQNTFYIGIDPVKENLFDISKKIIKKPSKGGLSNVVFVIAAAESMPFELKNIADSISILFPWGTLLEYVIKPNRDILSNVADMAKKEAHFEFVTTYSDKAYFLSEQYKAELSNSGFRIDDVKELDNEYVKQFNSMWAKRLAFGRKRSFFRVSGHV 3pb7 X 1.4 BS01 PBD X 1 D186 E225 E226 W231 D269 V324 E325 F346 W350 H351 D113 E152 E153 W158 D196 V251 E252 F273 W277 H278 2.3.2.5 0016603 Ki=1.817uM remove_due_to_license_issue Q9NXS2 21288892 390 GSLPEARLRRVVGQLDPQRLWSTYLRPLLVVRTPGSPGNLQVRKFLEATLRSLTAGWHVELDPFTASTPLGPVDFGNVVATLDPRAARHLTLACHYDSKLFPPGSTPFVGATDSAVPCALLLELAQALDLELSRAKKQAAPVTLQLLFLDGEEALKEWGPKDSLYGSRHLAQLMESIPHSPGPTRIQAIELFMLLDLLGAPNPTFYSHFPRTVRWFHRLRSIEKRLHRLNLLQSHPQEVMYFQPGEPFGSVEDDHIPFLRRGVPVLHLISTPFPAVWHTPADTEVNLHPPTVHNLCRILAVFLAEYLGL 3pb8 X 1.13 BS01 AHN X 1 D186 D269 E325 H351 D117 D200 E256 H282 2.3.2.5 0016603 Ki=5.748uM remove_due_to_license_issue Q9NXS2 21288892 390 VPLIGSLPEARLRRVVGQLDPQRLWSTYLRPLLVVRTPGSPGNLQVRKFLEATLRSLTAGWHVELDPFTASTPLGPVDFGNVVATLDPRAARHLTLACHYDSKLFPPGSTPFVGATDSAVPCALLLELAQALDLELSRAKKQAAPVTLQLLFLDGEEALKEWGPKDSLYGSRHLAQLMESIPHSPGPTRIQAIELFMLLDLLGAPNPTFYSHFPRTVRWFHRLRSIEKRLHRLNLLQSHPQEVMYFQPGEPFGSVEDDHIPFLRRGVPVLHLISTPFPAVWHTPADTEVNLHPPTVHNLCRILAVFLAEYLGL 3pb9 X 1.12 BS01 1BN X 1 D186 E225 E226 W231 D269 E325 F346 W350 H351 D113 E152 E153 W158 D196 E252 F273 W277 H278 2.3.2.5 0016603 Ki=0.262uM remove_due_to_license_issue Q9NXS2 21288892 390 GSLPEARLRRVVGQLDPQRLWSTYLRPLLVVRTPGSPGNLQVRKFLEATLRSLTAGWHVELDPFTASTPLGPVDFGNVVATLDPRAARHLTLACHYDSKLFPPGSTPFVGATDSAVPCALLLELAQALDLELSRAKKQAAPVTLQLLFLDGEEALKEWGPKDSLYGSRHLAQLMESIPHSPGPTRIQAIELFMLLDLLGAPNPTFYSHFPRTVRWFHRLRSIEKRLHRLNLLQSHPQEVMYFQPGEPFGSVEDDHIPFLRRGVPVLHLISTPFPAVWHTPADTEVNLHPPTVHNLCRILAVFLAEYLGL 3pbb A 1.95 BS01 PBD A 1 E201 E202 W207 D248 Q304 F325 H330 E163 E164 W169 D210 Q266 F287 H292 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Ki=0.095uM remove_due_to_license_issue Ki=60nM, IC50=5300nM Q16769 21288892 380 ASAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPYGYRSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 3pcb M 2.19 BS02 3HB M 1 Y324 Y447 W449 R457 I491 Y24 Y144 W146 R154 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=4mM remove_due_to_license_issue P00437 9254599 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pce M 2.06 BS02 3HP M 1 Y408 Y447 W449 R457 H462 I491 Y105 Y144 W146 R154 H159 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=10mM remove_due_to_license_issue P00437 9254599 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pce P 2.06 BS02 3HP P 1 Y408 Y447 W449 R457 H462 I491 Y105 Y144 W146 R154 H159 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=10mM remove_due_to_license_issue P00437 9254599 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pcf A 2.15 BS01 FHB M 1 G14 P15 G14 P15 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 9254599 550 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 3pcf B 2.15 BS01 FHB N 1 G14 P15 G14 P15 Y79 V114 Y79 V114 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 9254599 550 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 3pcf M 2.15 BS02 FHB M 1 Y324 Y447 W449 R457 H460 H462 I491 Y24 Y144 W146 R154 H157 H159 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=0.9uM remove_due_to_license_issue P00437 9254599 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pcf M 2.15 BS03 FHB N 2 P322 I328 P22 I28 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=0.9uM remove_due_to_license_issue P00437 9254599 551 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pcg M 1.96 BS02 4HP M 1 Y324 Y408 Y447 W449 R457 H462 I491 Y24 Y105 Y144 W146 R154 H159 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=5mM remove_due_to_license_issue P00437 9254599 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pch A 2.05 BS01 CHB M 1 G14 P15 R133 G14 P15 R133 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 9254599 550 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 3pch B 2.05 BS01 CHB N 1 G14 P15 G14 P15 Y79 V114 Y79 V114 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 9254599 550 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 3pch M 2.05 BS02 CHB M 1 Y324 Y447 W449 R457 H460 H462 Q477 I491 Y24 Y144 W146 R154 H157 H159 Q174 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Ki=4uM remove_due_to_license_issue P00437 9254599 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pcj M 2.13 BS02 INO M 1 Y324 Y447 W449 R457 H460 H462 Y24 Y144 W146 R154 H157 H159 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Kd=0.06uM remove_due_to_license_issue P00437 9254600 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pck M 2.13 BS02 NNO M 1 Y324 Y408 W449 R457 H460 H462 I491 Y24 Y105 W146 R154 H157 H159 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Kd=0.2uM remove_due_to_license_issue P00437 9254600 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pcn A 2.4 BS01 DHY M 1 P15 Y16 P15 Y16 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 9298971 550 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 3pcn M 2.4 BS02 DHY M 1 Y324 Y408 Y447 W449 R457 H460 H462 I491 Y24 Y105 Y144 W146 R154 H157 H159 I188 Y408 Y447 R457 H460 H462 Y105 Y144 R154 H157 H159 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0019619,0042952,0046872,0051213 Kd=220uM remove_due_to_license_issue P00437 9298971 550 PAQDNSRFVIRDRNWHPKALTPDYKTSIARSPRQALVSIPQSISETTGPNFSHLGFGAHDHDLLLNFGLPIGERIIVAGRVVDQYGKPVPNTLVEMWQANAGGRYRHKNDRYLAPLDPNFGGVGRCLTDSDGYYSFRTIKPGPYPWRNGPNDWRPAHIHFGISGPSIATKLITQLYFEGDPLIPMCPIVKSIANPEAVQQLIAKLDMNNANPMDCLAYRFDIVLRGQRKTHFE 3pcu A 2.0 BS02 LX8 A 1 I268 A271 A272 Q275 L309 F313 R316 L326 A327 V342 I345 C432 H435 L436 F439 I21 A24 A25 Q28 L62 F66 R69 L79 A80 V95 I98 C185 H188 L189 F192 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 22384078 1 DMPVERILEAELAVEDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 3pd2 A 1.86 BS01 A3S A 1 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 6.1.1.3 0004829,0005524,0005737,0008270 Kd=3.4uM remove_due_to_license_issue Q9UZ14 21098258 500 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYKAFKISCKGHPLAELSRTIVPEEARVE 3pd2 B 1.86 BS01 A3S B 1 V45 F81 A82 A94 F117 G118 Y119 K121 V45 F81 A82 A94 F117 G118 Y119 K121 6.1.1.3 0004829,0005524,0005737,0008270 Kd=3.4uM remove_due_to_license_issue Q9UZ14 21098258 501 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYKAFKISCKGHPLAELSRTIVPEE 3pd3 A 1.86 BS01 A3T A 1 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 K121 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 K121 6.1.1.3 0004829,0005524,0005737,0008270 Kd=36.2uM remove_due_to_license_issue Q9UZ14 21098258 148 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYKAFKISCKGHPLAELSRTIVPEEAR 3pd3 B 1.86 BS01 A3T B 1 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 K121 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 K121 6.1.1.3 0004829,0005524,0005737,0008270 Kd=36.2uM remove_due_to_license_issue Q9UZ14 21098258 148 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYKAFKISCKGHPLAELSRTIVPEE 3pd4 A 2.4 BS01 A3G A 1 A19 V45 F81 A82 L88 A94 F117 G118 Y119 A19 V45 F81 A82 L88 A94 F117 G118 Y119 6.1.1.3 0004829,0005524,0005737,0008270 Kd=33.3uM remove_due_to_license_issue Q9UZ14 21098258 500 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYKAFKISCKGHPLAELSRTIVPEEARV 3pd4 B 2.4 BS01 A3G B 1 A19 L20 V45 F81 F117 G118 Y119 A19 L20 V45 F81 F117 G118 Y119 6.1.1.3 0004829,0005524,0005737,0008270 Kd=33.3uM remove_due_to_license_issue Q9UZ14 21098258 501 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYKAFKISCKGHPLAELSRTIVPEE 3pd8 A 2.476 BS02 HA7 A 1 Y58 P86 L87 T88 R93 L135 G138 S139 T140 E190 M193 Y58 P86 L87 T88 R93 L135 G138 S139 T140 E190 M193 ? 0015276,0016020 Ki=108nM remove_due_to_license_issue P19491 21067182 261 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 3pd9 A 2.1 BS01 HA5 A 1 Y58 P86 L87 T88 R93 G138 S139 T140 E190 M193 Y58 P86 L87 T88 R93 G138 S139 T140 E190 M193 ? 0015276,0016020 Ki=494nM remove_due_to_license_issue P19491 21067182 260 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3pdc A 2.6 BS01 ZYI A 1 F265 D333 M337 T358 Y381 Y465 H523 W524 F42 D110 M114 T135 Y158 Y241 H299 W300 F265 H332 D333 W334 N357 N376 Y381 Y465 D495 H523 F42 H109 D110 W111 N134 N153 Y158 Y241 D271 H299 3.1.3.76,3.3.2.10 0003824 remove_due_to_license_issue P34913 21302953 1 APLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 3pdq A 1.989 BS02 KC6 A 1 Y132 D135 Y177 F185 H188 E190 K206 W208 K241 H276 Y130 D133 Y175 F183 H186 E188 K204 W206 K239 H274 G170 Y177 H188 E190 H276 S288 G168 Y175 H186 E188 H274 S286 1.14.11.66,1.14.11.69 ic50=0.18uM remove_due_to_license_issue O75164 21412984 503 SESETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 3pe1 A 1.6 BS01 3NG A 1 L45 G46 V53 V66 K68 F113 V116 H160 M163 I174 D175 L43 G44 V51 V64 K66 F111 V114 H158 M161 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.223nM remove_due_to_license_issue IC50=2000nM, Kd=0.562341nM, Ki=0.380000nM P68400 21870818 338 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 3pe2 A 1.9 BS01 E1B A 1 L45 G46 R47 V53 V66 K68 F113 H115 V116 I174 D175 L43 G44 R45 V51 V64 K66 F111 H113 V114 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.175nM remove_due_to_license_issue IC50=6nM, Ki=420nM P68400 21870818 338 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 3peq A 2.4 BS01 3EQ A 1 V281 F282 C285 T289 H323 L330 V341 V348 I363 I364 K367 F368 H449 M453 L469 Y473 V61 F62 C65 T69 H103 L110 V121 V128 I143 I144 K147 F148 H229 M233 L249 Y253 ? 0003677,0004879,0005634,0006355 ic50=31.6nM remove_due_to_license_issue Q03181 21414782 1 ADLKAFSKHIYNAYLKNFNMTKKKARSILTAPFVIHDIETLWQAEKGLVWLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKD 3pf4 B 1.38 BS01 rna R 0 K7 W8 N10 F15 F17 D25 F27 H29 K7 W8 N10 F15 F17 D25 F27 H29 ? 0003676,0003677,0005737,0009295,0010468 remove_due_to_license_issue P32081 22128343 1 ~ 5 MLEGKVKWFNSEKGFGFIEVEGQDDVFVHFSAIQGEGFKTLEEGQAVSFEIVEGNRGPQAANVTKE 3pf5 A 1.68 BS01 rna S 0 W8 F17 D25 W8 F17 D25 ? 0003676,0003677,0005737,0009295,0010468 remove_due_to_license_issue P32081 22128343 1 MLEGKVKWFNSEKGFGFIEVEGQDDVFVHFSAIQGEGFKTLEEGQAVSFEIVEGNRGPQAANVTKE 3pf5 B 1.68 BS01 rna R 0 W8 N10 F15 F17 D25 F27 H29 W8 N10 F15 F17 D25 F27 H29 ? 0003676,0003677,0005737,0009295,0010468 remove_due_to_license_issue P32081 22128343 1 ~ 5 MLEGKVKWFNSEKGFGFIEVEGQDDVFVHFSAIQGEGFKTLEEGQAVSFEIVEGNRGPQAANVTKEA 3pfp B 2.35 BS02 036 B 1 R126 K133 P134 R135 S136 G282 E283 R284 K306 R337 H369 K380 R128 K135 P136 R137 S138 G284 E285 R286 K308 R339 H371 K382 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 remove_due_to_license_issue O53512 21454647 463 GAMNWTVDIPIDQLPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 3pgl A 2.35 BS02 RZX A 1 F106 Y158 R178 F30 Y82 R102 3.1.3.16 0008420,0016791 Ki=5uM remove_due_to_license_issue Q9GZU7 21348431 257 QYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEIDGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRESCVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPFFEQLSRVDDVYSVLRQ 3phe A 2.2 BS01 C9A A 1 L419 R422 M423 H475 S476 Y477 P479 I482 A486 L489 P496 L497 W528 L414 R417 M418 H470 S471 Y472 P474 I477 A481 L484 P491 L492 W523 2.7.7.48,3.6.4.13 0000166,0001172,0003689,0003723,0003968,0004386,0006338,0006508,0008236,0016020,0016887,0034062,0039694,0061775,0140584,0140588,0140665,0140849 ic50=0.016uM remove_due_to_license_issue D0PY27 21145235 999 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3pi5 A 2.4 BS01 3P5 A 1 D32 G34 S35 Y71 T72 Q73 F108 I110 Y198 D228 G230 D35 G37 S38 Y74 T75 Q76 F111 I113 Y190 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.95uM remove_due_to_license_issue IC50=950nM P56817 21388807 387 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3pih A 2.9 BS01 dna D 0 G670 S675 T679 Y680 R688 S705 S708 N710 L711 G590 S595 T599 Y600 R608 S625 S628 N630 L631 ? 0003677,0003824,0004518,0005524,0005737,0006281,0006289,0008270,0009380,0009381,0009432,0016887,0046872 remove_due_to_license_issue Q9WYV0 21240268 1 ~ 32 NEIVVKGARVHNLKNITVRIPKNRLVVITGVSGSGKSSLAMDTIYAEGQRRYLESLSTYKKPDVDEIEGLSPAIAIDQKTSHNPRSTVGTVTEIYDYLRVLYARIGKAHCPECGRPLEKKSIDEILQDLFNSFKEGSRIYILAPLVVDRLILETRNEHRILDSLELAMREGKGFVEIRNVDTGESKIFSENLMCPVCGIGFPEITPKLFSFNSPYGACPNCHGLGFTFEVDPSLVAIIPYRWDRRLSRWVAREIEKRGVSPPEDVKEFILYGDFEGVVPKVQRWHRETEMKEWLEKNFIVQRTCSVCGGRRLNREALSVKINGLNIHEFTELSISEELEFLKNLNLTEREREIVGELLKEIEKRLEFLVDVGLEYLTLSRSATTLSGGESQRIRLATQIGSGLTGVIYVLDEPTIGLHPRDTERLIKTLKKLRDLGNTVIVVEHDEEVIRNADHIIDIGPGGGTNGGRVVFQGTVDELLKNPDSSLTGEYLSGKRKITVNKTRRLPYASLKIKGVRHNNLKNIDVEIPLGVFVCVTGVSGSGKSSLVMETLYPALMNLLHKTKLPAGEFDSIEGHENIDKMIAIDQSPIGRTPRSNPATYTKVFDEIRSLFAMTPAAKARGYNKSRFSFNLKGGRCEACQGQGYVKIEMLFLPDVYVECDVCKGKRYNRETLEITYKGKNISDILDMTVDEALEFFKNIPSIKRTLQVLHDVGLGYVKLGQPATTLSGGEAQRIKLASELRKRDTGRTLYILDEPTVGLHFEDVRKLVEVLHRLVDRGNTVIVIEHNLDVIKNADHIIDLGPEGGKEGGYIVATGTPEEIAKNPHSYTGRFLKNVL 3pix A 1.85 BS01 027 A 1 A428 Y476 M477 A478 G480 L528 A38 Y86 M87 A88 G90 L138 D521 A523 R525 N526 D539 F559 D131 A133 R135 N136 D149 F169 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.1uM remove_due_to_license_issue Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 3piy A 2.55 BS01 585 A 1 V416 A428 M477 G480 L528 L542 V546 V26 A38 M81 G84 L132 L146 V150 D521 A523 R525 N526 D539 F559 D125 A127 R129 N130 D143 F163 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=190nM Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 3piz A 2.21 BS01 03C A 1 L408 A428 K430 E445 T474 Y476 M477 G480 L528 L18 A35 K37 E47 T76 Y78 M79 G82 L130 D521 A523 R525 N526 D539 F559 D123 A125 R127 N128 D141 F145 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3.5uM remove_due_to_license_issue Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGVVKYGKWRGQYDVAIKMISEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 3pj1 A 2.0 BS01 LHL A 1 L408 V416 A428 I429 K430 E445 I472 T474 M477 G480 L528 L18 V23 A35 I36 K37 E47 I72 T74 M77 G80 L126 D521 A523 R525 N526 D539 F559 D119 A121 R123 N124 D137 F141 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.048uM remove_due_to_license_issue Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGVVKYGKWRGQYDVAIKMISEDEFIEEAKVMMNLSHEKLVQLYGVCTKQIFIITEYMANGCLLNYLREMRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 3pj1 A 2.0 BS02 LHL A 2 Y425 Q459 Y461 Y32 Q61 Y63 D521 A523 R525 N526 D539 F559 D119 A121 R123 N124 D137 F141 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.048uM remove_due_to_license_issue Q06187 21280133 2 GYGSWEIDPKDLTFLKELGTGVVKYGKWRGQYDVAIKMISEDEFIEEAKVMMNLSHEKLVQLYGVCTKQIFIITEYMANGCLLNYLREMRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 3pj2 A 1.75 BS01 04K A 1 E407 L408 V416 A428 M449 M477 G480 L528 D539 E17 L18 V23 A35 M56 M84 G87 L135 D146 D521 A523 R525 N526 D539 F559 D128 A130 R132 N133 D146 F148 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7.2uM remove_due_to_license_issue Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 3pj3 A 1.85 BS01 04L A 1 A428 K430 E445 M449 T474 Y476 M477 G480 F517 L528 S538 D539 A35 K37 E45 M49 T74 Y76 M77 G80 F117 L128 S138 D139 D521 A523 R525 N526 D539 F559 D121 A123 R125 N126 D139 F140 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5.6uM remove_due_to_license_issue Q06187 21280133 1 GYGSWEIDPKDLTFLKELGTGVVKYGKWRGQYDVAIKMIDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 3pj8 A 1.96 BS01 404 A 1 I10 A31 F80 F82 L83 L134 I11 A32 F78 F80 L81 L132 D127 K129 Q131 N132 D145 T165 D125 K127 Q129 N130 D143 T155 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 21417417 299 GMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pjc A 2.2 BS01 PJC A 1 L828 F833 V836 A853 V884 M902 E903 Y904 R953 L956 D967 L14 F19 V22 A39 V70 M84 E85 Y86 R135 L138 D149 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 ic50=27nM remove_due_to_license_issue IC50=27nM P52333 21155605 800 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGCERDVPALCRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSRG 3pjg A 2.7 BS01 UGA A 1 F142 L143 R144 K197 N201 V208 Y242 N244 S246 Y249 G250 Y252 M306 D388 F143 L144 R145 K198 N202 V209 Y243 N245 S247 Y250 G251 Y253 M307 D389 T118 E145 K197 N201 C253 D257 T119 E146 K198 N202 C254 D258 1.1.1.22 0000166,0000271,0003979,0006065,0016491,0016616,0051287 remove_due_to_license_issue A0A0J9WZA6 21536136 901 FMKITISGTGYVGLSNGVLIAQNHEVVALDIVQAKVDMLNQKISPIVDKEIQEYLAEKPLNFRATTDKHDAYRNADYVIIATPTDYDPKTNYFNTSTVEAVIRDVTEINPNAVMIIKSTIPVGFTRDIKERLGIDNVIFSPEFLREGRALYDNLHPSRIVIGERSARAERFADLLKEGAIKQDIPTLFTDSTEAEAIKLFANTYLALRVAYFNELDSYAESQGLNSKQIIEGVCLDPRIGNHYNNPSFGYGGYCLPKDTKQLLANYESVPNNIIAAIVDANRTRKDFIADSILARKPKVVGVYRLIMKSGSDNFRASSIQGIMKRIKAKGIPVIIYEPVMQEDEFFNSRVVRDLNAFKQEADVIISNRMAEELADVADKVYTRDLFGND 3pjg A 2.7 BS02 UGA A 2 K256 D257 K284 Q319 G320 K323 K326 F345 K257 D258 K285 Q320 G321 K324 K327 F346 T118 E145 K197 N201 C253 D257 T119 E146 K198 N202 C254 D258 1.1.1.22 0000166,0000271,0003979,0006065,0016491,0016616,0051287 remove_due_to_license_issue A0A0J9WZA6 21536136 902 FMKITISGTGYVGLSNGVLIAQNHEVVALDIVQAKVDMLNQKISPIVDKEIQEYLAEKPLNFRATTDKHDAYRNADYVIIATPTDYDPKTNYFNTSTVEAVIRDVTEINPNAVMIIKSTIPVGFTRDIKERLGIDNVIFSPEFLREGRALYDNLHPSRIVIGERSARAERFADLLKEGAIKQDIPTLFTDSTEAEAIKLFANTYLALRVAYFNELDSYAESQGLNSKQIIEGVCLDPRIGNHYNNPSFGYGGYCLPKDTKQLLANYESVPNNIIAAIVDANRTRKDFIADSILARKPKVVGVYRLIMKSGSDNFRASSIQGIMKRIKAKGIPVIIYEPVMQEDEFFNSRVVRDLNAFKQEADVIISNRMAEELADVADKVYTRDLFGND 3pjt A 2.5154 BS01 C2E A 1 Q431 K446 L448 S449 R450 A461 G462 L465 M481 N499 Q560 R561 R618 E620 G638 Q639 Q23 K38 L40 S41 R42 A53 G54 L57 M73 N91 Q152 R153 R210 E212 G230 Q231 ? 0071111 Kd=13.1uM (21304926) remove_due_to_license_issue Q3KK31 21304926 2256 DHHAWHRLLDQALNQRRFELFFQPVVAAQDTQLVLHYKVLSRLLDEQGQTIPAGRFLPWLERFGWTARLDRLMLERVLEQMAGHEESLALNLSSATLADPQALNKVFEILRAHSNLGARLTLEIGEEQLPEQAVLEQLTRRLRELGFSLSLQRFGGRFSMIGNLARLGLAYLKIDGSYIRAIDQESDKRLFIEAIQRAAHSIDLPLIAERVETEGELSVIREMGLYGVQGQLFGEPKPWG 3pju A 2.4991 BS01 C2E A 1 Q431 K446 L448 S449 R450 A461 G462 L465 M481 N499 Q560 R561 R618 E620 G638 Q639 Q32 K47 L49 S50 R51 A62 G63 L66 M82 N100 Q161 R162 R219 E221 G239 Q240 ? 0071111 Kd=13.1uM remove_due_to_license_issue Q3KK31 21304926 2256 QSLVADVGDDHHAWHRLLDQALNQRRFELFFQPVVAAQDTQLVLHYKVLSRLLDEQGQTIPAGRFLPWLERFGWTARLDRLMLERVLEQMAGHEESLALNLSSATLADPQALNKVFEILRAHSNLGARLTLEIGEEQLPEQAVLEQLTRRLRELGFSLSLQRFGGRFSMIGNLARLGLAYLKIDGSYIRAIDQESDKRLFIEAIQRAAHSIDLPLIAERVETEGELSVIREMGLYGVQGQLFGEPKPWG 3pka A 1.25 BS03 Y02 A 1 Y97 H114 D131 D142 T203 H205 F211 H212 E238 E269 Y96 H113 D130 D141 T202 H204 F210 H211 E237 E268 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=0.54uM remove_due_to_license_issue P9WK19 21465667 288 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3pkb A 1.25 BS01 Y16 A 1 Y97 H114 D131 D142 F202 T203 H205 H212 E238 E269 Y96 H113 D130 D141 F201 T202 H204 H211 E237 E268 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=0.62uM remove_due_to_license_issue P9WK19 21465667 286 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3pkc A 1.47 BS03 Y08 A 1 E35 Y97 H114 D131 D142 T203 H205 F211 H212 E238 E269 E32 Y94 H111 D128 D139 T200 H202 F208 H209 E235 E266 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H111 D128 D139 G201 H202 G205 H209 L212 E235 N239 E266 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=0.96uM remove_due_to_license_issue P9WK19 21465667 288 RTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTC 3pkd A 1.47 BS03 Y10 A 1 Y97 H114 D131 D142 T203 H205 F211 H212 E238 E269 Y94 H111 D128 D139 T200 H202 F208 H209 E235 E266 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H111 D128 D139 G201 H202 G205 H209 L212 E235 N239 E266 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 ic50=0.76uM remove_due_to_license_issue P9WK19 21465667 288 RTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3pke A 1.6 BS01 Y10 A 1 Y97 H114 D131 D142 T203 H205 F211 H212 E238 E269 Y96 H113 D130 D141 T202 H204 F210 H211 E237 E268 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H113 D130 D141 G203 H204 G207 H211 L214 E237 N241 E268 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0050897,0070006 remove_due_to_license_issue P9WK19 21465667 286 PSRTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTCL 3pm1 A 2.8 BS01 ET A 1 W61 S86 Q90 E120 Y123 N157 W59 S84 Q88 E118 Y121 N155 ? 0003677,0003700,0045892 remove_due_to_license_issue P0A0N3 21264225 205 LKDKILGVAKELFIKNGYNATTTGEIVKLSESSKGNLYYHFKTKENLFLEILNIEESKWQEQWKSEQIKAKTNREKFYLYNELSLTTQYYYPLQNAIIEFYTEYYKTNSINEKMNKLENKYIDAYHVIFKEGNLNGEWSINDVNAVSKIAANAVNGIVTFTHEQNINERIKLMNKFSQIFLNGLS 3pn1 A 2.0 BS01 IVH A 1 L82 E114 K116 L117 E174 Y226 V289 K291 P308 L82 E114 K116 L117 E174 Y226 V289 K291 P308 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 Ki=110nM remove_due_to_license_issue P43813 21189350 319 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFPA 3pn3 A 1.3 BS01 PN3 A 1 Y80 V102 P104 R146 Y80 V102 P104 R146 G43 Q48 C91 L92 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 3.5.1.88 0042586 Ki=400nM remove_due_to_license_issue Q9FUZ2 21629676 194 MEIVEYPDPILRAKNKRIDIFDENLKNLVDAMFDVMYKTDGIGLSAPQVGLNVQLMVFNPAGEPGEGKEIVLVNPKIKKYSDKLVPFDEGCLSFPGIYAEVVRPQSVKIDARDITGERFSISLSRLPARIFQHEYDHLEGVLFFDRMTDQVLDSIREELEALEKKYEEKTGLPSPERVEAR 3pn4 A 1.9 BS01 BB2 A 1 G41 I42 G43 Q48 D88 G90 C91 L92 Y98 R129 H133 E134 H137 G41 I42 G43 Q48 D88 G90 C91 L92 Y98 R129 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 G43 Q48 C91 L92 H133 E134 H137 3.5.1.88 0042586 Ki=140nM remove_due_to_license_issue Q9FUZ2 21629676 501 MEIVEYPDPILRAKNKRIDIFDENLKNLVDAMFDVMYKTDGIGLSAPQVGLNVQLMVFNPAGEPGEGKEIVLVNPKIKKYSDKLVPFDEGCLSFPGIYAEVVRPQSVKIDARDITGERFSISLSRLPARIFQHEYDHLEGVLFFDRMTDQVLDSIREELEALEKKYEEKTGLPSPERVEAR 3po1 B 1.65 BS03 MKY C 1 H79 Y83 W86 L132 H43 Y47 W50 L96 H79 D135 H43 D99 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 22726924 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKET 3po1 C 1.65 BS02 MKY C 1 D229 A230 E232 V255 S256 W257 G258 D45 A46 E48 V71 S72 W73 G74 E232 G233 D234 S235 G236 E48 G49 D50 S51 G52 3.4.21.5 0004252,0006508 Kd=95uM remove_due_to_license_issue P00734 22726924 1 GQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 3po6 A 1.47 BS02 DT9 A 1 N67 Q92 H94 H96 F131 L198 T199 T200 N65 Q90 H92 H94 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 21395315 262 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3pov A 2.5 BS01 dna C 0 R248 F249 K250 Y373 R221 F222 K223 Y346 ? 0003677,0004519,0004527,0005515,0030430,0042025,0046872 remove_due_to_license_issue P88925 21421561 2 ~ 20 TPTPADLFSEDYLVDTLDGLTVDDQQAVLASLSFSKFLKHAKVRDWCAQAKIQPSMPALRMAYNYFLFSKVGEFIGSEDVCNFFVDRVFGGVRLLDVASVYAACSQMNAHQRHHICCLVERATSSQSLNPVWDALRDGIISSSKFHWAVKQQKIFSPAFGLRCEEVVKTLLATLLHPDETNCLDYGFMQSPQNGIFGVSLDFAANVKTFDPNCKVYEIKCRFKYTFAKMECDPIYAAYQRLYEAPGKLALKDFFYSISKPAVEYVGLGKLPSESDYLVAYDQEWEACPRKKRKLTPLHNLIRECILHNSTTESDVYVLTDPQDTRGQISIKARFKANLFVNVRHSYFYQVLLQSSIVEEYIGSPKYYIATGFFRKRGYQDPVNCTIGGDALDPHVEIPTLLIVTPVYFPRGAKHRLLHQAANFWSRSAKDTFPYIKWDFSYLSAN 3pov A 2.5 BS02 dna D 0 S299 E300 K317 K318 R319 R370 S272 E273 K290 K291 R292 R343 ? 0003677,0004519,0004527,0005515,0030430,0042025,0046872 remove_due_to_license_issue P88925 21421561 21 ~ 39 TPTPADLFSEDYLVDTLDGLTVDDQQAVLASLSFSKFLKHAKVRDWCAQAKIQPSMPALRMAYNYFLFSKVGEFIGSEDVCNFFVDRVFGGVRLLDVASVYAACSQMNAHQRHHICCLVERATSSQSLNPVWDALRDGIISSSKFHWAVKQQKIFSPAFGLRCEEVVKTLLATLLHPDETNCLDYGFMQSPQNGIFGVSLDFAANVKTFDPNCKVYEIKCRFKYTFAKMECDPIYAAYQRLYEAPGKLALKDFFYSISKPAVEYVGLGKLPSESDYLVAYDQEWEACPRKKRKLTPLHNLIRECILHNSTTESDVYVLTDPQDTRGQISIKARFKANLFVNVRHSYFYQVLLQSSIVEEYIGSPKYYIATGFFRKRGYQDPVNCTIGGDALDPHVEIPTLLIVTPVYFPRGAKHRLLHQAANFWSRSAKDTFPYIKWDFSYLSAN 3poz A 1.5 BS01 03P A 1 V726 A743 K745 M766 C775 R776 L788 T790 M793 L844 T854 D855 F856 V26 A39 K41 M55 C64 R65 L77 T79 M82 L133 T143 D144 F145 D837 A839 R841 N842 D855 D126 A128 R130 N131 D144 2.7.10.1 0004672,0004713,0005524,0006468 ic50=23nM remove_due_to_license_issue IC50=4.0nM P00533 21454582 1023 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPVKIPVAIKELANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDVVDADEYL 3pp0 A 2.25 BS01 03Q A 1 L726 V734 A751 K753 E770 M774 L785 L796 T798 L800 M801 R849 L852 T862 D863 F864 L21 V29 A46 K48 E65 M69 L80 L91 T93 L95 M96 R144 L147 T157 D158 F159 D845 A847 R849 N850 D863 D140 A142 R144 N145 D158 2.7.10.1 0004672,0004713,0005524,0006468 ic50=11nM remove_due_to_license_issue IC50=11nM P04626 21454582 1 APNQALLRILKETELRKVKVLGSGAFGTVYKGIWIPDGENVKIPVAIKVLRENTSPKANKEILDEAYVMAGVGSPYVSRLLGICLTSTVQLVTQLMPYGCLLDHVRENRGRLGSQDLLNWCMQIAKGMSYLEDVRLVHRDLAARNVLVKSPNHVKITDFGLARLLDIDETEYHAGKVPIKWMALESILRRRFTHQSDVWSYGVTVWELMTFGAKPYDGIPAREIPDLLEKGERLPQPPICTIDVYMIMVKCWMIDSECRPRFRELVSEFSRMARDPQRFVVIQNED 3pp1 A 2.7 BS03 IZG A 1 G80 K97 V127 I141 M143 D208 F209 G210 V211 L215 G20 K37 V67 I81 M83 D148 F149 G150 V151 L155 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T166 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.8nM Q02750 21310613 500 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3pp7 B 2.35 BS01 SVR B 1 P29 N51 H54 G55 Y59 G331 A334 P29 N51 H54 G55 Y59 G331 A334 R49 R90 K238 T296 R49 R90 K238 T296 2.7.1.40 0000287,0003824,0004743,0005524,0006096,0016301,0030955,0046872 remove_due_to_license_issue Q27686 21733839 499 SQLAHNLTLSIFDPVANYRAARIICTIGPSTQSVEALKGLIQSGMSVARMNFSHGSHEYHQTTINNVRQAAAELGVNIAIALDTKGPEIRTGQFVGGDAVMERGATCYVTTDPAFADKGTKDKFYIDYQNLSKVVRPGNYIYIDDGILILQVQSHEDEQTLECTVTNSHTISDRRGVNLPGCDVDLPAVSAKDRVDLQFGVEQGVDMIFASFIRSAEQVGDVRKALGPKGRDIMIICKIENHQGVQNIDSIIEESDGIMVARGDLGVEIPAEKVVVAQKILISKCNVAGKPVICATQMLESMTYNPRPTRAEVSDVANAVFNGADCVMLSGETAKGKYPNEVVQYMARICLEAQSALNEYVFFNSIKKLQHIPMSADEAVCSSAVNSVYETKAKAMVVLSNTGRSARLVAKYRPNCPIVCVTTRLQTCRQLNITQGVESVFFDADKLGHDEGKEHRVAAGVEFAKSKGYVQTGDYCVVIHAKGYANQTRILLVE 3ppj A 3.7 BS01 FOI A 1 I463 V471 A481 K483 E501 L514 I527 T529 W531 C532 F583 D594 I16 V24 A34 K36 E54 L67 I80 T82 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21251822 727 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3ppk A 3.0 BS01 FNI A 1 V471 A481 K483 E501 I527 T529 W531 C532 F583 D594 V24 A34 K36 E54 I80 T82 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21251822 727 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3ppm A 1.78 BS01 JG1 A 1 M191 F192 S217 T236 I238 S241 G268 L278 T488 M495 M159 F160 S185 T204 I206 S209 G236 L246 T456 M463 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 Ki=0.29nM remove_due_to_license_issue Ki=0.29nM P97612 21355555 600 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQP 3ppo A 2.7 BS01 DCK A 1 Q39 S71 N72 Y91 T94 N135 Y137 Y217 Y241 Q8 S40 N41 Y60 T63 N104 Y106 Y186 Y210 ? 0022857,0043190,0055085 remove_due_to_license_issue O32243 21366542 401 DTIKIGAQSMTESEIVANMIAQLIEHDTDLNTALVKNLGSNYVQHQAMLGGDIDISATRYSGTDLTSTLGKEAEKDPKKALNIVQNEFQKRFSYKWFDSYGFDNTYAFTVTKKFAEKEHINTVSDLKKNASQYKLGVDNAWLKRKGDGYKGFVSTYGFEFGTTYPMQIGLVYDAVKNGKMDAVLAYSTDGRIKAYDLKILKDDKRFFPPYDCSPVIPEKVLKEHPELEGVINKLIGQIDTETMQELNYEVDGKLKEPSVVAKEFLEKHHYFD 3ppq A 1.91 BS01 CHT A 1 N135 Y137 Y217 Y241 N103 Y105 Y185 Y209 ? 0022857,0043190,0055085 Kd=28uM remove_due_to_license_issue O32243 21366542 401 TIKIGAQSMTESEIVANMIAQLIEHDTDLNTALVKNLGSNYVQHQAMLGGDIDISATRYSGTDLTSTLGKEAEKDPKKALNIVQNEFQKRFSYKWFDSYGFDNTYAFTVTKKFAEKEHINTVSDLKKNASQYKLGVDNAWLKRKGDGYKGFVSTYGFEFGTTYPMQIGLVYDAVKNGKMDAVLAYSTDGRIKAYDLKILKDDKRFFPPYDCSPVIPEKVLKEHPELEGVINKLIGQIDTETMQELNYEVDGKLKEPSVVAKEFLEKHHYFD 3ppr A 2.1 BS01 4CS A 1 Y91 N135 Y137 Y217 Y241 Y59 N103 Y105 Y185 Y209 ? 0022857,0043190,0055085 Kd=1.5mM remove_due_to_license_issue O32243 21366542 401 TIKIGAQSMTESEIVANMIAQLIEHDTDLNTALVKNLGSNYVQHQAMLGGDIDISATRYSGTDLTSTLGKEAEKDPKKALNIVQNEFQKRFSYKWFDSYGFDNTYAFTVTKKFAEKEHINTVSDLKKNASQYKLGVDNAWLKRKGDGYKGFVSTYGFEFGTTYPMQIGLVYDAVKNGKMDAVLAYSTDGRIKAYDLKILKDDKRFFPPYDCSPVIPEKVLKEHPELEGVINKLIGQIDTETMQELNYEVDGKLKEPSVVAKEFLEKHHYFD 3pr0 A 2.2 BS01 JG2 A 1 M191 F192 S193 S217 D237 I238 G239 S241 T488 M159 F160 S161 S185 D205 I206 G207 S209 T456 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 21355555 600 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQ 3prf A 2.9 BS01 FP3 A 1 I463 A481 E501 W531 C532 F583 G593 D594 I16 A34 E54 W84 C85 F136 G146 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21251822 727 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3prs A 1.38 BS01 RIT A 1 D15 D33 D35 G37 S78 Y79 G80 D81 D119 F194 D219 G221 T222 T223 Y226 I304 D15 D33 D35 G37 S78 Y79 G80 D81 D119 F194 D219 G221 T222 T223 Y226 I304 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 remove_due_to_license_issue P11838 22213702 1001 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 3prz A 2.6 BS01 3RZ A 1 I831 K833 D836 Y867 I879 V882 M953 D964 I590 K592 D595 Y626 I638 V641 M712 D723 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 21269826 1 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEVSLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNYCHPIALPRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLG 3ps1 A 1.85 BS02 ZH2 A 1 L62 C63 E78 H79 T191 I198 G210 S211 F212 A215 H238 K239 D242 H265 L62 C63 E78 H79 T191 I198 G210 S211 F212 A215 H238 K239 D242 H265 0009245,0103117 remove_due_to_license_issue 21194954 401 MIKQRTLKRIVQATGVGLHTGKKVTLTLRPAPANTGVIYRRTDLNPPVDFPADAKSVRDTMLCTCLVNEHDVRISTVEHLNAALAGLGIDNIVIEVNAPEIPIMDGSAAPFVYLLLDAGIDELNCAKKFVRIKETVRVEDGDKWAEFKPYNGFSLDFTIDFNHPAIDSSNQRYAMNFSADAFMRQISRARTFGFMRDIEYLQSRGLCLGGSFDCAIVVDDYRVLNEDGLRFEDEFVRHKMLDAIGDLFMCGHNIIGAFTAYKSGHALNNKLLQAVLAKQEAWEYVTFQDDAELPLAFKAP 3ps6 A 2.6 BS01 3PS A 1 I831 K833 D841 Y867 I879 V882 M953 I963 D964 I587 K589 D597 Y623 I635 V638 M709 I719 D720 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 21269826 1 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNYPIALPRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLG 3psb A 3.4 BS01 SM6 A 1 I463 A481 K483 E501 T529 W531 C532 F583 D594 I16 A34 K36 E54 T82 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21211972 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3psd A 3.6 BS01 SM7 A 1 I463 V471 A481 K483 E501 I527 T529 Q530 W531 C532 F583 D594 I16 V24 A34 K36 E54 I80 T82 Q83 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21536432 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3ptg A 2.43 BS02 932 A 1 I70 V78 A91 E147 L148 M149 A151 N152 V196 L206 I25 V33 A46 E102 L103 M104 A106 N107 V151 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T168 2.7.11.24 0004672,0004707,0005524,0006468 ic50=25nM remove_due_to_license_issue IC50=<100nM P53779 21316234 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLAVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPAHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIYDKQLDEREHTIEEWKELIYKEVMNS 3pty A 2.0 BS01 AFO A 1 G737 N740 R1055 G3 N6 R272 2.4.2.- remove_due_to_license_issue P9WNL5 21383969 1 SVGRSNLQALAGKTCGLAEDVLVELDPNAGMLAPVTAPLADALGAGLSEAFTPNGIPADVGTTAAPGINGSRARLPYNLDPARTPVLGSWRAGVQVPAMLRSGWYRLPTNEQRDRAPLLVVTAAGRFDSREVRLQWATDEQAAAGHHGGSMEFADVGAAPAWRNLRAPLSAIPSTATQVRLVADDQDLAPQHWIALTPPRIPRVRTLQNVVGAADPVFLDWLVGLAFPCQRPFGHQYGVDETPKWRILPDRITELLMRATTVASYLKDDWFRDWGALQRLTPYY 3pup A 2.99 BS01 OS1 A 1 I62 G63 A83 K85 D133 Y134 V135 P136 Q185 N186 L188 D200 I28 G29 A49 K51 D98 Y99 V100 P101 Q150 N151 L153 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 21446733 421 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 3pvp A 2.3 BS01 dna C 0 K436 R444 Q445 R468 D469 T471 T472 Y475 K479 K26 R34 Q35 R58 D59 T61 T62 Y65 K69 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 101 ~ 113 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRSK 3pvp A 2.3 BS02 dna D 0 K436 R438 R452 S458 L459 P460 H470 M474 K26 R28 R42 S48 L49 P50 H60 M64 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 201 ~ 213 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRSK 3pvp B 2.3 BS01 dna E 0 K436 R444 Q445 R468 D469 T471 T472 Y475 K479 K26 R34 Q35 R58 D59 T61 T62 Y65 K69 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 101 ~ 113 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRS 3pvp B 2.3 BS02 dna F 0 K436 R438 S458 L459 P460 H470 M474 K26 R28 S48 L49 P50 H60 M64 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 201 ~ 213 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRS 3pvu A 2.48 BS01 QRW A 1 G200 F202 G203 V205 K220 L222 L324 D335 G171 F173 G174 V176 K191 L193 L295 D306 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 ic50=290nM remove_due_to_license_issue IC50=30nM P21146 21596927 800 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKMGWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 3pvv A 2.0 BS01 dna C 0 R444 Q445 R468 D469 T471 T472 Y475 K479 R34 Q35 R58 D59 T61 T62 Y65 K69 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 101 ~ 113 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRSK 3pvv A 2.0 BS02 dna D 0 K436 T437 R438 R452 S458 L459 P460 H470 M474 K26 T27 R28 R42 S48 L49 P50 H60 M64 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 201 ~ 213 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRSK 3pvv B 2.0 BS01 dna E 0 K436 R468 T471 T472 Y475 K479 K26 R58 T61 T62 Y65 K69 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 101 ~ 113 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRS 3pvv B 2.0 BS02 dna F 0 G435 K436 T437 R438 S458 L459 P460 H470 M474 G25 K26 T27 R28 S48 L49 P50 H60 M64 ? 0003677,0003688,0005524,0006270,0006275,0043565 remove_due_to_license_issue P9WNW3 21620858 201 ~ 213 ISAATIMAATAEYFDTTVEELRGPGKTRALAQSRQIAMYLCRELTDLSLPKIGQAFGRDHTTVMYAQRKILSEMAERREVFDHVKELTTRIRQRS 3pvw A 2.49 BS01 QRX A 1 G200 G201 F202 G203 V205 K220 L222 L324 D335 G337 G172 G173 F174 G175 V177 K192 L194 L296 D307 G309 D317 K319 N322 D335 K344 T353 D289 K291 N294 D307 K316 T325 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 ic50=54nM remove_due_to_license_issue IC50=20nM P21146 21596927 800 SKKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKMGWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 3pwd A 2.2 BS01 CZ0 A 1 V45 K68 F113 M163 I174 D175 V39 K62 F107 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Ki=0.22uM remove_due_to_license_issue P28523 21720886 1 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 3pwh A 3.296 BS01 ZMA A 1 A63 S67 F168 M177 L249 N253 Y271 I274 A57 S61 F154 M163 L235 N239 Y257 I260 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue Ki=1.9nM, Kd=0.22nM, IC50=42nM P29274 21885291 401 SVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLKQMESQPLPGERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 3pwk A 1.5 BS02 L14 A 1 R99 N127 G159 A160 E220 K223 R245 R98 N126 G158 A159 E219 K222 R244 0004073,0008652,0009086,0009088,0009089,0009097,0016620,0046983,0050661,0051287 Ki=0.45mM remove_due_to_license_issue 22039970 368 GYTVAVVGATGAVGAQMIKMLEESTLPIDKIRYLASARSAGKSLKFKDQDITIEETTETAFEGVDIALFSAGSSTSAKYAPYAVKAGVVVVDNTSYFRQNPDVPLVVPEVNAHALDAHNGIIACPNCSTIQMMVALEPVRQKWGLDRIIVSTYQAVSGAGMGAILETQRELREVLNDGVKPCDLHAEILPSGGDKKHYPIAFNALPQIDVFTDNDYTYEEMKMTKETKKIMEDDSIAVSATCVRIPVLSAHSESVYIETKEVAPIEEVKAAIAAFPGAVLEDDVAHQIYPQAINAVGSRDTFVGRIRKDLDAEKGIHMWVVSDNLLKGAAWNSVQIAETLHERGLVRPTAELKFELK 3pwm A 1.46 BS01 017 B 1 D25 A28 D30 G48 P81 V82 I84 D25 A28 D30 G48 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 21446746 402 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 3pwm B 1.46 BS01 017 B 1 D125 G127 D129 D130 G148 G149 I150 D25 G27 D29 D30 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 21446746 402 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 3pww A 1.22 BS01 ROC A 1 D15 D33 D35 G37 Y79 G80 F116 L125 F194 I217 D219 G221 T222 T223 D15 D33 D35 G37 Y79 G80 F116 L125 F194 I217 D219 G221 T222 T223 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 remove_due_to_license_issue P11838 22213702 1001 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 3px8 X 1.29 BS01 JP2 X 1 Y80 V81 G121 N122 Y123 I172 R180 Y77 V78 G118 N119 Y120 I169 R177 V81 V78 3.2.2.22 0017148,0030598 ic50=230uM remove_due_to_license_issue P02879 21641093 1 KQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAP 3px9 X 1.89 BS01 JP3 X 1 Y80 V81 G121 Y123 I172 R180 Y77 V78 G118 Y120 I169 R177 V81 V78 3.2.2.22 0017148,0030598 ic50=380uM remove_due_to_license_issue IC50=380000nM P02879 21641093 1 KQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAP 3pxf A 1.8 BS01 2AN A 1 I52 K56 H71 L76 I56 K60 H75 L80 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=37uM remove_due_to_license_issue Kd=37000nM, IC50=91000nM P24941 21291269 304 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pxf A 1.8 BS02 2AN A 2 Y15 K33 I35 L55 K56 V64 F80 A144 D145 Y19 K37 I39 L59 K60 V68 F84 A148 D149 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=37uM remove_due_to_license_issue Kd=37000nM, IC50=91000nM P24941 21291269 305 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pxq A 1.9 BS01 2AN A 1 I10 G11 E12 V18 K33 V64 F80 L83 D86 Q131 L134 D145 I14 G15 E16 V22 K37 V64 F80 L83 D86 Q131 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=37uM remove_due_to_license_issue Kd=37000nM, IC50=91000nM P24941 21291269 300 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pxq A 1.9 BS02 2AN A 2 I52 K56 H71 L76 F152 I52 K56 H71 L76 F152 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=37uM remove_due_to_license_issue Kd=37000nM, IC50=91000nM P24941 21291269 301 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pxq A 1.9 BS03 2AN A 3 K33 I35 L55 K56 V64 F80 A144 D145 F146 F152 K37 I39 L55 K56 V64 F80 A144 D145 F146 F152 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=37uM remove_due_to_license_issue Kd=37000nM, IC50=91000nM P24941 21291269 302 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pxy A 1.8 BS01 JWS A 1 I10 A31 F80 F82 L83 H84 Q85 L134 D145 I10 A31 F76 F78 L79 H80 Q81 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=5.9uM remove_due_to_license_issue P24941 21291269 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pxz A 1.7 BS03 JWS A 1 I10 A31 K33 V64 F80 L83 H84 Q85 L134 I14 A35 K37 V68 F84 L87 H88 Q89 L138 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=5.9uM remove_due_to_license_issue P24941 21291269 301 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3py0 A 1.75 BS01 SU9 A 1 I10 A31 F80 F82 L83 H84 L134 I10 A31 F76 F78 L79 H80 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.13uM remove_due_to_license_issue IC50=22nM P24941 21291269 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3py1 A 2.05 BS01 SU9 A 1 I10 A31 F80 F82 L83 H84 K89 L134 D145 I14 A35 F84 F86 L87 H88 K93 L138 D149 D127 K129 Q131 N132 D145 T158 T165 D131 K133 Q135 N136 D149 T162 T169 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.13uM remove_due_to_license_issue IC50=22nM P24941 21291269 300 SPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3pyy A 1.85 BS02 3YY A 1 A356 L359 L360 L448 I451 A452 G482 C483 P484 A102 L105 L106 L194 I197 A198 G228 C229 P230 D382 A384 R386 N387 D400 P421 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=398nM, EC50=794nM P00519 21338916 538 YDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 3pz1 B 1.95 BS01 3PZ B 1 Y44 W52 D238 W244 F289 H290 Y37 W45 D231 W237 F282 H283 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=724nM remove_due_to_license_issue Q08603 21520375 1 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3pz2 B 2.35 BS03 3PZ B 1 Y44 D238 W244 D287 F289 H290 Y35 D229 W235 D278 F280 H281 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H181 R223 K226 D229 C231 Y232 D271 D278 H281 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=724nM remove_due_to_license_issue Q08603 21520375 333 QKDVTIKSDAPDTLLLEKHADYIASYGSEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3pz3 B 2.0 BS03 PZ3 B 1 Y44 Y51 W52 L99 F147 D238 W244 P288 F289 H290 Y37 Y44 W45 L92 F140 D231 W237 P281 F282 H283 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=141nM remove_due_to_license_issue Q08603 21520375 333 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 3pz4 B 2.1 BS03 3PZ B 1 L96 W102 D297 D359 Y361 H362 L76 W82 D277 D339 Y341 H342 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H228 R271 K274 D277 C279 Y280 D332 D339 H342 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=6nM remove_due_to_license_issue Q02293 21520375 429 EPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 3q05 A 2.4 BS01 dna K 0 S241 R248 R273 A276 R280 S148 R155 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 3 ~ 28 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q05 A 2.4 BS02 dna L 0 V122 R248 R283 V29 R155 R190 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q05 B 2.4 BS01 dna K 0 K120 S121 K27 S28 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 3 ~ 28 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q05 B 2.4 BS02 dna L 0 S241 R273 A276 R280 S148 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q05 C 2.4 BS01 dna K 0 S241 R273 A276 R280 S148 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 3 ~ 28 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q05 C 2.4 BS02 dna L 0 K120 R248 K27 R155 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q05 D 2.4 BS01 dna L 0 S241 R273 A276 R280 S148 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 21522129 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 3q0b X 2.2 BS01 dna A 0 Y378 R379 S391 Q392 S393 G394 S413 G415 Y416 D418 Y428 T429 Q431 Y486 Y17 R18 S30 Q31 S32 G33 S52 G54 Y55 D57 Y67 T68 Q70 Y110 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKDDGGELVATSIVSSGGYNDVLDNSDVLIYTGQGGNVGEPPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0d A 2.3704 BS01 dna B 0 Y378 R379 S391 Q392 S393 G394 S412 S413 G415 Y416 D418 Y428 T429 Q431 Y17 R18 S30 Q31 S32 G33 S49 S50 G52 Y53 D55 Y65 T66 Q68 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKDGELVATSIVSSGGYNDVLDNSDVLIYTGQGGNVEPPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0d A 2.3704 BS02 dna C 0 N383 R389 S391 Q392 Y397 N22 R28 S30 Q31 Y36 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKDGELVATSIVSSGGYNDVLDNSDVLIYTGQGGNVEPPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0d X 2.3704 BS01 dna B 0 M380 R389 S391 Q392 Y397 M19 R28 S30 Q31 Y36 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKLVATSIVSSGGYNDVLDNSDVLIYTGQGGNVPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0d X 2.3704 BS02 dna C 0 Y378 R379 S391 Q392 V411 S413 G415 Y416 D418 Y428 Q431 Y486 Y17 R18 S30 Q31 V45 S47 G49 Y50 D52 Y62 Q65 Y102 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKLVATSIVSSGGYNDVLDNSDVLIYTGQGGNVPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0f A 2.75 BS01 dna B 0 Y378 R379 Q392 S393 G394 S413 G414 Y416 D418 Y428 T429 Q431 Y486 Y17 R18 Q31 S32 G33 S52 G53 Y55 D57 Y67 T68 Q70 Y108 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 11 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKDDGGELVATSIVSSGGYNDVLDNSDVLIYTGQGGNEPPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0f X 2.75 BS01 dna C 0 Y378 R379 Q392 S393 G394 S412 S413 G414 Y416 D418 Y428 T429 Q431 Y486 Y17 R18 Q31 S32 G33 S51 S52 G53 Y55 D57 Y67 T68 Q70 Y107 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 21245167 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKDDGGELVATSIVSSGGYNDVLDNSDVLIYTGQGGNPPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 3q0l A 2.503 BS01 rna C 0 Q860 R864 Q867 F897 N899 Y900 Y933 R936 Q939 H972 Q975 C1007 R1008 Q1011 N1043 Y1044 Q1047 N1080 E1083 Y1120 N1122 Y1123 H1159 Q33 R37 Q40 F70 N72 Y73 Y106 R109 Q112 H145 Q148 C180 R181 Q184 N216 Y217 Q220 N253 E256 Y293 N295 Y296 H332 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 3q0l B 2.503 BS01 rna D 0 Q860 R864 Q867 F897 N899 Y900 Y933 C935 R936 Q939 Q968 H972 Q975 Y1005 C1007 R1008 Q1011 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 H1159 Q33 R37 Q40 F70 N72 Y73 Y106 C108 R109 Q112 Q141 H145 Q148 Y178 C180 R181 Q184 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 H332 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 3q0m A 2.705 BS01 rna C 0 Q860 R864 Q867 N899 Y900 R936 Q939 Q968 H972 Q975 Y1005 R1008 Q1011 N1043 Y1044 Q1047 S1079 N1080 E1083 N1122 Y1123 Q1126 Y1156 H1159 Q32 R36 Q39 N71 Y72 R108 Q111 Q140 H144 Q147 Y177 R180 Q183 N215 Y216 Q219 S251 N252 E255 N294 Y295 Q298 Y328 H331 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 RSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLE 3q0m B 2.705 BS01 rna D 0 Q860 R864 Q867 F897 N899 Y900 Q903 Y933 R936 Q939 Q968 H972 Q975 Y1005 R1008 N1043 Y1044 F1077 N1080 E1083 N1122 Y1123 Q1126 Y1156 H1159 Q31 R35 Q38 F68 N70 Y71 Q74 Y104 R107 Q110 Q139 H143 Q146 Y176 R179 N214 Y215 F248 N251 E254 N293 Y294 Q297 Y327 H330 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 SRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 3q0n A 2.4 BS01 rna C 0 Q860 Q867 F897 N899 Y900 Q903 R936 Q939 H972 C1007 R1008 Q1011 N1043 Y1044 Q1047 K1076 F1077 S1079 N1080 E1083 N1122 Y1123 Q1126 H1159 Q33 Q40 F70 N72 Y73 Q76 R109 Q112 H145 C180 R181 Q184 N216 Y217 Q220 K249 F250 S252 N253 E256 N295 Y296 Q299 H332 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 3q0n B 2.4 BS01 rna D 0 N899 Y900 Q903 M932 R936 Q939 H972 C1007 R1008 Q1011 N1043 Y1044 Q1047 F1077 S1079 N1080 E1083 Y1120 N1122 Y1123 H1159 N72 Y73 Q76 M105 R109 Q112 H145 C180 R181 Q184 N216 Y217 Q220 F250 S252 N253 E256 Y293 N295 Y296 H332 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 7 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 3q0p A 2.6 BS01 rna C 0 Q860 R864 Q867 F897 N899 Y900 M932 Y933 R936 Q939 H972 R1008 Y1041 N1043 Y1044 K1076 F1077 N1080 E1083 Y1120 N1122 Y1123 Y1156 H1159 Q33 R37 Q40 F70 N72 Y73 M105 Y106 R109 Q112 H145 R181 Y214 N216 Y217 K249 F250 N253 E256 Y293 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKYY 3q0p B 2.6 BS01 rna D 0 Q860 R864 Q867 N899 Y900 Y933 R936 Q939 H972 C1007 R1008 Q1011 N1043 Y1044 F1077 N1080 E1083 Y1120 N1122 Y1123 Y1156 H1159 Q33 R37 Q40 N72 Y73 Y106 R109 Q112 H145 C180 R181 Q184 N216 Y217 F250 N253 E256 Y293 N295 Y296 Y329 H332 ? 0003723 remove_due_to_license_issue Q14671 21397187 1 ~ 8 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFALSTHPYGCRVIQRILEHCLPDQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 3q0q A 2.0 BS01 rna B 0 Q738 R742 Q745 N777 Y778 Q781 M810 Y811 C813 R814 Q817 Q848 N849 N851 H852 Q855 Y885 R888 Q891 Y921 N923 Y924 Q927 S959 N960 E963 Y1000 N1002 Y1003 Q1006 Y1036 H1039 Q33 R37 Q40 N72 Y73 Q76 M105 Y106 C108 R109 Q112 Q143 N144 N146 H147 Q150 Y180 R183 Q186 Y216 N218 Y219 Q222 S254 N255 E258 Y295 N297 Y298 Q301 Y331 H334 ? 0003723 remove_due_to_license_issue Q8TB72 21397187 1 ~ 8 GRSRLLEDFRNNRFPNLQLRDLIGHIVEFSQDQHGSRFIQQKLERATPAERQMVFNEILQAAYQLMTDVFGNYVIQKFFEFGSLDQKLALATRIRGHVLPLALQMYGCRVIQKALESISSDQQVISEMVKELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFVLSTHPYGCRVIQRILEHCTAEQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVSEIRGKVLALSQHKFASNVVEKCVTHASRAERALLIDEVCCQNDGPHSALYTMMKDQYANYVVQKMIDMAEPAQRKIIMHKIRPHITTLRKYTYGKHILAKLEKYY 3q0r A 2.0 BS01 rna B 0 Q738 R742 Q745 N777 Y778 Q781 Y811 C813 R814 Q817 Q848 N849 H852 Q855 Y885 C887 R888 Q891 Y921 N923 Y924 Q927 S959 N960 E963 Y1000 N1002 Y1003 Q1006 Y1036 H1039 Q33 R37 Q40 N72 Y73 Q76 Y106 C108 R109 Q112 Q143 N144 H147 Q150 Y180 C182 R183 Q186 Y216 N218 Y219 Q222 S254 N255 E258 Y295 N297 Y298 Q301 Y331 H334 ? 0003723 remove_due_to_license_issue Q8TB72 21397187 1 ~ 8 GRSRLLEDFRNNRFPNLQLRDLIGHIVEFSQDQHGSRFIQQKLERATPAERQMVFNEILQAAYQLMTDVFGNYVIQKFFEFGSLDQKLALATRIRGHVLPLALQMYGCRVIQKALESISSDQQVISEMVKELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFVLSTHPYGCRVIQRILEHCTAEQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVSEIRGKVLALSQHKFASNVVEKCVTHASRAERALLIDEVCCQNDGPHSALYTMMKDQYANYVVQKMIDMAEPAQRKIIMHKIRPHITTLRKYTYGKHILAKLEKYY 3q0s A 2.0 BS01 rna B 0 R742 Q745 N777 Y778 Q781 Y811 R814 Q817 H852 C887 R888 Q891 N923 Y924 Q927 S959 N960 E963 Y1000 N1002 Y1003 Y1036 H1039 R37 Q40 N72 Y73 Q76 Y106 R109 Q112 H147 C182 R183 Q186 N218 Y219 Q222 S254 N255 E258 Y295 N297 Y298 Y331 H334 ? 0003723 remove_due_to_license_issue Q8TB72 21397187 1 ~ 8 GRSRLLEDFRNNRFPNLQLRDLIGHIVEFSQDQHGSRFIQQKLERATPAERQMVFNEILQAAYQLMTDVFGNYVIQKFFEFGSLDQKLALATRIRGHVLPLALQMYGCRVIQKALESISSDQQVISEMVKELDGHVLKCVKDQNGNHVVQKCIECVQPQSLQFIIDAFKGQVFVLSTHPYGCRVIQRILEHCTAEQTLPILEELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVSEIRGKVLALSQHKFASNVVEKCVTHASRAERALLIDEVCCQNDGPHSALYTMMKDQYANYVVQKMIDMAEPAQRKIIMHKIRPHITTLRKYTYGKHILAKLEKYY 3q0z A 2.29 BS01 23E A 1 L392 A395 A396 I424 H428 G493 V494 P495 P496 R498 W500 R503 L370 A373 A374 I402 H406 G471 V472 P473 P474 R476 W478 R481 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 21486696 601 SMSYTWTGALITPCVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSLSRARPRWFM 3q1x A 1.59 BS01 SER A 1 H208 R222 H223 H208 R222 H223 2.3.1.30 0008652,0009001,0016746 remove_due_to_license_issue Q9U8X2 21297164 314 MDNYIYSIAHQLYEMYLQDEDAFHSKRDYPHKKVFTELQKLRKIFFPDFFMKHQKITESHIASELTKLVDYIKDSVTAYNDELFAHQCVMAILEKLPSIKRTLKTDLIAAYAGDPAAPGLSLIIRCYPGFQAVIVYRIAHVLYECGERYYCREMMESVHSYTSIDIHPGASIKGHFFIDHGVGVVIGETAIIGEWCRIYQSVTLGAMHFQEEGGVIKRGTKRHPTVGDYVTIGTGAKVLGNIIVGSHVRIGANCWIDRDVDSNQTVY 3q2a A 1.99 BS03 PAB A 1 W338 E391 T392 L393 T463 L464 W337 E390 T391 L392 T462 L463 E104 E134 H137 E197 E231 H234 E103 E133 H136 E196 E230 H233 1.14.13.236 0004497,0009056,0016491,0018638,0042203,0046872 remove_due_to_license_issue Q00456 22264099 519 AMHPRKDWYELTRATNWTPSYVTEEQLFPERMSGHMGIPLEKWESYDEPYKTSYPEYVSIQREKDAGAYSVKAALERAKIYENSDPGWISTLKSHYGAIAVGEYAAVTGEGRMARFSKAPGNRNMATFGMMDELRHGQLQLFFPHEYCKKDRQFDWAWRAYHSNEWAAIAAKHFFDDIITGRDAISVAIMLTFSFETGFTNMQFLGLAADAAEAGDYTFANLISSIQTDESRHAQQGGPALQLLIENGKREEAQKKVDMAIWRAWRLFAVLTGPVMDYYTPLEDRSQSFKEFMYEWIIGQFERSLIDLGLDKPWYWDLFLKDIDELHHSYHMGVWYWRTTAWWNPAAGVTPEERDWLEEKYPGWNKRWGRCWDVITENVLNDRMDLVSPETLPSVCNMSQIPLVGVPGDDWNIEVFSLEHNGRLYHFGSEVDRWVFQQDPVQYQNHMNIVDRFLAGQIQPMTLEGALKYMGFQSIEEMGKDAHDFAWADKC 3q2a A 1.99 BS04 PAB A 2 W167 P403 M471 W166 P402 M470 E104 E134 H137 E197 E231 H234 E103 E133 H136 E196 E230 H233 1.14.13.236 0004497,0009056,0016491,0018638,0042203,0046872 remove_due_to_license_issue Q00456 22264099 520 AMHPRKDWYELTRATNWTPSYVTEEQLFPERMSGHMGIPLEKWESYDEPYKTSYPEYVSIQREKDAGAYSVKAALERAKIYENSDPGWISTLKSHYGAIAVGEYAAVTGEGRMARFSKAPGNRNMATFGMMDELRHGQLQLFFPHEYCKKDRQFDWAWRAYHSNEWAAIAAKHFFDDIITGRDAISVAIMLTFSFETGFTNMQFLGLAADAAEAGDYTFANLISSIQTDESRHAQQGGPALQLLIENGKREEAQKKVDMAIWRAWRLFAVLTGPVMDYYTPLEDRSQSFKEFMYEWIIGQFERSLIDLGLDKPWYWDLFLKDIDELHHSYHMGVWYWRTTAWWNPAAGVTPEERDWLEEKYPGWNKRWGRCWDVITENVLNDRMDLVSPETLPSVCNMSQIPLVGVPGDDWNIEVFSLEHNGRLYHFGSEVDRWVFQQDPVQYQNHMNIVDRFLAGQIQPMTLEGALKYMGFQSIEEMGKDAHDFAWADKC 3q2a A 1.99 BS05 PAB A 3 E104 E134 F176 I180 E197 E231 E103 E133 F175 I179 E196 E230 E104 E134 H137 E197 E231 H234 E103 E133 H136 E196 E230 H233 1.14.13.236 0004497,0009056,0016491,0018638,0042203,0046872 remove_due_to_license_issue Q00456 22264099 521 AMHPRKDWYELTRATNWTPSYVTEEQLFPERMSGHMGIPLEKWESYDEPYKTSYPEYVSIQREKDAGAYSVKAALERAKIYENSDPGWISTLKSHYGAIAVGEYAAVTGEGRMARFSKAPGNRNMATFGMMDELRHGQLQLFFPHEYCKKDRQFDWAWRAYHSNEWAAIAAKHFFDDIITGRDAISVAIMLTFSFETGFTNMQFLGLAADAAEAGDYTFANLISSIQTDESRHAQQGGPALQLLIENGKREEAQKKVDMAIWRAWRLFAVLTGPVMDYYTPLEDRSQSFKEFMYEWIIGQFERSLIDLGLDKPWYWDLFLKDIDELHHSYHMGVWYWRTTAWWNPAAGVTPEERDWLEEKYPGWNKRWGRCWDVITENVLNDRMDLVSPETLPSVCNMSQIPLVGVPGDDWNIEVFSLEHNGRLYHFGSEVDRWVFQQDPVQYQNHMNIVDRFLAGQIQPMTLEGALKYMGFQSIEEMGKDAHDFAWADKC 3q2a A 1.99 BS06 PAB A 4 H447 M448 R453 Q458 H446 M447 R452 Q457 E104 E134 H137 E197 E231 H234 E103 E133 H136 E196 E230 H233 1.14.13.236 0004497,0009056,0016491,0018638,0042203,0046872 remove_due_to_license_issue Q00456 22264099 522 AMHPRKDWYELTRATNWTPSYVTEEQLFPERMSGHMGIPLEKWESYDEPYKTSYPEYVSIQREKDAGAYSVKAALERAKIYENSDPGWISTLKSHYGAIAVGEYAAVTGEGRMARFSKAPGNRNMATFGMMDELRHGQLQLFFPHEYCKKDRQFDWAWRAYHSNEWAAIAAKHFFDDIITGRDAISVAIMLTFSFETGFTNMQFLGLAADAAEAGDYTFANLISSIQTDESRHAQQGGPALQLLIENGKREEAQKKVDMAIWRAWRLFAVLTGPVMDYYTPLEDRSQSFKEFMYEWIIGQFERSLIDLGLDKPWYWDLFLKDIDELHHSYHMGVWYWRTTAWWNPAAGVTPEERDWLEEKYPGWNKRWGRCWDVITENVLNDRMDLVSPETLPSVCNMSQIPLVGVPGDDWNIEVFSLEHNGRLYHFGSEVDRWVFQQDPVQYQNHMNIVDRFLAGQIQPMTLEGALKYMGFQSIEEMGKDAHDFAWADKC 3q2g A 2.3 BS01 QGF A 1 T117 L118 G119 F145 T146 H149 E150 H153 H159 L182 F274 T114 L115 G116 F142 T143 H146 E147 H150 H156 L174 F257 3.4.24.- 0004222,0006508,0008237 ic50=3.5nM remove_due_to_license_issue Q9UHI8 21300546 1 SHRYVETMLVADQSMAEFHGSGLKHYLLTLFSVAARLYKHPSIRNSVSLVVVKILVIHDEQKGPEVTSNAALTLRNFCNWQKQHNPPSDRDAEHYDTAILFTRQDLCGSQTCDTLGMADVGTVCDPSRSCSVIEDDGLQAAFTTAHELGHVFNMPHDDAKQCASLNSHMMASMLSNLDHSQPWSPCSAYMITSFLDNGHGECLMDKPQNPIQLPGDLPGTSYDANRQCQFTFGEDSKHCPTCSTLWCTGLVCQTKHFPWADGTSCGEGKWCINGKCVNKLVP 3q2h A 2.33 BS03 QHF A 1 T117 G119 F145 H149 E150 H153 H159 S180 L182 T114 G116 F142 H146 E147 H150 H156 S173 L175 3.4.24.- 0004222,0006508,0008237 ic50=0.69nM remove_due_to_license_issue Q9UHI8 21300546 1 SHRYVETMLVADQSMAEFHGSGLKHYLLTLFSVAARLYKHPSIRNSVSLVVVKILVIHDEQKGPEVTSNAALTLRNFCNWQKQHNPPSDRDAEHYDTAILFTRQDLCGSQTCDTLGMADVGTVCDPSRSCSVIEDDGLQAAFTTAHELGHVFNMPHDDAKQCASLNDSHMMASMLSNLDHSQPWSPCSAYMITSFLDNGHGECLMDKPQNPIQLPGDLPGTSYDANRQCQFTFGEDSKHCPTCSTLWCTGVLVCQTKHFPWADGTSCGEGKWCINGKCVNKLVP 3q2j A 2.1501 BS02 CKI A 1 M26 Y42 M90 E92 A93 L97 S194 F197 I207 M23 Y39 M87 E89 A90 L94 S191 F194 I204 K44 D190 N195 D208 K41 D187 N192 D205 2.7.1.95 0005524,0008910,0016301,0016773,0046677 remove_due_to_license_issue P0A3Y5 21573013 300 MRISPELKKLIEKYRCVKDTEGMSPAKVYKLVGENENLYLKMTDSRYKGTTYDVEREKDMMLWLEGKLPVPKVLHFERHDGWSNLLMSEADGVLCSEEYEDEQSPEKIIELYAECIRLFHSIDISDCPYTNSLDSRLAELDYLLNNDLADVDCENWEEDTPFKDPRELYDFLKTEKPEEELVFSHGDLGDSNIFVKDGKVSGFIDLGRSGRADKWYDIAFCVRSIREDIGEEQYVELFFDLLGIKPDWEKIKYYILLDELF 3q2m A 2.9 BS01 CKI A 1 F50 F102 I103 A105 F48 F100 I101 A103 ? 0000166,0016740,0046872 remove_due_to_license_issue O06916 21573013 400 KQPIQAQQLIELLKVHYGIDIHTAQFIQGGADTNAFAYQADSESKSYFIKLKYGYHDEINLSIIRLLHDSGIKEIIFPIHTLEAKLFQQLKHFKIIAYPFIHAPNGFTQNLTGKQWKQLGKVLRQIHETSVPISIQQQLRKEIYSPKWREIVRSFYNQIEFDNSDDKLTAAFKSFFNQNSAAIHRLVDTSEKLSKKIQPDLDKYVLCHSDIHAGNVLVGNEESIYIIDWDEPMLAPKERDLMFIGGGVGNVWNKPHEIQYFYEGYGEINVDKTILSYYRHERIVEDIAVYGQDLLSRNQNNQSRLESFKYFKEMFDPNNVVEIAFATEQ 3q32 A 2.5 BS01 J2I A 1 L855 G856 K857 S862 V863 A880 M929 E930 Y931 L932 G935 R980 N981 L983 D994 L16 G17 K18 S23 V24 A41 M90 E91 Y92 L93 G96 R141 N142 L144 D155 D976 A978 R980 N981 D994 S1016 D137 A139 R141 N142 D155 S177 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.0018uM remove_due_to_license_issue IC50=1.8nM O60674 21282055 1 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 3q3b A 2.7 BS01 55E A 1 N64 F67 A83 K85 D133 Y134 V135 L188 D200 N30 F33 A49 K51 D95 Y96 V97 L150 D162 D181 K183 N186 D200 S219 D143 K145 N148 D162 S181 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 21295469 421 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARIQA 3q3k A 2.0 BS03 D90 A 1 T98 Y99 F174 D189 A190 Q192 V213 W215 G216 G218 C220 G226 I227 Y228 T84 Y85 F162 D179 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=7.4nM remove_due_to_license_issue IC50=7.4nM P00742 21345673 700 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 3q3t A 2.6 BS01 RX0 A 1 T12 Q13 Y14 D32 S76 T77 F117 D215 G217 T15 Q16 Y17 D35 S81 T82 F121 D223 G225 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=37nM P00797 21741239 500 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3q43 A 1.8 BS02 D66 A 1 E319 V459 G460 A461 M462 E463 H496 E497 H500 E519 Y575 Y580 E124 V264 G265 A266 M267 E268 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=43nM remove_due_to_license_issue Ki=43nM O96935 21366301 1087 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 3q44 A 1.8 BS02 D50 A 1 E319 V459 G460 A461 E463 H496 E497 H500 E519 M571 E572 Y575 Y580 M1034 E124 V264 G265 A266 E268 H301 E302 H305 E324 M376 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=490nM remove_due_to_license_issue Ki=490nM O96935 21366301 1086 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 3q4b A 2.19 BS01 RX5 A 1 T12 Q13 Y14 D32 G34 Y75 S76 T77 P111 F112 F117 D215 T216 G217 A218 T15 Q16 Y17 D35 G37 Y80 S81 T82 P115 F116 F121 D223 T224 G225 A226 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.47nM P00797 24900262 335 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3q4c A 3.2 BS01 RSW A 1 I462 W530 C531 G533 H538 F582 I16 W84 C85 G87 H92 F136 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 19371126 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3q5h A 2.16 BS01 RX6 A 1 T12 Q13 Y14 V30 D32 G34 S76 T77 P111 F112 F117 D215 T216 G217 A218 T15 Q16 Y17 V33 D35 G37 S81 T82 P115 F116 F121 D223 T224 G225 A226 D32 S35 N37 W39 Y75 D215 A218 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.48nM P00797 24900262 335 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3q6k A 2.52 BS01 SRO A 1 T29 Q91 F223 T327 N342 F344 T29 Q91 F223 T327 N342 F344 ? 0005576 Kd=4.3nM (21795673) remove_due_to_license_issue Q5WPU9 21795673 383 ADTQGYKWKQLLYNNVTPGSYNPDNMISTAFAYDAEGEKLFLAVPRKLPRVPYTLAEVDTKNSLGVKGKHSPLLNKFSGHKTGKELTSIYQPVIDDCRRLWVVDIGSVEYRSRGAKDYPSHRPAIVAYDLKQPNYPEVVRYYFPTRLVEKPTYFGGFAVDVANPKGDCSETFVYITNFLRGALFIYDHKKQDSWNVTHPTFKAERPTKFDYGGKEYEFKAGIFGITLGDRDSEGNRPAYYLAGSAIKVYSVNTKELKQKGGKLNPELLGNRGKYNDAIALAYDPKTKVIFFAEANTKQVSCWNTQKMPLRMKNTDVVYTSSRFVFGTDISVDSKGGLWFMSNGFPPIRKSEKFKYDFPRYRLMRIMDTQEAIAGTACDMN 3q6w A 1.75 BS01 Q6W A 1 I1084 G1085 R1086 V1092 A1108 Y1159 M1160 K1161 G1163 D1164 R1208 M1211 I35 G36 R37 V43 A59 Y110 M111 K112 G114 D115 R159 M162 D1204 A1206 R1208 N1209 D1222 D155 A157 R159 N160 D173 2.7.10.1 0004672,0004713,0005524,0006468 Kd=27nM remove_due_to_license_issue IC50=85nM P08581 21247903 1 TVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHHHHH 3q6z A 2.23 BS01 APR A 1 A822 N824 G831 G832 L833 S922 G924 V925 F926 D961 A31 N33 G40 G41 L42 S131 G133 V134 F135 D168 2.4.2.- remove_due_to_license_issue Q460N5 23473667 1 CFSRTVLAPGVVLIVQQGDLARLPVDVVVNASNEDLKHYGGLAAALSKAAGPELQADCDQIVKREGRLLPGNATISKAGKLPYHHVIHAVGPRWSGYEAPRCVYLLRRAVQLSLCLAEKYKYRSIAIPAISSGVFGFPLGRCVETIVSAIKENFQFKKHCLKEIYLVDVSEKTVEAFAEAVKTVF 3q71 A 2.2 BS01 AR6 A 1 G1022 V1023 S1034 P1036 G1044 P1045 L1046 S1049 A1131 G1133 T1134 G1135 N1136 L1137 H1172 D1175 G34 V35 S46 P48 G56 P57 L58 S61 A143 G145 T146 G147 N148 L149 H184 D187 Q1015 Q27 2.4.2.- remove_due_to_license_issue Q460N5 23473667 800 GTENLYFQSMGKTSWEKGSLVSPGGLQMLLVKEGVQNAKTDVVVNSVPLDLVLSRGPLSKSLLEKAGPELQEELDTVGQGVAVSMGTVLKTSSWNLDCRYVLHVVAPEWRNGSTSSLKIMEDIIRECMEITESLSLKSIAFPAIGTGNLGFPKNIFAELIISEVFKFSSKNQLKTLQEVHFLLHPSDHENIQAFSDEFARRAN 3q72 A 1.655 BS01 GNP A 1 G101 V102 G103 K104 S105 A106 N203 K204 D206 L207 S233 A234 A235 G12 V13 G14 K15 S16 A17 N86 K87 D89 L90 S116 A117 A118 ? 0003924,0005525 remove_due_to_license_issue P55042 21903096 256 SVYKVLLLGAPGVGKSALARIFGGVHTYDRSIVVDGEEASLMVYDIWGDAYVIVYSVTDKGSFEKASELRVQLRRARDVPIILVGNKSDLVRSREVSVDEGRACAVVFDCKFIETSAALHHNVQALFEGVVRQIRLRR 3q77 A 1.998 BS02 2HY A 1 H57 Y94 L99B D102 V190 C191 F192 D194 S195 A213 S214 F215 V216 H41 Y80 L85 D88 V168 C169 F170 D172 S173 A187 S188 F189 V190 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G167 C169 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=6nM remove_due_to_license_issue P08246 21549129 500 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 3q7j A 2.91 BS02 FBO A 1 H99 Q101 A229 G230 A231 E233 E266 T292 R316 E348 Y351 G352 H99 Q101 A229 G230 A231 E233 E266 T292 R316 E348 Y351 G352 E233 H265 E266 H269 E288 S343 Y351 E233 H265 E266 H269 E288 S343 Y351 3.4.11.- 0004177,0005615,0005737,0006508,0008237,0008270,0016020,0042277,0043171,0046872,0070006 remove_due_to_license_issue O93655 21493078 900 MEVEKYDLTLDFDIQKRTFNGTETITADAGDIVLDAVGLQINWMKVNGRDTAFTYDGQTVRAPGDSQPQKIEISFAGKVSDSLSGIYYAGRENGMITTHFQATDARRMFPCVDHPAYKAVFAITVVIDKDYDAISNMPPKRIEVSERKVVEFQDTPRMSTYLLYVGIGKFRYEYEKYRDIDLILASLKDIRSKYPLDMARKSVEFYENYFGIPYALPKMHLISVPEFGAGAMENWGAITFREIYMDIAENSAVTVKRNSATVIAHEIAHQWFGDLVTMKWWNDLWLNESFATFMSYKTMDTLFPEWSFWGDFFVSRTSGALRSDSLKNTHPIEVDVRDPDEISQIFDEISYGKGASILRMIEDYAGYEEFRKGISKYLNDHKFGNAEGSDLWTAIEDVSGKPVKRVMEYWIKNPGYPVIKLKRNGRKITMYQTRFLLNGEEEGRWPVPVNIKKKDGVERILLEDEASIEADGLIKINADSAGFYRVLYDDATFSDVMGHYRDLSPLDRIGLVDDLFAFLLSGHIDPETYRQRIRNFFDDEDHNVITAIVGQMEYLRMLTHAFDDDARAFCRSRMQFLTGKQDENLKIALGRVSRLYVMVDESYAEEMSKLFKDFDSAEPEMRSSIATAYALVTGDLKGLLEKFRSVDRDEDRVRIISAFGKLKSNTDLSTVYGMVEKTEIKKQDMISFFSSALETLPGREFIFANLDRIIRLVIRYFTGNRTASRTVEMMIPVIGLDHPDAEDIVRNIGSKNISMGLAKGIEMLAVNRKLVERIRQTAVK 3q7p A 2.5 BS01 GNP A 1 G101 V102 G103 K104 S105 A106 E147 N203 K204 D206 L207 S233 A234 A235 G12 V13 G14 K15 S16 A17 E47 N90 K91 D93 L94 S120 A121 A122 ? 0003924,0005525 remove_due_to_license_issue P55042 21903096 256 SVYKVLLLGAPGVGKSALARIFGGHTYDRSIVVDGEEASLMVYDIWECMAMGDAYVIVYSVTDKGSFEKASELRVQLRRARDVPIILVGNKSDLVRSREVSVDEGRACAVVFDCKFIETSAALHHNVQALFEGVVRQIRLRR 3q7q A 2.3 BS01 GNP A 1 P100 G101 V102 G103 K104 S105 A106 K204 D206 L207 A234 A235 P11 G12 V13 G14 K15 S16 A17 K95 D97 L98 A125 A126 ? 0003924,0005525 remove_due_to_license_issue P55042 21903096 1 SVYKVLLLGAPGVGKSALARIFGGVEDGHTYDRSIVVDGEEASLMVYDIWEMGDAYVIVYSVTDKGSFEKASELRVQLRRARQTDDVPIILVGNKSDLVRSREVSVDEGRACAVVFDCKFIETSAALHHNVQALFEGVVRQIRLRR 3q8h A 1.75 BS02 AO9 A 1 H36 D58 I59 G60 F63 H36 D58 I59 G60 F63 4.6.1.12 0008299,0008685,0016114,0016829,0019288,0046872 remove_due_to_license_issue Q63T71 24157367 165 MDFRIGQGYDVHQLVPGRPLIIGGVTIPYERGLLGHSDADVLLHAITDALFGAAALGDIGRHFSADSRALLRECASRVAQAGFAIRNVDSTIIAQAPKLAPHIDAMRANIAADLDLPLDRVNVKAKTNEKLGYLGRGEGIEAQAAALVVRE 3q8h A 1.75 BS03 AO9 A 2 L107 A108 A133 L99 A100 A125 4.6.1.12 0008299,0008685,0016114,0016829,0019288,0046872 remove_due_to_license_issue Q63T71 24157367 164 MDFRIGQGYDVHQLVPGRPLIIGGVTIPYERGLLGHSDADVLLHAITDALFGAAALGDIGRHFSADSRALLRECASRVAQAGFAIRNVDSTIIAQAPKLAPHIDAMRANIAADLDLPLDRVNVKAKTNEKLGYLGRGEGIEAQAAALVVRE 3q8h B 1.75 BS01 AO9 A 1 K106 L107 A108 A133 K102 L103 A104 A129 4.6.1.12 0008299,0008685,0016114,0016829,0019288,0046872 remove_due_to_license_issue Q63T71 24157367 165 MDFRIGQGYDVHQLVPGRPLIIGGVTIPYERGLLGHSDADVLLHAITDALFGAAALGDIGRHFPRFKGADSRALLRECASRVAQAGFAIRNVDSTIIAQAPKLAPHIDAMRANIAADLDLPLDRVNVKAKTNEKLGYLGRGEGIEAQAAALVVRE 3q8h B 1.75 BS03 AO9 B 1 H36 D58 I59 G60 F63 H36 D58 I59 G60 F63 4.6.1.12 0008299,0008685,0016114,0016829,0019288,0046872 remove_due_to_license_issue Q63T71 24157367 165 MDFRIGQGYDVHQLVPGRPLIIGGVTIPYERGLLGHSDADVLLHAITDALFGAAALGDIGRHFPRFKGADSRALLRECASRVAQAGFAIRNVDSTIIAQAPKLAPHIDAMRANIAADLDLPLDRVNVKAKTNEKLGYLGRGEGIEAQAAALVVRE 3q92 A 2.8 BS01 XNB A 1 A224 A226 E227 G229 P246 V250 G257 F260 C282 A222 A224 E225 G227 P244 V248 G255 F258 C280 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=<500nM P50053 24900346 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3q92 B 2.8 BS01 XNB B 1 A226 G229 F245 P246 V250 G257 F260 C289 A229 G232 F248 P249 V253 G260 F263 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=<500nM P50053 24900346 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3q96 A 3.1 BS01 0NF A 1 A481 K483 E501 L514 T529 Q530 W531 C532 H574 D594 F595 A33 K35 E53 L66 T81 Q82 W83 C84 H126 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S150 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21341678 1 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP 3qa2 A 2.519 BS01 XNA A 1 A224 A226 P246 V250 A256 G257 F260 A223 A225 P245 V249 A255 G256 F259 G255 A256 G257 D258 G254 A255 G256 D257 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=2400nM P50053 24900346 302 RGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3qa2 B 2.519 BS01 XNA B 1 A224 A226 E227 P246 V250 A256 G257 F260 C289 A227 A229 E230 P249 V253 A259 G260 F263 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=2400nM P50053 24900346 303 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3qaa A 1.4 BS01 G04 A 1 D25 A28 D30 I47 G48 P81 V82 I84 D25 A28 D30 I47 G48 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 22509432 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3qaa B 1.4 BS01 G04 A 1 D125 G127 D129 D130 G148 G149 I150 D25 G27 D29 D30 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 22509432 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3qai A 2.7 BS01 XNN A 1 N107 A224 A226 G229 P246 V250 A256 G257 F260 A285 N105 A222 A224 G227 P244 V248 A254 G255 F258 A283 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=8nM P50053 24900346 302 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3qai B 2.7 BS01 XNN B 1 A226 E227 G229 F245 P246 V250 T253 C289 A229 E230 G232 F248 P249 V253 T256 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=8nM P50053 24900346 303 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3qak A 2.71 BS01 UKA A 1 T88 F168 E169 M177 W246 N253 T256 H264 L267 M270 Y271 I274 S277 H278 T86 F157 E158 M166 W382 N389 T392 H400 L403 M406 Y407 I410 S413 H414 E1011 D1020 E207 D216 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P29274 21393508 1200 IMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYRSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVL 3qaq A 2.9 BS01 QAQ A 1 M804 W812 I831 D841 Y867 E880 I881 V882 A885 M953 I963 D964 M567 W575 I594 D604 Y630 E643 I644 V645 A648 M714 I724 D725 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=100nM, Ki=120nM P48736 21376583 1103 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKETVSLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNHPIALPKHQVRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 3qar A 2.65 BS01 QAR A 1 I831 Y867 I879 V882 K890 M953 I963 D964 I584 Y620 I632 V635 K643 M706 I716 D717 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 21376583 1103 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKESLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISFNADKLTSATNPDKENSMSISILLDNPIALPKHQEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 3qbc A 1.65 BS01 B55 A 1 T43 A44 V46 F54 N56 F123 T45 A46 V48 F56 N58 F125 R83 R92 D95 D97 R85 R94 D97 D99 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656 Kd=10.8uM remove_due_to_license_issue A0A0H3JXR3 22276115 159 SHMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRYK 3qbc A 1.65 BS02 B55 B 1 P109 K110 P111 K112 R83 R92 D95 D97 R85 R94 D97 D99 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656 Kd=10.8uM remove_due_to_license_issue A0A0H3JXR3 22276115 163 SHMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRYK 3qbh A 2.24 BS01 QBH A 1 S10 G13 D32 G34 S35 Y71 T72 Q73 F108 I110 I126 Y198 D228 G230 T231 T232 S13 G16 D35 G37 S38 Y74 T75 Q76 F111 I113 I129 Y188 D218 G220 T221 T222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=0.15uM remove_due_to_license_issue IC50=150nM P56817 21388807 387 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3qbn A 3.5 BS01 E9Z A 1 R137 L139 V147 A160 A213 G216 L263 R12 L14 V22 A35 A88 G91 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T154 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 21671622 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADTLSGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3qc4 A 1.8 BS01 MP7 A 1 A109 K111 Y126 M134 L137 F142 V143 L159 Y161 L212 I221 T222 D223 F224 G225 A227 A34 K36 Y51 M59 L62 F67 V68 L84 Y86 L137 I146 T147 D148 F149 G150 A152 D205 K207 E209 N210 D223 T245 D130 K132 E134 N135 D148 T163 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.002uM remove_due_to_license_issue EC50=1nM O15530 21459573 1 KKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPAAFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3qc9 A 2.7 BS01 ADP A 1 L193 G194 R195 G196 V201 A214 K216 M267 L321 D332 L163 G164 R165 G166 V171 A184 K186 M237 L291 D302 D314 K316 E318 N319 D332 A341 T352 D284 K286 E288 N289 D302 A311 T322 2.7.11.14 0001750,0004672,0004674,0004703,0005515,0005524,0005737,0006468,0007165,0007601,0009966,0016020,0022400,0042995,0046777,0050254,0097381 remove_due_to_license_issue P28327 21265573 700 RDRKYLARLKLPPLSKCEALRESLDLGFEGMCLEQPIGKRLFQQFLRTHEQHGPALQLWKDIEDYDTADDALRPQKAQALRAAYLEPQAQLFCSFLDAETVARARAGAGDGLFQPLLRAVLAHLGQAPFQEFLDSLYFLRFLQWKWLEAQPMGEDWFLDFRVLGRGGFGEVFACQMKATGKLYACKKLNKKRLKKRKGYQGAMVEKKILAKVHSRFIVSLAYAFETKTDLCLVMTIMNGGDIRYHIYNVDEDNPGFQEPRAIFYTAQIVSGLEHLHQRNIIYRDLKPENVLLDDDGNVRISDLGLAVELKAGQTKTKGYAGTPGFMAPELLLGEEYDFSVDYFALGVTLYEMIAARGPFRARGEKVENKELKQRVLEQAVTYPDKFSPASKDFCEALLQKDPEKRLGFRDGSCDGLRTHPLFRDISWRQLEAGMLTPPFVPDVKGVAFEKADTEFFQEFASGTCPIPWQEEMIETGVFGDLNVWRP 3qce B 2.1 BS01 NXY B 1 I950 Y1023 W1026 V1031 V1038 F1041 R1066 Y1070 Q1108 F1111 I125 Y185 W188 V193 V200 F203 R228 Y232 Q270 F273 E955 D1028 C1060 R1066 T1067 Q1104 E130 D190 C222 R228 T229 Q266 3.1.3.48 0004725,0006470,0016311 Ki=2.5uM remove_due_to_license_issue Ki=2500nM, IC50=2500nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRCTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPGKSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENSEEYGNIIVTLKSTKIHACYTVRRFSIRNTKNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILG 3qcf B 2.5 BS01 NXY B 1 I950 Y1023 W1026 V1031 P1032 V1038 F1041 R1066 Y1070 Q1108 F1111 I125 Y185 W188 V193 P194 V200 F203 R228 Y232 Q270 F273 E955 D1028 C1060 R1066 T1067 Q1104 E130 D190 C222 R228 T229 Q266 3.1.3.48 0004725,0006470,0016311 Ki=2.5uM remove_due_to_license_issue Ki=2500nM, IC50=2500nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRCTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPGKSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENSEEYGNIIVTLKSTKIHACYTVRRFSIRNTKNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILG 3qch A 2.4 BS01 NX2 A 1 I950 Y1023 W1026 V1031 P1032 V1038 F1041 R1066 Y1070 Q1108 F1111 I123 Y184 W187 V192 P193 V199 F202 R227 Y231 Q269 F272 E955 D1028 C1060 R1066 T1067 Q1104 E128 D189 C221 R227 T228 Q265 3.1.3.48 0004725,0006470,0016311 ic50=3.3uM remove_due_to_license_issue IC50=3300nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRCTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENSEEYGNIIVTLKSTKIHACYTVRRFSIRNTKQNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILGK 3qci A 2.27 BS01 NX3 A 1 I950 Y1023 W1026 V1031 P1032 V1038 F1041 R1066 Y1070 Q1104 E1107 Q1108 F1111 I123 Y186 W189 V194 P195 V201 F204 R229 Y233 Q267 E270 Q271 F274 E955 D1028 C1060 R1066 T1067 Q1104 E128 D191 C223 R229 T230 Q267 3.1.3.48 0004725,0006470,0016311 ic50=3.8uM remove_due_to_license_issue IC50=3800nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRCTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENSEEYGNIIVTLKSTKIHACYTVRRFSIRNTKVKQNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILG 3qcj A 2.26 BS01 NX4 A 1 I950 Y1023 W1026 V1031 P1032 V1038 F1041 G1065 R1066 Y1070 Q1104 E1107 Q1108 F1111 I124 Y185 W188 V193 P194 V200 F203 G227 R228 Y232 Q266 E269 Q270 F273 E955 D1028 C1060 R1066 T1067 Q1104 E129 D190 C222 R228 T229 Q266 3.1.3.48 0004725,0006470,0016311 ic50=0.5uM remove_due_to_license_issue IC50=500nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRCTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPGSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENSEEYGNIIVTLKSTKIHACYTVRRFSIRNTKQNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILGK 3qck A 2.05 BS01 NX5 A 1 I950 Y1023 W1026 V1031 P1032 V1038 F1041 R1066 Y1070 Q1108 F1111 I123 Y186 W189 V194 P195 V201 F204 R229 Y233 Q271 F274 E955 D1028 C1060 R1066 T1067 Q1104 E128 D191 C223 R229 T230 Q267 3.1.3.48 0004725,0006470,0016311 ic50=5.8uM remove_due_to_license_issue IC50=5800nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRCTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENSEEYGNIIVTLKSTKIHACYTVRRFSIRNTKVKQNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILGKETE 3qcl A 2.4 BS01 NXV A 1 I950 Y1023 W1026 V1031 P1032 V1038 F1041 R1066 T1069 Y1070 E1107 I1110 F1111 I124 Y187 W190 V195 P196 V202 F205 R230 T233 Y234 E271 I274 F275 E955 D1028 C1060 R1066 T1067 Q1104 E129 D192 C224 R230 T231 Q268 3.1.3.48 0004725,0006470,0016311 ic50=4uM remove_due_to_license_issue IC50=4000nM P23470 21882820 2001 MEAIPVKQFVKHIGELYSNNQHGFSEDFEEVQRSTADMNITAEHSNHPENKHKNRYINILAYDHSRVKLRPLPGSKHSDYINANYVDGYNKAKAYIATQGPLKSTFEDFWRMIWEQNTGIIVMITNLVEKGRRKCDQYWPTENTEEYGNIIVTLKSTKIHACYTVRRFSIRNTKVKQNERVVIQYHYTQWPDMGVPEYALPVLTFVRRSSAARMPETGPVLVHCSAGVGRTGTYIVIDSMLQQIKDKSTVNVLGFLKHIRTQRNYLVQTEEQYIFIHDALLEAILGKET 3qcq A 2.501 BS01 3Q0 A 1 V96 A109 K111 S160 A162 L212 T222 D223 V24 A37 K39 S88 A90 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.158uM remove_due_to_license_issue IC50=158nM O15530 21341675 370 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qcs A 2.487 BS01 3Q1 A 1 V96 A109 K111 S160 A162 L212 T222 D223 V24 A37 K39 S88 A90 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.316uM remove_due_to_license_issue IC50=316nM O15530 21341675 370 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qcx A 2.3 BS01 3Q2 A 1 G91 V96 A109 K111 E130 S160 A162 L212 T222 D223 G19 V24 A37 K39 E58 S88 A90 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 ic50=63nM remove_due_to_license_issue IC50=63nM O15530 21341675 370 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qcy A 2.2 BS01 3Q3 A 1 G91 S92 F93 V96 A109 K111 E130 L159 S160 A162 L212 T222 D223 G225 T226 G19 S20 F21 V24 A37 K39 E58 L87 S88 A90 L140 T150 D151 G153 T154 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T162 2.7.11.1 0004672,0004674,0005524,0006468 ic50=20nM remove_due_to_license_issue IC50=20nM O15530 21341675 371 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qd0 A 1.99 BS01 3Q4 A 1 V96 A109 K111 Y126 E130 L159 S160 Y161 A162 L212 T222 D223 G225 V24 A37 K39 Y54 E58 L87 S88 Y89 A90 L140 T150 D151 G153 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T161 2.7.11.1 0004672,0004674,0005524,0006468 ic50=3.16nM remove_due_to_license_issue IC50=333nM O15530 21341675 370 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qd3 A 2.0 BS01 3Q5 A 1 G91 S94 V96 A109 K111 E130 S160 Y161 A162 L212 T222 D223 G21 S24 V26 A39 K41 E60 S90 Y91 A92 L142 T152 D153 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T166 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.00000001M remove_due_to_license_issue IC50=10.0nM O15530 21341675 360 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qd4 A 2.3 BS01 3Q6 A 1 E90 S94 V96 A109 K111 E130 L159 S160 A162 L212 T222 D223 E20 S24 V26 A39 K41 E60 L89 S90 A92 L142 T152 D153 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T163 2.7.11.1 0004672,0004674,0005524,0006468 ic50=6.31nM remove_due_to_license_issue IC50=74nM O15530 21341675 360 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3qdd A 1.79 BS01 94M A 1 A55 G97 M98 L107 F138 W162 A39 G81 M82 L91 F122 W146 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=1.7nM remove_due_to_license_issue Ki=1.7nM, EC50=38nM, IC50=5.1nM P07900 22938030 999 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3qei A 2.178 BS01 dna T 0 D86 D87 S360 P361 I362 K363 Y391 P392 G393 A394 G565 G568 N572 W574 K705 K706 R707 P799 K800 F803 K844 K874 D86 D87 S360 P361 I362 K363 Y391 P392 G393 A394 G565 G568 N572 W574 K705 K706 R707 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22304682 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3qei A 2.178 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22304682 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3qel A 2.6 BS01 QEL B 1 Y109 T110 S132 L135 Y82 T83 S105 L108 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 21677647 1 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 3qel B 2.6 BS01 QEL B 1 Q110 I111 F114 F176 P177 E236 Q70 I71 F74 F136 P137 E196 ? remove_due_to_license_issue IC50=20nM, Ki=11nM Q00960 21677647 1 PPSIGIAVILVGTSDEVAIKDLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPR 3qem A 3.003 BS01 QEM B 1 Y109 T110 R115 S132 L135 Y82 T83 R88 S105 L108 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 21677647 396 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 3qem B 3.003 BS01 QEM B 1 Q110 I111 F114 T174 Y175 F176 P177 E236 Q73 I74 F77 T137 Y138 F139 P140 E199 ? remove_due_to_license_issue IC50=6nM Q00960 21677647 396 PPSIGIAVILVGTSDEVAIKDAHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPR 3qer A 1.96 BS01 dna T 0 D86 D87 S360 P361 I362 K363 Y391 P392 G393 A394 G565 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 D86 D87 S360 P361 I362 K363 Y391 P392 G393 A394 G565 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22304682 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3qer A 1.96 BS02 dna P 0 N284 D621 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 N284 D621 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22304682 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3qes A 1.98 BS01 dna T 0 E219 I253 E254 M256 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 E219 I253 E254 M256 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22304682 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 3qes A 1.98 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22304682 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 3qfq A 2.9001 BS01 dna W 0 S324 A326 Y328 S329 N330 K331 N403 S16 A18 Y20 S21 N22 K23 N95 ? 0003688,0006260 remove_due_to_license_issue E2IPT4 21501625 1 ~ 26 TPVPTDFPIDLSDYLSHAVYSNKTVSCFAIYTTSDKAIELYDKIEKFKVDFKSRHACELGCILLFITLSKHRVSAIKNFCSTFCTISFLICKGVNKMPEMYNNLCKPPYKLLQENKPLL 3qfq A 2.9001 BS02 dna C 0 N330 T332 K378 H379 R380 A383 N22 T24 K70 H71 R72 A75 ? 0003688,0006260 remove_due_to_license_issue E2IPT4 21501625 1 ~ 26 TPVPTDFPIDLSDYLSHAVYSNKTVSCFAIYTTSDKAIELYDKIEKFKVDFKSRHACELGCILLFITLSKHRVSAIKNFCSTFCTISFLICKGVNKMPEMYNNLCKPPYKLLQENKPLL 3qfq B 2.9001 BS01 dna W 0 T332 K378 H379 R380 A383 T24 K70 H71 R72 A75 ? 0003688,0006260 remove_due_to_license_issue E2IPT4 21501625 1 ~ 26 TPVPTDFPIDLSDYLSHAVYSNKTVSCFAIYTTSDKAIELYDKIEKFKVDFKSRHACELGCILLFITLSKHRVSAIKNFCSTFCTISFLICKGVNKMPEMYNNLCKPPYKLLQENKPLLN 3qfq B 2.9001 BS02 dna C 0 S324 A326 Y328 S329 N330 K331 S16 A18 Y20 S21 N22 K23 ? 0003688,0006260 remove_due_to_license_issue E2IPT4 21501625 1 ~ 26 TPVPTDFPIDLSDYLSHAVYSNKTVSCFAIYTTSDKAIELYDKIEKFKVDFKSRHACELGCILLFITLSKHRVSAIKNFCSTFCTISFLICKGVNKMPEMYNNLCKPPYKLLQENKPLLN 3qfq E 2.9001 BS01 dna W 0 S324 Y328 S329 N330 K331 N403 S14 Y18 S19 N20 K21 N93 ? 0003688,0006260 remove_due_to_license_issue E2IPT4 21501625 1 ~ 26 VPTDFPIDLSDYLSHAVYSNKTVSCFAIYTTSDKAIELYDKIEKFKVDFKSRHACELGCILLFITLSKHRVSAIKNFCSTFCTISFLICKGVNKMPEMYNNLCKPPYKLLQENKPLL 3qfq E 2.9001 BS02 dna C 0 K331 T332 K378 H379 R380 A383 N386 K21 T22 K68 H69 R70 A73 N76 ? 0003688,0006260 remove_due_to_license_issue E2IPT4 21501625 1 ~ 26 VPTDFPIDLSDYLSHAVYSNKTVSCFAIYTTSDKAIELYDKIEKFKVDFKSRHACELGCILLFITLSKHRVSAIKNFCSTFCTISFLICKGVNKMPEMYNNLCKPPYKLLQENKPLL 3qfv A 2.65 BS01 NM7 A 1 I82 G83 V90 T137 M153 Y156 F370 I81 G82 V89 T136 M152 Y155 F369 D200 K202 N205 D218 T239 D199 K201 N204 D217 T238 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9Y5S2 21949762 416 SAKVRLKKLEQLLLDGPWRNESALSVETLLDVLVCLYTECSHSALRRDKYVAEFLEWAKPFTQLVKEMQLHREDFEIIKVIGRGAFGEVAVVKMKNTERIYAMKILNKWEMLKRAETACFREERDVLVNGDCQWITALHYAFQDENHLYLVMDYYVGGDLLTLLSKFEDKLPEDMARFYIGEMVLAIDSIHQLHYVHRDIKPDNVLLDVNGHIRLADFGSCLKMNDDGTVQSSVAVGTPDYISPEILQAMEDGMGKYGPECDWWSLGVCMYEMLYGETPFYAESLVETYGKIMNHEERFQFPSHVTDVSEEAKDLIQRLICSRERRLGQNGIEDFKKHAFFEGLNWENIRNLEAPYIPDVSSPSDTSNFDVSGLHLPFIGFTFTTESCFSDRGSL 3qfy A 2.3 BS02 IFM A 1 R367 D368 W488 D490 E659 F664 R367 D368 W488 D490 E659 F664 2.4.1.20 0003824,0005975,0016757,0030246 remove_due_to_license_issue O66264 1903 MRYGHFDDAAREYVITTPHTPYPWINYLGSEQFFSLLSHQAGGYSFYRDAKMRRLTRYRYNNIPADAGGRYLYVNDGGDVWTPSWLPVKADLDHFEARHGLGYSRITGERNGLKVETLFFVPLGENAEVQKVTVTNTSDAPKTATLFSFVEFCLWNAQDDQTNYQRNLSIGEVEVEQDGPHGSAIYHKTEYRERRDHYAVFGVNTRADGFDTDRDTFVGAYNSLGEASVPRAGKSADSVASGWYPIGSHSVAVTLQPGESRDLVYVLGYLENPDEEKWADDAHQVVNKAPAHALLGRFATSEQVDAALEALNSYWTNLLSTYSVSSTDEKLDRMVNIWNQYQCMVTFNMSRSASFFETGIGRGMGFRDSNQDLLGFVHLIPERARERIIDIASTQFADGSAYHQYQPLTKRGNNDIGSGFNDDPLWLIAGVAAYIKESGDWGILDEPVPFDNEPGSEVPLFEHLTRSFQFTVQNRGPHGLPLIGRADWNDCLNLNCFSTTPGESFQTTENQAGGVAESVFIAAQFVLYGAEYATLAERRGLADVATEARKYVDEVRAAVLEHGWDGQWFLRAYDYYGNPVGTDAKPEGKIWIEPQGFAVMAGIGVGEGPDDADAPAVKALDSVNEMLGTPHGLVLQYPAYTTYQIELGEVSTYPPGYKENGGIFCHNNPWVIIAETVVGRGAQAFDYYKRITPAYREDISDTHKLEPYVYAQMIAGKEAVRAGEAKNSWLTGTAAWNFVAVSQYLLGVRPDYDGLVVDPQIGPDVPSYTVTRVARGATYEITVTNSGAPGARASLTVDGAPVDGRTVPYAPAGSTVRVEVTV 3qfy B 2.3 BS02 IFM B 1 R367 D368 W488 N489 D490 E659 F664 R367 D368 W488 N489 D490 E659 F664 2.4.1.20 0003824,0005975,0016757,0030246 remove_due_to_license_issue O66264 2903 MRYGHFDDAAREYVITTPHTPYPWINYLGSEQFFSLLSHQAGGYSFYRDAKMRRLTRYRYNNIPADAGGRYLYVNDGGDVWTPSWLPVKADLDHFEARHGLGYSRITGERNGLKVETLFFVPLGENAEVQKVTVTNTSDAPKTATLFSFVEFCLWNAQDDQTNYQRNLSIGEVEVEQDGPHGSAIYHKTEYRERRDHYAVFGVNTRADGFDTDRDTFVGAYNSLGEASVPRAGKSADSVASGWYPIGSHSVAVTLQPGESRDLVYVLGYLENPDEEKWADDAHQVVNKAPAHALLGRFATSEQVDAALEALNSYWTNLLSTYSVSSTDEKLDRMVNIWNQYQCMVTFNMSRSASFFETGIGRGMGFRDSNQDLLGFVHLIPERARERIIDIASTQFADGSAYHQYQPLTKRGNNDIGSGFNDDPLWLIAGVAAYIKESGDWGILDEPVPFDNEPGSEVPLFEHLTRSFQFTVQNRGPHGLPLIGRADWNDCLNLNCFSTTPGESFQTTENQAGGVAESVFIAAQFVLYGAEYATLAERRGLADVATEARKYVDEVRAAVLEHGWDGQWFLRAYDYYGNPVGTDAKPEGKIWIEPQGFAVMAGIGVGEGPDDADAPAVKALDSVNEMLGTPHGLVLQYPAYTTYQIELGEVSTYPPGYKENGGIFCHNNPWVIIAETVVGRGAQAFDYYKRITPAYREDISDTHKLEPYVYAQMIAGKEAVRAGEAKNSWLTGTAAWNFVAVSQYLLGVRPDYDGLVVDPQIGPDVPSYTVTRVARGATYEITVTNSGAPGARASLTVDGAPVDGRTVPYAPAGSTVRVEVTV 3qfz A 2.39 BS02 NOJ A 1 R362 R367 D368 W488 D490 E659 F664 R362 R367 D368 W488 D490 E659 F664 2.4.1.20 0003824,0005975,0016757,0030246 remove_due_to_license_issue O66264 1903 MRYGHFDDAAREYVITTPHTPYPWINYLGSEQFFSLLSHQAGGYSFYRDAKMRRLTRYRYNNIPADAGGRYLYVNDGGDVWTPSWLPVKADLDHFEARHGLGYSRITGERNGLKVETLFFVPLGENAEVQKVTVTNTSDAPKTATLFSFVEFCLWNAQDDQTNYQRNLSIGEVEVEQDGPHGSAIYHKTEYRERRDHYAVFGVNTRADGFDTDRDTFVGAYNSLGEASVPRAGKSADSVASGWYPIGSHSVAVTLQPGESRDLVYVLGYLENPDEEKWADDAHQVVNKAPAHALLGRFATSEQVDAALEALNSYWTNLLSTYSVSSTDEKLDRMVNIWNQYQCMVTFNMSRSASFFETGIGRGMGFRDSNQDLLGFVHLIPERARERIIDIASTQFADGSAYHQYQPLTKRGNNDIGSGFNDDPLWLIAGVAAYIKESGDWGILDEPVPFDNEPGSEVPLFEHLTRSFQFTVQNRGPHGLPLIGRADWNDCLNLNCFSTTPGESFQTTENQAGGVAESVFIAAQFVLYGAEYATLAERRGLADVATEARKYVDEVRAAVLEHGWDGQWFLRAYDYYGNPVGTDAKPEGKIWIEPQGFAVMAGIGVGEGPDDADAPAVKALDSVNEMLGTPHGLVLQYPAYTTYQIELGEVSTYPPGYKENGGIFCHNNPWVIIAETVVGRGAQAFDYYKRITPAYREDISDTHKLEPYVYAQMIAGKEAVRAGEAKNSWLTGTAAWNFVAVSQYLLGVRPDYDGLVVDPQIGPDVPSYTVTRVARGATYEITVTNSGAPGARASLTVDGAPVDGRTVPYAPAGSTVRVEVTV 3qfz B 2.39 BS02 NOJ B 1 R362 R367 D368 W488 N489 D490 E659 F664 R362 R367 D368 W488 N489 D490 E659 F664 2.4.1.20 0003824,0005975,0016757,0030246 remove_due_to_license_issue O66264 2903 MRYGHFDDAAREYVITTPHTPYPWINYLGSEQFFSLLSHQAGGYSFYRDAKMRRLTRYRYNNIPADAGGRYLYVNDGGDVWTPSWLPVKADLDHFEARHGLGYSRITGERNGLKVETLFFVPLGENAEVQKVTVTNTSDAPKTATLFSFVEFCLWNAQDDQTNYQRNLSIGEVEVEQDGPHGSAIYHKTEYRERRDHYAVFGVNTRADGFDTDRDTFVGAYNSLGEASVPRAGKSADSVASGWYPIGSHSVAVTLQPGESRDLVYVLGYLENPDEEKWADDAHQVVNKAPAHALLGRFATSEQVDAALEALNSYWTNLLSTYSVSSTDEKLDRMVNIWNQYQCMVTFNMSRSASFFETGIGRGMGFRDSNQDLLGFVHLIPERARERIIDIASTQFADGSAYHQYQPLTKRGNNDIGSGFNDDPLWLIAGVAAYIKESGDWGILDEPVPFDNEPGSEVPLFEHLTRSFQFTVQNRGPHGLPLIGRADWNDCLNLNCFSTTPGESFQTTENQAGGVAESVFIAAQFVLYGAEYATLAERRGLADVATEARKYVDEVRAAVLEHGWDGQWFLRAYDYYGNPVGTDAKPEGKIWIEPQGFAVMAGIGVGEGPDDADAPAVKALDSVNEMLGTPHGLVLQYPAYTTYQIELGEVSTYPPGYKENGGIFCHNNPWVIIAETVVGRGAQAFDYYKRITPAYREDISDTHKLEPYVYAQMIAGKEAVRAGEAKNSWLTGTAAWNFVAVSQYLLGVRPDYDGLVVDPQIGPDVPSYTVTRVARGATYEITVTNSGAPGARASLTVDGAPVDGRTVPYAPAGSTVRVEVTV 3qg9 A 2.25 BS01 rna B 0 E208 F242 N244 Y245 Q248 R288 H326 K360 Y361 R364 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S554 K557 E41 F75 N77 Y78 Q81 R121 H159 K193 Y194 R197 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 Q337 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 21372189 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3qgb A 2.4 BS01 rna B 0 K201 E208 F242 N244 Y245 Q248 Y288 Q291 H326 K360 Y361 R364 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 K557 K34 E41 F75 N77 Y78 Q81 Y121 Q124 H159 K193 Y194 R197 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 K390 ? 0003723 remove_due_to_license_issue Q09312 21372189 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACYVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3qgc A 1.9 BS01 rna B 0 K201 E208 F242 N244 Y245 Y288 Q291 N323 H326 K360 Y361 R364 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S554 K557 K34 E41 F75 N77 Y78 Y121 Q124 N156 H159 K193 Y194 R197 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 Q337 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 21372189 1 ~ 9 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACYVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3qgw B 2.1 BS01 L7A B 1 I369 V377 A389 K391 F435 E436 F437 M438 G441 L489 S499 I12 V20 A32 K34 F78 E79 F80 M81 G84 L132 S142 D482 A484 R486 N487 D500 P521 D125 A127 R129 N130 D143 P145 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=1.3uM remove_due_to_license_issue Ki=1300nM Q08881 21391610 1 IDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIKEGSMSEDDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIA 3qgy B 2.1 BS01 L7O B 1 V377 A389 K391 F435 E436 F437 M438 E439 G441 L489 D500 V22 A34 K36 F80 E81 F82 M83 E84 G86 L134 D145 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P150 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=0.016uM remove_due_to_license_issue Ki=16nM Q08881 21391610 1 MVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIKEGSMSEDDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIA 3qi1 A 2.3 BS01 C6A A 1 D38 G40 P76 Y77 T78 F114 Y204 K230 D234 G236 D36 G38 P74 Y75 T76 F112 Y195 K221 D225 G227 D38 S41 N43 A45 Y77 D234 T237 D36 S39 N41 A43 Y75 D225 T228 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 23856050 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3qi3 A 2.3 BS01 PDB A 1 H252 L420 Y424 A452 E453 F456 H72 L240 Y244 A272 E273 F276 3.1.4.35 0004114,0004115,0004117,0005515,0005654,0005737,0005783,0005794,0005829,0005886,0007165,0008081,0010613,0016787,0019933,0032587,0042383,0042995,0043204,0046068,0046069,0046872,0047555,0048101,0048471,1900273,2000178 remove_due_to_license_issue O76083 21483814 600 PTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAEIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 3qi5 A 2.2 BS01 dna C 0 Y127 H136 M149 Y159 I161 Y162 Y165 N169 L180 R197 K202 G217 P218 S219 K220 G263 Y48 H57 M70 Y80 I82 Y83 Y86 N90 L101 R118 K123 G133 P134 S135 K136 G179 3.2.2.21 0003677,0003824,0003905,0006284 remove_due_to_license_issue P29372 21349833 1 ~ 13 GPHMTRLGLEFFDQPAVPLARAFLGQVLVRRLPNGTELRGRIVETEAYLGPEDEAAHSRGGRQTPRNRGMFMKPGTLYVYIIYGMYFCMNISSQGDGACVLLRALEPLEGLETMRQLRSTLRKVLKDRELCSGPSKLCQALAINKSFDQRDLAQDEAVWLERGPLEPSEPAVVAAARVGVEWARKPLRFYVRGSPWVSVVDRVAEQ 3qi5 A 2.2 BS02 dna D 0 T143 R145 Y162 G163 M164 K229 T64 R66 Y83 G84 M85 K145 3.2.2.21 0003677,0003824,0003905,0006284 remove_due_to_license_issue P29372 21349833 14 ~ 26 GPHMTRLGLEFFDQPAVPLARAFLGQVLVRRLPNGTELRGRIVETEAYLGPEDEAAHSRGGRQTPRNRGMFMKPGTLYVYIIYGMYFCMNISSQGDGACVLLRALEPLEGLETMRQLRSTLRKVLKDRELCSGPSKLCQALAINKSFDQRDLAQDEAVWLERGPLEPSEPAVVAAARVGVEWARKPLRFYVRGSPWVSVVDRVAEQ 3qi5 B 2.2 BS01 dna E 0 Y127 H136 M149 Y159 I161 Y162 Y165 C167 N169 L180 R182 R197 R201 G217 P218 S219 K220 G263 Y48 H57 M70 Y80 I82 Y83 Y86 C88 N90 L101 R103 R118 R122 G136 P137 S138 K139 G182 3.2.2.21 0003677,0003824,0003905,0006284 remove_due_to_license_issue P29372 21349833 1 ~ 13 GPHMTRLGLEFFDQPAVPLARAFLGQVLVRRLPNGTELRGRIVETEAYLGPEDEAAHSRGGRQTPRNRGMFMKPGTLYVYIIYGMYFCMNISSQGDGACVLLRALEPLEGLETMRQLRSTLRKGTRVLKDRELCSGPSKLCQALAINKSFDQRDLAQDEAVWLERGPLEPSEPAVVAAARVGVAGEWARKPLRFYVRGSPWVSVVDRVAE 3qi5 B 2.2 BS02 dna F 0 T143 P144 R145 I160 Y162 G163 M164 K229 T64 P65 R66 I81 Y83 G84 M85 K148 3.2.2.21 0003677,0003824,0003905,0006284 remove_due_to_license_issue P29372 21349833 14 ~ 26 GPHMTRLGLEFFDQPAVPLARAFLGQVLVRRLPNGTELRGRIVETEAYLGPEDEAAHSRGGRQTPRNRGMFMKPGTLYVYIIYGMYFCMNISSQGDGACVLLRALEPLEGLETMRQLRSTLRKGTRVLKDRELCSGPSKLCQALAINKSFDQRDLAQDEAVWLERGPLEPSEPAVVAAARVGVAGEWARKPLRFYVRGSPWVSVVDRVAE 3qin A 1.6967 BS03 P1Y A 1 D443 E478 D498 A538 H539 D18 E53 D73 A116 H117 D443 G444 E478 D498 H539 D549 D18 G19 E53 D73 H117 D127 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.1.26.4,3.4.23.16 0003676,0004523 Kd=136nM remove_due_to_license_issue P04585,P0A7Y4 21464257 700 MYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIITQWIHNWKVKNVDLVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRKV 3qio A 1.4011 BS03 QID A 1 D443 D498 H539 R557 D18 D73 H116 R134 D443 G444 E478 D498 H539 D549 D18 G19 E53 D73 H116 D126 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.1.26.4,3.4.23.16 0003676,0004523 Kd=144nM remove_due_to_license_issue P04585,P0A7Y4 21464257 700 MYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIITQWIHNWKKNVDLVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRKV 3qip A 2.0926 BS03 P4Y A 1 D443 E478 D498 A538 H539 D441 E476 D496 A536 H537 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 21464257 900 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGI 3qiy A 2.3 BS02 QI1 A 1 V68 P69 F163 F194 H223 E224 H227 E262 R363 Y366 N368 V65 P66 F160 F191 H208 E209 H212 E234 R333 Y336 N338 H223 E224 H227 E262 R363 H208 E209 H212 E234 R333 0004222,0006508,0008270 Ki=4.6uM remove_due_to_license_issue 21434688 432 GFVNKQFNYKDPVNGVDIAYIKIPNAGQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPAKQVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEEGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGTTASLQYMKNVFKEKYLLSTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKNFTG 3qiz A 2.0 BS02 QI2 A 1 V68 P69 F163 F194 H223 E224 H227 E262 R363 Y366 L367 N368 V67 P68 F162 F193 H212 E213 H216 E240 R341 Y344 L345 N346 H223 E224 H227 E262 R363 H212 E213 H216 E240 R341 0004222,0006508,0008270 Ki=6.1uM remove_due_to_license_issue 21434688 432 GFVNKQFNYKDPVNGVDIAYIKIPNAGQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPPEAKQVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEEGAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFKLEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGTTASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKNFTG 3qj0 A 2.301 BS02 QI3 A 1 P69 F163 F194 H223 E224 H227 E262 Y366 F369 P68 F162 F193 H211 E212 H215 E237 Y341 F344 H223 E224 H227 E262 R363 H211 E212 H215 E237 R338 0004222,0006508,0008270 Ki=6.3uM remove_due_to_license_issue 21434688 432 GFVNKQFNYKDPVNGVDIAYIKIPNAGQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPPEAKQVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEEAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGTTASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKNFT 3qj9 A 2.3 BS01 QJ9 A 1 L192 S193 F194 I238 L404 I407 L429 M436 G485 T488 I491 W531 L164 S165 F166 I210 L376 I379 L401 M408 G457 T460 I463 W503 K142 S217 S218 T236 I238 G239 G240 S241 F244 K114 S189 S190 T208 I210 G211 G212 S213 F216 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 ic50=951nM remove_due_to_license_issue IC50=60nM P97612 21502526 600 ELETGRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMLSFDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSAGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNSMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAISYTVLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQ 3qk0 A 2.85 BS01 QK0 A 1 P810 W812 I831 K833 Y867 I881 V882 A885 M953 I963 D964 P550 W552 I571 K573 Y607 I621 V622 A625 M693 I703 D704 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=4.7nM P48736 21332118 1103 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 3qk5 A 2.2 BS01 QK5 A 1 L192 S193 I238 G239 G240 S241 F244 L404 I407 M436 G485 T488 I491 W531 L164 S165 I210 G211 G212 S213 F216 L376 I379 M408 G457 T460 I463 W503 K142 S217 S218 T236 I238 G239 G240 S241 F244 K114 S189 S190 T208 I210 G211 G212 S213 F216 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 ic50=0.018uM remove_due_to_license_issue IC50=18nM P97612 21392988 600 ELETGRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMLSFDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSAGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNSMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAISYTVLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQ 3qkd A 2.02 BS01 HI0 A 1 A93 E96 F97 R100 Y101 F105 V126 E129 L130 G138 R139 V141 Y195 A36 E39 F40 R43 Y44 F48 V69 E72 L73 G81 R82 V84 Y138 ? 0042981 ic50=3nM remove_due_to_license_issue IC50=7nM, Kd=4.2nM Q07817 21366295 218 SNRELVVDFLSYKLSQKGYSWSQFSSEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGN 3qkk A 2.3 BS02 SMH A 1 G157 K158 G159 F161 G162 V164 A177 M227 E278 M281 T291 D292 F438 G14 K15 G16 F18 G19 V21 A34 M84 E135 M138 T148 D149 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P31749 21392984 1 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITIMECVDSERRPHFPQFDYSASS 3qkl A 1.9 BS02 SMR A 1 G157 K158 G159 F161 G162 K163 V164 A177 M227 Y229 E278 M281 T291 D292 G14 K15 G16 F18 G19 K20 V21 A34 M84 Y86 E135 M138 T148 D149 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P31749 21392984 1 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITRPHFPQFDYSASS 3qkm A 2.2 BS01 SM9 A 1 G157 K158 G159 F161 G162 K163 V164 A177 E191 M227 A230 E234 E278 M281 D292 F438 G14 K15 G16 F18 G19 K20 V21 A34 E48 M84 A87 E91 E135 M138 D149 F295 D274 K276 N279 D292 T312 D131 K133 N136 D149 T169 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.038uM remove_due_to_license_issue P31749 21420856 1 RVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITITPSMECVDSERRPHFPQFDYSASS 3qkv B 3.1 BS01 QKV B 1 L192 S193 I238 G239 S241 F381 T488 L158 S159 I204 G205 S207 F347 T454 K142 S217 S218 T236 I238 G239 G240 S241 F244 K108 S183 S184 T202 I204 G205 G206 S207 F210 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 21502526 580 QKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMLSFDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSAGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNSMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAISYTVLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQKQ 3qlb A 3.26 BS01 EFE A 1 F92 P244 R245 Y329 F331 Y370 F70 P222 R223 Y307 F309 Y348 ? 0009279,0015343,0015891,0038023 remove_due_to_license_issue C5I2D9 21902256 701 PDSATGPQAGYVAKRSLSGTKTDASLSEIPQSISVITRDQMDAQQVQSVNEALRYTAGVQANTTAASQRFDTLSIRGFDVTTGMLRDGLKGNTAQAWPKVEAYGLERIDVLKGPASVLFGQNSPGGVVNQISKRPLDKPFHEVQIQGGSFDRAQGQFDFSGPLDDEGQFLYRLVGLERDSGTQFDHIKDDKQYFAPSFTWKPNDDTSLTLLADYTQDTFGAPRVFLPAQGTLLGNPNGKVRHNVFLDEPGLDNDRTQYSLGYLLEHRLNDVWSLNSSARYGHVNLLTNTASGMSLAPDLRTLNRAAYRFRIVGDTYSLDNNAQARWNLGSTQMVSLLGIDYRRTREDYYLRGGSASPIDIYNPVHHHHGVFDPSTPFTNTVQRADQVGVYAQQQFTFDEHWVLTVGGRQDRSSARTDNRMNDSGSKQDDEKFTYRTGLVYLADNGLAPYISYSTSFDPVLGTNFYGTPYKPTSAKQSEVGVKYQPPGIDSYITLSLFDLTQENVLTTDPAQRLNKIQTGEINVRGIELEGKASLARGLDLLAALTYNDAEVSKSNNPLEKGKRPTDTPEKMASLWADYTLPEGPLSGLGFGAGVRYIGSTEADAANTQRVPSYTLLDAAVHYDFDKLIPAAKGLRLAVNATNLTDKHYYEGCSLTNCSAGYDRSVIASLRYRW 3qmb A 2.06 BS01 dna B 0 K202 I203 R204 K35 I36 R37 ? 0003677,0008270 remove_due_to_license_issue Q9P0U4 21407193 1 ~ 12 RSARMCGECEACRRTEDCGHCDFCRDMKKFGGPNKIRQKCRLRQCQLRARESYK 3qmb A 2.06 BS02 dna C 0 R171 R204 Q205 K206 R210 R217 R4 R37 Q38 K39 R43 R50 ? 0003677,0008270 remove_due_to_license_issue Q9P0U4 21407193 1 ~ 12 RSARMCGECEACRRTEDCGHCDFCRDMKKFGGPNKIRQKCRLRQCQLRARESYK 3qmh A 2.5 BS01 dna B 0 R167 R200 Q201 K202 R213 R2 R35 Q36 K37 R48 ? 0003677,0008270 remove_due_to_license_issue Q9P0U4 21407193 1 ~ 12 ARMCGECEACRRTEDCGHCDFCRDMKKFGGPNKIRQKCRLRQCQLRARESYKY 3qmh A 2.5 BS02 dna C 0 I199 R200 Q201 S215 I34 R35 Q36 S50 ? 0003677,0008270 remove_due_to_license_issue Q9P0U4 21407193 1 ~ 12 ARMCGECEACRRTEDCGHCDFCRDMKKFGGPNKIRQKCRLRQCQLRARESYKY 3qmi A 2.1 BS01 dna B 0 R167 R200 Q201 K202 R213 R2 R35 Q36 K37 R48 ? 0003677,0008270 remove_due_to_license_issue Q9P0U4 21407193 1 ~ 12 ARMCGECEACRRTEDCGHCDFCRDMKKFGGPNKIRQKCRLRQCQLRARESYK 3qmi A 2.1 BS02 dna C 0 K198 I199 R200 K33 I34 R35 ? 0003677,0008270 remove_due_to_license_issue Q9P0U4 21407193 1 ~ 12 ARMCGECEACRRTEDCGHCDFCRDMKKFGGPNKIRQKCRLRQCQLRARESYK 3qmk A 2.21 BS01 SGN C 1 H307 K422 H16 K131 ? 0016020 remove_due_to_license_issue P51693 21930949 1 DGVDIYFGMPGEISEHEGFLRAKMDLEERRMRQINEVMREWAMADNQSKNLPKADRQALNEHFQSILQTLEEQVSGERQRLVETHATRVIALINDQRRAALEGFLAALQADPPQAERVLLALRRYLRAEQKEQRHTLRHYQHVAAVDPEKAQQMRFQVHTHLQVIEERVNQSLGLLDQNPHLAQELRPQIQELLH 3qmk A 2.21 BS02 IDS C 1 H307 H426 R429 H16 H135 R138 ? 0016020 remove_due_to_license_issue P51693 21930949 2 DGVDIYFGMPGEISEHEGFLRAKMDLEERRMRQINEVMREWAMADNQSKNLPKADRQALNEHFQSILQTLEEQVSGERQRLVETHATRVIALINDQRRAALEGFLAALQADPPQAERVLLALRRYLRAEQKEQRHTLRHYQHVAAVDPEKAQQMRFQVHTHLQVIEERVNQSLGLLDQNPHLAQELRPQIQELLH 3qmk A 2.21 BS03 SGN C 2 R429 H430 H433 R138 H139 H142 ? 0016020 remove_due_to_license_issue P51693 21930949 3 DGVDIYFGMPGEISEHEGFLRAKMDLEERRMRQINEVMREWAMADNQSKNLPKADRQALNEHFQSILQTLEEQVSGERQRLVETHATRVIALINDQRRAALEGFLAALQADPPQAERVLLALRRYLRAEQKEQRHTLRHYQHVAAVDPEKAQQMRFQVHTHLQVIEERVNQSLGLLDQNPHLAQELRPQIQELLH 3qmk A 2.21 BS04 IDS C 2 F310 V373 H433 F19 V82 H142 ? 0016020 remove_due_to_license_issue P51693 21930949 4 DGVDIYFGMPGEISEHEGFLRAKMDLEERRMRQINEVMREWAMADNQSKNLPKADRQALNEHFQSILQTLEEQVSGERQRLVETHATRVIALINDQRRAALEGFLAALQADPPQAERVLLALRRYLRAEQKEQRHTLRHYQHVAAVDPEKAQQMRFQVHTHLQVIEERVNQSLGLLDQNPHLAQELRPQIQELLH 3qnd A 2.4 BS02 SIA A 1 Y312 P317 D318 K345 Y131 P136 D137 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 21648036 1 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 3qnd C 2.4 BS02 SIA C 1 Y312 P317 P320 K345 Y130 P135 P138 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 21648036 1 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 3qnn A 1.92 BS01 dna T 0 E219 I253 Y257 R260 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 N572 K705 R707 S784 N786 K800 F803 K844 K874 E219 I253 Y257 R260 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 N572 K705 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22616982 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 3qnn A 1.92 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22616982 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 3qno A 1.88 BS01 dna T 0 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 N572 K705 K706 R707 K800 F803 K844 K874 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 N572 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22616982 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 3qno A 1.88 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22616982 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 3qo3 A 2.15 BS01 ATP A 1 Y25 G29 T61 Y21 G25 T57 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 23226421 66 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3qo3 B 2.15 BS01 ATP A 1 I30 L32 I26 L28 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 23226421 66 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3qo3 B 2.15 BS02 ATP B 1 Y25 G29 K31 T61 Y21 G25 K27 T57 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 23226421 66 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3qo9 A 2.6 BS01 QO9 A 1 K102 K103 V106 Y181 Y183 Y188 F227 W229 L234 P236 Y318 K103 K104 V107 Y182 Y184 Y189 F228 W230 L235 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 21446702 556 VPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAISQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 3qox A 2.3 BS01 SAH A 1 P133 G137 E138 T139 D161 G163 S164 E186 K187 D222 F223 N241 F245 P127 G131 E132 T133 D155 G157 S158 E180 K181 D216 F217 N235 F239 2.1.1.360 0031151,0051726 Ki=0.27uM remove_due_to_license_issue Ki=160nM, IC50=600nM, Kd=150nM Q8TEK3 21564555 417 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLKNP 3qpn A 2.0 BS02 PFK A 1 Y683 F686 P702 M703 G715 Q716 F719 Y231 F234 P250 M251 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=17nM remove_due_to_license_issue IC50=17nM Q9QYJ6 21650160 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3qpo A 1.8 BS02 PFR A 1 Y683 M703 G715 Q716 F719 V723 Y231 M251 G263 Q264 F267 V271 3.1.4.17 0004114,0007165,0008081 ic50=247nM remove_due_to_license_issue IC50=247nM Q9QYJ6 21650160 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3qpp A 1.8 BS02 PFW A 1 Y683 F686 P702 M703 G715 Q716 F719 V723 Y231 F234 P250 M251 G263 Q264 F267 V271 3.1.4.17 0004114,0007165,0008081 ic50=12nM remove_due_to_license_issue IC50=12nM Q9QYJ6 21650160 999 NLPARICRDIELFHFDIGPFENMWPGIFVYMIHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIR 3qqa A 2.2 BS01 TCH A 1 H72 F103 I115 H67 F98 I110 ? 0003677 Kd=1.5uM remove_due_to_license_issue Q7B8P6 21328631 211 TPSQKVLARQEKIKAVALELFLTKGYQETSLSDIIKLSGGSYSNIYDGFKSKEGLFFEILDDICKKHFHLIYSKTQEIKNGTLKEILTSFGLAFIEIFNQPEAVAFGKIIYSQVYDKDRHLANWIENNQQNFSYNILMGFFKQQNNSYMKKNAEKLAVLFCTMLKEPYHHLNVLINAPLKNKKEQKEHVEFVVNVFLNGI 3qqk A 1.86 BS01 X02 A 1 I10 A31 F82 L83 L134 D145 I10 A31 F78 L79 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=15000nM P24941 23600925 497 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qqs A 1.97 BS04 17C A 1 P180 H183 Y186 R187 A190 R193 R194 P156 H159 Y162 R163 A166 R169 R170 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 404 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3qqu A 2.9 BS01 01P A 1 Q1004 V1010 A1028 E1077 M1079 M1139 D1150 M1153 Q17 V23 A41 E90 M92 M142 D153 M156 D1132 R1136 N1137 D1150 E1159 D135 R139 N140 D153 E162 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=2.4nM P08069 21414779 1 EWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEEN 3qri A 2.1 BS01 919 A 1 L248 A269 K271 E286 M290 E316 F317 M318 G321 H361 L370 A380 D381 F382 L25 A46 K48 E63 M67 E93 F94 M95 G98 H138 L147 A157 D158 F159 D363 A365 R367 N368 D381 P402 D140 A142 R144 N145 D158 P179 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.8nM remove_due_to_license_issue P00519 21481795 500 SMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ 3qrj A 1.82 BS01 919 A 1 L248 A269 E282 E286 M290 I315 F317 M318 L370 A380 D381 F382 L15 A36 E44 E48 M52 I77 F79 M80 L132 A142 D143 F144 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4nM remove_due_to_license_issue P00519 21481795 2 KWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETM 3qrk A 2.3 BS01 9DP A 1 A269 K271 E282 E286 M290 V299 I313 T315 A380 D381 F382 A43 K45 E56 E60 M64 V73 I87 T89 A154 D155 F156 D363 A365 R367 N368 D381 P402 D137 A139 R141 N142 D155 P176 2.7.10.2 0004672,0004713,0005524,0006468 ic50=57nM remove_due_to_license_issue P00519 21481795 1 PSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETM 3qs1 A 3.1 BS01 006 A 1 D32 G34 Y75 V76 S77 D215 G217 T218 S219 D33 G35 Y76 V77 S78 D213 G215 T216 S217 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D213 T216 3.4.23.38 0004190,0006508 remove_due_to_license_issue IC50=280nM P39898 21521654 330 AGDSVTLNDVANVMYYGEAQIGDNKQKFAFIFDTGSANLWVPSAQCNTIGCKTKNLYDSNKSKTYEKDGTKVEMNYVSGTVSGFFSKDIVTIANLSFPYKFIEVTDTNGFEPAYTLGQFDGIVGLGWKDLSIGSVDPVVVELKNQNKIEQAVFTFYLPFDDKHKGYLTIGGIEDRFYEGQLTYEKLNHDLYWQVDLDLHFGNLTVEKATAIVDSGTSSITAPTEFLNKFFEGLDVVKIPFLPLYITTCNNPKLPTLEFRSATNVYTLEPEYYLQQIFDFGISLCMVSIIPVDLNKNTFILGDPFMRKYFTVFDYDNHTVGFALAKKK 3qs1 B 3.1 BS01 006 B 1 D32 G34 N74 Y75 V76 S77 L128 D215 G217 T218 S219 I300 D33 G35 N75 Y76 V77 S78 L130 D213 G215 T216 S217 I299 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D213 T216 3.4.23.38 0004190,0006508 remove_due_to_license_issue IC50=280nM P39898 21521654 330 AGDSVTLNDVANVMYYGEAQIGDNKQKFAFIFDTGSANLWVPSAQCNTIGCKTKNLYDSNKSKTYEKDGTKVEMNYVSGTVSGFFSKDIVTIANLSFPYKFIEVTDTNGFEPAYTLGQFDGIVGLGWKDLSIGSVDPVVVELKNQNKIEQAVFTFYLPFDDKHKGYLTIGGIEDRFYEGQLTYEKLNHDLYWQVDLDLHFGNLTVEKATAIVDSGTSSITAPTEFLNKFFEGLDVVKIPFLPLYITTCNNPKLPTLEFRSATNVYTLEPEYYLQQIFDFGISLCMVSIIPVDLNKNTFILGDPFMRKYFTVFDYDNHTVGFALAKKK 3qs4 A 2.631 BS01 TRP A 1 A22 G24 G26 N27 Y108 F253 T254 S256 V259 A18 G20 G22 N23 Y104 F246 T247 S249 V252 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 21952050 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGVGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3qs4 A 2.631 BS02 TRP A 2 R30 G249 F253 D404 G408 T409 R26 G242 F246 D397 G401 T402 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 21952050 602 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGVGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3qs4 A 2.631 BS03 TRP A 3 R11 D272 Q273 D274 G439 R7 D265 Q266 D267 G432 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 21952050 603 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGVGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 3qs5 A 2.6 BS01 TRP A 1 N21 A22 G24 G26 F253 T254 S256 F259 A261 S355 A358 Q359 N17 A18 G20 G22 F247 T248 S250 F253 A255 S349 A352 Q353 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 21952050 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAQMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3qs6 A 2.801 BS01 TRP A 1 N21 A22 G24 G26 Y108 F253 T254 S256 V259 S355 Q359 N17 A18 G20 G22 Y104 F247 T248 S250 V253 S349 Q353 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 21952050 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGVGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAQMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 3qs8 A 2.0 BS04 17D A 1 N138 A179 P180 Y186 A190 R193 R194 N114 A155 P156 Y162 A166 R169 R170 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 600 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3qs8 A 2.0 BS05 17D A 2 M86 G107 N138 A179 Y186 R193 L205 G206 M62 G83 N114 A155 Y162 R169 L181 G182 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 602 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3qsb A 1.9 BS01 743 A 1 T172 G174 V247 V360 M362 T172 G174 V247 V360 M362 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 ic50=8.3uM remove_due_to_license_issue P0A988 21604761 367 MKFTVEREHLLKPLQQVSGPLGGRPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 3qsd A 1.3 BS01 074 A 1 Q94 G98 C100 W101 G143 G144 L146 H180 H181 G269 H270 W292 Q24 G28 C30 W31 G73 G74 L76 H110 H111 G199 H200 W222 Q94 C100 H270 N290 Q24 C30 H200 N220 3.4.22.1 0006508,0008234 remove_due_to_license_issue Q8MNY2 21832058 324 EIPSSFDSRKKWPRCKSIATIRDQSRCGSCWAFGAVEAMSDRSCIQSGGKQNVELSAVDLLSCCESCGLGCEGGILGPAWDYWVKEGIVTGSSKENHAGCEPYPFPKCEHHTKGKYPPCGSKIYKTPRCKQTCQKKYKTPYTQDKHRGKSSYNVKNDEKAIQKEIMKYGPVEAGFTVYEDFLNYKSGIYKHITGETLGGHAIRIIGWGVENKAPYWLIANSWNEDWGENGYFRIVRGRDECSIESEVTAGRIN 3qsu A 2.2 BS01 rna R 0 F25 F26 N28 G29 F30 Q31 S61 T62 F20 F21 N23 G24 F25 Q26 S56 T57 0003723,0006355 remove_due_to_license_issue 22965117 1 ~ 4 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTV 3qsu B 2.2 BS01 rna R 0 N28 F30 N23 F25 0003723,0006355 remove_due_to_license_issue 22965117 1 ~ 4 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTVE 3qsu C 2.2 BS01 rna P 0 N28 F30 N23 F25 0003723,0006355 remove_due_to_license_issue 22965117 5 ~ 8 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTV 3qsu E 2.2 BS01 rna P 0 F25 F26 N28 G29 F30 Q31 S61 T62 F21 F22 N24 G25 F26 Q27 S57 T58 0003723,0006355 remove_due_to_license_issue 22965117 5 ~ 8 ENIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTV 3qsu F 2.2 BS01 rna P 0 F25 G29 S61 T62 F20 G24 S56 T57 0003723,0006355 remove_due_to_license_issue 22965117 5 ~ 8 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTV 3qsu H 2.2 BS01 rna R 0 F25 G29 S61 T62 F20 G24 S56 T57 0003723,0006355 remove_due_to_license_issue 22965117 1 ~ 4 NIQDKALENFKANQTEVTVFFLNGFQMKGVIEEYDKYVVSLNSQGKQHLIYKHAISTYTVE 3qt6 A 2.047 BS01 2P0 A 1 K17 Y18 K21 S139 G140 S141 R144 S192 R193 D283 K18 Y19 K22 S140 G141 S142 R145 S193 R194 D284 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 Ki=4.3uM remove_due_to_license_issue Q9FD73 21561869 328 SMVKSGKARAHTNIALIKYWGKADETYIIPMNNSLSVTLDRFYTETKVTFDPDFTEDCLILNGNEVNAKEKEKIQNYMNIVRDLAGNRLHARIESENYVPTAAGLASSASAYAALAAACNEALSLNLSDTDLSRLARRGSGSASRSIFGGFAEWEKGHDDLTSYAHGINSNGWEKDLSMIFVVINNQSKKVSSRSGMSLTRDTSRFYQYWLDHVDEDLNEAKEAVKNQDFQRLGEVIEANGLRMHATNLGAQPPFTYLVQESYDAMAIVEQCRKANLPCYFTMDAGPNVKVLVEKKNKQAVMEQFLKVFDESKIIASDIISSGVEIIK 3qt7 A 2.199 BS01 FM0 A 1 A14 Y18 W19 K21 S139 G140 S141 R144 S192 R193 M196 D283 A284 A14 Y18 W19 K21 S139 G140 S141 R144 S189 R190 M193 D280 A281 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 Ki=49uM remove_due_to_license_issue Q9FD73 21561869 328 MVKSGKARAHTNIALIKYWGKADETYIIPMNNSLSVTLDRFYTETKVTFDPDFTEDCLILNGNEVNAKEKEKIQNYMNIVRDLAGNRLHARIESENYVPTAAGLASSASAYAALAAACNEALSLNLSDTDLSRLARRGSGSASRSIFGGFAEWEKGHDDLTSYAHGINSNGWEKDLSMIFVVINNQVSSRSGMSLTRDTSRFYQYWLDHVDEDLNEAKEAVKNQDFQRLGEVIEANGLRMHATNLGAQPPFTYLVQESYDAMAIVEQCRKANLPCYFTMDAGPNVKVLVEKKNKQAVMEQFLKVFDESKIIASDIISSGVEIIK 3qtf A 1.5703 BS01 05S A 1 N51 M98 L107 F138 Y139 W162 N35 M82 L91 F122 Y123 W146 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.11uM remove_due_to_license_issue IC50=110nM P07900 21420297 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3qti A 2.0 BS01 3QT A 1 I1084 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I33 A53 Y104 M105 D109 R153 M156 A166 D167 Y175 D1204 A1206 R1208 N1209 D1222 D149 A151 R153 N154 D167 2.7.10.1 0004672,0004713,0005524,0006468 ic50=14nM remove_due_to_license_issue IC50=14nM P08581 21697284 1 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEFLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK 3qto H 1.52 BS03 10P H 1 Y60A W60D L99 A190 E192 S195 S214 W215 G216 G219 Y47 W50 L96 A193 E195 S198 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=74.8uM remove_due_to_license_issue P00734 22366545 1001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3qtq A 1.8 BS01 X35 A 1 I10 V18 A31 K33 L83 Q85 D86 L134 D145 I10 V18 A31 K33 L79 Q81 D82 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 476 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qtr A 1.85 BS01 X36 A 1 A31 F82 L83 H84 K89 L134 D145 A31 F74 L75 H76 K81 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 497 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qts A 1.9 BS01 X46 A 1 G11 E12 V18 A31 K33 F82 L83 H84 Q131 L134 G11 E12 V18 A31 K33 F74 L75 H76 Q123 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qtu A 1.82 BS01 X44 A 1 I10 G13 V18 A31 F80 F82 L83 H84 Q85 D86 K89 N132 L134 D145 I10 G13 V18 A31 F76 F78 L79 H80 Q81 D82 K85 N128 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 451 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qtv H 1.63 BS03 06P H 1 Y60A W60D D189 E192 S195 S214 W215 G216 G219 Y47 W50 D192 E195 S198 S219 W220 G221 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=22.5uM remove_due_to_license_issue P00734 22366545 1001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3qtw A 1.85 BS01 X3A A 1 I10 V18 A31 K33 F80 L83 H84 K89 L134 D145 I10 V18 A31 K33 F76 L79 H80 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 451 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qtx A 1.95 BS01 X43 A 1 G13 V18 A31 K33 F80 L83 H84 Q85 D86 K89 L134 D145 G13 V18 A31 K33 F76 L79 H80 Q81 D82 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qtz A 2.0 BS01 X42 A 1 I10 V18 A31 K33 F82 L83 H84 Q85 D86 K89 L134 D145 I10 V18 A31 K33 F78 L79 H80 Q81 D82 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 453 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qu0 A 1.95 BS01 X40 A 1 I10 V18 A31 F80 F82 L83 H84 Q85 D86 K89 N132 L134 D145 I10 V18 A31 F76 F78 L79 H80 Q81 D82 K85 N128 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=0.900000nM P24941 23600925 454 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3que A 2.7 BS01 3FF A 1 V30 A51 K53 I84 L104 T106 M109 G110 A111 L167 L171 V26 A47 K49 I80 L100 T102 M105 G106 A107 L163 L167 D150 K152 N155 D168 T185 D146 K148 N151 D164 T175 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=40nM Q16539 22198732 362 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3qup A 1.9 BS01 LUN A 1 F519 L593 P594 F595 M596 R649 M652 A662 D663 F18 L72 P73 F74 M75 R125 M128 A138 D139 D645 A647 R649 N650 D663 D121 A123 R125 N126 D139 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.476uM remove_due_to_license_issue P55144 22119469 1 EDVLIPFTLGRMLGKGEFGSVREAQLVKVAVKMLSSDIEEFLREAACMKEFDHPHVAKLVGVSLRSIPMVILPFMKHGDLHAFLLASRIPFNLPLQTLVRFMVDIACGMEYLSSRNFIHRDLAARNCMLAEDMTVCVADFGLLPVKWLALESLADNLYTVHSDVWAFGVTMWEIMTRGQTPYAGIENAEIYNYLIGGNRLKQPPECMEEVYDLMYQCWSADPKQRPSFTCLRMELENILGH 3qvu A 2.5 BS01 NPO A 1 F81 K106 H108 F142 F74 K99 H101 F135 K48 H108 S138 K41 H101 S131 2.8.2.1 0004062,0005515,0005737,0005829,0006068,0006584,0006805,0008146,0008202,0008210,0009308,0009812,0016740,0047894,0050294,0050427,0050656,0051923 Ki=283uM remove_due_to_license_issue P50225 21723874 296 SRQPLEYVKGVPLIKYFAEALGPLQSFQARPDDLLISTYPKSGTTWVSQILDMIYQGGDLEKCHRAPIFNRVPFLEFKAPGIPSGMETLKDTPAPRLLKTHLPLALLPQTLLDQKVKVVYVARNAKDVAVSYYHFYHMAKVHPDPGTWDSFLEKFMVGEVCYGSWYQHVQEWWELSRTHPVLYLFYEDMKENPKREIQKILEFVGHSLPEETVDFMVQHTSFKEMKKNPMTNYTTIPQEIMDHSISPFMRKGMAGDWKTTFTVAQNERFDADYAEKMAGCSLSFRSEL 3qvv A 2.35 BS02 3QV A 1 F81 F84 K106 H108 V148 I247 F74 F77 K99 H101 V141 I240 K48 H108 S138 K41 H101 S131 2.8.2.1 0004062,0005515,0005737,0005829,0006068,0006584,0006805,0008146,0008202,0008210,0009308,0009812,0016740,0047894,0050294,0050427,0050656,0051923 Ki=38uM remove_due_to_license_issue P50225 21723874 296 SRQPLEYVKGVPLIKYFAEALGPLQSFQARPDDLLISTYPKSGTTWVSQILDMIYQGGDLEKCHRAPIFNRVPFLEFKAPGIPSGMETLKDTPAPRLLKTHLPLALLPQTLLDQKVKVVYVARNAKDVAVSYYHFYHMAKVHPDPGTWDSFLEKFMVGEVCYGSWYQHVQEWWELSRTHPVLYLFYEDMKENPKREIQKILEFVGHSLPEETVDFMVQHTSFKEMKKNPMTNYTTIPQEIMDHSISPFMRKGMAGDWKTTFTVAQNERFDADYAEKMAGCSLSFRSEL 3qwc H 1.75 BS03 98P H 1 H57 Y60A L99 S195 S214 W215 G216 G219 C220 H43 Y47 L96 S198 S219 W220 G221 G223 C224 3.4.21.5 0004252,0005509,0006508,0007596 Ki=55.4uM remove_due_to_license_issue P00734 22366545 2001 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3qx5 H 1.35 BS03 02P H 1 H57 Y60A W60D N98 V213 S214 W215 G216 F227 H43 Y47 W50 N95 V218 S219 W220 G221 F232 3.4.21.5 0004252,0005509,0006508,0007596 Ki=63.5uM remove_due_to_license_issue P00734 22366545 5 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3qx8 A 2.3 BS01 GTG A 1 L522 G524 K525 T526 Y529 K533 Q545 C546 Q548 K570 L83 G85 K86 T87 Y90 K94 Q106 C107 Q109 K131 3.1.26.n2 0003676 Kd=1.37mM remove_due_to_license_issue Q9UKV8 21475248 28 KQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLG 3qx9 A 2.0 BS01 ATP A 1 K525 T526 Y529 K533 Q545 C546 Q548 K566 K570 K86 T87 Y90 K94 Q106 C107 Q109 K127 K131 3.1.26.n2 0003676 Kd=0.09mM remove_due_to_license_issue Q9UKV8 21475248 1 KQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGV 3qxc A 1.34 BS01 ATP A 1 T9 N10 G12 K13 T14 T15 E116 N175 K177 T13 N14 G16 K17 T18 T19 E120 N179 K181 T9 N10 K13 T14 K35 T39 D50 E116 T13 N14 K17 T18 K39 T43 D54 E120 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 Kd=1.7uM remove_due_to_license_issue O24872 22284390 221 FQGHMLFISATNTNAGKTTCARLLAQYCNACGVKTILLKPIETGVNDAINHSSDAHLFLQDNRLLDRSLTLKDISFYRYHKVSAPLIAQQEEDPNAPIDTDNLTQRLHNFTKTYDLVIVEGAGGLCVPITLEENMLDFALKLKAKMLLISHDNLGLINDCLLNDFLLKSHQLDYKIAINLKGNNTAFHSISLPYIELFNTRSNNPIVIFQQSLKVLMSFALKGS 3qxh A 1.36 BS02 ADP A 1 N10 G12 K13 T14 T15 N175 K177 N14 G16 K17 T18 T19 N179 K181 T9 N10 K13 T14 K35 T39 D50 E116 T13 N14 K17 T18 K39 T43 D54 E120 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 Kd=5.8uM remove_due_to_license_issue O24872 22284390 222 FQGHMLFISATNTNAGKTTCARLLAQYCNACGVKTILLKPIETGVNDAINHSSDAHLFLQDNRLLDRSLTLKDISFYRYHKVSAPLIAQQEEDPNAPIDTDNLTQRLHNFTKTYDLVIVEGAGGLCVPITLEENMLDFALKLKAKMLLISHDNLGLINDCLLNDFLLKSHQLDYKIAINLKGNNTAFHSISLPYIELFNTRSNNPIVIFQQSLKVLMSFALKGS 3qxm A 1.65 BS01 NDZ A 1 Y457 P485 L486 A487 R492 V654 G657 A658 T659 M706 E707 T710 Y58 P86 L87 A88 R93 V135 G138 A139 T140 M187 E188 T191 ? 0015276,0016020 Ki=33nM remove_due_to_license_issue Q13002 21893069 301 RSLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDANGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWWR 3qxp A 1.75 BS01 X64 A 1 V18 A31 K33 F80 F82 L83 H84 Q85 D86 K89 N132 L134 D145 V18 A31 K33 F76 F78 L79 H80 Q81 D82 K85 N128 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=1.1nM P24941 23600925 300 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3qxt A 1.7 BS01 MTX A 1 V4 A26 R28 R29 S30 R32 W34 M36 R74 N79 T80 V81 V2 A24 R26 R27 S28 R30 W32 M34 R72 N77 T78 V79 Kd=6700nM remove_due_to_license_issue 21557375 2000 QVQLVESGGGLVQAGGSLRLSCAASRRSSRSWAMAWFRQAPGKEREFVAKISGDGRLTTYGDSVKGRFTISRDKGKNTVYLQMDSLKPEDTAVYYCAADDNYVTASWRSGPDYWGQGTQVTVSS 3qxv A 2.5 BS01 MTX A 1 V4 A26 S30 S31 W34 M36 R74 N76 Y79 L80 V81 V1 A23 S27 S28 W31 M33 R71 N73 Y76 L77 V78 Kd=5nM remove_due_to_license_issue 21557375 2000 VQLVESGGGLVQAGGSLRLSCAASRRSSRSWAMAWFRQAPGKEREFVAKISGDGRLTTYGDSVKGRFTISRDNAEYLVYLQMDSLKPEDTAVYYCAADDNYVTASWRSGPDYWGQGTQVTVSS 3qym A 3.2 BS01 dna I 0 R304 A307 R311 R176 A179 R183 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 SPSNTDYPGPHSFDVSFQTAKSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qym B 3.2 BS01 dna J 0 S272 R279 R304 A307 R311 S143 R150 R175 A178 R182 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 PSNTDYPGPHSFDVSFQQSSSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qym C 3.2 BS01 dna K 0 N270 R304 A307 R311 N145 R179 A182 R186 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 SPSNTDYPGPHSFDVSFQQSSTAKSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qym D 3.2 BS01 dna L 0 S272 R304 A307 R311 S148 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 ASPSNTDYPGPHSFDVSFQQSSTAKSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qym E 3.2 BS01 dna M 0 S272 R304 A307 R311 S148 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 ASPSNTDYPGPHSFDVSFQQSSTAKSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSIR 3qym F 3.2 BS01 dna N 0 R304 A307 R311 R179 A182 R186 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 SPSNTDYPGPHSFDVSFQQSSTAKSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qym G 3.2 BS01 dna O 0 S272 R279 R304 A307 R311 S142 R149 R174 A177 R181 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 SNTDYPGPHSFDVSFQQSKSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qym H 3.2 BS01 dna P 0 N270 R304 A307 R311 N139 R173 A176 R180 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue Q9H3D4 21464285 1 ~ 10 PSNTDYPGPHSFDVSFQQSATWTYSTELKKLYCQIAKTCPIQIKVMTPPPQGAVIRAMPVYKKAEHVTEVVKRCPNHELSREFNEGQIAPPSHLIRVEGNSHAQYVEDPITGRQSVLVPYEPPQVGTEFTTVLYNFMCNSSCVGGMNRRPILIIVTLETRDGQVLGRRCFEARICACPGRDRKADEDSI 3qyy A 1.9 BS01 C2E A 1 L177 K178 N181 H186 G189 D190 R212 G215 D216 L44 K45 N48 H53 G56 D57 R79 G82 D83 2.7.7.65 Ki=6.54uM (22120736) Kd=8.26uM remove_due_to_license_issue Q8P559 22120736 487 HALFDPLTEALNRRGCEQAMRDSVTAAQREGWPFVLFVLDMDNLKPINDRFGHLAGDRVLVRLVESAYGWLGAQDWIGRWGGDEFLIGVHASEDEATLKLNQWLSMLEREAPLHVSAGSAVCEVGIDATELYRRADAAMYRAKFSGGRRLVRD 3qyy A 1.9 BS03 C2E B 1 R146 W213 G214 G215 E217 R13 W80 G81 G82 E84 2.7.7.65 Ki=6.54uM (22120736) Kd=8.26uM remove_due_to_license_issue Q8P559 22120736 486 HALFDPLTEALNRRGCEQAMRDSVTAAQREGWPFVLFVLDMDNLKPINDRFGHLAGDRVLVRLVESAYGWLGAQDWIGRWGGDEFLIGVHASEDEATLKLNQWLSMLEREAPLHVSAGSAVCEVGIDATELYRRADAAMYRAKFSGGRRLVRD 3qyy B 1.9 BS01 C2E A 1 R146 W213 G214 G215 E217 R17 W84 G85 G86 E88 2.7.7.65 Ki=6.54uM (22120736) Kd=8.26uM remove_due_to_license_issue Q8P559 22120736 487 DLKRHALFDPLTEALNRRGCEQAMRDSVTAAQREGWPFVLFVLDMDNLKPINDRFGHLAGDRVLVRLVESAYGWLGAQDWIGRWGGDEFLIGVHASEDEATLKLNQWLSMLEEAPLHVSAGSAVCEVGIDATELYRRADAAMYRAKFSGGRRLVRD 3qyy B 1.9 BS02 C2E B 1 L177 K178 N181 H186 G189 D190 L193 R212 G215 D216 L48 K49 N52 H57 G60 D61 L64 R83 G86 D87 2.7.7.65 Ki=6.54uM (22120736) Kd=8.26uM remove_due_to_license_issue Q8P559 22120736 486 DLKRHALFDPLTEALNRRGCEQAMRDSVTAAQREGWPFVLFVLDMDNLKPINDRFGHLAGDRVLVRLVESAYGWLGAQDWIGRWGGDEFLIGVHASEDEATLKLNQWLSMLEEAPLHVSAGSAVCEVGIDATELYRRADAAMYRAKFSGGRRLVRD 3qzq A 1.7001 BS01 AG7 A 1 R39 H40 L125 N126 L127 S128 K130 T142 K143 A144 C147 H161 G163 G164 N165 F170 R35 H36 L121 N122 L123 S124 K126 T138 K139 A140 C143 H157 G159 G160 N161 F166 H40 D71 G145 C147 H36 D67 G141 C143 ? 0004197,0006508,0008234,0019062,0030430,0039618,0046718 remove_due_to_license_issue E7E815 21813612 501 DFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNVLDAVELVDEQGVNLDLTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKIIGIHIGGNGRQGFCAGLKRSYFA 3r00 A 2.1 BS01 UNJ A 1 A65 K67 I104 E121 R122 L174 I185 D186 A33 K35 I72 E89 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=8.5uM remove_due_to_license_issue IC50=9000nM P11309 21507633 1 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 3r01 A 2.6 BS01 UNE A 1 V52 A65 K67 R122 L174 D186 V20 A33 K35 R90 L142 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=6000nM P11309 21507633 1 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 3r02 A 1.95 BS01 UNM A 1 V52 A65 K67 R122 D128 L174 I185 D186 V18 A31 K33 R88 D94 L140 I151 D152 D167 K169 N172 D186 L193 T204 D133 K135 N138 D152 L159 T170 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.001uM remove_due_to_license_issue IC50=1nM P11309 21507633 555 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3r04 A 1.7 BS01 UNQ A 1 L44 A65 K67 I104 L120 E121 R122 D128 L174 I185 D186 L10 A31 K33 I70 L86 E87 R88 D94 L140 I151 D152 D167 K169 N172 D186 L193 T204 D133 K135 N138 D152 L159 T170 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.12uM remove_due_to_license_issue IC50=120nM P11309 21507633 555 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3r0i A 2.1 BS02 C0K A 1 E152 G185 S186 S222 N227 K228 S254 M276 E152 G185 S186 S217 N222 K223 S249 M271 1.1.1.267 0008299,0016491,0019288,0030145,0030604,0042802,0046872,0051484,0070402,1990065 ic50=0.12uM remove_due_to_license_issue P45568 21866890 991 MKQLTILGSTGSIGCSTLDVVRHNPEHFRVVALVAGKNVTRMVEQCLEFSPRYAVMDDEASAKLLKTMLQQQGSRTEVLSGQQAACDMAALEDVDQVMAAIVGAAGLLPTLAAIRAGKTILLANKESLVTCGRLFMDAVKQSKAQLLPVDSEHNAIFQSLPQPIQHNLGYADLEQNGVVSILLTGSGGPFRETPLRDLATMTPDQACSMGRKISVDSATMMNKGLEYIEARWLFNASASQMEVLIHPQSVIHSMVRYQDGSVLAQLGEPDMRTPIAHTMAWPNRVNSGVKPLDFCKLSALTFAAPDYDRYPCLKLAMEAFEQGQAATTALNAANEITVAAFLAQQIRFTDIAALNLSVLEKMDMREPQCVDDVLSVDANAREVARKEVMRLAS 3r0t A 1.75 BS01 FU9 A 1 L45 G46 V53 V66 K68 F113 H115 V116 M163 I174 D175 L43 G44 V51 V64 K66 F111 H113 V114 M161 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.91nM remove_due_to_license_issue IC50=>750nM P68400 21870818 338 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 3r0w A 1.7 BS01 RSY A 1 N25 G27 A28 V32 V84 N25 G27 A28 V32 V84 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=30.3uM remove_due_to_license_issue Q000H7 22469467 301 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3r0w B 1.7 BS01 RSY A 1 N25 G27 G48 P81 T82 V84 N25 G27 G48 P81 T82 V84 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q000H7 22469467 301 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3r0y A 1.65 BS01 RSZ A 1 N25 G27 I50 T80 P81 T82 V84 N25 G27 I50 T80 P81 T82 V84 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=14.53uM remove_due_to_license_issue Q000H7 22469467 301 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3r0y B 1.65 BS01 RSZ A 1 N25 P81 T82 N25 P81 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q000H7 22469467 301 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3r16 A 1.6 BS02 5UN A 1 H94 H96 H119 F131 L198 T199 T200 P202 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=50nM remove_due_to_license_issue Ki=50nM P00918 21620713 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3r17 B 1.7 BS02 5UM B 1 H94 H119 L198 T199 T200 P202 H91 H116 L194 T195 T196 P198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=390nM remove_due_to_license_issue Ki=390nM P00918 21620713 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3r1v A 2.19 BS01 AZB A 1 I50 L69 F111 F120 L124 I47 L66 F108 F117 L121 ? 0005549 Kd=0.12uM remove_due_to_license_issue Q7PXT9 22019737 128 FEIPDRYKKPAKMLHEICIAESGASEEQLRTCLDGTVPTAPAAKCYIHCLFDKIDVVDEATGRILLDRLLYIIPDDVKAAVDHLTRECSHIVTPDKCETAYETVKCYFNAHDEVIKFCHLLVLE 3r21 A 2.9 BS01 D36 A 1 L139 G140 V147 A160 Y212 A213 G216 T217 R220 L263 L13 G14 V21 A34 Y86 A87 G90 T91 R94 L137 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=180nM O14965 21798738 1 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3r22 A 2.9 BS01 D37 A 1 L139 G140 K141 V147 L194 Y212 A213 G216 T217 R220 L263 L14 G15 K16 V22 L69 Y87 A88 G91 T92 R95 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=17nM O14965 21798738 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3r24 A 2.0 BS01 SAM A 1 N43 G71 G73 P80 G81 D99 L100 D114 C115 D130 M131 Y132 N41 G69 G71 P78 G79 D97 L98 D112 C113 D128 M129 Y130 G39 T120 R283 V288 V289 G37 T118 R281 V286 V287 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0004483 remove_due_to_license_issue P0C6X7 22022266 302 QAWQPGVAMPNLYKMQRMLLEKCDLQNYGENAVIPKGIMMNVAKYTQLCQYLNTLTLAVPYNMRVIHFGAGSDKGVAPGTAVLRQWLPTGTLLVDSDLNDFVSDADSTLIGDCATVHTANKWDLIISDMYDPRTKHVTKENDSKEGFFTYLCGFIKQKLALGGSIAVKITEHSWNADLYKLMGHFSWWTAFVTNVNASSSEAFLIGANYLGKPKEQIDGYTMHANYIFWRNTNPIQLSSYSLFDMSKFPLKLRGTAVMSLKENQINDMIYSLLEKGRLIIRENNRVVVSSDI 3r2a A 3.0 BS01 RHN A 1 I268 N306 L436 I26 N64 L194 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 21613212 1 ANEDMPVERILEAELAVEPKDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLME 3r2a C 3.0 BS01 RHN C 1 N306 L309 C432 L436 N56 L59 C182 L186 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 21613212 2 EDMPVERILEAELAVEPICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLME 3r2b A 2.9 BS01 05B A 1 L70 G71 L72 V78 A91 K93 E139 C140 L141 E190 N191 L193 D207 L24 G25 L26 V32 A45 K47 E93 C94 L95 E140 N141 L143 D157 D186 K188 E190 N191 D207 D136 K138 E140 N141 D157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue EC50=620nM P49137 21565500 1000 HVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTPYYVAPEVLYDKSCDMWSLGVIMYILLCGYPPFYSGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKED 3r2f A 2.53 BS01 PB0 A 1 D32 G34 Y71 T72 Q73 F108 I110 W115 Y198 D228 G230 T231 T232 R235 D34 G36 Y73 T74 Q75 F110 I112 W117 Y200 D230 G232 T233 T234 R237 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=1.4nM P56817 21782431 394 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 3r2y A 3.0 BS01 P4O A 1 L70 L72 A91 K93 L141 D142 L193 D207 L25 L27 A46 K48 L96 D97 L142 D156 D186 K188 E190 N191 D207 D135 K137 E139 N140 D156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=8.5nM, EC50=49nM P49137 21565500 3 FHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTDKSCDMWSLGVIMYILLCGYPPFYMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKED 3r4m A 1.7 BS01 WOE A 1 N51 A55 G97 M98 N106 F138 T184 N41 A45 G87 M88 N96 F128 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=1.2uM remove_due_to_license_issue Ki=1200nM P07900 21438541 501 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3r4n A 2.0 BS01 FU5 A 1 N51 S52 D54 A55 D93 G97 M98 L107 F138 N42 S43 D45 A46 D84 G88 M89 L98 F129 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.13uM remove_due_to_license_issue Ki=130nM P07900 21438541 901 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKELEHHH 3r4o A 2.65 BS01 FU3 A 1 D54 A55 I96 G97 M98 D102 N106 L107 F138 D38 A39 I80 G81 M82 D86 N90 L91 F122 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Ki=7nM P07900 21438541 901 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKEL 3r4p A 1.7 BS01 FU7 A 1 N51 S52 A55 K58 I96 G97 M98 N106 L107 F138 N43 S44 A47 K50 I88 G89 M90 N98 L99 F130 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.011uM remove_due_to_license_issue Ki=11nM P07900 21438541 901 DQPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKELEHHH 3r5m A 2.8 BS02 MLO A 1 I268 A272 L309 F313 F346 C432 L436 I25 A29 L66 F70 F103 C189 L193 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 22140563 1 NEDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 3r5n A 2.0 BS01 MLO A 1 F264 G284 C285 R288 I341 S342 M364 F56 G67 C68 R71 I124 S125 M147 ? 0003677,0004879,0005634,0006355 Kd=1.67uM remove_due_to_license_issue P37231 22140563 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTKSPFVIYDMNSLMMGEDKIKFSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTSLHPLLQEIYKDLY 3r5n A 2.0 BS02 MLO A 2 F282 C285 R288 S289 I326 F363 M364 F65 C68 R71 S72 I109 F146 M147 ? 0003677,0004879,0005634,0006355 Kd=1.67uM remove_due_to_license_issue P37231 22140563 2 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTKSPFVIYDMNSLMMGEDKIKFSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTSLHPLLQEIYKDLY 3r5t A 1.45 BS01 VBN A 1 Q80 G124 A125 D126 S197 H199 H239 F242 R244 F296 R297 Q50 G94 A95 D96 S167 H169 H209 F212 R214 F266 R267 ? 0030288,0030313,1901678 remove_due_to_license_issue Q9RCF6 22291019 1 NVWPRTFQNADGSITTIPSQPKRILSTAVTVTGTLLAIDAPVIASAATTQSTFFEQWRKLAELRQVKKLWPAGSVDLESVYVEQPDLIVVSMIGADSARDQIPLLQAIAPTILVDYSDQTWQSLAQQLGLATGLEEQAERTIHNFEQWTKQVRDVLDLPKGRANIVSYHGPGVVNAVAKAQSAHAQLLQSVGVVLEEPDPAWQAGSIVHRDFLRIHYEHLTQLQAETTFLITMTDQQAQAFLHDPILKNLPSIQRKQVYGLGENSFRIDLFSAREIINSLLRRFAGEQAQSLVMPL 3r6c A 1.83 BS04 17N A 1 M86 N138 A179 P180 H183 Y186 A190 R193 G206 T209 M62 N114 A155 P156 H159 Y162 A166 R169 G182 T185 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 404 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3r6c A 1.83 BS05 17N A 2 R263 A265 D270 V325 A334 W336 R239 A241 D246 V301 A310 W312 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 405 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3r6t A 1.2 BS02 LU1 A 1 W81 M83 E133 I134 S162 D184 H185 W186 K187 N213 P217 L241 E242 W36 M38 E88 I89 S117 D139 H140 W141 K142 N168 P172 L196 E197 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 ic50=1368nM remove_due_to_license_issue P22734 22349227 307 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3r6u A 1.61 BS01 CHT A 1 Y71 D74 N115 Y117 Y197 Y221 Y60 D63 N104 Y106 Y186 Y210 ? 0005886,0006865,0022857,0043190,0055085 Kd=30.5uM remove_due_to_license_issue Q45462 21658392 285 QTIKIGAQSMSESEIIASMLGQLIEHHTDLKTTTIKNLGSNAVQQQALMNGEIDIAATRYTGDALTGTLRMEPEKDPDKALALTQREFKKRYDLKWYDSYGFDNTYAFTVSKELADQYHLETVSDVKKWAPQLKLGVDNYWMKLKGNGYQDFTKTYGMTFGGTYPMQIGLVYDAVKSGKMDIVLAYSTDGRIKSYGLKMLKDDKQFFPPYDCSPVVPEKVLKEHPELEGIIKKMLGKIDTATMQELNYEVDGNLKEPSVVAKEYLEKHRYFE 3r7o A 2.3 BS01 M61 A 1 I1084 G1085 R1086 V1092 A1108 Y1159 M1160 K1161 G1163 D1164 R1208 M1211 D1222 I37 G38 R39 V45 A61 Y112 M113 K114 G116 D117 R161 M164 D175 D1204 A1206 R1208 N1209 D1222 D157 A159 R161 N162 D175 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=3.0nM P08581 21247903 1 QNTVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHHHHH 3r7q A 2.5 BS01 FAV A 1 M804 I831 Y867 I881 V882 M953 I963 D964 M567 I594 Y630 I644 V645 M712 I722 D723 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=0.108uM remove_due_to_license_issue P48736 21636270 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNYCHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3r7r A 2.9 BS01 FAZ A 1 W812 K833 Y867 E880 V882 A885 M953 I963 D964 W572 K593 Y627 E640 V642 A645 M713 I723 D724 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 21636270 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3r88 B 1.73 BS04 14F B 1 N138 A179 P180 H183 Y186 R187 A190 N114 A155 P156 H159 Y162 R163 A166 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 404 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3r8f A 3.366 BS01 dna E 0 K188 E189 R190 T191 K112 E113 R114 T115 ? 0003677,0003688,0005524,0006270,0006275,0016887,0043565 remove_due_to_license_issue O66659 21964332 1 ~ 12 DFLNPKYTLENFIVGEGNRLAYEVVKEALENLGSLYNPIFIYGSVGTGKTHLLQAAGNEAKKRGYRVIYSSADDFAQAMVEHLKKGTINEFRNMYKSVDLLLLDDVQFLSGKERTQIEFFHIFNTLYLLEKQIILASDRHPQKLDGVSDRLVSRFEGGILVEIELDNKTRFKIIKEKLKEFNLELRKEVIDYLLENTKNVREIEGKIKLIKLKGFEGLERKERKERDKLMQIVEFVANYYAVKVEDILSDKNKRTSEARKIAMYLCRKVCSASLIEIARAFKRKDHTTVIHAIRSVEEEKRKFKHLVGFLEKQAFDKIC 3r8f B 3.366 BS01 dna E 0 K188 E189 R190 T191 K112 E113 R114 T115 ? 0003677,0003688,0005524,0006270,0006275,0016887,0043565 remove_due_to_license_issue O66659 21964332 1 ~ 12 DFLNPKYTLENFIVGEGNRLAYEVVKEALENLGSLYNPIFIYGSVGTGKTHLLQAAGNEAKKRGYRVIYSSADDFAQAMVEHLKKGTINEFRNMYKSVDLLLLDDVQFLSGKERTQIEFFHIFNTLYLLEKQIILASDRHPQKLDGVSDRLVSRFEGGILVEIELDNKTRFKIIKEKLKEFNLELRKEVIDYLLENTKNVREIEGKIKLIKLKGFEGLERKERKERDKLMQIVEFVANYYAVKVEDILSDKNKRTSEARKIAMYLCRKVCSASLIEIARAFKRKDHTTVIHAIRSVEEEKRKFKHLVGFLEKQAFDKIC 3r8f C 3.366 BS01 dna E 0 L159 K188 R190 T191 L83 K112 R114 T115 ? 0003677,0003688,0005524,0006270,0006275,0016887,0043565 remove_due_to_license_issue O66659 21964332 1 ~ 12 DFLNPKYTLENFIVGEGNRLAYEVVKEALENLGSLYNPIFIYGSVGTGKTHLLQAAGNEAKKRGYRVIYSSADDFAQAMVEHLKKGTINEFRNMYKSVDLLLLDDVQFLSGKERTQIEFFHIFNTLYLLEKQIILASDRHPQKLDGVSDRLVSRFEGGILVEIELDNKTRFKIIKEKLKEFNLELRKEVIDYLLENTKNVREIEGKIKLIKLKGFEGLERKERKERDKLMQIVEFVANYYAVKVEDILSDKNKRTSEARKIAMYLCRKVCSASLIEIARAFKRKDHTTVIHAIRSVEEEKRKFKHLVGFLEKQAFDKIC 3r8f D 3.366 BS01 dna E 0 K188 R190 T191 K112 R114 T115 ? 0003677,0003688,0005524,0006270,0006275,0016887,0043565 remove_due_to_license_issue O66659 21964332 1 ~ 12 DFLNPKYTLENFIVGEGNRLAYEVVKEALENLGSLYNPIFIYGSVGTGKTHLLQAAGNEAKKRGYRVIYSSADDFAQAMVEHLKKGTINEFRNMYKSVDLLLLDDVQFLSGKERTQIEFFHIFNTLYLLEKQIILASDRHPQKLDGVSDRLVSRFEGGILVEIELDNKTRFKIIKEKLKEFNLELRKEVIDYLLENTKNVREIEGKIKLIKLKGFEGLERKERKERDKLMQIVEFVANYYAVKVEDILSDKNKRTSEARKIAMYLCRKVCSASLIEIARAFKRKDHTTVIHAIRSVEEEKRKFKHLVGFLEKQAFDKIC 3r8i A 2.3 BS01 XCX A 1 I281 C285 R288 S289 H323 L340 I341 M364 H449 Y473 I75 C79 R82 S83 H117 L134 I135 M158 H243 Y267 ? 0003677,0004879,0005634,0006355 Kd=4.5uM remove_due_to_license_issue EC50=110nM, Kd=4500nM P37231 22081932 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3r8u A 2.0 BS01 Z31 A 1 I10 E12 V18 A31 K33 F82 L83 Q85 Q131 L134 I10 E12 V18 A31 K33 F78 L79 Q81 Q127 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 465 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r8v A 1.9 BS01 Z62 A 1 I10 G11 E12 V18 A31 K33 F82 L83 L134 I10 G11 E12 V18 A31 K33 F78 L79 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 473 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r8z A 1.85 BS01 Z63 A 1 V18 A31 E81 F82 L83 D86 L134 D145 V18 A31 E77 F78 L79 D82 L130 D141 D127 K129 Q131 N132 D145 T165 D123 K125 Q127 N128 D141 T157 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 440 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r91 A 1.579 BS01 06H A 1 N51 A55 K58 M98 L107 F138 Y139 W162 N35 A39 K42 M82 L91 F122 Y123 W146 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.092uM remove_due_to_license_issue P07900 21515049 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 3r92 A 1.5801 BS01 06J A 1 N51 A55 M98 L107 F138 Y139 W162 T184 N35 A39 M82 L91 F122 Y123 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.883uM remove_due_to_license_issue IC50=96nM P07900 21605975 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3r9d A 1.95 BS01 X6B A 1 I10 V18 A31 K33 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 V18 A31 K33 F76 F78 L79 H80 Q81 D82 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 590 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r9h A 2.1 BS01 Z67 A 1 I10 A31 K33 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 K33 F76 E77 F78 L79 H80 Q81 D82 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 606 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r9n A 1.75 BS01 Z68 A 1 G11 E12 V18 A31 K33 F82 L83 Q85 Q131 L134 G11 E12 V18 A31 K33 F74 L75 Q77 Q123 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 529 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r9o A 1.9 BS01 Z71 A 1 I10 A31 K33 F80 E81 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 K33 F72 E73 F74 L75 H76 Q77 D78 K81 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 401 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3r9w A 2.05 BS01 rna B 0 K66 T206 R207 E208 E209 G224 D225 A226 M230 R241 N243 L244 K245 P246 I247 I249 G250 K251 K252 R255 L256 K257 G260 K261 R264 V275 Y276 L277 W280 V281 R289 K67 T207 R208 E209 E210 G225 D226 A227 M231 R242 N244 L245 K246 P247 I248 I250 G251 K252 K253 R256 L257 K258 G261 K262 R265 V276 Y277 L278 W281 V282 R290 ? 0000028,0003723,0003924,0005525,0005737,0005829,0005886,0019843,0042254,0042274,0043024,0070181 remove_due_to_license_issue O67800 21646538 1506 ~ 1539 HMKVGYVAIVGKPNVGKSTLLNNLLGTKVSIISPKAGTTRMRVLGVKNIPNEAQIIFLDTPGIYEPKKSDVLGHSMVEIAKQSLEEADVILFMIDATEGWRPRDEEIYQNFIKPLNKPVIVVINKIDKIGPAKNVLPLIDEIHKKHPELTEIVPISALKGANLDELVKTILKYLPEGEPLFPEDMITDLPLRLLAAEIVREKAMMLTREEVPTSIAVKINEIKPGDANPNMLVIKGEIIVDRENLKPIIIGKKGQRLKEIGKRARQELELILGRPVYLELWVKVVPDWRRRPEYVRLFGYAL 3rah A 1.75 BS01 O1Z A 1 E12 G13 V18 A31 K33 F82 L83 Q85 Q131 N132 L134 E12 G13 V18 A31 K33 F74 L75 Q77 Q123 N124 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 516 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rak A 1.75 BS01 03Z A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F72 F74 L75 H76 Q77 D78 K81 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 497 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ral A 1.75 BS01 04Z A 1 I10 G13 V18 A31 K33 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 G13 V18 A31 K33 F72 F74 L75 H76 Q77 D78 K81 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 499 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rbm A 2.61 BS03 B73 A 1 F122 D126 R135 V156 Q195 K243 T244 D287 K301 F88 D92 R101 V122 Q161 K205 T206 D249 K263 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILF 3rbm A 2.61 BS04 B73 B 1 V153 L157 V119 L123 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILF 3rbm B 2.61 BS01 B73 A 1 V153 L157 V119 L123 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K209 F249 D253 D254 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSDAHREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3rbm B 2.61 BS04 B73 B 1 F122 A125 D126 R135 V153 V156 Q195 K243 T244 D287 K301 F88 A91 D92 R101 V119 V122 Q161 K209 T210 D253 K267 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K209 F249 D253 D254 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSDAHREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3rbu A 1.6 BS04 G88 A 1 R210 N257 D387 E424 E425 L428 G518 Y552 H553 K699 Y700 R156 N203 D333 E370 E371 L374 G464 Y494 H495 K640 Y641 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=370pM remove_due_to_license_issue Ki=0.280000nM, IC50=300nM, Kd=0.5nM, EC50=0.620000nM Q04609 22178733 1800 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3rcd A 3.21 BS01 03P A 1 G727 V734 A751 K753 S783 L785 T798 L800 M801 G804 L852 T862 D863 G18 V25 A42 K44 S70 L72 T85 L87 M88 G91 L139 T149 D150 D845 A847 R849 N850 D863 D132 A134 R136 N137 D150 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=17nM P04626 22003817 9001 ALLRILKETELRKVKVLGSGAFGTVYKGIWIPDGENVKIPVAIKVLRPKANKEILDEAYVMAGVGSPYVSRLLGICLTSTVQLVTQLMPYGCLLDHVRENRGRLGSQDLLNWCMQIAKGMSYLEDVRLVHRDLAARNVLVKSPNHVKITDFGLVPIKWMALESILRRRFTHQSDVWSYGVTVWELMTFGAKPYDGIPAREIPDLLEKGERLPQPPICTIDVYMIMVKCWMIDSECRPRFRELVSEFSRMARDPQRFVVIQNLDSTFYRSLLEDDDLVDAEE 3rcj A 1.7 BS01 3RC A 1 S94 V96 A109 S160 Y161 A162 L212 T222 S18 V20 A33 S84 Y85 A86 L136 T146 D205 K207 E209 N210 D223 T245 D129 K131 E133 N134 D147 T169 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.8uM remove_due_to_license_issue O15530 21625704 0 KRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 3rde A 1.892 BS02 OYP A 1 F175 L179 E357 H361 H366 R403 A404 L408 I593 Q596 L597 F64 L68 E246 H250 H255 R292 A293 L297 I482 Q485 L486 H361 H366 H541 H545 I663 H250 H255 H430 H434 I552 1.13.11.-,1.13.11.12,1.13.11.31,1.13.11.33 0005506,0016702,0034440,0046872 remove_due_to_license_issue IC50=35nM P16469 22795085 664 GTARTVVDDPQGLFKKHREEELAERRKLYRWGNWKDGLILNIASTGIHDLPVDERFLEDKRIDFEASLAKGLADLAVKDSLNVLMSWNSLDSFNRIFWSGQSKLAERVRDSWKEDALFGYQFLNGTNPMLLRHSVELPARLKFPPGMEELQAQLEKELQGGTLFEADFSLLDGIKANVILSSQQYLAVPLVMLKLQPDGKLLPMVIQLQLPREGSPLPPLFLPTDPPMVWLLAKCWVRSSDFQLHELHSHLLRGHLMAEVIAVATMRCLPSIHPIFKLLIPHFRYTMEINVRARNGLVSDLGIFDQVVSTGGGGHVELLRRAAALLTYSSFCPPDDLADRGLLGVESSFYAQDALRLWEVISRYVEGIVSLHYKTDESVKEDFELQAWCREFTEIGLLGAQDRGFPVSLQSKEQLCHFVTMCIFTCTGQHSSNHLGQLDWYTWVPNAPCTMRLPPPTTKDATLETVMATLPNFHQASLQMSITWQLGRCQPTMVALGQHEEEYFSGPGPKAVLTKFREELAALDKDIEVRNAKLALPYEYLRPSRVENSVAI 3rdh A 2.39 BS01 3RD A 1 K120 I217 K123 I220 ? 0000122,0001525,0003016,0003723,0005515,0005615,0005634,0005654,0005737,0005829,0005925,0006468,0006605,0007165,0008039,0008104,0019901,0019904,0030324,0031625,0031647,0031982,0035148,0042149,0042470,0042802,0043066,0043067,0044325,0045296,0045824,0050815,0051683,0070062,0070371,0070372,0072562,0090128,0090168,0098686,0098978,0140297,0140311,1900181,1904262 remove_due_to_license_issue IC50=9300nM P63104 21908710 246 GSHMDKNELVQKAKLAEQAERYDDMAACMKSVTEQGAELSNEERNLLSVAYKNVVGARRSSWRVVSSIEQKTEGAEKKQQMAREYREKIETELRDICNDVLSLLEKFLIPNASQAESKVFYLKMKGDYYRYLAEVAAGDDKKGIVDQSQQAYQEAFEISKKEMQPTHPIRLGLALNFSVFYYEILNSPEKACSLAKTAFDEAIAELDTLSEESYKDSTLIMQLLRDNLTLWTS 3rdo A 1.404 BS01 BTN A 1 L25 S27 Y43 S45 V47 N49 W79 A86 S88 D128 L19 S21 Y37 S39 V41 N43 W73 A80 S82 D122 ? 0009374 Kd=0.14nM remove_due_to_license_issue Kd=1.000000nM P22629 21520321 300 HHHHSTAEAGITGTWYNQLGSTLIVTAGADGALTGTYESAVGNAEGSYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSASTWSGQYVGGAEARINTQVLTTSGTTEANAWKSTLVGHDTFTKVKP 3rdq A 1.6 BS01 DTB A 1 L25 S27 Y43 S45 V47 G48 N49 W79 A86 S88 D128 L16 S18 Y34 S36 V38 G39 N40 W70 A77 S79 D119 ? 0009374 Kd=0.49nM remove_due_to_license_issue P22629 21520321 300 HHTAEAGITGTWYNQLGSTLIVTAGADGALTGTYESAVGNAEGSYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSASTWSGQYVGGAEARINTQVLTTSGTTEANAWKSTLVGHDTFTKVK 3re4 A 1.997 BS01 TO1 A 1 S56 A78 M147 F149 I150 I211 S54 A76 M141 F143 I144 I205 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004711,0005524,0006338,0006468,0016787,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0046872,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 Kd~40nM remove_due_to_license_issue O28471 22629386 259 DLKKIESYLDKLRIKEKDGEERKIYAEVLDGRTLKTLYKLSAKGYITAMGGVISTGKEANVFYADGVFDGKPVAMAVKIYRIEDKMDEYLYGDERFDMRRISPKEKVFIWTEKEFRNLERAKEAGVSVPQPYTYMKNVLLMEFIGEDELPAPTLVELGRELKELDVEGIFNDVVENVKRLYQEAELVHADLSEYNIMYIDKVYFIDMGQAVTLRHPMAESYLERDVRNIIRFFSKYGVKADFEEMLKEVKGE 3rer A 1.7 BS01 rna K 0 Q8 Q41 F42 H57 Q3 Q36 F37 H52 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 21979921 1 ~ 8 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3rer B 1.7 BS01 rna K 0 S6 Q8 D9 Q41 F42 Y55 H57 S3 Q5 D6 Q38 F39 Y52 H54 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 21979921 1 ~ 8 GQSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3rer C 1.7 BS01 rna K 0 Q5 Q8 Q41 F42 K56 H57 Q4 Q7 Q40 F41 K55 H56 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 21979921 1 ~ 8 AKGQSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3rer D 1.7 BS01 rna K 0 Q8 Q41 F42 K56 H57 Q3 Q36 F37 K51 H52 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 21979921 1 ~ 8 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3rer E 1.7 BS01 rna K 0 F42 H57 F37 H52 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 21979921 1 ~ 8 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3rer F 1.7 BS01 rna K 0 Q8 Q41 H57 Q4 Q37 H53 ? 0003723,0006355 remove_due_to_license_issue P0A6X3 21979921 1 ~ 8 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 3rey A 3.309 BS01 XAC A 1 A81 F168 M177 L249 H250 N253 M270 Y271 I274 A75 F154 M163 L235 H236 N239 M256 Y257 I260 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue Ki=63nM P29274 21885291 999 SVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLKQMESQPLPGERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 3rf4 A 1.8 BS01 FUN A 1 P1 M2 K32 R36 I64 V106 F108 V113 P1 M2 K32 R36 I64 V106 F108 V113 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=0.56uM remove_due_to_license_issue A4GRE3 21944748 201 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf4 C 1.8 BS01 FUN C 1 P1 M2 K32 R36 I64 V106 F108 V113 P1 M2 K32 R36 I64 V106 F108 V113 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=0.56uM remove_due_to_license_issue A4GRE3 21944748 203 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf5 A 2.1 BS01 FUZ A 1 P1 M2 K32 R36 I64 V106 F108 V113 P1 M2 K32 R36 I64 V106 F108 V113 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=2.37uM remove_due_to_license_issue A4GRE3 21944748 202 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf5 C 2.1 BS01 FUZ A 1 H49 I95 H49 I95 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=2.37uM remove_due_to_license_issue A4GRE3 21944748 202 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf5 C 2.1 BS02 FUZ C 1 P1 M2 K32 R36 I64 F108 P1 M2 K32 R36 I64 F108 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=2.37uM remove_due_to_license_issue A4GRE3 21944748 203 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rg2 A 3.1 BS01 SVS A 1 N235 Y236 G309 A310 R311 V331 F332 G333 M334 A335 D415 N234 Y235 G308 A309 R310 V330 F331 G332 M333 A334 D414 S190 S210 H234 A335 E336 N436 K441 K520 S189 S209 H233 A334 E335 N435 K440 K519 3.3.2.1,6.2.1.71,6.3.2.14 0005515,0005524,0005829,0008668,0009239,0016020,0016746,0016874,0016877,0019290,0047527 remove_due_to_license_issue P0ADI4,P10378 22365602 698 SIPFTRWPEEFARRYREKGYWQDLPLTDILTRHAASDSIAVIDGERQLSYRELNQAADNLACSLRRQGIKPGETALVQLGNVAELYITFFALLKLGVAPVLALFSHQRSELNAYASQIEPALLIADRQHALFSGDDFLNTFVTEHSSIRVVQLLNDSGEHNLQDAINHPAEDFTATPSPADEVAYFQLSGGTTGTPKLIPRTHNDYYYSVRRSVEICQFTQQTRYLCAIPAAHNYAMSSPGSLGVFLAGGTVVLAADPSATLCFPLIEKHQVNVTALVPPAVSLWLQALIEGESRAQLASLKLLQVGGARLSATLAARIPAEIGCQLQQVFGMAEGLVNYTRLDDSAEKIIHTQGYPMCPDDEVWVADAEGNPLPQGEVGRLMTRGPYTFRGYYKSPQHNASAFDANGFYCSGDLISIDPEGYITVQGREKDQINRGGEKIAAEEIENLLLRHPAVIYAALVSMEDELMGEKSCAYLVVKEPLRAVQVRRFLREQGIAEFKLPDRVECVDSLPLTAVGKVDKKQLRQWLASRASAGRASIPASKAALREVILPLLDESDEPFDDDNLIDYGLDSVRMMALAARWRKVHGDIDFVMLAKNPTIDAWWKLLSR 3rg2 A 3.1 BS02 PNS B 1 P231 H234 V279 G438 G439 P230 H233 V278 G437 G438 S190 S210 H234 A335 E336 N436 K441 K520 S189 S209 H233 A334 E335 N435 K440 K519 3.3.2.1,6.2.1.71,6.3.2.14 0005515,0005524,0005829,0008668,0009239,0016020,0016746,0016874,0016877,0019290,0047527 remove_due_to_license_issue P0ADI4,P10378 22365602 991 SIPFTRWPEEFARRYREKGYWQDLPLTDILTRHAASDSIAVIDGERQLSYRELNQAADNLACSLRRQGIKPGETALVQLGNVAELYITFFALLKLGVAPVLALFSHQRSELNAYASQIEPALLIADRQHALFSGDDFLNTFVTEHSSIRVVQLLNDSGEHNLQDAINHPAEDFTATPSPADEVAYFQLSGGTTGTPKLIPRTHNDYYYSVRRSVEICQFTQQTRYLCAIPAAHNYAMSSPGSLGVFLAGGTVVLAADPSATLCFPLIEKHQVNVTALVPPAVSLWLQALIEGESRAQLASLKLLQVGGARLSATLAARIPAEIGCQLQQVFGMAEGLVNYTRLDDSAEKIIHTQGYPMCPDDEVWVADAEGNPLPQGEVGRLMTRGPYTFRGYYKSPQHNASAFDANGFYCSGDLISIDPEGYITVQGREKDQINRGGEKIAAEEIENLLLRHPAVIYAALVSMEDELMGEKSCAYLVVKEPLRAVQVRRFLREQGIAEFKLPDRVECVDSLPLTAVGKVDKKQLRQWLASRASAGRASIPASKAALREVILPLLDESDEPFDDDNLIDYGLDSVRMMALAARWRKVHGDIDFVMLAKNPTIDAWWKLLSR 3rg2 B 3.1 BS01 PNS A 1 P231 H234 V279 G438 G439 P230 H233 V278 G437 G438 S190 S210 H234 A335 E336 N436 K441 K520 S189 S209 H233 A334 E335 N435 K440 K519 3.3.2.1,6.2.1.71,6.3.2.14 0005515,0005524,0005829,0008668,0009239,0016020,0016746,0016874,0016877,0019290,0047527 remove_due_to_license_issue P0ADI4,P10378 22365602 991 SIPFTRWPEEFARRYREKGYWQDLPLTDILTRHAASDSIAVIDGERQLSYRELNQAADNLACSLRRQGIKPGETALVQLGNVAELYITFFALLKLGVAPVLALFSHQRSELNAYASQIEPALLIADRQHALFSGDDFLNTFVTEHSSIRVVQLLNDSGEHNLQDAINHPAEDFTATPSPADEVAYFQLSGGTTGTPKLIPRTHNDYYYSVRRSVEICQFTQQTRYLCAIPAAHNYAMSSPGSLGVFLAGGTVVLAADPSATLCFPLIEKHQVNVTALVPPAVSLWLQALIEGESRAQLASLKLLQVGGARLSATLAARIPAEIGCQLQQVFGMAEGLVNYTRLDDSAEKIIHTQGYPMCPDDEVWVADAEGNPLPQGEVGRLMTRGPYTFRGYYKSPQHNASAFDANGFYCSGDLISIDPEGYITVQGREKDQINRGGEKIAAEEIENLLLRHPAVIYAALVSMEDELMGEKSCAYLVVKEPLRAVQVRRFLREQGIAEFKLPDRVECVDSLPLTAVGKVDKKQLRQWLASRASSIPASKAALREVILPLLDESDEPFDDDNLIDYGLDSVRMMALAARWRKVHGDIDFVMLAKNPTIDAWWKLLS 3rg2 B 3.1 BS02 SVS B 1 N235 Y236 G309 A310 R311 V331 F332 G333 M334 A335 D415 N234 Y235 G308 A309 R310 V330 F331 G332 M333 A334 D414 S190 S210 H234 A335 E336 N436 K441 K520 S189 S209 H233 A334 E335 N435 K440 K519 3.3.2.1,6.2.1.71,6.3.2.14 0005515,0005524,0005829,0008668,0009239,0016020,0016746,0016874,0016877,0019290,0047527 remove_due_to_license_issue P0ADI4,P10378 22365602 698 SIPFTRWPEEFARRYREKGYWQDLPLTDILTRHAASDSIAVIDGERQLSYRELNQAADNLACSLRRQGIKPGETALVQLGNVAELYITFFALLKLGVAPVLALFSHQRSELNAYASQIEPALLIADRQHALFSGDDFLNTFVTEHSSIRVVQLLNDSGEHNLQDAINHPAEDFTATPSPADEVAYFQLSGGTTGTPKLIPRTHNDYYYSVRRSVEICQFTQQTRYLCAIPAAHNYAMSSPGSLGVFLAGGTVVLAADPSATLCFPLIEKHQVNVTALVPPAVSLWLQALIEGESRAQLASLKLLQVGGARLSATLAARIPAEIGCQLQQVFGMAEGLVNYTRLDDSAEKIIHTQGYPMCPDDEVWVADAEGNPLPQGEVGRLMTRGPYTFRGYYKSPQHNASAFDANGFYCSGDLISIDPEGYITVQGREKDQINRGGEKIAAEEIENLLLRHPAVIYAALVSMEDELMGEKSCAYLVVKEPLRAVQVRRFLREQGIAEFKLPDRVECVDSLPLTAVGKVDKKQLRQWLASRASSIPASKAALREVILPLLDESDEPFDDDNLIDYGLDSVRMMALAARWRKVHGDIDFVMLAKNPTIDAWWKLLS 3rhk A 1.94 BS01 M97 A 1 I1084 G1085 F1089 V1092 A1108 K1110 Y1159 M1160 G1163 M1211 F1223 I36 G37 F41 V44 A60 K62 Y111 M112 G115 M163 F175 D1204 A1206 R1208 N1209 D1222 A1243 D156 A158 R160 N161 D174 A195 2.7.10.1 0004672,0004713,0005524,0006468 ic50=520nM remove_due_to_license_issue P08581 21454604 1 NTVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 3rhx B 2.01 BS01 3RH B 1 V492 A512 V561 Y563 A564 L630 V32 A48 V97 Y99 A100 L150 D623 A625 R627 N628 D641 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=0.84uM remove_due_to_license_issue IC50=840nM P11362 21454610 1 SEYELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLADYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALT 3ri1 A 2.1 BS01 3RH A 1 V495 A515 K517 M538 V564 A567 L633 V28 A48 K50 M71 V97 A100 L153 D626 A628 R630 N631 D644 D146 A148 R150 N151 D164 2.7.10.1 0004672,0004713,0005524,0006468 Kd=5uM remove_due_to_license_issue IC50=1230nM P21802 21454610 2 LPEDPKWEFPRDKLTLGKPLGEGCFGQVVMAEAVGIDKDKPKEAVTVAVKMLKDDATEKDLSDLVSEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLRARRPPEQMTFKDLVSCTYQLARGMEYLASQKCIHRDLAARNVLVTENNVMKIADFGLARDINNIDYYKKTTNGRLPVKWMAPEALFDRVYTHQSDVWSFGVLMWEIFTLGGSPYPGIPVEELFKLLKEGHRMDKPANCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRILTLTT 3rik B 2.48 BS01 3RI B 1 D127 F128 W179 N234 E235 W312 Y313 E340 W381 D127 F128 W179 N234 E235 W312 Y313 E340 W381 E235 E340 C342 N370 E235 E340 C342 N370 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 ic50=3.4mM remove_due_to_license_issue P04062 22047104 501 ARPCIPKSFGYSSVVCVCNATYCDSFDPPTFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 3ril A 2.4 BS01 3RK A 1 D127 F128 W179 N234 E235 F246 E340 W381 D127 F128 W179 N234 E235 F246 E339 W380 E235 E340 C342 N370 E235 E339 C341 N369 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 ic50=146uM remove_due_to_license_issue Ki=12800nM P04062 22047104 513 ARPCIPKSFGYSSVVCVCNATYCDSFDPPTFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 3ril B 2.4 BS01 3RK B 1 D127 F128 W179 N234 E235 E340 C342 W381 D127 F128 W179 N234 E235 E340 C342 W381 E235 E340 C342 N370 E235 E340 C342 N370 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 ic50=146uM remove_due_to_license_issue Ki=12800nM P04062 22047104 509 ARPCIPKSFGYSSVVCVCNATYCDSFDPPTFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWHRQ 3rin A 2.2 BS01 I2O A 1 Y35 A51 E71 T106 L108 M109 G110 A111 L167 D168 F169 L171 Y32 A48 E68 T103 L105 M106 G107 A108 L164 D165 F166 L168 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=1.3nM remove_due_to_license_issue IC50=1.3nM Q16539 21696951 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3rj7 A 1.2 BS02 RCS A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22344779 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rj7 A 1.2 BS03 RCS A 2 H4 W5 H10 N11 H15 W16 D19 H2 W3 H8 N9 H13 W14 D17 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22344779 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rjc A 1.85 BS01 06Z A 1 I10 V18 A31 F82 L83 H84 L134 D145 I10 V18 A31 F78 L79 H80 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 450 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rjw A 2.56 BS06 CIQ A 1 Y1067 D1074 A1077 D1078 R1080 D1083 L1086 D1088 Y1154 F1158 Y150 D157 A160 D161 R163 D166 L169 D171 Y237 F241 Y1067 Y1154 Y150 Y237 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue IC50=<15nM, Ki=3.7nM, Kd=1420nM Q96KQ7 21743462 2000 TEKIICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLDNKDGEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKYFTCQCGSEKCKHSAEAIALEQS 3rk5 A 2.0 BS01 07Z A 1 V18 A31 F82 L83 H84 K89 L134 V18 A31 F78 L79 H80 K85 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 436 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rk7 A 1.8 BS01 08Z A 1 V18 A31 K33 F80 F82 L83 H84 L134 D145 V18 A31 K33 F76 F78 L79 H80 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 467 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rk9 A 1.85 BS01 09Z A 1 I10 V18 A31 L83 L134 D145 I10 V18 A31 L79 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 483 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rkb A 2.0 BS01 12Z A 1 I10 V18 A31 F82 L83 L134 D145 I10 V18 A31 F78 L79 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 457 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rkz A 1.5693 BS01 06T A 1 N51 M98 L107 F138 Y139 W162 T184 N35 M82 L91 F122 Y123 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.083uM remove_due_to_license_issue IC50=83nM P07900 21715165 1 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3rl3 A 1.42 BS06 5GP A 1 H67 D86 N117 H118 F183 K225 I253 H254 E255 H57 D76 N107 H108 F168 K210 I238 H239 E240 3.1.-.- 0000166,0008081,0016208,0016787,0019002,0030145,0046872 ic50=67nM remove_due_to_license_issue B1WBP0 21824479 951 VTITVDEYSSNPTQAFTHYNINQSRFQPPHVHMVDPIPYDTPKPAGHTRFVCISDTHSRTDGIQMPYGDILLHTGDFTELGLPSEVKKFNDWLGNLPYEYKIVIAGNHELTFDKEFMADLVRFPSVSKLKPEDFDNVQSLLTNSIYLQDSEVTVKGFRIYGAPWTPWFNGWGFNLPRGQSLLDKWNLIPEGTDILMTHGPPLGFRDWVPKELQRVGCVELLNTVQRRVRPKLHVFGGIHEGYGTMTDGYTTYINASTCTVSFQPTNPPIIFDLPNP 3rl4 A 1.29 BS06 5GP A 1 H67 D86 N117 H118 F183 E226 H252 H254 E255 H57 D76 N107 H108 F167 E210 H236 H238 E239 3.1.-.- 0000166,0008081,0016208,0016787,0019002,0030145,0046872 ic50=3800nM remove_due_to_license_issue B1WBP0 21824479 951 VTITVDEYSSNPTQAFTHYNINQSRFQPPHVHMVDPIPYDTPKPAGHTRFVCISDTHSRTDGIQMPYGDILLHTGDFTELGLPSEVKKFNDWLGNLPYEYKIVIAGNHELTFDKEFMADLVFPSVSKLKPEDFDNVQSLLTNSIYLQDSEVTVKGFRIYGAPWTPWFNGWGFNLPRGQSLLDKWNLIPEGTDILMTHGPPLGFRDWVPKELQRVGCVELLNTVQRRVRPKLHVFGHIHEGYGTMTDGYTTYINASTCTVSFQPTNPPIIFDLPNP 3rlb A 2.0 BS01 VIB A 1 W34 E84 Y85 H125 W133 Y146 W28 E78 Y79 H119 W127 Y140 0005886,0015234,0015888 Kd=120pM remove_due_to_license_issue 21706007 191 NVRLLTEIAFMAALAFIISLIPNTVYGWIIVEIACIPILLLSLRRGLTAGLVGGLIWGILSMITGHAYILSLSQAFLEYLVAPVSLGIAGLFRQKTAPLKLAPVLLGTFVAVLLKYFFHFIAGIIFWSQYAWKGWGAVAYSLAVNGISGILTAIAAFVILIIFVKKFPKLFIHSNY 3rlp A 1.7 BS01 3RP A 1 S52 A55 M98 L107 F138 S43 A46 M89 L98 F129 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.084uM remove_due_to_license_issue P07900 21612924 901 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKEL 3rlq A 1.9 BS01 3RQ A 1 N51 A55 D93 M98 L107 F138 T184 N43 A47 D85 M90 L99 F130 T176 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.04uM remove_due_to_license_issue P07900 21612924 901 DQPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKELEHHH 3rlr A 1.7 BS01 3RR A 1 L48 N51 A55 D93 M98 L107 F138 T184 V186 L40 N43 A47 D85 M90 L99 F130 T176 V178 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.03uM remove_due_to_license_issue P07900 21612924 901 DQPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKELE 3rm4 A 1.9 BS01 3RM A 1 Y27 D138 E140 M210 Y212 D213 Y267 E297 I300 W360 L364 Y6 D117 E119 M189 Y191 D192 Y246 E276 I279 W339 L343 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 Kd=1.69uM remove_due_to_license_issue IC50=210nM, Kd=1690nM Q9BZP6 20666458 1 YQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNVKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASC 3rm8 A 1.8 BS01 RM8 A 1 W99 D138 E140 M210 Y212 D213 Y267 E297 I300 W360 W78 D117 E119 M189 Y191 D192 Y246 E276 I279 W339 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 ic50=0.7uM remove_due_to_license_issue IC50=700nM Q9BZP6 20666458 417 YQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNVKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTAPA 3rm9 A 2.1 BS01 613 A 1 E140 D213 Y267 E297 I300 W360 L364 E119 D192 Y246 E276 I279 W339 L343 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 Kd=17uM remove_due_to_license_issue Kd=17000nM, IC50=13000nM Q9BZP6 20666458 1 YQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNVKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTAPA 3rme A 1.8 BS01 RME A 1 W31 F58 G98 D138 E140 Y212 D213 Y267 W360 W10 F37 G77 D117 E119 Y191 D192 Y246 W339 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 ic50=22uM remove_due_to_license_issue IC50=22000nM Q9BZP6 20666458 418 YQLTCYFTNWAQYRPGLGRFMPDDINPCLCTHLIYAFAGMQNNEITTIEWNDVTLYQAFNGLKNKNSQLKTLLAIGGWNFGTAPFTAMVSTPENRQTFITSVIKFLRQYEFDGLDFDWEYPGSRGSPPQDKHLFTVLVQEMREAFEQEAKQINKPRLMVTAAVAAGISNIQSGYEIPQLSQYLDYIHVMTYDLHGSWEGYTGENSPLYKYPTDTGSNAYLNVDYVMNYWKDNGAPAEKLIVGFPTYGHNFILSNPSNTGIGAPTSGAGPAGPYAKESGIWAYYEICTFLKNGATQGWDAPQEVPYAYQGNVWVGYDNVKSFDIKAQWLKHNKFGGAMVWAIDLDDFTGTFCNQGKFPLISTLKKALGLQSASCTAPA 3rmf A 1.75 BS01 20Z A 1 I10 V18 A31 F82 L83 H84 Q85 D86 K89 L134 D145 I10 V18 A31 F75 L76 H77 Q78 D79 K82 L127 D138 D127 K129 Q131 N132 D145 T165 D120 K122 Q124 N125 D138 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 496 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rn2 A 2.55 BS01 dna K 0 L267 K309 R311 K340 L121 K163 R165 K194 ? 0002218,0035458 remove_due_to_license_issue O14862 22483801 1 ~ 20 EGFQKRCLPVMVLKAKKPFTFETQEGKQEMFHATVATEKEFFFVKVFNTLLKDKFIPKRIIIIARYYRHSGFLEVNSASRVLDAESDQKVNVPLNIIRKAGETPKINTLQTQPLGTIVNGLFVVQKVTEKKKNILFDLSDNTGKMEVLGVRNEDTMKCKEGDKVRLTFFTLSKNGEKLQLTSGVHSTIKVIKAK 3rn2 A 2.55 BS02 dna L 0 K162 K163 R244 N287 K16 K17 R98 N141 ? 0002218,0035458 remove_due_to_license_issue O14862 22483801 1 ~ 20 EGFQKRCLPVMVLKAKKPFTFETQEGKQEMFHATVATEKEFFFVKVFNTLLKDKFIPKRIIIIARYYRHSGFLEVNSASRVLDAESDQKVNVPLNIIRKAGETPKINTLQTQPLGTIVNGLFVVQKVTEKKKNILFDLSDNTGKMEVLGVRNEDTMKCKEGDKVRLTFFTLSKNGEKLQLTSGVHSTIKVIKAK 3rn2 B 2.55 BS01 dna K 0 K204 G247 E248 T249 K58 G101 E102 T103 ? 0002218,0035458 remove_due_to_license_issue O14862 22483801 1 ~ 20 EGFQKRCLPVMVLKAKKPFTFETQEGKQEMFHATVATEKEFFFVKVFNTLLKDKFIPKRIIIIARYYRHSGFLEVNSASRVLDAESDQKVNVPLNIIRKAGETPKINTLQTQPLGTIVNGLFVVQKVTEKKKNILFDLSDNTGKMEVLGVRNEDTMKCKEGDKVRLTFFTLSKNGEKLQLTSGVHSTIKVIKA 3rn2 B 2.55 BS02 dna L 0 K162 K163 K198 R311 K335 I337 K16 K17 K52 R165 K189 I191 ? 0002218,0035458 remove_due_to_license_issue O14862 22483801 1 ~ 20 EGFQKRCLPVMVLKAKKPFTFETQEGKQEMFHATVATEKEFFFVKVFNTLLKDKFIPKRIIIIARYYRHSGFLEVNSASRVLDAESDQKVNVPLNIIRKAGETPKINTLQTQPLGTIVNGLFVVQKVTEKKKNILFDLSDNTGKMEVLGVRNEDTMKCKEGDKVRLTFFTLSKNGEKLQLTSGVHSTIKVIKA 3rni A 1.95 BS01 21Z A 1 V18 A31 F82 L83 H84 L134 D145 V18 A31 F78 L79 H80 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 424 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ro0 A 1.5 BS01 TPT A 1 F10 F13 N19 T45 A139 F142 C144 H168 F9 F12 N18 T44 A138 F141 C143 H167 E81 R91 C144 H168 E80 R90 C143 H167 3.4.19.3 0005737,0005829,0006508,0008234,0016920 remove_due_to_license_issue P46107 21875148 480 EKKVLLTGFDPFGGETVNPSWEAVKRLNGAAEGPASIVSEQVPTVFYKSLAVLREAMKKHQPDIIICVGQAGGRMQITPERVAINLNEARIPDNEGNQPVGEDISQGGPAAYWTGLPIKRIVEEIKKEGIPAAVSYTAGTFVCNHLFYGLMDEISRHHPHIRGGFIHIPYIPEQTLQKSAPSLSLDHITKALKIAAVTAAAHEDDIE 3ro4 A 2.6 BS01 LJ9 B 1 R108 A226 E227 P246 T253 A256 A285 R106 A224 E225 P244 T251 A254 A283 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=5360nM P50053 21767952 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3roc A 1.7 BS01 29A A 1 V30 A51 K53 I84 L104 T106 M109 G110 A111 V26 A47 K49 I80 L100 T102 M105 G106 A107 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Ki=193nM, IC50=12nM Q16539 21620699 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3rpr A 1.75 BS01 25Z A 1 I10 G11 E12 G13 V18 A31 K33 F82 L83 D86 K89 Q131 L134 I10 G11 E12 G13 V18 A31 K33 F74 L75 D78 K81 Q123 L126 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 529 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rpv A 1.8 BS01 26Z A 1 I10 V18 A31 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 V18 A31 F76 F78 L79 H80 Q81 D82 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 495 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rpy A 1.9 BS01 27Z A 1 I10 A31 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F74 L75 H76 Q77 D78 K81 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 470 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rqw A 2.913 BS01 ACH A 1 F19 Y38 N103 F9 Y28 N93 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802 remove_due_to_license_issue E0SJQ4 22395605 323 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 3rqw A 2.913 BS02 ACH E 1 E131 Y175 L178 F188 E121 Y165 L168 F178 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802 remove_due_to_license_issue E0SJQ4 22395605 323 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 3rqw B 2.913 BS01 ACH A 1 E131 F133 Y175 L178 F188 E121 F123 Y165 L168 F178 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802 remove_due_to_license_issue E0SJQ4 22395605 323 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 3rqw B 2.913 BS02 ACH B 1 F19 Y38 N103 F9 Y28 N93 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802 remove_due_to_license_issue E0SJQ4 22395605 323 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 3rr4 A 1.68 BS02 HRD A 1 S103 Y106 D156 C158 G229 L231 A232 M260 G261 S93 Y96 D142 C144 G215 L217 A218 M246 G247 D102 D280 C318 C320 C323 H349 D92 D266 C304 C306 C309 H335 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=28050nM remove_due_to_license_issue P28720 22736391 501 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSLTKQSEEGVTFKSHSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 3rsb A 2.8 BS01 GTP A 1 M6 A7 T12 R13 S50 E82 S99 M6 A7 T8 R9 S46 E70 S87 2.7.7.62 0005525,0008820,0009236,0016779,0043752 remove_due_to_license_issue Q58517 21542645 197 MDALIMATRMGGVEKPLIKLCGRCLIDYVVSPLLKSKVNNIFIATSPNTPKTKEYINSAYKDYKNIVVIEDLNECIGYFSEPFLVVSSDLINLKSKIINSIVDYFYCIKAKTPEALAVMIPKEKYPNPSIDFNGLVPADINVVSPKHGYQKEEIMVIDELIFNINTKDDLKLAEMLL 3rsr A 2.3 BS01 N5P A 1 D226 S227 I228 R256 I262 A263 G264 T265 D138 S139 I140 R168 I174 A175 G176 T177 C218 N406 C408 E410 C423 Y693 Y694 C130 N318 C320 E322 C335 Y605 Y606 1.17.4.1 0000166,0004748,0005515,0005524,0005634,0005737,0005971,0009263,0016491,0042802 Kd=44uM remove_due_to_license_issue P21524 22933704 841 QTTKQFSKVVEDLYRYVNAATGKPAPMISDDVYNIVMENKDKLNSAIVYDRDFQYSYFGFKTLERSYLLRINGQVAERPQHLIMRVALGIHGRDIEAALETYNLMSLKYFTHASPTLFNAGTPKPQMSSCFLVAMKEDSIEGIYDTLKECALISKTAGGIGLHIHNIRSTGSYIAGTNGTSNGLIPMIRVFNNTARYVFALYLEPWHADIFDFIDIRKDLFPALWIPDLFMKRVEENGTWTLFSPTSAPGLSDCYGDEFEALYTRYEKEGRGKTIKAQKLWYSILEAQTETGTPFVVYKDACNRKSNQKNLGVIKSSNLCCEIVEYSAPDETAVCNLASVALPAFIETSKTSTYNFKKLHEIAKVVTRNLNRVIDRNYYPVEEARKSNMRHRPIALGVQGLADTFMLLRLPFDSEEARLLNIQIFETIYHASMEASCELAQKDGPYETFQGSPASQGILQFDMWDQKPYGMWDWDTLRKDIMKHGVRNSLTMAPMPTTSQILGYNECFEPNPYLLRDLVDLGIWQYLITQNGSIQGLPNVPQELKDLYKTVWEISQKTIINMAADRSVYIDQSHSLNLFLRAPTMGKLTSMHFYGWKKGLKTGMYYLRTQ 3rsv A 2.5 BS01 3RS A 1 D32 G34 Y71 K75 W76 F108 R128 Y198 D228 D34 G36 Y73 K77 W78 F110 R130 Y190 D220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.0007uM remove_due_to_license_issue IC50=0.700000nM P56817 21707077 400 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rsx A 2.48 BS01 RSV A 1 D32 Y71 K75 W76 F108 D228 D34 Y73 K77 W78 F110 D221 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D221 T224 3.4.23.46 0004190,0006508,0016020 Kd=38.8uM remove_due_to_license_issue Kd=38800nM P56817 21707077 397 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rt4 C 1.7 BS01 LP5 C 1 L64 W66 A92 H93 G95 P96 N99 L64 W66 A92 H93 G95 P96 N99 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 Kd=1.6nM remove_due_to_license_issue Q9GK12 21454594 501 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3rt4 D 1.7 BS01 LP5 C 1 G95 P96 T97 W98 K144 D148 V149 Q150 P151 G95 P96 T97 W98 K144 D148 V149 Q150 P151 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 21454594 501 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3rt6 B 2.836 BS01 FWD B 1 Y61 P89 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y58 P86 L87 T88 R93 L135 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 remove_due_to_license_issue Ki=18nM, EC50=20900nM P19492 21464198 401 RTIVVTTILESPYVMYKKNHEQLEGNERYEGYCVDLAYEIAKHVRIKYKLSIVGDGKYGARDPETKIWNGMVGELVYGRADIAVAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWSYMKSAEPSVFTKTTADGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSALGTPVNLAVLKLSEQGILDKLKNKWWYDKGEC 3rt8 A 2.426 BS01 CWD A 1 Y61 T91 R96 G141 S142 T143 L192 E193 Y58 T88 R93 G138 S139 T140 L189 E190 ? 0015276,0016020 remove_due_to_license_issue Ki=451nM P19492 21464198 401 RTIVVTTILESPYVMYKKNHEQLEGNERYEGYCVDLAYEIAKHVRIKYKLSIVGDGKYGARDPETKIWNGMVGELVYGRADIAVAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWSYMKSAEPSVFTKTTADGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSALGTPVNLAVLKLSEQGILDKLKNKWWYDKGEC 3rtf B 1.7 BS01 CWD B 1 Y61 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y58 T88 R93 L135 G138 S139 T140 L189 E190 M193 ? 0015276,0016020 remove_due_to_license_issue Ki=45nM, EC50=2110nM P19491 21464198 800 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3rth A 2.7 BS01 RTH A 1 D32 Y71 K75 W76 F108 I118 D228 D34 Y73 K77 W78 F110 I120 D220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue Kd=6100nM P56817 21707077 397 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rti A 2.8 BS01 FMP A 1 Y80 V81 G121 N122 Y123 I172 E177 R180 Y75 V76 G116 N117 Y118 I167 E172 R175 V81 E177 R180 V76 E172 R175 3.2.2.22 0017148,0030598 remove_due_to_license_issue P02879 1433290 301 YPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPP 3rtm A 2.76 BS01 RTM A 1 D32 S35 D228 G230 T231 D34 S37 D219 G221 T222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue Kd=38400nM P56817 21707077 395 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rtn A 2.7 BS01 RTN A 1 D32 G34 Y71 K75 W76 Y198 D228 D34 G36 Y73 K77 W78 Y189 D219 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=74nM P56817 21707077 401 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQATPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rtp A 2.4 BS01 34I A 1 I70 V78 A91 M146 E147 L148 M149 D150 A151 V196 L206 I25 V30 A43 M98 E99 L100 M101 D102 A103 V148 L158 D189 K191 N194 D207 T226 D141 K143 N146 D159 T163 2.7.11.24 0004672,0004707,0005524,0006468 ic50=7nM remove_due_to_license_issue IC50=<100nM P53779 21813278 1 NQFYSVEVGDSTFTVLKRYQNLKPIGSGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPLDEREHTIEEWKELIYKEVMN 3ru1 A 2.3 BS01 3RU A 1 D32 G34 S35 V69 Y71 Y198 D228 D34 G36 S37 V71 Y73 Y189 D219 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 Kd=14.2uM remove_due_to_license_issue Kd=14200nM P56817 21707077 398 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rup A 1.99 BS01 ADP A 1 Y82 G83 G164 G165 R167 F193 K238 R292 V295 E296 R338 D382 Y82 G83 G164 G165 R167 F193 K238 R292 V295 E296 R338 D382 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 remove_due_to_license_issue P24182 21592965 1000 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKL 3rup A 1.99 BS02 ADP A 2 K116 K159 G164 G166 M169 E201 K202 Y203 L204 H209 Q233 H236 L278 E288 I437 K116 K159 G164 G166 M169 E201 K202 Y203 L204 H209 Q233 H236 L278 E288 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 remove_due_to_license_issue P24182 21592965 1002 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKL 3rux A 1.7 BS01 BS5 A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 I83 N130 K138 G141 I142 V155 G156 N158 V166 D167 A170 S37 T38 N39 Q62 G65 R66 G67 R68 R71 G72 W73 A74 I82 N129 K137 G140 I141 V154 G155 N157 V165 D166 A169 R69 K138 R266 R68 K137 R265 6.3.4.15 0004077,0005737,0016874,0036094,0036211,0043687 Kd=0.53nM remove_due_to_license_issue Kd=0.865000nM P96884 22118677 1001 TDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 3rv3 A 1.91 BS01 ADP A 1 Y82 G83 G164 G165 R167 F193 K238 R292 Q294 V295 E296 R338 D382 Y85 G86 G167 G168 R170 F196 K241 R295 Q297 V298 E299 R341 D385 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K119 K162 D199 H212 R238 T277 E279 E291 N293 R295 E299 R341 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 remove_due_to_license_issue P24182 21592965 1000 GSHMLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKL 3rv3 A 1.91 BS02 ADP A 2 K116 K159 G164 G165 G166 M169 E201 K202 Y203 L204 H209 Q233 H236 L278 E288 I437 K119 K162 G167 G168 G169 M172 E204 K205 Y206 L207 H212 Q236 H239 L281 E291 I440 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K119 K162 D199 H212 R238 T277 E279 E291 N293 R295 E299 R341 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 remove_due_to_license_issue P24182 21592965 1002 GSHMLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKL 3rv4 A 1.98 BS01 ADP A 1 K116 K159 G164 G166 M169 K202 Y203 L204 H209 Q233 H236 L278 I287 E288 I437 K116 K159 G164 G166 M169 K202 Y203 L204 H209 Q233 H236 L278 I287 E288 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 remove_due_to_license_issue P24182 21592965 1000 MLDKIVIANRGEIALEILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 3rv6 A 2.04 BS01 VAE A 1 L268 G270 E297 Y385 L404 A418 G419 K438 L254 G256 E271 Y352 L371 A385 G386 K405 K205 E252 A269 E297 T361 Y385 R405 G421 E434 K438 K191 E238 A255 E271 T328 Y352 R372 G388 E401 K405 4.2.99.21,5.4.4.2,5.4.99.5 0000162,0000287,0004106,0005886,0008909,0009058,0009697,0010106,0016829,0016833,0016853,0019540,0043904,0046872,0052572 Ki=21uM remove_due_to_license_issue P9WFX1 22607697 451 SSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTRADDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVARQ 3rv7 A 2.5 BS01 RVB A 1 P251 L268 T271 H334 T361 Y385 L404 R405 A418 G419 K438 P237 L254 T257 H301 T328 Y352 L371 R372 A385 G386 K405 K205 E252 A269 E297 H334 T361 Y385 R405 G421 E434 K438 K191 E238 A255 E270 H301 T328 Y352 R372 G388 E401 K405 4.2.99.21,5.4.4.2,5.4.99.5 0000162,0000287,0004106,0005886,0008909,0009058,0009697,0010106,0016829,0016833,0016853,0019540,0043904,0046872,0052572 Ki=14uM remove_due_to_license_issue P9WFX1 22607697 451 SSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTRDDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRHLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVAR 3rv8 A 2.29 BS01 RVC A 1 L268 T361 Y385 L404 R405 G419 K438 L254 T329 Y353 L372 R373 G387 K406 K205 E252 A269 E297 H334 T361 Y385 R405 G421 E434 K438 K191 E238 A255 E269 H302 T329 Y353 R373 G389 E402 K406 4.2.99.21,5.4.4.2,5.4.99.5 0000162,0000287,0004106,0005886,0008909,0009058,0009697,0010106,0016829,0016833,0016853,0019540,0043904,0046872,0052572 Ki=12uM remove_due_to_license_issue P9WFX1 22607697 451 SSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTDDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRVQHLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVARQ 3rv9 A 2.14 BS01 RVD A 1 T361 Y385 L404 R405 A418 G419 K438 T331 Y355 L374 R375 A388 G389 K408 K205 E252 A269 E297 H334 T361 Y385 R405 G421 E434 K438 K191 E238 A255 E272 H304 T331 Y355 R375 G391 E404 K408 4.2.99.21,5.4.4.2,5.4.99.5 0000162,0000287,0004106,0005886,0008909,0009058,0009697,0010106,0016829,0016833,0016853,0019540,0043904,0046872,0052572 Ki=12uM remove_due_to_license_issue P9WFX1 22607697 451 SSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTLARDDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRQHLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVARQ 3rvg A 2.498 BS01 17P A 1 L855 A880 E930 Y931 L932 G935 L983 L15 A40 E90 Y91 L92 G95 L143 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5nM remove_due_to_license_issue O60674 21942426 2000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVSPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 3rvi A 2.65 BS01 RVI A 1 D32 G34 S35 Y71 K75 W76 F108 Y198 I226 D228 D34 G36 S37 Y73 K77 W78 F110 Y189 I217 D219 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=11nM P56817 21707077 402 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3rw6 A 2.3 BS01 rna H 0 T123 Y126 E151 H153 Y154 R158 I190 N192 R233 V246 N248 N275 R276 Y278 K304 S305 T6 Y9 E34 H36 Y37 R41 I73 N75 R116 V129 N131 N158 R159 Y161 K187 S188 ? 0003676,0003723,0005737,0006406 remove_due_to_license_issue Q9UBU9 21822283 1 ~ 62 NWFKITIPYGRKYDKAWLLSMIQSKCSVPFTPIEFHYENTRAQFFVEDASTASALKAVNYKILDRENRRISIIINSSAPPHTILNELKPEQVEQLKLIMSKRYDGSQQALDLKGLRSDPDLVAQNIDVVLNRRSCMAATLRIIEENIPELLSLNLSNNRLYRLDDMSSIVQKAPNLKILNLSGNELKSERELDKIKGLKLEELWLDGNSLCDTFRDQSTYISAIRERFPKLLRLDGHELPPPIAF 3rw6 B 2.3 BS01 rna F 0 T123 P125 Y126 E151 H153 Y154 N156 R158 Y177 N192 H198 R233 V246 N248 N275 R276 Y278 R279 K304 S305 T7 P9 Y10 E35 H37 Y38 N40 R42 Y61 N76 H82 R117 V130 N132 N159 R160 Y162 R163 K188 S189 ? 0003676,0003723,0005737,0006406 remove_due_to_license_issue Q9UBU9 21822283 1 ~ 62 KNWFKITIPYGRKYDKAWLLSMIQSKCSVPFTPIEFHYENTRAQFFVEDASTASALKAVNYKILDRENRRISIIINSSAPPHTILNELKPEQVEQLKLIMSKRYDGSQQALDLKGLRSDPDLVAQNIDVVLNRRSCMAATLRIIEENIPELLSLNLSNNRLYRLDDMSSIVQKAPNLKILNLSGNELKSERELDKIKGLKLEELWLDGNSLCDTFRDQSTYISAIRERFPKLLRLDGHELPPPI 3rw9 A 2.0 BS01 DSH A 1 Q49 Q70 G101 G103 E124 I125 D155 G156 D173 S174 P180 A181 L184 Q35 Q56 G87 G89 E110 I111 D141 G142 D159 S160 P162 A163 L166 2.5.1.16 0003824,0004766,0005515,0005829,0006595,0008295,0016740,0042802,0042803,1990830 Kd=1.1uM remove_due_to_license_issue P19623 21898642 303 AIREGWFRETCSLWPGQALSLQVEQLLHHRRSRYQDILVFRSKTYGNVLVLDGVIQCTERDEFSYQEMIANLPLCSHPNPRKVLIIGGGDGGVLREVVKHPSVESVVQCEIDEDVIQVSKKFLPGMAIGYSSSKLTLHVGDGFEFMKQNQDAFDVIITDSGPAESLFKESYYQLMKTALKEDGVLCCQGECQWLHLDLIKEMRQFCQSLFPVVAYAYCTIPTYPSGQIGFMLCSKNPSTNFQEPVQPLTQQQVAQMQLKYYNSDVHRAAFVLPEFARKALND 3rwp A 1.92 BS01 ABQ A 1 L88 G89 E90 G91 T95 V96 A109 K111 A162 E166 E209 L212 T222 D223 L16 G17 E18 G19 T23 V24 A37 K39 A90 E94 E137 L140 T150 D151 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T164 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.6nM remove_due_to_license_issue Ki=0.600000nM O15530 22040023 360 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3rwq A 2.55 BS01 3RW A 1 L88 G89 E90 G91 V96 A109 K111 A162 L212 T222 D223 L17 G18 E19 G20 V25 A38 K40 A91 L141 T151 D152 D205 K207 E209 N210 D223 T245 D134 K136 E138 N139 D152 T170 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=35nM O15530 22040023 1 PQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3rx5 A 1.99 BS04 G2I A 1 A144 D146 Y300 W343 W401 Q487 E515 Y519 W520 A140 D142 Y296 W339 W397 Q483 E511 Y515 W516 D143 D146 Y300 E515 D139 D142 Y296 E511 3.2.1.4 0004553,0005975,0008810,0016798,0030245,0046872 remove_due_to_license_issue Q9AJS0 21785782 604 VPKSIFYNQVGYLISGDKRFWIQAHEPQPFALRTPEGQAVFAGMTKPVGGNWYVGDFTALRVPGTYTLTVGTLEARVVIHRRAYRDVLEAMLRFFDYQLCGVVLPEDEAGPWAHGACHTSDAKVFGTERALACPGGWHDAGDYGKYTVPAAKAVADLLLAHEYFPAALAHVRPMRSVHRAPHLPPALEVAREEIAWLLTMQDPATGGVYHKVTTPSFPPLDTRPEDDDAPLVLSPISYAATATFCAAMAHAALVYRPFDPALSSCCADAARRAYAWLGAHEMQPFHNPDGILTGEYGDAELRDELLWASCALLRMTGDSAWARVCEPLLDLDLPWELGWADVALYGVMDYLRTPRAAVSDDVRNKVKSRLLRELDALAAMAESHPFGIPMRDDDFIWGSNMVLLNRAMAFLLAEGVGVLHPAAHTVAQRAADYLFGANPLGQCYVTGFGQRPVRHPHHRPSVADDVDHPVPGMVVGGPNRHLQDEIARAQLAGRPAMEAYIDHQDSYSTNEVAVYWNSPAVFVIAALLEA 3rx7 A 2.02 BS03 G3I A 1 A144 D146 Y300 W343 W401 H485 E515 Y519 A140 D142 Y296 W339 W397 H481 E511 Y515 D143 D146 Y300 E515 D139 D142 Y296 E511 3.2.1.4 0004553,0005975,0008810,0016798,0030245,0046872 remove_due_to_license_issue Q9AJS0 21785782 604 VPKSIFYNQVGYLISGDKRFWIQAHEPQPFALRTPEGQAVFAGMTKPVGGNWYVGDFTALRVPGTYTLTVGTLEARVVIHRRAYRDVLEAMLRFFDYQLCGVVLPEDEAGPWAHGACHTSDAKVFGTERALACPGGWHDAGDYGKYTVPAAKAVADLLLAHEYFPAALAHVRPMRSVHRAPHLPPALEVAREEIAWLLTMQDPATGGVYHKVTTPSFPPLDTRPEDDDAPLVLSPISYAATATFCAAMAHAALVYRPFDPALSSCCADAARRAYAWLGAHEMQPFHNPDGILTGEYGDAELRDELLWASCALLRMTGDSAWARVCEPLLDLDLPWELGWADVALYGVMDYLRTPRAAVSDDVRNKVKSRLLRELDALAAMAESHPFGIPMRDDDFIWGSNMVLLNRAMAFLLAEGVGVLHPAAHTVAQRAADYLFGANPLGQCYVTGFGQRPVRHPHHRPSVADDVDHPVPGMVVGGPNRHLQDEIARAQLAGRPAMEAYIDHQDSYSTNEVAVYWNSPAVFVIAALLEA 3rx8 A 2.56 BS03 9MR A 1 F221 H461 R463 Y511 E515 F215 H455 R457 Y505 E509 D143 D146 Y300 E515 D137 D140 Y294 E509 3.2.1.4 0004553,0005975,0008810,0016798,0030245,0046872 remove_due_to_license_issue Q9AJS0 21785782 603 KSIFYNQVGYLISGDKRFWIQAHEPQPFALRTPEGQAVFAGMTKPVGGNWYVGDFTALRVPGTYTLTVGTLEARVVIHRRAYRDVLEAMLRFFDYQLCGVVLPEDEAGPWAHGACHTSDAKVFGTERALACPGGWHDAGDYGKYTVPAAKAVADLLLAHEYFPAALAHVRPMRSVHRAPHLPPALEVAREEIAWLLTMQDPATGGVYHKVTTPSFPPLDTRPEDDDAPLVLSPISYAATATFCAAMAHAALVYRPFDPALSSCCADAARRAYAWLGAHEMQPFHNPDGILTGEYGDAELRDELLWASCALLRMTGDSAWARVCEPLLDLDLPWELGWADVALYGVMDYLRTPRAAVSDDVRNKVKSRLLRELDALAAMAESHPFGIPMRDDDFIWGSNMVLLNRAMAFLLAEGVGVLHPAAHTVAQRAADYLFGANPLGQCYVTGFGQRPVRHPHHRPSVADDVDHPVPGMVVGGPNRHLQDEIARAQLAGRPAMEAYIDHQDSYSTNEVAVYWNSPAVFVIAALLEA 3rx8 A 2.56 BS04 9MR A 2 D143 D146 G298 Y300 W343 W401 E515 Y519 D137 D140 G292 Y294 W337 W395 E509 Y513 D143 D146 Y300 E515 D137 D140 Y294 E509 3.2.1.4 0004553,0005975,0008810,0016798,0030245,0046872 remove_due_to_license_issue Q9AJS0 21785782 601 KSIFYNQVGYLISGDKRFWIQAHEPQPFALRTPEGQAVFAGMTKPVGGNWYVGDFTALRVPGTYTLTVGTLEARVVIHRRAYRDVLEAMLRFFDYQLCGVVLPEDEAGPWAHGACHTSDAKVFGTERALACPGGWHDAGDYGKYTVPAAKAVADLLLAHEYFPAALAHVRPMRSVHRAPHLPPALEVAREEIAWLLTMQDPATGGVYHKVTTPSFPPLDTRPEDDDAPLVLSPISYAATATFCAAMAHAALVYRPFDPALSSCCADAARRAYAWLGAHEMQPFHNPDGILTGEYGDAELRDELLWASCALLRMTGDSAWARVCEPLLDLDLPWELGWADVALYGVMDYLRTPRAAVSDDVRNKVKSRLLRELDALAAMAESHPFGIPMRDDDFIWGSNMVLLNRAMAFLLAEGVGVLHPAAHTVAQRAADYLFGANPLGQCYVTGFGQRPVRHPHHRPSVADDVDHPVPGMVVGGPNRHLQDEIARAQLAGRPAMEAYIDHQDSYSTNEVAVYWNSPAVFVIAALLEA 3rxa A 1.7 BS02 SZ1 A 1 S190 V209 S172 V191 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 7 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxb A 1.7 BS02 ALG A 1 D189 S190 C191 W211 G214 D171 S172 C173 W193 G196 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 6 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxd A 1.7 BS02 SZ4 A 1 D189 S190 C191 Q192 V209 W211 G214 D171 S172 C173 Q174 V191 W193 G196 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 6 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxg A 1.7 BS02 SZ3 A 1 S190 C191 V209 W211 S172 C173 V191 W193 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 8 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxh A 1.7 BS02 HSM A 1 S190 C191 Q192 S195 S172 C173 Q174 S177 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 7 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxi A 1.6 BS02 TSS A 1 S190 C191 Q192 S195 W211 C215 S172 C173 Q174 S177 W193 C197 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 6 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxj A 1.7 BS02 GBS A 1 H58 D189 S190 S195 V209 S210 W211 G212 G214 H40 D171 S172 S177 V191 S192 W193 G194 G196 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 9 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxk A 1.6 BS02 SZ8 A 1 S190 Q192 C215 S172 Q174 C197 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 8 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxl A 1.7 BS02 SZ9 A 1 D189 S190 C191 S195 V209 W211 G212 G214 D171 S172 C173 S177 V191 W193 G194 G196 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 6 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxm A 1.7 BS02 SW1 A 1 D189 S190 C191 Q192 W211 D171 S172 C173 Q174 W193 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 8 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxo A 1.6 BS02 SW2 A 1 D189 S190 C191 Q192 V209 W211 G214 D171 S172 C173 Q174 V191 W193 G196 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 7 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3rxp A 1.6 BS02 SW3 A 1 D189 S190 C191 S195 V209 W211 D171 S172 C173 S177 V191 W193 H58 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 7 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 3ry8 A 1.4 BS01 FLC A 1 N355 R356 D385 N127 R128 D157 ? Kd=460uM remove_due_to_license_issue Q5F4T5 22031945 1 KPFTLPILTLGELTNSRFPLPIDVLYTNPNESAIVQCQNGRCTLDGELQGTTQLLPTGICAFRGKVTQQVQGTHWNMTVTNLNGTPFDPTEDVPAPLGTPDFSGQIYGVISQRNTNTVPGEGNLPANRAHEAVIATYSPKFTPKLGNIQFSTWETQDVSSGQPTKFTPVGLASVDANSHFDQWTLPSYSGALTLNMNLAPSVAPVFPGECLLFFRSFIPLKGGYGNPAIDCLMPQEWVQHLYQESAPSLSDVALVRYVNPETGRTLFEAKLHRNGFLTVARNSAGPVVAPTNGYFRFDSWVNQFYTLAPM 3ryj B 1.39 BS02 RYJ B 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=16nM remove_due_to_license_issue P00918 21790183 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ryv B 1.2 BS02 RYV B 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=86nM remove_due_to_license_issue P00918 21790183 1 HWGYGGHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ryw A 2.9 BS01 K9H A 1 F122 A125 D126 R135 Q195 K243 D287 K301 F88 A91 D92 R101 Q161 K205 D249 K263 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3ryw A 2.9 BS04 K9H D 1 V153 L157 V119 L123 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3ryw D 2.9 BS01 K9H A 1 V153 L157 V119 L123 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3ryw D 2.9 BS02 K9H D 1 F122 A125 D126 D130 R135 T191 Q195 K243 D287 K301 F88 A91 D92 D96 R101 T157 Q161 K205 D249 K263 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A87 D92 D96 R101 D164 K205 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 22392982 2001 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIAVDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVGSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 3ryx B 1.6 BS02 RYX B 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=7.3nM remove_due_to_license_issue P00918 21790183 1 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ryy A 1.16 BS02 RYY A 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=38nM remove_due_to_license_issue P00918 21790183 262 HWGYGGHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ryy A 1.16 BS03 RYY A 2 D180 G183 D176 G179 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=38nM remove_due_to_license_issue P00918 21790183 263 HWGYGGHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3ryz A 1.37 BS02 RYZ A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=2.4nM remove_due_to_license_issue P00918 21790183 262 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rz0 B 1.798 BS02 RZ0 B 1 H94 H119 F131 L198 T199 T200 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=28nM remove_due_to_license_issue P00918 21790183 1 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rz1 B 1.51 BS02 RZ1 B 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.8nM remove_due_to_license_issue P00918 21790183 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rz3 A 2.3 BS01 U94 A 1 I45 P48 T51 Y52 Y53 F58 I128 N132 Y161 I40 P43 T46 Y47 Y48 F53 I109 N113 Y142 C93 C88 2.3.2.23,2.3.2.24 ic50=1.72uM remove_due_to_license_issue P49427 21683433 1 SPSSQKALLLELKGLQEEPVEGFRVTLVDEGDLYNWEVAIFGPPNTYYEGGYFKARLKFPIDYPYSPPAFRFLTKMWHPNIYETGDVCISILERWNPTQNVRTILLSVISLLNEPNTFSPANVDASVMYRKWKESKGKDREYTDIIRKQVLGTKVDAERDGVKV 3rz5 A 1.65 BS02 RZ5 A 1 H94 H119 F131 V135 L198 T199 T200 H92 H117 F128 V132 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=13nM remove_due_to_license_issue P00918 21790183 262 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rz7 A 1.8 BS02 RZ7 A 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.1nM remove_due_to_license_issue P00918 21790183 262 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rz8 A 1.7 BS02 RZ8 A 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=6.7nM remove_due_to_license_issue P00918 21790183 262 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3rzb A 1.9 BS01 02Z A 1 I10 A31 E81 F82 L83 H84 D86 L134 D145 I10 A31 E73 F74 L75 H76 D78 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 458 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3rzi A 1.95 BS03 TRP A 1 K123 L194 N237 L238 T240 K118 L189 N232 L233 T235 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 remove_due_to_license_issue O53512 22154807 465 NWTVDIPIDQPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 3rzi B 1.95 BS03 TRP B 1 K123 A192 N237 L238 T240 A241 K118 A187 N232 L233 T235 A236 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 remove_due_to_license_issue O53512 22154807 466 MNWTVDIPILPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 3s00 A 1.8 BS01 Z60 A 1 I10 A31 K33 F82 L83 H84 N132 L134 I10 A31 K33 F78 L79 H80 N128 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 461 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3s0b A 1.22 BS01 FNA A 1 L51 F54 I68 V71 M72 L75 L103 V104 V107 T112 M113 L51 F54 I68 V71 M72 L75 L103 V104 V107 T112 M113 0005549 Kd=0.32uM remove_due_to_license_issue 22075131 120 MTIEELKTRLHTEQSVCKTETGIDQQKANDVIEGNIDVEDKKVQLYCECILKNFNILDKNNVFKPQGIKAVMELLIDENSVKQLVSDCSTISEENPHLKASKLVQCVSKYKTMKSVDFL 3s0d A 1.24 BS01 CTV A 1 F54 V71 V104 V107 K111 M113 F54 V71 V104 V107 K111 M113 0005549 Kd=280nM remove_due_to_license_issue 22075131 120 MTIEELKTRLHTEQSVCKTETGIDQQKANDVIEGNIDVEDKKVQLYCECILKNFNILDKNNVFKPQGIKAVMELLIDENSVKQLVSDCSTISEENPHLKASKLVQCVSKYKTMKSVDFL 3s0e A 1.6 BS01 EOL A 1 I56 V71 V107 S108 K111 T112 M113 I56 V71 V107 S108 K111 T112 M113 0005549 Kd=90nM remove_due_to_license_issue 22075131 120 MTIEELKTRLHTEQSVCKTETGIDQQKANDVIEGNIDVEDKKVQLYCECILKNFNILDKNNVFKPQGIKAVMELLIDENSVKQLVSDCSTISEENPHLKASKLVQCVSKYKTMKSVDFL 3s0j A 2.0 BS01 Z15 A 1 G135 L136 D283 N284 D339 H341 H377 T378 N484 E672 S674 G675 G124 L125 D266 N267 D313 H315 H351 T352 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=169.9uM remove_due_to_license_issue IC50=169900nM P00489 21821421 998 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3s0n A 1.95 BS02 0BB A 1 H45 L86 A177 F178 K179 S182 S197 Y198 G199 R200 H45 L86 A177 F178 K179 S182 S197 Y198 G199 R200 H45 D89 K179 G180 D181 S182 G183 H45 D89 K179 G180 D181 S182 G183 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 ic50=180nM remove_due_to_license_issue IC50=180nM P23946 21733690 230 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPSQKNFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 3s0o A 2.0 BS01 50Z A 1 I10 V18 A31 F82 L83 L134 D145 I10 V18 A31 F79 L80 L131 D142 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T153 T160 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 446 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3s1g A 1.82 BS02 ITE A 1 Y106 D156 C158 G229 G230 L231 A232 M260 G261 Y96 D132 C134 G205 G206 L207 A208 M236 G237 D102 D280 C318 C320 C323 H349 D92 D256 C294 C296 C299 H325 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=6500nM remove_due_to_license_issue P28720 22736391 501 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVKQSEEGVTFKHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 3s1h A 1.75 BS01 56Z A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F72 F74 L75 H76 Q77 D78 K81 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 479 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3s1y A 1.4 BS01 S1Y A 1 S90 Q146 Y177 N179 V239 G240 P241 G242 Y249 T343 G344 S345 S62 Q118 Y149 N151 V211 G212 P213 G214 Y221 T315 G316 S317 S90 K93 Y177 E299 K342 S345 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 21676616 398 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLEQ 3s22 A 1.65 BS01 3S2 A 1 S90 Q146 Y177 N179 Y249 T343 G344 S345 S62 Q118 Y149 N151 Y221 T315 G316 S317 S90 K93 Y177 E299 K342 S345 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 21676616 1 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLEQ 3s2a A 2.55 BS01 2NQ A 1 P810 I831 K833 Y867 I879 E880 V882 N951 M953 I963 D964 P567 I588 K590 Y624 I636 E637 V639 N708 M710 I720 D721 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=8.1nM P48736 21612232 1103 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAIDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKETVSLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNHPIALPKHQEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 3s2o A 2.6 BS01 EV6 A 1 D32 Y71 W76 D228 G230 N385 D34 Y73 W78 D220 G222 N377 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=8900nM P56817 20656487 393 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3s2p A 2.3 BS01 PMU A 1 F82 L83 H84 Q85 D86 K89 Q131 N132 L134 D145 F74 L75 H76 Q77 D78 K81 Q123 N124 L126 D137 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T146 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.068uM remove_due_to_license_issue IC50=68nM P24941 21684737 500 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3s2v A 2.5 BS01 3HU A 1 E13 Y16 Y61 P88 L89 T90 R95 V137 S141 T142 E190 S193 E10 Y13 Y58 P85 L86 T87 R92 V134 S138 T139 E187 S190 ? 0015276,0016020 Ki=157nM remove_due_to_license_issue Ki=157nM P22756 21619066 258 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 3s3i A 1.8 BS01 CQ0 A 1 A51 K53 E71 T106 L108 L167 D168 F169 A48 K50 E68 T103 L105 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 22521646 1 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3s3k B 3.2 BS01 CSN B 1 K154 C242 A244 V246 Q286 K134 C222 A224 V226 Q266 D210 C242 R248 S249 Q286 D190 C222 R228 S229 Q266 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P35992 22007620 308 MASRPILIKNFAEHYRLMSADSDFRFSEEFEELKHVGRDQPCTFADLPCNRPKNRFTNILPYDHSRFKLQPVDDDEGSDYINANYVPGHNSPREFIVTQGPLHSTRDDFWRMCWESNSRAIVMLTRCFEKGREKCDQYWPNDTVPVFYGDIKVQILNDSHYADWVMTEFMLCRGSEQRILRHFHFTTWPDFGVPNPPQTLVRFVRAFRDRIGAEQRPIVVHCSAGVGRSGTFITLDRILQQINTSDYVDIFGIVYAMRKERVWMVQTEQQYICIHQCLLAVLEGK 3s3m A 2.49 BS06 DLU A 1 D128 D185 G187 Y212 P214 E221 D121 D178 G180 Y205 P207 E214 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0015074 remove_due_to_license_issue P14350 21719464 398 LDAELDQLLQGHYIKGYPKQYTYFLEDGKVKVSRPEGVKIIPPQSDRQKIVLQAHNLAHTGREATLLKIANLYWWPNMRKDVVKQLGRCQQCLITNASNKASGPILRPDRPQKPFDKFFIDYIGPLPPSQGYLYVLVVVDGMTGFTWLYPTKAPSTSATVKSLNVLTSIAIPKVIHSDQGAAFTSSTFAEWAKERGIHLEFSTPYHPQSSGKVERKNSDIKRLLTKLLVGRPTKWYDLLPVVQLALNNTYSPVLKYTPHQLLFGIDSNTPFANQDTLDLTREEELSLLQEIRTSLYHPSTPPASSRSWSPVVGQLVQERVARPASLRPRWHKPSTVLKVLNPRTVVILDHLGNNRTVSIDNLKPTSHQ 3s3n A 2.49 BS06 DLU A 1 D128 D185 P214 Q215 E221 D121 D178 P207 Q208 E214 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0015074 remove_due_to_license_issue P14350 21719464 398 LDAELDQLLQGHYIKGYPKQYTYFLEDGKVKVSRPEGVKIIPPQSDRQKIVLQAHNLAHTGREATLLKIANLYWWPNMRKDVVKQLGRCQQCLITNASNKASGPILRPDRPQKPFDKFFIDYIGPLPPSQGYLYVLVVVDGMTGFTWLYPTKAPSTSATVKSLNVLTSIAIPKVIHSDQGAAFTSSTFAEWAKERGIHLEFSTPYHPQSHGKVERKNSDIKRLLTKLLVGRPTKWYDLLPVVQLALNNTYSPVLKYTPHQLLFGIDSNTPFANQDTLDLTREEELSLLQEIRTSLYHPSTPPASSRSWSPVVGQLVQERVARPASLRPRWHKPSTVLKVLNPRTVVILDHLGNNRTVSIDNLKPTSHQ 3s3o A 2.55 BS06 DLU A 1 D128 D185 Y212 P214 E221 D121 D178 Y205 P207 E214 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0015074 remove_due_to_license_issue P14350 21719464 399 LDAELDQLLQGHYIKGYPKQYTYFLEDGKVKVSRPEGVKIIPPQSDRQKIVLQAHNLAHTGREATLLKIANLYWWPNMRKDVVKQLGRCQQCLITNASNKASGPILRPDRPQKPFDKFFIDYIGPLPPSQGYLYVLVVVDGMTGFTWLYPTKAPSTSATVKSLNVLTSIAIPKVIHSDQGAAFTSSTFAEWAKERGIHLEFSTPYHPQSSGKVERKHSDIKRLLTKLLVGRPTKWYDLLPVVQLALNNTYSPVLKYTPHQLLFGIDSNTPFANQDTLDLTREEELSLLQEIRTSLYHPSTPPASSRSWSPVVGQLVQERVARPASLRPRWHKPSTVLKVLNPRTVVILDHLGNNRTVSIDNLKPTSHQ 3s3q A 1.8 BS01 C1P A 1 Q94 G98 C100 W101 E142 G143 G144 L146 I193 V247 G269 H270 W292 Q25 G29 C31 W32 E73 G74 G75 L77 I124 V178 G200 H201 W223 Q94 C100 H270 N290 Q25 C31 H201 N221 3.4.22.1 0006508,0008234 remove_due_to_license_issue Q8MNY2 21832058 1 VEIPSSFDSRKKWPRCKSIATIRDQSRCGSCWAFGAVEAMSDRSCIQSGGKQNVELSAVDLLSCCESCGLGCEGGILGPAWDYWVKEGIVTGSSKENHAGCEPYPFPKCEHHTKGKYPPCGSKIYKTPRCKQTCQKKYKTPYTQDKHRGKSSYNVKNDEKAIQKEIMKYGPVEAGFTVYEDFLNYKSGIYKHITGETLGGHAIRIIGWGVENKAPYWLIANSWNEDWGENGYFRIVRGRDECSIESEVTAGRIN 3s3r A 2.64 BS01 0IW A 1 Q94 G98 C100 W101 L139 E142 G143 G144 L146 G269 H270 Q25 G29 C31 W32 L70 E73 G74 G75 L77 G200 H201 Q94 C100 H270 N290 Q25 C31 H201 N221 3.4.22.1 0006508,0008234 remove_due_to_license_issue Q8MNY2 21832058 324 VEIPSSFDSRKKWPRCKSIATIRDQSRCGSCWAFGAVEAMSDRSCIQSGGKQNVELSAVDLLSCCESCGLGCEGGILGPAWDYWVKEGIVTGSSKENHAGCEPYPFPKCEHHTKGKYPPCGSKIYKTPRCKQTCQKKYKTPYTQDKHRGKSSYNVKNDEKAIQKEIMKYGPVEAGFTVYEDFLNYKSGIYKHITGETLGGHAIRIIGWGVENKAPYWLIANSWNEDWGENGYFRIVRGRDECSIESEVTAGRIN 3s3r A 2.64 BS02 0IW B 1 R79 P83 R10 P14 Q94 C100 H270 N290 Q25 C31 H201 N221 3.4.22.1 0006508,0008234 remove_due_to_license_issue Q8MNY2 21832058 324 VEIPSSFDSRKKWPRCKSIATIRDQSRCGSCWAFGAVEAMSDRSCIQSGGKQNVELSAVDLLSCCESCGLGCEGGILGPAWDYWVKEGIVTGSSKENHAGCEPYPFPKCEHHTKGKYPPCGSKIYKTPRCKQTCQKKYKTPYTQDKHRGKSSYNVKNDEKAIQKEIMKYGPVEAGFTVYEDFLNYKSGIYKHITGETLGGHAIRIIGWGVENKAPYWLIANSWNEDWGENGYFRIVRGRDECSIESEVTAGRIN 3s3v A 1.53 BS01 TOP A 1 V8 E30 F31 F34 K35 I60 L67 V8 E30 F31 F34 K35 I60 L67 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=593nM remove_due_to_license_issue IC50=680000nM, Ki=19070nM P00374 21684339 187 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFKRMTTTSSVEGKQNLVIMGKKTWFSIPEKFRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3s3v A 1.53 BS02 TOP A 2 S59 P61 F64 S59 P61 F64 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=593nM remove_due_to_license_issue IC50=680000nM, Ki=19070nM P00374 21684339 193 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFKRMTTTSSVEGKQNLVIMGKKTWFSIPEKFRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3s43 A 1.26 BS01 478 A 1 D25 G27 A28 D30 G48 I82 D25 G27 A28 D30 G48 I82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=2.53nM remove_due_to_license_issue Q7SSE3 22238126 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDEIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s43 B 1.26 BS01 478 A 1 D125 G127 A128 D130 V147 G149 I150 D25 G27 A28 D30 V47 G49 I50 D125 T126 G127 D25 T26 G27 ? 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 22238126 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s45 A 1.51 BS01 478 B 1 D25 A28 D30 I32 I82 I84 D25 A28 D30 I32 I82 I84 D25 T26 G27 D25 T26 G27 3.4.23.47 0004190,0006508,0046872 remove_due_to_license_issue Q9W9R3 22238126 201 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 3s45 B 1.51 BS01 478 B 1 D25 G27 A28 D30 G49 I50 I84 D25 G27 A28 D30 G49 I50 I84 D25 T26 G27 D25 T26 G27 3.4.23.47 0004190,0006508,0046872 Ki=3.24nM remove_due_to_license_issue Q9W9R3 22238126 201 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 3s4q A 2.27 BS01 NK0 A 1 K53 E71 I84 T106 L108 M109 G110 A111 L167 D168 F169 L171 K45 E63 I76 T98 L100 M101 G102 A103 L157 D158 F159 L161 D150 K152 N155 D168 T185 D140 K142 N145 D158 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=4nM remove_due_to_license_issue IC50=4nM Q16539 21705217 361 ERPTFYRQELNKTIWEVPERYQNLSPVGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAATRWYRAPEIMYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3s53 A 1.5 BS01 017 A 1 D25 G27 D29 D30 G48 I50 D25 G27 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.23nM remove_due_to_license_issue Q7SSI0 22238126 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s53 B 1.5 BS01 017 A 1 D25 A28 D30 I32 P81 D25 A28 D30 I32 P81 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.23nM remove_due_to_license_issue Q7SSI0 22238126 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s53 B 1.5 BS02 017 B 1 W42 P44 K55 V56 R57 V77 W42 P44 K55 V56 R57 V77 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.23nM remove_due_to_license_issue Q7SSI0 22238126 203 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s54 A 1.42 BS01 017 B 1 D25 A28 D30 P81 I82 I84 D25 A28 D30 P81 I82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 22238126 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s54 B 1.42 BS01 017 B 1 D25 G27 D29 D30 V47 G48 G49 I50 D25 G27 D29 D30 V47 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.23nM remove_due_to_license_issue Q7SSI0 22238126 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s56 A 1.88 BS01 ROC A 1 D25 G27 A28 D29 D30 G48 G49 I50 P81 I82 D25 G27 A28 D29 D30 G48 G49 I50 P81 I82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.24nM remove_due_to_license_issue Q7SSI0 22238126 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s56 B 1.88 BS01 ROC A 1 R8 D25 G48 G49 I50 I82 I84 R8 D25 G48 G49 I50 I82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.24nM remove_due_to_license_issue Q7SSI0 22238126 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s56 B 1.88 BS02 ROC B 1 R8 L10 E21 P81 I82 R8 L10 E21 P81 I82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.24nM remove_due_to_license_issue Q7SSI0 22238126 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF 3s5y A 2.105 BS02 DGJ A 1 W47 D92 D93 C142 K168 D170 E203 R227 D231 W16 D61 D62 C111 K137 D139 E172 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 Ki=39nM remove_due_to_license_issue IC50=70nM P06280 22195554 801 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTM 3s5y B 2.105 BS02 DGJ B 1 W47 D92 D93 C142 K168 D170 E203 R227 D231 W16 D61 D62 C111 K137 D139 E172 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 Ki=39nM remove_due_to_license_issue IC50=70nM P06280 22195554 802 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTMQ 3s68 A 1.85 BS02 TCW A 1 W38 W143 K144 N170 P174 E199 W36 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue IC50=2.2nM P22734 22349227 227 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 3s6t A 2.3 BS01 OAN A 1 R220 D367 W424 W448 Y475 D477 W490 W524 E526 R201 D348 W405 W429 Y456 D458 W471 W505 E507 D367 E368 D348 E349 3.2.1.52 0004553,0004563,0005975 Ki=0.045uM remove_due_to_license_issue Q06GJ0 21692744 1 VAAEDVVWRWSCDNGKCVKLKNDPRSSEPALSLEACKMFCNEYGLLWPRPTGEADLGNFLSKINLNSIEVKILKKGATDDLMEAAAKRFKEQVSLAIPRGSTPKLTGKAVDVYLVNENPNEKAFSLEMDESYGLRVSPSGADRVNATITANSFFGMRHGLETLSQLFVFDDIRDHLLMVRDVNISDKPVYPYRGILLDTARNYYSIESIKRTIEAMAAVKLNTFHWHITDSQSFPFVTTKRPNLYKFGALSPQKVYTKAAIREVVRFGLERGVRVLPEFDAPAHVGEGWQDTDLTVCFKAEPWKSYCGEPPCGQLNPTKDELYQYLEDIYSDMAEVFDTTDIFHMGGDEVSEACWNSSDSIQNFMMQNRWDLDKESFLKLWNYFQQKAQDKAYKAFGKKLPLILWTSTLTNYKHIDDYLNKDDYIIQVWTTGVDPQIKGLLEKGYRLIMSNYDALYFDCGYGAWVGAGNNWCSPYIGWQKVYDNSPAVIALEHRDQVLGGEAALWSEQSDTSTLDGRLWPRAAALAERLWAEPATSWQDAEYRMLHIRERLVRMGIQAESLQPEWCYQNEGYCYS 3s71 B 1.25 BS02 EVD B 1 H94 H119 V121 L198 T199 T200 H92 H117 V119 L195 T196 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue IC50=8nM P00918 22011572 1 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s71 B 1.25 BS03 EVD B 2 W5 H15 W16 D19 W3 H13 W14 D17 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue IC50=8nM P00918 22011572 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s72 B 1.6 BS02 EVE B 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s73 B 1.75 BS02 EVF B 1 H94 H119 V121 L198 T199 T200 H91 H116 V118 L194 T195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=30nM P00918 22011572 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s73 B 1.75 BS03 EVF B 2 H15 W16 D19 H12 W13 D16 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=30nM P00918 22011572 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s74 B 1.4 BS02 03T B 1 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue IC50=5.2nM P00918 22011572 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s74 B 1.4 BS03 03T B 2 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue IC50=5.2nM P00918 22011572 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s75 B 1.5 BS02 EVG B 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 1 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s75 B 1.5 BS03 EVG B 2 W5 H15 D19 W2 H12 D16 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s76 A 1.6 BS02 EVH A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 262 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s77 B 1.86 BS02 EVI B 1 H94 L198 T199 T200 H92 L195 T196 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 1 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s77 B 1.86 BS03 EVI B 2 W5 H10 N11 H15 D19 W3 H8 N9 H13 D17 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s78 B 1.98 BS02 EVJ B 1 H94 H119 V121 L198 T199 H92 H117 V119 L195 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 1 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s78 B 1.98 BS03 EVJ B 2 H4 W5 D19 H2 W3 D17 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 22011572 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s7a A 1.8 BS04 684 A 1 I7 V8 A9 L22 E30 F31 F34 S59 I60 P61 N64 I7 V8 A9 L22 E30 F31 F34 S59 I60 P61 N64 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 remove_due_to_license_issue IC50=9.9nM P00374 21931219 192 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFQRMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 3s7b A 2.42 BS06 NH5 A 1 K145 I149 N180 N182 G183 F184 T185 A203 T238 Y240 S257 Y258 K141 I145 N176 N178 G179 F180 T181 A199 T234 Y236 S253 Y254 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 Kd=0.5uM remove_due_to_license_issue IC50=120nM, Kd=500nM, Ki=300nM Q9NRG4 21782458 439 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIESH 3s7l A 2.162 BS01 591 A 1 G73 Q74 G75 D94 S97 V131 Y133 Q135 F170 I172 I180 D290 G292 G14 Q15 G16 D35 S38 V72 Y74 Q76 F111 I113 I121 D224 G226 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.08uM remove_due_to_license_issue IC50=80nM, EC50=1700nM P56817 21835615 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGY 3s7m A 2.2 BS01 532 A 1 G73 Q74 G75 L92 D94 Y133 F170 I172 W177 I180 D290 G292 G14 Q15 G16 L33 D35 Y74 F111 I113 W118 I121 D226 G228 D94 S97 N99 A101 Y133 D290 T293 D35 S38 N40 A42 Y74 D226 T229 3.4.23.46 0004190,0006508,0016020 ic50=0.06uM remove_due_to_license_issue IC50=60nM, EC50=420nM P56817 21835615 1 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDCGY 3s8x A 1.3 BS02 E59 A 1 H94 H96 H119 F131 L198 T199 T200 P202 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.07uM remove_due_to_license_issue Kd=67nM P00918 22440859 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s9e A 1.6 BS01 GLU A 1 Y63 L91 T92 R97 G142 A143 T144 E191 Y61 L89 T90 R95 G140 A141 T142 E189 ? 0015276,0016020 remove_due_to_license_issue P42264 21907808 259 GTNRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRCP 3s9i A 1.9 BS01 XI7 A 1 R339 E434 G459 L461 D462 M515 W541 D633 R329 E422 G447 L449 D450 M503 W529 D621 D271 E273 R339 E434 D462 D633 D270 E272 R329 E422 D450 D621 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 23261599 742 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAALRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNADVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 3s9t A 1.3 BS02 E49 A 1 Q92 H94 H119 V121 L198 T199 T200 Q90 H92 H117 V119 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.22uM remove_due_to_license_issue Kd=222nM P00918 22440859 266 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3s9y A 1.7 BS01 FNU A 1 D23 K102 N104 D136 K138 T194 T195 P264 Q269 G293 R294 D31 K110 N112 D144 K146 T202 T203 P272 Q277 G301 R302 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=16.6uM remove_due_to_license_issue Q8IJH3 19260677 324 SGLVPRGSMGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNMES 3s9y A 1.7 BS02 FNU B 1 D141 I142 T145 D149 I150 T153 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=16.6uM remove_due_to_license_issue Q8IJH3 19260677 324 SGLVPRGSMGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNMES 3s9y B 1.7 BS01 FNU A 1 D141 I142 T145 D142 I143 T146 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=16.6uM remove_due_to_license_issue Q8IJH3 19260677 324 SMGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNME 3s9y B 1.7 BS02 FNU B 1 D23 K102 N104 D136 K138 T194 T195 P264 Q269 G293 R294 D24 K103 N105 D137 K139 T195 T196 P265 Q270 G294 R295 4.1.1.23 0004590,0005515,0006207,0006221,0016831,0044205 Ki=16.6uM remove_due_to_license_issue Q8IJH3 19260677 324 SMGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILKQNME 3s9z A 1.793 BS02 I92 A 1 V118 R339 E434 G459 L461 D462 M515 W541 M631 D633 V117 R330 E423 G448 L450 D451 M504 W530 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R330 E423 D451 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 23261599 803 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAALRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNADVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 3sad A 1.82 BS02 040 A 1 R339 E434 G459 L461 D462 M515 W541 M631 D633 R326 E418 G443 L445 D446 M499 W525 M615 D617 D271 E273 R339 E434 D462 D633 D267 E269 R326 E418 D446 D617 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 23261599 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAALRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDVLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 3sap A 1.75 BS02 E2I A 1 H94 H96 H119 F131 V135 Q136 L198 T199 T200 P202 H91 H93 H116 F127 V131 Q132 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.014uM remove_due_to_license_issue Kd=14nM P00918 22440859 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3sax A 1.1 BS02 E50 A 1 Q92 H94 H119 V121 L198 T199 T200 P202 Q90 H92 H117 V119 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.14uM remove_due_to_license_issue Kd=270nM P00918 22440859 263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3saz A 2.04 BS01 043 A 1 R339 G459 L461 D462 M515 W541 M631 D633 R330 G446 L448 D449 M502 W528 M618 D620 D271 E273 R339 E434 D462 D633 D270 E272 R330 E421 D449 D620 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 23261599 801 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAFLRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 3sb0 A 2.199 BS02 I93 A 1 V118 R339 G459 L461 D462 M515 W541 M631 D633 V113 R324 G440 L442 D443 M496 W522 M612 D614 D271 E273 R339 E434 D462 D633 D266 E268 R324 E415 D443 D614 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 23261599 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 3sbh A 1.65 BS02 E65 A 1 H94 H96 H119 L198 T199 T200 P202 H93 H95 H118 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.22uM remove_due_to_license_issue Kd=33nM P00918 22440859 266 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3sbi A 1.4 BS02 E90 A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.017uM remove_due_to_license_issue Kd=17nM, kon=1600000M-1-s-1, koff=0.0080s-1 P00918 22440859 266 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3sc1 A 2.7 BS01 3S1 A 1 G89 E90 A109 S160 Y161 A162 E166 L212 G17 E18 A37 S88 Y89 A90 E94 L140 D205 K207 E209 N210 D223 T245 D133 K135 E137 N138 D151 T165 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 21779981 900 QPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSNSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 3sd5 A 3.2 BS01 SD5 A 1 M804 P810 I831 I879 E880 V882 T887 D964 M546 P552 I571 I619 E620 V622 T627 D702 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Kd=130nM, IC50=262nM P48736 22188813 1 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKCDRKFRVKIRGIDIPVLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGNADKLTSATNPDKENSMSISILLDNMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTANETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNRVPFVLTPDFLFVMGTSKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 3sdg A 1.87 BS01 3SE A 1 M102 G106 F110 W145 Y148 T149 N176 N179 E180 W207 M72 G76 F80 W115 Y118 T119 N146 N149 E150 W177 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=2.8uM remove_due_to_license_issue IC50=2800nM, EC50=500nM P9WMC1 22098589 217 ELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAEDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 3sdi K 2.65 BS02 3SD K 1 A20 T21 A27 K33 M45 G47 G48 A49 A20 T21 A27 K33 M45 G47 G48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20875739 302 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3sdi L 2.65 BS01 3SD K 1 D114 P115 S118 D126 P127 S130 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20875739 302 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3sdk K 2.7 BS02 P3N K 1 A20 T21 A27 V31 K33 M45 G47 A49 A20 T21 A27 V31 K33 M45 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 20875739 302 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3sdk L 2.7 BS01 P3N K 1 D114 P115 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 20875739 302 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3sfc A 2.1 BS01 S53 A 1 Q13 V30 D32 Y75 S76 T77 P111 F117 V120 D215 G217 A218 M289 Q19 V36 D38 Y83 S84 T85 P118 F124 V127 D226 G228 A229 M303 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y83 D226 A229 3.4.23.15 0004190,0006508 ic50=0.003uM remove_due_to_license_issue IC50=192nM P00797 21840218 330 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3sfc A 2.1 BS02 S53 A 2 L110 L114 R240 L242 F243 L117 L121 R251 L252 F253 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y83 D226 A229 3.4.23.15 0004190,0006508 ic50=0.003uM remove_due_to_license_issue IC50=192nM P00797 21840218 331 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3sff A 2.0 BS01 0DI A 1 I34 G140 W141 H142 H143 G151 F152 C153 D178 H180 F208 G303 G304 Y306 I21 G104 W105 H106 H107 G115 F116 C117 D142 H144 F172 G267 G268 Y270 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=200nM remove_due_to_license_issue IC50=200nM Q9BY41 21723733 378 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 3sfg A 2.209 BS01 2TU A 1 D250 S303 N312 Y344 D346 D246 S299 N308 Y340 D342 2.7.7.48,3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 Kd=0.865uM remove_due_to_license_issue Q80J95 22341781 601 LPRPSGTYAGLPIADYGDAPPLSTKTMFWRTSPEKLPPGAWEPAYLGSKDERVDGPSLQQVMRDQLKPYSEPRGLLPPQEILDAVCDAIENRLENTLEPQKPWTFKKACESLDKNTSSGYPYHKQKSKDWTGSAFIGDLGDQATHANNMYEMGKSMRPIYTAALKDELVKPDKIYGKIKKRLLWGSDLGTMIRAARAFGPFCDALKETCIFNPIRVGMSMNEDGPFIFARHANFRYHMDADYTRWDSTQQRAILKRAGDIMVRLSPEPDLARVVMDDLLAPSLLDVGDYKIVVEEGLPSGCPCTTQLNSLAHWILTLCAMVEVTRVDPDIVMQESEFSFYGDDEVVSTNLELDMVKYTMALRRYGLLPTRADKEEGPLERRQTLQGISFLRRAIVGDQFGWYGRLDRASIDRQLLWTKGPNHQNPFETLPGHAQRPSQLMALLGEAAMHGEKYYRTVASRVSKMVVPRHRSVLRWVRFGT 3sfh A 2.7 BS05 1DI A 1 I34 R37 G140 W141 H142 H143 G151 F152 H180 F208 G303 G304 I21 R24 G105 W106 H107 H108 G116 F117 H145 F173 G268 G269 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue IC50=90nM Q9BY41 21723733 501 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 3sfi A 2.31 BS01 3SF A 1 M102 G106 F110 F114 W138 W145 Y148 T149 N176 N179 E180 W207 M81 G85 F89 F93 W117 W124 Y127 T128 N155 N158 E159 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.4uM remove_due_to_license_issue IC50=400nM, EC50=60nM P9WMC1 22098589 217 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 3sgt B 1.85 BS01 P09 B 1 A69 L85 M86 F89 A92 L93 F116 I141 A142 A143 N144 A57 L70 M71 F74 A77 L78 F101 I126 A127 A128 N129 D26 H43 L137 D14 H31 L122 2.5.1.31 0000287,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0045547,0046872,0071555 remove_due_to_license_issue P60473 23248302 1001 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 3sgv B 1.61 BS01 2BJ B 1 K44 A47 K48 V50 R51 L88 A92 E96 K32 A35 K36 V38 R39 L65 A69 E73 D26 H43 L137 D14 H31 L114 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 5001 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 3sgv B 1.61 BS02 2BJ B 2 M25 D26 G27 N28 G29 H43 A69 L85 F89 M13 D14 G15 N16 G17 H31 A57 L62 F66 D26 H43 L137 D14 H31 L114 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 1001 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 3sgx A 2.45 BS01 0FW A 1 A47 V50 R51 V54 S55 A58 N59 W91 A92 E96 S99 L100 H103 A31 V34 R35 V38 S39 A42 N43 W64 A65 E69 S72 L73 H76 D26 H43 L137 D10 H27 L110 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 1001 GCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSELMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFAN 3sgx A 2.45 BS02 0FW A 2 N28 R39 H43 F70 S71 M86 F89 A92 I141 N12 R23 H27 F54 S55 M59 F62 A65 I114 D26 H43 L137 D10 H27 L110 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 2001 GCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSELMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFAN 3sh0 B 1.84 BS01 SAX B 1 A47 L85 M86 L88 E96 F116 A142 A143 N144 A35 L67 M68 L70 E78 F98 A124 A125 N126 D26 H43 L137 D14 H31 L119 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 1001 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 3sh0 B 1.84 BS02 SAX B 2 S55 A58 N59 E96 S99 L100 H103 S43 A46 N47 E78 S81 L82 H85 D26 H43 L137 D14 H31 L119 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 1002 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 3sh1 A 2.9 BS02 MLK A 1 Y93 K143 W147 Y149 R186 Y195 D197 Y99 K149 W153 Y155 R192 Y201 D203 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 301 DDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRSERFYECCKEPYPDVNLVVKFRERR 3sh1 A 2.9 BS03 MLK B 1 W55 S167 W61 S173 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 301 DDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRSERFYECCKEPYPDVNLVVKFRERR 3sh1 E 2.9 BS01 MLK A 1 W55 L118 S167 W62 L125 S174 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 301 KDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRSERFYECCKEPYPDVNLVVKFRERR 3sh1 E 2.9 BS03 MLK E 1 Y93 K143 W147 Y149 R186 Y188 Y195 D197 Y100 K150 W154 Y156 R193 Y195 Y202 D204 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 301 KDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRSERFYECCKEPYPDVNLVVKFRERR 3sha H 1.52 BS03 P97 H 1 H57 Y60A W60D L99 I174 S195 S214 W215 G216 H43 Y47 W50 L96 I172 S198 S219 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=2.6uM remove_due_to_license_issue P00734 22366545 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3shc H 1.9 BS03 B01 H 1 H57 N98 A190 S195 V213 S214 W215 G216 F227 H43 N95 A193 S198 V218 S219 W220 G221 F232 3.4.21.5 0004252,0005509,0006508,0007596 Ki=1.9uM remove_due_to_license_issue P00734 22366545 3 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3shj K 2.8 BS01 H10 K 1 T1 A20 T21 V31 M45 A49 T1 A20 T21 V31 M45 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 22105886 2I TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 3shj L 2.8 BS01 H10 K 1 S112 F113 S118 E122 R125 S124 F125 S130 E134 R137 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 22105886 2I QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 3shy A 2.647 BS01 5FO A 1 V782 F786 M816 Q817 F820 V239 F243 M254 Q255 F258 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue Kd=1700nM O76074 21714539 1 ETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 3shz A 2.449 BS01 5CO A 1 A783 F786 M816 Q817 F820 A240 F243 M253 Q254 F257 3.1.4.35 0004114,0007165,0008081 ic50=35.9nM remove_due_to_license_issue Kd=770nM O76074 21714539 1 ETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 3si3 H 1.55 BS03 B03 H 1 Y60A W60D N98 L99 I174 V213 S214 W215 G216 Y47 W50 N95 L96 I172 V218 S219 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=69.3uM remove_due_to_license_issue P00734 22366545 5 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3si4 H 1.27 BS03 B04 H 1 Y60A W60D N98 V213 S214 W215 G216 Y47 W50 N95 V218 S219 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=132.2uM remove_due_to_license_issue P00734 22366545 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3sie A 1.93 BS01 5BO A 1 Y612 V782 F786 L804 M816 Q817 G819 F820 Y75 V223 F227 L241 M253 Q254 G256 F257 3.1.4.35 0004114,0007165,0008081 ic50=13.3nM remove_due_to_license_issue Kd=420nM O76074 21714539 1 RELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 3sio A 2.32 BS01 MLK A 1 Y93 K143 W147 Y149 Y188 C190 Y195 D197 Y100 K150 W154 Y156 Y195 C197 Y202 D204 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 260 KDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3sio A 2.32 BS02 MLK B 1 W55 Q116 S167 W62 Q123 S174 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 260 KDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3sio E 2.32 BS01 MLK A 1 W55 S167 W64 S176 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 260 DYKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3sio E 2.32 BS02 MLK E 1 Y93 K143 W147 Q186 Y188 Y195 Y102 K152 W156 Q195 Y197 Y204 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 22009746 260 DYKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVYLSFSLLDIVKADSSTNEVDLVYWEQQSWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQNALVNSSGHVQYLPAQRLSFMCDPTGVDSEEGATCAVKFGSWSYGGWEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 3siu A 2.626 BS01 rna C 0 R36 K37 G38 A39 N40 E41 K44 E61 I65 V95 R97 V99 I100 R33 K34 G35 A36 N37 E38 K41 E58 I62 V92 R94 V96 I97 ? 0000398,0001651,0003723,0005515,0005634,0005654,0005681,0005690,0005730,0006397,0008380,0030490,0030515,0030621,0030622,0031428,0032040,0032991,0034511,0034512,0042254,0042274,0046540,0051117,0071005,0071011,1990904 remove_due_to_license_issue P55769 21784869 28 ~ 55 ADVNPKAYPLADAHLTKKLLDLVQQSCNYKQLRKGANEATKTLNRGISEFIVMAADAEPLEIILHLPLLCEDKNVPYVFVRSKQALGRACGVSRPVIACSVTIKEGSQLKQQIQSIQQSIERLLV 3siu B 2.626 BS01 rna C 0 C247 N248 M250 L251 H270 R289 R293 A297 K298 C162 N163 M165 L166 H173 R192 R196 A200 K201 ? 0000244,0000398,0046540 remove_due_to_license_issue Q8WWY3 21784869 28 ~ 55 AAPEYRVIVDANNLTVEIENELNIIHKFIRDKYSKRFPELESLVPNALDYIRTVKELGNSLDKCKNNENLQQILTNATIMVVSVTASTTQGQQLSEEELERLEEACDMALELNASKHRIYEYVESRMSFIAPNLSIIIGASTAAKIMGVAGGLTNLSKMPACNIMLLGAQLPHTGYIYHSDIVQSLPPDLRRKAARLVAAKCTLAARVDSFHESTEGKVGYELKDEIERKFDKWQ 3siu D 2.626 BS01 rna F 0 K37 G38 A39 N40 E41 K44 R48 A60 E61 I65 V95 R97 V99 I100 K34 G35 A36 N37 E38 K41 R45 A57 E58 I62 V92 R94 V96 I97 ? 0000398,0001651,0003723,0005515,0005634,0005654,0005681,0005690,0005730,0006397,0008380,0030490,0030515,0030621,0030622,0031428,0032040,0032991,0034511,0034512,0042254,0042274,0046540,0051117,0071005,0071011,1990904 remove_due_to_license_issue P55769 21784869 28 ~ 55 ADVNPKAYPLADAHLTKKLLDLVQQSCNYKQLRKGANEATKTLNRGISEFIVMAADAEPLEIILHLPLLCEDKNVPYVFVRSKQALGRACGVSRPVIACSVTIKEGSQLKQQIQSIQQSIERLLV 3siu E 2.626 BS01 rna F 0 C247 N248 M250 L251 L252 H270 R289 R293 A297 K298 K327 C162 N163 M165 L166 L167 H174 R193 R197 A201 K202 K231 ? 0000244,0000398,0046540 remove_due_to_license_issue Q8WWY3 21784869 28 ~ 55 AAPEYRVIVDANNLTVEIENELNIIHKFIRDKYSKRFPELESLVPNALDYIRTVKELGNSLDKCKNNENLQQILTNATIMVVSVTASTTQGQQLSEEELERLEEACDMALELNASKHRIYEYVESRMSFIAPNLSIIIGASTAAKIMGVAGGLTNLSKMPACNIMLLGASVLPHTGYIYHSDIVQSLPPDLRRKAARLVAAKCTLAARVDSFHESTEGKVGYELKDEIERKFDKWQ 3sjf A 1.65 BS04 JRG A 1 R210 N257 E424 L428 R463 D465 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 L374 R409 D411 G464 N465 R480 R482 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=23nM remove_due_to_license_issue Ki=23nM Q04609 21923190 1 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 3sji A 1.798 BS01 AG7 A 1 H40 E71 L125 L127 S128 K130 T142 K143 A144 C147 H161 I162 G163 G164 N165 H37 E68 L122 L124 S125 K127 T139 K140 A141 C144 H158 I159 G160 G161 N162 H40 E71 G145 C147 H37 E68 G142 C144 3.4.22.28 0004197,0006508 remove_due_to_license_issue C8CIL7 21795339 501 LDFALSLLRRNIRQVQTDQGHFTMLGVRDRLAILPRHSQPGKTIWVEHKLINVLDAVELVDEQGVNLELTLVTLDTNEKFRDVTKFIPETITGASDATLIINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKIIGIHIGGNGRQGFCAGLKRGYFASE 3sjo A 1.702 BS01 AG7 A 1 R39 H40 E71 L127 S128 K130 T142 A144 C147 H161 G163 G164 N165 F170 R36 H37 E68 L124 S125 K127 T139 A141 C144 H158 G160 G161 N162 F167 H40 E71 G145 C147 H37 E68 G142 C144 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue E0WWC7 21795339 501 LDFALSLLRRNIRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNVLDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFASE 3sjt A 1.597 BS03 5AB A 1 D124 H126 D128 S137 H141 D183 D232 D119 H121 D123 S132 H136 D178 D227 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue P05089 21728378 551 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 3sk2 A 1.01 BS01 GRI A 1 V108 F109 V111 F112 ? 0042803,0043177,0046677 Kd=244uM remove_due_to_license_issue Q8GPH6 21849072 130 GSHMTDLAGPTITPNLQLVYVSNVERSTDFYRFIFKKEPVFVTPRYVAFPSSGDALFAIWSGGEEPVAEIPRFSEIGIMLPTGEDVDKLFNEWTKQKSHQIIVIKEPYTDVFGRTFLISDPDGHIIRVCPLD 3sk2 B 1.01 BS01 GRI A 1 R42 Y43 W57 R45 Y46 W60 ? 0042803,0043177,0046677 remove_due_to_license_issue Q8GPH6 21849072 130 GSHMTDLAGPTITPNLQLVYVSNVERSTDFYRFIFKKEPVFVTPRYVAFPSSGDALFAIWSGGEEPVAEIPRFSEIGIMLPTGEDVDKLFNEWTKQKSHQIIVIKEPYTDVFGRTFLISDPDGHIIRVCPLD 3ska A 1.73 BS01 053 A 1 P197 N316 C366 S368 L384 G410 M414 Y415 Q446 I447 Y448 P192 N311 C361 S363 L379 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.017uM remove_due_to_license_issue O92972 21840715 578 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3skc A 3.2 BS01 BR2 A 1 A481 K483 L505 L514 I527 T529 W531 C532 D594 A34 K36 L58 L67 I80 T82 W84 C85 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S153 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 21802293 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3ske A 1.97 BS01 054 A 1 N316 C366 S368 L384 G410 N411 M414 Y415 Q446 I447 Y448 N311 C361 S363 L379 G405 N406 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.032uM remove_due_to_license_issue O92972 21840715 578 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3skf A 3.0 BS01 PB7 A 1 G11 Q12 D32 G34 S35 P70 Y71 T72 Q73 F108 D228 G230 T231 T232 G13 Q14 D34 G36 S37 P72 Y73 T74 Q75 F110 D230 G232 T233 T234 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 21974952 394 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3skg A 2.88 BS01 PB8 A 1 G11 Q12 L30 D32 G34 Y71 T72 Q73 F108 I110 W115 Y198 D228 G230 T231 T232 R235 G13 Q14 L32 D34 G36 Y73 T74 Q75 F110 I112 W117 Y200 D230 G232 T233 T234 R237 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=9.5nM P56817 21974952 394 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 3skh A 2.5 BS01 058 A 1 C366 L384 G410 M414 Y415 Y448 C361 L379 G405 M409 Y410 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.9uM remove_due_to_license_issue O92972 21840715 577 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3skk A 1.701 BS03 4U7 A 1 D124 H126 D128 S137 H141 D183 D232 D119 H121 D123 S132 H136 D178 D227 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue P05089 21728378 551 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 3sl0 A 1.997 BS03 FB5 A 1 D216 H218 D220 N222 S229 H233 G234 D274 D323 D325 D113 H115 D117 N119 S126 H130 G131 D171 D220 D222 H193 D216 H218 D220 H233 D323 D325 E368 H90 D113 H115 D117 H130 D220 D222 E265 3.5.3.1 0000050,0004053,0005737,0005829,0006525,0016787,0019547,0030145,0042802,0046872 remove_due_to_license_issue Q8I384 21728378 414 KNVSIIGSPLAAGQPLGGVQLACDDLRKLGLHNVIDVLGWKYEDIGNIDNCYYDNIRNIKEIGIFSKNLFDTMSNELRKKNFVLNIGGDHGVAFSSILSSLQMYQNLRVIWIDAHGDINIPETSPSGNYHGMTLAHTLGLFKKKVPYFEWSENLTYLKPENTAIIGIRDIDAYEKIILKKCNINYYTIFDIEKNGIYNTICTALEKIDPNSNCPIHISLDIDSVDNVFAPGTGTVAKGGLNYREINLLMKILAETKRVVSMDLVEYNPSLDEVDKKVHGDSLPILDNATKTGKLCLELIARVLGYDIV 3sl1 A 1.902 BS03 FB6 A 1 D216 H218 D220 S229 H233 G234 D274 D323 D325 D113 H115 D117 S126 H130 G131 D171 D220 D222 H193 D216 H218 D220 H233 D323 D325 E368 H90 D113 H115 D117 H130 D220 D222 E265 3.5.3.1 0000050,0004053,0005737,0005829,0006525,0016787,0019547,0030145,0042802,0046872 remove_due_to_license_issue Q8I384 21728378 414 KNVSIIGSPLAAGQPLGGVQLACDDLRKLGLHNVIDVLGWKYEDIGNIDNCYYDNIRNIKEIGIFSKNLFDTMSNELRKKNFVLNIGGDHGVAFSSILSSLQMYQNLRVIWIDAHGDINIPETSPSGNYHGMTLAHTLGLFKKKVPYFEWSENLTYLKPENTAIIGIRDIDAYEKIILKKCNINYYTIFDIEKNGIYNTICTALEKIDPNSNCPIHISLDIDSVDNVFAPGTGTVAKGGLNYREINLLMKILAETKRVVSMDLVEYNPSLDEVDKKVHGDSLPILDNATKTGKLCLELIARVLGYDIV 3sl4 A 1.9 BS02 JN4 A 1 Y159 L319 N321 P322 Y329 I336 M357 Q369 F372 Y77 L237 N239 P240 Y247 I254 M275 Q287 F290 3.1.4.53 0004114,0007165,0008081 ic50=0.027uM remove_due_to_license_issue Q08499 22030030 23 GVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 3sl5 A 2.65 BS02 J25 A 1 Y159 N321 P322 Y329 M357 Q369 F372 Y77 N239 P240 Y247 M275 Q287 F290 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=22nM Q08499 22030030 1 GVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTI 3sl8 A 2.6 BS02 JN7 A 1 Y159 N321 T333 I336 F340 S368 Q369 F372 I376 Y76 N238 T250 I253 F257 S285 Q286 F289 I293 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 22030030 18 VKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTI 3slz A 1.4 BS01 3TL A 1 D32 G34 Q36 A52 V54 Q55 G56 A57 W65 P89 Y90 D22 G24 Q26 A42 V44 Q45 G46 A47 W55 P79 Y80 ? 0004190,0006508 Ki=102nM remove_due_to_license_issue Q9E7M1 21951660 126 EPPPEPRITLKVGGQPVTFLVDTGAQHSVLTQNPGPLSDKSAWVQGATGGKRYRWTTDRKVHLATGKVTHSFLHVPDCPYPLLGRDLLTKLKAQIHFEGSGAQVVGPMGQPLQV 3slz B 1.4 BS01 3TL A 1 D32 G34 Q36 H37 V54 Q55 G56 A57 W65 P89 Y90 L92 D22 G24 Q26 H27 V44 Q45 G46 A47 W55 P79 Y80 L82 ? 0004190,0006508 remove_due_to_license_issue Q9E7M1 21951660 126 EPPPEPRITLKVGGQPVTFLVDTGAQHSVLTQNPGPLSDKSAWVQGATGGKRYRWTTDRKVHLATGKVTHSFLHVPDCPYPLLGRDLLTKLKAQIHFEGSGAQVVGPMGQPLQV 3sm0 A 1.57 BS02 AEK A 1 V45 N70 D102 Y106 Q107 D156 C158 G229 A232 M260 G261 D280 V35 N60 D92 Y96 Q97 D138 C140 G211 A214 M242 G243 D262 D102 D280 C318 C320 C323 H349 D92 D262 C300 C302 C305 H331 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=740nM remove_due_to_license_issue P28720 22736391 501 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 3sm2 A 1.75 BS01 478 A 1 D32 G34 H37 V54 G56 A57 D22 G24 H27 V44 G46 A47 ? 0004190,0006508 Ki=0.2nM remove_due_to_license_issue Q9E7M1 21951660 126 EPPPEPRITLKVGGQPVTFLVDTGAQHSVLTQNPGPLSDKSAWVQGATGGKRYRWTTDRKVHLATGKVTHSFLHVPDCPYPLLGRDLLTKLKAQIHFEGSGAQVVGPMGQPLQV 3sm2 B 1.75 BS01 478 A 1 D32 G34 A35 H37 V54 A57 P89 Y90 D22 G24 A25 H27 V44 A47 P79 Y80 ? 0004190,0006508 remove_due_to_license_issue Q9E7M1 21951660 126 EPPPEPRITLKVGGQPVTFLVDTGAQHSVLTQNPGPLSDKSAWVQGATGGKRYRWTTDRKVHLATGKVTHSFLHVPDCPYPLLGRDLLTKLKAQIHFEGSGAQVVGPMGQPLQV 3smq A 2.0 BS01 TDU A 1 K392 H393 R396 V420 E422 L424 T466 A467 K150 H151 R154 V178 E180 L182 T224 A225 D253 E346 E355 H496 D11 E104 E113 H254 2.1.1.319 0016274,0018216 remove_due_to_license_issue IC50=2500nM O60678 22795084 1 HYGIHEEMLKDKIRTESYRDFIYQNPHIFKDKVVLDVGCGTGILSMFAAKAGAKKVLGVDQSEILYQAMDIIRLNKLEDTITLIKGKIEEVHLPVEKVDVIISEWMGYFLLFESMLDSVLYAKNKYLAKGGSVYPDICTISLVAVSDVNKHADRIAFWDDVYGFKMSCMKKAVIPEAVVEVLDPKTLISEPCGIKHIDCHTTSISDLEFSSDFTLKITRTSMCTAIAGYFDIYFEKNCHNRVVFSTGPQSTKTHWKQTVFLLEKPFSVKAGEALKGKVTVHKSLTVTLTLNNSTQTYGL 3sn7 A 1.82 BS01 540 A 1 L665 I682 Y683 F686 M703 Q716 F719 L228 I245 Y246 F249 M266 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=0.7nM remove_due_to_license_issue IC50=0.700000nM Q9Y233 21988093 780 MSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3sn8 A 1.99 BS01 S89 A 1 M49 F140 L141 N142 G143 C145 M165 E166 R188 M49 F140 L141 N142 G143 C145 M165 E166 R188 H41 G143 C145 H41 G143 C145 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0008233,0019082 remove_due_to_license_issue P0C6U8 21854807 307 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 3sni A 1.9 BS02 546 A 1 Y514 H515 I682 F686 M703 Q716 F719 Y77 H78 I245 F249 M266 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=11nM remove_due_to_license_issue IC50=11nM Q9Y233 21988093 782 MSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3snl B 2.4 BS02 548 B 1 Y514 I682 Y683 F686 M703 Q716 Y78 I233 Y234 F237 M254 Q267 3.1.4.17 0004114,0007165,0008081 ic50=0.7nM remove_due_to_license_issue IC50=0.700000nM Q9Y233 21988093 1 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3so9 A 2.87 BS01 017 A 1 G27 A28 D29 D30 G48 I50 G27 A28 D29 D30 G48 I50 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q000H7 21871444 100 PQITLWKRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3so9 B 2.87 BS01 017 A 1 N25 A28 D30 I47 I50 T82 N25 A28 D30 I47 I50 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q000H7 21871444 100 PQITLWKRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3spf A 1.7 BS01 B50 A 1 F97 Y101 F105 L108 E129 F42 Y46 F50 L53 E74 ? 0042981 Ki=138uM remove_due_to_license_issue Ki=138000nM, IC50=453000nM Q07817 22448988 501 FMSQSNRELVVDFLSYKLSQKGYSWSESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGN 3spk A 1.24 BS01 TPV A 1 R8 N25 D29 D30 I47 G48 G49 I50 P81 T82 R8 N25 D29 D30 I47 G48 G49 I50 P81 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=3.02nM remove_due_to_license_issue Q000H7 21871444 100 PQITLWKRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3spk A 1.24 BS02 TPV B 1 R8 L23 N25 A28 I50 T82 R8 L23 N25 A28 I50 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=3.02nM remove_due_to_license_issue Q000H7 21871444 100 PQITLWKRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3spk B 1.24 BS01 TPV A 1 R8 L23 N25 I50 T82 R8 L23 N25 I50 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=3.02nM remove_due_to_license_issue Q000H7 21871444 100 PQITLWKRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3spk B 1.24 BS02 TPV B 1 R8 N25 D29 D30 I47 G48 G49 I50 P81 T82 R8 N25 D29 D30 I47 G48 G49 I50 P81 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=3.02nM remove_due_to_license_issue Q000H7 21871444 100 PQITLWKRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 3sq2 A 2.1 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 V396 N564 S565 Y567 G568 G571 N572 W574 K705 K706 R707 K800 K844 K874 K878 S360 P361 I362 Y391 P392 G393 A394 V396 N564 S565 Y567 G568 G571 N572 W574 K705 K706 R707 K800 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 3sq2 A 2.1 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 K800 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 3sq4 A 2.23 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 N564 S565 Y567 G568 G571 N572 W574 K705 K706 R707 K800 K844 K874 S360 P361 I362 Y391 P392 G393 N564 S565 Y567 G568 G571 N572 W574 K705 K706 R707 K800 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 3sq4 A 2.23 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 H804 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 3sqq A 1.85 BS01 99Z A 1 I10 V18 A31 F80 L83 H84 Q85 D86 K89 L134 D145 I10 V18 A31 F76 L79 H80 Q81 D82 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T148 T155 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 23600925 456 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3sr4 A 2.5 BS01 TT8 A 1 G137 E138 T139 D161 G163 S164 Q168 V169 E186 K187 G221 D222 F223 F245 G133 E134 T135 D157 G159 S160 Q164 V165 E182 K183 G217 D218 F219 F241 2.1.1.360 0031151,0051726 Ki=0.29uM remove_due_to_license_issue Ki=290nM Q8TEK3 21936531 417 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLKNP 3srb A 1.8 BS01 28S B 1 L169 L170 L141 L142 3.5.1.97 0016787,0016811,0017000 remove_due_to_license_issue Q9I194 21892836 1 TGLAADIRWTAYGVPHIRAKDERGLGYGIGYAYARDNACLLAEEIVTARGERARYFGSEGKSSAELDNLPSDIFYAWLNQPEALQAFWQAQTPAVRQLLEGYAAGFNRFLREADGKTTSCLGQPWLRAIATDDLLRLTRRLLVEGGVGQFADALVAAAPPGAE 3srb B 1.8 BS01 28S B 1 L269 N273 V374 L375 W378 W402 L53 N57 V158 L159 W162 W186 S217 H239 V286 N485 T695 S1 H23 V70 N269 T479 3.5.1.97 0016787,0017000 ic50=65uM remove_due_to_license_issue Q9I194 21892836 1 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIRE 3src B 2.0 BS01 28N B 1 L266 L269 N273 V374 W378 W402 L50 L53 N57 V158 W162 W186 S217 H239 V286 N485 T695 S1 H23 V70 N269 T479 3.5.1.97 0016787,0017000 ic50=130uM remove_due_to_license_issue Q9I194 21892836 1 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIRE 3srg A 2.19 BS03 OCH A 1 E53 Y71 I74 H115 N168 N224 D269 H285 F292 E35 Y53 I56 H97 N150 N206 D251 H267 F274 0004064,0005576 remove_due_to_license_issue 22387469 1358 RQKSSFQTRFNVHREVTPVELPNCNLVKGIDNGSEDLEILPNGLAFISSGLKYPGIMSFDPDKSGKILLMDLNEKEPAVSELEIIGNTLDISSFNPHGISTFIDDDNTVYLLVVNHPGSSSTVEVFKFQEEEKSLLHLKTIRHKLLPSVNDIVAVGPEHFYATNDHYFIDPYLKSWEMHLGLAWSFVTYYSPNDVRVVAEGFDFANGINISPDGKYVYIAELLAHKIHVYEKHANWTLTPLRVLSFDTLVDNISVDPVTGDLWVGCHPNGMRIFFYDAENPPGSEVLRIQDILSEEPKVTVVYAENGTVLQGSTVAAVYKGKLLIGTVFHKALYCDL 3srv A 1.95 BS01 S19 A 1 L377 A400 M448 G454 P455 R498 L501 D512 L14 A35 M77 G83 P84 R127 L130 D141 D494 A496 R498 N499 D512 K533 D123 A125 R127 N128 D141 K162 2.7.10.2 0004672,0004713,0005524,0006468 ic50=31.6nM remove_due_to_license_issue IC50=32nM P43405 21903390 1 YLDRKLLTLEDKELGNFGTVKKGYYQMKKVVKTVAVKILKALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV 3st5 A 1.45 BS01 G89 B 1 D25 A28 D30 P81 D25 A28 D30 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 21800876 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3st5 B 1.45 BS01 G89 B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=5pM remove_due_to_license_issue P03367 21800876 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3st6 A 1.75 BS01 RVE A 1 H334 T361 Y385 L404 R405 A418 G419 G421 K438 H320 T347 Y371 L390 R391 A404 G405 G407 K424 K205 E252 A269 E297 H334 T361 Y385 R405 G421 E434 K438 K191 E238 A255 E283 H320 T347 Y371 R391 G407 E420 K424 4.2.99.21,5.4.4.2,5.4.99.5 0000162,0000287,0004106,0005886,0008909,0009058,0009697,0010106,0016829,0016833,0016853,0019540,0043904,0046872,0052572 Ki=240uM remove_due_to_license_issue P9WFX1 22607697 451 SSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTRALGRGPAIDRLARDDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRERGSVQHLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVARQ 3std A 1.65 BS01 MQ0 A 1 Y30 Y50 F53 V108 A127 N131 L147 P149 I151 G165 Y22 Y42 F45 V100 A119 N123 L139 P141 I143 G157 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=7.7pM remove_due_to_license_issue P56221 9922139 503 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFG 3std B 1.65 BS02 MQ0 B 1 Y30 Y50 F53 V75 V108 L147 P149 I151 F162 G165 Y22 Y42 F45 V67 V100 L139 P141 I143 F154 G157 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=7.7pM remove_due_to_license_issue P56221 9922139 505 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFG 3str P 1.75 BS01 3LI P 1 Q57 G70 V71 G72 Q77 E126 G127 E128 G129 C130 L131 Y166 H173 E174 H177 Q56 G69 V70 G71 Q76 E116 G117 E118 G119 C120 L121 Y156 H163 E164 H167 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=334nM remove_due_to_license_issue Q939R9 21711014 209 SAIERITKAAHLIDMNDIIREGNPTLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNIAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLILE 3su0 A 1.159 BS01 TSV A 1 Q1041 F1043 H1057 D1081 L1135 K1136 G1137 A1139 F1154 K1155 A1156 A1157 Q59 F61 H75 D99 L153 K154 G155 A157 F172 K173 A174 A175 H1057 D1081 G1137 A1139 H75 D99 G155 A157 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=162nM remove_due_to_license_issue A8DG50 22910833 100 MASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFKAAVSTRGVAKAVDFIPVESLETTMR 3su1 A 1.399 BS01 TSV A 1 Q1041 F1043 H1057 D1081 L1135 K1136 G1137 A1139 F1154 R1155 A1156 A1157 Q61 F63 H77 D101 L155 K156 G157 A159 F174 R175 A176 A177 H1057 D1081 G1137 A1139 H77 D101 G157 A159 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=208nM remove_due_to_license_issue A8DG50 22910833 100 SHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRAAVSTRGVAKAVAFIPVESLETTMR 3su2 A 1.496 BS01 TSV A 1 Q1041 F1043 H1057 V1078 D1081 L1135 K1136 G1137 A1139 F1154 R1155 T1156 A1157 Q60 F62 H76 V97 D100 L154 K155 G156 A158 F173 R174 T175 A176 H1057 D1081 G1137 A1139 H76 D100 G156 A158 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=44.8nM remove_due_to_license_issue A8DG50 22910833 100 HMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTM 3su3 A 1.3 BS01 SU3 A 1 Q1041 F1043 H1057 D1081 L1135 K1136 G1137 A1139 F1154 R1155 A1156 A1157 Q62 F64 H78 D102 L156 K157 G158 A160 F175 R176 A177 A178 H1057 D1081 G1137 A1139 H78 D102 G158 A160 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=0.74nM remove_due_to_license_issue A8DG50 22910833 1 GSHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRAAVSTRGVAKAVDFIPVESLETTMR 3su4 A 2.255 BS01 SU3 A 1 Q1041 F1043 H1057 V1078 D1081 R1123 I1132 L1135 K1136 G1137 A1139 F1154 K1155 A1156 A1157 Q52 F54 H68 V89 D92 R134 I143 L146 K147 G148 A150 F165 K166 A167 A168 H1057 D1081 G1137 A1139 H68 D92 G148 A150 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=554nM remove_due_to_license_issue P26664 22910833 1 GSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFKAAVSTRGVAKAVDFIPVESLETTMRS 3su5 A 1.55 BS01 SU3 A 1 Q1041 F1043 H1057 D1081 L1135 K1136 G1137 A1139 F1154 R1155 A1156 A1157 Q61 F63 H77 D101 L155 K156 G157 A159 F174 R175 A176 A177 H1057 D1081 G1137 A1139 H77 D101 G157 A159 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=2635nM remove_due_to_license_issue A8DG50 22910833 1 SHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRAAVSTRGVAKAVAFIPVESLETTMRS 3su6 A 1.1 BS01 SU3 A 1 F1043 H1057 D1081 L1135 K1136 G1137 A1139 F1154 R1155 T1156 A1157 F63 H77 D101 L155 K156 G157 A159 F174 R175 T176 A177 H1057 D1081 G1137 A1139 H77 D101 G157 A159 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=958nM remove_due_to_license_issue A8DG50 22910833 1 SHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTM 3sud A 1.96 BS01 SUE A 1 Q1041 F1043 Y1056 H1057 V1078 D1081 L1135 K1136 G1137 A1139 F1154 R1155 A1156 A1157 Q53 F55 Y68 H69 V90 D93 L147 K148 G149 A151 F166 R167 A168 A169 H1057 D1081 G1137 A1139 H69 D93 G149 A151 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=0.14nM remove_due_to_license_issue A8DG50 22910833 1201 KGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRAAVSTRGVAKAVDFIPVESLETTM 3sue A 2.2 BS01 SUE A 1 Q1041 F1043 Y1056 H1057 V1078 D1081 I1132 L1135 K1136 G1137 S1139 F1154 K1155 A1156 A1157 Q52 F54 Y67 H68 V89 D92 I143 L146 K147 G148 S150 F165 K166 A167 A168 H1057 D1081 G1137 S1139 H68 D92 G148 S150 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=0.84nM remove_due_to_license_issue A8DG50 22910833 1201 GSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFKAAVSTRGVAKAVDFIPVESLETTM 3suf A 2.19 BS01 SUE A 1 Q1041 H1057 V1078 D1081 L1135 K1136 G1137 S1139 F1154 R1155 A1156 A1157 Q52 H68 V89 D92 L146 K147 G148 S150 F165 R166 A167 A168 H1057 D1081 G1137 S1139 H68 D92 G148 S150 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=27.8nM remove_due_to_license_issue A8DG50 22910833 1201 GSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVAFIPVESLETTM 3sug A 1.8 BS01 SUE A 1 Q1041 F1043 Y1056 H1057 G1058 V1078 L1135 K1136 G1137 A1139 F1154 R1155 T1156 A1157 Q61 F63 Y76 H77 G78 V98 L155 K156 G157 A159 F174 R175 T176 A177 H1057 D1081 G1137 A1139 H77 D101 G157 A159 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=620nM remove_due_to_license_issue A8DG50 22910833 1201 SHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTMRS 3sun A 2.42 BS01 dna T 0 S360 I362 Y391 P392 G393 A394 N564 S565 G568 N572 W574 K705 R707 K800 K844 K874 K878 S360 I362 Y391 P392 G393 A394 N564 S565 G568 N572 W574 K705 R707 K800 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKA 3sun A 2.42 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 K790 Y791 K800 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 K790 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKA 3suo A 2.23 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 V396 N564 S565 G568 N572 W574 K705 K706 R707 K800 K844 K874 K878 S360 P361 I362 Y391 P392 G393 A394 V396 N564 S565 G568 N572 W574 K705 K706 R707 K800 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDM 3suo A 2.23 BS02 dna P 0 N284 K706 Y708 M728 G729 S735 S784 N786 H804 N284 K706 Y708 M728 G729 S735 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDM 3sup A 2.32 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 W574 K705 K706 R707 P799 K800 K844 K874 K878 S360 P361 I362 Y391 P392 G393 A394 N564 S565 G568 N572 W574 K705 K706 R707 P799 K800 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3sup A 2.32 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 3suq A 3.15 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 V396 S565 G568 N572 W574 K705 R707 K800 K874 S360 P361 I362 Y391 P392 G393 A394 V396 S565 G568 N572 W574 K705 R707 K800 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASL 3suq A 3.15 BS02 dna P 0 N284 D621 T622 K706 Y708 M728 G729 Q733 K734 S735 S783 S784 N786 Y791 K800 H804 N284 D621 T622 K706 Y708 M728 G729 Q733 K734 S735 S783 S784 N786 Y791 K800 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22023103 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASL 3sur A 1.9 BS01 NGT A 1 R170 D321 E322 W352 W370 Y395 D397 W410 W441 E443 R172 D323 E324 W354 W372 Y397 D399 W412 W443 E445 L19 Y25 D321 E322 L21 Y27 D323 E324 3.2.1.52 0004553,0004563,0005975 Ki=70uM remove_due_to_license_issue D2KW09 22367352 2000 HHHHSSGLVPRGSHMSQPSILPKPVSYTVGSGQFVLTKNASIFVAGNNVGETDELFNIGQALAKKLNASTGYTISVVKSNQPTAGSIYLTTVGGNAALGNEGYDLITTSNQVTLTANKPEGVFRGNQTLLQLLPAGIEKNTVVSGVQWVIPHSNISDKPEYEYRGLMLDVARHFFTVDEVKRQIDLASQYKINKFHMHLSDDQGWRIEIKSWPDLIEIGSKGQVGGGPGGYYTQEQFKDIVSYAAERYIEVIPEIDMPGHTNAALASYGELNPDGKRKAMRTDTAVGYSTLMPRAEITYQFVEDVISELAAISPSPYIHLGGDESNATSAADYDYFFGRVTAIANSYGKKVVGWDPSDTSSGATSDSVLQNWTCSASTGTAAKAKGMKVIVSPANAYLDMKYYSDSPIGLQWRGFVNTNRAYNWDPTDCIKGANIYGVESTLWTETFVTQDHLDYMLYPKLLSNAEVGWTARGDRNWDDFKERLIEHTPRLQNKGIKFFADPIV 3sus A 1.8 BS01 GNL A 1 R170 D321 E322 W370 Y395 D397 W410 W441 E443 R172 D323 E324 W372 Y397 D399 W412 W443 E445 L19 Y25 D321 E322 L21 Y27 D323 E324 3.2.1.52 0004553,0004563,0005975 Ki=71uM remove_due_to_license_issue D2KW09 22367352 2000 HHHHSSGLVPRGSHMSQPSILPKPVSYTVGSGQFVLTKNASIFVAGNNVGETDELFNIGQALAKKLNASTGYTISVVKSNQPTAGSIYLTTVGGNAALGNEGYDLITTSNQVTLTANKPEGVFRGNQTLLQLLPAGIEKNTVVSGVQWVIPHSNISDKPEYEYRGLMLDVARHFFTVDEVKRQIDLASQYKINKFHMHLSDDQGWRIEIKSWPDLIEIGSKGQVGGGPGGYYTQEQFKDIVSYAAERYIEVIPEIDMPGHTNAALASYGELNPDGKRKAMRTDTAVGYSTLMPRAEITYQFVEDVISELAAISPSPYIHLGGDESNATSAADYDYFFGRVTAIANSYGKKVVGWDPSDTSSGATSDSVLQNWTCSASTGTAAKAKGMKVIVSPANAYLDMKYYSDSPIGLQWRGFVNTNRAYNWDPTDCIKGANIYGVESTLWTETFVTQDHLDYMLYPKLLSNAEVGWTARGDRNWDDFKERLIEHTPRLQNKGIKFFADPIV 3sut A 1.9 BS01 OAN A 1 R170 D321 E322 W370 Y395 D397 W410 W441 E443 R172 D323 E324 W372 Y397 D399 W412 W443 E445 L19 Y25 D321 E322 L21 Y27 D323 E324 3.2.1.52 0004553,0004563,0005975 Ki=0.014uM remove_due_to_license_issue D2KW09 22367352 2000 HHHHSSGLVPRGSHMSQPSILPKPVSYTVGSGQFVLTKNASIFVAGNNVGETDELFNIGQALAKKLNASTGYTISVVKSNQPTAGSIYLTTVGGNAALGNEGYDLITTSNQVTLTANKPEGVFRGNQTLLQLLPAGIEKNTVVSGVQWVIPHSNISDKPEYEYRGLMLDVARHFFTVDEVKRQIDLASQYKINKFHMHLSDDQGWRIEIKSWPDLIEIGSKGQVGGGPGGYYTQEQFKDIVSYAAERYIEVIPEIDMPGHTNAALASYGELNPDGKRKAMRTDTAVGYSTLMPRAEITYQFVEDVISELAAISPSPYIHLGGDESNATSAADYDYFFGRVTAIANSYGKKVVGWDPSDTSSGATSDSVLQNWTCSASTGTAAKAKGMKVIVSPANAYLDMKYYSDSPIGLQWRGFVNTNRAYNWDPTDCIKGANIYGVESTLWTETFVTQDHLDYMLYPKLLSNAEVGWTARGDRNWDDFKERLIEHTPRLQNKGIKFFADPIV 3suu A 1.6 BS01 OGN A 1 R170 D321 E322 W370 Y395 D397 W410 W441 E443 R172 D323 E324 W372 Y397 D399 W412 W443 E445 L19 Y25 D321 E322 L21 Y27 D323 E324 3.2.1.52 0004553,0004563,0005975 Ki=0.003uM remove_due_to_license_issue D2KW09 22367352 2000 HHHHSSGLVPRGSHMSQPSILPKPVSYTVGSGQFVLTKNASIFVAGNNVGETDELFNIGQALAKKLNASTGYTISVVKSNQPTAGSIYLTTVGGNAALGNEGYDLITTSNQVTLTANKPEGVFRGNQTLLQLLPAGIEKNTVVSGVQWVIPHSNISDKPEYEYRGLMLDVARHFFTVDEVKRQIDLASQYKINKFHMHLSDDQGWRIEIKSWPDLIEIGSKGQVGGGPGGYYTQEQFKDIVSYAAERYIEVIPEIDMPGHTNAALASYGELNPDGKRKAMRTDTAVGYSTLMPRAEITYQFVEDVISELAAISPSPYIHLGGDESNATSAADYDYFFGRVTAIANSYGKKVVGWDPSDTSSGATSDSVLQNWTCSASTGTAAKAKGMKVIVSPANAYLDMKYYSDSPIGLQWRGFVNTNRAYNWDPTDCIKGANIYGVESTLWTETFVTQDHLDYMLYPKLLSNAEVGWTARGDRNWDDFKERLIEHTPRLQNKGIKFFADPIV 3suv A 1.6 BS01 NOK A 1 R170 D321 E322 W352 W370 Y395 W410 W441 E443 R172 D323 E324 W354 W372 Y397 W412 W443 E445 L19 Y25 D321 E322 L21 Y27 D323 E324 3.2.1.52 0004553,0004563,0005975 remove_due_to_license_issue D2KW09 22367352 2000 HHHHSSGLVPRGSHMSQPSILPKPVSYTVGSGQFVLTKNASIFVAGNNVGETDELFNIGQALAKKLNASTGYTISVVKSNQPTAGSIYLTTVGGNAALGNEGYDLITTSNQVTLTANKPEGVFRGNQTLLQLLPAGIEKNTVVSGVQWVIPHSNISDKPEYEYRGLMLDVARHFFTVDEVKRQIDLASQYKINKFHMHLSDDQGWRIEIKSWPDLIEIGSKGQVGGGPGGYYTQEQFKDIVSYAAERYIEVIPEIDMPGHTNAALASYGELNPDGKRKAMRTDTAVGYSTLMPRAEITYQFVEDVISELAAISPSPYIHLGGDESNATSAADYDYFFGRVTAIANSYGKKVVGWDPSDTSSGATSDSVLQNWTCSASTGTAAKAKGMKVIVSPANAYLDMKYYSDSPIGLQWRGFVNTNRAYNWDPTDCIKGANIYGVESTLWTETFVTQDHLDYMLYPKLLSNAEVGWTARGDRNWDDFKERLIEHTPRLQNKGIKFFADPIV 3suw A 1.9 BS01 GC2 A 1 R170 D321 E322 W352 W370 Y395 W410 W441 E443 R172 D323 E324 W354 W372 Y397 W412 W443 E445 L19 Y25 D321 E322 L21 Y27 D323 E324 3.2.1.52 0004553,0004563,0005975 Ki=20uM remove_due_to_license_issue D2KW09 22367352 2000 HHHHSSGLVPRGSHMSQPSILPKPVSYTVGSGQFVLTKNASIFVAGNNVGETDELFNIGQALAKKLNASTGYTISVVKSNQPTAGSIYLTTVGGNAALGNEGYDLITTSNQVTLTANKPEGVFRGNQTLLQLLPAGIEKNTVVSGVQWVIPHSNISDKPEYEYRGLMLDVARHFFTVDEVKRQIDLASQYKINKFHMHLSDDQGWRIEIKSWPDLIEIGSKGQVGGGPGGYYTQEQFKDIVSYAAERYIEVIPEIDMPGHTNAALASYGELNPDGKRKAMRTDTAVGYSTLMPRAEITYQFVEDVISELAAISPSPYIHLGGDESNATSAADYDYFFGRVTAIANSYGKKVVGWDPSDTSSGATSDSVLQNWTCSASTGTAAKAKGMKVIVSPANAYLDMKYYSDSPIGLQWRGFVNTNRAYNWDPTDCIKGANIYGVESTLWTETFVTQDHLDYMLYPKLLSNAEVGWTARGDRNWDDFKERLIEHTPRLQNKGIKFFADPIV 3sv2 H 1.3 BS03 P05 H 1 Y60A W60D E192 S195 S214 W215 G216 Y47 W50 E195 S198 S219 W220 G221 3.4.21.5 0004252,0005509,0006508,0007596 Ki=64uM remove_due_to_license_issue P00734 22366545 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3sv6 A 1.4 BS01 SV6 A 1 Q1041 H1057 R1123 L1135 G1137 S1139 R1155 A1156 A1157 S1159 Q62 H78 R144 L156 G158 S160 R176 A177 A178 S180 H1057 D1081 G1137 S1139 H78 D102 G158 S160 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue A8DG50 22910833 1 GSHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVDFIPVESLETTMRS 3sv7 A 1.55 BS01 SV6 A 1 H1057 L1135 G1137 S1139 K1155 A1156 A1157 S1159 H78 L156 G158 S160 K176 A177 A178 S180 H1057 D1081 G1137 S1139 H78 D102 G158 S160 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue A8DG50 22910833 1 GSHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFKAAVSTRGVAKAVDFIPVESLETTMR 3sv8 A 2.5 BS01 SV6 A 1 H1057 K1136 G1137 S1139 R1155 A1156 A1157 V1158 S1159 H69 K148 G149 S151 R167 A168 A169 V170 S171 H1057 D1081 G1137 S1139 H69 D93 G149 S151 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue A8DG50 22910833 1 KGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVAFIPVESLETTMRS 3sv9 A 1.6 BS01 SV6 A 1 H1057 K1136 G1137 S1139 F1154 T1156 A1157 S1159 D1168 H76 K155 G156 S158 F173 T175 A176 S178 D187 H1057 D1081 G1137 S1139 H76 D100 G156 S158 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue A8DG50 22910833 1 HMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTMR 3svj P 1.55 BS01 4LI P 1 G69 V71 E126 G127 E128 G129 H173 G68 V70 E116 G117 E118 G119 H163 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=117nM remove_due_to_license_issue Ki=117nM Q8DP79 21711014 207 SAIERITKAAHLIDMNDIIREGNPTLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNIAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLILE 3svv A 2.204 BS01 VSP A 1 A293 K295 E310 V323 L325 C338 Y340 M341 L393 A36 K38 E53 V66 L68 C81 Y83 M84 L136 D386 R388 A390 N391 D404 D129 R131 A133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 21852571 600 KDAWEIPRESLRLEVKLGQGFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVCEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3sw2 B 2.42 BS01 FI1 B 1 E97 T98 Y99 F174 A190 Q192 V213 W215 G216 G218 G226 I227 Y228 E83 T84 Y85 F162 A180 Q182 V203 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=4.71nM remove_due_to_license_issue IC50=13nM, Ki=4.71nM P00742 22041058 1 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMK 3sw8 P 1.702 BS01 5LI P 1 G70 V71 G72 Q77 E128 G129 C130 L131 V170 H173 E174 H177 G69 V70 G71 Q76 E119 G120 C121 L122 V161 H164 E165 H168 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=25910nM remove_due_to_license_issue Q939R9 21711014 205 SAIERITKAAHLIDMNDIIREGNPTLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNIEAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLILE 3sww A 2.0 BS01 KXB A 1 R125 E205 E206 Y547 S630 Y662 Y666 N710 H740 R86 E166 E167 Y508 S591 Y623 Y627 N671 H701 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=4nM remove_due_to_license_issue Ki=4nM P27487 21996520 1 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3sx4 A 2.6 BS01 KXA A 1 R125 E205 E206 Y547 S630 Y631 W659 Y662 Y666 N710 H740 R86 E166 E167 Y507 S590 Y591 W619 Y622 Y626 N670 H700 Y547 S630 Y631 D708 H740 Y507 S590 Y591 D668 H700 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue Ki=3nM P27487 21996520 1 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDSLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3sx9 A 2.65 BS01 BK7 A 1 V65 A78 K80 M112 L126 Y131 E135 L181 I194 V24 A37 K39 M71 L85 Y90 E94 L140 I153 D174 K176 E178 N179 D195 T214 D133 K135 E137 N138 D154 T173 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue IC50=3.80nM Q9BJF5 22369268 701 HSTAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3sxf A 2.04 BS01 BK5 A 1 V65 A78 K80 M112 L126 Y131 L181 I194 V21 A34 K36 M68 L82 Y87 L137 I150 D174 K176 E178 N179 D195 T214 D130 K132 E134 N135 D151 T170 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 Ki=0.0025uM remove_due_to_license_issue IC50=5.00nM Q9BJF5 22369268 701 AIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3sym A 2.4 BS01 GP0 A 1 G135 L136 D283 N284 H377 T378 N484 E672 S674 G675 X680 G124 L125 D263 N264 H348 T349 N455 E643 S645 G646 X651 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=27.1uM remove_due_to_license_issue P00489 22296957 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3syr A 2.4 BS01 GPK A 1 G135 L136 D283 N284 H377 T378 N484 E672 A673 S674 G675 G124 L125 D263 N264 H348 T349 N455 E643 A644 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=7.9uM remove_due_to_license_issue Ki=5500nM P00489 22296957 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3sz1 B 2.3 BS01 LU2 B 1 F264 K265 H266 G284 C285 F287 R288 I341 F54 K55 H56 G68 C69 F71 R72 I125 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 22391103 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKSPFVIYDMNSLMMGEDKIKFKHITKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDLHPLLQEIYKDL 3sz9 A 2.1 BS01 I3E A 1 F170 C301 C302 D457 F459 F465 F164 C295 C296 D451 F453 F459 N169 K192 E268 C302 E399 E476 N163 K186 E262 C296 E393 E470 1.2.1.3 0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627 remove_due_to_license_issue P05091 22021038 8001 AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS 3szb A 1.51 BS01 I1E A 1 Y115 L119 C243 I394 Y115 L119 C243 I394 N114 K137 E209 C243 E333 Y412 N114 K137 E209 C243 E333 Y412 1.2.1.5 0004028,0004029,0004030,0005515,0005615,0005737,0005783,0005829,0005886,0006081,0006629,0006805,0008106,0016020,0016491,0016620,0018479 remove_due_to_license_issue P30838 22021038 1001 SKISEAVKRARAAFSSGRTRPLQFRIQQLEALQRLIQEQEQELVGALAADLHKNEWNAYYEEVVYVLEEIEYMIQKLPEWAADEPVEKTPQTQQDELYIHSEPLGVVLVIGTWNYPFNLTIQPMVGAIAAGNAVVLKPSELSENMASLLATIIPQYLDKDLYPVINGGVPETTELLKERFDHILYTGSTGVGKIIMTAAAKHLTPVTLELGGKSPCYVDKNCDLDVACRRIAWGKFMNSGQTCVAPDYILCDPSIQNQIVEKLKKSLKEFYGEDAKKSRDYGRIISARHFQRVMGLIEGQKVAYGGTGDAATRYIAPTILTDVDPQSPVMQEEIFGPVLPIVCVRSLEEAIQFINQREKPLALYMFSSNDKVIKKMIAETSSGGVAANDVIVHITLHSLPFGGVGNSGMGSYHGKKSFETFSHRRSCLVRPLMNDEGLKVRYPPSPA 3szq A 2.353 BS01 dna B 0 F34 F65 K67 S142 M143 K161 H165 S229 V230 F3 F34 K36 S111 M112 K130 H134 S198 V199 3.6.1.71,3.6.1.72 0003824 remove_due_to_license_issue O74859 21984210 1 ~ 5 QSFRDNLKVYIESPESYKNVIYYDDDVVLVRDMFPKSKMHLLLMTRDPHLTHVHPLEIMMKHRSLVEKLVSYVQGDLSGLIFDEARNCLSQQLTNEALCNYIKVGFHAGPSMNNLHLHIMTLDHVSPSLKNSAHYISFTSPFFVKIDTPTSNLPTRGTLTSLFQEDLKCWRCGETFGRHFTKLKAHLQEEYDDWLDKSV 3szq A 2.353 BS02 dna C 0 F34 R209 F211 T212 F3 R178 F180 T181 3.6.1.71,3.6.1.72 0003824 remove_due_to_license_issue O74859 21984210 7 ~ 14 QSFRDNLKVYIESPESYKNVIYYDDDVVLVRDMFPKSKMHLLLMTRDPHLTHVHPLEIMMKHRSLVEKLVSYVQGDLSGLIFDEARNCLSQQLTNEALCNYIKVGFHAGPSMNNLHLHIMTLDHVSPSLKNSAHYISFTSPFFVKIDTPTSNLPTRGTLTSLFQEDLKCWRCGETFGRHFTKLKAHLQEEYDDWLDKSV 3t01 A 1.6 BS03 PPF A 1 T68 D211 I287 H377 T65 D208 I284 H374 3.6.1.9 0016787,0046872,0047400,0106379 Ki=33uM remove_due_to_license_issue Q92UV8 22035792 503 MSKISVTVNGRRYPWPRVPAIAVCLDGCEPAYLDAAIDAGLMPALKRIKERGAVRLAHSVIPSFTNPNNLSIATGSPPAVHGICGNYLYEPSTGEEVMMNDPKFLRAPTIFQAFYDAGARVAVVTAKDKLRALLGKGLRFDEGRAVCFSSEKSDKATRAEHGIDNASAWLGRPVPEVYSAALSEFVFAAGVKLLREFRPDIMYLTTTDYVQHKYAPGVPEANSFYEMFDRYLAELDGLGAAIVVTADHGMKPKHKADGSPDVIYVQDLLDEWLGKDAARVILPITDPYVVHHGALGSFATAYLPDGCDRSEIMARLKAIQGVDVVLGREEACRRFELPEDRIGDIVLVSSENKTLGTSEHRHDLAALDEPLRSHGGLTEQEVPFIVNRVLPELPNAPRLRNFDAFFYAVTAAA 3t03 A 2.1 BS02 3T0 A 1 I309 C313 R316 S317 A320 I354 L361 L381 F391 M392 I69 C73 R76 S77 A80 I114 L121 L141 F151 M152 ? 0003677,0004879,0005634,0006355 Ki=160nM remove_due_to_license_issue P37231 22584573 2 DLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHIQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3t07 A 3.3 BS01 09C B 1 A358 I361 H365 N369 A358 I361 H365 N369 R32 R73 K219 T277 R32 R73 K219 T277 2.7.1.40 0000287,0003824,0004743,0005524,0006096,0016301,0016310,0016772,0030955,0046872 remove_due_to_license_issue IC50=16nM Q6GG09 22030393 586 MRKTKIVCTIGPASESEEMIEKLINAGMNVARLNFSHGSHEEHKGRIDTIRKVAKRLDKIVAILLDTKGPEIRTHNMKDGIIELERGNEVIVSMNEVEGTPEKFSVTYENLINDVQVGSYILLDDGLIELQVKDIDHAKKEVKCDILNSGELKNKKGVNLPGVRVSLPGITEKDAEDIRFGIKENVDFIAASFVRRPSDVLEIREILEEQKANISVFPKIENQEGIDNIEEILEVSDGLMVARGDMGVEIPPEKVPMVQKDLIRQCNKLGKPVITATQMLDSMQRNPRATRAEASDVANAIYDGTDAVMLSGETAAGLYPEEAVKTMRNIAVSAEAAQDYKKLLSDRTKLVETSLVNAIGISVAHTALNLNVKAIVAATESGSTARTISKYRPHSDIIAVTPSEETARQCSIVWGVQPVVKKGRKSTDALLNNAVATAVETGRVTNGDLIIITAGVPTGETGTTNMMKIHLVGDEIANGQGIGRGSVVGTTLVAETVKDLEGKDLSDKVIVTNSIDETFVPYVEKALGLITEENGITSPSAIVGLEKGIPTVVGVEKAVKNISNNVLVTIDAAQGKIFEGYAN 3t07 B 3.3 BS01 09C B 1 A358 I361 H365 N369 L370 A358 I361 H365 N369 L370 R32 R73 K219 T277 R32 R73 K219 T277 2.7.1.40 0000287,0003824,0004743,0005524,0006096,0016301,0016310,0016772,0030955,0046872 remove_due_to_license_issue IC50=16nM Q6GG09 22030393 586 MRKTKIVCTIGPASESEEMIEKLINAGMNVARLNFSHGSHEEHKGRIDTIRKVAKRLDKIVAILLDTKGPEIRTHNMKDGIIELERGNEVIVSMNEVEGTPEKFSVTYENLINDVQVGSYILLDDGLIELQVKDIDHAKKEVKCDILNSGELKNKKGVNLPGVRVSLPGITEKDAEDIRFGIKENVDFIAASFVRRPSDVLEIREILEEQKANISVFPKIENQEGIDNIEEILEVSDGLMVARGDMGVEIPPEKVPMVQKDLIRQCNKLGKPVITATQMLDSMQRNPRATRAEASDVANAIYDGTDAVMLSGETAAGLYPEEAVKTMRNIAVSAEAAQDYKKLLSDRTKLVETSLVNAIGISVAHTALNLNVKAIVAATESGSTARTISKYRPHSDIIAVTPSEETARQCSIVWGVQPVVKKGRKSTDALLNNAVATAVETGRVTNGDLIIITAGVPTGETGTTNMMKIHLVGDEIANGQGIGRGSVVGTTLVAETVKDLEGKDLSDKVIVTNSIDETFVPYVEKALGLITEENGITSPSAIVGLEKGIPTVVGVEKAVKNISNNVLVTIDAAQGKIFEGYAN 3t08 A 2.0 BS03 IPT A 1 N102 D201 E461 Y503 E537 H540 N604 W999 N94 D193 E453 Y495 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.91mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVAEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t08 D 2.0 BS03 IPT D 1 D201 E461 Y503 E537 H540 N604 W999 D193 E453 Y495 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.91mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVAEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t09 A 1.75 BS01 149 A 1 D201 H391 N460 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 N452 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.16mM remove_due_to_license_issue P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVAEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t09 D 1.75 BS01 149 D 1 D201 H391 N460 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 N452 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.16mM remove_due_to_license_issue P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVAEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t0b A 2.4 BS03 IPT A 1 N102 D201 E461 E537 H540 N604 W999 N93 D192 E452 E528 H531 N595 W990 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D192 H348 H382 E407 H409 E452 Y494 E528 N588 F592 N595 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.05mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22155115 2001 VLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVTEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t0b D 2.4 BS03 IPT D 1 N102 D201 E461 Y503 E537 H540 N604 W999 N94 D193 E453 Y495 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.05mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVTEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t0d A 1.93 BS01 149 A 1 D201 H391 N460 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 N452 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=4.3mM remove_due_to_license_issue P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVTEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t0d D 1.93 BS01 149 D 1 D201 H391 N460 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 N452 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=4.3mM remove_due_to_license_issue P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVTEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t0l A 1.6 BS01 1CT A 1 G53 R56 R60 R129 Y130 N175 G57 R60 R64 R127 Y128 N173 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 232 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNKGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 3t0m A 1.62 BS01 2CT A 1 G53 R56 R60 R129 Y130 L174 N175 G57 R60 R64 R127 Y128 L172 N173 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 232 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNKGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 3t0t A 3.1 BS01 I30 A 1 T353 A358 I361 S362 H365 N369 T353 A358 I361 S362 H365 N369 R32 R73 K219 T277 R32 R73 K219 T277 2.7.1.40 0000287,0003824,0004743,0005524,0006096,0016301,0016310,0016772,0030955,0046872 remove_due_to_license_issue IC50=91nM Q6GG09 22066782 586 MRKTKIVCTIGPASESEEMIEKLINAGMNVARLNFSHGSHEEHKGRIDTIRKVAKRLDKIVAILLDTKGPEIRTHNMKDGIIELERGNEVIVSMNEVEGTPEKFSVTYENLINDVQVGSYILLDDGLIELQVKDIDHAKKEVKCDILNSGELKNKKGVNLPGVRVSLPGITEKDAEDIRFGIKENVDFIAASFVRRPSDVLEIREILEEQKANISVFPKIENQEGIDNIEEILEVSDGLMVARGDMGVEIPPEKVPMVQKDLIRQCNKLGKPVITATQMLDSMQRNPRATRAEASDVANAIYDGTDAVMLSGETAAGLYPEEAVKTMRNIAVSAEAAQDYKKLLSDRTKLVETSLVNAIGISVAHTALNLNVKAIVAATESGSTARTISKYRPHSDIIAVTPSEETARQCSIVWGVQPVVKKGRKSTDALLNNAVATAVETGRVTNGDLIIITAGVPTGETGTTNMMKIHLVGDEIANGQGIGRGSVVGTTLVAETVKDLEGKDLSDKVIVTNSIDETFVPYVEKALGLITEENGITSPSAIVGLEKGIPTVVGVEKAVKNISNNVLVTIDAAQGKIFEGYAN 3t0t B 3.1 BS01 I30 A 1 I361 S362 H365 T366 N369 L370 I361 S362 H365 T366 N369 L370 R32 R73 K219 T277 R32 R73 K219 T277 2.7.1.40 0000287,0003824,0004743,0005524,0006096,0016301,0016310,0016772,0030955,0046872 remove_due_to_license_issue IC50=91nM Q6GG09 22066782 586 MRKTKIVCTIGPASESEEMIEKLINAGMNVARLNFSHGSHEEHKGRIDTIRKVAKRLDKIVAILLDTKGPEIRTHNMKDGIIELERGNEVIVSMNEVEGTPEKFSVTYENLINDVQVGSYILLDDGLIELQVKDIDHAKKEVKCDILNSGELKNKKGVNLPGVRVSLPGITEKDAEDIRFGIKENVDFIAASFVRRPSDVLEIREILEEQKANISVFPKIENQEGIDNIEEILEVSDGLMVARGDMGVEIPPEKVPMVQKDLIRQCNKLGKPVITATQMLDSMQRNPRATRAEASDVANAIYDGTDAVMLSGETAAGLYPEEAVKTMRNIAVSAEAAQDYKKLLSDRTKLVETSLVNAIGISVAHTALNLNVKAIVAATESGSTARTISKYRPHSDIIAVTPSEETARQCSIVWGVQPVVKKGRKSTDALLNNAVATAVETGRVTNGDLIIITAGVPTGETGTTNMMKIHLVGDEIANGQGIGRGSVVGTTLVAETVKDLEGKDLSDKVIVTNSIDETFVPYVEKALGLITEENGITSPSAIVGLEKGIPTVVGVEKAVKNISNNVLVTIDAAQGKIFEGYAN 3t0w A 1.501 BS01 DIW A 1 Y34 V46 Y49 S55 S56 L89 W96 F98 Y35 V47 Y50 S56 S57 L90 W99 F101 remove_due_to_license_issue 22390683 204 QPVLTQSPSVSGTPGQKVTIFCSGSSSNVEDNSVYWYQQFPGTTPKVLIYNDDRRSSGVPDRFSGSKSGTSASLAISGLRSEDEADYYCLSWDDSLNGWVFGGGTKVTVLD 3t0x A 1.96 BS01 DIW A 1 Y34 Y49 P55 S56 L89 W96 Y35 Y50 P56 S57 L90 W99 remove_due_to_license_issue 22390683 201 QPVLTQSPSVSGTPGQKVTIFCSGSSSNVEDNSVYWYQQFPGTTPKVLIYNDDRRPSGVPDRFSGSKSGTSASLAISGLRSEDEADYYCLSWDDSLNGWVFGGGTKVTVLD 3t0x B 1.96 BS01 DIW A 1 Y34 Y49 W96 Y35 Y50 W99 remove_due_to_license_issue 22390683 201 QPVLTQSPSVSGTPGQKVTIFCSGSSSNVEDNSVYWYQQFPGTTPKVLIYNDDRRPSGVPDRFSGSKSGTSASLAISGLRSEDEADYYCLSWDDSLNGWVFGGGTKVTV 3t19 A 2.6 BS01 5MA A 1 L100 K101 K103 V106 Y188 G190 P225 F227 W229 L234 H235 P236 Y318 L97 K98 K100 V103 Y185 G187 P222 F224 W226 L231 H232 P233 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 21985673 561 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3t1a A 2.4 BS01 5MA A 1 P95 L100 K101 N103 V106 V108 Y181 Y188 V189 F227 W229 L234 H235 P236 Y318 P92 L97 K98 N100 V103 V105 Y178 Y185 V186 F224 W226 L231 H232 P233 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 Ki=4.3nM remove_due_to_license_issue P04585 21985673 561 SPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3t1l A 1.6 BS01 MQT A 1 R144 H158 R162 N174 W181 E184 R32 H46 R50 N62 W69 E72 ? 0030246 Kd=0.55mM remove_due_to_license_issue Kd=550000nM P17931 22136701 1 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 3t1m A 1.55 BS01 DQT A 1 N143 R144 A146 H158 R162 N174 W181 E184 N30 R31 A33 H45 R49 N61 W68 E71 ? 0030246 Kd=0.91mM remove_due_to_license_issue P17931 22136701 1 LIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 3t2p A 2.6 BS01 IPT A 1 D201 E461 Y503 E537 H540 N604 W999 D192 E452 Y494 E528 H531 N595 W990 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D192 H348 H382 E407 H409 E452 Y494 E528 N588 F592 N595 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 22155115 2001 VLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVDEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t2p D 2.6 BS01 IPT D 1 N102 D201 E461 E537 H540 W999 N94 D193 E453 E529 H532 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVDEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t2q A 2.4 BS01 149 A 1 D201 E461 M502 Y503 E537 H540 W568 F601 N604 D193 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.22mM remove_due_to_license_issue P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVDEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t2q D 2.4 BS01 149 D 1 D201 H391 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.22mM remove_due_to_license_issue P00722 22155115 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGNESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVDEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3t2t A 1.9 BS01 MQT A 1 V31 H44 R48 H52 N61 E71 V31 H44 R48 H52 N61 E71 ? 0002317,0003723,0005515,0005576,0005615,0005737,0005788,0005829,0005886,0006915,0007165,0030246,0030395,0031295,0042981,0043065,0043123,0043236,0045445,0046598,0048018,0050729,0062023,0070062,0098609,1990724,2000329,2001200 remove_due_to_license_issue Kd=>4000000nM P09382 22136701 135 ACGLVASNLNLKPGECLRVRGEVAPDAKSFVLNLGKDSNNLCLHFNPRFNAHGDANTIVCNSKDGGAWGTEQREAVFPFQPGSVAEVCITFDQANLTVKLPDGYEFKFPNRLNLEAINYMAADGDFKIKCVAFD 3t2v B 2.51 BS01 KKJ D 1 D2 C6 L134 D2 C6 L134 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 23149273 172 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3t2v D 2.51 BS01 KKJ D 1 R31 R138 R31 R138 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 23149273 172 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3t2w A 1.5 BS01 BTN A 1 N15 S19 Y36 N38 W67 C74 S76 T78 W97 D115 N12 S16 Y33 N35 W64 C71 S73 T75 W92 D110 ? 0009374 Kd=0.000000064M remove_due_to_license_issue Q12QS6 22493427 600 AQELTAMSAWVNQDGSTLYINSINAQGELTGSYINRAAGAACQNSPYPVNGWVFGTAISFSTKWLNSVESCNSITSWSGFYINGQGKISTLWQLVVNGSSSPSQILKGQDVFSQT 3t3c A 2.1 BS01 017 A 1 D25 G27 A28 D29 D30 A48 I50 D25 G27 A28 D29 D30 A48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.059nM remove_due_to_license_issue P03367 22644035 201 PQISLWQRPVVTARIGGQLIEVLLDTGADDTVIEDIDLPGKWSPKMIAGIGGFVKVRQYDQILIEFCGKKAIGSVLVGPTPANVIGRNIMSQIGCTLNF 3t3c B 2.1 BS01 017 A 1 D25 A28 D30 V32 A82 D25 A28 D30 V32 A82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22644035 201 PQISLWQRPVVTARIGGQLIEVLLDTGADDTVIEDIDLPGKWSPKMIAGIGGFVKVRQYDQILIEFCGKKAIGSVLVGPTPANVIGRNIMSQIGCTLNF 3t3d A 2.5 BS01 CJB A 1 G135 L136 D283 N284 H377 N484 E672 S674 G675 G124 L125 D266 N267 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=12.39uM remove_due_to_license_issue Ki=6100nM P00489 22267166 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3t3e A 2.15 BS01 GPQ A 1 G135 L136 D283 N284 H377 T378 N484 E672 A673 S674 G675 G124 L125 D266 N267 H351 T352 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=1.02uM remove_due_to_license_issue Ki=1020nM P00489 22267166 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3t3g A 2.4 BS01 GPU A 1 G135 L136 D283 N284 H377 T378 N484 E672 A673 S674 G675 G124 L125 D263 N264 H348 T349 N455 E643 A644 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=3.27uM remove_due_to_license_issue P00489 22267166 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3t3h A 2.6 BS01 GPV A 1 G135 L136 D283 N284 D339 H377 T378 N484 E672 A673 S674 G675 G124 L125 D263 N264 D310 H348 T349 N455 E643 A644 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 22267166 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3t3i A 2.65 BS01 GPW A 1 G135 L136 D283 N284 H377 T378 N484 E672 A673 S674 G675 G124 L125 D266 N267 H351 T352 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 22267166 843 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 3t3u A 2.1 BS01 BK6 A 1 V65 A78 K80 M112 L126 Y131 E135 L181 I194 V21 A34 K36 M68 L82 Y87 E91 L137 I150 D174 K176 E178 N179 D195 T214 D130 K132 E134 N135 D151 T170 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 Ki=0.0025uM remove_due_to_license_issue IC50=4.90nM Q9BJF5 22369268 701 AIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3t3v A 2.04 BS01 BK4 A 1 G58 V65 A78 K80 M112 L126 Y131 L181 I194 G14 V21 A34 K36 M68 L82 Y87 L137 I150 D174 K176 E178 N179 D195 T214 D130 K132 E134 N135 D151 T170 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 Ki=0.003uM remove_due_to_license_issue IC50=6.00nM Q9BJF5 22369268 701 AIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMSMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3t3y A 2.001 BS02 MD6 A 1 Y122 L128 H131 D133 S145 W178 H187 I189 R204 N206 T208 Y107 L113 H116 D118 S130 W163 H172 I174 R189 N191 T193 1.14.11.33 0005515,0005737,0005829,0006281,0006307,0008198,0035513,0035515,0035516,0042245,0046872,0051213,0070989,0072702 ic50=3.4uM remove_due_to_license_issue P05050 22263962 401 AAGAVILRRFAFNAAEQLIRDINDVASQSPFRQMVTPGGYTMSVAMTNCGHLGWTTHRQGYLYSPIDPQTNKPWPAMPQSFHNLCQRAATAAGYPDFQPDACLINRYAPGAKLSLHQDKDEPDLRAPIVSVSLGLPAIFQFGGLKRNDPLKRLLLEHGDVVVWGGESRLFYHGIQPLKAGFHPLTIDCRYNLTFRQAGK 3t4h B 1.65 BS02 MD5 B 1 N120 Y122 L128 H131 S145 F154 W178 S182 H187 I189 R204 N206 T208 R210 N107 Y109 L115 H118 S132 F141 W165 S169 H174 I176 R191 N193 T195 R197 1.14.11.33 0005515,0005737,0005829,0006281,0006307,0008198,0035513,0035515,0035516,0042245,0046872,0051213,0070989,0072702 ic50=5.2uM remove_due_to_license_issue P05050 22263962 217 PLAAGAVILRRFAFNAAEQLIRDINDVASQSPFRQMVTPGGYTMSVAMTNCGHLGWTTHRQGYLYSPIDPQTNKPWPAMPQSFHNLCQRAATAAGYPDFQPDACLINRYAPGAKLSLHQDKDEPDLRAPIVSVSLGLPAIFQFGGLKRNDPLKRLLLEHGDVVVWGGESRLFYHGIQPLKAGFHPLTIDCRYNLTFRQAGK 3t4n C 2.3 BS01 ADP C 1 T196 M200 K201 V221 S222 V308 T310 S312 D313 T185 M189 K190 V210 S211 V297 T299 S301 D302 ? 0004679,0005515,0005524,0005634,0005641,0005737,0005829,0005886,0006110,0006357,0006914,0007031,0016208,0019887,0019901,0030447,0031588,0042149,0042802,0043539,0043609,0045722,1904547,2000217 Kd=72uM remove_due_to_license_issue P12904 22019086 324 SQEKVSIEQQLAVESIRKFLNSKTSYDVLPVSYRLIVLDTSLLVKKSLNVLLQNSIVSAPLWDSKTSRFAGLLTTTDFINVIQYYFSNPDKFELVDKLQLDGLKDIERALGVTASIHPSRPLFEACLKMLESRSGRIPLIDQDEETHREIVVSVLTQYRILKFVALNCRETHFLKIPIGDLNIITQDNMKSCQMTTPVIDVIQMLTQGRVSSVPIIDENGYLINVYEAYDVLGLIKGGIYNDLSLSVGEALMRRSDDFEGVYTCTKNDKLSTIMDNIRKARVHRFFVVDDVGRLVGVLTLSDILKYILLGS 3t4v A 1.732 BS02 MD3 A 1 N120 Y122 L128 H131 D133 I143 S145 F154 W178 R183 H187 I189 R204 N206 T208 R210 N106 Y108 L114 H117 D119 I129 S131 F140 W164 R169 H173 I175 R190 N192 T194 R196 1.14.11.33 0005515,0005737,0005829,0006281,0006307,0008198,0035513,0035515,0035516,0042245,0046872,0051213,0070989,0072702 ic50=0.5uM remove_due_to_license_issue P05050 22263962 401 LAAGAVILRRFAFNAAEQLIRDINDVASQSPFRQMVTPGGYTMSVAMTNCGHLGWTTHRQGYLYSPIDPQTNKPWPAMPQSFHNLCQRAATAAGYPDFQPDACLINRYAPGAKLSLHQDKDEPDLRAPIVSVSLGLPAIFQFGGLKRNDPLKRLLLEHGDVVVWGGESRLFYHGIQPLKAGFHPLTIDCRYNLTFRQAG 3t5u A 1.75 BS02 A09 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.47uM remove_due_to_license_issue Ki=26nM P00918 21952494 263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3t5u A 1.75 BS03 A09 A 2 W5 H10 N11 H15 W16 D19 W2 H7 N8 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.47uM remove_due_to_license_issue Ki=26nM P00918 21952494 264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3t5u A 1.75 BS04 A09 A 3 Y7 D243 W245 Y4 D239 W241 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.47uM remove_due_to_license_issue Ki=26nM P00918 21952494 265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3t5u A 1.75 BS05 A09 A 4 E69 I91 Q92 E66 I88 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.47uM remove_due_to_license_issue Ki=26nM P00918 21952494 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 3t60 A 2.396 BS01 DUA A 1 F46 N103 G106 Y112 I117 F39 N80 G83 Y89 I94 S27 R91 S93 L99 D109 S20 R68 S70 L76 D86 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.2uM remove_due_to_license_issue Ki=200nM Q8II92 22049550 182 MHLKIVCLSDEVREMYKNDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFG 3t60 A 2.396 BS02 DUA C 1 S92 S93 S69 S70 S27 R91 S93 L99 D109 S20 R68 S70 L76 D86 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.2uM remove_due_to_license_issue Ki=200nM Q8II92 22049550 182 MHLKIVCLSDEVREMYKNDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFG 3t60 B 2.396 BS01 DUA A 1 S92 S93 S71 S72 S27 R91 S93 L99 D109 S20 R70 S72 L78 D88 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.2uM remove_due_to_license_issue Ki=200nM Q8II92 22049550 182 MHLKIVCLSDEVREMYKNDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELV 3t60 B 2.396 BS02 DUA B 1 F46 N103 G106 Y112 I117 A119 F39 N82 G85 Y91 I96 A98 S27 R91 S93 L99 D109 S20 R70 S72 L78 D88 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.2uM remove_due_to_license_issue Ki=200nM Q8II92 22049550 182 MHLKIVCLSDEVREMYKNDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELV 3t64 A 1.65 BS02 DU3 A 1 F46 N103 G106 I108 Y112 I117 F46 N89 G92 I94 Y98 I103 S27 R91 S93 L99 D109 S27 R77 S79 L85 D95 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.2uM remove_due_to_license_issue Q8II92 22049550 201 MHLKIVCLSDEVREMYKNHKTHHEGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFGS 3t64 B 1.65 BS02 DU3 B 1 F46 N103 G106 I108 Y112 I116 I117 F40 N83 G86 I88 Y92 I96 I97 S27 R91 S93 L99 D109 S21 R71 S73 L79 D89 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.2uM remove_due_to_license_issue Q8II92 22049550 201 MHLKIVCLSDEVREMYKNHDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEEL 3t6y A 2.6 BS02 DU2 A 1 F46 N103 G106 I108 Y112 I116 I117 F42 N86 G89 I91 Y95 I99 I100 S27 R91 S93 L99 D109 S23 R74 S76 L82 D92 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 remove_due_to_license_issue Q8II92 22049550 400 MHLKIVCLSDEVREMYKNHKGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKSNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFGS 3t6y B 2.6 BS02 DU2 B 1 F46 N103 G106 I108 Y112 I116 I117 F41 N85 G88 I90 Y94 I98 I99 S27 R91 S93 L99 D109 S22 R73 S75 L81 D91 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 remove_due_to_license_issue Q8II92 22049550 400 MHLKIVCLSDEVREMYKNHGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKSNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEEL 3t70 A 1.8 BS02 DU4 A 1 F46 N103 G106 I108 Y112 I117 A119 F42 N85 G88 I90 Y94 I99 A101 S27 R91 S93 L99 D109 S23 R73 S75 L81 D91 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.5uM remove_due_to_license_issue Q8II92 22049550 400 MHLKIVCLSDEVREMYKNHKGDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELDETSRGEGGFGS 3t70 B 1.8 BS02 DU4 A 1 S92 K96 S73 K77 S27 R91 S93 L99 D109 S21 R72 S74 L80 D90 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.5uM remove_due_to_license_issue Q8II92 22049550 400 MHLKIVCLSDEVREMYKNHDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKCNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELD 3t70 B 1.8 BS03 DU4 B 1 F46 N103 G106 I108 Y112 I117 F40 N84 G87 I89 Y93 I98 S27 R91 S93 L99 D109 S21 R72 S74 L80 D90 3.6.1.23 0000287,0004170,0006226,0006260,0006399,0009117,0016787,0042802,0046081,0046872 Ki=0.5uM remove_due_to_license_issue Q8II92 22049550 400 MHLKIVCLSDEVREMYKNHDSGLDLFIVKDEVLKPKSTTFVKLGIKAIALQYKSNYYYKCNIVNTSFLLFPRSSISKTPLRLANSIGLIDAGYRGEIIAALDNTSDQEYHIKKNDKLVQLVSFTGEPLSFELVEELD 3t82 A 2.002 BS02 SG4 A 1 N62 N67 Q92 H94 L197 T198 T199 N59 N64 Q89 H91 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=101nM remove_due_to_license_issue P00918 21958118 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3t83 A 1.8 BS02 SG5 A 1 N62 A65 F66 N67 Q92 H94 L197 T198 T199 N59 A62 F63 N64 Q89 H91 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=105nM remove_due_to_license_issue P00918 21958118 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3t84 A 2.0 BS02 SG6 A 1 N62 N67 Q92 H94 V121 L197 T198 T199 N59 N64 Q89 H91 V118 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=106nM remove_due_to_license_issue P00918 21958118 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3t85 A 2.4 BS02 SG7 A 1 N67 Q92 H94 F130 T198 T199 N64 Q89 H91 F127 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11.3nM remove_due_to_license_issue P00918 21958118 300 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3t8s B 3.77 BS01 I3P B 1 R265 T267 Y567 R568 R251 T253 Y469 R470 ? 0005220,0005262,0005783,0006816,0016020,0070588,0070679 remove_due_to_license_issue Kd=8.7nM, EC50=209nM P29994 21892169 603 SFLHIGDICSLYAEGSTNGFISTLGLVDDRCVVQPEAGDLNNPPKKFRDCLFKLCPMNRYSAQKQFWKTTDAVLLNKLHHAADLEKKQNETENRKLLGTVIQYGNVIQLLHLKSNKYLTVNKRLPALLEKNAMRVTLDEAGNEGSWFYIQPFYKLRSIGDSVVIGDKVVLNPVNAGQPLHASSHQLVDNPGCNEVNSVNCNTSWKIVLFMKWSDNKDDILKGGDVVRLFHAEQEKFLTCDEHRKKQHVFLRTTSATSSKALWEVEVVQHDPWNSLFRFKHLATGHYLAAEVDYSLVSVPEGNDISSIFELDPLVPRNSYVRLRHLCTNTWVHSTNIPIDKEEEKPVMLKIGTSPLKEDKEAFAIVPVSPAEVRDLDFANDASKVLGSIAGKLEKGTITQNERRSVTKLLEDLVYFVTGEVVFSKPNRERQKLMREQNILKQIFKLLQAPPFRHICRLCYRVLRHSQQDYRKNQEYIAKQFGF 3t8v A 1.8 BS02 BTJ A 1 Q317 E319 V459 G460 A461 M462 H496 E497 H500 E519 A572 Y575 Y580 M1034 Q1038 Q122 E124 V264 G265 A266 M267 H301 E302 H305 E324 A377 Y380 Y385 M839 Q843 E463 H496 E497 H500 E519 A572 Y580 E268 H301 E302 H305 E324 A377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=260nM remove_due_to_license_issue O96935 21844374 1092 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMANFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 3t8w A 2.0 BS04 DGZ A 1 K374 D379 A388 G390 M392 M396 F398 D399 N457 D459 E461 T486 L487 T488 G489 A490 Y493 I547 K290 D295 A304 G306 M308 M312 F314 D315 N373 D375 E377 T402 L403 T404 G405 A406 Y409 I463 K386 R463 K302 R379 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=330nM remove_due_to_license_issue Q8IL11 21844374 615 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3t8w B 2.0 BS04 DGZ B 1 K374 D379 A388 P389 G390 M392 M396 F398 D399 N457 D459 E461 T486 L487 G489 A490 Y493 I547 K288 D293 A302 P303 G304 M306 M310 F312 D313 N371 D373 E375 T400 L401 G403 A404 Y407 I461 K386 R463 K300 R377 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=330nM remove_due_to_license_issue Q8IL11 21844374 615 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3t8w D 2.0 BS04 DGZ D 1 K374 D379 A388 P389 G390 M392 F398 D399 N457 D459 E461 T486 L487 T488 G489 A490 Y493 I547 S550 K285 D290 A299 P300 G301 M303 F309 D310 N368 D370 E372 T397 L398 T399 G400 A401 Y404 I458 S461 K386 R463 K297 R374 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=330nM remove_due_to_license_issue Q8IL11 21844374 615 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3t8w F 2.0 BS04 DGZ F 1 K374 D379 A388 P389 M392 M396 F398 D399 N457 D459 E461 T486 L487 T488 G489 A490 Y493 I547 V551 K282 D287 A296 P297 M300 M304 F306 D307 N365 D367 E369 T394 L395 T396 G397 A398 Y401 I455 V459 K386 R463 K294 R371 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=330nM remove_due_to_license_issue Q8IL11 21844374 615 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 3t9t A 1.65 BS01 IAQ A 1 I369 S371 G372 V377 A389 K391 L433 T435 F437 M438 C442 L489 S499 I14 S16 G17 V22 A34 K36 L78 T80 F82 M83 C87 L134 S144 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Q08881 21958547 800 WVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVTEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 3ta0 A 2.3 BS01 ATP A 1 G35 R36 G37 E38 Q39 F86 G87 G89 R90 G35 R36 G37 E38 Q39 F73 G74 G76 R77 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 200 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEQVDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVA 3ta0 A 2.3 BS02 ATP C 1 G27 M28 T29 V63 V64 R103 G27 M28 T29 V50 V51 R90 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 200 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEQVDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVA 3ta0 B 2.3 BS01 ATP A 1 G27 M28 T29 V63 V64 R103 G27 M28 T29 V48 V49 R88 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 200 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVAAA 3ta0 B 2.3 BS02 ATP B 1 G35 R36 G37 E38 G87 G89 R90 G35 R36 G37 E38 G72 G74 R75 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 200 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVAAA 3ta1 A 1.9 BS01 ADP A 1 G35 R36 G37 E38 Q39 G87 G89 R90 G35 R36 G37 E38 Q39 G85 G87 R88 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 119 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEQKGIRLQFRGVEVDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVAAA 3ta1 A 1.9 BS02 ADP D 1 G27 M28 T29 V63 V64 K101 R103 G27 M28 T29 V61 V62 K99 R101 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 119 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEQKGIRLQFRGVEVDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVAAA 3ta1 C 1.9 BS01 ADP A 1 G27 M28 T29 V63 V64 R103 G27 M28 T29 V54 V55 R94 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 119 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEQKGIEVDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVAAA 3ta1 C 1.9 BS02 ADP C 1 G35 R36 G37 E38 K58 F86 G87 G89 R90 G35 R36 G37 E38 K49 F77 G78 G80 R81 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue O28524 22039461 119 MKMVVAVIRPEKLECVKKALEERGFVGMTVTEVKGRGEQKGIEVDLLQKTKVEVVVSDDAVDEVVEAIVSSARTGKFGDGRIFVIPVEKSVKIRTGDEEVAAA 3tam A 2.51 BS01 M06 A 1 N103 V106 V108 Y188 F227 W229 L234 H235 P236 Y318 N99 V102 V104 Y184 F223 W225 L230 H231 P232 Y314 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 22071300 561 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 3tao A 1.45 BS01 PGH A 1 K12 H100 I177 G178 G217 S218 L237 G239 G240 K11 H99 I176 G177 G216 S217 L236 G238 G239 N10 K12 H100 E102 E172 G178 S218 N9 K11 H99 E101 E171 G177 S217 5.3.1.1 0004807,0005515,0005576,0005737,0005829,0005886,0006094,0006096,0016853,0019563,0046166 Kd=7.28uM remove_due_to_license_issue P9WG43 22120738 268 SRKPLIAGNWKMNLNHYEAIALVQKIAFSLPDKYYDRVDVAVIPPFTDLRSVQTLVDGDKLRLTYGAQDLSPHDSGAYTGDVSGAFLAKLGCSYVVVGHSERRTYHNEDDALVAAKAATALKHGLTPIVCIGEHLDVREAGNHVAHNIEQLRGSLAGLLAEQIGSVVIAYEPVWAIGTGRVASAADAQEVCAAIRKELASLASPRIADTVRVLYGGSVNAKNVGDIVAQDDVDGGLVGGASLDGEHFATLAAIAAG 3tao A 1.45 BS02 PGH A 2 R51 S52 T55 R50 S51 T54 N10 K12 H100 E102 E172 G178 S218 N9 K11 H99 E101 E171 G177 S217 5.3.1.1 0004807,0005515,0005576,0005737,0005829,0005886,0006094,0006096,0016853,0019563,0046166 Kd=7.28uM remove_due_to_license_issue P9WG43 22120738 269 SRKPLIAGNWKMNLNHYEAIALVQKIAFSLPDKYYDRVDVAVIPPFTDLRSVQTLVDGDKLRLTYGAQDLSPHDSGAYTGDVSGAFLAKLGCSYVVVGHSERRTYHNEDDALVAAKAATALKHGLTPIVCIGEHLDVREAGNHVAHNIEQLRGSLAGLLAEQIGSVVIAYEPVWAIGTGRVASAADAQEVCAAIRKELASLASPRIADTVRVLYGGSVNAKNVGDIVAQDDVDGGLVGGASLDGEHFATLAAIAAG 3tay A 1.85 BS01 MN0 A 1 R101 Y188 Y189 S190 R40 Y127 Y128 S129 ? 0019028,0019058 Kd=0.42mM remove_due_to_license_issue P0C6Y8 23035213 1000 GSLLDGPYQPTTFNPPTSYWILLAPTVEGVVIQGTNNIDRWLATILIEPNVQTTNRIYNLFGQQVTLSVENTSQTQWKFIDVSKTTPTGNYTQHGSLFSTPKLYAVMKFSGRIYTYNGTTPNATTGYYSTTNYDTVNMTSFCDFYIIPRNQEEKCTEYINHGL 3tb6 A 2.21 BS01 ARB A 1 Y92 N170 Q214 R218 N273 D301 Y14 N92 Q136 R140 N195 D223 ? 0006355 remove_due_to_license_issue P96711 22281747 400 NKTIGVLTTYISDYIFPSIIRGIESYLSEQGYSMLLTSTNNNPDNERRGLENLLSQHIDGLIVEPTKSALQTPNIGYYLNLEKNGIPFAMINASYAELAAPSFTLDDVKGGMMAAEHLLSLGHTHMMGIFKADDTQGVKRMNGFIQAHRERELFPSPDMIVTFTTEEKESKLLEKVKATLEKNSKHMPTAILCYNDEIALKVIDMLREMDLKVPEDMSIVGYDDSHFAQISEVKLTSVKHPKSVLGKAAAKYVIDCLEHKKPKQEDVIFEPELIIRQSARKLN 3tc5 A 1.4 BS01 3T5 A 1 K63 R68 R69 F125 Q129 M130 Q131 F134 S154 H157 K44 R49 R50 F106 Q110 M111 Q112 F115 S135 H138 H59 C113 Q131 S154 H157 H40 C94 Q112 S135 H138 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0006626,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0071456,0080090,0090263,0098978,0099524,0140839,0140840,1900180,1902430,1990757,2000146 remove_due_to_license_issue Q13526 21797253 164 LPPGWEKAMSRSSGRVYYFNHITNASQWERPEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3tcp A 2.69 BS01 CKJ A 1 V601 A617 F673 M674 K675 R727 M730 V20 A36 F86 M87 K88 R140 M143 D723 A725 R727 N728 D741 D136 A138 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=2.9nM, Ki=4.3nM Q12866 22662287 1 LEDVVIDRNLLILGKILGSVMEGNLKQEDGTSLKVAVKTMKLDNSSQREIEEFLSEAACMKDFSHPNVIRLLGVCIEPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESLPD 3tct A 1.3 BS01 3MI A 1 L110 S117 T118 L100 S107 T108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3nM remove_due_to_license_issue IC50=3100nM, Kd=274nM P02766 22645360 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 3tct B 1.3 BS01 3MI B 1 K15 L17 S117 T118 K5 L7 S107 T108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3nM remove_due_to_license_issue IC50=3100nM, Kd=274nM P02766 22645360 128 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 3tcy A 1.55 BS01 PHE A 1 A158 Y159 K165 L175 T254 P256 D257 F258 A152 Y153 K159 L169 T248 P250 D251 F252 H138 H143 E184 S203 H132 H137 E178 S197 1.14.16.1 0004497,0004505,0005506,0006559,0009072,0016714,0019293,0046872 remove_due_to_license_issue P30967 23860686 302 FVVPDITTRKNVGLSHDANDFTLPQPLDRYSAEDHATWATLYQRQCKLLPGRACDEFLEGLERLEVDADRVPDFNKLNEKLMAATGWKIVAVPGLIPDDVFFEHLANRRFPVTWWLREPHQLDYLQEPDVFHDLFGHVPLLINPVFADYLEAYGKGGVKAKALGALPMLARLYWYTVEFGLINTPAGMRIYGAGILSSKSESIYCLDSASPNRVGFDLMRIMNTRYRIDTFQKTYFVIDSFKQLFDATAPDFAPLYLQLADAQPWGAGDIAPDDLVL 3td4 A 1.79 BS01 API A 1 T236 N237 T270 D271 T273 G274 N279 L282 R286 R329 T19 N20 T53 D54 T56 G57 N62 L65 R69 R112 ? 0016020 Kd=2.2uM remove_due_to_license_issue Q6RYW5 21965596 401 SHMELTEDLNMELRVFFDTNKSNIKDQYKPEIAKVAEKLSEYPNATARIEGHTDNTGPRKLNERLSLARANSVKSALVNEYNVDASRLSTQGFAWDQPIADNKTKEGRAMNRRVFATITGSR 3tdc A 2.41 BS01 0EU A 1 T1985 A1989 L1990 V1993 T267 A271 L272 V275 6.4.1.2 0003989,0016874 ic50=5.4nM remove_due_to_license_issue IC50=5.4nM O00763 21944854 3000 TPYVTKDLLQAKRFQAQTLGTTYIYDFPEMFRQALFKLWGSPDKYPKDILTYTELVLDSQGQLVEMNRLPGGNEVGMVAFKMRFKTQEYPEGRDVIVIGNDITFRIGSFGPGEDLLYLRASEMARAEGIPKIYVAANSGARIGMAEEIKHMFHVAWVDPEDPHKGFKYLYLTPQDYTRISSLNSVHCKHIEEGGESRYMITDIIGKDDGLGVENLRGSGMIAGESSLAYEEIVTISLVTCRAIGIGAYLVRLGQRVIQVENSHIILTGASALNKVLGREVYTSNNQLGGVQIMHYNGVSHITVPDDFEGVYTILEWLSYMPKDNHSPVPIITPTDPIDREIEFLPSRAPYDPRWMLAGRPHPTLKGTWQSGFFDHGSFKEIMAPWAQTVVTGRARLGGIPVGVIAVETRTVEVAVPADPANLDSEAKIIQQAGQVWFPDSAYKTAQAIKDFNREKLPLMIFANWRGFSGGMKDMYDQVLKFGAYIVDGLRQYKQPILIYIPPYAELRGGSWVVIDATINPLCIEMYADKESRGGVLEPEGTVEIKFRKKDLIKSMRRIDPAYKKLMEQLGEPDLSDKDRKDLEGRLKAREDLLLPIYHQVAVQFADFHDTPGRMLEKGVISDILEWKTARTFLYWRLRRLLLEDQVKQEILQASGELSHVHIQSMLRRWFVETEGAVKAYLWDNNQVVVQWLEQHWITYLKHDSVLKTIRGLVEENPEVA 3tdh C 2.3 BS01 AMP C 1 T195 M199 K200 V220 S221 T309 S311 D312 T190 M194 K195 V215 S216 T304 S306 D307 ? 0004679,0005515,0005524,0005634,0005641,0005737,0005829,0005886,0006110,0006357,0006914,0007031,0016208,0019887,0019901,0030447,0031588,0042149,0042802,0043539,0043609,0045722,1904547,2000217 Kd=55uM remove_due_to_license_issue P12904 22019086 323 DSQEKVSIEQQLAVESIRKFLNSKTSYDVLPVSYRLIVLDTSLLVKKSLNVLLQNSIVSAPLWDSKTSRFAGLLTTTDFINVIQYYFSNPDKFELVDKLQLDGLKDIERALGVDQLDTASIHPSRPLFEACLKMLESRSGRIPLIDQDEETHREIVVSVLTQYRILKFVALNCRETHFLKIPIGDLNIITQDNMKSCQMTTPVIDVIQMLTQGRVSSVPIIDENGYLINVYEAYDVLGLIKGGIYNDLSLSVGEALMRRSDDFEGVYTCTKNDKLSTIMDNIRKARVHRFFVVDDVGRLVGVLTLSDILKYILLGS 3tdj A 1.95 BS02 3TJ B 1 P105 F106 M107 S108 P102 F103 M104 S105 ? 0015276,0016020 remove_due_to_license_issue P19491 21895609 400 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 3tdj A 1.95 BS03 3TJ B 2 P105 S108 S217 K218 G219 P102 S105 S214 K215 G216 ? 0015276,0016020 remove_due_to_license_issue P19491 21895609 265 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 3tdj B 1.95 BS01 3TJ B 1 P105 S108 S217 K218 G219 P104 S107 S216 K217 G218 ? 0015276,0016020 remove_due_to_license_issue P19491 21895609 400 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGEC 3tdj B 1.95 BS02 3TJ B 2 P105 F106 M107 S108 P104 F105 M106 S107 ? 0015276,0016020 remove_due_to_license_issue P19491 21895609 265 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGEC 3tf6 A 2.35 BS01 DBH A 1 Y106 F123 K125 Y132 F133 K134 Y104 F121 K123 Y130 F131 K132 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 remove_due_to_license_issue P80188 216 STSDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 3tfn A 2.07 BS01 2CJ A 1 M15 H18 S19 F22 F26 Y41 G138 L141 G161 L164 N168 R171 Y248 M15 H18 S19 F22 F26 Y41 G138 L141 G161 L164 N168 R171 Y248 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=0.27uM remove_due_to_license_issue A9JQL9 22290830 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 3tfp A 2.0 BS01 03L A 1 F22 Y41 R45 D48 V133 V137 A157 L160 G161 L164 F22 Y41 R45 D48 V133 V137 A157 L160 G161 L164 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 remove_due_to_license_issue A9JQL9 22290830 303 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 3tfu A 1.94 BS01 PL8 A 1 W64 G124 S125 Y157 H158 D254 I256 K283 W58 G118 S119 Y151 H152 D238 I240 K267 Y25 Y157 E220 D254 A257 K283 Y407 Y19 Y151 E204 D238 A241 K267 Y391 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 21988601 501 GLTPEQIIAVDGAHLWHPYSSIGREAVSPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLV 3tfu A 1.94 BS02 PL8 B 1 P317 T318 P301 T302 Y25 Y157 E220 D254 A257 K283 Y407 Y19 Y151 E204 D238 A241 K267 Y391 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 21988601 501 GLTPEQIIAVDGAHLWHPYSSIGREAVSPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLV 3tfu B 1.94 BS01 PL8 A 1 G93 P317 T318 G82 P296 T297 Y25 Y157 E220 D254 A257 K283 Y407 Y19 Y146 E199 D233 A236 K262 Y386 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 21988601 501 GLTPEQIIAVDGAHLWHPYSSISPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLV 3tfu B 1.94 BS02 PL8 B 1 G124 S125 Y157 H158 G159 D254 I256 K283 F402 G113 S114 Y146 H147 G148 D233 I235 K262 F381 Y25 Y157 E220 D254 A257 K283 Y407 Y19 Y146 E199 D233 A236 K262 Y386 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 21988601 501 GLTPEQIIAVDGAHLWHPYSSISPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLV 3tfv A 3.0 BS01 2CN A 1 F22 Y41 C44 R45 D48 D114 V133 A134 V137 L160 F22 Y41 C44 R45 D48 D114 V133 A134 V137 L160 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 remove_due_to_license_issue A9JQL9 22290830 289 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 3tge A 1.96 BS02 TGE A 1 A767 I768 Q775 V782 L804 M816 Q817 F820 A233 I234 Q241 V248 L270 M282 Q283 F286 3.1.4.35 0004114,0007165,0008081 ic50=0.07nM remove_due_to_license_issue IC50=0.070000nM O76074 21955943 999 ETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHPGVSNQFLINTNSELALMYNDESVLEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHEKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGDRERKELNIEPTDLMNREKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 3tgs A 2.7 BS01 03G A 1 V255 E370 F376 N377 F382 I424 N425 M426 W427 E429 V430 G473 M475 V139 E229 F235 N236 F241 I280 N281 M282 W283 E285 V286 G326 M328 ? 0019031 remove_due_to_license_issue C6G099 22451932 507 VWKEAKTTLFCASDAKAYEKEVHNVWATHACVPTDPNPQEMVLANVTENFNMWKNDMVEQMHEDIISLWDESLKPCVKLTGGSAITQACPKVSFDPIPLHYCAPAGFAILKCNNKTFNGTGPCRNVSTVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNESVNIVCTRPNNIRQAHCNINESKWNNTLQKVGEELAKHFPSKTIKFEPSSGGDLEITTHSFNCRGEFFYCNTSDLFNGTYRNGTYNHTGRSSNGTITLQCKIKQIINMWQEVGRAIYAPPIEGEITCNSNITGLLLLRDGGNDTETFRPGGGDMRDNWRSELYKYKVVEIK 3th0 A 1.75 BS01 RAM B 1 S237 E359 K363 Q366 W391 D395 S125 E247 K251 Q254 W279 D283 3.2.1.- remove_due_to_license_issue P12528 23292517 1 YSIEADKKFKYSVKLSDYPTLQDAASAAVDGLLIDRDYNFYGGETVDFGGKVLTIECKAKFIGDGNLIFTKLGKGSRIAGVFMESTTTPWVIKPWTDDNQWLTDAAAVVATLKQSKTDGYQPTVSDYVKFPGIETLLPPNAKGQNITSTLEIRECIGVEVHRASGLMAGFLFRGCHFCKMVDANNPSGGKDGIITFENLSGDWGKGNYVIGGRTSYGSVSSAQFLRNNGGFERDGGVIGFTSYRAGESGVKTWQGTVGSTTSRNYNLQFRDSVVIYPVWDGFDLGADTDMNPELDRPGDYPITQYPLHQLPLNHLIDNLLVRGALGVGFGMDGKGMYVSNITVEDCAGSGAYLLTHESVFTNIAIIDTNTKDFQANQIYISGACRVNGLRLIGIRSGQSLTIDAPNSTVSGITGMVDPSRINVANLAEEGLGNIRANSFGYDSAAIKLRIHKLSKTLDSGALYSHINGGAGSGSAYTQLTAISGSTPDAVSLKVNHKDCRGAEIPFVPDIASDDFIKDSSCFLPYWENNSTSLKALVKKPNGELVRLTLATL 3th0 A 1.75 BS02 MAN B 1 K363 Q366 K251 Q254 3.2.1.- remove_due_to_license_issue P12528 23292517 2 YSIEADKKFKYSVKLSDYPTLQDAASAAVDGLLIDRDYNFYGGETVDFGGKVLTIECKAKFIGDGNLIFTKLGKGSRIAGVFMESTTTPWVIKPWTDDNQWLTDAAAVVATLKQSKTDGYQPTVSDYVKFPGIETLLPPNAKGQNITSTLEIRECIGVEVHRASGLMAGFLFRGCHFCKMVDANNPSGGKDGIITFENLSGDWGKGNYVIGGRTSYGSVSSAQFLRNNGGFERDGGVIGFTSYRAGESGVKTWQGTVGSTTSRNYNLQFRDSVVIYPVWDGFDLGADTDMNPELDRPGDYPITQYPLHQLPLNHLIDNLLVRGALGVGFGMDGKGMYVSNITVEDCAGSGAYLLTHESVFTNIAIIDTNTKDFQANQIYISGACRVNGLRLIGIRSGQSLTIDAPNSTVSGITGMVDPSRINVANLAEEGLGNIRANSFGYDSAAIKLRIHKLSKTLDSGALYSHINGGAGSGSAYTQLTAISGSTPDAVSLKVNHKDCRGAEIPFVPDIASDDFIKDSSCFLPYWENNSTSLKALVKKPNGELVRLTLATL 3th0 A 1.75 BS03 GLA B 1 E359 W365 E247 W253 3.2.1.- remove_due_to_license_issue P12528 23292517 3 YSIEADKKFKYSVKLSDYPTLQDAASAAVDGLLIDRDYNFYGGETVDFGGKVLTIECKAKFIGDGNLIFTKLGKGSRIAGVFMESTTTPWVIKPWTDDNQWLTDAAAVVATLKQSKTDGYQPTVSDYVKFPGIETLLPPNAKGQNITSTLEIRECIGVEVHRASGLMAGFLFRGCHFCKMVDANNPSGGKDGIITFENLSGDWGKGNYVIGGRTSYGSVSSAQFLRNNGGFERDGGVIGFTSYRAGESGVKTWQGTVGSTTSRNYNLQFRDSVVIYPVWDGFDLGADTDMNPELDRPGDYPITQYPLHQLPLNHLIDNLLVRGALGVGFGMDGKGMYVSNITVEDCAGSGAYLLTHESVFTNIAIIDTNTKDFQANQIYISGACRVNGLRLIGIRSGQSLTIDAPNSTVSGITGMVDPSRINVANLAEEGLGNIRANSFGYDSAAIKLRIHKLSKTLDSGALYSHINGGAGSGSAYTQLTAISGSTPDAVSLKVNHKDCRGAEIPFVPDIASDDFIKDSSCFLPYWENNSTSLKALVKKPNGELVRLTLATL 3th8 B 2.114 BS01 TH9 B 1 D26 N28 G29 R39 H43 A47 A69 F70 I141 D13 N15 G16 R26 H30 A34 A56 F57 I113 D26 H43 L137 D13 H30 L109 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 22662288 289 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 3th9 A 1.34 BS01 9Y9 A 1 D25 A28 D29 D30 G48 I50 P81 V82 I84 D25 A28 D29 D30 G48 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P0C6F2 21916489 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3th9 A 1.34 BS02 9Y9 B 1 D25 G27 G49 I50 D25 G27 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P0C6F2 21916489 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3th9 B 1.34 BS01 9Y9 A 1 D25 G27 G48 G49 I50 D25 G27 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P0C6F2 21916489 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3th9 B 1.34 BS02 9Y9 B 1 D25 G27 A28 D29 D30 I50 P81 V82 I84 D25 G27 A28 D29 D30 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P0C6F2 21916489 100 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3thb A 2.5 BS02 3TA A 1 L59 G60 K61 C67 A80 L132 C133 R136 E140 F183 D194 L18 G19 K20 C26 A39 L91 C92 R95 E99 F142 D153 D176 K178 G180 N181 D194 T214 D135 K137 G139 N140 D153 T173 2.7.11.21 0004672,0005524,0006468 ic50=2nM remove_due_to_license_issue P53350 22070629 1 EVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 3thd A 1.79 BS01 DGJ A 1 Y83 C127 A128 E129 N187 E188 E268 Y333 Y55 C99 A100 E101 N159 E160 E240 Y305 3.2.1.23 0004553,0004565,0005515,0005576,0005615,0005737,0005764,0005773,0005794,0005975,0006516,0006689,0016020,0016787,0016798,0016936,0019388,0030200,0035578,0042340,0042803,0043202,0043231,0046479,0048471,0051413,0070062,1904016,1904813 remove_due_to_license_issue IC50=90000nM P16278 22128166 900 QRMFEIDYSRDSFLKDGQPFRYISGSIHYSRVPRFYWKDRLLKMKMAGLNAIQTYVPWNFHEPWPGQYQFSEDHDVEYFLRLAHELGLLVILRPGPYICAEWEMGGLPAWLLEKESILLRSSDPDYLAAVDKWLGVLLPKMKPLLYQNGGPVITVQVENEYGSYFACDFDYLRFLQKRFRHHLGDDVVLFTTDGAHKTFLKCGALQGLYTTVDFGTGSNITDAFLSQRKCEPKGPLINSEFYTGWLDHWGQPHSTIKTEAVASSLYDILARGASVNLYMFIGGTNFAYWNGANSPYAAQPTSYDYDAPLSEAGDLTEKYFALRNIIQKFEKVPEGPIPPSTPKFAYGKVTLEKLKTVGAALDILCPSGPIKSLYPLTFIQVKQHYGFVLYRTTLPQDCSNPAPLSSPLNGVHDRAYVAVDGIPQGVLERNNVITLNITGKAGATLDLLVENMGRVNYGAYINDFKGLVSNLTLSSNILTDWTIFPLDTEDAVRSHLGGWGHRNYTLPAFYMGNFSIPSGIPDLPQDTFIQFPGWTKGQVWINGFNLGRYWPARGPQLTLFVPQHILMTSAPNTITVLELEWAPCSSDDPELCAVTFVDRPVIGSS 3thw B 3.09 BS01 dna D 0 T221 P222 L223 G244 Y245 I263 Y264 H266 H269 S275 H279 H284 Q300 R313 S314 L316 F317 V738 S739 T765 K766 R770 T6 P7 L8 G29 Y30 I48 Y49 H51 H54 S60 H64 H69 Q85 R98 S99 L101 F102 V506 S507 T533 K534 R538 ? 0005524,0006298,0030983,0140664 remove_due_to_license_issue P20585 22179786 1 ~ 53 SKSIYTPLELQYIEMKQQHKDAVLCVECGYKYRFFGEDAEIAARELNIYCHLDHNFMTASIPTHRLFVHVRRLVAKGYKVGVVKQTETAALKAIGDNRSSLFSRKLTALYTKSTLIGEDVNPLIKLAVNVDEIMTDTSTSYLLCISENKENKKKGNIFIGIVGVQPATGEVVFDSFQDSASRSELETRMSSLQPVELLLPSALSEQTEALIHRATSVSVQDDRIRVERMDNIYFEYSHAFQAVTEFYAKGIVNLEKPVICSLAAIIKYLKEFNLEKMLSKPENFKQLSSKMEFMTINGTTLRNLEILQNQTDMKTKGSLLWVLDHTKTSFGRRKLKKWVTQPLLKLREINARLDAVSEVLHSESSVFGQIENHLRKLPDIERGLCSIYHKKCSTQEFFLIVKTLYHLKSEFQAIIPAVNSHIQSDLLRTVILEIPELLSPVEHYLKILNEQAAKVGDKTELFKDLSDFPLIKKRKDEIQGVIDEIRMHLQEIRKILKNPSAQYVTVSGQEFMIEIKNSAVSCIPTDWVKVGSTKAVSRFHSPFIVENYRHLNQLREQLVLDCSAEWLDFLEKFSEHYHSLCKAVHHLATVDCIFSLAKVAKQGDYCRPTVQEERKIVIKNGRHPVIDVLLGEQDQYVPNNTDLSEDSERVMIITGPNMGGKSSYIKQVALITIMAQIGSYVPAEEATIGIVDGIFTRMGAAGRSTFMEELTDTAEIIRKATSQSLVILDELGRGTSTHDGIAIAYATLEYFIRDVKSLTLFVTHYPPVCELEKNYSHQVGNYHMGFLVFVTFLYQITRGIAARSYGLNVAKLADVPGEILKKAAHKSKELEGLINTKRKRLKYFAKLWTMHNAQDLQKWT 3thx A 2.7 BS01 dna E 0 F42 T526 C527 F31 T492 C493 ? 0000287,0000400,0000781,0001701,0002204,0003677,0003682,0003684,0003690,0003697,0005515,0005524,0005634,0005654,0005694,0006119,0006281,0006298,0006301,0006302,0006312,0006974,0007281,0008094,0008340,0008584,0008630,0010165,0010224,0016020,0016446,0016447,0016887,0019237,0019724,0030183,0030983,0031573,0032137,0032139,0032142,0032143,0032181,0032301,0032302,0032357,0032405,0042771,0042803,0043524,0043531,0043570,0045190,0045910,0048298,0048304,0051096,0051726,0071168,0140664 remove_due_to_license_issue P43246 22179786 26 ~ 50 ESAAEVGFVRFFQGMPEKPTTTVRLFDRGDFYTAHGEDALLAAREVFKTQGVIKYMGPAGAKNLQSVVLSKMNFESFVKDLLLVRQYRVEVYKNRASKENDWYLAYKASPGNLSQFEDILFIGVVGVKMSAVDGQRQVGVGYVDSIQRKLGLCEFPDNDQFSNLEALLIQIGPKECVLPGGETAGDMGKLRQIIQRGGILITERKKADFSTKDIYQDLNRLLKGKKGEQMNSAVLPEMENQVAVSSLSAVIKFLELLSDDSNFGQFELTTFDFSQYMKLDIAAVRALNLFQQSLAALLNKCKTPQGQRLVNQWIKQPLMDKNRIEERLNLVEAFVEDAELRQTLQEDLLRRFPDLNRLAKKFQRQAANLQDCYRLYQGINQLPNVIQALEKHEGKHQKLLLAVFVTPLTDLRSDFSKFQEMIETTLDMDQVENHEFLVKPSFDPNLSELREIMNDLEKKMQSTLISAARDLGLDPGKQIKLDSSAGYYFRVTCKEEKVLRNNKNFSTVDIQGVKFTNSKLTSLNEEYTKNKTEYEEAQDAIVKEIVNISSGYVEPMQTLNDVLAQLDAVVSFAHVSNGAPVPYVRPAILEKGQGRIILKASRHACVEVQIAFIPNDVYFEKDKQMFHIITGPNMGGKSTYIRQTGVIVLMAQIGCFVPCESAEVSIVDCILARVGSTFMAEMLETASILRSATKDSLIIIDELGRGTSTYDGFGLAWAISEYIATKIGAFCMFATHFHELTALANQIPTVNNLHVTALTTEETLTMLYQVKKGVCDQSFGIHVAELANFPKHVIECAKQKALELEEFQYKCYLEREQGEKIIQEFLSKVKQMPFTEMSEENITIKLKQLKAEVIAKNNSFVNEIISRI 3thx B 2.7 BS01 dna D 0 T221 P222 L223 C243 G244 Y245 H269 Q300 L316 F317 R319 T5 P6 L7 C27 G28 Y29 H53 Q84 L100 F101 R103 ? 0005524,0006298,0030983,0140664 remove_due_to_license_issue P20585 22179786 3 ~ 23 KSIYTPLELQYIEMKQQHKDAVLCVECGYKYRFFGEDAEIAARELNIYCHLDHNFMTASIPTHRLFVHVRRLVAKGYKVGVVKQTETAALKAIGDNRSSLFSRKLTALYTKSTLIGEDVNPLIKLAVNVDEIMTDTSTSYLLCISENKNIFIGIVGVQPATGEVVFDSFQDSASRSELETRMSSLQPVELLLPSALSEQTEALIHRATSVSVQDDRIRVERMDNIYFEYSHAFQAVTEFYAIVNLEKPVICSLAAIIKYLKEFNLEKMLSKPENFKQLSSKMEFMTINGTTLRNLEILQNQTDMKTKGSLLWVLDHTKTSFGRRKLKKWVTQPLLKLREINARLDAVSEVLHSESSVFGQIENHLRKLPDIERGLCSIYHKKCSTQEFFLIVKTLYHLKSEFQAIIPAVNSHIQSDLLRTVILEIPELLSPVEHYLKILNEQAAKVGDKTELFKDLSDFPLIKKRKDEIQGVIDEIRMHLQEIRKILKNPSAQYVTVSGQEFMIEIKNSAVSCIPTDWVKVGSTKAVSRFHSPFIVENYRHLNQLREQLVLDCSAEWLDFLEKFSEHYHSLCKAVHHLATVDCIFSLAKVAKQGDYCRPTVQEERKIVIKNGRHPVIDVLLGEQDQYVPNNTDLSEDSERVMIITGPNMGGKSSYIKQVALITIMAQIGSYVPAEEATIGIVDGIFTRMSTFMEELTDTAEIIRKATSQSLVILDELGRGTSTHDGIAIAYATLEYFIRDVKSLTLFVTHYPPVCELEKNYSHQVGNYHMGFLVSVTFLYQITRGIAARSYGLNVAKLADVPGEILKKAAHKSKELEGLINTKRKRLKYFAKLWTMHNAQDLQKWTEEFNME 3thx B 2.7 BS02 dna E 0 Y245 K246 I263 Y264 S275 P277 R280 H284 S314 S739 T765 K766 R770 Y29 K30 I47 Y48 S59 P61 R64 H68 S98 S498 T524 K525 R529 ? 0005524,0006298,0030983,0140664 remove_due_to_license_issue P20585 22179786 26 ~ 50 KSIYTPLELQYIEMKQQHKDAVLCVECGYKYRFFGEDAEIAARELNIYCHLDHNFMTASIPTHRLFVHVRRLVAKGYKVGVVKQTETAALKAIGDNRSSLFSRKLTALYTKSTLIGEDVNPLIKLAVNVDEIMTDTSTSYLLCISENKNIFIGIVGVQPATGEVVFDSFQDSASRSELETRMSSLQPVELLLPSALSEQTEALIHRATSVSVQDDRIRVERMDNIYFEYSHAFQAVTEFYAIVNLEKPVICSLAAIIKYLKEFNLEKMLSKPENFKQLSSKMEFMTINGTTLRNLEILQNQTDMKTKGSLLWVLDHTKTSFGRRKLKKWVTQPLLKLREINARLDAVSEVLHSESSVFGQIENHLRKLPDIERGLCSIYHKKCSTQEFFLIVKTLYHLKSEFQAIIPAVNSHIQSDLLRTVILEIPELLSPVEHYLKILNEQAAKVGDKTELFKDLSDFPLIKKRKDEIQGVIDEIRMHLQEIRKILKNPSAQYVTVSGQEFMIEIKNSAVSCIPTDWVKVGSTKAVSRFHSPFIVENYRHLNQLREQLVLDCSAEWLDFLEKFSEHYHSLCKAVHHLATVDCIFSLAKVAKQGDYCRPTVQEERKIVIKNGRHPVIDVLLGEQDQYVPNNTDLSEDSERVMIITGPNMGGKSSYIKQVALITIMAQIGSYVPAEEATIGIVDGIFTRMSTFMEELTDTAEIIRKATSQSLVILDELGRGTSTHDGIAIAYATLEYFIRDVKSLTLFVTHYPPVCELEKNYSHQVGNYHMGFLVSVTFLYQITRGIAARSYGLNVAKLADVPGEILKKAAHKSKELEGLINTKRKRLKYFAKLWTMHNAQDLQKWTEEFNME 3thz B 4.3 BS01 dna D 0 S216 T221 L223 C243 G244 Y245 L316 F317 S750 S1 T6 L8 C28 G29 Y30 L101 F102 S504 ? 0005524,0006298,0030983,0140664 remove_due_to_license_issue P20585 22179786 4 ~ 23 SKSIYTPLELQYIEMKQQHKDAVLCVECGYKYRFFGEDAEIAARELNIYCHLDHNFMTASIPTHRLFVHVRRLVAKGYKVGVVKQTETAALKAIGDNRSSLFSRKLTALYTKSTLIGEDVNPTDTSTSYLLCISENKKKKGNIFIGIVGVQPATGEVVFDSFQDSASRSELETRMSSLQPVELLLPSALSEQTEALIHRATSVSVQDDRIRVERMDNIYFEYSHAFQAVTEFYAKGIVNLEKPVICSLAAIIKYLKEFNLEKMLSKPENFKQLSSKMEFMTINGTTLRNLEILQNQTDMKTKGSLLWVLDHTKTSFGRRKLKKWVTQPLLKLREINARLDAVSEVLHSESSVFGQIENHLRKLPDIERGLCSIYHKKCSTQEFFLIVKTLYHLKSEFQAIIPAVNSHIQSDLLRTVILEIPELLSPVEHYLKILNEQAAKVGDKTELFKDLSDFPLIKKRKDEIQGVIDEIRMHLQEIRKILKNPSAQYVTVSGQEFMIEIKNSAVSCIPTDWVKVGSTKAVSRFHSPFIVENYRHLNQLREQLVLDCSAEWLDFLEKFSEHYHSLCKAVHHLATVDCIFSLAKVAKQGDYCRPTVQEERKIVIKNGRHPVIDVLLGEQDQYVPNNTDLSEDSERVMIITGPNMGGKSSYIKQVALITIMAQIGSYVPAEEATIGIVDGIFTRMGAAGRSTFMEELTDTAEIIRKATSQSLVILDELGRGTSTHDGIAIAYATLEYFIRDVKSLTLFVTHYPPVCELEKNYSHQVGNYHMGFLVFVTFLYQITRGIAARSYGLNVAKLADVPGEILKKAAHKSKELEGLINTKRKRLKYFAKLWTMHNAQDLQKWT 3thz B 4.3 BS02 dna E 0 Y245 I263 Y264 S275 P277 R280 H284 S314 T737 V738 S739 T765 K766 R770 Y30 I48 Y49 S60 P62 R65 H69 S99 T491 V492 S493 T519 K520 R524 ? 0005524,0006298,0030983,0140664 remove_due_to_license_issue P20585 22179786 27 ~ 53 SKSIYTPLELQYIEMKQQHKDAVLCVECGYKYRFFGEDAEIAARELNIYCHLDHNFMTASIPTHRLFVHVRRLVAKGYKVGVVKQTETAALKAIGDNRSSLFSRKLTALYTKSTLIGEDVNPTDTSTSYLLCISENKKKKGNIFIGIVGVQPATGEVVFDSFQDSASRSELETRMSSLQPVELLLPSALSEQTEALIHRATSVSVQDDRIRVERMDNIYFEYSHAFQAVTEFYAKGIVNLEKPVICSLAAIIKYLKEFNLEKMLSKPENFKQLSSKMEFMTINGTTLRNLEILQNQTDMKTKGSLLWVLDHTKTSFGRRKLKKWVTQPLLKLREINARLDAVSEVLHSESSVFGQIENHLRKLPDIERGLCSIYHKKCSTQEFFLIVKTLYHLKSEFQAIIPAVNSHIQSDLLRTVILEIPELLSPVEHYLKILNEQAAKVGDKTELFKDLSDFPLIKKRKDEIQGVIDEIRMHLQEIRKILKNPSAQYVTVSGQEFMIEIKNSAVSCIPTDWVKVGSTKAVSRFHSPFIVENYRHLNQLREQLVLDCSAEWLDFLEKFSEHYHSLCKAVHHLATVDCIFSLAKVAKQGDYCRPTVQEERKIVIKNGRHPVIDVLLGEQDQYVPNNTDLSEDSERVMIITGPNMGGKSSYIKQVALITIMAQIGSYVPAEEATIGIVDGIFTRMGAAGRSTFMEELTDTAEIIRKATSQSLVILDELGRGTSTHDGIAIAYATLEYFIRDVKSLTLFVTHYPPVCELEKNYSHQVGNYHMGFLVFVTFLYQITRGIAARSYGLNVAKLADVPGEILKKAAHKSKELEGLINTKRKRLKYFAKLWTMHNAQDLQKWT 3ti1 A 1.99 BS01 B49 A 1 I10 A31 F80 F82 L83 H84 D86 K88 L134 D145 I10 A31 F76 F78 L79 H80 D82 K84 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue Kd=>10000nM, IC50=1.30e+5nM P24941 22893598 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3ti3 A 1.8 BS03 LNV A 1 R118 E119 D151 R152 W178 E227 S246 E276 R292 R371 Y406 R37 E38 D70 R71 W98 E147 S166 E196 R212 R287 Y321 D151 E277 R292 R371 Y406 D70 E197 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=1.83nM remove_due_to_license_issue C3W5S3 22028647 801 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 3ti4 A 1.602 BS03 LVO A 1 R118 E119 D151 R152 W178 E227 S246 R292 N294 R371 Y406 R37 E38 D70 R71 W98 E147 S166 R212 N214 R287 Y321 D151 E277 R292 R371 Y406 D70 E197 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=947nM remove_due_to_license_issue C3W5S3 22028647 801 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 3ti5 A 1.9 BS03 ZMR A 1 R118 E119 D151 R152 W178 S246 E276 R292 R371 Y406 R37 E38 D70 R71 W98 S166 E196 R212 R287 Y321 D151 E277 R292 R371 Y406 D70 E197 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=1.11nM remove_due_to_license_issue C3W5S3 22028647 1002 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 3ti6 A 1.69 BS03 G39 A 1 R118 E119 D151 R152 W178 R224 E276 R292 N294 R371 Y406 R37 E38 D70 R71 W98 R144 E196 R212 N214 R287 Y321 D151 E277 R292 R371 Y406 D70 E197 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.54nM remove_due_to_license_issue C3W5S3 22028647 801 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 3ti8 A 1.601 BS02 LNV A 1 R118 E119 D151 R152 W178 E227 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W98 E147 A166 E196 R212 R292 Y326 D151 E277 R292 R371 Y406 D70 E197 R212 R292 Y326 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.9nM remove_due_to_license_issue A1ILL9 22028647 901 PEFLNNTEPLCNVSGFAIVSKDNGIRIGSRGHVFVIREPFVACGPTECRTFFLTQGALLNDKHSNNTVKDRSPYRALMSVPLGSSPNAYQAKFESVAWSATACHDGKKWLAVGISGADDDAYAVIHYGGMPTDVVRSWRKQILRTQESSCVCMNGNCYWVMTDGPANSQASYKIFKSHEGMVTNEREVSFQGGHIEECSCYPNLGKVECVCRDNWNGMNRPILIFDEDLDYEVGYLCAGIPTDTPRVQDSSFTGSCTNAVGGSGTNNYGVKGFGFRQGNSVWAGRTVSISSRSGFEILLIEDGWIRTSKTIVKKVEVLNNKNWSGYSGAFTIPITMTSKQCLVPCFWLEMIRGKPEERTSIWTSSSSTVFCGVSSEVPGWSWDDGAILPFDIDK 3tia A 1.8 BS04 LNV A 1 R118 E119 D151 R152 W178 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W97 A165 E195 R211 R290 Y325 D151 E277 R292 R371 Y406 D70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 ic50=3.12nM remove_due_to_license_issue IC50=3100nM Q194T1 22028647 801 VEYRNWSKPQCQITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPGKCYQFALGQGTTLDNKHSNDTVHDRIPHRTLLMNELGVPFHLGTRQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYDGRLVDSIGSWSQNILRTQESECVCINGTCTVVMTDGSASGRADTRILFIEEGKIVHISPLSGSAQHIEECSCYPRYPGVRCICRDNWKGSNRPVVDINMEDYSIDSSYVCSGLVGDTPRNDDSSSNSNCRNPNNERGTQGVKGWAFDNGNDLWMGRTISKESRSGYETFKVIGGWSTPNSKSQVNRQVIVDNNNWSGYSGIFSVEGKSCINRCFYVELIRGRPQETRVWWTSNSIVVFCGTSGTYGTGSWPDGANINFMPI 3tib A 2.201 BS04 LVO A 1 R118 E119 D151 R152 W178 I222 R224 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W97 I141 R143 A165 E195 R211 R290 Y325 D151 E277 R292 R371 Y406 D70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 ic50=129nM remove_due_to_license_issue Q194T1 22028647 801 VEYRNWSKPQCQITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPGKCYQFALGQGTTLDNKHSNDTVHDRIPHRTLLMNELGVPFHLGTRQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYDGRLVDSIGSWSQNILRTQESECVCINGTCTVVMTDGSASGRADTRILFIEEGKIVHISPLSGSAQHIEECSCYPRYPGVRCICRDNWKGSNRPVVDINMEDYSIDSSYVCSGLVGDTPRNDDSSSNSNCRNPNNERGTQGVKGWAFDNGNDLWMGRTISKESRSGYETFKVIGGWSTPNSKSQVNRQVIVDNNNWSGYSGIFSVEGKSCINRCFYVELIRGRPQETRVWWTSNSIVVFCGTSGTYGTGSWPDGANINFMPI 3tic A 1.89 BS04 ZMR A 1 R118 E119 D151 R152 W178 E227 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W97 E146 A165 E195 R211 R290 Y325 D151 E277 R292 R371 Y406 D70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 ic50=1.36nM remove_due_to_license_issue IC50=1400nM Q194T1 22028647 1002 VEYRNWSKPQCQITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPGKCYQFALGQGTTLDNKHSNDTVHDRIPHRTLLMNELGVPFHLGTRQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYDGRLVDSIGSWSQNILRTQESECVCINGTCTVVMTDGSASGRADTRILFIEEGKIVHISPLSGSAQHIEECSCYPRYPGVRCICRDNWKGSNRPVVDINMEDYSIDSSYVCSGLVGDTPRNDDSSSNSNCRNPNNERGTQGVKGWAFDNGNDLWMGRTISKESRSGYETFKVIGGWSTPNSKSQVNRQVIVDNNNWSGYSGIFSVEGKSCINRCFYVELIRGRPQETRVWWTSNSIVVFCGTSGTYGTGSWPDGANINFMPI 3tif A 1.7995 BS01 ADP A 1 Y11 G41 S42 G43 K44 S45 T46 Y11 G41 S42 G43 K44 S45 T46 ? 0005524,0005886,0016887,0022857,0055085 remove_due_to_license_issue Q58206 22158619 236 MVKLKNVTKTYKMGEEIIYALKNVNLNIKEGEFVSIMGPSGSGKSTMLNIIGCLDKPTEGEVYIDNIKTNDLDDDELTKIRRDKIGFVFQQFNLIPLLTALENVELPLIFKYRGAMSGEERRKRALECLKMAELEERFANHKPNQLSGGQQQRVAIARALANNPPIILADQPTWALDSKTGEKIMQLLKKLNEEDGKTVVVVTHDINVARFGERIIYLKDGEVEREEKLR 3tif A 1.7995 BS02 ADP B 1 Q145 S147 Q145 S147 ? 0005524,0005886,0016887,0022857,0055085 remove_due_to_license_issue Q58206 22158619 1 MVKLKNVTKTYKMGEEIIYALKNVNLNIKEGEFVSIMGPSGSGKSTMLNIIGCLDKPTEGEVYIDNIKTNDLDDDELTKIRRDKIGFVFQQFNLIPLLTALENVELPLIFKYRGAMSGEERRKRALECLKMAELEERFANHKPNQLSGGQQQRVAIARALANNPPIILADQPTWALDSKTGEKIMQLLKKLNEEDGKTVVVVTHDINVARFGERIIYLKDGEVEREEKLR 3tif B 1.7995 BS01 ADP A 1 F1138 Q1145 S1147 Q1150 F138 Q145 S147 Q150 ? 0005524,0005886,0016887,0022857,0055085 remove_due_to_license_issue Q58206 22158619 236 MVKLKNVTKTYKMGEEIIYALKNVNLNIKEGEFVSIMGPSGSGKSTMLNIIGCLDKPTEGEVYIDNIKTNDLDDDELTKIRRDKIGFVFQQFNLIPLLTALENVELPLIFKYRGAMSGEERRKRALECLKMAELEERFANHKPNQLSGGQQQRVAIARALANNPPIILADQPTWALDSKTGEKIMQLLKKLNEEDGKTVVVVTHDINVARFGERIIYLKDGEVEREEKLRGF 3tif B 1.7995 BS02 ADP B 1 Y1011 G1041 G1043 K1044 S1045 T1046 Y11 G41 G43 K44 S45 T46 ? 0005524,0005886,0016887,0022857,0055085 remove_due_to_license_issue Q58206 22158619 1 MVKLKNVTKTYKMGEEIIYALKNVNLNIKEGEFVSIMGPSGSGKSTMLNIIGCLDKPTEGEVYIDNIKTNDLDDDELTKIRRDKIGFVFQQFNLIPLLTALENVELPLIFKYRGAMSGEERRKRALECLKMAELEERFANHKPNQLSGGQQQRVAIARALANNPPIILADQPTWALDSKTGEKIMQLLKKLNEEDGKTVVVVTHDINVARFGERIIYLKDGEVEREEKLRGF 3tiy A 1.84 BS01 TIY A 1 V18 A31 K33 F80 E81 L83 L134 D145 V17 A30 K32 F75 E76 L78 L129 D140 D127 K129 Q131 N132 D145 T158 T165 D122 K124 Q126 N127 D140 T153 T160 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=1.7e+4nM P24941 22893598 311 ENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3tiz A 2.02 BS01 3TI A 1 I10 A31 F82 L83 H84 K89 L134 A144 D145 I9 A30 F77 L78 H79 K84 L129 A139 D140 D127 K129 Q131 N132 D145 T158 T165 D122 K124 Q126 N127 D140 T153 T160 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=>1.50e+5nM P24941 22893598 299 ENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3tjc A 2.4 BS01 0TP A 1 L855 G856 Y931 L932 G935 N981 L983 D994 L13 G14 Y85 L86 G89 N135 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.031uM remove_due_to_license_issue IC50=3940nM O60674 22087750 1 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 3tjd A 2.9 BS01 6TP A 1 L855 K857 G861 A880 Y931 L932 G935 L983 D994 L13 K15 G19 A38 Y85 L86 G89 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1nM O60674 22087750 1 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 3tjm A 1.48 BS01 7FA A 1 P2249 I2250 S2308 Y2309 Y2347 Y2351 E2366 F2370 L2427 R2428 E2431 P32 I33 S91 Y92 Y130 Y134 E149 F153 L210 R211 E214 1.1.1.100,1.3.1.39,2.3.1.38,2.3.1.39,2.3.1.41,2.3.1.85,3.1.2.14,4.2.1.59 0009058 remove_due_to_license_issue P49327 21908709 500 NLRSLLVNPEGPTLMRLNSVQSSERPLFLVHPIEGSTTVFHSLASRLSIPTYGLQCTRAAPLDSIHSLAAYYIDCIRQVQPEGPYRVAGYSYGACVAFEMCSQLQAQQSPAPTHNSLFLFDGSPTYVLAYTGSYRAKLTPGCEAEAETEAICFFVQQFTDMEHNRVLEALLPLKGLEERVAAAVDLIIKSHQGLDRQELSFAARSFYYKLRAAEQYTPKAKYHGNVMLLRAAAGADYNLSQVCDGKVSVHVIEGDHATLLEGSGLESIISIIHSS 3tk2 A 1.35 BS01 PHE A 1 A158 Y159 K165 L175 T254 P256 F258 A152 Y153 K159 L169 T248 P250 F252 H138 H143 E184 S203 H132 H137 E178 S197 1.14.16.1 0004497,0004505,0005506,0006559,0009072,0016714,0019293,0046872 remove_due_to_license_issue P30967 23860686 298 FVVPDITTRKNVGLSHDANDFTLPQPLDRYSAEDHATWATLYQRQCKLLPGRACDEFMEGLERLEVDADRVPDFNKLNQKLMAATGWKIVAVPGLIPDDVFFEHLANRRFPVTWWLREPHQLDYLQEPDVFHDLFGHVPLLINPVFADYLEAYGKGGVKAKALGALPMLARLYWYTVEFGLINTPAGMRIYGAGILSSKSESIYCLDSASPNRVGFDLMRIMNTRYRIDTFQKTYFVIDSFKQLFDATAPDFAPLYLQLADAQPWGAGDVAPDDLVL 3tkh A 1.79 BS01 07S A 1 L15 V23 A36 Y86 C87 S88 G90 L137 L14 V22 A35 Y75 C76 S77 G79 L126 D130 K132 E134 N135 D148 T170 D119 K121 E123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=47nM remove_due_to_license_issue O14757 22374217 325 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 3tki A 1.6 BS01 S25 A 1 Q13 L15 Y20 A36 K38 Y86 C87 G90 L137 D148 Q12 L14 Y19 A35 K37 Y78 C79 G82 L129 D140 D130 K132 E134 N135 D148 T170 D122 K124 E126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.05nM remove_due_to_license_issue O14757 22374217 325 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 3tkm A 1.953 BS01 GW0 A 1 F246 R248 C249 T253 H287 V305 V312 I327 H413 L433 Y437 F75 R77 C78 T82 H116 V134 V141 I156 H242 L262 Y266 ? 0003677,0004879,0005634,0006355 Kd=22nM remove_due_to_license_issue EC50=13nM, Kd=0.400000nM Q03181 22606221 1 GSHMQVADLKAFSKHIYNAYLKNFNMTKKKARSILTGKASHTAPFVIHDIETLWQAEKGLVWGLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKDMY 3tku A 2.15 BS01 M77 A 1 I82 G83 V90 A103 Y155 D204 N205 L207 F370 I81 G82 V89 A102 Y154 D203 N204 L206 F369 D200 K202 N205 D218 T239 D199 K201 N204 D217 T238 2.7.11.1 0004672,0004674,0005524,0006468 ic50=1.92uM remove_due_to_license_issue Q9Y5S2 21949762 418 SAKVRLKKLEQLLLDGPWRNESALSVETLLDVLVCLYTECSHSALRRDKYVAEFLEWAKPFTQLVKEMQLHREDFEIIKVIGRGAFGEVAVVKMKNTERIYAMKILNKWEMLKRAETACFREERDVLVNGDCQWITALHYAFQDENHLYLVMDYYVGGDLLTLLSKFEDKLPEDMARFYIGEMVLAIDSIHQLHYVHRDIKPDNVLLDVNGHIRLADFGSCLKMNDDGTVQSSVAVGTPDYISPEILQAMEDGMGKYGPECDWWSLGVCMYEMLYGETPFYAESLVETYGKIMNHEERFQFPSHVTDVSEEAKDLIQRLICSRERRLGQNGIEDFKKHAFFEGLNWENIRNLEAPYIPDVSSPSDTSNFDVSGLHLPFIGFTFTTESCFSDRGSL 3tkw A 1.55 BS01 017 B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 22242794 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3tkw B 1.55 BS01 017 B 1 D25 G27 A28 D30 V82 I84 D29 G31 A32 D34 V86 I88 D25 T26 G27 D29 T30 G31 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 22242794 401 SFNFPQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3tl5 A 2.788 BS01 980 A 1 K802 M804 I831 I879 I881 V882 M953 F961 I963 D964 K569 M571 I598 I646 I648 V649 M720 F728 I730 D731 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=36nM, Kd=2.6nM P48736 21981714 1 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNYCHPIALPRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 3tlh A 2.0 BS01 3TL A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.5nM remove_due_to_license_issue P03366 10651036 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 3tll A 1.37 BS02 62D A 1 S103 Y106 M153 D156 C158 I201 G229 G230 L231 A232 M260 G261 S93 Y96 M137 D140 C142 I185 G213 G214 L215 A216 M244 G245 D102 D280 C318 C320 C323 H349 D92 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=40830nM remove_due_to_license_issue P28720 22736391 501 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSTKQSEEGVTFKSHRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYF 3tmk A 2.0 BS01 T5A A 1 D14 R15 G17 K18 T19 T20 K37 F38 P39 R41 L53 F69 R73 R94 G99 Y102 E142 K143 S144 Y151 G188 I189 D14 R15 G17 K18 T19 T20 K37 F38 P39 R41 L53 F69 R73 R94 G99 Y102 E142 K143 S144 Y151 G188 I189 2.7.4.9 0004550,0004798,0005515,0005524,0005634,0005737,0006227,0006233,0006235,0009041,0009165,0016301,0046940 Kd=135nM remove_due_to_license_issue P00572 9521686 217 MMGRGKLILIEGLDRTGKTTQCNILYKKLQPNCKLLKFPERSTRIGGLINEYLTDDSFQLSDQAIHLLFSANRWEIVDKIKKDLLEGKNIVMDRYVYSGVAYSAAKGTNGMDLDWCLQPDVGLLKPDLTLFLSTQDVDNNAEKSGFGDERYETVKFQEKVKQTFMKLLDKEIRKGDESITIVDVTNKGIQEVEALIWQIVEPVLSTHIDHDKFSFF 3tmm A 2.5001 BS01 dna B 0 S13 S14 Y15 L16 S19 T36 I39 R40 A43 W46 R47 Y61 W65 R98 M101 K105 K114 R115 R117 N121 V124 A125 F128 P136 L140 S13 S14 Y15 L16 S19 T36 I39 R40 A43 W46 R47 Y61 W65 R98 M101 K105 K114 R115 R117 N121 V124 A125 F128 P136 L140 ? remove_due_to_license_issue Q00059 22037171 1 ~ 28 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKK 3tmm A 2.5001 BS02 dna C 0 K9 L16 T35 H95 R98 M101 K105 T108 R115 Y120 Q137 L140 K144 Y169 R190 R191 T192 K9 L16 T35 H95 R98 M101 K105 T108 R115 Y120 Q137 L140 K144 Y169 R190 R191 T192 ? remove_due_to_license_issue Q00059 22037171 1 ~ 28 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKK 3tn8 A 2.95 BS01 F18 A 1 A46 E66 F103 C106 L156 D167 A39 E59 F87 C90 L140 D151 D149 K151 A153 N154 D167 T191 D133 K135 A137 N138 D151 T171 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=3.5e+2nM P50750 22292676 332 VECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLQPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLK 3tne A 2.4 BS01 RIT A 1 D32 G34 Y78 G79 D80 S82 V113 N125 D220 G222 T223 T224 Y227 I303 D32 G34 Y78 G79 D80 S82 V113 N125 D220 G222 T223 T224 Y227 I303 D32 S35 D37 W39 Y78 D220 T223 D32 S35 D37 W39 Y78 D220 T223 3.4.23.24 0004190,0005576,0006508 remove_due_to_license_issue P32951 22146051 401 DSISLSLINEGPSYASKVSVGSNKQQQTVIIDTGSSDFWVVDSNAQCGKGVDCKSSGTFTPSSSSSYKNLGAAFTIRYGDGSTSQGTWGKDTVTINGVSITGQQIADVTQTSVDQGILGIGYTSNEAVYDTSGRQTTPNYDNVPVTLKKQGKIRTNAYSLYLNSPSAETGTIIFGGVDNAKYSGKLVAEQVTSSQALTISLASVNLKGSSFSFGDGALLDSGTTLTYFPSDFAAQLADKAGARLVQVARDQYLYFIDCNTDTSGTTVFNFGNGAKITVPNTEYVYQNGDGTCLWGIQPSDDTILGDNFLRHAYLLYNLDANTISIAQVKYTTDSSISAV 3tnh A 3.202 BS01 F18 A 1 A46 E66 F103 C106 L156 D167 A39 E59 F86 C89 L139 D150 D149 K151 A153 N154 D167 T191 D132 K134 A136 N137 D150 T167 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=3.5e+2nM P50750 22292676 400 VECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKGML 3tpp A 1.6 BS01 5HA A 1 G11 Q12 G13 L30 D32 G34 Y71 T72 Q73 F108 W115 I118 I226 D228 G230 T231 T232 N233 R235 G16 Q17 G18 L35 D37 G39 Y76 T77 Q78 F113 W120 I123 I219 D221 G223 T224 T225 N226 R228 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=15nM remove_due_to_license_issue IC50=15nM, EC50=43nM, Ki=233nM P56817 22194329 999 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVETSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3tpr A 2.55 BS01 5HA A 1 G11 G13 D32 G34 F108 I118 D228 G230 T232 N233 R235 N385 G13 G15 D34 G36 F110 I120 D218 G220 T222 N223 R225 N368 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D218 T221 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=15nM, EC50=43nM, Ki=233nM P56817 22194329 400 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3ts4 A 1.587 BS06 EEG A 1 I180 L181 A182 H183 L214 H218 E219 H222 H228 K233 A234 P238 T239 Y240 I76 L77 A78 H79 L110 H114 E115 H118 H124 K129 A130 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=1.9nM remove_due_to_license_issue Ki=1.92nM P39900 22689580 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3tsd A 2.653 BS01 XMP A 1 M51 G305 S306 I307 C308 D341 G364 S365 Y388 G390 M55 G308 S309 I310 C311 D344 G367 S368 Y385 G387 1.1.1.205 0000166,0003824,0003938,0006164,0006177,0006183,0016491,0046872 remove_due_to_license_issue A0A6L8P2U9 22788966 500 QSNAMWESKFVKEGLTFDDVLLVPAKSDVLPREVSVKTVLSESLQLNIPLISAGMDTVTEADMAIAMARQGGLGIIHKNMSIEQQAEQVDKVKRSESGVISDPFFLTPEHQVYDAEHLMGKYRISGVPVVNNLDERKLVGIITNRDMRFIQDYSIKISDVMKEQLITAPVGTTLSEAEKILQKYKIEKLPLVDNNGVLQGLITIKDIEKVIEFPNSAKDKQGRLLVGAAVGVTADAMTRIDALVKASVDAIVLDTAHGHSQGVIDKVKEVRAKYPSLNIIAGNVATAEATKALIEAGANVVKVGIGPGSICTTRVVAGVGVPQLTAVYDCATEARKHGIPVIADGGIKYSGDMVKALAAGAHVVMLGSMFAGVAESPGERQFKVYRGEGRVPYKGPLADTVHQLVGGLRAGMGYCGAQDLEFLRENAQFIRMSGAGLLESHP 3tsk A 2.0 BS06 QEG A 1 G179 I180 H218 K233 P238 T239 Y240 K241 V243 G75 I76 H114 K129 P134 T135 Y136 K137 V139 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=317nM P39900 22689580 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3tt0 A 2.8 BS01 07J A 1 V492 A512 K514 E531 M535 I545 V561 Y563 A564 G567 L630 A640 D641 V32 A52 K54 E71 M75 I85 V101 Y103 A104 G107 L170 A180 D181 T521 L525 L528 G567 R576 S588 Q606 D623 A625 R627 N628 V629 D641 G697 T61 L65 L68 G107 R116 S128 Q146 D163 A165 R167 N168 V169 D181 G237 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue IC50=1.0nM P11362 21936542 1 SEYELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 3tt4 A 1.88 BS05 E1S A 1 I159 L160 A161 H197 E198 H201 H207 L214 Y216 P217 N218 Y219 A220 R222 I76 L77 A78 H114 E115 H118 H124 L131 Y133 P134 N135 Y136 A137 R139 H197 E198 H201 H207 H114 E115 H118 H124 3.4.24.34 0004222,0006508,0008237,0008270,0031012 Ki=5.3nM remove_due_to_license_issue Ki=5.3nM P22894 22689580 1 GNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3tti A 2.2 BS01 KBI A 1 I70 V78 A91 K93 I124 M146 M149 A151 Q155 L206 I25 V33 A46 K48 I79 M101 M104 A106 Q110 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T176 2.7.11.24 0000165,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0005886,0006468,0007165,0007254,0009416,0016020,0033554,0038095,0042752,0048511,0090398,0106310 ic50=0.006uM remove_due_to_license_issue IC50=6.0nM P53779 22244937 465 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPREHTIEEWKELIYKEVMN 3ttj A 2.1 BS01 JBI A 1 V78 A91 K93 I124 M146 M149 A151 N152 Q155 V196 L206 V31 A44 K46 I77 M99 M102 A104 N105 Q108 V149 L159 D189 K191 N194 D207 T226 D142 K144 N147 D160 T170 2.7.11.24 0000165,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0005886,0006468,0007165,0007254,0009416,0016020,0033554,0038095,0042752,0048511,0090398,0106310 ic50=0.21uM remove_due_to_license_issue IC50=210nM P53779 22226655 465 NQFYSVEVSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPEHTIEEWKELIYKEVMN 3ttm A 2.0 BS01 PUT A 1 W35 S36 D37 Y38 Y241 D244 F273 D275 F311 W10 S11 D12 Y13 Y216 D219 F248 D250 F286 ? 0015846,0019808,0019810,0042597 Kd=3nM remove_due_to_license_issue Q9I6J1 22300763 367 DNKVLHVYNWSDYIAPDTLEKFTKETGIKVVYDVYDSNEVLEAKLLAGKSGYDVVVPSNSFLAKQIKAGVYQKLDKSKLPNWKNLNKDLMHTLEVSDPGNEHAIPYMWGTIGIGYNPDKVKAAFGDNAPVDSWDLVFKPENIQKLKQCGVSFLDSPTEILPAALHYLGYKPDTDNPKELKAAEELFLKIRPYVTYFHSSKYISDLANGNICVAIGYSGDIYQAKSRAEEAKNKVTVKYNIPKEGAGSFFDMVAIPKDAENTEGALAFVNFLMKPEIMAEITDVVQFPNGNAAATPLVSEAIRNDPGIYPSEEVMKKLYTFPDLPAKTQRAMTRSWTKIKSG 3ttn A 2.0 BS01 SPD A 1 W34 T35 Y37 S82 E181 Y239 D242 W271 D273 W7 T8 Y10 S55 E154 Y212 D215 W244 D246 ? 0005615,0015846,0019808,0019809,0042597 Kd=14.3nM remove_due_to_license_issue Q9I6J0 22300763 363 SLHIYNWTDYIAPTTLKDFTKESGIDVSYDVFDSNETLEGKLVSGHSGYDIVVPSNNFLGKQIQAGAFQKLDKSKLPNWKNLDPALLKQLEVSDPGNQYAVPYLWGTNGIGYNVAKVKEVLGDQPIDSWAILFEPENMKKLAKCGVAFMDSGDEMLPAALNYLGLDPNTHDPKDYKKAEEVLTKVRPYVSYFHSSKYISDLANGNICVAFGYSGDVFQAAARAEEAGKGIDIQYVIPKEGANLWFDLMAIPADAKAADNAYAFIDYLLRPEVIAKVSDYVGYANAIPGARPLMDKSVSDSEEVYPPQAVLDKLYVSAVLPAKVLRLQTRTWTRIK 3ttp A 2.23 BS01 017 A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 24785545 201 PQITLWQRPLVTVKIGGQLREALLDTGADDTIFEDINLPGKWTPKMVGGIGGFMKVRQYDQVVIEICGHKVTSPVLVGPTPLNIIGRNVLTQLGCTLNF 3ttp B 2.23 BS01 017 A 1 D25 G27 A28 D30 G48 P81 I84 D25 G27 A28 D30 G48 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 24785545 201 PQITLWQRPLVTVKIGGQLREALLDTGADDTIFEDINLPGKWTPKMVGGIGGFMKVRQYDQVVIEICGHKVTSPVLVGPTPLNIIGRNVLTQLGCTLNF 3ttz A 1.63 BS01 07N A 1 N54 E58 D81 R84 G85 I86 P87 R144 T173 N41 E45 D68 R71 G72 I73 P74 R108 T137 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.004uM remove_due_to_license_issue IC50=4nM P0A0K8 22041057 1 YGAGQIQVLEGLEAVRKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYE 3tu1 A 1.603 BS01 07G A 1 L54 G58 I61 M62 V93 H96 I99 L37 G41 I44 M45 V76 H79 I82 2.3.2.27 0005634,0043066,0051726 Ki=0.25uM remove_due_to_license_issue Q00987 21954050 1 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 3tu7 H 2.49 BS02 0BM H 1 Y60A N98 L99 I174 D189 A190 E192 S214 W215 G216 G219 Y47 N95 L96 I171 D191 A192 E194 S218 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 Ki=8.17nM remove_due_to_license_issue Ki=8.2nM, IC50=46nM P00734 11738570 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3tu9 A 2.09 BS01 5MM A 1 A31 D33 E34 S35 S38 K107 K146 E187 K229 S271 G272 Y301 G302 R303 A31 D33 E34 S35 S38 K107 K146 E187 K229 S271 G272 Y301 G302 R303 D33 K146 E187 E189 K229 S300 Y363 D33 K146 E187 E189 K229 S300 Y349 4.1.2.13 0004332,0005515,0005737,0006096,0016829,0030335,0031430,0031674,0034316,0051289 remove_due_to_license_issue IC50=7500nM P00883 24900268 364 PHSHPALTPEQKKELSDIAHRIVAPGKGILAADESTGSIAKRLQSIGTENTEENRRFYRQLLLTADDRVNPCIGGVILFHETLYQKADDGRPFPQVIKSKGGVVGIKVDKGVVPLAGTNGETTTQGLDGLSERCAQYKKDGADFAKWRCVLKIGEHTPSALAIMENANVLARYASICQQNGIVPIVEPEILPDGDHDLKRCQYVTEKVLAAVYKALSDHHIYLEGTLLKPNMVTPGHACTQKYSHEEIAMATVTALRRTVPPAVTGVTFLSGGQSEEEASINLNAINKCPLLKPWALTFSYGRALQASALKAWGGKKENLKAAQEEYVKRALANSLACQGKYTPSNHAY 3tv4 A 3.4 BS01 TV4 A 1 A481 K483 L505 L514 I527 T529 W531 C532 F583 D594 F595 G596 A32 K34 L56 L65 I78 T80 W82 C83 F134 D145 F146 G147 D576 K578 N580 N581 D594 S616 D127 K129 N131 N132 D145 S157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1200nM P15056 24900315 1 DDWEIPDGQITVGQRIGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3tv5 A 2.8 BS01 RCP A 1 V1923 R1954 S1957 E2026 E2028 G2029 E2032 I2033 V444 R475 S478 E547 E549 G550 E553 I554 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 21953464 1 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 3tv5 B 2.8 BS01 RCP B 1 V1923 R1954 F1956 S1957 G1958 E2026 E2028 G2029 E2032 V444 R475 F477 S478 G479 E547 E549 G550 E553 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 21953464 1 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3tv5 B 2.8 BS02 RCP C 1 A1761 V1765 A282 V286 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 21953464 1 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3tv6 A 3.3 BS01 B0R A 1 A481 K483 L505 L514 I527 T529 W531 C532 F583 D594 F595 G596 A34 K36 L58 L67 I80 T82 W84 C85 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 24900315 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3tv7 A 2.75 BS01 07Q A 1 G85 F87 G88 V90 A103 K105 Y155 M156 L205 A215 D216 G77 F79 G80 V82 A95 K97 Y147 M148 L197 A207 D208 D198 K200 N203 D216 T237 D190 K192 N195 D208 T229 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=30nM Q13464 23275831 1 TRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3tv8 A 2.639 BS01 DGJ A 1 W47 D92 D93 Y134 C142 K168 E203 R227 D231 W16 D61 D62 Y103 C111 K137 E172 R196 D200 A170 D231 A139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue IC50=70nM P06280 22195554 801 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFAGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTM 3tv8 B 2.639 BS01 DGJ B 1 W47 D92 D93 Y134 C142 K168 E203 R227 D231 W16 D61 D62 Y103 C111 K137 E172 R196 D200 A170 D231 A139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue IC50=70nM P06280 22195554 802 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFAGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTMQ 3tvc A 2.43 BS06 E3P A 1 L184 L185 A186 L218 V219 H222 E223 H226 H232 L239 F241 I243 Y244 T245 T247 F252 L81 L82 A83 L115 V116 H119 E120 H123 H129 L136 F138 I140 Y141 T142 T144 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=18nM remove_due_to_license_issue Ki=18nM P45452 22689580 1 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDED 3tvl A 2.3 BS01 3PO A 1 K11 R55 R57 K65 R125 K8 R52 R54 K62 R122 3.6.1.28 0000287,0005515,0005737,0005829,0006091,0006772,0009229,0016311,0016462,0016787,0042357,0046872,0050333 remove_due_to_license_issue Q9BU02 23707715 231 GLIEVERKFLPGPGTEERLQELGGTLEYRVTFRDTYYDTPELSLMQADHWLRRREDSGWELKCPGAAGVLGPHTEYKELTAEPTIVAQLCKVLRADGLGAGDVAAVLGPLGLQEVASFVTKRSAWKLVLPQLRVDLDTADFGYAVGEVEALVHEEAEVPTALEKIHRLSSMLGVPAQETAPAKLIVYLQRFRPQDYQRLLEVNS 3tvw A 2.8 BS01 07H A 1 V1923 R1954 F1956 L2025 E2026 E2028 G2029 E2032 I2033 V444 R475 F477 L546 E547 E549 G550 E553 I554 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 21953464 1 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 3tvw B 2.8 BS01 07H B 1 V1923 R1954 L2025 E2026 E2028 G2029 E2032 V444 R475 L546 E547 E549 G550 E553 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 21953464 1 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3tvw B 2.8 BS02 07H C 1 A1761 K1764 A282 K285 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 21953464 1 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 3tvx A 2.84 BS03 PNX A 1 Y371 N533 I548 M569 Q581 F584 Y83 N245 I260 M281 Q293 F296 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=168000nM P27815 22223051 902 MNIPRFGVKTDQEELLAQELENLNKWGLNIFCVSDYAGGRSLTCIMYMIFQERDLLKKFRIPVDTMVTYMLTLEDHYHADVAYHNSLHAADVLQSTHVLLATPALDAVFTDLEILAALFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEDNCDIFQNLSKRQRQSLRKMVIDMVLATDMSKHMTLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLRNMVHCADLSNPTKPLELYRQWTDRIMAEFFQQGDRERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVHPDAQEILDTLEDNRDWYYSAI 3twd A 1.9 BS01 GOB A 1 N377 G379 F402 G404 S405 T420 A422 L436 R440 N146 G148 F171 G173 S174 T189 A191 L205 R209 2.3.1.157,2.7.7.23 0003977,0006048,0016740,0019134 ic50=0.018uM remove_due_to_license_issue IC50=20nM P0ACC7 21984832 1 ASRLERVYQSEQAEKLLLAGVMLRDPARFDLRGTLTHGRDVEIDTNVIIEGNVTLGHRVKIGTGCVIKNSVIGDDCEISPYTVVEDANLAAACTIGPFARLRPGAELLEGAHVGNFVEMKKARLGKGSKAGHLTYLGDAEIGDNVNIGAGTITCNYDGANKFKTIIGDDVFVGSDTQLVAPVTVGKGATIAAGTTVTRNVGENALAISRVPQTQKEGWRRPA 3twd B 1.9 BS01 GOB B 1 C385 Y387 D388 V410 C154 Y156 D157 V179 2.3.1.157,2.7.7.23 0003977,0006048,0016740,0019134 ic50=0.018uM remove_due_to_license_issue IC50=20nM P0ACC7 21984832 454 ASRLERVYQSEQAEKLLLAGVMLRDPARFDLRGTLTHGRDVEIDTNVIIEGNVTLGHRVKIGTGCVIKNSVIGDDCEISPYTVVEDANLAAACTIGPFARLRPGAELLEGAHVGNFVEMKKARLGKGSKAGHLTYLGDAEIGDNVNIGAGTITCNYDGANKFKTIIGDDVFVGSDTQLVAPVTVGKGATIAAGTTVTRNVGENALAISRVPQTQKEGWRRPA 3twj A 2.9 BS01 07R A 1 G85 G88 E89 K105 M128 M153 E154 Y155 M156 L205 A215 D216 G79 G82 E83 K99 M122 M147 E148 Y149 M150 L199 A209 D210 D198 K200 N203 D216 T237 D192 K194 N197 D210 T231 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=8nM Q13464 22846914 1 FETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3txo A 2.05 BS01 07U A 1 F366 V369 A382 K384 E434 V436 D440 L486 D497 F14 V17 A30 K32 E82 V84 D88 L134 D145 D479 K481 D483 N484 D497 T517 D127 K129 D131 N132 D145 T156 2.7.11.13 0004672,0004674,0004697,0005524,0006468 ic50=9nM remove_due_to_license_issue IC50=9.0nM P24723 22078216 1 DNFEFIRVLGKGSFGKVMLARVKETGDLYAVKVLKKDVILQDDDVECTMTEKRILSLARNHPFLTQLFCCFQTPDRLFFVMEFVNGGDLMFHIQKSRRFDEARARFYAAEIISALMFLHDKGIIYRDLKLDNVLLDHEGHCKLADFGMCKEGICGTPDYIAPEILQEMLYGPAVDWWAMGVLLYEMLCGHAPFEAENEDDLFEAILNDEVVYPTWLHEDATGILKSFMTKNPTMRLGSLTQGGEHAILRHPFFKEIDWAQLNHRQIEPPFRPRIKSREDVSNFDPDFIKEEPVLTPIDEGHLPMINQDEFRNFEYVSP 3ty0 A 2.0 BS01 082 A 1 H266 G284 C285 R288 A292 I326 M329 L330 I341 S342 M364 H66 G84 C85 R88 A92 I126 M129 L130 I141 S142 M164 ? 0003677,0004879,0005634,0006355 ic50=83.1nM remove_due_to_license_issue P37231 22070604 1 GSQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 3tyq A 1.6 BS01 HI4 A 1 N316 D319 C366 G410 M414 Y415 Q446 I447 Y448 N311 D314 C361 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 22247956 577 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3tyv A 1.65 BS01 HI3 A 1 F193 C366 S367 G410 M414 Y415 Q446 I447 Y448 S556 F188 C361 S362 G405 M409 Y410 Q441 I442 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.008uM remove_due_to_license_issue O92972 22148957 578 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3tz0 A 2.5 BS01 03H A 1 I72 Y99 H132 R167 I170 R171 I35 Y62 H95 R130 I133 R134 Y241 E245 K248 N249 Y204 E208 K211 N212 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 389 VRLTPTMMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHID 3tz2 A 2.85 BS01 CLT A 1 L68 Y99 L128 L129 H132 R167 I170 R171 L30 Y61 L90 L91 H94 R129 I132 R133 Y241 E245 K248 N249 Y203 E207 K210 N211 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 389 RLTPTMMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHID 3tz4 A 2.25 BS02 03H A 1 I72 Y99 H132 R167 I170 R171 I35 Y62 H95 R130 I133 R134 Y241 E245 K248 N249 Y204 E208 K211 N212 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 390 VRLTPTMMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYHFTTAGFGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHIDG 3tza A 1.9 BS01 TZG A 1 Y58 P86 L87 T88 R93 L135 T140 E190 M193 Y60 P88 L89 T90 R95 L137 T142 E192 M195 ? 0015276,0016020 Ki=3.15uM remove_due_to_license_issue P19491 21923187 261 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 3tzm A 1.7 BS01 085 A 1 G214 A230 K232 L278 S280 Y282 H283 K337 L340 D351 G15 A31 K33 L79 S81 Y83 H84 K138 L141 D152 D333 K335 N338 D351 T375 D134 K136 N139 D152 T174 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=94nM, Ki=17nM, EC50=172nM P36897 21983015 1 TIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLS 3u0d A 2.51 BS01 DBH A 1 S68 R72 W79 K134 S65 R69 W76 K131 ? 0036094 remove_due_to_license_issue P80188 22928018 180 TSDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 3u0d A 2.51 BS02 DBH A 2 W79 R81 L94 L103 Y106 K125 W76 R78 L91 L100 Y103 K122 ? 0036094 remove_due_to_license_issue P80188 22928018 181 TSDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 3u0d A 2.51 BS03 DBH A 3 Y106 K125 K134 Y103 K122 K131 ? 0036094 remove_due_to_license_issue P80188 22928018 182 TSDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 3u0p A 2.8 BS01 LSC A 1 S76 R79 D80 L90 W131 W153 S71 R74 D75 L85 W126 W148 ? remove_due_to_license_issue P15813 22395072 305 RLFPLRCLQISSFANSSWTRTDGLAWLGELQTHSWSQDSDTVRSLKPWSQGTFSDQQWETLQHIFRVYRSSFTRDVKEFAKMLRLSYPLELQVSAGCEVHPGQASNNFFHVAFQGKDILSFQGTSWEPTQEAPLWVNLAIQVLNQDKWTRETVQWLLQGTCPQFVSGLLESGKSELKKQVKPKAWLSRGPSPGPGRLLLVCHVSGFYPKPVWVKWMRGEQEQQGTQPGDILPNADETWYLRATLDVVAGEAAGLSCRVKHSSLEGQDIVLYWH 3u10 A 2.3 BS01 CMP A 1 V591 M599 F607 G608 E609 I610 C611 R618 T619 A620 R659 I663 V122 M130 F138 G139 E140 I141 C142 R149 T150 A151 R190 I194 ? Kd=82.0nM (22006928) remove_due_to_license_issue Q9UL51 22006928 701 DSSRRQYQEKYKQVEQYMSFHKLPADFRQKIHDYYEHRYQGKMFDEDSILGELNGPLREEIVNFNCRKLVASMPLFANADPNFVTAMLTKLKFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKEMKLSDGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVAIDRLDRIGKKNSILL 3u15 A 1.8 BS01 03M A 1 I60 M61 Y66 Q71 I35 M36 Y41 Q46 ? 0005634,0043066,0051726 Kd=0.078uM remove_due_to_license_issue O15151 22745160 1 QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV 3u15 A 1.8 BS02 03M B 1 M53 L56 G57 F90 V92 M28 L31 G32 F65 V67 ? 0005634,0043066,0051726 Kd=0.078uM remove_due_to_license_issue O15151 22745160 1 QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV 3u15 B 1.8 BS01 03M A 1 M53 G57 F90 V92 M28 G32 F65 V67 ? 0005634,0043066,0051726 Kd=0.078uM remove_due_to_license_issue O15151 22745160 1 QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV 3u15 B 1.8 BS02 03M B 1 I60 M61 Y66 Q71 V92 I35 M36 Y41 Q46 V67 ? 0005634,0043066,0051726 Kd=0.078uM remove_due_to_license_issue O15151 22745160 1 QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV 3u18 A 1.9 BS01 Y0X A 1 K32 Y36 I64 G65 K66 W108 N109 N110 F113 K32 Y36 I64 G65 K66 W108 N109 N110 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 ic50=0.81uM remove_due_to_license_issue P14174 22782901 999 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3u1y A 2.0 BS02 03I A 1 M62 E77 T190 F191 G192 F193 I197 V216 H237 K238 D241 H264 M62 E77 T190 F191 G192 F193 I197 V216 H237 K238 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50<2.13nM remove_due_to_license_issue IC50=0.172nM P47205 22175825 405 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 3u2k A 1.64 BS01 087 A 1 N54 E58 D81 R84 G85 I86 P87 R144 T173 N41 E45 D68 R71 G72 I73 P74 R108 T137 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue IC50=30nM P0A0K8 22183167 1 YGAGQIQVLEGLEAVRKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYE 3u3u C 2.5 BS01 EAH C 1 H53 W59 V126 H130 K133 H53 W59 V126 H130 K133 ? 0005576,0035821,0090729 Kd=133.3nM remove_due_to_license_issue F8QQG5 22311975 236 VNYCRLPCRGDNYHVGCGEPAYAQECGQSPRTRELLKEHRNEILSKINDVRDHVAKGSWGLPVAARMKVVVWDAELAGLAKRHTKGCVGETHACRNTERFWLPGQLNFKYSGDKLPRIKELIDDAVKKGHLQKHNITREIIENYRENGPNGDVKELALAISDRVTAVGCGLTTWEDGAKARALLTCNFSSQNTRGRPVYKIGNSPGEKCIEKDETYKNLCSATEPIDPNKSN 3u4h A 1.878 BS01 C8R A 1 L124 W125 S126 R127 L145 E146 W189 S220 T221 F222 E226 L77 W78 S79 R80 L98 E99 W142 S173 T174 F175 E179 E146 T221 E226 E99 T174 E179 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue P28907 23840430 401 QTWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFDTSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVEVHNLQPEKVQTLEAWVIHGSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKNPEDSSC 3u4i A 2.118 BS01 CVR A 1 W125 S126 R127 L145 E146 W189 S193 S220 T221 F222 E226 W81 S82 R83 L101 E102 W145 S149 S176 T177 F178 E182 E146 T221 E226 E102 T177 E182 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue P28907 23840430 401 RWRQTWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFDTSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVEVHNLQPEKVQTLEAWVIHSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKNPEDSSC 3u4m A 2.0 BS01 rna B 0 H3 G4 K5 R6 Y7 A35 K36 F37 T40 E42 H44 P133 R134 D166 K167 T168 H172 P174 S211 Y213 T215 T217 M218 G219 S221 H3 G4 K5 R6 Y7 A35 K36 F37 T40 E42 H44 P133 R134 D166 K167 T168 H172 P174 S211 Y213 T215 T217 M218 G219 S221 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 22868771 2105 ~ 2184 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMGPSVRINPHS 3u4o A 1.77 BS01 08E A 1 N316 C366 L384 G410 M414 Y415 Q446 I447 Y448 N311 C361 L379 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.053uM remove_due_to_license_issue O92972 22104146 579 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3u4r A 2.0 BS01 08F A 1 F193 S288 N291 N316 D318 D319 C366 L384 G410 M414 Y415 Y448 G449 S556 F188 S283 N286 N311 D313 D314 C361 L379 G405 M409 Y410 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.039uM remove_due_to_license_issue O92972 22104146 579 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 3u4u A 2.2 BS01 LNH A 1 L45 G46 V53 V66 K68 F113 V116 M163 I174 D175 L44 G45 V52 V65 K67 F112 V115 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=<3.0nM P68400 24900464 334 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 3u5j A 1.6 BS01 08H A 1 W81 P82 F83 L92 I146 W40 P41 F42 L51 I105 ? Kd=2.46uM remove_due_to_license_issue Kd=2460nM O60885 22137933 1 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 3u5l A 1.39 BS01 08K A 1 W81 P82 F83 L92 N140 I146 W40 P41 F42 L51 N99 I105 ? Kd=0.64uM remove_due_to_license_issue Kd=640nM O60885 22137933 1 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 3u6a A 2.199 BS01 18P A 1 Q12 G13 L30 D32 Y71 F108 D228 G230 T231 T232 Q15 G16 L33 D35 Y74 F111 D221 G223 T224 T225 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=36nM P56817 22071305 386 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3u6h A 2.0 BS01 03X A 1 I1084 F1089 V1092 A1108 F1124 E1127 M1131 L1157 Y1159 M1160 M1211 D1222 F1223 I34 F39 V42 A58 F74 E77 M81 L107 Y109 M110 M161 D172 F173 D1204 A1206 R1208 N1209 D1222 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005524,0006468 Ki=1nM remove_due_to_license_issue IC50=1.000000nM, Ki=1nM P08581 22320343 1 VHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 3u6i A 2.1 BS01 044 A 1 I1084 F1089 V1092 A1108 F1124 E1127 G1128 M1131 L1157 Y1159 M1160 M1211 D1222 F1223 I34 F39 V42 A58 F74 E77 G78 M81 L107 Y109 M110 M161 D172 F173 D1204 A1206 R1208 N1209 D1222 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1nM, Ki=1.9nM P08581 22320343 1 VHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVH 3u6j A 2.15 BS01 03X A 1 L840 V848 A866 K868 E885 L889 C919 L1019 H1026 L1035 C1045 D1046 F1047 L26 V34 A50 K52 E69 L73 C103 L153 H160 L169 C179 D180 F181 D1028 A1030 R1032 N1033 D1046 K1055 D1064 D162 A164 R166 N167 D180 K189 D198 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=10nM P35968 22320343 1 EHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHH 3u6w A 2.21 BS02 KIV A 1 R80 L143 P252 T254 H285 H287 R62 L125 P234 T236 H267 H269 2.3.3.13 0003824,0003852,0009098,0019752,0046912 Kd=120nM remove_due_to_license_issue P9WQB3 22352945 427 IVKPAGPPRVGQPSWNPQRASSMPVNRYRPFAEEVEPIRLRNRTWPDRVIDRAPLWCAVDLRDGNQALIDPMSPARKRRMFDLLVRMGYKEIEVGFPSASQTDFDFVREIIEQGAIPDDVTIQVLTQCRPELIERTFQACSGAPRAIVHFYNSTSILQRRVVFRANRAEVQAIATDGARKCVEQAAKYPGTQWRFEYSPESYTGTELEYAKQVCDAVGEVIAPTPERPIIFNLPATVEMTTPNVYADSIEWMSRNLANRESVILSLHPHNDRGTAVAAAELGFAAGADRIEGCLFGNGERTGNVCLVTLGLNLFSRGVDPQIDFSNIDEIRRTVEYCNQLPVHERHPYGGDLVYTAFSGSHQDAINKGLDAMKDVDDMLWQVPYLPIDPRDVGRTYEAV 3u6w B 2.21 BS02 KIV B 1 R80 L143 E218 P252 T254 H285 H287 R63 L126 E201 P235 T237 H268 H270 2.3.3.13 0003824,0003852,0009098,0019752,0046912 Kd=120nM remove_due_to_license_issue P9WQB3 22352945 427 TIVKPAGPPRVGQPSWNPQRASSMPVNRYRPFAEEVEPIRLRNRTWPDRVIDRAPLWCAVDLRDGNQALIDPMSPARKRRMFDLLVRMGYKEIEVGFPSASQTDFDFVREIIEQGAIPDDVTIQVLTQCRPELIERTFQACSGAPRAIVHFYNSTSILQRRVVFRANRAEVQAIATDGARKCVEQAAKYPGTQWRFEYSPESYTGTELEYAKQVCDAVGEVIAPTPERPIIFNLPATVEMTTPNVYADSIEWMSRNLANRESVILSLHPHNDRGTAVAAAELGFAAGADRIEGCLFGNGERTGNVCLVTLGLNLFSRGVDPQIDFSNIDEIRRTVEYCNQLPVHERHPYGGDLVYTAFSGSHQDAINKGLDAMKLDADCDVDDMLWQVPYLPIDPRDVGRTYEAV 3u78 A 2.689 BS02 E67 A 1 Q200 T279 H282 D284 F285 P391 D392 Q87 T166 H169 D171 F172 P278 D279 1.14.11.65 remove_due_to_license_issue Q6ZMT4 22227394 707 PVQAGTRTFIKELRSRVFPSADEIIIKMHGSQLTQRYLEKHGFDVPIMVPKLDDLGLRLPSPTFSVMDVERYVGGDKVIDVIDVARQADSKMTLHNYVKYFMNPNRPKVLNVISLEFSDTKMSELVEVPDIAKKLSWVENYWPDDSVFPKPFVQKYCLMGVQDSYTDFHIDFGGTSVWYHVLWGEKIFYLIKPTDENLARYESWSSSVTQSEVFFGDKVDKCYKCVVKQGHTLFVPTGWIHAVLTSQDCMAFGGNFLHNLNIGMQLRCYEMEKRLKTPDLFKFPFFEAICWFVAKNLLETLKELREDGFQPQTYLVQGVKALHTALKLWMKKELVSEHAFEIPDNVRPGHLIKELSKVIRAIEEEN 3u7f B 1.8 BS01 dna X 0 D172 N217 Q218 G220 R258 F305 D31 N76 Q77 G79 R117 F164 2.7.1.78,3.1.3.32 0006281,0046403,0046404 remove_due_to_license_issue Q9JLV6 22171004 401 ~ 402 SSLGWESLKKLLVFTASGVKPQGKVAAFALDGTLITTRSGKVFPTSPSDWRILYPEIPKKLQELAAEGYKLVIFTNQMGIGRGKLPAEVFKGKVEAVLEKLGVPFQVLVATHAGLNRKPVSGMWDHLQEQANEGIPISVEDSVFVGDAAGRLANWAPGRKKKDFSCADRLFALNVGLPFATPEEFFLKWPAARFELPAFDPRTISSAGPLYLPESSSLLSPNPEVVVAVGFPGAGKSTFIQEHLVSAGYVHVNRDTLGSWQRCVSSCQAALRQGKRVVIDNTNPDVPSRARYIQCAKDAGVPCRCFNFCATIEQARHNNRFREMTDPSHAPVSDMVMFSYRKQFEPPTLAEGFLEILEIPFRLQLDPALQRLYRQFSEG 3u7k A 1.9 BS01 MDB A 1 Q45 R56 S57 G58 V59 G60 Q65 E109 G110 A111 L112 H154 E155 H158 Q45 R56 S57 G58 V59 G60 Q65 E109 G110 A111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 3.5.1.88 0006412,0016787,0042586,0043686,0046872 remove_due_to_license_issue Q5HGZ3 22751663 301 MLTMKDIIRDGHPTLRQKAAELELPLTKEEKETLIAMREFLVNSQDEEIAKRYGLRSGVGLAAPQINISKRMIAVLIPDDGSGKSYDYMLVNPKIVSHSVQEAYLPTGEGCLSVDDNVAGLVHRHNRITIKAKDIEGNDIQLRLKGYPAIVFQHEIDHLNGVMFYDHIDKDHPLQPHTDAVEVLE 3u7l A 2.01 BS02 UDB A 1 R56 S57 G58 V59 G60 Q65 G110 A111 L112 H154 E155 H158 R56 S57 G58 V59 G60 Q65 G110 A111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 3.5.1.88 0006412,0016787,0042586,0043686,0046872 remove_due_to_license_issue Q5HGZ3 22751663 192 MLTMKDIIRDGHPTLRQKAAELELPLTKEEKETLIAMREFLVNSQDEEIAKRYGLRSGVGLAAPQINISKRMIAVLIPDDGSGKSYDYMLVNPKIVSHSVQEAYLPTGEGCLSVDDNVAGLVHRHNRITIKAKDIEGNDIQLRLKGYPAIVFQHEIDHLNGVMFYDHIDKDHPLQPHTDAVEVLE 3u7m A 2.15 BS02 FHF A 1 S57 G58 V59 G60 Q65 G110 A111 L112 H154 E155 H158 S57 G58 V59 G60 Q65 G110 A111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 3.5.1.88 0006412,0016787,0042586,0043686,0046872 remove_due_to_license_issue Q5HGZ3 22751663 192 MLTMKDIIRDGHPTLRQKAAELELPLTKEEKETLIAMREFLVNSQDEEIAKRYGLRSGVGLAAPQINISKRMIAVLIPDDGSGKSYDYMLVNPKIVSHSVQEAYLPTGEGCLSVDDNVAGLVHRHNRITIKAKDIEGNDIQLRLKGYPAIVFQHEIDHLNGVMFYDHIDKDHPLQPHTDAVEVLE 3u7n A 2.3 BS02 UHF A 1 S57 G58 V59 G60 Q65 G110 A111 L112 H154 E155 H158 S57 G58 V59 G60 Q65 G110 A111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 G60 Q65 C111 L112 H154 E155 H158 3.5.1.88 0006412,0016787,0042586,0043686,0046872 remove_due_to_license_issue Q5HGZ3 22751663 192 MLTMKDIIRDGHPTLRQKAAELELPLTKEEKETLIAMREFLVNSQDEEIAKRYGLRSGVGLAAPQINISKRMIAVLIPDDGSGKSYDYMLVNPKIVSHSVQEAYLPTGEGCLSVDDNVAGLVHRHNRITIKAKDIEGNDIQLRLKGYPAIVFQHEIDHLNGVMFYDHIDKDHPLQPHTDAVEVLE 3u7s A 2.05 BS01 017 A 1 D25 G27 A28 D29 D30 I50 D25 G27 A28 D29 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3700pM remove_due_to_license_issue P35963 19535439 201 PQITLWQRPLVVVKVGGQLMEALLDTGADDTIFEEMNLPGRWTPKMIGGIGGFLNVRQYDQVPIEICGHKVVSTVLIGPTPLNVIGRNVMTQIGCTLNF 3u7s A 2.05 BS02 017 A 2 D25 G48 G49 I50 P81 L82 D25 G48 G49 I50 P81 L82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3700pM remove_due_to_license_issue P35963 19535439 202 PQITLWQRPLVVVKVGGQLMEALLDTGADDTIFEEMNLPGRWTPKMIGGIGGFLNVRQYDQVPIEICGHKVVSTVLIGPTPLNVIGRNVMTQIGCTLNF 3u7s B 2.05 BS01 017 A 1 D25 G48 G49 P81 L82 D25 G48 G49 P81 L82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 19535439 201 PQITLWQRPLVVVKVGGQLMEALLDTGADDTIFEEMNLPGRWTPKMIGGIGGFLNVRQYDQVPIEICGHKVVSTVLIGPTPLNVIGRNVMTQIGCTLNF 3u7s B 2.05 BS02 017 A 2 D25 G27 A28 D29 D30 I50 D25 G27 A28 D29 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 19535439 202 PQITLWQRPLVVVKVGGQLMEALLDTGADDTIFEEMNLPGRWTPKMIGGIGGFLNVRQYDQVPIEICGHKVVSTVLIGPTPLNVIGRNVMTQIGCTLNF 3u81 A 1.13 BS01 SAH A 1 K46 G66 Y68 S72 E90 I91 A118 S119 D141 H142 K45 G65 Y67 S71 E89 I90 A117 S118 D140 H141 D141 K144 D169 N170 E199 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 Ki=36uM remove_due_to_license_issue P22734 22349227 222 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSPD 3u8d A 1.805 BS01 U8D A 1 L2 F5 H6 Y21 C28 G29 G31 H47 D48 K62 F98 L2 F5 H6 Y21 C28 G29 G31 H47 D48 K62 F98 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 remove_due_to_license_issue IC50=470nM P14555 23482564 201 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 3u8h A 2.3 BS01 BHP A 1 L2 F5 H6 A17 G22 G29 V30 G31 C44 H47 D48 Y51 L2 F5 H6 A17 G22 G29 V30 G31 C44 H47 D48 Y51 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 remove_due_to_license_issue P14555 23482564 125 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 3u8h A 2.3 BS04 BHP B 1 A18 F23 A18 F23 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 remove_due_to_license_issue P14555 23482564 125 NLVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRITCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRC 3u8j B 2.35 BS01 09O B 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=3.1nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSEIL 3u8j B 2.35 BS02 09O A 1 L112 M114 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=3.1nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSEIL 3u8j C 2.35 BS01 09O C 1 Y89 W143 Y185 Y192 Y89 W143 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=3.1nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 3u8k A 2.47 BS01 09P A 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=2.2nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSEI 3u8k A 2.47 BS02 09P E 1 R104 L112 M114 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=2.2nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSEI 3u8k B 2.47 BS01 09P A 1 L112 M114 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=2.2nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8k B 2.47 BS02 09P B 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y180 Y187 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=2.2nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l A 2.32 BS01 09Q A 1 Y89 W143 Y185 C188 Y192 Y89 W143 Y182 C185 Y189 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l A 2.32 BS02 09Q B 2 Y89 K139 Y89 K139 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 212 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l A 2.32 BS03 09Q E 1 Q73 R104 L112 M114 Q73 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l B 2.32 BS01 09Q A 1 Q73 R104 Q73 R104 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l B 2.32 BS02 09Q B 1 Y89 W143 Y185 C188 Y192 Y89 W143 Y185 C188 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l B 2.32 BS03 09Q B 2 W53 D160 E163 Y164 W53 D160 E163 Y164 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 212 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8l B 2.32 BS04 09Q B 3 L33 K34 F35 E157 D161 S162 I173 V176 Q178 L33 K34 F35 E157 D161 S162 I173 V176 Q178 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=8.9nM P58154 22170047 213 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8m A 2.7 BS01 09R A 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y181 Y188 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=1.3nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGR 3u8m A 2.7 BS02 09R E 1 R104 L112 M114 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=1.3nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGR 3u8m B 2.7 BS01 09R A 1 R104 L112 M114 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=1.3nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8m B 2.7 BS02 09R B 1 Y89 W143 T144 Y185 C187 Y192 Y89 W143 T144 Y179 C181 Y186 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=1.3nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8n A 2.35 BS01 09S A 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y182 Y189 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=0.067nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8n A 2.35 BS02 09S E 1 R104 L112 M114 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=0.067nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8n B 2.35 BS01 09S A 1 A103 R104 L112 M114 A103 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=0.067nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTNSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8n B 2.35 BS02 09S B 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y183 Y190 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=0.067nM P58154 22170047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTNSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3u8w A 2.15 BS01 09J A 1 K53 E71 L75 T106 D112 L167 D168 F169 K50 E68 L72 T103 D109 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=1nM remove_due_to_license_issue IC50=1nM Q16539 22196117 500 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3u90 A 1.9 BS01 SDS A 1 S27 R59 E63 S26 R58 E62 ? 0005506,0005737,0005764,0005776,0006826,0006879,0008198,0008199,0031410,0044754,0046872,0070288 remove_due_to_license_issue P02791 22525747 175 SQIRQNYSTEVEAAVNRLVNLYLRASYTYLSLGFYFDRDDVALEGVCHFFRELAEEKREGAERLLKMQNQRGGRALFQDLQKPSQDEWGTTLDAMKAAIVLEKSLNQALLDLHALGSAQADPHLCDFLESHFLDEEVKLIKKMGDHLTNIQRLVQAGLGEYLFERLTL 3u92 A 1.9 BS01 KAI A 1 E13 Y61 P88 T90 R95 G140 A141 T142 E189 E11 Y59 P86 T88 R93 G138 A139 T140 E187 ? 0015276,0016020 remove_due_to_license_issue Ki=32.8nM P42264 23141068 258 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 3u93 A 1.881 BS01 GLU A 1 Y61 T90 R95 G140 A141 T142 E189 Y59 T88 R93 G138 A139 T140 E187 ? 0015276,0016020 remove_due_to_license_issue P42264 23141068 258 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGCP 3u9c A 3.2 BS01 04G A 1 V66 K68 F113 V116 I174 D175 V65 K67 F112 V115 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 22868753 404 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 3u9n A 1.85 BS01 09H A 1 L15 Y20 A36 K38 E85 C87 E91 E134 L137 D148 K270 K271 L9 Y14 A30 K32 E71 C73 E77 E120 L123 D134 K256 K257 D130 K132 E134 N135 D148 T170 D116 K118 E120 N121 D134 T156 2.7.11.1 0000077,0004672,0004674,0005524,0006468 remove_due_to_license_issue EC50=10000nM, IC50=75nM O14757 301 EDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 3u9q A 1.522 BS02 DKA A 1 I281 F282 C285 S289 H323 F363 H449 L469 Y473 I62 F63 C66 S70 H104 F144 H230 L250 Y254 ? 0003677,0004879,0005634,0006355 Ki=41.7uM remove_due_to_license_issue P37231 22039047 1 SADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 3ua8 A 1.9 BS01 08W A 1 E13 Y61 P89 L90 T91 R96 T174 E193 M196 E9 Y57 P85 L86 T87 R92 T170 E189 M192 ? 0015276,0016020 ic50=14nM remove_due_to_license_issue P42262 22197388 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLRNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3ua9 A 2.15 BS02 IWR A 1 F1035 A1038 G1043 F1044 D1045 H1048 Y1050 Y1060 Y1071 F84 A87 G92 F93 D94 H97 Y99 Y109 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=135nM Q9H2K2 22233320 2 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 3ubd A 1.53 BS01 SL0 A 1 I50 F79 K100 V131 L147 D148 E197 L200 I2 F31 K52 V77 L93 D94 E143 L146 D193 K195 E197 N198 D211 T231 D139 K141 E143 N144 D157 T172 2.7.11.1 0004672,0004674,0005524,0006468 Kd=2.9uM remove_due_to_license_issue P18654 22846040 400 EIAITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKP 3ubx A 3.1 BS01 09N A 1 C12 S28 F70 Y73 S76 D80 L84 W133 W142 L150 D153 G155 T156 C7 S23 F65 Y68 S71 D75 L79 W128 W137 L145 D148 G150 T151 ? remove_due_to_license_issue P11609 22110136 287 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYWHHHHHHH 3ubx L 3.1 BS01 09N A 1 N31 R32 G50 N31 R32 G50 remove_due_to_license_issue 22110136 287 DIQMTQSSSSFSVSLGDRATITCKASEDIYNRIAWYQQKPGNVPRLLISGATSLETGVPSRFSGSGSGKDYTLSITSLQTEDVATYYCQHYWSSPLTFGAGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 3uby A 2.0 BS01 dna C 0 Y127 H136 M149 Y159 I161 Y162 Y165 C167 N169 L180 R197 G217 P218 S219 K220 V262 G263 Y48 H57 M70 Y80 I82 Y83 Y86 C88 N90 L101 R118 G130 P131 S132 K133 V175 G176 3.2.2.21 0003677,0003824,0003905,0006284 remove_due_to_license_issue P29372 22148158 1 ~ 11 GPHMTRLGLEFFDQPAVPLARAFLGQVLVRRLPNGTELRGRIVETEAYLGPEDEAAHSRGGRQTPRNRGMFMKPGTLYVYIIYGMYFCMNISSQGDGACVLLRALEPLEGLETMRQLRSTLLKDRELCSGPSKLCQALAINKSFDQRDLAQDEAVWLERGPLEPSEPAVVAAARVGVAGEWARKPLRFYVRGSPWVSVVDRVAE 3uby A 2.0 BS02 dna D 0 R141 T143 P144 R145 Y162 G163 R62 T64 P65 R66 Y83 G84 3.2.2.21 0003677,0003824,0003905,0006284 remove_due_to_license_issue P29372 22148158 1 ~ 8 GPHMTRLGLEFFDQPAVPLARAFLGQVLVRRLPNGTELRGRIVETEAYLGPEDEAAHSRGGRQTPRNRGMFMKPGTLYVYIIYGMYFCMNISSQGDGACVLLRALEPLEGLETMRQLRSTLLKDRELCSGPSKLCQALAINKSFDQRDLAQDEAVWLERGPLEPSEPAVVAAARVGVAGEWARKPLRFYVRGSPWVSVVDRVAE 3ucj A 1.85 BS02 AZM A 1 C47 D49 H103 G107 A108 A111 W115 T123 C42 D44 H98 G102 A103 A106 W110 T118 C47 D49 R51 H103 C106 C42 D44 R46 H98 C101 4.2.1.1 0004089,0008270,0015976,0016829,0046872 Ki=1uM remove_due_to_license_issue Q96554 22162771 229 TADLSPLLEANRKWADECAAKDSTYFSKVAGSQAPEYLYIGCADSRVSPAQLFNMAPGEVFVQRNVGNLVSNKDLNCMSCLEYTVDHLKIKHILVCGHYNCGACKAGLVWHPKTAGVTNLWISDVREVRDKNAAKLHGLSADDAWDKMVELNVEAQVFNVCASPIVQAAWARGQPLSVHGIVYTPGTGLVKELIKPITGMEDAGALLRADLKQHCFFSESLA 3ucj A 1.85 BS03 AZM B 1 F66 Y88 F61 Y83 C47 D49 R51 H103 C106 C42 D44 R46 H98 C101 4.2.1.1 0004089,0008270,0015976,0016829,0046872 Ki=1uM remove_due_to_license_issue Q96554 22162771 229 TADLSPLLEANRKWADECAAKDSTYFSKVAGSQAPEYLYIGCADSRVSPAQLFNMAPGEVFVQRNVGNLVSNKDLNCMSCLEYTVDHLKIKHILVCGHYNCGACKAGLVWHPKTAGVTNLWISDVREVRDKNAAKLHGLSADDAWDKMVELNVEAQVFNVCASPIVQAAWARGQPLSVHGIVYTPGTGLVKELIKPITGMEDAGALLRADLKQHCFFSESLA 3ucj B 1.85 BS01 AZM A 1 F66 Y88 F61 Y83 C47 D49 R51 H103 C106 C42 D44 R46 H98 C101 4.2.1.1 0004089,0008270,0015976,0016829,0046872 Ki=1uM remove_due_to_license_issue Q96554 22162771 229 TADLSPLLEANRKWADECAAKDSTYFSKVAGSQAPEYLYIGCADSRVSPAQLFNMAPGEVFVQRNVGNLVSNKDLNCMSCLEYTVDHLKIKHILVCGHYNCGACKAGLVWHPKTAGVTNLWISDVREVRDKNAAKLHGLSADDAWDKMVELNVEAQVFNVCASPIVQAAWARGQPLSVHGIVYTPGTGLVKELIKPITGMEDAGALLRADLKQHCFFSESLA 3ucj B 1.85 BS03 AZM B 1 C47 D49 V71 H103 G107 A108 A111 W115 T123 C42 D44 V66 H98 G102 A103 A106 W110 T118 C47 D49 R51 H103 C106 C42 D44 R46 H98 C101 4.2.1.1 0004089,0008270,0015976,0016829,0046872 Ki=1uM remove_due_to_license_issue Q96554 22162771 229 TADLSPLLEANRKWADECAAKDSTYFSKVAGSQAPEYLYIGCADSRVSPAQLFNMAPGEVFVQRNVGNLVSNKDLNCMSCLEYTVDHLKIKHILVCGHYNCGACKAGLVWHPKTAGVTNLWISDVREVRDKNAAKLHGLSADDAWDKMVELNVEAQVFNVCASPIVQAAWARGQPLSVHGIVYTPGTGLVKELIKPITGMEDAGALLRADLKQHCFFSESLA 3ud5 A 2.0 BS01 J1A A 1 T42 P43 L45 Y53 N55 Q74 D95 D97 I98 R110 L111 T112 F123 T42 P43 L45 Y53 N55 Q74 D95 D97 I98 R110 L111 T112 F123 R82 R92 D95 D97 R82 R92 D95 D97 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 remove_due_to_license_issue Kd=>150000nM, IC50=>100000nM P26281 22169600 171 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 3ud7 B 2.8 BS01 IDY D 1 N18 K113 Q127 K128 A129 N8 K103 Q117 K118 A119 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 1 PKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3ud7 B 2.8 BS02 GNS D 1 K112 K118 K102 K108 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 2 PKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3ud8 A 2.37 BS01 IDY D 1 N18 K113 Q127 K128 A129 N10 K105 Q119 K120 A121 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 1 KKPKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3ud8 A 2.37 BS02 GNX D 1 N18 K112 K113 K118 N10 K104 K105 K110 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 2 KKPKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3ud9 B 2.34 BS01 IDY D 1 N18 K113 Q127 K128 A129 N9 K104 Q118 K119 A120 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 1 KPKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3ud9 B 2.34 BS02 SGN D 1 N18 K112 K113 K118 N9 K103 K104 K109 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 2 KPKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3uda B 2.51 BS01 IDY D 1 N18 K113 Q127 A129 N8 K103 Q117 A119 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 1 PKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3uda B 2.51 BS02 SUS D 1 K112 K113 K118 K102 K103 K108 ? 0001525,0001759,0005104,0005178,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005938,0007165,0008083,0008201,0008284,0008543,0009653,0010595,0022008,0030154,0030324,0030334,0030335,0030544,0031012,0032148,0034605,0042060,0043406,0043410,0044548,0045542,0045766,0045944,0050673,0050679,0051781,0060681,0070374,0072163,1901509,1902533,1903672,2000347,2000544 remove_due_to_license_issue P05230 23240683 2 PKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPV 3udd A 1.95 BS02 34M A 1 H1184 P1187 F1188 A1191 I1192 F1197 D1198 H1201 Y1203 Y1213 G1227 I1228 H80 P83 F84 A87 I88 F93 D94 H97 Y99 Y109 G123 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Kd=79nM O95271 22260203 1 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKPEA 3udh A 1.7 BS01 091 A 1 L30 D32 Y71 Q73 F108 D228 G230 L32 D34 Y73 Q75 F110 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 Kd=1.4mM remove_due_to_license_issue P56817 22468999 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udj A 1.8 BS01 092 A 1 L30 D32 G34 Y71 F108 D228 G230 L32 D34 G36 Y73 F110 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=242uM remove_due_to_license_issue P56817 22468999 401 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udk A 2.51 BS01 095 A 1 L30 D32 G34 Y71 I226 D228 V332 L32 D34 G36 Y73 I222 D224 V328 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 22468999 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udm A 1.94 BS01 09A A 1 L30 D32 G34 Y71 Q73 F108 Y198 D228 G230 L32 D34 G36 Y73 Q75 F110 Y194 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=33uM remove_due_to_license_issue P56817 22468999 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udn A 2.193 BS01 09B A 1 L30 D32 G34 Y71 Q73 F108 R128 Y198 D228 G230 L32 D34 G36 Y73 Q75 F110 R130 Y194 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=7uM remove_due_to_license_issue P56817 22468999 401 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udp A 1.95 BS01 09D A 1 L30 D32 G34 Y71 T72 Q73 F108 R128 Y198 D228 G230 L32 D34 G36 Y73 T74 Q75 F110 R130 Y194 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=6uM remove_due_to_license_issue P56817 22468999 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udq A 2.73 BS01 09E A 1 L30 D32 G34 Y71 T72 Q73 F108 W115 Y198 D228 G230 L32 D34 G36 Y73 T74 Q75 F110 W117 Y194 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 22468999 4000 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udr A 1.95 BS01 09F A 1 L30 D32 G34 Y71 Q73 F108 Y198 I226 D228 G230 L32 D34 G36 Y73 Q75 F110 Y194 I222 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=11uM remove_due_to_license_issue P56817 22468999 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3udv A 1.88 BS01 J1C A 1 T42 L45 Y53 N55 W89 G90 R92 D95 D97 I98 R110 L111 T112 F123 T42 L45 Y53 N55 W85 G86 R88 D91 D93 I94 R106 L107 T108 F119 R82 R92 D95 D97 R82 R88 D91 D93 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=2.55uM remove_due_to_license_issue Kd=2550nM, IC50=3160nM P26281 22169600 171 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 3udy A 2.0 BS01 09G A 1 L30 D32 G34 Y71 Q73 F108 R128 Y198 D228 G230 L32 D34 G36 Y73 Q75 F110 R130 Y194 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=2uM remove_due_to_license_issue P56817 22468999 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 3ue4 A 2.424 BS01 DB8 A 1 L248 A269 K271 V299 I313 T315 F317 M318 T319 L370 F382 L16 A37 K39 V67 I81 T83 F85 M86 T87 L138 F150 D363 A365 R367 N368 D381 P402 D131 A133 R135 N136 D149 P170 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1.1nM, Kd=0.057000nM P00519 22493660 601 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSI 3uew A 2.0 BS01 PLM A 1 L46 L54 K60 I71 I84 F105 M107 L45 L53 K59 I70 I83 F104 M106 ? 0005515,0005576,0019841,0036041,0036094,0042802 Ka=2043000M^-1 remove_due_to_license_issue P02754 22425630 1000 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 3uf9 A 2.68 BS03 FST A 1 H24 D256 C258 I261 W263 T265 A266 H24 D256 C258 I261 W263 T265 A266 H22 H24 K137 H170 H199 D202 R223 D256 H22 H24 K137 H170 H199 D202 R223 D256 3.1.8.1 0004063,0008270,0009056,0016787,0016788,0046872 remove_due_to_license_issue Q97VT7 23139857 317 MRIPLVGKDSIESKDIGFTLIHEHLRVFSEAVRQQWPHLYNEDEEFRNAVNEVKRAMQFGVKTIVDPTVMGLGRDIRFMEKVVKATGINLVAGTGIYIYIDLPFYFLNRSIDEIADLFIHDIKEGIQGTLNKAGFVKIAADEPGITKDVEKVIRAAAIANKETKVPIITHSNAHNNTGLEQQRILTEEGVDPGKILIGHLGDTDNIDYIKKIADKGSFIGLDRYGLDLFLPVDKRNETTLRLIKDGYSDKIMISHDYCCTIDWGTAKPEYKPKLAPRWSITLIFEDTIPFLKRNGVNEEVIATIFKENPKKFFS 3uf9 C 2.68 BS03 FST C 1 H24 R223 L226 F229 D256 C258 W263 T265 A266 H24 R223 L226 F229 D256 C258 W263 T265 A266 H22 H24 K137 H170 H199 D202 R223 D256 H22 H24 K137 H170 H199 D202 R223 D256 3.1.8.1 0004063,0008270,0009056,0016787,0016788,0046872 remove_due_to_license_issue Q97VT7 23139857 317 MRIPLVGKDSIESKDIGFTLIHEHLRVFSEAVRQQWPHLYNEDEEFRNAVNEVKRAMQFGVKTIVDPTVMGLGRDIRFMEKVVKATGINLVAGTGIYIYIDLPFYFLNRSIDEIADLFIHDIKEGIQGTLNKAGFVKIAADEPGITKDVEKVIRAAAIANKETKVPIITHSNAHNNTGLEQQRILTEEGVDPGKILIGHLGDTDNIDYIKKIADKGSFIGLDRYGLDLFLPVDKRNETTLRLIKDGYSDKIMISHDYCCTIDWGTAKPEYKPKLAPRWSITLIFEDTIPFLKRNGVNEEVIATIFKENPKKFFS 3ufa A 1.8 BS01 VPF A 1 H39 A149 Q150 P151 G152 S154 L169 A171 N181 H39 A149 Q150 P151 G152 S154 L169 A171 N180 3.4.21.- 0004252,0005576,0006508,0008236 remove_due_to_license_issue Q2FXC2 24375505 201 EKNVKEITDATKEPYNSVVAFVGGTGVVVGKNTIVTNKHIAKSNDIFKNRVSAHHSSKGKGGGNYDVKDIVEYPGKEDLAIVHVHETSTEGLNFNKNVSYTKFADGAKVKDRISVIGYPKGAQTKYKMFESTGTINHISGTFMEFDAYAQPGNSGSPVLNSKHELIGILYAGSGDESEKNFGVYFTPQLKEFIQNNIEK 3ufd A 2.8 BS01 dna C 0 R17 T23 Q24 R35 S39 R43 N44 R16 T22 Q23 R34 S38 R42 N43 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 3ufd A 2.8 BS02 dna D 0 L33 D34 T36 Y37 R46 N47 L48 T49 S52 L32 D33 T35 Y36 R45 N46 L47 T48 S51 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 3ufd B 2.8 BS01 dna C 0 L33 D34 T36 Y37 R46 N47 L48 T49 S52 L32 D33 T35 Y36 R45 N46 L47 T48 S51 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILKH 3ufd B 2.8 BS02 dna D 0 T23 Q24 R35 S39 R43 N44 T22 Q23 R34 S38 R42 N43 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILKH 3ufd E 2.8 BS01 dna G 0 T23 Q24 R35 S39 R43 T22 Q23 R34 S38 R42 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 3ufd E 2.8 BS02 dna H 0 L33 D34 T36 Y37 R46 N47 L48 T49 S52 L32 D33 T35 Y36 R45 N46 L47 T48 S51 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 3ufd F 2.8 BS01 dna G 0 L33 D34 T36 Y37 R46 N47 T49 S52 L31 D32 T34 Y35 R44 N45 T47 S50 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 SFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILKH 3ufd F 2.8 BS02 dna H 0 T23 Q24 R35 R43 T21 Q22 R33 R41 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 22941636 1 ~ 19 SFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTYISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILKH 3ufl A 1.9 BS01 508 A 1 D32 G34 V69 P70 Y71 K75 F108 I118 D228 G230 T231 D36 G38 V73 P74 Y75 K79 F112 I122 D221 G223 T224 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.15uM remove_due_to_license_issue IC50=150nM P56817 22130130 449 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3ug2 A 2.5 BS01 IRE A 1 S719 A743 K745 L788 M790 M793 D800 S23 A44 K46 L84 M86 M89 D96 D837 A839 R841 N842 D855 G874 D133 A135 R137 N138 D151 G170 2.7.10.1 0004672,0004713,0005524,0006468 Kd=5.6nM remove_due_to_license_issue P00533 22349823 1 EAPNQALLRILKETEFKKIKVLSSGTVYKGLWIPEGEKVKIPVAIKESPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLEDMDDVVDADEYLI 3ugc A 1.34 BS01 046 A 1 L855 V863 A880 K882 E898 L902 V911 L927 Y931 L932 G935 I973 H974 L983 G993 D994 F995 L13 V21 A38 K40 E56 L60 V69 L85 Y89 L90 G93 I131 H132 L141 G151 D152 F153 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S161 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue O60674 22684457 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDN 3uh2 A 2.0 BS02 P34 A 1 H1184 G1185 G1206 Y1213 A1215 S1221 Y1224 I1228 H80 G81 G99 Y106 A108 S114 Y117 I121 2.4.2.-,2.4.2.30 0003950 ic50=1uM remove_due_to_license_issue IC50=39nM O95271 22297980 1 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKP 3uh2 A 2.0 BS03 P34 A 2 F1188 I1192 F1197 D1198 H1201 F84 I88 F93 D94 H97 2.4.2.-,2.4.2.30 0003950 ic50=1uM remove_due_to_license_issue IC50=39nM O95271 22297980 2 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKP 3uh4 A 2.0 BS02 XAV A 1 H1184 G1185 S1186 P1187 F1188 Y1213 F1214 A1215 S1221 Y1224 H80 G81 S82 P83 F84 Y106 F107 A108 S114 Y117 2.4.2.-,2.4.2.30 0003950 ic50=0.011uM remove_due_to_license_issue IC50=11nM, Kd=100nM O95271 22297980 1 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEAP 3uhm A 1.26 BS02 RFN A 1 L18 M62 E77 T190 F191 H237 D241 H264 L18 M62 E77 T190 F191 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=3.6nM remove_due_to_license_issue IC50=3.6nM P47205 22257165 303 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 3ui7 A 2.28 BS01 C1L A 1 H525 L675 I692 M713 Q726 F729 H70 L220 I237 M258 Q271 F274 3.1.4.17 0004114,0007165,0008081 Ki=1nM remove_due_to_license_issue Ki=1nM Q9Y233 22142545 1 WQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 3uib A 2.65 BS01 SB2 A 1 A49 T112 M115 H160 L165 C175 D176 A29 T74 M77 H122 L127 C137 D138 D158 H160 N163 D176 H195 D120 H122 N125 D138 H145 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q4QHJ8 22884419 362 AAMRDLIAELVQRYGAVCAGVDSEGIPVAIKRVFNTNILSDSFLCKRVLREIRLLNHFHHPNILGLRDILYLVTELMRTDLAQVIHDQRIVISPQHIQYFMYHILLGLHVLHEAGVVHRDLHPGNILLADNNDITICDFNLYVTHRWYRAPELVMQFKGFTKLVDMWSAGCVMAEMFNRKALFRGSTFYNQLNKIVEVVGTPKIEDVVMFSSPSARDYLRNSLSNVPARAWTAVVPTADPVALDLIAKMLEFNPQRRISTEQALRHPYFESLFDPLDLTEGLSERFHFDESVTDVYDMHKIFTAEVERF 3uix A 2.2 BS01 Q17 A 1 F49 V52 A65 K67 D128 E171 L174 I185 D186 F13 V16 A29 K31 D89 E132 L135 I146 D147 D167 K169 N172 D186 L193 T204 D128 K130 N133 D147 L154 T165 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.151uM remove_due_to_license_issue P11309 22306408 400 QYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3uj9 A 1.24 BS01 PC A 1 Y19 Y27 I36 D128 Y160 Y175 R179 Y181 K247 Y11 Y19 I28 D120 Y152 Y167 R171 Y173 K239 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 Kd=23.4uM remove_due_to_license_issue Q8IDQ9 22117061 301 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 3ujb A 1.521 BS02 SAH A 1 Y19 I36 S37 G63 D85 I86 I111 R127 H132 Y9 I26 S27 G53 D75 I76 I101 R117 H122 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 remove_due_to_license_issue Q8IDQ9 22117061 502 KTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 3ujc A 1.19 BS01 PC A 1 Y19 Y27 I36 D128 Y160 Y175 R179 Y181 K247 Y11 Y19 I28 D120 Y152 Y167 R171 Y173 K239 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 Kd=26uM remove_due_to_license_issue Q8IDQ9 22117061 301 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILALSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 3ujd A 1.5 BS01 PC A 1 Y27 I36 D128 Y160 Y175 R179 Y181 K247 Y18 I27 D119 Y151 Y166 R170 Y172 K238 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 Kd=20.2uM remove_due_to_license_issue Q8IDQ9 22117061 301 DKTFLENNQFTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 3ukr A 2.48 BS01 CKH B 1 L117 S188 L105 S176 ? 0003779,0005515,0005524,0005634,0005737,0005829,0005856,0005885,0010592,0030030,0034314,0035861,0042995,0045944,0051015,0060271 remove_due_to_license_issue P61157 22623398 401 GRLPACVVDCGTGYTKLGYAGNTEPQFIIPSCIAIKESVMKGVDDLDFFIGDEAIEKPTYATKWPIRHGIVEDWDLMERFMEQVIFKYLRAEPEDHYFLLTEPPLNTPENREYTAEIMFESFNVPGLYIAVQAVLALAASWTSRQVGERTLTGTVIDSGDGVTHVIPVAEGYVIGSCIKHIPIAGRDITYFIQQLLRDREVGIPPEQSLETAKAVKERYSYVCPDLVKEFNKYDTDGSKWIKQYTGINAISKKEFSIDVGYERFLGPEIFFHPEFANPDFTQPISEVVDEVIQNCPIDVRRPLYKNIVLSGGSTMFRDFGRRLQRDLKRTVDARLKLSEELSKPKPIDVQVITHHMQRYAVWFGGSMLASTPEFYQVCHTKKDYEEIGPSICRHNPVFGVM 3ukr B 2.48 BS01 CKH B 1 Y202 A203 F204 D209 L246 P247 D248 Y49 A50 F51 D56 L93 P94 D95 ? 0003779,0005515,0005524,0005634,0005737,0005829,0005856,0005885,0005938,0010592,0034314,0035861,0042995,0045944,0051015,1905168,2001032 ic50=12uM remove_due_to_license_issue A7MB62 22623398 401 GVVVDSGDGVTHICPVYEGFSLPHLTRRLDIAGRDITRYLIKLLLLRGYAFNHSADFETVRMIKEKLCYVGYNIEQEQKLALETTVLVESYTLPDGRIIKVGGERFEAPEALFQPHLINVEGVGVAELLFNTIQAADIDTRSEFYKHIVLSGGSTMYPGLPSRLERELKQLYLERVLKGDVEKLSKFKIRIED 3uli A 2.0 BS01 1N3 A 1 I10 E12 V18 A31 K33 F80 L83 H84 D86 K89 N132 L134 D145 I10 E12 V18 A31 K33 F75 L78 H79 D81 K84 N127 L129 D140 D127 K129 Q131 N132 D145 T165 D122 K124 Q126 N127 D140 T153 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.07uM remove_due_to_license_issue P24941 22305584 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3umo A 1.696 BS01 ATP A 1 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 313 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3umo A 1.696 BS02 ATP A 2 Y23 G26 K27 Y23 G26 K27 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 315 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3umo A 1.696 BS03 ATP B 1 N187 K189 N187 K189 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 312 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3umo B 1.696 BS01 ATP A 2 N187 K189 N187 K189 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 315 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3umo B 1.696 BS02 ATP B 1 Y23 G26 K27 Y23 G26 K27 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 312 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3umo B 1.696 BS03 ATP B 2 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 313 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3ump A 1.849 BS01 ATP A 1 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 313 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3ump A 1.849 BS02 ATP A 2 Y23 G26 K27 Y23 G26 K27 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 314 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLSR 3ump B 1.849 BS01 ATP B 1 Y23 G26 K27 Y23 G26 K27 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 312 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLS 3ump B 1.849 BS02 ATP B 2 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 K185 N187 S224 G226 P227 G229 A254 G255 M258 V280 G283 S284 T287 G253 A254 G255 D256 G253 A254 G255 D256 2.7.1.11 0000287,0003872,0005515,0005524,0005829,0005975,0006096,0006974,0009024,0016301,0016772,0016773,0042802,0042803,0046872,0061615 remove_due_to_license_issue P06999 23823238 313 MVRIYTLTLAPSLDSATITPQIYPEGKLRCTAPVFEPGGGGINVARAIAHLGGSATAIFPAGGATGEHLVSLLADENVPVATVEAKDWTRQNLHVHVEASGEQYRFVMPGAALNEDEFRQLEEQVLEIESGAILVISGSLPPGVKLEKLTQLISAAQKQGIRCIVDSSGEALSAALAIGNIELVKPNQKELSALVNRELTQPDDVRKAAQEIVNSGKAKRVVVSLGPQGALGVDSENCIQVVPPPVKSQSTVGAGDSMVGAMTLKLAENASLEEMVRFGVAAGSAATLNQGTRLCSHDDTQKIYAYLS 3umw A 2.08 BS01 596 A 1 F49 V52 A65 K67 I104 L120 E121 D128 E171 L174 I185 D186 F13 V16 A29 K31 I64 L80 E81 D88 E131 L134 I145 D146 D167 K169 N172 D186 L193 T204 D127 K129 N132 D146 L153 T164 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=3nM remove_due_to_license_issue IC50=6nM P11309 22540945 400 QYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHL 3umx A 2.55 BS01 Q18 A 1 L44 F49 V52 A65 K67 L120 E121 E171 L174 D186 L8 F13 V16 A27 K29 L77 E78 E128 L131 D143 D167 K169 N172 D186 L193 T204 D124 K126 N129 D143 L150 T161 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=410nM P11309 22869110 400 QYQVGPLLGSGGFGSVYSGIRVNLPVAIKHVEKDRISDWGERVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHL 3unj A 1.9001 BS01 0BX A 1 I10 A31 F80 F82 L83 H84 K89 L134 D145 I10 A31 F76 F78 L79 H80 K85 L130 D141 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=11uM remove_due_to_license_issue P24941 22248356 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3unk A 2.1 BS01 0BY A 1 I10 V18 A31 K33 F80 F82 L83 H84 K89 N132 L134 D145 I10 V18 A31 K33 F77 F79 L80 H81 K86 N129 L131 D142 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=15uM remove_due_to_license_issue P24941 22248356 299 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3unz A 2.8 BS01 0BZ A 1 L139 G140 A160 L194 Y212 A213 G216 R220 L263 V279 L13 G14 A34 L68 Y86 A87 G90 R94 L137 V153 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=3.7nM, Kd=16nM O14965 22248356 2 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uo4 A 2.45 BS01 0C0 A 1 R137 L139 V147 A213 G216 R220 E260 N261 L263 A273 R14 L16 V24 A90 G93 R97 E137 N138 L140 A150 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Kd=299nM remove_due_to_license_issue IC50=149.0nM, Kd=299nM O14965 22248356 1 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uo5 A 2.7012 BS01 0BX A 1 R137 L139 G140 V147 L194 A213 T217 R220 L263 R14 L16 G17 V24 L71 A90 T94 R97 L140 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=10.0nM, Kd=39nM O14965 22248356 501 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 3uo6 A 2.8002 BS01 0BY A 1 R137 L139 L194 Y212 A213 G216 T217 L263 V279 R12 L14 L69 Y87 A88 G91 T92 L138 V154 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=2.5nM, Kd=15nM O14965 22248356 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uo9 A 2.3 BS01 04A B 1 K320 L321 F322 L323 D327 Y394 K184 L185 F186 L187 D191 Y258 S286 K289 Y414 Y466 V484 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=100nM, Kd=200nM O94925 22049910 2 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREGE 3uo9 B 2.3 BS01 04A B 1 K320 L321 F322 L323 N324 E325 Y394 K174 L175 F176 L177 N178 E179 Y248 S286 K289 Y414 Y466 V484 S145 K148 Y268 Y320 V338 3.5.1.2 0004359,0006541 ic50=0.08uM remove_due_to_license_issue IC50=100nM, Kd=200nM O94925 22049910 2 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREGE 3uo9 D 2.3 BS01 04A C 1 K320 L321 F322 L323 N324 E325 Y394 K182 L183 F184 L185 N186 E187 Y256 S286 K289 Y414 Y466 V484 S148 K151 Y276 Y328 V346 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=100nM, Kd=200nM O94925 22049910 1 LEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREE 3uod A 2.5002 BS01 0C3 A 1 R137 L139 V147 A213 G216 T217 R220 E260 L263 A273 R14 L16 V24 A90 G93 T94 R97 E137 L140 A150 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Kd=49nM remove_due_to_license_issue IC50=35.0nM, Kd=49nM O14965 22248356 1 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uoh A 2.8002 BS01 0C4 A 1 R137 L139 L194 Y212 A213 G216 T217 R220 L263 V279 R12 L14 L69 Y87 A88 G91 T92 R95 L138 V154 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=2.1nM, Kd=13nM O14965 22248356 2 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uoj A 2.9003 BS01 0C5 A 1 R137 A213 G216 T217 L263 V279 R11 A87 G90 T91 L137 V153 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=43nM, Kd=51nM O14965 22248356 1 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uok A 2.9506 BS01 0C6 A 1 R137 A160 L194 A213 G216 T217 L263 V279 R13 A36 L70 A89 G92 T93 L139 V155 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=0.8nM O14965 22248356 2 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3uol A 2.4 BS01 0C7 A 1 L139 L194 A213 G216 T217 L263 V279 L13 L68 A87 G90 T91 L137 V153 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=3.1nM remove_due_to_license_issue IC50=3.1nM, Kd=18nM O14965 22248356 2 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3up2 A 2.3001 BS01 0C8 A 1 R137 L139 G140 V147 A213 G216 R220 L263 A273 R14 L16 G17 V24 A90 G93 R97 L140 A150 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Kd=40nM remove_due_to_license_issue IC50=28nM, Kd=40nM O14965 22248356 1 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 3up7 A 3.05 BS01 0C9 A 1 R137 L139 G140 V147 A160 A213 G216 R220 D274 R14 L16 G17 V24 A37 A90 G93 R97 D151 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=6.1nM, Kd=34nM O14965 22803810 1 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANS 3upf A 2.6 BS01 0BU A 1 W42 D65 Q66 P69 E168 V170 K171 K174 K180 R182 R245 R392 W41 D64 Q65 P68 E167 V169 K170 K173 K179 R181 R244 R389 2.7.7.48,3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 remove_due_to_license_issue Q80J95 22446684 600 LPRPSGTYAGLPIADYGDAPPLSTKTMFWRTSPEKLPPGAWEPAYLGSKDERVDGPSLQQVMRDQLKPYSEPRGLLPPQEILDAVCDAIENRLENTLEPQKPWTFKKACESLDKNTSSGYPYHKQKSKDWTGSAFIGDLGDQATHANNMYEMGKSMRPIYTAALKDELVKPDKIYGKIKKRLLWGSDLGTMIRAARAFGPFCDALKETCIFNPIRVGMSMNEDGPFIFARHANFRYHMDADYTRWDSTQQRAILKRAGDIMVRLSPEPDLARVVMDDLLAPSLLDVGDYKIVVEEGLPSCPCTTQLNSLAHWILTLCAMVEVTRVDPDIVMQESEFSFYGDDEVVSTNLELDMVKYTMALRRYGLLPTRADKEEPLERRQTLQGISFLRRAIVGDQFGWYGRLDRASIDRQLLWTKGPNHQNPFETLPGHRPQLMALLGEAAMHGEKYYRTVASRVSKEAAVVPRHRSVLRWVRFG 3uph A 2.0 BS01 0C1 A 1 F193 C366 S367 G410 M414 Y415 I447 Y448 G449 S556 F188 C361 S362 G405 M409 Y410 I442 Y443 G444 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=15nM remove_due_to_license_issue O92972 22220815 578 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3upi A 2.0 BS01 0C2 A 1 F193 P197 N316 D319 C366 S367 G410 M414 Y415 I447 Y448 F188 P192 N311 D314 C361 S362 G405 M409 Y410 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=6nM remove_due_to_license_issue O92972 22220815 587 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 3upk A 2.0 BS01 UD1 A 1 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 F328 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 F328 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 22378791 427 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 3upx A 2.27 BS01 B6A A 1 V65 A78 K80 M112 L126 Y131 E135 L181 I194 D195 V22 A35 K37 M69 L83 Y88 E92 L138 I151 D152 D174 K176 E178 N179 D195 T214 D131 K133 E135 N136 D152 T171 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 Ki=0.0075uM remove_due_to_license_issue IC50=15nM Q9BJF5 22369268 1 TAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRDASMLDASAVEHEVDQVLDIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3upy A 1.8 BS02 FOM A 1 E168 K191 K193 F223 E232 H323 E167 K190 K192 F222 E231 H322 ? 0016491,0046872,0050661 ic50=2.39uM remove_due_to_license_issue Q2YIM3 22442144 447 TTNVALVGLARDLAARAETGKPIRIGLIGAGEMGTDIVTQVARMQGIEVGALSARRLPNTFKAIRTAYGDEENAREATTESAMTRAIEAGKIAVTDDNDLILSNPLIDVIIDATGIPEVGAETGIAAIRNGKHLVMMNVEADVTIGPYLKAQADKQGVIYSLGAGDEPSSCMELIEFVSALGYEVVSAGKGKNNPLNFDATPDDYRQEADRRNMNVRLLVEFIDGSKTMVEMAAIANATGLVPDIAGMHGPRASIDQLSHTLIPQAEGGVLSKSGVVDYSIGKGVSPGVFVVAKMDHPRLNERLEDLKIGKGPYFTFHRPYHLTSLEVPLTVARVVLHGKTDMVPLPKPVAEVCAVAKKDMQPGEHLDAIGQYCYRSWIMTVPEARAAKAIPCGLLQNGTVIAPIKKGELITYANAAPQPGSRIAELRALQDAMLG 3upz A 2.2 BS01 B5A A 1 V65 A78 M112 Y131 E135 L181 V22 A35 M69 Y88 E92 L138 D174 K176 E178 N179 D195 T214 D131 K133 E135 N136 D152 T171 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue Q9BJF5 22369268 1 TAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3uqf A 2.27 BS01 BK5 A 1 A293 K295 T338 M341 L393 A36 K38 T81 M84 L136 D386 R388 A390 N391 D404 D129 R131 A133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.2uM remove_due_to_license_issue P00523 22369268 1 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLAPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3uqg A 2.2 BS01 B5A A 1 A293 Y340 M341 L393 A36 Y83 M84 L136 D386 R388 A390 N391 D404 D129 R131 A133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 22369268 1 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3ur0 B 2.45 BS01 SVR B 1 P38 P39 G40 A41 W42 A409 R413 P37 P38 G39 A40 W41 A407 R411 2.7.7.48,3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 ic50=70nM remove_due_to_license_issue Q80J95 22446684 516 LPRPSGTYAGLPIADYGDAPPLSTKTMFWRTSPEKLPPGAWEPAYLGSKDERVDGPSLQQVMRDQLKPYSEPRGLLPPQEILDAVCDAIENRLENTLEPQKPWTFKKACESLDKNTSSGYPYHKQKSKDWTGSAFIGDLGDQATHANNMYEMGKSMRPIYTAALKDELVKPDKIYGKIKKRLLWGSDLGTMIRAARAFGPFCDALKETCIFNPIRVGMSMNEDGPFIFARHANFRYHMDADYTRWDSTQQRAILKRAGDIMVRLSPEPDLARVVMDDLLAPSLLDVGDYKIVVEEGLPSGPCTTQLNSLAHWILTLCAMVEVTRVDPDIVMQESEFSFYGDDEVVSTNLELDMVKYTMALRRYGLLPTRADKEEGPLERRQTLQGISFLRRAIVGDQFGWYGRLDRASIDRQLLWTKGPNHQNPFETLPGRPSQLMALLGEAAMHGEKYYRTVASRVSKEAVVPRHRSVLRWVRFG 3ur9 A 1.65 BS01 K36 A 1 H30 Q110 T134 C139 H157 A158 A159 A160 H32 Q112 T126 C131 H149 A150 A151 A152 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 22915796 203 HMAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSNTVVCAVQA 3usn A -1.00 BS06 ATT A 1 F4 A83 A85 A87 E120 H123 F4 A83 A85 A87 E120 H123 H119 E120 H123 H129 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=710nM P08254 9827994 174 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHSLTDLTRFRLSQDDINGIQSLYGPPP 3usx B 2.28 BS01 MYR B 1 P3 A5 C6 L134 P3 A5 C6 L134 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 23149273 172 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 3utu H 1.55 BS03 1TS H 1 Y60A W60D E97A N98 L99 D189 A190 V213 W215 G216 E217 G219 R221A Y46 W49 E93 N94 L95 D190 A191 V216 W218 G219 E220 G221 R224 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.012nM remove_due_to_license_issue P00734 22907907 901 VEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 3uu1 A 1.82 BS04 14B A 1 N138 A179 P180 H183 Y186 A190 N114 A151 P152 H155 Y158 A162 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 23363292 404 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRASGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 3uug A 1.75 BS01 BDP A 1 R17 D91 R92 D143 N145 W183 Y212 D242 K262 R16 D90 R91 D142 N144 W182 Y211 D241 K261 ? remove_due_to_license_issue P25548 23267119 331 DKGSVGIAMPTKSSARWIDDGNNIVKQLQEAGYKTDLQYADDDIPNQLSQIENMVTKGVKVLVIASIDGTTLSDVLKQAGEQGIKVIAYDRLIRNSGDVSYYATFDNFQVGVLQATSITDKLGLKDGKGPFNIELFGGSPDDNNAFFFYDGAMSVLKPYIDSGKLVVKSGQMGMDKVGTLRWDPATAQARMDNLLSAYYTDAKVDAVLSPYDGLSIGIISSLKGVGYGTKDQPLPVVSGQDAEVPSVKSIIAGEQYSTIFKDTRELAKVTVNMVNAVMEGKEPEVNDTKTYENGVKVVPSYLLKPVAVTKENYKQVLVDGGYYKEDQLK 3uuo A 2.11 BS01 0CV A 1 L675 I692 F696 Q726 F729 L211 I228 F232 Q262 F265 3.1.4.17 0004114,0007165,0008081 Ki=11nM remove_due_to_license_issue Ki=11nM, IC50=858nM Q9Y233 22222034 1 PVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3uvp A 2.4 BS01 048 A 1 A51 K53 E71 T106 L108 M109 L167 D168 A44 K46 E64 T99 L101 M102 L160 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.035uM remove_due_to_license_issue IC50=35nM Q16539 22897496 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 3uvq A 2.2 BS01 FS8 A 1 A51 K53 E71 I84 L104 L108 M109 G110 A111 L167 D168 A47 K49 E67 I80 L100 L104 M105 G106 A107 L160 D161 D150 K152 N155 D168 T185 D143 K145 N148 D161 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=1.000000nM Q16539 23270382 361 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3uwk A 1.91 BS01 0DF A 1 E12 E39 M70 R74 R96 A100 T101 Y104 Q105 F155 E10 E37 M68 R72 R94 A98 T99 Y102 Q103 F150 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=58uM remove_due_to_license_issue Q9HZN8 22243413 800 GLFVTLEGPEGAGKSTNRDYLAERLRERGIEVQLTREPGGTPLAERIRELLLAPSDEPMAADTELLLMFAARAQHLAGVIRPALARGAVVLCDRFTDATYAYQGGGRGLPEARIAALESFVQGDLRPDLTLVFDLPVEIGLARAAARDRFEQEDRRFFEAVRQTYLQRAAQAPERYQVLDAGLPLAEVQAGLDRLLPNLLER 3uwo A 1.7 BS01 0DJ A 1 E39 M70 R74 R96 A100 T101 Y104 Q105 F155 E37 M68 R72 R94 A98 T99 Y102 Q103 F142 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=0.44uM remove_due_to_license_issue Q9HZN8 22243413 800 GLFVTLEGPEGAGKSTNRDYLAERLRERGIEVQLTREPGGTPLAERIRELLLAPSDEPMAADTELLLMFAARAQHLAGVIRPALARGAVVLCDRFTDATYAYQGGGRGLPEARIAALESFVQGDLRPDLTLVFDLPVRLDRFEQEDRRFFEAVRQTYLQRAAQAPERYQVLDAGLPLAEVQAGLDRLLPNLLER 3uxd A 1.8 BS01 0CU A 1 W110 G131 I133 V159 E231 W109 G130 I132 V158 E230 0004425 remove_due_to_license_issue 22685214 291 PRYLKGALKDVVQLSLRRPSLRASRQRPIISLRERILEFNKRNITAIIAVYKRKSPSGLDVERDPIEYAKFMERYAVGLVILTEEKYFNGSYEDLRKIASSVSIPILMWDFIVKESQIDDAYNLGADTVGLIVKILTERELESLLEYARSYGMEPAIVINDEEDLDIALRIGARIIIISSRDLETLEINKENQRKLISMIPSNVVKVAASGISERNEIEELRKLGVNAFEIGSSLMRNPEKIKELIL 3uxk A 2.201 BS02 BHO A 1 V22 K164 K166 D195 N197 E247 H297 L319 V20 K162 K164 D193 N195 E245 H295 L317 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=11.7uM remove_due_to_license_issue Ki=12000nM P11444 22264153 361 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 3uxk C 2.201 BS02 BHO C 1 V22 K164 K166 D195 N197 E247 H297 V20 K162 K164 D193 N195 E245 H295 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=11.7uM remove_due_to_license_issue Ki=12000nM P11444 22264153 361 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 3uxl A 2.201 BS02 CFI A 1 K164 K166 D195 N197 E247 H297 K162 K164 D193 N195 E245 H295 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=2.7uM remove_due_to_license_issue Ki=2670nM P11444 22264153 361 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 3uxl C 2.201 BS02 CFI C 1 K164 K166 D195 E247 H297 K162 K164 D193 E245 H295 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=2.7uM remove_due_to_license_issue Ki=2670nM P11444 22264153 361 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 3uxm A 1.95 BS03 0DN A 1 E12 E39 P40 R50 L54 M70 R74 R96 A100 T101 Y104 Q105 F155 E10 E33 P34 R44 L48 M64 R68 R90 A94 T95 Y98 Q99 F144 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=20uM remove_due_to_license_issue Q9HZN8 22243413 800 GLFVTLEGPEGTNRDYLAERLRERGIEVQLTREPGGTPLAERIRELLLAPSDEPMAADTELLLMFAARAQHLAGVIRPALARGAVVLCDRFTDATYAYQGGGRGLPEARIAALESFVQGDLRPDLTLVFDLPVEIGLARRLDRFEQEDRRFFEAVRQTYLQRAAQAPERYQVLDAGLPLAEVQAGLDRLLPNLLERL 3uyt A 2.0 BS01 0CK A 1 I15 I23 A36 M80 M82 L85 L135 I148 I11 I19 A32 M73 M75 L78 L128 I141 D128 K130 D121 K123 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=13nM P48730 22168824 295 VGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 3uz5 A 1.9 BS01 0CU A 1 W110 G131 I133 V159 E231 W109 G130 I132 V158 E230 0004425 remove_due_to_license_issue 22685214 291 PRYLKGWLEDVVQRSQRRPSVRASRQRPIISLKERILEFNKRNITAIMAVYKRKSPSGLDVERDPIEYAKFMERGVVGLAILTEEKYFNGSYEDLRKIASSVSVPILMWDIIVKESQIDDAYNLGADTVGLIVKILTERELESLLEYARSLGMEPAIVIHDENDLDIALRIGARFIIITSHDLETLEINNENQRKLISMIPSNVVKVVASGISERNEIEELYKLGVNAFEIGTSLMRNPEKIKEFIQ 3uza A 3.273 BS01 T4G A 1 F168 M177 L249 H250 N253 I274 F154 M163 L235 H236 N239 I260 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue Ki=7.76nM P29274 22220592 330 SVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLKQMESQPLPGERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 3uzc A 3.341 BS01 T4E A 1 V84 F168 M177 L249 H250 N253 I274 H278 V78 F154 M163 L235 H236 N239 I260 H264 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue Ki=1.41nM P29274 22220592 330 SVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLKQMESQPLPGERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 3uzj A 1.69 BS01 0CT A 1 W110 I133 V159 I178 E231 W109 I132 V158 I177 E230 0004425 remove_due_to_license_issue 22685214 301 PRYLKGWLEDVVQRSQRRPSVRASRQRPIISLKERILEFNKRNITAIMAVYKRKSPSGLDVERDPIEYAKFMERGVVGLAILTEEKYFNGSYEDLRKIASSVSVPILMWDIIVKESQIDDAYNLGADTVGLIVKILTERELESLLEYARSLGMEPAIVIHDENDLDIALRIGARFIIITSHDLETLEINNENQRKLISMIPSNVVKVVASGISERNEIEELYKLGVNAFEIGTSLMRNPEKIKEFIQ 3uzp A 1.94 BS01 0CK A 1 I23 A36 K38 M80 M82 L85 L135 I148 I21 A34 K36 M78 M80 L83 L133 I146 D128 K130 D126 K128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=13nM P48730 22168824 295 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 3uzt A 3.51 BS01 rna B 0 I197 R199 G200 V205 A218 M274 H280 A321 L324 D335 I168 R170 G171 V176 A189 M245 H251 A292 L295 D306 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 remove_due_to_license_issue P21146 22727813 47 ~ 53 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKDYALGKDCIMHGYMSKMWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQ 3v01 A 2.705 BS01 3V0 A 1 G77 N78 K97 V127 D208 F209 G210 V211 S212 L215 I216 G17 N18 K37 V67 D148 F149 G150 V151 S152 L155 I156 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T163 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=25nM, EC50=6.3nM Q02750 22506516 501 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3v04 A 2.7 BS01 V04 A 1 K97 V127 I141 D208 F209 V211 S212 L215 K37 V67 I81 D148 F149 V151 S152 L155 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T163 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue EC50=0.4nM, IC50=13nM Q02750 22506516 501 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3v0l A 1.75 BS02 2GW A 1 F121 A122 I123 Y126 W181 R188 D211 V212 D213 G267 A268 W300 H301 D302 F57 A58 I59 Y62 W114 R121 D144 V145 D146 G200 A201 W233 H234 D235 H233 G266 W300 E303 A343 H166 G199 W233 E236 A276 2.4.1.37,2.4.1.40 0005975,0016020,0016758 Ki=3uM remove_due_to_license_issue P16442 23836908 450 SLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVP 3v0p A 1.9 BS02 4GW A 1 F121 I123 Y126 W181 R188 D211 V212 D213 A350 V351 F64 I66 Y69 W124 R131 D154 V155 D156 A293 V294 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 remove_due_to_license_issue P16442 23836908 402 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPKNHQAVRN 3v11 A 5.0 BS02 rna D 0 S35 H37 S38 E39 F221 V223 P226 S278 R280 A296 S29 H31 S32 E33 F215 V217 P220 S267 R269 A285 D19 K22 T23 T46 H97 D13 K16 T17 T40 H91 3.6.5.3 0000049,0001731,0003743,0003746,0003924,0005515,0005525,0006412,0006413,0006414,0016787,0046872,1990606 remove_due_to_license_issue Q980A5 22447243 2 ~ 76 QPEVNIGVVGHVDHGKTTLVQAITGIWTSKHSEELKRGMTIKLGYAETNIGVCESCKKPEAYVTEPSCKSCGSDDEPKFLRRISFIDAPGHEVLMATMLSGAALMDGAILVVAANEPFPQPQTREHFVALGIIGVKNLIIVQNKVDVVSKEEALSQYRQIKQFTKGTWAENVPIIPVSALHKINIDSLIEGIEEYIKTPYRDLSQKPVMLVIRSFDVNKPGTQFNELKGGVIGGSIIQGLFKVDQEIKVLPGLRVVSYEPIFTKISSIRFGDEEFKEAKPGGLVAIGTYLDPSLTKADNLLGSIITLADAEVPVLWNIRIKYNLLERVVGAKEMLKVDPIRAKETLMLSVGSSTTLGIVTSVKKDEIEVELRRPVAVWSNNIRTVISRQIAGRWRMIGWGLVEI 3v11 B 5.0 BS01 rna D 0 N53 R62 N94 W97 Q101 K105 N48 R57 N89 W92 Q96 K100 ? 0003676,0003723,0003743,0005515,0006412,0006413,0043022 remove_due_to_license_issue Q97Z79 22447243 2 ~ 76 MIYSRSKLPSEGEILIATVKQVFDYGSYVSLDEYGGLQAFLPWSEVSNIRDVLKENRKVIVKVIRVDRRKGTVDVSLKKVTDDERRKKNLQWKKIQRLDKILELVSQKLKLSEKDAWEQVAWKLEAKYGDPITAIEKAVKEGEKILIDAGVPEIWVKPLLEEASRKVKMSGLITVRTNEPLGVEKIKEVISKALENIEQDYESLLNIKIYTIGAPRYRVDVVGTNPKEASEALNQIISNLIKIGKEENVDISVV 3v1r A 2.8 BS03 JTH A 1 D524 E562 H638 R657 D22 E60 H136 R155 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0003676,0004523 remove_due_to_license_issue Q2F7J3 22366278 675 HGTRPDLTDQPIPDADYTWYTDGSSFLQEGQRRAGAAVTTETEVIWARALPAGTSAQRAELIALTQALKMAEGKKLNVYTDSRYAFATAHVHGEIYRRRGLLTSEGREIKNKNEILALLKALFLPKRLSIIHCPGHQKGNSAEARGNRMADQAAREAAMKAVLET 3v2w A 3.35 BS01 ML5 A 1 Y29 K34 N101 E121 M124 F125 L128 L276 L297 Y13 K18 N78 E98 M101 F102 L105 L393 L414 E1011 D1020 E211 D220 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P21453 22344443 1201 SDYVNYDIIVRHYNYTGKLNISALTSVVFILICCFIILENIFVLLTIWKTKKFHRPMYYFIGNLALSDLLAGVAYTANLLLSGATTYKLTPAQWFLREGSMFVALSASVFSLLAIAIERYITMLKNNFRLFLLISACWVISLILGGLPIMGWNCISALSSCSTVLPLYHKHYILFCTTVFTLLLLSIVILYCRIYSLVRTRNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYASRSSENVALLKTVIIVLSVFIACWAPLFILLLLDVGCKVKTCDILFRAEYFLVLAVLNSGTNPIIYTLTNKEMRRAFIRI 3v3l A 1.65 BS01 V3L A 1 Y107 R110 W114 Y116 I139 Y144 Q153 R161 R163 K175 G179 Y7 R10 W14 Y16 I39 Y44 Q53 R61 R63 K75 G79 2.3.2.27 0008270,0016055,0061630,0072572 Kd~370nM remove_due_to_license_issue Q9NTX7 22267412 1 GEYAWYYEGRNGWWQYDERTSRELEDAFSKGKKNTEMLIAGFLYVADLENMVQYRRNEHGRRRKIKRDIIDIPKKGVAGLRLD 3v3l A 1.65 BS02 V3L B 1 R110 R161 R10 R61 2.3.2.27 0008270,0016055,0061630,0072572 Kd~370nM remove_due_to_license_issue Q9NTX7 22267412 1 GEYAWYYEGRNGWWQYDERTSRELEDAFSKGKKNTEMLIAGFLYVADLENMVQYRRNEHGRRRKIKRDIIDIPKKGVAGLRLD 3v3m A 1.96 BS01 0EN A 1 H41 F140 L141 N142 G143 S144 C145 H163 H164 M165 E166 H41 F140 L141 N142 G143 S144 C145 H163 H164 M165 E166 H41 G143 C145 H41 G143 C145 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0008233,0019082 ic50=4.8uM remove_due_to_license_issue IC50=1500nM P0C6U8 23231439 401 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 3v3q A 2.22 BS01 TMY A 1 E109 S110 A111 F112 L113 E114 R232 C235 L239 I260 T264 E82 S83 A84 F85 L86 E87 R201 C204 L208 I229 T233 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P22736 22983157 301 DAPANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKWAEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFGDWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVAAVAPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPFL 3v3q A 2.22 BS02 TMY A 2 H41 L42 P46 Y122 R123 L162 H163 L166 V167 V169 H14 L15 P19 Y95 R96 L135 H136 L139 V140 V142 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P22736 22983157 302 DAPANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKWAEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFGDWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVAAVAPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPFL 3v3v A 2.7 BS02 MYU A 1 K55 E73 M108 L110 M111 A113 V158 L168 D169 K49 E67 M102 L104 M105 A107 V152 L162 D163 D151 K153 N156 D169 T188 D145 K147 N150 D163 T178 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P45983 23142567 401 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSPEVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMIKGGVLFPGTDHIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDL 3v49 A 1.7 BS02 PK0 A 1 L704 N705 L707 G708 W741 M742 M745 V746 M749 F764 M780 H874 T877 I899 L34 N35 L37 G38 W71 M72 M75 V76 M79 F94 M110 H199 T202 I224 ? ic50=9.6nM remove_due_to_license_issue IC50=9.6nM P10275 22897611 950 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 3v4j A 2.04 BS03 PQR A 1 R278 C308 K310 K334 R83 C113 K115 K139 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q9HC16 22181350 403 SMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAIL 3v4t A 2.5 BS01 UD1 A 1 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 I327 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 I327 K22 N23 D49 R91 D115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 D115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 22378791 501 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGDAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 3v4t B 2.5 BS01 UD1 B 1 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 I327 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 I327 K22 N23 D49 R91 D115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 D115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 22378791 501 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGDAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 3v4t D 2.5 BS01 UD1 D 1 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 I327 F328 N23 W95 R120 P121 V122 D123 L124 K160 S162 V163 G164 T304 D305 I327 F328 K22 N23 D49 R91 D115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 D115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 remove_due_to_license_issue P33038 22378791 501 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGDAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 3v4v A 3.1 BS04 0DU B 1 Y187 F214 Y187 F214 ? 0007155,0008305 remove_due_to_license_issue IC50=32nM P13612 22232704 4000 YNVDTESALLYQGPHNTLFGYSVVLHSHGANRWLLVGAPTANWLANASVINPGAIYRCRIGKNPGQTCEQLQLGSPNGEPCGKTCLEERDNQWLGVTLSRQPGENGSIVTCGHRWKNIFYIKNENKLPTGGCYGVPPDLRTELSKRIAPCYQDYVKKFGENFASCQAGISSFYTKDLIVMGAPGSSYWTGSLFVYNITTNKYKAFLDKQNQVKFGSYLGYSVGAGHFRSQHTTEVVGGAPQHEQIGKAYIFSIDEKELNILHEMKGKKLGSYFGASVCAVDLNADGFSDLLVGAPMQSTIREEGRVFVYINSGSGAVMNAMETNLVGSDKYAARFGESIVNLGDIDNDGFEDVAIGAPQEDDLQGAIYIYNGRADGISSTFSQRIEGLQISKSLSMFGQSISGQIDADNNGYVDVAVGAFRSDSAVLLRTRPVVIVDASLSHPESVNRTKFDCVENGWPSVCIDLTLCFSYKGKEVPGYIVLFYNMSLDVNRKAESPPRFYFSSNGTSDVITGSIQVSSREANCRTHQAFMRKDVRDILTPIQIEAAYHLGPHSTEEFPPLQPILQQKKEKDIMKKTINFAR 3v4v B 3.1 BS04 0DU B 1 S142 Y143 G234 N235 L236 D237 S238 S62 Y63 G154 N155 L156 D157 S158 ? remove_due_to_license_issue IC50=42nM P26010 22232704 4000 RGQQEVLQDQPLSQGARGEGATQLAPQRVRVTLRPGEPQQLQVRFLRAEGYPVDLYYLMDLSYSMKDDLERVRQLGHALLVRLQEVTHSVRIGFGSFVDKTVLPFVSTVPSKLRHPCPTRLERCQSPFSFHHVLSLTGDAQAFEREVGRQSVSGNLDSPEGGFDAILQAALCQEQIGWRNVSRLLVFTSDDTFHTAGDGKLGGIFMPSDGHCHLDSNGLYSRSTEFDYPSVGQVAQALSAANIQPIFAVTSAALPVYQELSKLIPKSAVGELSEDSSNVVQLIMDAYNSLSSTVTLEHSSLPPGVHISYESQCEGPEKREGKAEDRGQCNHVRINQTVTFWVSLQATHCLPEPHLLRLRALGFSEELIVELHTLC 3v4x A 1.952 BS01 F24 A 1 E79 A110 C111 Y143 G148 G149 F185 H233 Y277 G307 S308 E83 A114 C115 Y147 G152 G153 F189 H237 Y281 G311 S312 2.3.3.10 0004421,0006084,0008299,0010142,0016746 remove_due_to_license_issue Q9FD71 22510038 500 STGSMTIGIDKISFFVPPYYIDMTALAEARNVDPGKFHIGIGQDQMAVNPISQDIVTFAANAAEAILTKEDKEAIDMVIVGTESSIDESKAAAVVLHRLMGIQPFARSFEIKEACYGATAGLQLAKNHVALHPDKKVLVVAADIAKYGLNSGGEPTQGAGAVAMLVSSEPRILALKEDNVMLTQDIYDFWRPTGHPYPMVDGPLSNETYIQSFAQVWDEHKKRTGLDFADYDALAFHIPYTKMGKKALLAKISDQTEAEQERILARYEESIIYSRRVGNLYTGSLYLGLISLLENATTLTAGNQIGLFSYGSGAVAEFFTGELVAGYQNHLQKETHLALLDNRTELSIAEYEAMFAETLDTDIDQTLEDELKYSISAINNTVRSYRN 3v51 A 1.95 BS01 I76 A 1 G58 V65 A78 K80 V100 L103 M112 L126 Y131 L181 I194 G197 L198 G16 V23 A36 K38 V58 L61 M70 L84 Y89 L139 I152 G155 L156 D174 K176 E178 N179 D195 T214 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue IC50=5.50nM Q9BJF5 22369268 701 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNDGEVDFDEFQQMLLKLCGN 3v5g A 1.5 BS02 0F3 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=74nM remove_due_to_license_issue Ki=74nM P00918 22775345 800 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3v5g A 1.5 BS03 0F3 A 2 H4 H15 W16 D19 F20 H1 H12 W13 D16 F17 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=74nM remove_due_to_license_issue Ki=74nM P00918 22775345 801 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3v5g A 1.5 BS04 0F3 A 3 F70 D72 I91 F67 D69 I88 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=74nM remove_due_to_license_issue Ki=74nM P00918 22775345 802 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3v5j A 2.59 BS01 0F2 A 1 I369 V377 A389 F435 E436 F437 M438 G441 L489 I15 V22 A34 F78 E79 F80 M81 G84 L132 D482 A484 R486 N487 D500 P521 D125 A127 R129 N130 D143 P146 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue IC50=10.9nM Q08881 22464456 701 GSVIDPSELTFVQEIGSGQGLVHLGYWLNKDKVAIKTIREGSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYERSNSEVVEDISTGRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAES 3v5l A 1.86 BS01 0G1 A 1 I369 V377 A389 F435 F437 M438 H440 G441 C442 L489 I15 V21 A33 F75 F77 M78 H80 G81 C82 L129 D482 A484 R486 N487 D500 P521 D122 A124 R126 N127 D140 P145 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=7nM remove_due_to_license_issue IC50=7nM Q08881 22464456 701 GSVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIA 3v5p A 2.1 BS01 C88 A 1 V65 A78 K80 M112 Y131 E135 L181 I194 D195 V23 A36 K38 M70 Y89 E93 L139 I152 D153 D174 K176 E178 N179 D195 T214 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 Ki=0.0011uM remove_due_to_license_issue Q9BJF5 22369268 1 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3v5q A 2.2001 BS01 0F4 A 1 A570 K572 E588 L592 F617 E618 Y619 M620 K621 G623 F675 H677 L686 I695 G696 D697 F698 A38 K40 E54 L58 F83 E84 Y85 M86 K87 G89 F126 H128 L137 I146 G147 D148 F149 D679 R683 N684 D697 S706 D130 R134 N135 D148 S155 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=40nM Q16288 24900443 902 GIHVQHIKRRDIVLKRELKVFLAECYNLSPTKDKMLVAVKALPTLAARKDFQREAELLTNLQHEHIVKFYGVCGDGDPLIMVFEYMKHGDLNKFLRAHGPELGLSQMLHIASQIASGMVYLASQHFVHRDLATRNCLVGANLLVKIGDFGMDVYSTDYYRTMLPIRWMPPESIMYRKFTTESDVWSFGVILWEIFTYGKQPWFQLSNTEVIECITQGRVLERPRVCPKEVYDVMLGCWQREPQQRLNIKEIYKILHALGKATP 3v5t A 2.13 BS01 UW9 A 1 L57 G58 V65 A78 K80 M112 L126 Y131 L181 I194 D195 L15 G16 V23 A36 K38 M70 L84 Y89 L139 I152 D153 D174 K176 E178 N179 D195 T214 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue Q9BJF5 22369268 700 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 3v66 A 1.8 BS01 D3A A 1 S53 F54 Y73 V179 G180 L183 G208 L211 Y276 F288 M295 M325 S18 F19 Y38 V144 G145 L148 G173 L176 Y241 F253 M260 M290 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=1.3nM remove_due_to_license_issue P37268 22464687 402 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVKIRKGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQN 3v6r A 2.6 BS01 CQQ A 1 V78 A91 M149 N152 C154 Q155 S193 L206 Y229 V34 A47 M105 N108 C110 Q111 S149 L162 Y181 D189 K191 N194 D207 T226 D145 K147 N150 D163 T178 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 22284361 403 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIQLDEREHTIEEWKELIYKEVMNS 3v6s A 2.97 BS01 0F0 A 1 G71 S72 V78 A91 M149 N152 C154 Q155 L206 I261 G27 S28 V34 A47 M105 N108 C110 Q111 L162 I212 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 22284361 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIQLDEREHTIEEWKELIYKEVMNS 3v6y A 2.5 BS01 rna B 0 K201 E208 N244 Y245 R288 Q291 H326 K360 Y361 R364 N415 Y416 Q419 K450 S453 H454 E457 F495 N500 Y501 Q504 F552 S553 S554 K557 K35 E42 N78 Y79 R122 Q125 H160 K194 Y195 R198 N249 Y250 Q253 K284 S287 H288 E291 F321 N326 Y327 Q330 F378 S379 S380 K383 ? 0003723 remove_due_to_license_issue Q09312 3 ~ 13 VLPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3v71 A 2.902 BS01 rna B 0 Q214 K252 Y253 R256 Q259 F300 N302 Y303 Q306 K338 S341 H342 E345 F383 Q385 N388 Y389 Q392 F439 S440 S441 K444 Q133 K171 Y172 R175 Q178 F219 N221 Y222 Q225 K257 S260 H261 E264 F300 Q302 N305 Y306 Q309 F351 S352 S353 K356 ? 0003723 remove_due_to_license_issue O44169 1 ISLEDVLLNGQLIDFAIDPSGVKFLEANYPLDSEDQIRKAVFEKFTESTTLFVGLCHSRNGNFIVQKLVELATPAEQRELLRQMIDGGLLAMCKDKFACRVVQLALQKFDHSNVFQLIQELSTFDLAAMCTDQISIHVIQRVVKQLPVDMWTFFVHFLSSGDSLMAVCQDKYGCRLVQQVIDRLAENPKLPCFKFRIQLLHSLMTCIVRNCYRLSSNEFANYVIQYVIKSSGIMEMYRDTIIDKCLLRNLLSMSQDKYASHVIEGAFLFAPPALLHEMMEEIFSVKDVESNRDALDILLFHQYGNYVVQQMISICTAALIELPPAILLLYSGWYEKMKQRVLQHASRLERFSSGKKIIDSVMRH 3v74 A 2.3 BS01 rna B 0 K201 E208 N244 Y245 Q248 R288 Q291 H326 K360 Y361 R364 N415 Y416 Q419 K450 S453 H454 E457 F495 N500 Y501 Q504 F552 S553 S554 K556 K557 K34 E41 N77 Y78 Q81 R121 Q124 H159 K193 Y194 R197 N248 Y249 Q252 K283 S286 H287 E290 F322 N327 Y328 Q331 F379 S380 S381 K383 K384 ? 0003723 remove_due_to_license_issue Q09312 2 ~ 12 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRS 3v78 A 2.299 BS01 ET A 1 S73 L76 W80 Y101 Y115 W131 F155 D156 T159 S61 L64 W68 Y89 Y103 W119 F143 D144 T147 ? 0000976,0003677,0003700,0006355 Kd=2.9uM remove_due_to_license_issue P95092 22821564 301 AGRRQAIVEAAERVIARQGLGGLSHRRVAAEANVPVGSTTYYFNDLDALREAALAHAANASADLLAQWRSDLDKDRDLAATLARLTTVYLADQDRYRTLNELYMAAAHRPELQRLARLWPDGLLALLEPRIGRRAANAVTVFFDGATLHALITGTPLSTDELTDAIARLVAD 3v78 B 2.299 BS01 ET B 1 S73 W80 Y101 N112 Y115 W131 F155 D156 T159 S62 W69 Y90 N101 Y104 W120 F144 D145 T148 ? 0000976,0003677,0003700,0006355 Kd=2.9uM remove_due_to_license_issue P95092 22821564 301 PAGRRQAIVEAAERVIARQGLGGLSHRRVAAEANVPVGSTTYYFNDLDALREAALAHAANASADLLAQWRSDLDKDRDLAATLARLTTVYLADQDRYRTLNELYMAAAHRPELQRLARLWPDGLLALLEPRIGRRAANAVTVFFDGATLHALITGTPLSTDELTDAIARLVAD 3v7c A 2.7 BS01 C77 A 1 S93 T94 Q116 G119 R120 G121 R122 R125 W127 S128 M137 K187 G190 F191 G208 I209 G210 N212 I224 R227 S92 T93 Q115 G118 R119 G120 R121 R124 W126 S127 M136 K186 G189 F190 G207 I208 G209 N211 I223 R226 0004077,0006355,0036211 remove_due_to_license_issue 22437830 401 SKYSQDVLQLLYKNKPNYISGQSIAESLNISRTAVKKVIDQLKLEGCKIDSVNHKGHLLQQLPDIWYQGIIDQYTKSSALFDFSEVYDSIDSTQLAAKKSLVGNQSSFFILSDEQTKGRGRFNRHWSSSKGQGLWMSVVLRPNVAFSMISKFNLFIALGIRDAIQHFSQDEVKVKWPNDIYIDNGKVCGFLTEMVANNDGIEAIICGIGINLTQQLENFDESIRHRATSIQLHDKNKLDRYQFLERLLQEIEKRYNQFLTLPFSEIREEYIAASNIWNRTLLFTENDKQFKGQAIDLDYDGYLIVRDEAGESHRLISADIDF 3v7e A 2.8 BS01 rna C 0 I514 G515 Q518 A537 D538 L541 M562 V573 G574 A575 A576 I13 G14 Q17 A36 D37 L40 M61 V72 G73 A74 A75 ? 0003723,0005737,0005840,1990904 remove_due_to_license_issue P46350 22355167 1 ~ 126 SYDKVSQAKSIIIGTKQTVKALKRGSVKEVVVAKDADPILTSSVVSLAEDQGISVSMVESMKKLGKACGIEVGAAAVAIIL 3v7e B 2.8 BS01 rna D 0 G615 K617 Q618 A637 L641 M662 V673 G674 A676 G14 K16 Q17 A36 L40 M61 V72 G73 A75 ? 0003723,0005737,0005840,1990904 remove_due_to_license_issue P46350 22355167 201 ~ 326 SYDKVSQAKSIIIGTKQTVKALKRGSVKEVVVAKDADPILTSSVVSLAEDQGISVSMVESMKKLGKACGIEVGAAAV 3v7s A 3.1 BS01 36F A 1 S93 T94 Q95 Q116 G119 R120 G121 R125 S128 M137 D180 G190 F191 G208 I209 G210 S92 T93 Q94 Q115 G118 R119 G120 R124 S127 M136 D179 G189 F190 G207 I208 G209 0004077,0006355,0036211 remove_due_to_license_issue 22437830 401 SKYSQDVLQLLYKNKPNYISGQSIAESLNISRTAVKKVIDQLKLEGCKIDSVNHKGHLLQQLPDIWYQGIIDQYTKSSALFDFSEVYDSIDSTQLAAKKSLVGNQSSFFILSDEQTKGRGRFNRHWSSSKGQGLWMSVVLRPNVAFSMISKFNLFIALGIRDAIQHFSQDEVKVKWPNDIYIDNGKVCGFLTEMVANNDGIEAIICGIGINLTQQLENFDESIRHRATSIQLHDKNKLDRYQFLERLLQEIEKRYNQFLTLPFSEIREEYIAASNIWNRTLLFTENDKQFKGQAIDLDYDGYLIVRDEAGESHRLISADIDF 3v7t A 2.09 BS01 0GX A 1 Q102 D203 S204 C205 Q206 S209 V227 W229 G230 G232 Q87 D188 S189 C190 Q191 S194 V212 W214 G215 G217 H59 D106 Q206 G207 D208 S209 G210 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=62nM remove_due_to_license_issue P20231 22264487 301 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 3v7t A 2.09 BS03 0GX C 1 P63 Y99 P48 Y84 H59 D106 Q206 G207 D208 S209 G210 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=62nM remove_due_to_license_issue P20231 22264487 301 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 3v7t C 2.09 BS01 0GX A 1 P63 Y99 P48 Y84 H59 D106 Q206 G207 D208 S209 G210 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=62nM remove_due_to_license_issue P20231 22264487 301 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 3v7t C 2.09 BS02 0GX C 1 Q102 D203 S204 C205 Q206 S209 V227 W229 G230 G232 Q87 D188 S189 C190 Q191 S194 V212 W214 G215 G217 H59 D106 Q206 G207 D208 S209 G210 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=62nM remove_due_to_license_issue P20231 22264487 301 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 3v7x A 1.03 BS02 D7A A 1 H1094 H1119 F1131 L1198 T1199 T1200 H92 H117 F128 L195 T196 T197 H1064 H1094 H1096 E1106 H1119 T1199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.7nM remove_due_to_license_issue Ki=2.7nM P00918 22443141 2002 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3v8s A 2.286 BS01 0HD A 1 R84 G85 G88 E89 V90 A103 K105 M153 E154 Y155 M156 L205 D216 R77 G78 G81 E82 V83 A96 K98 M146 E147 Y148 M149 L198 D209 D198 K200 N203 D216 T237 D191 K193 N196 D209 T230 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.65uM remove_due_to_license_issue IC50=650nM Q13464 22272748 501 ETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3v8t A 2.0 BS01 477 A 1 I369 A389 K391 F435 E436 F437 M438 H440 G441 L489 I15 A32 K34 F78 E79 F80 M81 H83 G84 L132 D482 A484 R486 N487 D500 P521 D125 A127 R129 N130 D143 P147 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=0.3nM remove_due_to_license_issue Q08881 22464456 701 GSVIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAES 3v8w A 2.27 BS01 0G2 A 1 I369 A389 F435 E436 F437 M438 G441 L489 S499 I15 A33 F78 E79 F80 M81 G84 L132 S142 D482 A484 R486 N487 D500 P521 D125 A127 R129 N130 D143 P146 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=8.6nM remove_due_to_license_issue Q08881 22464456 701 GSVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIRGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYERSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 3v9b A 2.1 BS01 IHM A 1 S208 T271 M273 N321 Y329 W332 T333 F340 Q343 M357 S368 Q369 F372 S127 T190 M192 N240 Y248 W251 T252 F259 Q262 M276 S287 Q288 F291 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=500nM Q08499 22371117 1 FGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 3vap A 2.66 BS01 0FY A 1 R137 L139 G140 F144 V147 K162 L194 L210 A213 P214 L215 G216 L263 D274 R11 L13 G14 F18 V21 K36 L68 L84 A87 P88 L89 G90 L137 D148 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T153 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 22503250 1 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 3vbd A 1.05 BS02 0FZ A 1 Q1092 H1094 H1119 F1131 L1198 T1199 T1200 Q90 H92 H117 F128 L195 T196 T197 H1064 H1094 H1096 E1106 H1119 T1199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8.6nM remove_due_to_license_issue Ki=8.6nM P00918 22443141 2002 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3vbg A 2.8 BS01 03M A 1 I61 M62 R65 Y67 Q72 I36 M37 R40 Y42 Q47 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 22745160 1 TLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 3vbg A 2.8 BS02 03M B 1 L57 V93 I99 L32 V68 I74 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 22745160 1 TLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 3vbg B 2.8 BS01 03M A 1 L54 L57 G58 V93 L30 L33 G34 V69 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 22745160 1 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 3vbg B 2.8 BS02 03M B 1 I61 M62 Y67 Q72 I37 M38 Y43 Q48 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 22745160 1 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 3vbq A 1.85 BS01 0F5 A 1 F49 V52 A65 K67 L120 E121 L174 I185 D186 F15 V18 A31 K33 L86 E87 L140 I151 D152 D167 K169 N172 D186 L193 T204 D133 K135 N138 D152 L159 T170 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=470pM remove_due_to_license_issue P11309 22339127 555 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3vbt A 2.23 BS01 0F9 A 1 F49 V52 A65 E121 R122 L174 I185 D186 F15 V18 A31 E83 R84 L136 I147 D148 D167 K169 N172 D186 L193 T204 D129 K131 N134 D148 L155 T166 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=37uM remove_due_to_license_issue IC50=37000nM P11309 22339127 1 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGETRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3vbv A 2.08 BS01 0FK A 1 L44 V52 A65 K67 I104 L120 L174 I185 D186 L10 V18 A31 K33 I67 L83 L137 I148 D149 D167 K169 N172 D186 L193 T204 D130 K132 N135 D149 L156 T167 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=10uM remove_due_to_license_issue IC50=10000nM P11309 22339127 1 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3vbw A 2.48 BS01 0FN A 1 L44 V52 A65 K67 E121 L174 I185 D186 L10 V14 A27 K29 E80 L133 I144 D145 D167 K169 N172 D186 L193 T204 D126 K128 N131 D145 L152 T163 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=6uM remove_due_to_license_issue IC50=6000nM P11309 22339127 1 ESQYQVGPLLGGSVYSGIRVSDNLPVAIKHVEKDRISDWGELTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3vbx A 2.03 BS01 0FO A 1 V52 A65 K67 E121 L174 I185 V18 A31 K33 E84 L137 I148 D167 K169 N172 D186 L193 T204 D130 K132 N135 D149 L156 T167 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=17uM remove_due_to_license_issue IC50=17000nM P11309 22339127 1 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3vby A 2.27 BS01 0FR A 1 F49 V52 A65 K67 L174 I185 D186 F15 V18 A31 K33 L136 I147 D148 D167 K169 N172 D186 L193 T204 D129 K131 N134 D148 L155 T166 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=28uM remove_due_to_license_issue IC50=28000nM P11309 22339127 1 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGETRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 3vc4 A 2.23 BS01 0FS A 1 L44 V52 K67 R122 L174 I185 D186 L12 V20 K35 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=24nM remove_due_to_license_issue IC50=17nM P11309 22339127 1 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 3vd4 A 2.0 BS03 IPT A 1 N102 D201 E461 Y503 E537 H540 N604 W999 N94 D193 E453 Y495 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.015mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGDESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vd4 D 2.0 BS03 IPT D 1 N102 D201 E461 E537 H540 N604 W999 N94 D193 E453 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.015mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGDESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vd7 A 2.87 BS01 GTZ A 1 D201 E461 M502 Y503 E537 H540 W568 N604 W999 D189 E449 M490 Y491 E525 H528 W556 N592 W987 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue P00722 22446164 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGSESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vd7 D 2.87 BS01 GTZ D 1 D201 E461 Y503 E537 H540 W568 N604 W999 D189 E449 Y491 E525 H528 W556 N592 W987 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D189 H345 H379 E404 H406 E449 Y491 E525 N585 F589 N592 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue P00722 22446164 2001 RRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGSESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vd9 A 2.05 BS03 IPT A 1 N102 D201 E461 Y503 E537 H540 N604 W999 N94 D193 E453 Y495 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.1mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGSESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vd9 D 2.05 BS03 IPT D 1 N102 D201 E461 E537 H540 N604 W999 N94 D193 E453 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=0.1mM remove_due_to_license_issue Ki=7.6e+4nM P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGSESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vdb A 2.05 BS01 149 A 1 D201 H391 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=3.03mM remove_due_to_license_issue P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGTESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vdb D 2.05 BS01 149 D 1 D201 H391 E461 M502 Y503 E537 H540 W568 F601 N604 D193 H383 E453 M494 Y495 E529 H532 W560 F593 N596 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 Ki=3.03mM remove_due_to_license_issue P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGTESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vdc A 2.55 BS01 IPT A 1 N102 D201 E461 Y503 E537 H540 N604 W999 N94 D193 E453 Y495 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGTESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3vdc D 2.55 BS01 IPT D 1 N102 D201 E461 E537 H540 N604 W999 N94 D193 E453 E529 H532 N596 W991 D201 H357 H391 E416 H418 E461 Y503 E537 N597 F601 N604 D193 H349 H383 E408 H410 E453 Y495 E529 N589 F593 N596 3.2.1.23 0000287,0003824,0004553,0004565,0005975,0005990,0009056,0009341,0016798,0030246,0031420,0042802,0046872 remove_due_to_license_issue Ki=7.6e+4nM P00722 22446164 2001 VVLQRRDWENPGVTQLNRLAAHPPFASWRNSEEARTDRPSQQLRSLNGEWRFAWFPAPEAVPESWLECDLPEADTVVVPSNWQMHGYDAPIYTNVTYPITVNPPFVPTENPTGCYSLTFNVDESWLQEGQTRIIFDGVNSAFHLWCNGRWVGYGQDSRLPSEFDLSAFLRAGENRLAVMVLRWSDGSYLEDQDMWRMSGIFRDVSLLHKPTTQISDFHVATRFNDDFSRAVLEAEVQMCGELRDYLRVTVSLWQGETQVASGTAPFGGEIIDERGGYADRVTLRLNVENPKLWSAEIPNLYRAVVELHTADGTLIEAEACDVGFREVRIENGLLLLNGKPLLIRGVNRHEHHPLHGQVMDEQTMVQDILLMKQNNFNAVRCSHYPNHPLWYTLCDRYGLYVVDEANIETHGMVPMNRLTDDPRWLPAMSERVTRMVQRDRNHPSVIIWSLGTESGHGANHDALYRWIKSVDPSRPVQYEGGGADTTATDIICPMYARVDEDQPFPAVPKWSIKKWLSLPGETRPLILCEYAHAMGNSLGGFAKYWQAFRQYPRLQGGFVWDWVDQSLIKYDENGNPWSAYGGDFGDTPNDRQFCMNGLVFADRTPHPALTEAKHQQQFFQFRLSGQTIEVTSEYLFRHSDNELLHWMVALDGKPLASGEVPLDVAPQGKQLIELPELPQPESAGQLWLTVRVVQPNATAWSEAGHISAWQQWRLAENLSVTLPAASHAIPHLTTSEMDFCIELGNKRWQFNRQSGFLSQMWIGDKKQLLTPLRDQFTRAPLDNDIGVSEATRIDPNAWVERWKAAGHYQAEAALLQCTADTLADAVLITTAHAWQHQGKTLFISRKTYRIDGSGQMAITVDVEVASDTPHPARIGLNCQLAQVAERVNWLGLGPQENYPDRLTAACFDRWDLPLSDMYTPYVFPSENGLRCGTRELNYGPHQWRGDFQFNISRYSQQQLMETSHRHLLHAEEGTWLNIDGFHMGIGGDDSWSPSVSAEFQLSAGRYHYQLVWCQK 3veh A 2.0 BS01 0GA A 1 P251 L268 T271 H334 T361 Y385 L404 A418 G419 K438 P237 L254 T257 H320 T347 Y371 L390 A404 G405 K424 K205 E252 A269 E297 H334 T361 Y385 R405 G421 E434 K438 K191 E238 A255 E283 H320 T347 Y371 R391 G407 E420 K424 4.2.99.21,5.4.4.2,5.4.99.5 0000162,0000287,0004106,0005886,0008909,0009058,0009697,0010106,0016829,0016833,0016853,0019540,0043904,0046872,0052572 Ki=11uM remove_due_to_license_issue P9WFX1 22607697 501 SSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTRALGRGPAIDRLARDDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRERGSVQHLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVAR 3veu A 1.52 BS01 0GO A 1 G13 D32 G34 S35 Y71 T72 Q73 F108 I126 D219 G221 T222 T223 G16 D35 G37 S38 Y74 T75 Q76 F111 I129 D222 G224 T225 T226 D32 S35 N37 A39 Y71 D219 T222 D35 S38 N40 A42 Y74 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=55nM remove_due_to_license_issue P56817 22380629 378 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3vf3 A 1.48 BS01 0GS A 1 D32 G34 S35 Y71 T72 Q73 F108 Y185 D215 G217 D35 G37 S38 Y74 T75 Q76 F111 Y188 D218 G220 D32 S35 N37 A39 Y71 D215 T218 D35 S38 N40 A42 Y74 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=1.37uM remove_due_to_license_issue P56817 22380629 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3vf5 A 1.25 BS01 031 B 1 D25 G27 A28 D30 P81 V82 D25 G27 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3vf5 B 1.25 BS01 031 B 1 D25 G27 A28 D29 V47 G48 G49 I50 V82 D25 G27 A28 D29 V47 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 3vf7 A 1.3 BS01 031 A 1 L23 D25 G27 A28 D29 G48 G49 I50 L23 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 3vf7 B 1.3 BS01 031 A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 3vf8 A 2.08 BS01 0JE A 1 L377 A400 M450 A451 E452 G454 P455 L501 S511 L15 A36 M80 A81 E82 G84 P85 L131 S141 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=150nM remove_due_to_license_issue P43405 22464456 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 3vf9 A 2.3 BS01 477 A 1 L377 A400 M448 E449 M450 A451 L453 G454 P455 L501 L14 A36 M78 E79 M80 A81 L83 G84 P85 L131 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=358.2nM remove_due_to_license_issue P43405 22464456 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 3vfa A 1.43 BS01 031 A 1 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 3vfa B 1.43 BS01 031 A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 3vfb A 1.55 BS01 031 A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRDLLTQIGATLNF 3vfb B 1.55 BS01 031 A 1 D25 G27 A28 D30 V82 D25 G27 A28 D30 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22401672 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRDLLTQIGATLNF 3vfq A 2.8 BS01 AR6 A 1 G1022 V1023 S1034 P1036 G1044 P1045 L1046 S1049 A1131 G1133 T1134 G1135 N1136 L1137 H1172 D1175 G206 V207 S218 P220 G228 P229 L230 S233 A315 G317 T318 G319 N320 L321 H356 D359 2.4.2.- remove_due_to_license_issue Q460N5 23473667 1201 KCFSRTVLAPGVVLIVQQGDLARLPVDVVVNASNEDLKHYGGLAAALSKAAGPELQADCDQIVKREGRLLPGNATISKAGKLPYHHVIHAVGPRWSGYEAPRCVYLLRRAVQLSLCLAEKYKYRSIAIPAISSGVFGFPLGRCVETIVSAIKENFQFKKDGHCLKEIYLVDVSEKTVEAFAEAVKTVFKGSLVSPGGLQMLLVKEGVQNAKTDVVVNSVPLDLVLSRGPLSKSLLEKAGPELQEELDTVGQGVAVSMGTVLKTSSWNLDCRYVLHVVAPEWRNGSTSSLKIMEDIIRECMEITESLSLKSIAFPAIGTGNLGFPKNIFAELIISEVFKFSSKNQLKTLQEVHFLLHPSDHENIQAFSDEFARRAN 3vg1 A 1.77 BS01 0GT A 1 D32 G34 S35 Y71 T72 F108 I110 W115 I126 Y186 D216 G218 T219 R223 D35 G37 S38 Y74 T75 F111 I113 W118 I129 Y189 D219 G221 T222 R226 D32 S35 N37 A39 Y71 D216 T219 D35 S38 N40 A42 Y74 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.055uM remove_due_to_license_issue P56817 22380629 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3vgc C 1.67 BS02 SRB C 1 S190 M192 S195 V213 S214 W215 G216 S217 S40 M42 S45 V63 S64 W65 G66 S67 M192 G193 D194 S195 G196 M42 G43 D44 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 9425066 358 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 3vh9 A 1.29 BS03 HQY A 1 D117 E152 D179 Y225 Y251 I255 H256 D117 E152 D179 Y225 Y251 I255 H256 H97 D117 E151 E152 D179 H256 H97 D117 E151 E152 D179 H256 3.4.11.10 0006508,0008235 Ki=0.58uM remove_due_to_license_issue Q01693 22311113 303 MPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATG 3vha A 1.39 BS01 VHA A 1 A55 G97 M98 N106 L107 F138 T184 A45 G87 M88 N96 L97 F128 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=40nM remove_due_to_license_issue Kd=40nM P07900 22192591 237 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3vhc A 1.41 BS01 VHC A 1 A55 K58 G97 M98 N106 L107 K112 F138 T184 A46 K49 G88 M89 N97 L98 K103 F129 T175 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=1.3nM remove_due_to_license_issue Kd=1.3nM P07900 22192591 1 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 3vhd A 1.52 BS01 VHE A 1 A55 K58 I96 G97 M98 N106 L107 F138 T184 A44 K47 I85 G86 M87 N95 L96 F127 T173 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.52nM remove_due_to_license_issue Kd=0.52nM P07900 22192591 1 MEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3vhe A 1.55 BS01 42Q A 1 L840 V848 A866 K868 E885 L889 V916 F918 C919 L1035 C1045 D1046 F1047 L30 V38 A56 K58 E75 L79 V106 F108 C109 L171 C181 D182 F183 D1028 R1032 N1033 D1046 K1055 D164 R168 N169 D182 K191 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=6.2nM remove_due_to_license_issue Ki=4.6nM, Kd=19nM, IC50=4.7nM P35968 20833055 1170 LPLDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQ 3vhk A 2.49 BS01 BPK A 1 V848 K868 E885 L1019 C1045 D1046 F1047 V35 K55 E72 L150 C176 D177 F178 D1028 R1032 N1033 D1046 K1055 D159 R163 N164 D177 K186 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue Ki=25000nM, IC50=100000nM P35968 24900475 2001 DEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 3vhu A 2.11 BS01 SNL A 1 L766 L769 N770 Q776 M807 L810 F829 M845 M852 L938 C942 T945 F956 L39 L42 N43 Q49 M80 L83 F102 M118 M125 L205 C209 T212 F223 ? ic50=49nM remove_due_to_license_issue IC50=11nM, Ki=2.323nM P08235 22074142 1001 STISRALTPSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFH 3vhv A 1.35 BS01 LD1 A 1 N770 Q776 M807 L810 S811 L814 F829 M845 M852 L938 F941 C942 T945 N46 Q52 M83 L86 S87 L90 F105 M121 M128 L209 F212 C213 T216 ? ic50=510nM remove_due_to_license_issue IC50=510nM P08235 22074142 1 GSLSTISRALTPSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNVKPLYFHRK 3vi2 A 2.1 BS01 HMZ A 1 D23 T195 A268 Q269 N291 G293 R294 D23 T195 A268 Q269 N291 G293 R294 4.1.1.23 0004590,0006207,0006221,0016831,0044205 remove_due_to_license_issue Q8T6J6 22740703 500 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILK 3vi2 B 2.1 BS01 HMZ B 1 D23 T195 A268 Q269 N291 G293 R294 D23 T195 A268 Q269 N291 G293 R294 4.1.1.23 0004590,0006207,0006221,0016831,0044205 remove_due_to_license_issue Q8T6J6 22740703 600 MGFKVKLEKRRNAINTCLCIGLDPDEKDIENFMKNEKENNYNNIKKNLKEKYINNVSIKKDILLKAPDNIIREEKSEEFFYFFNHFCFYIINETNKYALTFKMNFAFYIPYGSVGIDVLKNVFDYLYELNIPTILDMKINDIGNTVKNYRKFIFEYLKSDSCTVNIYMGTNMLKDICYDEEKNKYYSAFVLVKTTNPDSAIFQKNLSLDNKQAYVIMAQEALNMSSYLNLEQNNEFIGFVVGANSYDEMNYIRTYFPNCYILSPGIGAQNGDLHKTLTNGYHKSYEKILINIGRAITKNPYPQKAAQMYYDQINAILK 3vi5 D 2.0 BS01 M4M D 1 G613 R614 K650 M699 W704 G12 R13 K49 M98 W103 Y608 R614 R619 W704 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 remove_due_to_license_issue O60760 22418579 804 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 3vi7 A 2.0 BS02 CBD A 1 R14 M99 W104 A105 K107 K198 L199 R13 M98 W103 A104 K106 K197 L198 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 remove_due_to_license_issue IC50=2E2nM O60760 22418579 201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 3vid A 2.3 BS01 4TT A 1 V848 A866 E917 F918 C919 G922 L1035 V36 A54 E105 F106 C107 G110 L173 D1028 R1032 N1033 D1046 K1055 D166 R170 N171 D184 K186 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue P35968 24900475 2001 LDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKEAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 3vjc A 1.89 BS01 ZGA A 1 S51 R52 S53 F54 Y73 R77 D80 V175 V179 M295 A296 S16 R17 S18 F19 Y38 R42 D45 V140 V144 M260 A261 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 remove_due_to_license_issue IC50=5nM P37268 22474324 400 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVKIRKGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQ 3vjc B 1.89 BS01 ZGA B 1 T50 S51 R52 S53 F54 Y73 R77 D80 V175 V179 N215 T14 S15 R16 S17 F18 Y37 R41 D44 V139 V143 N179 Y171 R218 R228 F288 Y135 R182 R192 F252 2.5.1.21 0008610,0009058,0016765,0045338,0051996 remove_due_to_license_issue IC50=5nM P37268 22474324 400 SSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVKIRKGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQ 3vje A 2.12 BS01 ZGA A 1 H18 S19 K20 S21 F22 F26 Y41 C44 R45 D48 L107 V137 L164 N168 R171 A244 R265 H18 S19 K20 S21 F22 F26 Y41 C44 R45 D48 L107 V137 L164 N168 R171 A244 R265 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 remove_due_to_license_issue A9JQL9 22474324 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIAIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 3vjk A 2.49 BS01 M51 A 1 E205 E206 S209 F357 R358 S630 Y631 Y662 Y666 E168 E169 S172 F320 R321 S593 Y594 Y625 Y629 Y547 S630 Y631 D708 H740 Y510 S593 Y594 D671 H703 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.37nM remove_due_to_license_issue Kd=12nM, IC50=0.37nM P27487 22959556 1000 DSRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3vjl A 2.393 BS01 W94 A 1 E205 E206 F357 R358 S630 Y631 Y662 Y666 N710 E168 E169 F320 R321 S593 Y594 Y625 Y629 N673 Y547 S630 Y631 D708 H740 Y510 S593 Y594 D671 H703 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=5.6nM remove_due_to_license_issue IC50=5.6nM P27487 22959556 1000 DSRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3vjm A 2.1 BS01 W61 A 1 E205 E206 F357 R358 S630 Y631 Y662 Y666 N710 E168 E169 F320 R321 S593 Y594 Y625 Y629 N673 Y547 S630 Y631 D708 H740 Y510 S593 Y594 D671 H703 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.37nM remove_due_to_license_issue IC50=0.37nM P27487 22824762 1000 DSRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3vjs A 1.93 BS02 10S A 1 V230 S233 I267 R270 S271 S274 W282 V296 H301 H393 V48 S51 I85 R88 S89 S92 W100 V114 H119 H211 ? 0003677,0004879,0006355 ic50=0.64uM remove_due_to_license_issue P13053 22066785 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNE 3vjt A 2.0 BS02 10R A 1 V230 S233 I267 R270 S271 W282 V296 H301 H393 V48 S51 I85 R88 S89 W100 V114 H119 H211 ? 0003677,0004879,0006355 ic50=4.1uM remove_due_to_license_issue P13053 22066785 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3vnt A 1.64 BS01 0JA A 1 V848 A866 K868 E885 L889 I892 V898 V899 V916 F918 C919 K920 G922 L1019 L1035 C1045 D1046 F1047 V37 A55 K57 E74 L78 I81 V87 V88 V105 F107 C108 K109 G111 L152 L168 C178 D179 F180 D1028 A1030 R1032 N1033 D1046 K1055 D161 A163 R165 N166 D179 K188 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=2.2nM remove_due_to_license_issue P35968 22376051 2001 PLDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 3vo3 A 1.52 BS01 0KF A 1 L840 V848 A866 K868 E885 L889 V916 F918 C919 G922 L1035 C1045 D1046 F1047 L29 V37 A55 K57 E74 L78 V105 F107 C108 G111 L170 C180 D181 F182 D1028 A1030 R1032 N1033 D1046 K1055 D163 A165 R167 N168 D181 K190 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=1.4nM remove_due_to_license_issue IC50=1.8nM P35968 23498918 2001 PLDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 3vok A 2.0 BS01 dna U 0 P45 Q51 P44 Q50 ? 0003677,0046872 remove_due_to_license_issue Q9CHR1 22798069 1 ~ 15 PKSTYFSLSDEKRNRVYDACLNEFQTHSFHEAKIMHIVKALDIPRGSFYQYFEDLKDAYFYVLSQETLEIHDLFFNLLKDNSIEESLDKYKYLLLENLIDSPQYKLYKYRFLDWTYELERDWKDNPISQVLKSVVHNLVYRLFSENWTEKTFIENYDKEIKLVTEGLLNYITDRKN 3voz A 2.4 BS01 04A A 1 F318 L321 F322 L323 N324 E325 Y394 F100 L103 F104 L105 N106 E107 Y176 S286 K289 Y414 Y466 V484 S68 K71 Y196 Y248 V266 3.5.1.2 0004359,0006541 ic50=0.14uM remove_due_to_license_issue IC50=100nM, Kd=200nM O94925 22538822 601 SMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 3vp1 A 2.3 BS01 04A A 1 R317 F318 L321 L323 N324 E325 Y394 R99 F100 L103 L105 N106 E107 Y176 S286 K289 Y414 Y466 V484 S68 K71 Y196 Y248 V266 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=100nM, Kd=200nM O94925 22538822 601 SMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 3vp2 A 2.7 BS01 BP0 A 1 L323 Y394 L103 Y174 S286 K289 Y414 Y466 V484 S68 K71 Y194 Y246 V264 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=100000nM O94925 22538822 601 SMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 3vp3 A 2.7 BS01 BP8 A 1 F322 Y394 F102 Y174 S286 K289 Y414 Y466 V484 S68 K71 Y194 Y246 V264 3.5.1.2 0004359,0006541 remove_due_to_license_issue O94925 22538822 601 SMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 3vp4 A 2.45 BS01 BP9 A 1 L323 Y394 L104 Y175 S286 K289 Y414 Y466 V484 S69 K72 Y195 Y247 V265 3.5.1.2 0004359,0006541 remove_due_to_license_issue O94925 22538822 601 QSMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 3vqh A 1.95 BS02 IQB A 1 L49 G50 T51 G52 F54 V57 A70 M120 V123 E127 E170 L173 T183 D184 F327 L46 G47 T48 G49 F51 V54 A67 M117 V120 E124 E167 L170 T180 D181 F324 D166 K168 E170 N171 D184 T201 D163 K165 E167 N168 D181 T198 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue Ki=48nM P17612 22869112 401 AAAKKGSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3vqs A 1.9 BS01 JT1 A 1 V179 Y191 F193 Y195 S196 P197 R200 S288 C289 C366 S368 L384 M414 Y415 I447 Y448 Y452 L466 L547 F551 V179 Y191 F193 Y195 S196 P197 R200 S288 C289 C366 S368 L384 M414 Y415 I447 Y448 Y452 L466 L547 F551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.0178uM remove_due_to_license_issue P26663 22615294 1000 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVA 3vqu A 2.4 BS01 O22 A 1 V539 A551 M602 E603 C604 I607 L654 I663 P673 V24 A36 M86 E87 C88 I91 L138 I147 P157 D647 K649 N652 D664 D674 T686 D131 K133 N136 D148 D158 T160 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 24900510 909 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMSISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 3vrt A 2.4 BS02 YS2 A 1 Y143 S233 I264 R270 S271 S274 W282 C284 V296 H393 Y20 S52 I83 R89 S90 S93 W101 C103 V115 H212 ? 0003677,0004879,0006355 ic50=2.7nM remove_due_to_license_issue P13053 22512505 501 LSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 3vru A 2.0 BS02 YS3 A 1 Y143 V230 S233 R270 S271 S274 W282 C284 V296 H301 H393 Y21 V48 S51 R88 S89 S92 W100 C102 V114 H119 H211 ? 0003677,0004879,0006355 ic50=0.1nM remove_due_to_license_issue P13053 22512505 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3vrv A 1.9 BS02 YSD A 1 Y143 L223 V230 S233 R270 S271 S274 W282 C284 V296 H301 H393 Y21 L41 V48 S51 R88 S89 S92 W100 C102 V114 H119 H211 ? 0003677,0004879,0006355 ic50=0.029nM remove_due_to_license_issue P13053 22512505 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 3vrw A 2.4 BS02 YS5 A 1 Y143 S233 R270 S271 S274 W282 C284 V296 H301 L305 H393 Y21 S52 R89 S90 S93 W101 C103 V115 H120 L124 H212 ? 0003677,0004879,0006355 ic50=0.41nM remove_due_to_license_issue P13053 22512505 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 3vry A 2.481 BS01 B43 A 1 L273 V281 A293 K295 V323 T338 M341 L393 A403 D404 F405 L183 V191 A203 K205 V233 T248 M251 L303 A313 D314 F315 D386 R388 A390 N391 D404 F424 D296 R298 A300 N301 D314 F322 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7.7nM remove_due_to_license_issue P08631 23596204 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 3vs3 A 2.17 BS01 VSE A 1 L273 V281 A293 K295 M314 V323 T338 M341 S345 D348 L393 D404 F405 L189 V197 A209 K211 M230 V239 T254 M257 S261 D264 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F328 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=0.426580nM P08631 23596204 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 3vsw A 3.0 BS01 R31 A 1 T18 Y20 D38 G40 S41 R82 Y83 T85 P118 F119 A122 F124 D226 G228 A229 S230 I305 T18 Y20 D38 G40 S41 R82 Y83 T85 P118 F119 A122 F124 D226 G228 A229 S230 I305 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D226 A229 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=130nM P00797 22726934 402 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3vsx A 2.8 BS01 R32 A 1 D38 G40 S41 R82 Y83 T85 F119 V127 D226 G228 D38 G40 S41 R82 Y83 T85 F119 V127 D226 G228 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D226 A229 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=1.4nM P00797 22726934 402 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3vtb A 2.0 BS02 TKA A 1 Y143 L223 V230 S233 R270 S271 S274 W282 C284 H301 H393 F418 Y21 L43 V50 S53 R90 S91 S94 W102 C104 H121 H213 F238 ? 0003677,0004879,0006355 ic50=0.5nM remove_due_to_license_issue P13053 24773565 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3vtc A 1.5 BS02 TK3 A 1 Y143 V230 S233 R270 S271 S274 W282 C284 H301 L309 H393 L400 Y21 V50 S53 R90 S91 S94 W102 C104 H121 L129 H213 L220 ? 0003677,0004879,0006355 ic50=13nM remove_due_to_license_issue P13053 24773565 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3vtd A 2.7 BS02 TKD A 1 Y143 L223 A227 V230 S233 M268 R270 S271 S274 W282 V296 H301 H393 Y21 L43 A47 V50 S53 M88 R90 S91 S94 W102 V116 H121 H213 ? 0003677,0004879,0006355 remove_due_to_license_issue P13053 24773565 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3vuc A 2.6 BS01 HHE A 1 D38 G40 S41 Y83 T85 P118 F119 F124 V127 L224 D226 G228 D38 G40 S41 Y83 T85 P118 F119 F124 V127 L224 D226 G228 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D226 A229 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 24900544 402 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3vv6 A 2.05 BS01 B00 A 1 D32 Y71 F108 I118 D228 D36 Y75 F112 I122 D220 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=157uM remove_due_to_license_issue P56817 22998419 510 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEFPDGFWLGEQLVCNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3vv7 A 2.1 BS01 0B1 A 1 G13 D32 Y71 F108 I118 D228 G230 G17 D36 Y75 F112 I122 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=4.6uM remove_due_to_license_issue P56817 22998419 509 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEFPDGFWLGEQLVCWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3vv8 A 2.5 BS01 B02 A 1 D32 Y71 F108 I118 D228 G230 D34 Y73 F110 I120 D219 G221 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=17.1uM remove_due_to_license_issue P56817 22998419 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTFPDGFWLGEQLVCWNIFPVISLYLMGEVTNQSFRITILPQQYLRPDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3vva A 2.59 BS03 CHW A 1 C95 R96 F99 R118 F121 L122 L212 E215 A216 T219 C66 R67 F70 R89 F92 L93 L183 E186 A187 T190 1.-.-.- 0005739,0005743,0008199,0009916,0010230,0016491,0046872 remove_due_to_license_issue Q26710 23487766 504 TPVWGHTQLNRLSFLETVPVVPLRVSDESSEDRPTWSLPDIENVAITHKKPNGLVDTLAYRSVRTCRWLFDTFSLYRFGSITESKVISRCLFLETVAGVPGMVGGMLRHLSSLRYMTRDKGWINTLLVEAENERMHLMTFIELRQPGLPLRVSIIITQAIMYLFLLVAYVISPRFVHRFVGYLEEEAVITYTGVMRAIDEGRLRPTKNDVPEVARVYWNLSKNATFRDLINVIRADEAEHRVVNHTFADMHEKRLQNSVNPFVVLK 3vvy A 1.63 BS01 ET A 1 T85 I88 W89 Y92 L130 C134 D152 F155 M184 T78 I81 W82 Y85 L123 C127 D145 F148 M177 ? 0003677 remove_due_to_license_issue A0A0F6AY66 23800819 301 DKKQALLEAATQAIAQSGIAASTAVIARNAGVAEGTLFRYFATKDELINTLYLHLKQDLCQSMIMELDRSITDAKMMTRFIWNSYISWGLNHPARHRAIRQLAVSEKLTKETEQRADDMFPELRDLCHRSVLMVFMSDEYRAFGDGLFLALAETTMDFAARDPARAGEYIALGFEAMWRALTRE 3vvz A 2.51 BS01 RHQ A 1 L66 T85 I88 W89 I106 C134 H135 R148 D152 F155 L59 T78 I81 W82 I99 C127 H128 R141 D145 F148 ? 0003677 remove_due_to_license_issue A0A0F6AY66 23800819 301 DKKQALLEAATQAIAQSGIAASTAVIARNAGVAEGTLFRYFATKDELINTLYLHLKQDLCQSMIMELDRSITDAKMMTRFIWNSYISWGLNHPARHRAIRQLAVSEKLTKETEQRADDMFPELRDLCHRSVLMVFMSDEYRAFGDGLFLALAETTMDFAARDPARAGEYIALGFEAMWRALTRE 3vw0 B 2.6 BS01 DEQ B 1 M70 I88 Y92 A110 C134 D152 F155 L156 M64 I82 Y86 A104 C128 D146 F149 L150 ? 0003677 remove_due_to_license_issue A0A0F6AY66 23800819 301 EDKKQALLEAATQAIAQSGIAASTAVIARNAGVAEGTLFRYFATKDELINTLYLHLKQDLCQSMIMELDRSITDAKMMTRFIWNSYISWGLNHPARHRAIRQLAVSEKLTKETEQRADDMFPELRDLCHRSVLMVFMSDEYRAFGDGLFLALAETTMDFAARDPARAGEYIALGFEAMWRALTRE 3vw1 B 2.21 BS01 CVI B 1 Y59 L66 M70 I88 S91 Y92 I106 L130 F155 Y52 L59 M63 I81 S84 Y85 I99 L123 F148 ? 0003677 remove_due_to_license_issue A0A0F6AY66 23800819 301 DKKQALLEAATQAIAQSGIAASTAVIARNAGVAEGTLFRYFATKDELINTLYLHLKQDLCQSMIMELDRSITDAKMMTRFIWNSYISWGLNHPARHRAIRQLAVSEKLTKETEQRADDMFPELRDLCHRSVLMVFMSDEYRAFGDGLFLALAETTMDFAARDPARAGEYIALGFEAMWRALTRE 3vw2 A 2.34 BS01 BER A 1 T85 C134 V138 D152 F155 L156 M184 T78 C127 V131 D145 F148 L149 M177 ? 0003677 remove_due_to_license_issue A0A0F6AY66 23800819 301 DKKQALLEAATQAIAQSGIAASTAVIARNAGVAEGTLFRYFATKDELINTLYLHLKQDLCQSMIMELDRSITDAKMMTRFIWNSYISWGLNHPARHRAIRQLAVSEKLTKETEQRADDMFPELRDLCHRSVLMVFMSDEYRAFGDGLFLALAETTMDFAARDPARAGEYIALGFEAMWRALTRE 3vw2 B 2.34 BS01 BER B 1 T85 Y92 V138 D152 F155 T189 T78 Y85 V131 D145 F148 T182 ? 0003677 remove_due_to_license_issue A0A0F6AY66 23800819 301 DKKQALLEAATQAIAQSGIAASTAVIARNAGVAEGTLFRYFATKDELINTLYLHLKQDLCQSMIMELDRSITDAKMMTRFIWNSYISWGLNHPARHRAIRQLAVSEKLTKETEQRADDMFPELRDLCHRSVLMVFMSDEYRAFGDGLFLALAETTMDFAARDPARAGEYIALGFEAMWRALTRE 3vw3 H 2.5 BS01 dna A 0 W33 H35 T58 R95 Y97 Y100I W33 H35 T59 R99 Y101 Y105 remove_due_to_license_issue 23519658 1 ~ 18 EVQLQQSGTVLARPGASVKMSCKASGYTFTNYWMHWIKQRPGQGLEWIGTIYPGNSDTTYSQKFKGKAKLTAVTSTSTAYMELSSLTNEDSAVYYCSRRNYGSSYAMDYWGQGTSVTVSSAKTTPPSVYPLAPGSAAQTSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTSTWPSETVTCNVAHPASSTKVDKKIVPR 3vw3 L 2.5 BS01 dna A 0 Y30 Y32 S92 H93 Y34 Y36 S96 H97 remove_due_to_license_issue 23519658 1 ~ 18 VLMTQTPLSLPVSLGDQASISCRSSQNIVHSNGYTYLEWYLQKPGQSPKLLIYTVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFRGSHVPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRN 3vw3 L 2.5 BS02 dna B 0 Q27 N27A V27C N28 G29 Q26 N27 V29 N32 G33 remove_due_to_license_issue 23519658 1 ~ 18 VLMTQTPLSLPVSLGDQASISCRSSQNIVHSNGYTYLEWYLQKPGQSPKLLIYTVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFRGSHVPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRN 3vw6 A 2.4 BS01 IM6 A 1 L686 V694 K709 Q756 V757 G759 G760 L810 S821 L16 V24 K39 Q80 V81 G83 G84 L134 S145 D803 K805 D807 N808 D822 T842 D127 K129 D131 N132 D146 T158 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=14nM Q99683 23147077 1001 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPEQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 3vw7 A 2.2 BS01 VPX A 1 Y183 P236 L237 H255 V257 F271 L332 Y337 A349 Y353 Y93 P141 L142 H160 V162 F176 L396 Y401 A413 Y417 E1011 N1020 E216 N225 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P25116 23222541 2001 DASGYLTSSWLTLFVPSVYTGVFVVSLPLNIMAIVVFILKMKVKKPAVVYMLHLATADVLFVSVLPFKISYYFSGSDWQFGSELCRFVTAAFYCNMYASILLMTVISIDRFLAVVYPMRTLGRASFTCLAIWALAIAGVVPLLLKEQTIQVPGLGITTCHDVLSETLLEGYYAYYFSAFSAVFFFVPLIISTVCYVSIIRCLSSSANIFEMLRIDEGLRLKIYKNTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYANRSKKSRALFLSAAVFCIFIICFGPTNVLLIAHYSFLSHTSTTEAAYFAYLLCVCVSSISCCIDPLIYYYASSEC 3vw9 A 1.47 BS02 HPJ A 1 H126 M157 F162 E172 M179 M183 H119 M150 F155 E165 M172 M176 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 ic50=0.011uM remove_due_to_license_issue Ki=11nM, IC50=11nM Q04760 23122816 203 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 3vw9 A 1.47 BS04 HPJ B 1 Q33 C60 L69 E99 Q26 C53 L62 E92 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 ic50=0.011uM remove_due_to_license_issue Ki=11nM, IC50=11nM Q04760 23122816 202 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 3vw9 B 1.47 BS02 HPJ A 1 Q33 C60 M65 L69 E99 Q26 C53 M58 L62 E92 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 ic50=0.011uM remove_due_to_license_issue Ki=11nM, IC50=11nM Q04760 23122816 203 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 3vw9 B 1.47 BS04 HPJ B 1 H126 F162 E172 M179 H119 F155 E165 M172 Q33 E99 H126 E172 Q26 E92 H119 E165 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 ic50=0.011uM remove_due_to_license_issue Ki=11nM, IC50=11nM Q04760 23122816 202 GGLTDEAALSCCSDADPSTKDFLLQQTMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKMATLM 3vws A 2.1 BS03 VWS A 1 N405 V411 F412 T413 F485 W795 N123 V129 F130 T131 F194 W504 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 Kd=225uM remove_due_to_license_issue Q6YMS4 23408636 1003 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATSMINGVVKLLTKPWDVVPMVTQMAMTQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAAMGAVFTEENQWDSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMMGGKAKGSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 3vws A 2.1 BS04 VWS A 2 F412 N492 Q602 V603 G604 T605 Y606 I797 F130 N201 Q311 V312 G313 T314 Y315 I506 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 Kd=225uM remove_due_to_license_issue Q6YMS4 23408636 1004 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATSMINGVVKLLTKPWDVVPMVTQMAMTQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAAMGAVFTEENQWDSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMMGGKAKGSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 3vx3 A 2.1 BS01 ADP A 1 G30 V31 G32 K33 S34 L35 N187 F218 Y219 D223 G27 V28 G29 K30 S31 L32 N180 F205 Y206 D210 ? 0005524,0016226,0016787,0016887,0046872,0051536,0051539,0140663 remove_due_to_license_issue Q5JIH4 23399544 301 IDPREIAINARLEGVKRIIPVVSGKGGVGKSLVSTTLALVLAEKGYRVGLLDLDFHGASDHVILGFEPKEFPEEDRGVVPPTVHGIKFMTIAYYTTPLRGKEISDALIELLTITRWDELDYLVIDMPPGLGDQLLDVLRFLKRGEFLVVATPSKLSLNVVRKLIELLKEEGHKVIGVVENMKLREKDVEKLAEEFGVPYLVGIPFYPDLDAKVGNVEELMKTEFAGKVRELAGRL 3vx3 A 2.1 BS02 ADP B 1 K28 S160 K25 S153 ? 0005524,0016226,0016787,0016887,0046872,0051536,0051539,0140663 remove_due_to_license_issue Q5JIH4 23399544 301 IDPREIAINARLEGVKRIIPVVSGKGGVGKSLVSTTLALVLAEKGYRVGLLDLDFHGASDHVILGFEPKEFPEEDRGVVPPTVHGIKFMTIAYYTTPLRGKEISDALIELLTITRWDELDYLVIDMPPGLGDQLLDVLRFLKRGEFLVVATPSKLSLNVVRKLIELLKEEGHKVIGVVENMKLREKDVEKLAEEFGVPYLVGIPFYPDLDAKVGNVEELMKTEFAGKVRELAGRL 3vx3 B 2.1 BS01 ADP A 1 K28 S160 K25 S153 ? 0005524,0016226,0016787,0016887,0046872,0051536,0051539,0140663 remove_due_to_license_issue Q5JIH4 23399544 301 IDPREIAINARLEGVKRIIPVVSGKGGVGKSLVSTTLALVLAEKGYRVGLLDLDFHGASDHVILGFEPKEFPEEDRGVVPPTVHGIKFMTIAYYTTPLRGKEISDALIELLTITRWDELDYLVIDMPPGLGDQLLDVLRFLKRGEFLVVATPSKLSLNVVRKLIELLKEEGHKVIGVVENMKLREKDVEKLAEEFGVPYLVGIPFYPDLDAKVGNVEELMKTEFAGKVRELAGRL 3vx3 B 2.1 BS02 ADP B 1 G30 V31 G32 K33 S34 L35 N187 M188 F218 Y219 L222 D223 G27 V28 G29 K30 S31 L32 N180 M181 F205 Y206 L209 D210 ? 0005524,0016226,0016787,0016887,0046872,0051536,0051539,0140663 remove_due_to_license_issue Q5JIH4 23399544 301 IDPREIAINARLEGVKRIIPVVSGKGGVGKSLVSTTLALVLAEKGYRVGLLDLDFHGASDHVILGFEPKEFPEEDRGVVPPTVHGIKFMTIAYYTTPLRGKEISDALIELLTITRWDELDYLVIDMPPGLGDQLLDVLRFLKRGEFLVVATPSKLSLNVVRKLIELLKEEGHKVIGVVENMKLREKDVEKLAEEFGVPYLVGIPFYPDLDAKVGNVEELMKTEFAGKVRELAGRL 3vxv A 2.0 BS01 dna B 0 R106 S107 K108 R109 R36 S37 K38 R39 3.2.2.- 0003677 remove_due_to_license_issue Q9Z2D7 23316048 1 ~ 14 KPVPCGWERVVKQRLSGKTAGKFDVYFISPQGLKFRSKRSLANYLLKNGETFLKPEDFNFTVLPK 3vxv A 2.0 BS02 dna C 0 K82 R84 L85 S86 G87 K88 T89 K12 R14 L15 S16 G17 K18 T19 3.2.2.- 0003677 remove_due_to_license_issue Q9Z2D7 23316048 1 ~ 14 KPVPCGWERVVKQRLSGKTAGKFDVYFISPQGLKFRSKRSLANYLLKNGETFLKPEDFNFTVLPK 3vxx A 2.204 BS01 dna B 0 R106 S107 K108 R109 R35 S36 K37 R38 3.2.2.- 0003677 remove_due_to_license_issue Q9Z2D7 23316048 1 ~ 14 PVPCGWERVVKQRLSGKTAGKFDVYFISPQGLKFRSKRSLANYLLKNGETFLKPEDFNFTVLP 3vxx A 2.204 BS02 dna C 0 K82 R84 L85 S86 G87 K88 T89 K11 R13 L14 S15 G16 K17 T18 3.2.2.- 0003677 remove_due_to_license_issue Q9Z2D7 23316048 1 ~ 14 PVPCGWERVVKQRLSGKTAGKFDVYFISPQGLKFRSKRSLANYLLKNGETFLKPEDFNFTVLP 3vyb A 2.4 BS01 dna B 0 R106 S107 K108 R109 R35 S36 K37 R38 3.2.2.- 0003677 remove_due_to_license_issue Q9Z2D7 23316048 1 ~ 14 PVPCGWERVVKQRLSGKTAGKFDVYFISPQGLKFRSKRSLANYLLKNGETFLKPEDFNFTVLP 3vyb A 2.4 BS02 dna C 0 K82 R84 L85 S86 G87 K88 T89 K11 R13 L14 S15 G16 K17 T18 3.2.2.- 0003677 remove_due_to_license_issue Q9Z2D7 23316048 1 ~ 14 PVPCGWERVVKQRLSGKTAGKFDVYFISPQGLKFRSKRSLANYLLKNGETFLKPEDFNFTVLP 3vyd A 2.81 BS01 VYD A 1 Q19 D38 G40 S41 Y83 T85 F119 F124 D226 G228 Q19 D38 G40 S41 Y83 T85 F119 F124 D223 G225 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=406nM P00797 23122821 402 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3vye A 2.7 BS01 VYE A 1 Q19 D38 G40 Y83 S84 T85 F119 F124 D226 G228 Q19 D38 G40 Y83 S84 T85 F119 F124 D221 G223 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D221 A224 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=7.7nM P00797 23122821 402 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3vyf A 2.8 BS01 VYF A 1 Q19 D38 G40 S41 Y83 S84 T85 F119 F124 I137 D226 G228 Q19 D38 G40 S41 Y83 S84 T85 F119 F124 I137 D222 G224 D38 S41 N43 W45 Y83 D226 A229 D38 S41 N43 W45 Y83 D222 A225 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=1.6nM P00797 23122821 402 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 3vzd A 2.3 BS01 UUL A 1 F173 I174 V177 D178 T196 M272 F288 F303 M306 H311 F168 I169 V172 D173 T191 M257 F273 F288 M291 H296 2.3.1.-,2.7.1.91 0000287,0001568,0001727,0003376,0003677,0005515,0005516,0005524,0005634,0005654,0005737,0005768,0005829,0005886,0005905,0006473,0006629,0006670,0006954,0007420,0008283,0008284,0008289,0008481,0010008,0010800,0010803,0016020,0016301,0016407,0017050,0019722,0030100,0030139,0030148,0030307,0030335,0031398,0031901,0032651,0032740,0034612,0035556,0035924,0038036,0043066,0043231,0045202,0045766,0045840,0045931,0045987,0046512,0046521,0048146,0050764,0051092,0051721,0070301,0071363,0071897,0090520,0098793,0150077,1900060,1900745,1901224,1903978,1905364 remove_due_to_license_issue Ki=16000nM, IC50=35000nM Q9NYA1 23602659 401 MGSGVLPRPCRVLVLLNPRGGKGKALQLFRSHVQPLLAEAEISFTLMLTERRNHARELVRSEELGRWDALVVMSGDGLMHEVVNGLMERPDWETAIQKPLCSLPAGSGNALAASLNHYAGYEQVTNEDLLTNCTLLLCRRLLSPMNLLSLHTASGLRLFSVLSLAWGFIADVDLESEKYRRLGEMRFTLGTFLRLAALRTYRGRLAYLPVGRVGSQGPVDAHLVPLEEPVPSHWTVVPDEDFVLVLALLHSHLGSEMFAAPMGRCAAGVMHLFYVRAGVSRAMLLRLFLAMEKGRHMEYECPYLVYVPVVAFRLEPKDGKGVFAVDGELMVSEAVQGQVHPNYFWMVSG 3vzd A 2.3 BS02 UUL A 2 F197 L200 A201 R296 A297 F192 L195 A196 R281 A282 2.3.1.-,2.7.1.91 0000287,0001568,0001727,0003376,0003677,0005515,0005516,0005524,0005634,0005654,0005737,0005768,0005829,0005886,0005905,0006473,0006629,0006670,0006954,0007420,0008283,0008284,0008289,0008481,0010008,0010800,0010803,0016020,0016301,0016407,0017050,0019722,0030100,0030139,0030148,0030307,0030335,0031398,0031901,0032651,0032740,0034612,0035556,0035924,0038036,0043066,0043231,0045202,0045766,0045840,0045931,0045987,0046512,0046521,0048146,0050764,0051092,0051721,0070301,0071363,0071897,0090520,0098793,0150077,1900060,1900745,1901224,1903978,1905364 remove_due_to_license_issue Ki=16000nM, IC50=35000nM Q9NYA1 23602659 402 MGSGVLPRPCRVLVLLNPRGGKGKALQLFRSHVQPLLAEAEISFTLMLTERRNHARELVRSEELGRWDALVVMSGDGLMHEVVNGLMERPDWETAIQKPLCSLPAGSGNALAASLNHYAGYEQVTNEDLLTNCTLLLCRRLLSPMNLLSLHTASGLRLFSVLSLAWGFIADVDLESEKYRRLGEMRFTLGTFLRLAALRTYRGRLAYLPVGRVGSQGPVDAHLVPLEEPVPSHWTVVPDEDFVLVLALLHSHLGSEMFAAPMGRCAAGVMHLFYVRAGVSRAMLLRLFLAMEKGRHMEYECPYLVYVPVVAFRLEPKDGKGVFAVDGELMVSEAVQGQVHPNYFWMVSG 3vzg A 2.7 BS01 MAN A 1 G35 Y104 G147 S148 L149 D151 G14 Y83 G126 S127 L128 D130 ? 0005515,0005576,0005615,0005794,0005796,0015031,0030246,0031410,0042589,0042834,0050830,0052373,0062023,0070701 remove_due_to_license_issue O60844 24790092 202 RSSSYSGEYGSGGGKRFSHSGNQLDGPITALRVRVNTYYIVGLQVRYGKVWSDYVGGRNGDLEEIFLHPGESVIQVSGKYKWYLKKLVFVTDKGRYLSFGKDSGTSFNAVPLHPNTVLRFISGRSGSLIDAIGLHWDV 3vzv A 2.8 BS01 VZV A 1 L54 G58 M62 Y67 Q72 V93 H96 Y100 L30 G34 M38 Y43 Q48 V69 H72 Y76 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 23266121 200 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 3w07 A 1.03 BS01 U5P A 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D10 K32 D60 K62 M116 S117 P170 Q175 G192 R193 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Kd=0.00042M remove_due_to_license_issue O26232 23395822 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3w0l B 2.92 BS01 F6R B 1 C107 G108 T109 S179 C180 R259 E347 K513 C104 G105 T106 S176 C177 R256 E340 K506 ? 0004857,0005634,0005654,0005737,0005739,0005829,0009750,0019899,0030246,0033132,0042593,0070095,0097367,1901135 remove_due_to_license_issue Q91754 23733961 701 TRKYQHVIETPDPGKWELAGYEESLPISEKSNPMTRELDKADPSQLVQLLRDCDAEIFQEEDENLIHYHRLYSESVLKTMGDVAKRVQEVLKNPDDSLVVLSGCGTSGRLALLLANSFNGLLKGLHKTPCYCYIMSGGDRSIVTSQESSEDNPQLGAQELEKVCEGKKNVLFIGISCGLSAPFIAGQLDFCMRHLDVYLPVLVGFNPVSMARNERIEGWHSSFRQVAERLQTLHDSQKGFILNPAVGPEGVSGSSRMKGGSATKILLETLLLVAHKAEVTEKCLLEILRTYERAHKVTYSQSKKIAALMKQTATSLQKKGHLYILGWGTLGLVGIMDAVECVPTYQADWRDVRGFITGGYHSIENKEGDLSSLGPQFSISHEDFVKNVLPSVSETDTVLLIFTLDDDLNQIEKLVALVKEKTSNIQVICHATAGQYLPNSLKKTIPSIIGLTWPILFLEYEGAFIQKFQRELSTKWILDTVTSGAYTLRGKIFRNFMVDFKINNSKLFHRATSVLQRLTGQSQQRCTEVLLQSIYGEQTLSEQIRNTTIAGHVEAAASQDKVLPVAIVSLLRSCTIQDSRSRINSSLSIRSAIESSMN 3w1f A 2.7 BS01 1O5 A 1 K529 I531 Q541 A551 K553 M602 E603 C604 G605 N606 L654 I663 K14 I16 Q26 A36 K38 M87 E88 C89 G90 N91 L139 I148 D647 K649 N652 D664 D674 T686 D132 K134 N137 D149 D159 T161 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=198nM P33981 23634759 901 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMSISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 3w1k A 7.5 BS01 rna G 0 K2 L5 R6 I8 Q10 I11 S12 K13 V28 R32 R39 K2 L5 R6 I8 Q10 I11 S12 K13 V28 R32 R39 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w1k B 7.5 BS01 rna F 0 R6 I8 P9 Q10 I11 S12 K13 E16 R32 R39 R6 I8 P9 Q10 I11 S12 K13 E16 R32 R39 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w1k C 7.5 BS01 rna G 0 Q405 I422 R423 E424 Q405 I422 R423 E424 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w1k C 7.5 BS02 rna H 0 K257 S262 K257 S262 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w1k C 7.5 BS03 rna I 0 K2 L5 R6 I8 P9 Q10 I11 S12 E16 V28 R32 R39 K2 L5 R6 I8 P9 Q10 I11 S12 E16 V28 R32 R39 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w1k D 7.5 BS01 rna H 0 K2 L5 R6 I8 P9 Q10 I11 S12 E16 V28 R32 R39 K2 L5 R6 I8 P9 Q10 I11 S12 E16 V28 R32 R39 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w1k E 7.5 BS01 rna I 0 Q405 I422 Q405 I422 2.9.1.1 0001514,0001717,0004125,0005737,0006412,0016740,0042802 remove_due_to_license_issue O67140 23559248 1 ~ 73 MKSLLRQIPQISKVVEIFAKAYPEIYVVKAAREVAEKYRKEIIEGARADLNGFLEDVERKIKSLMKPNIKRVINATGVVINTNLGRAPLSKDVINFISEIANGYSNLEYNLEEGKRGSRIAHIEKYLNELTGAESSFVVNNNAGAVFLVLNTLAEGKEVIISRGELVEIGGSFRIPDIMKKSGAILREVGTTNKTKVSDYEGAINQNTALLMKVHKSNFYMEGFVEEVKLEDLVKLGHKYGIPTYYDAGSGLLINLKEFGISVDEPNFRDCISLGIDLVSGSGDKLLGGPQAGIIVGKKNLIEKIKKNPIARALRIDKLTLSGLEMTLKLYFEKRYEDIPVIRMLTQDEKALRQKAKRLEKLLKDIPGLKISVIKDKAKPGGGSLPELELPTYCVAIRHDRLSSQELSRRLRLAEPPIVCRIREDQLLFDMRTVFHEDLKTIKKTLQELLSI 3w2o A 2.35 BS01 03P A 1 S720 G721 V726 A743 K745 E762 M766 L788 M790 M793 S24 G25 V30 A47 K49 E66 M70 L92 M94 M97 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=4.0nM P00533 24900643 1101 HAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPMDDVVDADEYL 3w2p A 2.05 BS01 W2P A 1 L718 V726 A743 K745 I759 E762 M766 L788 M790 M793 C797 L22 V30 A47 K49 I63 E66 M70 L92 M94 M97 C101 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 24900643 1101 HAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSDMDDVVDADEYLI 3w2q A 2.2 BS01 HKI A 1 A743 K745 I759 E762 A763 M790 M793 P794 G796 C797 D800 L844 A47 K49 I63 E66 A67 M94 M97 P98 G100 C101 D104 L148 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 24900643 1101 HAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPMDDVVDADEYL 3w2r A 2.05 BS01 W2R A 1 F723 V726 A743 K745 M766 C775 L788 M790 M793 L844 T854 D855 F856 R858 F997 F26 V29 A46 K48 M69 C78 L91 M93 M96 L147 T157 D158 F159 R161 F277 D837 A839 R841 N842 D855 D140 A142 R144 N145 D158 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=6.9nM P00533 24900643 1101 APNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDESNFYRALMDEEDMDDVVDADEYL 3w2s A 1.9 BS01 W2R A 1 V726 A743 K745 M766 L788 T790 M793 R841 L844 T854 D855 F856 G857 V26 A43 K45 M66 L88 T90 M93 R141 L144 T154 D155 F156 G157 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=6.9nM P00533 24900643 1101 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDADEYLIP 3w2t A 2.36 BS01 LF7 A 1 E205 E206 Y547 S630 Y631 Y662 Y666 V711 E168 E169 Y510 S593 Y594 Y625 Y629 V674 Y547 S630 Y631 D708 H740 Y510 S593 Y594 D671 H703 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=3.5nM P27487 23501107 801 DSRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3w32 A 1.8 BS01 W32 A 1 A743 K745 C775 R776 L788 T790 M793 L844 T854 D855 F856 F997 A43 K45 C75 R76 L88 T90 M93 L144 T154 D155 F156 F297 D837 A839 R841 N842 D855 G874 D137 A139 R141 N142 D155 G174 2.7.10.1 0004672,0004713,0005524,0006468 ic50=75nM remove_due_to_license_issue IC50=75nM P00533 23490150 1101 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDADEYL 3w33 A 1.7 BS01 W19 A 1 A743 K745 C775 L777 L788 T790 M793 G796 L844 T854 D855 F856 L858 A43 K45 C70 L72 L83 T85 M88 G91 L139 T149 D150 F151 L153 D837 A839 R841 N842 D855 D132 A134 R136 N137 D150 2.7.10.1 0004672,0004713,0005524,0006468 ic50=36nM remove_due_to_license_issue IC50=36nM P00533 23490150 1101 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDDDVVDADEYLI 3w3c A 2.431 BS01 dna B 0 S150 Y151 K152 R162 T166 S20 Y21 K22 R32 T36 ? 0003677 remove_due_to_license_issue P0A247 23985969 1 ~ 26 EHSIRELGIGLNFLKVSGMSYKDIAKKENLSRAKVTRAFQAASVPQEIISLFPIASELNFNDYKILFNYYKGLEKANESLSSTLPILKEEIKDLDTNLPPDIYKKEILNIIKKSKN 3w3c A 2.431 BS02 dna C 0 K164 R167 N189 F190 K34 R37 N59 F60 ? 0003677 remove_due_to_license_issue P0A247 23985969 1 ~ 26 EHSIRELGIGLNFLKVSGMSYKDIAKKENLSRAKVTRAFQAASVPQEIISLFPIASELNFNDYKILFNYYKGLEKANESLSSTLPILKEEIKDLDTNLPPDIYKKEILNIIKKSKN 3w54 A 2.3 BS03 RNB A 1 V92 C95 R96 R118 L122 M190 L212 A216 T219 V61 C64 R65 R87 L91 M159 L181 A185 T188 1.-.-.- 0005739,0005743,0008199,0009916,0010230,0016491,0046872 ic50=0.2nM remove_due_to_license_issue IC50=4.0nM Q26710 23487766 504 VWGHTQLNRLSFLETVPVVPLRVSDESSEDRPTWSLPDIENVAITHKKPNGLVDTLAYRSVRTCRWLFDTFSLYRFGSITESKVISRCLFLETVAGVPGMVGGMLRHLSSLRYMTRDKGWINTLLVEAENERMHLMTFIELRQPGLPLRVSIIITQAIMYLFLLVAYVISPRFVHRFVGYLEEEAVITYTGVMRAIDEGRLRPTKNDVPEVARVYWNLSKNATFRDLINVIRADEAEHRVVNHTFADMHEKRLQNSVNPFVVLK 3w55 A 3.0 BS01 1FM A 1 I31 V39 K54 M108 S153 N154 L156 C166 I21 V29 K44 M98 S143 N144 L146 C156 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T168 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue IC50=738nM P28482 17194451 401 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 3w5e A 2.3 BS01 NVW A 1 Y233 N395 T407 I410 F414 S442 Q443 F446 L502 M503 F506 Y80 N242 T254 I257 F261 S289 Q290 F293 L336 M337 F340 3.1.4.53 0004114,0007165,0008081 ic50=11nM remove_due_to_license_issue IC50=11nM Q07343 23602400 901 SRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPCQGLMEKFQFELT 3w5t A 2.29 BS02 LHP A 1 Y143 A227 I267 S271 S274 W282 V296 H301 H393 V414 Y21 A47 I87 S91 S94 W102 V116 H121 H213 V234 ? 0003677,0004879,0006355 remove_due_to_license_issue P13053 23723390 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNEI 3w69 A 1.9 BS01 LTZ A 1 L54 G58 I61 M62 Y67 Q72 V93 H96 Y100 L30 G34 I37 M38 Y43 Q48 V69 H72 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.058uM remove_due_to_license_issue Q00987 23685175 201 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVV 3w6v A 2.95 BS01 dna B 0 D249 V250 R261 R262 D265 R269 A275 L277 D20 V21 R32 R33 D36 R40 A46 L48 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9S166 24019524 -3 ~ 12 SDPLAEVVAWALEHLHEQFDVETLAARAYMSRRTFDRRFRSLTGSAPLQWLITQRVLQAQRLLETSDYSVDEVAGRCGFRSPVALRGHFRRQLGSSPAAYRAAYRARRPQG 3w6v A 2.95 BS02 dna C 0 S260 R262 T263 R266 R309 H317 S31 R33 T34 R37 R80 H88 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9S166 24019524 -3 ~ 12 SDPLAEVVAWALEHLHEQFDVETLAARAYMSRRTFDRRFRSLTGSAPLQWLITQRVLQAQRLLETSDYSVDEVAGRCGFRSPVALRGHFRRQLGSSPAAYRAAYRARRPQG 3w8o A 1.85 BS01 WPC A 1 H32 P34 V37 T43 Y56 Y75 F78 H83 L85 R129 V137 Y138 M141 H32 P34 V37 T43 Y56 Y75 F78 H83 L85 R129 V137 Y138 M141 ? 0046872 remove_due_to_license_issue G3XD33 24604808 201 MSISISYSTTYSGWTVADYLADWSAYFGDVNHRPGQVVDGSNTGGFNPGPFDGSQYALKSTASDAAFIAGGDLHYTLFSNPSHTLWGKLDSIALGDTLTGGASSGGYALDSQEVSFSNLGLDSPIAQGRDGTVHKVVYGLMSGDSSALQGQIDALLKAVDPSLSINSTFDQLAAAGVAHATPAA 3w9k A 1.8 BS01 MYR A 1 F32 Y57 T104 A105 K109 F31 Y56 T103 A104 K108 ? Kd=0.48uM remove_due_to_license_issue Q973T5 23836863 201 MKVEKEIKTNQDIDVVMTIFSDPAFTIPQIFPGIASIKCIEPEIFEAEGKFLAFSYKVKGRVYKGVDEVRIIYDSDRGNGILYIRKKDNNTLQIILEHDNKLTAFLGKPYVSSNLDRLAENIDEIIRLERIKRKI 3w9r A 1.9 BS01 A8S A 1 K63 S94 L165 N169 K51 S82 L153 N157 ? 0004864,0005515,0005634,0005737,0005886,0009738,0010427,0038023,0042803 Kd=0.66uM remove_due_to_license_issue Q84MC7 24645846 201 GGLETVQYVRTHHQHLCRENQCTSALVKHIKAPLHLVWSLVRRFDQPQKYKPFVSRCTVIGDPEIGSLREVNVKSGLPATTSTERLELLDDEEHILGIKIIGGDHRLKNYSSILTVHPEIIEGRAGTMVIESFVVDVPQGNTKDETCYFVEALIRCNLKSLADVSERLASQ 3wab A 2.154 BS03 DDW A 1 H69 R127 N144 R145 H196 S207 Y248 D255 E270 H64 R122 N139 R140 H192 S203 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 remove_due_to_license_issue IC50=3.6nM P09955 24010887 403 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 3wav A 1.797 BS05 DWV A 1 L213 F273 F274 W275 Y306 L163 F223 F224 W225 Y256 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 ic50=180nM remove_due_to_license_issue IC50=180nM Q9R1E6 23688339 937 WTNTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPLDVYKKCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCDDKNKLEELNKRLHTKGSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 3waw A 1.954 BS05 DWW A 1 S169 F210 L213 F273 F274 W275 Y306 S119 F160 L163 F223 F224 W225 Y256 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 ic50=580nM remove_due_to_license_issue IC50=580nM Q9R1E6 23688339 937 WTNTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCDSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 3wax A 1.899 BS05 DWX A 1 D171 T209 L213 N230 L243 F273 F274 W275 Y306 D311 H474 D121 T159 L163 N180 L193 F223 F224 W225 Y256 D261 H414 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 ic50=13nM remove_due_to_license_issue IC50=13nM Q9R1E6 23688339 936 WTNTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCDDLEELNHTKGSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 3way A 1.746 BS05 DWY A 1 D171 T209 L213 F273 F274 W275 Y306 D311 H359 H474 D121 T159 L163 F223 F224 W225 Y256 D261 H309 H414 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 remove_due_to_license_issue IC50=22nM Q9R1E6 23688339 931 WTNTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCDDLEEHTKGSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 3wb4 A 2.25 BS01 0B3 A 1 L30 D32 Y71 D228 L32 D34 Y73 D220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 Kd=36.6uM remove_due_to_license_issue IC50=34000nM P56817 24051074 507 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAAEKFPDGFWLGEQLVCWQANIFPVISLYLMGEVTNQSFRITILPQQYLRPVCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3wb5 A 2.501 BS01 0B4 A 1 D32 Y71 F108 D228 D34 Y73 F110 D219 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 Kd=26.8uM remove_due_to_license_issue P56817 24051074 507 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGWNIFPVISLYLMGEVTNQSFRITILPQQYLRPYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDFRTAAVEGPFVTLDMEDCGYN 3wbl A 2.0 BS01 PDY A 1 I10 G13 V18 A31 L83 H84 Q85 N132 L134 D145 I10 G13 V18 A30 L77 H78 Q79 N126 L128 D139 D127 K129 Q131 N132 D145 T165 D121 K123 Q125 N126 D139 T150 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=23uM remove_due_to_license_issue IC50=23000nM P24941 24121337 302 MENFQKVEKIGEGTYGVVYKARNKTGEVVALKKIRLGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 3wc5 A 1.7 BS03 DDK A 1 H69 E72 R127 N144 R145 H196 S207 Y248 D255 E270 H64 E67 R122 N139 R140 H192 S203 Y244 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 remove_due_to_license_issue P09955 24010887 403 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 3wc7 A 1.9 BS03 EF1 A 1 H69 E72 R127 N144 R145 H196 S197 Y198 S207 I247 Y248 D255 E270 F279 H64 E67 R122 N139 R140 H192 S193 Y194 S203 I243 Y244 D251 E266 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 remove_due_to_license_issue IC50=4.9nM P09955 24010887 403 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 3wcb A 3.0 BS01 8PH A 1 S42 S44 F45 Y64 G172 M199 L203 S15 S17 F18 Y37 G145 M172 L176 Y163 R210 R222 F282 Y136 R183 R195 F255 2.5.1.21 0008610,0009058,0016765,0045338,0051996 remove_due_to_license_issue Q4CWB4 24789335 401 DEDLRFCYDILQAVSRSFAVVIMELDEEMRDAVCIFYLVLRALDTVEDDMSIPVEFKLRELPKFHEHLHDTTWCMSGVGVGRERELLERYTHVTRAYSRLGKAYQDVISGICERMANGMCDFLTRKVETKADYDLYCHYVAGLVGHGLTLLYVSSGLEDVRLADDLTNANHMGLFLQKTNIIRDFYEDICEVPPRVFWPREIWEKYTDDLHAFKDELHEAKAVECLNAMVADALVHVPHVVEYLASLRDPSVFTFSAIPQVMAMATLSLVFNNKDVFHTKVKTTRGATARIFHYSTELQATLQMLKTYTLRLAARMNAQDACYDRIEHLVNDAIRAMESHQ 3wcf A 2.22 BS01 BH8 A 1 R77 D80 G180 M207 L211 N215 R42 D45 G145 M172 L176 N180 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.053uM remove_due_to_license_issue P37268 24789335 401 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wcg A 2.8 BS01 BH3 A 1 S42 S44 Y64 R68 D71 V171 L175 L203 S15 S17 Y37 R41 D44 V144 L148 L176 Y163 R210 R222 F282 Y136 R183 R195 F255 2.5.1.21 0008610,0009058,0016765,0045338,0051996 remove_due_to_license_issue Q4CWB4 24789335 401 DEDLRFCYDILQAVSRSFAVVIMELDEEMRDAVCIFYLVLRALDTVEDDMSIPVEFKLRELPKFHEHLHDTTWCMSGVGVGRERELLERYTHVTRAYSRLGKAYQDVISGICERMANGMCDFLTRKVETKADYDLYCHYVAGLVGHGLTLLYVSSGLEDVRLADDLTNANHMGLFLQKTNIIRDFYEDICEVPPRVFWPREIWEKYTDDLHAFKDELHEAKAVECLNAMVADALVHVPHVVEYLASLRDPSVFAFSAIPQVMAMATLSLVFNNKDVFHTKVKTTRGATARIFHYSTELQATLQMLKTYTLRLAARMNAQDACYDRIEHLVNDAIRAMESHQ 3wch A 2.5 BS01 8PH A 1 R77 D80 D84 A176 G180 M207 Q212 R42 D45 D49 A141 G145 M172 Q177 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.089uM remove_due_to_license_issue P37268 24789335 401 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wch A 2.5 BS02 8PH A 2 F54 Y73 F19 Y38 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.089uM remove_due_to_license_issue P37268 24789335 402 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wch A 2.5 BS03 8PH A 3 S51 R52 S53 N215 S16 R17 S18 N180 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.089uM remove_due_to_license_issue P37268 24789335 403 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wci A 2.3 BS01 BH5 A 1 T50 S51 R52 Y73 R77 D80 V179 L211 T15 S16 R17 Y38 R42 D45 V144 L176 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.27uM remove_due_to_license_issue P37268 24789335 401 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wci C 2.3 BS01 BH5 C 1 R52 S53 Y73 R77 V179 L211 Y276 R17 S18 Y38 R42 V144 L176 Y241 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.27uM remove_due_to_license_issue P37268 24789335 401 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wcl A 2.24 BS01 BH3 A 1 S51 R52 S53 Y73 R77 D80 V179 M207 L211 S16 R17 S18 Y38 R42 D45 V144 M172 L176 Y171 R218 R228 F288 Y136 R183 R193 F253 2.5.1.21 0008610,0009058,0016765,0045338,0051996 ic50=0.26uM remove_due_to_license_issue P37268 24789335 401 LSSSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFALPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVLIRLGQAVTLMMDATNMPAVKAIIYQYMEEIYHRIPDSNPSSSKTRQIISTIRTQ 3wd1 A 2.3 BS01 ST7 A 1 Y10 F12 W97 D142 E144 M212 Y214 D215 P219 W220 Y292 R294 R338 I339 W403 Y9 F11 W96 D141 E143 M211 Y213 D214 P218 W219 Y291 R293 R337 I338 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 ic50=0.022uM remove_due_to_license_issue IC50=22nM P11797 24043811 514 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRL 3wd2 A 2.2 BS01 A1L A 1 Y10 W97 D142 E144 M212 Y214 D215 P219 R294 D316 R338 W403 Y9 W96 D141 E143 M211 Y213 D214 P218 R293 D315 R337 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 ic50=0.58uM remove_due_to_license_issue P11797 24043811 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRL 3wd9 A 2.5 BS01 QPC A 1 S282 N395 F414 S442 Q443 F446 L502 M503 F506 S129 N242 F261 S289 Q290 F293 L336 M337 F340 3.1.4.53 0004114,0007165,0008081 ic50=8.3nM remove_due_to_license_issue IC50=8.3nM Q07343 24094436 901 SRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPCQGLMEKFQFELT 3we4 A 1.995 BS02 5FI A 1 K99 G100 G103 V105 A121 K123 L125 E173 Y174 L175 M225 K241 K15 G16 G19 V21 A37 K39 L41 E89 Y90 L91 M141 K157 D218 K220 E222 N223 D236 T256 D134 K136 E138 N139 D152 T169 2.7.11.1 0004672,0004674,0005524,0006468 ic50=15nM remove_due_to_license_issue Ki=20nM, IC50=160nM P23443 25078151 402 KIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLLQ 3wf5 A 2.099 BS02 FZ8 A 1 K99 G100 V105 A121 E173 L175 K241 K15 G16 V21 A37 E77 L79 K145 D218 K220 E222 N223 D236 T256 D122 K124 E126 N127 D140 T160 2.7.11.1 0004672,0004674,0005524,0006468 ic50=81nM remove_due_to_license_issue P23443 25078151 402 KIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDGTVTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLLQ 3wf6 A 2.031 BS02 FZ9 A 1 G98 G100 V105 A121 E173 L175 M225 K241 G14 G16 V21 A37 E77 L79 M129 K145 D218 K220 E222 N223 D236 T256 D122 K124 E126 N127 D140 T160 2.7.11.1 0004672,0004674,0005524,0006468 ic50=33nM remove_due_to_license_issue P23443 25078151 402 KIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDGTVTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLLQ 3wf7 A 1.85 BS02 FS9 A 1 K99 G100 Y102 G103 K104 V105 A121 K123 L125 E173 L175 M225 K241 K17 G18 Y20 G21 K22 V23 A39 K41 L43 E91 L93 M143 K159 D218 K220 E222 N223 D236 T256 D136 K138 E140 N141 D154 T171 2.7.11.1 0004672,0004674,0005524,0006468 ic50=206nM remove_due_to_license_issue P23443 25078151 402 PEKIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLLQ 3wf8 A 1.975 BS02 F76 A 1 L97 K99 G100 Y102 G103 V105 L175 K241 L13 K15 G16 Y18 G19 V21 L91 K157 D218 K220 E222 N223 D236 T256 D134 K136 E138 N139 D152 T172 2.7.11.1 0004672,0004674,0005524,0006468 ic50=232nM remove_due_to_license_issue P23443 25078151 402 KIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDGTVTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPL 3wf9 A 2.035 BS02 FS7 A 1 L97 K99 G100 Y102 G103 L175 K241 L13 K15 G16 Y18 G19 L91 K157 D218 K220 E222 N223 D236 T256 D134 K136 E138 N139 D152 T172 2.7.11.1 0004672,0004674,0005524,0006468 ic50=567nM remove_due_to_license_issue P23443 25078151 402 KIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDGTVTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPL 3wff A 2.05 BS01 WFF A 1 N770 A773 M807 S811 L814 F829 M845 M852 L938 F941 C942 T945 N44 A47 M81 S85 L88 F103 M119 M126 L212 F215 C216 T219 ? remove_due_to_license_issue IC50=660nM P08235 23958516 1001 LSTISRALTPSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKCPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNVKPLYFHRK 3wfg A 1.4 BS01 WFG A 1 L769 N770 A773 M807 L814 F829 M845 M852 L938 F941 C942 T945 L35 N36 A39 M73 L80 F95 M111 M118 L204 F207 C208 T211 ? remove_due_to_license_issue IC50=120nM P08235 23958516 1001 TPSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKCPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNVKPLYFHR 3wgg A 2.1 BS01 8NA A 1 I90 G93 N94 L95 D117 I118 I154 P155 F177 P179 I87 G90 N91 L92 D114 I115 I151 P152 F174 P176 ? 0000166,0003677,0003700,0005737,0006355,0045892,0046872,0051775 remove_due_to_license_issue D5KM69 25527330 301 KTIVSMAVIRRLPRYHRYLEELLKNDVKRISSRELSEKMGVTASQIRQDLNNFGGFGQQGYGYNVEELYNNLTKILGLDKTYNTIIIGAGNLGQAIANYTSFEKSGFNLKGIFDINPRLFGLKIRDVEVMDVETVEDFIARNKIDIGILCIPKDNAQYTADRLVRAGIKAIWNFLPIDLKVPDDVILENVHLSDSLFTVSYRLNEEELFKKLK 3wgg A 2.1 BS05 8NA B 1 N101 Y102 S104 N98 Y99 S101 ? 0000166,0003677,0003700,0005737,0006355,0045892,0046872,0051775 remove_due_to_license_issue D5KM69 25527330 301 KTIVSMAVIRRLPRYHRYLEELLKNDVKRISSRELSEKMGVTASQIRQDLNNFGGFGQQGYGYNVEELYNNLTKILGLDKTYNTIIIGAGNLGQAIANYTSFEKSGFNLKGIFDINPRLFGLKIRDVEVMDVETVEDFIARNKIDIGILCIPKDNAQYTADRLVRAGIKAIWNFLPIDLKVPDDVILENVHLSDSLFTVSYRLNEEELFKKLK 3wgg B 2.1 BS01 8NA A 1 N101 Y102 S104 N98 Y99 S101 ? 0000166,0003677,0003700,0005737,0006355,0045892,0046872,0051775 remove_due_to_license_issue D5KM69 25527330 301 KTIVSMAVIRRLPRYHRYLEELLKNDVKRISSRELSEKMGVTASQIRQDLNNFGGFGQQGYGYNVEELYNNLTKILGLDKTYNTIIIGAGNLGQAIANYTSFEKSGFNLKGIFDINPRLFGLKIRDVEVMDVETVEDFIARNKIDIGILCIPKDNAQYTADRLVRAGIKAIWNFLPIDLKVPDDVILENVHLSDSLFTVSYRLNEEELFKKLK 3wgg B 2.1 BS03 8NA B 1 G93 N94 L95 D117 I118 I154 P155 F177 P179 G90 N91 L92 D114 I115 I151 P152 F174 P176 ? 0000166,0003677,0003700,0005737,0006355,0045892,0046872,0051775 remove_due_to_license_issue D5KM69 25527330 301 KTIVSMAVIRRLPRYHRYLEELLKNDVKRISSRELSEKMGVTASQIRQDLNNFGGFGQQGYGYNVEELYNNLTKILGLDKTYNTIIIGAGNLGQAIANYTSFEKSGFNLKGIFDINPRLFGLKIRDVEVMDVETVEDFIARNKIDIGILCIPKDNAQYTADRLVRAGIKAIWNFLPIDLKVPDDVILENVHLSDSLFTVSYRLNEEELFKKLK 3wgw A 2.8 BS01 T2B A 1 M40 L47 E124 G127 P129 P234 Y250 M40 L47 E124 G127 P129 P227 Y243 ? 0000122,0000307,0000701,0000781,0000785,0001673,0003677,0003682,0003684,0005515,0005634,0005652,0005654,0005657,0005813,0006260,0006272,0006275,0006281,0006287,0006298,0006979,0007507,0016604,0019899,0019985,0030331,0030337,0030855,0030894,0030971,0031297,0032077,0032139,0032355,0032405,0033993,0034644,0035035,0042802,0043596,0043626,0044849,0044877,0045739,0045740,0046686,0070062,0070182,0070301,0070557,0071466,0071548,0097421,1900264,1902065,1902990 remove_due_to_license_issue IC50=1300nM P12004 24474685 301 MFEARLVQGSILKKVLEALKDLINEACWDISSSGVNLQSMDSSHVSLVQLTLRSEGFDTYRCDRNLAMGVNLTSMSKILKCAGNEDIITLRAEDNADTLALVFEAPNQEKVSDYEMKLMDLDVEQLGIPEQEYSCVVKMPSGEFARICRDLSHIGDAVVISCAKDGVKFSASGELGNGNIKLSQTEAVTIEMNEPVQLTFALRYLNFFTKATPLSSTVTLSMSADVPLVVEYKIADMGHLKYYLAPKI 3wgw A 2.8 BS02 T2B A 2 D165 K181 L182 S183 D165 K181 L182 S183 ? 0000122,0000307,0000701,0000781,0000785,0001673,0003677,0003682,0003684,0005515,0005634,0005652,0005654,0005657,0005813,0006260,0006272,0006275,0006281,0006287,0006298,0006979,0007507,0016604,0019899,0019985,0030331,0030337,0030855,0030894,0030971,0031297,0032077,0032139,0032355,0032405,0033993,0034644,0035035,0042802,0043596,0043626,0044849,0044877,0045739,0045740,0046686,0070062,0070182,0070301,0070557,0071466,0071548,0097421,1900264,1902065,1902990 remove_due_to_license_issue IC50=1300nM P12004 24474685 303 MFEARLVQGSILKKVLEALKDLINEACWDISSSGVNLQSMDSSHVSLVQLTLRSEGFDTYRCDRNLAMGVNLTSMSKILKCAGNEDIITLRAEDNADTLALVFEAPNQEKVSDYEMKLMDLDVEQLGIPEQEYSCVVKMPSGEFARICRDLSHIGDAVVISCAKDGVKFSASGELGNGNIKLSQTEAVTIEMNEPVQLTFALRYLNFFTKATPLSSTVTLSMSADVPLVVEYKIADMGHLKYYLAPKI 3wha A 1.3 BS01 WHA A 1 A55 K58 I96 G97 M98 N106 L107 F138 Y139 A40 K43 I81 G82 M83 N91 L92 F123 Y124 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.48nM remove_due_to_license_issue Kd=0.480000nM P07900 24369839 302 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 3whw A 2.701 BS01 RUX A 1 Y7 T8 L9 F27 N33 G34 G36 G37 K38 M81 D119 D120 Y5 T6 L7 F25 N31 G32 G34 G35 K36 M79 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue P36639 24258965 204 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 3wi2 A 2.26 BS02 P98 A 1 I692 Y693 F696 P712 M713 E721 G725 Q726 F729 I246 Y247 F250 P266 M267 E275 G279 Q280 F283 3.1.4.17 0004114,0007165,0008081 ic50=92nM remove_due_to_license_issue Q9Y233 24238902 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 3wi6 A 2.99 BS01 YRZ A 1 A91 E139 L141 E190 N191 L193 D207 A46 E94 L96 E142 N143 L145 D159 D186 K188 E190 N191 D207 S216 D138 K140 E142 N143 D159 S168 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P49137 24316826 901 FHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILKLTDFGFAKETTSPYYVAPEVLGPEDKSCDMWSLGVIMYILLCGYPPFYSISPGMKTRIRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKE 3wig A 2.7 BS03 CHU A 1 L119 V128 I142 M144 R190 D191 C208 D209 F210 G211 V212 L216 I217 M220 N222 L55 V64 I78 M80 R126 D127 C144 D145 F146 G147 V148 L152 I153 M156 N158 D191 K193 S195 N196 D209 D218 T227 D127 K129 S131 N132 D145 D154 T163 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue Q02750 24746704 403 MELKDDDFEKISELGAGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIG 3wix A 1.9 BS01 LC3 A 1 A227 F228 M250 V253 F254 R263 T266 L267 F270 I294 A56 F57 M79 V82 F83 R92 T95 L96 F99 I123 ? 0042981 ic50=0.54uM remove_due_to_license_issue IC50=540nM Q07820 24215352 501 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 3wix A 1.9 BS02 LC3 C 1 P198 M199 R201 S202 R207 P27 M28 R30 S31 R36 ? 0042981 ic50=0.54uM remove_due_to_license_issue IC50=540nM Q07820 24215352 501 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 3wiy A 2.15 BS01 LC6 A 1 A227 F228 G230 M231 K234 M250 V253 R263 T266 L267 F270 A56 F57 G59 M60 K63 M79 V82 R92 T95 L96 F99 ? 0042981 ic50=0.61uM remove_due_to_license_issue IC50=610nM Q07820 24215352 501 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVED 3wiz A 2.45 BS01 LC6 A 1 E96 F97 Y101 L108 E129 L130 W137 G138 R139 V141 E41 F42 Y46 L53 E74 L75 W82 G83 R84 V86 ? 0042981 ic50=0.0044uM remove_due_to_license_issue IC50=4.4nM Q07817 24215352 501 QSNRELVVDFLSYKLSQKGYSWSQFTESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 3wiz B 2.45 BS01 LC6 B 1 E96 F97 Y101 F105 L108 W137 G138 R139 F146 E41 F42 Y46 F50 L53 W82 G83 R84 F91 ? 0042981 ic50=0.0044uM remove_due_to_license_issue IC50=4.4nM Q07817 24215352 501 QSNRELVVDFLSYKLSQKGYSWSQFTESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 3wjw A 1.59 BS01 U6M A 1 D20 K42 D70 K72 M126 S127 P180 Q185 G202 R203 D10 K32 D60 K62 M116 S117 P170 Q175 G192 R193 K42 D70 K72 D75 K32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=134uM remove_due_to_license_issue Ki=134000nM O26232 24151964 301 VMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESIKDL 3wk4 A 2.11 BS02 S0A A 1 F267 D335 W336 Y383 Y466 F266 D334 W335 Y382 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=7.4uM remove_due_to_license_issue IC50=7400nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wk5 A 2.77 BS02 S0C A 1 D335 W336 Y383 Y466 H524 D334 W335 Y382 Y465 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=15000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wk6 A 2.1 BS02 S0B A 1 D335 W336 Y383 L408 Y466 D334 W335 Y382 L407 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=6.3uM remove_due_to_license_issue IC50=6300nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wk7 A 2.2 BS02 S0D A 1 D335 W336 Y383 Y466 W525 D334 W335 Y382 Y465 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=127uM remove_due_to_license_issue IC50=127000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wk8 A 2.2 BS02 S0E A 1 F267 L408 M419 D496 V498 H524 F266 L407 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=49uM remove_due_to_license_issue IC50=49000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wk9 A 2.2 BS02 S0F A 1 F267 Y383 L408 M419 L428 D496 V498 H524 F266 Y382 L407 M418 L427 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=70uM remove_due_to_license_issue IC50=70000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wka A 2.01 BS02 S0G A 1 F267 M419 V498 H524 W525 F266 M418 V497 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=29uM remove_due_to_license_issue IC50=29000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wkb A 2.2 BS02 S0I A 1 W336 Y343 Q384 Y466 M469 N472 W335 Y342 Q383 Y465 M468 N471 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=61uM remove_due_to_license_issue IC50=61000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wkc A 2.2 BS02 S0J A 1 D335 W336 I375 D334 W335 I374 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=195uM remove_due_to_license_issue IC50=195000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wkd A 2.48 BS02 S0K A 1 W336 Y343 A365 Y466 M469 N472 W473 W335 Y342 A364 Y465 M468 N471 W472 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=171uM remove_due_to_license_issue IC50=171000nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wke A 2.75 BS02 AUB A 1 F267 D335 W336 Y383 M419 Y466 W525 F266 D334 W335 Y382 M418 Y465 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=1.5nM, Ki=1.5nM P34913 24656800 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 3wmb A 2.7 BS01 NF1 A 1 D367 W424 W448 Y475 W490 D345 W402 W426 Y453 W468 D367 E368 D345 E346 3.2.1.52 0000272,0004553,0004563,0005886,0005975,0006032,0016231,0016798,0030203 remove_due_to_license_issue Q06GJ0 25155420 601 EDVVWRWSCDNGKCVKLKNDPRSSEPALSLEACKMFCNEYGLLWPRPTGEADLGNFLSKINLNSIEVKILKKGATDDLMEAAAKRFKEQVSLAIPRGSTPKLTGKAVDVYLVNENPNEKAFSLEMDESYGLRVSPSGADRVNATITANSFFGMRHGLETLSQLFVFDDIRDHLLMVRDVNISDKPVYPYRGILLDTARNYYSIESIKRTIEAMAAVKLNTLHWHITDSQSFPFVTTKRPNLYKFGALSPQKVYTKAAIREVVRFGLERGVRVLPEFDAPAHVGEGWQDTDLTVCFKAEPWKSYCVEPPCGQLNPTKDELYQYLEDIYSDMAEVFDTTDIFHMGGDEVSEACWNSSDSIQNFMMQNRWDLDKESFLKLWNYFQQKAQDKAYKAFGKKLPLILWTSTLTNYKHIDDYLNKDDYIIQVWTTGVDPQIKGLLEKGYRLIMSNYDALYFDCGYGAWVGAGNNWCSPYIGWQKVYDNSPAVIALEHRDQVLGGEAALWSEQSDTSTLDGRLWPRAAALAERLWAEPATSWQDAEYRMLHIRERFVRMGIQAESLQPEWCYQNEGYCYS 3wmc A 2.095 BS01 NF6 A 1 V327 D367 E368 W424 W448 Y475 W490 W524 V305 D345 E346 W402 W426 Y453 W468 W502 D367 E368 D345 E346 3.2.1.52 0000272,0004553,0004563,0005886,0005975,0006032,0016231,0016798,0030203 Ki=0.31uM remove_due_to_license_issue Q06GJ0 25155420 601 EDVVWRWSCDNGKCVKLKNDPRSSEPALSLEACKMFCNEYGLLWPRPTGEADLGNFLSKINLNSIEVKILKKGATDDLMEAAAKRFKEQVSLAIPRGSTPKLTGKAVDVYLVNENPNEKAFSLEMDESYGLRVSPSGADRVNATITANSFFGMRHGLETLSQLFVFDDIRDHLLMVRDVNISDKPVYPYRGILLDTARNYYSIESIKRTIEAMAAVKLNTLHWHITDSQSFPFVTTKRPNLYKFGALSPQKVYTKAAIREVVRFGLERGVRVLPEFDAPAHVGEGWQDTDLTVCFKAEPWKSYCVEPPCGQLNPTKDELYQYLEDIYSDMAEVFDTTDIFHMGGDEVSEACWNSSDSIQNFMMQNRWDLDKESFLKLWNYFQQKAQDKAYKAFGKKLPLILWTSTLTNYKHIDDYLNKDDYIIQVWTTGVDPQIKGLLEKGYRLIMSNYDALYFDCGYGAWVGAGNNWCSPYIGWQKVYDNSPAVIALEHRDQVLGGEAALWSEQSDTSTLDGRLWPRAAALAERLWAEPATSWQDAEYRMLHIRERFVRMGIQAESLQPEWCYQNEGYCYS 3wnr A 2.008 BS01 9BE A 1 P2 Y37 I65 F114 P1 Y36 I64 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wnr A 2.008 BS02 9BE B 1 Y96 N98 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wnr C 2.008 BS01 9BE C 1 P2 K33 I65 F114 P1 K32 I64 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wns A 1.658 BS01 9AI A 1 P2 M3 Y37 V107 P1 M2 Y36 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wns C 1.658 BS01 9AI C 1 P2 M3 P1 M2 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wnt A 2.074 BS01 9BE A 1 P2 M3 H63 S64 I65 V107 P1 M2 H62 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wnt C 2.074 BS01 9BE C 1 P2 M3 S64 I65 V107 P1 M2 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 3wpc A 1.6 BS01 dna F 0 E616 H641 T642 E558 H583 T584 ? 0002224,0004888,0006955,0016020 remove_due_to_license_issue Q2EEY0 25686612 1 ~ 12 TLPPFLPCELQPHGLVNCNWLFLKSVPHFSAAAPRDNVTSLSLLSNRIHHLHDSDFAQLSNLQKLNLKWNCPPAGLSPMHFPCHMTIEPNTFLAVPTLEELNLSYNGITTVPALPSSLVSLILSRTNILQLDPTSLTGLHALRFLYMDGNCYYKNPCGRALEVAPGALLGLGNLTHLSLKYNNLTTVPRSLPPSLEYLLLSYNHIVTLAPEDLANLTALRVLDVGGNCRRCDHARNPCVECPHKFPQLHSDTFSHLSRLEGLVLKDSSLYQLNPRWFRGLGNLTVLDLSENFLYDCITKTKAFQGLAQLRRLNLSFNYHKKVSFAHLTLAPSFGSLLSLQELDMHGIFFRSLSQKTLQPLARLPMLQRLYLQMNFINQAQLGIFKDFPGLRYIDLSDNRISGAVEEDFMPSCKNLSFTLDLSRNNLVTVQPEMFAQLSRLQCLRLSHNSISQAVNGSQFVPLTSLQVLDLSHNKLDLYHGRSFTELPRLEALDLSYNSQPFSMRGVGHNLSFVAQLPTLRYLSLAHNGIHSRVSQQLCSTSLWALDFSGNSLSQMWAEGDLYLRFFQGLRSLIRLDLSQNRLHTLLPCTLGNLPKSLQLLRLRNNYLAFFNWSSLTLLPNLETLDLAGNQLKALSNGSLPSGTQLQRLDVSRNSIIFVVPGFFALATRLRELNLSANALRTVEPSWFGFLAGSLEVLDVSANPLHCACAAFVDFLLQVQAAVPGLPSRVKCGSPGQLQGRSIFAQDL 3wpc A 1.6 BS02 dna E 0 W47 F49 K51 S72 R74 H77 W96 S104 P105 M106 F108 Y132 R152 Y179 Y180 K181 Y208 Y229 R262 N263 W20 F22 K24 S45 R47 H50 W69 S77 P78 M79 F81 Y105 R125 Y152 Y153 K154 Y181 Y202 R235 N236 ? 0002224,0004888,0006955,0016020 remove_due_to_license_issue Q2EEY0 25686612 1 ~ 12 TLPPFLPCELQPHGLVNCNWLFLKSVPHFSAAAPRDNVTSLSLLSNRIHHLHDSDFAQLSNLQKLNLKWNCPPAGLSPMHFPCHMTIEPNTFLAVPTLEELNLSYNGITTVPALPSSLVSLILSRTNILQLDPTSLTGLHALRFLYMDGNCYYKNPCGRALEVAPGALLGLGNLTHLSLKYNNLTTVPRSLPPSLEYLLLSYNHIVTLAPEDLANLTALRVLDVGGNCRRCDHARNPCVECPHKFPQLHSDTFSHLSRLEGLVLKDSSLYQLNPRWFRGLGNLTVLDLSENFLYDCITKTKAFQGLAQLRRLNLSFNYHKKVSFAHLTLAPSFGSLLSLQELDMHGIFFRSLSQKTLQPLARLPMLQRLYLQMNFINQAQLGIFKDFPGLRYIDLSDNRISGAVEEDFMPSCKNLSFTLDLSRNNLVTVQPEMFAQLSRLQCLRLSHNSISQAVNGSQFVPLTSLQVLDLSHNKLDLYHGRSFTELPRLEALDLSYNSQPFSMRGVGHNLSFVAQLPTLRYLSLAHNGIHSRVSQQLCSTSLWALDFSGNSLSQMWAEGDLYLRFFQGLRSLIRLDLSQNRLHTLLPCTLGNLPKSLQLLRLRNNYLAFFNWSSLTLLPNLETLDLAGNQLKALSNGSLPSGTQLQRLDVSRNSIIFVVPGFFALATRLRELNLSANALRTVEPSWFGFLAGSLEVLDVSANPLHCACAAFVDFLLQVQAAVPGLPSRVKCGSPGQLQGRSIFAQDL 3wpc B 1.6 BS01 dna F 0 W47 F49 K51 S72 R74 H77 W96 S104 P105 M106 F108 Y132 R152 Y179 Y180 K181 Y208 R262 N263 W20 F22 K24 S45 R47 H50 W69 S77 P78 M79 F81 Y105 R125 Y152 Y153 K154 Y181 R235 N236 ? 0002224,0004888,0006955,0016020 remove_due_to_license_issue Q2EEY0 25686612 1 ~ 12 TLPPFLPCELQPHGLVNCNWLFLKSVPHFSAAAPRDNVTSLSLLSNRIHHLHDSDFAQLSNLQKLNLKWNCPPAGLSPMHFPCHMTIEPNTFLAVPTLEELNLSYNGITTVPALPSSLVSLILSRTNILQLDPTSLTGLHALRFLYMDGNCYYKNPCGRALEVAPGALLGLGNLTHLSLKYNNLTTVPRSLPPSLEYLLLSYNHIVTLAPEDLANLTALRVLDVGGNCRRCDHARNPCVECPHKFPQLHSDTFSHLSRLEGLVLKDSSLYQLNPRWFRGLGNLTVLDLSENFLYDCITKTKAFQGLAQLRRLNLSFNYHKKVSFAHLTLAPSFGSLLSLQELDMHGIFFRSLSQKTLQPLARLPMLQRLYLQMNFINQAQLGIFKDFPGLRYIDLSDNRISGAVESEDFMPSCKNLSFTLDLSRNNLVTVQPEMFAQLSRLQCLRLSHNSISQAVNGSQFVPLTSLQVLDLSHNKLDLYHGRSFTELPRLEALDLSYNSQPFSMRGVGHNLSFVAQLPTLRYLSLAHNGIHSRVSQQLCSTSLWALDFSGNSLSQMWAEGDLYLRFFQGLRSLIRLDLSQNRLHTLLPCTLGNLPKSLQLLRLRNNYLAFFNWSSLTLLPNLETLDLAGNQLKALSNGSLPSGTQLQRLDVSRNSIIFVVPGFFALATRLRELNLSANALRTVEPSWFGFLAGSLEVLDVSANPLHCACGAAFVDFLLQVQAAVPGLPSRVKCGSPGQLQGRSIFAQDL 3wpc B 1.6 BS02 dna E 0 E616 H641 T642 E559 H584 T585 ? 0002224,0004888,0006955,0016020 remove_due_to_license_issue Q2EEY0 25686612 1 ~ 12 TLPPFLPCELQPHGLVNCNWLFLKSVPHFSAAAPRDNVTSLSLLSNRIHHLHDSDFAQLSNLQKLNLKWNCPPAGLSPMHFPCHMTIEPNTFLAVPTLEELNLSYNGITTVPALPSSLVSLILSRTNILQLDPTSLTGLHALRFLYMDGNCYYKNPCGRALEVAPGALLGLGNLTHLSLKYNNLTTVPRSLPPSLEYLLLSYNHIVTLAPEDLANLTALRVLDVGGNCRRCDHARNPCVECPHKFPQLHSDTFSHLSRLEGLVLKDSSLYQLNPRWFRGLGNLTVLDLSENFLYDCITKTKAFQGLAQLRRLNLSFNYHKKVSFAHLTLAPSFGSLLSLQELDMHGIFFRSLSQKTLQPLARLPMLQRLYLQMNFINQAQLGIFKDFPGLRYIDLSDNRISGAVESEDFMPSCKNLSFTLDLSRNNLVTVQPEMFAQLSRLQCLRLSHNSISQAVNGSQFVPLTSLQVLDLSHNKLDLYHGRSFTELPRLEALDLSYNSQPFSMRGVGHNLSFVAQLPTLRYLSLAHNGIHSRVSQQLCSTSLWALDFSGNSLSQMWAEGDLYLRFFQGLRSLIRLDLSQNRLHTLLPCTLGNLPKSLQLLRLRNNYLAFFNWSSLTLLPNLETLDLAGNQLKALSNGSLPSGTQLQRLDVSRNSIIFVVPGFFALATRLRELNLSANALRTVEPSWFGFLAGSLEVLDVSANPLHCACGAAFVDFLLQVQAAVPGLPSRVKCGSPGQLQGRSIFAQDL 3wpd A 2.75 BS01 dna C 0 K95 Y132 I149 S151 Y173 D175 S205 K207 L226 Y229 V248 D250 R256 R262 N263 K292 S316 E317 R338 N340 S342 F343 H372 K68 Y105 I122 S124 Y146 D148 S178 K180 L199 Y202 V221 D223 R229 R235 N236 K265 S289 E290 R311 N313 S315 F316 H345 ? 0002224,0004888,0006955,0016020 remove_due_to_license_issue Q2EEY0 25686612 1 ~ 10 TLPPFLPCELQPHGLVNCNWLFLKSVPHFSAAAPRDNVTSLSLLSNRIHHLHDSDFAQLSNLQKLNLKWNCPPAGLSPMHFPCHMTIEPNTFLAVPTLEELNLSYNGITTVPALPSSLVSLILSRTNILQLDPTSLTGLHALRFLYMDGNCYYKNPCGRALEVAPGALLGLGNLTHLSLKYNNLTTVPRSLPPSLEYLLLSYNHIVTLAPEDLANLTALRVLDVGGNCRRCDHARNPCVECPHKFPQLHSDTFSHLSRLEGLVLKDSSLYQLNPRWFRGLGNLTVLDLSENFLYDCITKTKAFQGLAQLRRLNLSFNYHKKVSFAHLTLAPSFGSLLSLQELDMHGIFFRSLSQKTLQPLARLPMLQRLYLQMNFINQAQLGIFKDFPGLRYIDLSDNRISGAVEEDFMPSCKNLSFTLDLSRNNLVTVQPEMFAQLSRLQCLRLSHNSISQAVNGSQFVPLTSLQVLDLSHNKLDLYHGRSFTELPRLEALDLSYNSQPFSMRGVGHNLSFVAQLPTLRYLSLAHNGIHSRVSQQLCSTSLWALDFSGNSLSQMWAEGDLYLRFFQGLRSLIRLDLSQNRLHTLLPCTLGNLPKSLQLLRLRNNYLAFFNWSSLTLLPNLETLDLAGNQLKALSNGSLPSGTQLQRLDVSRNSIIFVVPGFFALATRLRELNLSANALRTVEPSWFGFLAGSLEVLDVSANPLHCACGAAFVDFLLQVQAAVPGLPSRVKCGSPGQLQGRSIFAQDLRLCL 3wpn A 2.8 BS01 B4S A 1 Y104 L292 L293 Y352 A353 Y88 L232 L233 Y292 A293 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=120nM P52732 25622007 401 KGKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGDKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTASSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVNQKL 3wq5 A 1.8 BS01 VPA A 1 Q53 H157 N202 E203 S206 Y345 F389 E416 W463 E470 W471 S473 Q477 F479 Q21 H125 N170 E171 S174 Y313 F357 E384 W431 E438 W439 S441 Q445 F447 R111 H157 E203 S206 N343 Y345 E416 R79 H125 E171 S174 N311 Y313 E384 3.2.1.149 0004553,0005975,0008422,0016798,0050535 remove_due_to_license_issue Q7X9A9 24753293 601 SFNRTSFPDGFVFGAASSAYQFEGAAKEGGKGPNIWDTFTHEFPGKISNGSTGDVADDFYHRYKEDVKVLKFIGLDGFRMSISWARVLPRGKLSGGVNKEGIAFYNNVINDLLSKGIQPFITIFHWDLPQALEDEYGGFLSPHIVNDFRDFAELCFKEFGDRVKHWITMNEPWSYSYGGYDAGLLAPGRCSAFMAFCPKGNSGTEPYIVTHNLLLSHAAAVKLYKEKYQAYQKGQIGITLVTYWMIPYSNSKADKDAAQRALDFMYGWFIEPLSFGEYPKSMRRLVGKRLPRFTKEQAMLVKGSFDFLGLNYYIANYVLNVPTSNSVNLSYTTDSLSNQTAFRNGVAIGRPTGVPAFFMYPKGLKDLLVYTKEKYNDPVIYITENGMGDNNNVTTEEGIKDPQRVYFYNQHLLSLKNAIAAGVKVKGYFTWAFLDNFEWLSGYTQRFGIVYVDFKDGLKRYPKHSALWFKKFLLK 3wq5 A 1.8 BS02 VPA A 2 A58 K59 K63 G64 P65 P121 R122 A163 A26 K27 K31 G32 P33 P89 R90 A131 R111 H157 E203 S206 N343 Y345 E416 R79 H125 E171 S174 N311 Y313 E384 3.2.1.149 0004553,0005975,0008422,0016798,0050535 remove_due_to_license_issue Q7X9A9 24753293 606 SFNRTSFPDGFVFGAASSAYQFEGAAKEGGKGPNIWDTFTHEFPGKISNGSTGDVADDFYHRYKEDVKVLKFIGLDGFRMSISWARVLPRGKLSGGVNKEGIAFYNNVINDLLSKGIQPFITIFHWDLPQALEDEYGGFLSPHIVNDFRDFAELCFKEFGDRVKHWITMNEPWSYSYGGYDAGLLAPGRCSAFMAFCPKGNSGTEPYIVTHNLLLSHAAAVKLYKEKYQAYQKGQIGITLVTYWMIPYSNSKADKDAAQRALDFMYGWFIEPLSFGEYPKSMRRLVGKRLPRFTKEQAMLVKGSFDFLGLNYYIANYVLNVPTSNSVNLSYTTDSLSNQTAFRNGVAIGRPTGVPAFFMYPKGLKDLLVYTKEKYNDPVIYITENGMGDNNNVTTEEGIKDPQRVYFYNQHLLSLKNAIAAGVKVKGYFTWAFLDNFEWLSGYTQRFGIVYVDFKDGLKRYPKHSALWFKKFLLK 3wq6 A 1.8 BS01 ZPA A 1 Q53 H157 W158 N202 E203 W205 S206 Y209 Y275 Y345 F389 E416 W463 E470 W471 S473 Q477 F479 Q22 H126 W127 N171 E172 W174 S175 Y178 Y244 Y314 F358 E385 W432 E439 W440 S442 Q446 F448 R111 H157 E203 S206 N343 Y345 E416 R80 H126 E172 S175 N312 Y314 E385 3.2.1.149 0004553,0005975,0008422,0016798,0050535 remove_due_to_license_issue Q7X9A9 24753293 601 SSFNRTSFPDGFVFGAASSAYQFEGAAKEGGKGPNIWDTFTHEFPGKISNGSTGDVADDFYHRYKEDVKVLKFIGLDGFRMSISWARVLPRGKLSGGVNKEGIAFYNNVINDLLSKGIQPFITIFHWDLPQALEDEYGGFLSPHIVNDFRDFAELCFKEFGDRVKHWITMNEPWSYSYGGYDAGLLAPGRCSAFMAFCPKGNSGTEPYIVTHNLLLSHAAAVKLYKEKYQAYQKGQIGITLVTYWMIPYSNSKADKDAAQRALDFMYGWFIEPLSFGEYPKSMRRLVGKRLPRFTKEQAMLVKGSFDFLGLNYYIANYVLNVPTSNSVNLSYTTDSLSNQTAFRNGVAIGRPTGVPAFFMYPKGLKDLLVYTKEKYNDPVIYITENGMGDNNNVTTEEGIKDPQRVYFYNQHLLSLKNAIAAGVKVKGYFTWAFLDNFEWLSGYTQRFGIVYVDFKDGLKRYPKHSALWFKKFLL 3wqh A 2.85 BS01 SKK A 1 E205 E206 F357 Y547 S630 Y662 Y666 E167 E168 F319 Y509 S592 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=3.8nM P27487 26147347 808 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 3wqm A 2.1 BS01 B29 A 1 G35 R37 R38 H41 G36 R38 R39 H42 D34 R38 Y51 Y90 D35 R39 Y49 Y88 2.5.1.153 0016102,0016740,0016765,0016791,0035440,0052572,0062204 Kd=560nM remove_due_to_license_issue P9WJ61 24475925 401 AMNLVSEKEFLDLPLVSVAEIVRCRGPKVSVFPFDGTRRWFHLECNDDYQQAALRQSIRILKMLFEHGIETVISPIFSDDLLDRGDRYIVQALEGMALLANDEEILSFYKEHEVHVLFYGDYKKRLPSTAQGAAVVKSFDDLTISTSSNTEHRLCFGVFGNDAAESVAQFSISWNETHGKPPTRREIIEGYYGEYVDKADMFIGFGRFSTFDFPLLSSGKTSLYFTVAPSYYMTETTLRRILYDHIYLRHFRPKPDYSAMSADQLNVLRNRYRAQPDRVFGVGCVHDGIWFAEG 3wqm A 2.1 BS02 B29 A 2 D34 T36 Y51 Q52 S59 F79 Y90 G97 Y233 D35 T37 Y49 Q50 S57 F77 Y88 G95 Y231 D34 R38 Y51 Y90 D35 R39 Y49 Y88 2.5.1.153 0016102,0016740,0016765,0016791,0035440,0052572,0062204 Kd=560nM remove_due_to_license_issue P9WJ61 24475925 402 AMNLVSEKEFLDLPLVSVAEIVRCRGPKVSVFPFDGTRRWFHLECNDDYQQAALRQSIRILKMLFEHGIETVISPIFSDDLLDRGDRYIVQALEGMALLANDEEILSFYKEHEVHVLFYGDYKKRLPSTAQGAAVVKSFDDLTISTSSNTEHRLCFGVFGNDAAESVAQFSISWNETHGKPPTRREIIEGYYGEYVDKADMFIGFGRFSTFDFPLLSSGKTSLYFTVAPSYYMTETTLRRILYDHIYLRHFRPKPDYSAMSADQLNVLRNRYRAQPDRVFGVGCVHDGIWFAEG 3wqv A 2.043 BS01 GCS B 1 F61 W107 D146 E148 M215 Y217 D218 W372 F38 W84 D123 E125 M192 Y194 D195 W349 D144 D146 E148 Y217 D121 D123 E125 Y194 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q2V6H4 24828498 1 RARVVCYFSNWAVYRPGVGRYGIEDIPVDMCTHIIYSFIGVTEDTQQVLIIDPELDVDKNGFKNFTSLRSKHPGVKFTVAVGGWAEGGSKYSKMVAAKSTRMAFVRSVVDFLNKYNFDGLDLDWEYPGAADRGGSFSDKDKFLYLVQELRRAFIREGKGWELTAAVPLANFRLMEGYHVPELCQELDAIHVMSYDLRGNWAGFADVHSPLYKRPHDQWAYEKLNVNDGLQLWEDKGCPTNKLVVGIPFYGRSFTLSSGNNNYNLGTYINKEAGGGDPAPYTNATGFWAYYEICTEVDTADSKWTKKWDEHGKCPYAYKGTQWVGYEDPRSVEIKMNWIKEKGYLGAMTWAIDMDDFQGLCGEKNILIKLLHKHMSAYTVPPPR 3wqv A 2.043 BS02 GCS B 2 F61 G106 A108 F38 G83 A85 D144 D146 E148 Y217 D121 D123 E125 Y194 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q2V6H4 24828498 2 RARVVCYFSNWAVYRPGVGRYGIEDIPVDMCTHIIYSFIGVTEDTQQVLIIDPELDVDKNGFKNFTSLRSKHPGVKFTVAVGGWAEGGSKYSKMVAAKSTRMAFVRSVVDFLNKYNFDGLDLDWEYPGAADRGGSFSDKDKFLYLVQELRRAFIREGKGWELTAAVPLANFRLMEGYHVPELCQELDAIHVMSYDLRGNWAGFADVHSPLYKRPHDQWAYEKLNVNDGLQLWEDKGCPTNKLVVGIPFYGRSFTLSSGNNNYNLGTYINKEAGGGDPAPYTNATGFWAYYEICTEVDTADSKWTKKWDEHGKCPYAYKGTQWVGYEDPRSVEIKMNWIKEKGYLGAMTWAIDMDDFQGLCGEKNILIKLLHKHMSAYTVPPPR 3wqw A 2.0 BS01 GCS B 1 G106 W107 D146 E148 Y217 D218 W372 G83 W84 D123 E125 Y194 D195 W349 D144 D146 E148 Y217 D121 D123 E125 Y194 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q2V6H4 24828498 1 RARVVCYFSNWAVYRPGVGRYGIEDIPVDMCTHIIYSFIGVTEDTQQVLIIDPELDVDKNGFKNFTSLRSKHPGVKFTVAVGGWAEGGSKYSKMVAAKSTRMAFVRSVVDFLNKYNFDGLDLDWEYPGAADRGGSFSDKDKFLYLVQELRRAFIREGKGWELTAAVPLANFRLMEGYHVPELCQELDAIHVMSYDLRGNWAGFADVHSPLYKRPHDQWAYEKLNVNDGLQLWEDKGCPTNKLVVGIPFYGRSFTLSSGNNNYNLGTYINKEAGGGDPAPYTNATGFWAYYEICTEVDTADSKWTKKWDEHGKCPYAYKGTQWVGYEDPRSVEIKMNWIKEKGYLGAMTWAIDMDDFQGLCGEKNILIKLLHKHMSAYTVPPPR 3wqw A 2.0 BS02 GCS B 2 F61 G106 A108 F38 G83 A85 D144 D146 E148 Y217 D121 D123 E125 Y194 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue Q2V6H4 24828498 2 RARVVCYFSNWAVYRPGVGRYGIEDIPVDMCTHIIYSFIGVTEDTQQVLIIDPELDVDKNGFKNFTSLRSKHPGVKFTVAVGGWAEGGSKYSKMVAAKSTRMAFVRSVVDFLNKYNFDGLDLDWEYPGAADRGGSFSDKDKFLYLVQELRRAFIREGKGWELTAAVPLANFRLMEGYHVPELCQELDAIHVMSYDLRGNWAGFADVHSPLYKRPHDQWAYEKLNVNDGLQLWEDKGCPTNKLVVGIPFYGRSFTLSSGNNNYNLGTYINKEAGGGDPAPYTNATGFWAYYEICTEVDTADSKWTKKWDEHGKCPYAYKGTQWVGYEDPRSVEIKMNWIKEKGYLGAMTWAIDMDDFQGLCGEKNILIKLLHKHMSAYTVPPPR 3ws8 A 2.6 BS02 X4C A 1 I692 Y693 F696 M713 Q726 F729 I246 Y247 F250 M267 Q280 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=210nM Q9Y233 24837154 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 3ws9 A 2.99 BS02 X4D A 1 Y693 F696 P712 M713 G725 Q726 F729 Y247 F250 P266 M267 G279 Q280 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=92nM Q9Y233 24837154 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 3wt5 A 1.9 BS02 YA1 A 1 Y143 V230 S233 I264 R270 S271 S274 W282 C284 H301 L309 H393 F418 Y21 V50 S53 I84 R90 S91 S94 W102 C104 H121 L129 H213 F238 ? 0003677,0004879,0006355 ic50=0.29nM remove_due_to_license_issue P13053 24742174 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3wt7 A 2.4 BS02 YA2 A 1 Y143 L229 S233 R270 S271 S274 W282 C284 V296 H301 H393 Y397 Y21 L49 S53 R90 S91 S94 W102 C104 V116 H121 H213 Y217 ? 0003677,0004879,0006355 ic50=1.79nM remove_due_to_license_issue P13053 24742174 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 3wth A 2.54 BS01 IM4 A 1 W143 T144 Y185 Y192 W144 T145 Y186 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=970nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wth A 2.54 BS02 IM4 E 1 W53 R104 L112 M114 W54 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=970nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wth B 2.54 BS01 IM4 A 1 W53 R55 A103 R104 L112 M114 W54 R56 A104 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=970nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 3wth B 2.54 BS02 IM4 B 1 W143 Y185 Y192 W144 Y186 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=970nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 3wti A 2.68 BS01 CT4 A 1 W143 Y185 C187 Y192 W143 Y185 C187 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wti A 2.68 BS02 CT4 E 1 W53 R104 L112 M114 W53 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wti B 2.68 BS01 CT4 A 1 W53 R104 L112 M114 W53 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 3wti B 2.68 BS02 CT4 B 1 Y185 Y192 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSE 3wtj A 2.24 BS01 TH4 A 1 Y89 W143 T144 T184 Y185 C187 C188 Y192 Y90 W144 T145 T185 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.297uM remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtj A 2.24 BS02 TH4 E 1 R104 M114 R105 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.297uM remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtj B 2.24 BS01 TH4 A 1 R104 M114 R105 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.297uM remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtj B 2.24 BS02 TH4 B 1 Y89 W143 T184 Y185 C187 Y192 Y90 W144 T185 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.297uM remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtk A 2.69 BS01 TH4 A 1 W53 R104 L112 M114 W54 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtk A 2.69 BS02 TH4 B 1 W143 T144 Y185 C187 Y192 W144 T145 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtk E 2.69 BS01 TH4 A 1 W143 T144 Y185 C187 Y192 W144 T145 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtk E 2.69 BS02 TH4 E 1 W53 A103 R104 L112 M114 W54 A104 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue Ki=220nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtl A 2.3 BS01 N1Y A 1 Y89 W143 T144 Y185 C187 Y192 Y90 W144 T145 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.092uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtl A 2.3 BS02 N1Y E 1 W53 R104 L112 M114 W54 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.092uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtl B 2.3 BS01 N1Y A 1 W53 R104 L112 M114 W54 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.092uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtl B 2.3 BS02 N1Y B 1 Y89 W143 Y185 C187 Y192 Y90 W144 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.092uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtm A 2.48 BS01 N1Y A 1 W53 R104 L112 M114 W53 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.1uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtm A 2.48 BS02 N1Y B 1 W143 T144 Y185 Y192 W143 T144 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.1uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtm E 2.48 BS01 N1Y A 1 Y89 W143 T144 Y185 C187 Y192 Y89 W143 T144 Y185 C187 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.1uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtm E 2.48 BS02 N1Y E 1 W53 R55 R104 L112 M114 W53 R55 R104 L112 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.1uM remove_due_to_license_issue Ki=80nM P58154 25267717 301 ADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRS 3wtn A 2.09 BS01 N2Y A 1 Y89 W143 Y192 Y92 W146 Y195 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.091uM remove_due_to_license_issue P58154 25267717 301 AEAADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wtn A 2.09 BS02 N2Y E 1 R104 L112 M114 R107 L115 M117 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.091uM remove_due_to_license_issue P58154 25267717 301 AEAADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wtn B 2.09 BS01 N2Y A 1 W53 R104 L112 M114 W56 R107 L115 M117 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.091uM remove_due_to_license_issue P58154 25267717 301 AEAADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wtn B 2.09 BS02 N2Y B 1 Y89 W143 Y192 Y92 W146 Y195 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.091uM remove_due_to_license_issue P58154 25267717 301 AEAADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wto A 2.25 BS01 N2Y A 1 Y89 W143 Y185 C187 Y192 Y90 W144 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.119uM remove_due_to_license_issue P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wto A 2.25 BS02 N2Y E 1 W53 R104 L112 M114 W54 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.119uM remove_due_to_license_issue P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wto B 2.25 BS01 N2Y A 1 R104 L112 M114 R105 L113 M115 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.119uM remove_due_to_license_issue P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wto B 2.25 BS02 N2Y B 1 Y89 W143 Y185 C187 Y192 Y90 W144 Y186 C188 Y193 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.119uM remove_due_to_license_issue P58154 25267717 301 AADRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQRTTWSDRTLAWDSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3wv1 A 1.98 BS06 WHH A 1 K140 N215 F217 L218 V219 H222 L239 F241 I243 Y244 T245 Y246 T247 K249 F252 M253 P255 K37 N112 F114 L115 V116 H119 L136 F138 I140 Y141 T142 Y143 T144 K146 F149 M150 P152 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.0039nM remove_due_to_license_issue IC50=0.003900nM P45452 25264600 307 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDEDP 3wv2 A 2.3 BS05 WGG A 1 L218 V219 H222 L239 F241 I243 Y244 T245 T247 F252 P255 L115 V116 H119 L136 F138 I140 Y141 T142 T144 F146 P149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=12nM remove_due_to_license_issue IC50=5.6nM P45452 25192810 306 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTHFMLPDDDVQGIQSLYGPGDED 3wv3 A 1.6 BS05 WLL A 1 L218 H222 L239 F241 I243 Y244 T245 F252 P255 L115 H119 L136 F138 I140 Y141 T142 F147 P150 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=24nM remove_due_to_license_issue P45452 25192810 308 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYKSHFMLPDDDVQGIQSLYGPGDEDP 3wyj A 2.1 BS01 H78 A 1 M25 N28 G29 R39 A40 H43 A47 A69 F70 S71 L85 L88 F89 M12 N15 G16 R26 A27 H30 A34 A56 F57 S58 L67 L70 F71 D26 H43 L137 D13 H30 L119 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 ic50=0.36uM remove_due_to_license_issue P60472 25574764 900 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 3wyk A 2.5 BS02 3KG A 1 L625 I682 F686 M703 Q716 F719 L181 I238 F242 M259 Q272 F275 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Q9Y233 25384088 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3wyl A 2.68 BS02 3KB A 1 L625 L665 I682 Y683 F686 M703 Q716 F719 L181 L221 I238 Y239 F242 M259 Q272 F275 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Q9Y233 25384088 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3wym A 2.0 BS02 3K9 A 1 H515 L625 L665 Y683 F686 M703 Q716 F719 H71 L181 L221 Y239 F242 M259 Q272 F275 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Q9Y233 25384088 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 3wyx A 2.9 BS01 O38 A 1 I531 Q541 A551 M602 E603 C604 G605 N606 I607 L654 I663 I16 Q26 A36 M87 E88 C89 G90 N91 I92 L139 I148 D647 K649 N652 D664 T686 D132 K134 N137 D149 T160 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 25801152 902 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPGTVNYMPPEAIKDMSISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 3wyy A 3.05 BS01 O17 A 1 I531 V539 Q541 A551 M602 E603 C604 N606 D608 L654 I663 I16 V24 Q26 A36 M87 E88 C89 N91 D93 L139 I148 D647 K649 N652 D664 T686 D132 K134 N137 D149 T160 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 25801152 901 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPGTVNYMPPEAIKDMSISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 3wz6 A 1.404 BS01 IXZ A 1 D35 G37 Y79 G80 D81 F116 D219 G221 T222 Y226 I300 D35 G37 Y79 G80 D81 F116 D219 G221 T222 Y226 I300 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=1.1uM remove_due_to_license_issue P11838 25630461 409 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 3wz7 A 1.9 BS01 IXY A 1 D33 D35 Y79 G80 D81 S83 F116 F194 D219 G221 T222 I300 I302 D33 D35 Y79 G80 D81 S83 F116 F194 D219 G221 T222 I300 I302 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=1.8uM remove_due_to_license_issue P11838 25630461 401 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 3wz8 A 1.45 BS01 IXV A 1 D15 G80 D81 F116 G221 T222 T223 Y226 I300 I304 D15 G80 D81 F116 G221 T222 T223 Y226 I300 I304 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=1.5uM remove_due_to_license_issue P11838 25630461 401 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 3wzj A 2.75 BS01 O43 A 1 I531 Q541 K553 E571 L575 M602 C604 G605 N606 L654 I663 M671 Q672 I16 Q26 K38 E56 L60 M87 C89 G90 N91 L139 I148 M156 Q157 D647 K649 N652 D664 D674 T686 D132 K134 N137 D149 D159 T161 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=5.6nM P33981 25625617 901 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 3wzk A 2.3 BS01 O23 A 1 I531 Q541 K553 E571 M602 C604 G605 N606 L654 I663 I16 Q26 K38 E56 M87 C89 G90 N91 L139 I148 D647 K649 N652 D664 D674 T686 D132 K134 N137 D149 D159 T161 2.7.12.1 0004672,0005524,0006468 ic50=58nM remove_due_to_license_issue IC50=561nM P33981 25625617 901 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMSISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 3wzn A 1.3 BS01 BTN A 1 D27 Y43 S45 V47 N49 W79 S88 T90 W108 D17 Y33 S35 V37 N39 W69 S78 T80 W98 ? 0009374 remove_due_to_license_issue Kd=1.000000nM P22629 25645976 1001 GPAEAGITGTWSDQLGDTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVK 3wzp A 1.2 BS01 ZOF A 1 L25 G48 N49 W79 S88 T90 W108 L110 D128 L14 G37 N38 W68 S77 T79 W97 L99 D117 ? 0009374 remove_due_to_license_issue P22629 25645976 201 PAEAGITGTWSDQLGDTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVK 3wzp C 1.2 BS01 ZOF C 1 L25 G48 N49 W79 S88 T90 W108 D128 L14 G37 N38 W68 S77 T79 W97 D117 ? 0009374 remove_due_to_license_issue P22629 25645976 201 PAEAGITGTWSDQLGDTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVK 3wzq A 1.7 BS01 ZOF A 1 L25 Y43 W79 S88 T90 W108 L15 Y33 W69 S78 T80 W98 ? 0009374 Kd=0.000000064M remove_due_to_license_issue P22629 25645976 1001 GSAEAGITGTWSDQLGDTFIVTAGADGALTGTYENAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVKP 3wzq C 1.7 BS01 ZOF C 1 L25 D27 Y43 W79 S88 T90 W108 L15 D17 Y33 W69 S78 T80 W98 ? 0009374 Kd=0.000000064M remove_due_to_license_issue P22629 25645976 1001 GSAEAGITGTWSDQLGDTFIVTAGADGALTGTYENAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVK 3wzu A 3.01 BS01 1FM A 1 G145 T146 M212 E213 M215 C218 K221 L266 G26 T27 M82 E83 M85 C88 K91 L136 D259 K261 S263 N264 D277 C296 D129 K131 S133 N134 D147 C152 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=1300nM O14733 25529738 600 GYLTIGGQRYQAEINDLENLGEMGSGTCGQVWKMRFRKTGHVIAVKQMRRSGNKVVLKSHDCPYIVQCFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGKMTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCDFGAGCAAYMAPERIDPPPDYDIRADVWSLGISLVELATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQSFVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFKDVMAKTE 3x00 A 1.3 BS01 ZOF A 1 D27 Y43 W79 A86 S88 T90 W108 D128 D17 Y33 W69 A76 S78 T80 W98 D118 ? 0009374 remove_due_to_license_issue P22629 25560769 201 GSAEAGITGTWSDQLGDTFIVTAGADGALTGTYENAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVK 3x00 D 1.3 BS01 ZOF D 1 D27 Y43 W79 S88 T90 W108 D128 D17 Y33 W69 S78 T80 W98 D118 ? 0009374 remove_due_to_license_issue P22629 25560769 201 GSAEAGITGTWSDQLGDTFIVTAGADGALTGTYENAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNSKNAHSATTWSGQYVGGADAKINTQWLLTSGTTNANAWKSTLVGHDTFTKVK 3x1k A 2.547 BS01 ANP A 1 Y6 G8 T9 G16 H17 L20 R87 G88 R90 D94 E98 P119 S127 S128 T129 Y5 G7 T8 G15 H16 L19 R86 G87 R89 D93 E97 P118 S126 S127 T128 H17 K41 R90 S128 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005524,0005737,0008771,0009058,0015937,0016779 remove_due_to_license_issue A0A0X1KGP2 27041211 1001 NRVLYPGTFDPITKGHGDLIERASRLFDHVIIAVAASPKKNPLFSLEQRVALAQEVTKHLPNVEVVGFSTLLAHFVKEQKANVFLRGLRAVSDFEYEFQLANMNRQLAPDVESMFLTPSEKYSFISSTLVREIAALGGDISKFVHPAVADALAERFK 3x1k E 2.547 BS01 ANP E 1 Y6 T9 F10 G16 H17 L20 R87 G88 R90 P119 S128 T129 Y5 T8 F9 G15 H16 L19 R86 G87 R89 P118 S127 T128 H17 K41 R90 S128 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005524,0005737,0008771,0009058,0015937,0016779 remove_due_to_license_issue A0A0X1KGP2 27041211 1001 NRVLYPGTFDPITKGHGDLIERASRLFDHVIIAVAASPKKNPLFSLEQRVALAQEVTKHLPNVEVVGFSTLLAHFVKEQKANVFLRGLRAVSDFEYEFQLANMNRQLAPDVESMFLTPSEKYSFISSTLVREIAALGGDISKFVHPAVADALAERFK 3zbf A 2.2 BS01 VGH A 1 L1951 A1978 M2029 G2032 D2033 N2084 L2086 G2101 D2102 S2229 L18 A42 M93 G96 D97 N148 L150 G165 D166 S281 D2079 A2081 R2083 N2084 D2102 D143 A145 R147 N148 D166 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=2.1nM remove_due_to_license_issue IC50=6.5nM, Kd=4.1nM, Ki=0.600000nM P08922 23724914 3000 IENLPAFPREKLTLRLLLGSGEVYEGTAVDILGVGSGEIKVAVKTLKKGSTDQEKIEFLKEAHLMSKFNHPNILKQLGVCLLNEPQYIILELMEGGDLLTYLRKARMATFYGPLLTLVDLVDLCVDISKGCVYLERMHFIHRDLAARNCLVSVKDYTSPRIVKIGDFGLARDIYLPVRWMAPESLMDGIFTTQSDVWSFGILIWEILTLGHQPYPAHSNLDVLNYVQTGGRLEPPRNCPDDLWNLMTQCWAQEPDQRPTFHRIQDQLQLFRNFFLNSIYKS 3zbx A 2.2 BS01 6XE A 1 I1084 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 F1344 I26 A46 Y97 M98 D102 R146 M149 A159 D160 Y168 F282 D1204 A1206 R1208 N1209 D1222 A1243 D142 A144 R146 N147 D160 A181 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.006uM remove_due_to_license_issue IC50=5nM, Ki=6nM P08581 23944843 2345 NPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 3zc5 A 2.2 BS01 W9Z A 1 I1084 A1108 Y1159 M1160 D1164 R1208 N1209 M1211 A1221 D1222 Y1230 F1344 I33 A53 Y104 M105 D109 R153 N154 M156 A166 D167 Y175 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.0103uM remove_due_to_license_issue IC50=6.0nM, Ki=10nM P08581 23944843 2345 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 3zc6 A 2.42 BS01 VFC A 1 L828 G829 K830 G831 G834 V836 A853 K855 E903 Y904 L905 G908 C909 L956 D967 L15 G16 K17 G18 G21 V23 A40 K42 E86 Y87 L88 G91 C92 L139 D150 D949 A951 R953 N954 D967 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM remove_due_to_license_issue IC50=0.600000nM P52333 23540648 2103 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 3zcl A 1.4 BS01 5TF A 1 I1084 A1108 L1157 M1160 M1211 A1221 D1222 Y1230 F1344 I33 A53 L102 M105 M156 A166 D167 Y175 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.0101uM remove_due_to_license_issue IC50=19nM, Ki=10nM P08581 23944843 1 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 3zcw A 1.691 BS02 4A2 A 1 Y104 S269 N289 L292 L293 L295 G296 R297 I299 T300 Y352 Y85 S242 N247 L250 L251 L253 G254 R255 I257 T258 Y310 ? 0003777,0005524,0007018,0008017 Kd=0.65uM remove_due_to_license_issue P52732 23305346 1366 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGDKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKP 3zcw A 1.691 BS03 4A2 A 2 E116 I136 L160 L172 I213 K216 G217 A218 K220 R221 M228 E97 I117 L141 L153 I186 K189 G190 A191 K193 R194 M201 ? 0003777,0005524,0007018,0008017 Kd=0.65uM remove_due_to_license_issue P52732 23305346 1367 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGDKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKP 3zcz A 2.6 BS01 TFR A 1 S49 W139 D142 Y147 S298 L349 G412 T413 S415 S49 W139 D142 Y147 S298 L349 G412 T413 S415 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue P39045 23484909 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 3zda A 1.5 BS01 dna B 0 A183 G184 G186 P187 K188 S189 A180 G181 G183 P184 K185 S186 3.1.-.- 0000287,0003677,0003824,0004518,0004519,0008409,0017108,0030955,0033567,0046872,0048256,0140640 remove_due_to_license_issue Q8X6R9 23821668 1 ~ 4 AVHLLIVDALNLIRRIHAVQGSPCVETCQHALDQLIMHSQPTHAVAVFDDRSSGWRHQRLPDYKAGRPPMPEELHDEMPALRAAFEQRGVPCWSTSGNEADDLAATLAVKVTQAGHQATIVSTDKGYCQLLSPTLRIRDYFQKRWLDAPFIDKEFGVQPQQLPDYWGLAGISSSKVPGVAGIGPKSATQLLVEFQSLEGIYENLDAVAEKWRKKLETHKEMAFLCRDIARLQTDLHIDGNLQQLRLV 3zdg K 2.48 BS01 XRX K 1 Y89 W143 T144 Y192 Y89 W143 T144 Y187 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Ki=0.079uM remove_due_to_license_issue Ki=79nM P58154 23256554 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 3zdg L 2.48 BS01 XRX L 1 Y89 W143 T144 Y185 Y192 Y89 W143 T144 Y180 Y187 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Ki=0.079uM remove_due_to_license_issue Ki=79nM P58154 23256554 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 3zdh A 2.195 BS01 XRS A 1 Y89 W143 Y192 Y89 W143 Y188 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Ki=0.045uM remove_due_to_license_issue Ki=45nM P58154 23256554 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 3zdh A 2.195 BS02 XRS E 1 W53 R104 W53 R104 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Ki=0.045uM remove_due_to_license_issue Ki=45nM P58154 23256554 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 3zdh B 2.195 BS01 XRS A 1 W53 M114 W53 M114 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Ki=0.045uM remove_due_to_license_issue Ki=45nM P58154 23256554 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3zdh B 2.195 BS02 XRS B 1 Y89 W143 T144 Y192 Y89 W143 T144 Y188 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Ki=0.045uM remove_due_to_license_issue Ki=45nM P58154 23256554 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 3zdv A 1.41 BS03 MMA A 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 23719508 201 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 3zdv A 1.41 BS04 F1A A 1 G24 D96 G24 D96 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 23719508 202 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 3zdv B 1.41 BS03 MMA B 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 23719508 201 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 3zdv B 1.41 BS04 F1A B 1 G24 D96 G24 D96 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 23719508 202 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 3zeb A 2.2 BS01 SV1 A 1 M149 H150 F153 N154 S201 Y205 W236 M249 M58 H59 F62 N63 S110 Y114 W145 M158 3.4.21.105 0004252,0006508,0016020 remove_due_to_license_issue P09391 23359682 401 RAGPVTWVMMIACVVVFIAMQILGDQEVMLWLAWPFDPTLKFEFWRYFTHALMHFSLMHILFNLLWWWYLGGAVEKRLGSGKLIVITLISALLSGYVQQKFSGPWFGGLSGVVYALMGYVWLRGERDPQSGIYLQRGLIIFALIWIVAGWFDLFGMSMANGAHIAGLAVGLAMAFVDSL 3zep A 2.35 BS01 1NX A 1 L828 K830 V836 A853 Y904 L905 G908 L956 D967 L15 K17 V23 A40 Y86 L87 G90 L138 D149 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.022uM remove_due_to_license_issue IC50=22nM P52333 23541670 2099 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 3zh2 A 2.1 BS01 dna E 0 D35 I36 A80 F82 K84 A85 P86 G87 K88 S89 D90 V229 H232 A233 S234 D33 I34 A78 F80 K82 A83 P84 G85 K86 S87 D88 V227 H230 A231 S232 R95 D155 R158 H182 R93 D153 R156 H180 1.1.1.27 0003824,0004459,0005515,0005737,0006096,0016491,0016616,0019752,0030060 remove_due_to_license_issue Q76NM3 24043813 1 ~ 27 PKAKIVLVGSGMIGGVMATLIVQKNLGDVVLFDIVKNMPHGKALDTSHTNVMAYSNCKVSGSNTYDDLAGADVVIVTAGFTKAPGKSDKEWNRDDLLPLNNKIMIEIGGHIKKNCPNAFIIVVTNPVDVMVQLLHQHSGVPKNKIIGLGGVLDTSRLKYYISQKLNVCPRDVNAHIVGAHGNKMVLLKRYITVGGIPLQEFINNKLISDAELEAIFDRTVNTALEIVNLHASPYVAPAAAIIEMAESYLKDLKKVLICSTLLEGQYGHSDIFGGTPVVLGANGVEQVIELQLNSEEKAKFDEAIAETKRMKALA 3zh2 B 2.1 BS01 dna E 0 I36 V37 M40 K44 A80 F82 I105 I34 V35 M38 K42 A78 F80 I97 R95 D155 R158 H182 R87 D147 R150 H174 1.1.1.27 0003824,0004459,0005515,0005737,0006096,0016491,0016616,0019752,0030060 remove_due_to_license_issue Q76NM3 24043813 1 ~ 27 PKAKIVLVGSGMIGGVMATLIVQKNLGDVVLFDIVKNMPHGKALDTSHTNVMAYSNCKVSGSNTYDDLAGADVVIVTAGFTKAEWNRDDLLPLNNKIMIEIGGHIKKNCPNAFIIVVTNPVDVMVQLLHQHSGVPKNKIIGLGGVLDTSRLKYYISQKLNVCPRDVNAHIVGAHGNKMVLLKRYITVGGIPLQEFINNKLISDAELEAIFDRTVNTALEIVNLHASPYVAPAAAIIEMAESYLKDLKKVLICSTLLEGQYGHSDIFGGTPVVLGANGVEQVIELQLNSEEKAKFDEAIAETKRMKALA 3zh2 C 2.1 BS01 dna G 0 D35 I36 A80 F82 K84 A85 P86 G87 K88 S89 D90 K91 V229 H232 A233 S234 D34 I35 A79 F81 K83 A84 P85 G86 K87 S88 D89 K90 V228 H231 A232 S233 R95 D155 R158 H182 R94 D154 R157 H181 1.1.1.27 0003824,0004459,0005515,0005737,0006096,0016491,0016616,0019752,0030060 remove_due_to_license_issue Q76NM3 24043813 1 ~ 27 APKAKIVLVGSGMIGGVMATLIVQKNLGDVVLFDIVKNMPHGKALDTSHTNVMAYSNCKVSGSNTYDDLAGADVVIVTAGFTKAPGKSDKEWNRDDLLPLNNKIMIEIGGHIKKNCPNAFIIVVTNPVDVMVQLLHQHSGVPKNKIIGLGGVLDTSRLKYYISQKLNVCPRDVNAHIVGAHGNKMVLLKRYITVGGIPLQEFINNKLISDAELEAIFDRTVNTALEIVNLHASPYVAPAAAIIEMAESYLKDLKKVLICSTLLEGQYGHSDIFGGTPVVLGANGVEQVIELQLNSEEKAKFDEAIAETKRMKALA 3zh2 D 2.1 BS01 dna G 0 G13 I36 V37 M40 K44 A80 F82 K84 I105 G11 I34 V35 M38 K42 A78 F80 K82 I100 R95 D155 R158 H182 R90 D150 R153 H177 1.1.1.27 0003824,0004459,0005515,0005737,0006096,0016491,0016616,0019752,0030060 remove_due_to_license_issue Q76NM3 24043813 1 ~ 27 PKAKIVLVGSGMIGGVMATLIVQKNLGDVVLFDIVKNMPHGKALDTSHTNVMAYSNCKVSGSNTYDDLAGADVVIVTAGFTKAPDKEWNRDDLLPLNNKIMIEIGGHIKKNCPNAFIIVVTNPVDVMVQLLHQHSGVPKNKIIGLGGVLDTSRLKYYISQKLNVCPRDVNAHIVGAHGNKMVLLKRYITVGGIPLQEFINNKLISDAELEAIFDRTVNTALEIVNLHASPYVAPAAAIIEMAESYLKDLKKVLICSTLLEGQYGHSDIFGGTPVVLGANGVEQVIELQLNSEEKAKFDEAIAETKRMKALA 3zh8 A 2.739 BS01 C58 A 1 I251 V259 V326 D330 L376 T386 D387 I13 V21 V88 D92 L138 T148 D149 D369 K371 N374 D387 T407 D131 K133 N136 D149 T169 2.7.11.13 0004672,0004674,0005524,0006468,0007163 remove_due_to_license_issue P41743 23418854 1582 SLGLQDFDLLRVIGRGSYAKVLLVRLKKTDRIYAMKVVKKELVNDDEDIDWVQTEKHVFEQASNHPFLVGLHSCFQTESRLFFVIEYVNGGDLMFHMQRQRKLPEEHARFYSAEISLALNYLHERGIIYRDLKLDNVLLDSEGHIKLTDYGMCKEGLRPGDTTSTFCGTPNYIAPEILRGEDYGFSVDWWALGVLMFEMMAGRSPFDIVNTEDYLFQVILEKQIRIPRSLSVKAASVLKSFLNKDPKERLGCHPQTGFADIQGHPFFRNVDWDMMEQKQVVPPFKPNISGEQLTPDDDDIVRKIDQSEFEGFEYINPLLM 3zhx A 2.0 BS02 FM6 A 1 D151 S152 A176 S177 S213 N218 K219 S245 P265 M267 D141 S142 A166 S167 S196 N201 K202 S228 P248 M250 1.1.1.267 0000287,0008299,0016491,0019288,0030145,0030604,0046872,0050897,0051483,0051484,0070402 remove_due_to_license_issue Kd=210nM, IC50=320nM P9WNS1 23819803 501 GRLRVVVLGSTGSIGTQALQVIADNPDRFEVVGLAAGGAHLDTLLRQRAQTGVTNIAVADEHAAQRVGDIPYHGSDAATRLVEQTEADVVLNALVGALGLRPTLAALKTGARLALANKESLVAGGSLVLRAARPGQIVPVDSEHSALAQCLRGGTPDEVAKLVLTASGGPFRGWSAADLEHVTPEQAGAPMNTLNSASLVNKGLEVIETHLLFGIPYDRIDVVVHPQSIIHSMVTFIDGSTIAQASPPDMKLPISLALGWPRRVSGAAAACDFHTASSWEFEPLDTDVFPAVELARQAGVAGGCMTAVYNAANEEAAAAFLAGRIGFPAIVGIIADVLHAADQWAVEPATVDDVLDAQRWARERAQRAVSGM 3zhz A 2.25 BS01 FM7 A 1 S152 E153 A176 S177 S213 N218 K219 M267 S135 E136 A159 S160 S189 N194 K195 M243 1.1.1.267 0000287,0008299,0016491,0019288,0030145,0030604,0046872,0050897,0051483,0051484,0070402 Kd=0.09uM remove_due_to_license_issue Kd=90nM, IC50=19000nM P9WNS1 23819803 1390 GRLRVVVLGSTGSIGTQALQVIADNPDRFEVVGLAAGGAHLDTLLRQRAQTGVTNIAVADEDIPYHGSDAATRLVEQTEADVVLNALVGALGLRPTLAALKTGARLALANKESLVAGGSLVLRAARPGQIVPVDSEHSALAQCLRGGTPDEVAKLVLTASGGPFRGWSAADLEHVTPEQAGAHPNTLNSASLVNKGLEVIETHLLFGIPYDRIDVVVHPQSIIHSMVTFIDGSTIAQASPPDMKLPISLALGWPRRVSGAAAACDFHTASSWEFEPLDTDVFPAVELARQAGVAGGCMTAVYNAANEEAAAAFLAGRIGFPAIVGIIADVLHAADQWAVEPATVDDVLDAQRWARERAQRAVSGM 3zi0 A 1.9 BS01 FM8 A 1 S152 E153 A176 S177 N209 S213 N218 K219 S245 P265 S130 E131 A154 S155 N179 S183 N188 K189 S215 P235 1.1.1.267 0000287,0008299,0016491,0019288,0030145,0030604,0046872,0050897,0051483,0051484,0070402 Kd=0.04uM remove_due_to_license_issue IC50=13000nM, Kd=40nM P9WNS1 23819803 501 RLRVVVLGSTGSIGTQALQVIADNPDRFEVVGLAAGGAHLDTLLRQRAQTGVTNIAVIPYHGSDAATRLVEQTEADVVLNALVGALGLRPTLAALKTGARLALANKESLVAGGSLVLRAARPGQIVPVDSEHSALAQCLRGGTPDEVAKLVLTASGGPFRGWSAADLEHVTPEQAGPMNTLNSASLVNKGLEVIETHLLFGIPYDRIDVVVHPQSIIHSMVTFIDGSTIAQASPPDMKLPISLALGWPRRVSGAAAACDFHTASSWEFEPLDTDVFPAVELARQAGVAGGCMTAVYNAANEEAAAAFLAGRIGFPAIVGIIADVLHAADQWAVEPATVDDVLDAQRWARERAQRAVS 3zi5 A 3.2 BS01 dna B 0 T225 Y227 N245 R246 R247 G248 R272 E276 N279 N280 R284 N337 T33 Y35 N53 R54 R55 G56 R80 E84 N87 N88 R92 N145 3.1.21.4 remove_due_to_license_issue Q9F4C9 24423868 1 ~ 12 LDETERVTLIVTLGHADTARIQAAPGTTAGQGTQYFWLSKDSYDFFPPLTIRNRRGTKATYSSLINMNYIDINYTDTQCRVTFEAENNFDFRLGTGKLRYTGVAKSNDIAAITRVGDSDYELRIIKQGTPEHSQLDPYAVSFIGNRGKRFGYISNEEFGRIIGVTF 3zi5 A 3.2 BS02 dna C 0 H207 A208 R212 Q223 G224 W229 S231 K232 N280 D282 I335 G336 R338 K340 H15 A16 R20 Q31 G32 W37 S39 K40 N88 D90 I143 G144 R146 K148 3.1.21.4 remove_due_to_license_issue Q9F4C9 24423868 1 ~ 12 LDETERVTLIVTLGHADTARIQAAPGTTAGQGTQYFWLSKDSYDFFPPLTIRNRRGTKATYSSLINMNYIDINYTDTQCRVTFEAENNFDFRLGTGKLRYTGVAKSNDIAAITRVGDSDYELRIIKQGTPEHSQLDPYAVSFIGNRGKRFGYISNEEFGRIIGVTF 3zi5 D 3.2 BS01 dna E 0 T225 Y227 N245 R247 G248 R272 E276 N279 N280 R284 N337 R338 T33 Y35 N53 R55 G56 R80 E84 N87 N88 R92 N145 R146 3.1.21.4 remove_due_to_license_issue Q9F4C9 24423868 1 ~ 12 LDETERVTLIVTLGHADTARIQAAPGTTAGQGTQYFWLSKDSYDFFPPLTIRNRRGTKATYSSLINMNYIDINYTDTQCRVTFEAENNFDFRLGTGKLRYTGVAKSNDIAAITRVGDSDYELRIIKQGTPEHSQLDPYAVSFIGNRGKRFGYISNEEFGRIIGVTF 3zi5 D 3.2 BS02 dna F 0 H207 A208 R212 T220 Q223 G224 W229 S231 K232 N280 D282 I335 G336 R338 K340 H15 A16 R20 T28 Q31 G32 W37 S39 K40 N88 D90 I143 G144 R146 K148 3.1.21.4 remove_due_to_license_issue Q9F4C9 24423868 1 ~ 12 LDETERVTLIVTLGHADTARIQAAPGTTAGQGTQYFWLSKDSYDFFPPLTIRNRRGTKATYSSLINMNYIDINYTDTQCRVTFEAENNFDFRLGTGKLRYTGVAKSNDIAAITRVGDSDYELRIIKQGTPEHSQLDPYAVSFIGNRGKRFGYISNEEFGRIIGVTF 3zim A 2.85 BS01 KKR A 1 M772 I800 D810 Y836 I848 E849 V850 V851 Q859 C862 M922 I932 D933 M626 I654 D664 Y690 I702 E703 V704 V705 Q713 C716 M776 I786 D787 2.7.11.1,2.7.1.137,2.7.1.153 0016301,0046854 remove_due_to_license_issue IC50=6.8nM, EC50=10nM P42336 23360348 2047 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRKSLWVINSALRIKILCATYVNVNDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREAGFSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGGLKGALQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDRERVPFVLTQDFLIVISCTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDA 3zj6 A 2.4 BS01 VM2 A 1 Q36 H140 E186 T189 H193 Y347 W392 E420 W469 E476 W477 Q24 H128 E174 T177 H181 Y310 W348 E376 W425 E432 W433 R94 H140 E186 T189 N345 Y347 E420 R82 H128 E174 T177 N308 Y310 E376 2.4.1.219,3.2.1.125 0004553,0005975,0008422,0009820,0009821,0016740,0016798,0050247,0050506 remove_due_to_license_issue Q9SPP9 25140865 1516 DATRISRSDFPADFIMGTGSSAYQIEGGARDGGRGPSIWDTFTHRRPDMIRGGTNGDVAVDSYHLYKEDVNILKNLGLDAYRFSISWSRVLPGGRLSGGVNKEGINYYNNLIDGLLANGIKPFVTLFHWDVPQALEDEYGGFLSPRIVDDFCEYAELCFWEFGDRVKHWMTLNEPWTFSVHGYATGLYAPGRGRTGNPGTEPYWVTHHLLLAHAAAVELYKNKFQRGQEGQIGISHATQWMEPWDENSASDVEAAARALDFMLGWFMEPITSGDYPKSMKKFVGSRLPKFSPEQSKMLKGSYDFVGLNYYTASYVTNASNFSYNTDIHVTYETDRNGVPIGPQSGSDWLLIYPEGIRKILVYTKKTYNVPLIYVTENGVDDVKNTNLTLSEARKDSMRLKYLQDHIFNVRQAMNDGVNVKGYFAWSLLDNFEWGEGYGVRFGIIHIDYNDNFARYPKDSAVWLMNSFHK 3zj8 A 3.01 BS01 LR1 A 1 Q57 E207 T210 Y345 W388 E416 W465 E472 W473 Y481 Q21 E171 T174 Y309 W347 E375 W424 E431 W432 Y440 R115 H161 E207 T210 N343 Y345 E416 R79 H125 E171 T174 N307 Y309 E375 3.2.1.105 0004553,0005975,0008422,0009820,0009821,0016798,0050422 remove_due_to_license_issue Q8GU20 25140865 1001 VVHRRDFPQDFIFGAGGSAYQCEGAYNEGNRGPSIWDTFTQRSPAKISDGSNGNQAINCYHMYKEDIKIMKQTGLESYRFSISWSRVLPGGRLAAGVNKDGVKFYHDFIDELLANGIKPSVTLFHWDLPQALEDEYGGFLSHRIVDDFCEYAEFCFWEFGDKIKYWTTFNEPHTFAVNGYALGEFAPGRGGKGDEGDPAIEPYVVTHNILLAHKAAVEEYRNKFQKCQEGEIGIVLNSMWMEPLSDVQADIDAQKRALDFMLGWFLEPLTTGDYPKSMRELVKGRLPKFSADDSEKLKGCYDFIGMNYYTATYVTNAVKLSYETDDQVTKTFERNQKPIGHALYGGWQHVVPWGLYKLLVYTKETYHVPVLYVTESGMVEENKTKILLSEARRDAERTDYHQKHLASVRDAIDDGVNVKGYFVWSFFDNFEWNLGYICRYGIIHVDYKSFERYPKESAIWYKNFIAGK 3zjc A 3.15 BS02 GNP A 1 T17 G18 G20 K21 S22 A23 S36 R37 I38 V43 T44 R133 E135 S168 N169 T10 G11 G13 K14 S15 A16 S29 R30 I31 V36 T37 R123 E125 S158 N159 ? 0003924,0005515,0005525,0005737,0005783,0005794,0005811,0042802,0042803,0046039 remove_due_to_license_issue Q8NHV1 23454188 1297 SLRIVLVGKTGSGKSATANTILGEEIFDSRIAAQAVTKNCQKASREWQGRDLLVVDTPGLFDSLDTTCKEISRCIISSCPGPHAIVLVLQLGRYTEEEQKTVALIKAVFGKSAMKHMVILFTRKEELEGQSFHDFIADADVGLKSIVKECGNRCCAFSNSTSKAEKESQVQELVELIEKMVQCNEGAYFSDDIYKDTEERLKQREEVLRKIYTDQLNEEIKLVEEDKHKSEEEKEKEIKLLKLKYDEKIKNIREEAERNIFKDVFNRIWKMLSEIWHRFLSKC 3zk6 A 2.48 BS01 H1I A 1 F97 R102 F105 S106 L108 L130 G138 R139 A142 S145 F146 F44 R49 F52 S53 L55 L77 G85 R86 A89 S92 F93 ? 0042981 Kd=0.46uM remove_due_to_license_issue IC50=500nM Q07817 23603658 1198 SQSNRELVVDFLSYKLSQKGYSWSQFSIPMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGN 3zk6 A 2.48 BS02 H1I B 1 Y101 A104 Y195 Y48 A51 Y142 ? 0042981 Kd=0.46uM remove_due_to_license_issue IC50=500nM Q07817 23603658 1198 SQSNRELVVDFLSYKLSQKGYSWSQFSIPMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGN 3zkc A 3.0 BS01 dna C 0 A27 S29 Y30 Q39 N41 P42 S43 A26 S28 Y29 Q38 N40 P41 S42 ? 0003677,0003700,0006355,0010629,0030435,0045892,0046983 remove_due_to_license_issue P06533 23430750 1 ~ 21 IGQRIKQYRKEKGYSLSELAEKAGVAKSYLSSIERNLQTNPSIQFLEKVSAVLDVSVHTLL 3zkc A 3.0 BS02 dna D 0 S16 L17 S18 K28 S29 S32 R36 S15 L16 S17 K27 S28 S31 R35 ? 0003677,0003700,0006355,0010629,0030435,0045892,0046983 remove_due_to_license_issue P06533 23430750 1 ~ 21 IGQRIKQYRKEKGYSLSELAEKAGVAKSYLSSIERNLQTNPSIQFLEKVSAVLDVSVHTLL 3zkc B 3.0 BS01 dna C 0 S16 L17 S29 S32 R36 S16 L17 S29 S32 R36 ? 0003677,0003700,0006355,0010629,0030435,0045892,0046983 remove_due_to_license_issue P06533 23430750 1 ~ 21 MIGQRIKQYRKEKGYSLSELAEKAGVAKSYLSSIERNLQTNPSIQFLEKVSAVLDVSVHTLLD 3zkc B 3.0 BS02 dna D 0 V26 A27 S29 Y30 P42 S43 V26 A27 S29 Y30 P42 S43 ? 0003677,0003700,0006355,0010629,0030435,0045892,0046983 remove_due_to_license_issue P06533 23430750 1 ~ 21 MIGQRIKQYRKEKGYSLSELAEKAGVAKSYLSSIERNLQTNPSIQFLEKVSAVLDVSVHTLLD 3zki A 2.4 BS01 WZV A 1 G27 R28 G29 L46 D48 Y87 W131 I134 D241 G243 T244 T245 A347 G14 R15 G16 L33 D35 Y74 W118 I121 D220 G222 T223 T224 A315 D48 S51 N53 A55 Y87 D241 T244 D35 S38 N40 A42 Y74 D220 T223 3.4.23.45 0004190,0006508,0016020 remove_due_to_license_issue Q9Y5Z0 23695257 1398 NFLAMVDNLQGDSGRGYYLEMLIGTPPQKLQILVDTGSSNFAVAGTPHSYIDTYFDTERSSTYRSKGFDVTVKYTQGSWTGFVGEDLVTIPKGFNTSFLVNIATIFESENFFLPGIKWNGILGLAYATLAKPSSSLETFFDSLVTQANIPNVFSMQMCGAGNGGSLVLGGIEPSLYKGDIWYTPIKEEWYYQIEILKLEIGGQSLNLDCREYNADKAIVDSGTTLLRLPQKVFDAVVEAVARASLIFSDGFWTGSQLACWTPWSYFPKISIYLRDENSSRSFRITILPQLYIQPMMYECYRFGISPSTNALVIGATVMEGFYVIFDRAQKRVGFAASPCAEIAGAAVSEISGPFSTEDVASNCVP 3zla A 3.2 BS01 rna I 0 F17 R47 K50 T75 R81 T91 R94 I123 P125 L126 K129 Y176 K179 R182 Q183 R184 E189 A190 F14 R44 K47 T72 R78 T88 R91 I120 P122 L123 K126 Y173 K176 R179 Q180 R181 E186 A187 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla B 3.2 BS01 rna I 0 T16 F17 I44 R47 K50 T75 R81 N82 R94 P125 L126 Y176 K179 R182 R184 E189 A190 N217 T13 F14 I41 R44 K47 T72 R78 N79 R91 P122 L123 Y173 K176 R179 R181 E186 A187 N214 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla C 3.2 BS01 rna I 0 T16 F17 K50 T75 R81 N82 T91 R94 P125 L126 K129 Y176 K179 R182 R184 E189 A190 N217 T13 F14 K47 T72 R78 N79 T88 R91 P122 L123 K126 Y173 K176 R179 R181 E186 A187 N214 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla D 3.2 BS01 rna I 0 I44 R47 K50 T75 R81 N82 L126 K175 Y176 K179 R182 Q183 R184 N217 I40 R43 K46 T71 R77 N78 L122 K171 Y172 K175 R178 Q179 R180 N213 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVTFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla E 3.2 BS01 rna J 0 T16 F17 I44 R47 K50 T75 R81 T91 R94 I123 P125 L126 K129 Y176 K179 R182 R184 E189 N217 T13 F14 I41 R44 K47 T72 R78 T88 R91 I120 P122 L123 K126 Y173 K176 R179 R181 E186 N214 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla F 3.2 BS01 rna J 0 T16 I44 R47 K50 T75 R81 N82 I123 P125 Y176 K179 R182 R184 E189 A190 N217 T13 I41 R44 K47 T72 R78 N79 I120 P122 Y173 K176 R179 R181 E186 A187 N214 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla G 3.2 BS01 rna J 0 T16 F17 R47 K50 T75 R81 T91 R94 I123 P125 L126 E128 K129 Y176 K179 R182 R184 E189 A190 N217 T13 F14 R44 K47 T72 R78 T88 R91 I120 P122 L123 E125 K126 Y173 K176 R179 R181 E186 A187 N214 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zla H 3.2 BS01 rna J 0 T16 F17 R47 K50 T75 R81 N82 V85 R94 P125 L126 E128 K175 Y176 K179 R182 R184 N217 T13 F14 R44 K47 T72 R78 N79 V82 R91 P122 L123 E125 K172 Y173 K176 R179 R181 N214 ? 0003723,0019013,0019029,0039657,1990904 remove_due_to_license_issue P16495 23595147 1 ~ 44 GSMIELEFHDVATFDPEVAYANFKRVHTTGLSYDHIRIFYIKGREIKTSLAKRSEWEVTLNLGGWKITVYNTNFPGNRNNPVPDDGLTLHRLSGFLARYLLEKMLKVSEPEKLIIKSKIINPLAEKNGITWNDGEEVYLSFFPGSEMFLGTFRFYPLAIGIYKVQRKEMEPKYLEKTMRQRYMGLEAATWTVSKLTEVQSALTVVSSLGWKKTNVSAAARDFLAKFGIN 3zlj A 3.1 BS01 dna E 0 T11 P12 M13 M33 G34 D35 F36 R58 S61 Q95 P99 P105 V106 R108 T10 P11 M12 M32 G33 D34 F35 R57 S60 Q94 P98 P104 V105 R107 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 23821665 1 ~ 19 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 3zlj A 3.1 BS02 dna F 0 F36 E38 I53 S54 R58 M68 G70 P72 Y79 L495 K496 R500 F35 E37 I52 S53 R57 M67 G69 P71 Y78 L494 K495 R499 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 23821665 5 ~ 21 SAIENFDAHTPMMQQYLRLKAQHPEILLFYRMGDFYELFYDDAKRASQLLDISLTKRGASAGEPIPMAGIPYHAVENYLAKLVNQGESVAICEQIGDPATSKGPVERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 3zlj B 3.1 BS01 dna E 0 L495 K496 R500 L438 K439 R443 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 23821665 1 ~ 19 EILLFYRMGDFYELFYDDAKRASQLLDISAVENYLAKLVNQGESVAICEERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGAADDLASGRSTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 3zlj B 3.1 BS02 dna F 0 H471 S478 H414 S421 ? 0000018,0003677,0003684,0005515,0005524,0005829,0006281,0006298,0006974,0008301,0016887,0030983,0032136,0032300,0042802,0043531,0140664,1990710 remove_due_to_license_issue P23909 23821665 5 ~ 21 EILLFYRMGDFYELFYDDAKRASQLLDISAVENYLAKLVNQGESVAICEERKVVRIVTPGTISDEALLQERQDNLLAAIWQDSKGFGYATLDISSGRFRLSEPADRETMAAELQRTNPAELLYAEDFAEMSLIEGRRGLRRRPLWEFEIDTARQQLNLQFGTRDLVGFGVENAPRGLCAAGCLLQYAKDTQRTTLPHIRSITMEREQDSIIMDAATRRNLEITQNLAGGAENTLASVLDCTVTPMGSRMLKRWLHMPVRDTRVLLERQQTIGALQDFTAGLQPVLRQVGDLERILARLALRTARPRDLARMRHAFQQLPELRAQLETVDSAPVQALREKMGEFAELRDLLERAIIDTPPVLVRDGGVIASGYNEELDEWRALADGATDYLERLEVRERERTGLDTLKVGFNAVHGYYIQISRGQSHLAPINYMRRQTLKNAERYIIPELKEYEDKVLTSKGKALALEKQLYEELFDLLLPHLEALQQSASALAELDVLVNLAERAYTLNYTCPTFIDKPGIRITEGRHPVVEQVLNEPFIANPLNLSPQRRMLIITGPNMGGKSTYMRQTALIALMAYIGSYVPAQKVEIGPIDRIFTRVGAADDLASGRSTFMVEMTETANILHNATEYSLVLMDEIGRGTSTYDGLSLAWACAENLANKIKALTLFATHYFELTQLPEKMEGVANVHLDALEHGDTIAFMHSVQDGAASKSYGLAVAALAGVPKEVIKRARQKLRELESIS 3zlk A 1.952 BS01 Y46 A 1 S41 L45 Y113 Y114 G115 V250 A251 E255 I256 S45 L49 Y117 Y118 G119 V254 A255 E259 I260 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=1.32uM remove_due_to_license_issue IC50=1.32e+3nM Q9HU22 23138692 400 HHHHHKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 3zlk C 1.952 BS01 Y46 C 1 S41 L45 Y113 Y114 G115 H119 V250 A251 E255 R259 S40 L44 Y112 Y113 G114 H118 V249 A250 E254 R258 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=1.32uM remove_due_to_license_issue IC50=1.32e+3nM Q9HU22 23138692 400 KRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 3zll A 2.0 BS01 4WF A 1 L45 E255 I256 R259 L49 E259 I260 R263 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 Kd=0.395uM remove_due_to_license_issue IC50=1.14e+3nM Q9HU22 23138692 400 HHHHHKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 3zln A 2.288 BS01 H0Y A 1 F97 F105 S106 D107 L108 T109 E129 L130 R132 N136 G138 R139 S145 F146 G196 F44 F52 S53 D54 L55 T56 E76 L77 R79 N83 G85 R86 S92 F93 G143 ? 0042981 Kd=3.4nM remove_due_to_license_issue IC50=20nM, Kd=4.1nM Q07817 23603658 1197 MSQSNRELVVDFLSYKLSQKGYSWSQFTESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 3zlo A 2.601 BS01 X8U A 1 A93 F97 Y101 F105 S106 L108 T109 L130 N136 G138 R139 A142 S145 F146 Y195 G196 A38 F42 Y46 F50 S51 L53 T54 L75 N81 G83 R84 A87 S90 F91 Y140 G141 ? 0042981 remove_due_to_license_issue IC50=1.5nM Q07817 23603658 1198 SQSNRELVVDFLSYKLSQKGYSWSQTESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 3zlq A 2.1 BS01 6T9 A 1 G29 Y30 L46 D48 Y87 F124 D241 S242 G243 T245 A347 G14 Y15 L31 D33 Y72 F109 D217 S218 G219 T221 A317 D48 S51 N53 A55 Y87 D241 T244 D33 S36 N38 A40 Y72 D217 T220 3.4.23.45 0004190,0006508,0016020 ic50=0.904uM remove_due_to_license_issue IC50=904nM Q9Y5Z0 23590342 1398 LAMVDNLQGDSGRGYYLEMLIGTPPQKLQILVDTGSSNFAVAGTPHSYIDTYFDTERSSTYRSKGFDVTVKYTQGSWTGFVGEDLVTIPKGFNTSFLVNIATIFESENFFLPGIKWNGILGLAYATLAKPSSSLETFFDSLVTQANIPNVFSMQMCGAGGGSLVLGGIEPSLYKGDIWYTPIKEEWYYQIEILKLEIGGQSLNLDCREYNADKAIVDSGTTLLRLPQKVFDAVVEAVARASDGFWTGSQLACWTNSETPWSYFPKISIYLRDENSSRSFRITILPQLYIQPMMGAGLNYECYRFGISPSTNALVIGATVMEGFYVIFDRAQKRVGFAASPCAEIAGAAVSEISGPFSTEDVASNCVP 3zlr A 2.026 BS01 X0B A 1 F97 Y101 R102 F105 S106 L108 L130 R132 G138 R139 S145 F146 F46 Y50 R51 F54 S55 L57 L79 R81 G87 R88 S94 F95 ? 0042981 Kd=0.55nM remove_due_to_license_issue IC50=3.0nM, EC50=48nM, Ki=1.1nM Q07817 23603658 1198 GPLGSMSQSNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGN 3zlr B 2.026 BS01 X0B B 1 E96 F97 Y101 R102 F105 S106 L108 E129 L130 G138 R139 F146 Y195 E37 F38 Y42 R43 F46 S47 L49 E70 L71 G79 R80 F87 Y136 ? 0042981 Kd=0.55nM remove_due_to_license_issue IC50=3.0nM, EC50=48nM, Ki=1.1nM Q07817 23603658 1204 SNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGNNAAAES 3zls A 2.5 BS01 92P A 1 L74 A95 M143 E144 M146 L197 C207 D208 L36 A57 M105 E106 M108 L159 C169 D170 D190 K192 S194 N195 D208 D217 T226 D152 K154 S156 N157 D170 D179 T188 2.7.12.2 0004672,0005524,0006468 ic50=39.4uM remove_due_to_license_issue IC50=39400nM Q02750 23648182 1383 ELELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3zlv A 2.5 BS01 HI6 A 1 Y124 W286 F297 Y341 Y124 W279 F290 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 23376121 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 3zlw A 2.12 BS01 MT8 A 1 L74 V82 A95 M143 M146 G149 L197 C207 L36 V44 A57 M105 M108 G111 L159 C169 D190 K192 N195 D208 D217 T226 D152 K154 N157 D170 D179 T185 2.7.12.2 0004672,0005524,0006468 ic50=198uM remove_due_to_license_issue IC50=18100nM Q02750 23648182 1383 ELELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAANGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3zlx A 2.2 BS01 5EZ A 1 L74 A76 G77 A95 M143 E144 H145 M146 D152 Q153 L197 L36 A38 G39 A57 M105 E106 H107 M108 D114 Q115 L159 D190 K192 S194 N195 D208 D217 T226 D152 K154 S156 N157 D170 D179 T185 2.7.12.2 0004672,0005524,0006468 ic50=157uM remove_due_to_license_issue IC50=157000nM Q02750 23648182 1383 ELELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3zly A 2.11 BS01 YSO A 1 V82 A95 M143 E144 M146 L197 V42 A55 M103 E104 M106 L157 D190 K192 S194 N195 D208 D217 T226 D150 K152 S154 N155 D168 D177 T183 2.7.12.2 0004672,0005524,0006468 ic50=300uM remove_due_to_license_issue IC50=300000nM Q02750 23648182 1383 LELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3zm4 A 2.37 BS01 22T A 1 L74 A76 G77 V82 A95 M143 E144 H145 M146 S194 L197 L35 A37 G38 V43 A56 M104 E105 H106 M107 S155 L158 D190 K192 S194 N195 D208 D217 T226 D151 K153 S155 N156 D169 D178 T183 2.7.12.2 0004672,0005524,0006468 ic50=1.1uM remove_due_to_license_issue IC50=1100nM Q02750 23648182 1383 LELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMAGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFGCPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 3zm5 A 2.94 BS01 IGM A 1 F31 D32 R34 R49 F54 Y135 N137 I139 N326 N328 P329 T330 A331 L334 L360 F31 D32 R34 R49 F54 Y135 N137 I139 N326 N328 P329 T330 A331 L334 L360 6.3.2.10 0005524,0005737,0008360,0008766,0009058,0009252,0016874,0016881,0047480,0051301,0071555 remove_due_to_license_issue Q8DNV6 23786712 1455 MKLTIHEIAQVVGAKNDISIFEDTQLEKAEFDSRLIGTGDLFVPLKGARDGHDFIETAFENGAAVTLSEKEVSNHPYILVDDVLTAFQSLASYYLEKTTVDVFAVTGSNGKTTTKDMLAHLLSTRYKTYKTQGNYNNEIGLPYTVLHMPEGTEKLVLEMGQDHLGDIHLLSELARPKTAIVTLVGEAHLAFFKDRSEIAKGKMQIADGMASGSLLLAPADPIVEDYLPIDKKVVRFGQGAELEITDLVERKDSLTFKANFLEQALDLPVTGKYNATNAMIASYVALQEGVSEEQIRLAFQHLELTRNRTEWKKAANGADILSDVYNANPTAMKLILETFSAIPANEGGKKIAVLADMKELGDQSVQLHNQMILSLSPDVLDIVIFYGEDIAQLAQLASQMFPIGHVYYFKKTEDQDQFEDLVKQVKESLGAHDQILLKGSNSMNLAKLVESLEN 3zm6 A 1.84 BS01 2GN A 1 F31 D32 R34 A48 R49 F54 Y135 N137 G140 N326 N328 T330 A331 L334 L360 Q363 F31 D32 R34 A48 R49 F54 Y135 N137 G140 N326 N328 T330 A331 L334 L360 Q363 6.3.2.10 0005524,0005737,0008360,0008766,0009058,0009252,0016874,0016881,0047480,0051301,0071555 ic50=0.3uM remove_due_to_license_issue Q8DNV6 23786712 500 MKLTIHEIAQVVGAKNDISIFEDTQLEKAEFDSRLIGTGDLFVPLKGARDGHDFIETAFENGAAVTLSEKEVSNHPYILVDDVLTAFQSLASYYLEKTTVDVFAVTGSNGKTTTKDMLAHLLSTRYKTYKTQGNYNNEIGLPYTVLHMPEGTEKLVLEMGQDHLGDIHLLSELARPKTAIVTLVGEAHLAFFKDRSEIAKGKMQIADGMASGSLLLAPADPIVEDYLPIDKKVVRFGQGAELEITDLVERKDSLTFKANFLEQALDLPVTGKYNATNAMIASYVALQEGVSEEQIRLAFQHLELTRNRTEWKKAANGADILSDVYNANPTAMKLILETFSAIPANEGGKKIAVLADMKELGDQSVQLHNQMILSLSPDVLDIVIFYGEDIAQLAQLASQMFPIGHVYYFKKTEDQDQFEDLVKQVKESLGAHDQILLKGSNSMNLAKLVESLEN 3zm9 A 1.9 BS01 QMQ A 1 I209 R213 G310 I329 Y354 W420 W423 I106 R110 G207 I226 Y251 W317 W320 2.7.1.32,2.7.1.82 remove_due_to_license_issue P35790 23441033 1458 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 3zmg A 1.74 BS01 6Z0 A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 D227 G229 T231 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D227 T230 3.4.23.46 0004190,0006508,0016020 ic50=0.023uM remove_due_to_license_issue P56817 23590342 1448 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 3zmh A 2.3 BS01 L62 A 1 M149 H150 F153 N154 W157 S201 V204 Y205 M208 W236 M247 H254 M59 H60 F63 N64 W67 S111 V114 Y115 M118 W146 M157 H164 3.4.21.105 0004252,0006508,0016020 remove_due_to_license_issue P09391 23665170 401 ERAGPVTWVMMIACVVVFIAMQILGDQEVMLWLAWPFDPTLKFEFWRYFTHALMHFSLMHILFNLLWWWYLGGAVEKRLGSGKLIVITLISALLSGYVQQKFSGPWFGGLSGVVYALMGYVWLRGERDPQSGIYLQRGLIIFALIWIVAGWFDLFGMSMANGAHIAGLAVGLAMAFVDSL 3zmi A 2.2 BS01 L6C A 1 M149 H150 N154 W157 S201 V204 Y205 W236 H254 M58 H59 N63 W66 S110 V113 Y114 W145 H158 3.4.21.105 0004252,0006508,0016020 remove_due_to_license_issue P09391 23665170 401 RAGPVTWVMMIACVVVFIAMQILGDQEVMLWLAWPFDPTLKFEFWRYFTHALMHFSLMHILFNLLWWWYLGGAVEKRLGSGKLIVITLISALLSGYVQQKFSGPWFGGLSGVVYALMGYVWLRGERDPQSGIYLQRGLIIFALIWIVAGWFDLANGAHIAGLAVGLAMAFVDSL 3zmj A 2.3 BS01 L61 A 1 M149 H150 N154 W157 S201 Y205 M208 W236 M247 H254 M58 H59 N63 W66 S110 Y114 M117 W145 M155 H162 3.4.21.105 0004252,0006508,0016020 remove_due_to_license_issue P09391 23665170 401 RAGPVTWVMMIACVVVFIAMQILGDQEVMLWLAWPFDPTLKFEFWRYFTHALMHFSLMHILFNLLWWWYLGGAVEKRLGSGKLIVITLISALLSGYVQQKFSGPWFGGLSGVVYALMGYVWLRGERDPQSGIYLQRGLIIFALIWIVAGWFDLGMSMANGAHIAGLAVGLAMAFVDSL 3zmm A 2.51 BS01 F9J A 1 L855 A880 M929 E930 Y931 L932 G935 N981 L983 G993 L12 A33 M78 E79 Y80 L81 G84 N130 L132 G142 D976 A978 R980 N981 D994 S1016 D125 A127 R129 N130 D143 S161 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=0.720000nM O60674 23562594 2133 FEERHLKFLQQLGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYRNLKLIMEYLPYGSLRDYLQAHAERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQM 3znc A 2.8 BS02 BZ1 A 1 Q92 H94 H96 F141 L198 T199 T200 W209 Q91 H93 H95 F127 L188 T189 T190 W199 H64 H94 H96 E106 H119 T199 H66 H93 H95 E105 H118 T189 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006885,0008270,0009897,0009986,0015670,0015701,0016020,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 remove_due_to_license_issue Q64444 9541386 500 WCYEIQTEDPRSSCLGPEKWPGACKENQQSPINIVTARTKVNPRLTPFILVGYDQKQQWPIKNNQHTVEMTLGGGACIIGGDLPARYEAVQLHLHWSNGNDNGSEHSIDGRHFAMEMHIVHKKLDKFAVLAFMIEVGDKVNKGFQPLVEALPSISKPHSTSTVRESSLQDMLPPSTKMYTYFRYNGSLTTPNCDETVIWTVYKQPIKIHKNQFLEFSKNLYYDEDQKLNMKDNVRPLQPLGKRQVFKSHA 3znr A 2.4 BS03 NU9 A 1 P542 E543 P667 H669 H670 G678 F679 D707 H709 F738 L810 E840 G841 H843 P27 E28 P134 H136 H137 G145 F146 D174 H176 F205 L277 E307 G308 H310 3.5.1.-,3.5.1.98 Ki=0.036uM remove_due_to_license_issue Ki=46nM, IC50=4.1nM Q8WUI4 23524983 1000 LPFTTGLIYDSVMLKHQCSCGDNSRHPEHAGRIQSIWSRLQERGLRSQCECLRGRKASLEELQSVHSERHVLLYGTNPLSVMLPCGGVGVDTDTIWNELHSSNAARWAAGSVTDLAFKVASRELKNGFAVVRPPGHHADHSTAMGFCFFNSVAIACRQLQQQSKASKILIVDWDVHHGNGTQQTFYQDPSVLYISLHRHDDGNFFPGSGAVDEVGAGSGEGFNVNVAWAGGLDPPMGDPEYLAAFRIVVMPIAREFSPDLVLVSAGFDAAEGHPAPLGGYHVSAKCFGYMTQQLMNLAGGAVVLALEGGHDLTAICDASEACVAALLGNRVDPLSEEGWKQKPNLNAIRSLEAVIRVHSKYWGCMQRL 3zns A 2.45 BS03 NU7 A 1 P542 P667 H669 H670 G678 F679 D707 H709 F738 L810 G841 P27 P134 H136 H137 G145 F146 D174 H176 F205 L277 G308 3.5.1.-,3.5.1.98 Ki=0.039uM remove_due_to_license_issue Ki=39nM Q8WUI4 23524983 1900 LPFTTGLIYDSVMLKHQCSCGDNSRHPEHAGRIQSIWSRLQERGLRSQCECLRGRKASLEELQSVHSERHVLLYGTNPLSVMLPCGGVGVDTDTIWNELHSSNAARWAAGSVTDLAFKVASRELKNGFAVVRPPGHHADHSTAMGFCFFNSVAIACRQLQQQSKASKILIVDWDVHHGNGTQQTFYQDPSVLYISLHRHDDGNFFPGSGAVDEVGAGSGEGFNVNVAWAGGLDPPMGDPEYLAAFRIVVMPIAREFSPDLVLVSAGFDAAEGHPAPLGGYHVSAKCFGYMTQQLMNLAGGAVVLALEGGHDLTAICDASEACVAALLGNRVDPLSEEGWKQKPNLNAIRSLEAVIRVHSKYWGCMQRL 3zo1 A 2.0 BS02 SIJ A 1 V57 A70 V104 M120 E121 Y122 V123 E127 E170 L173 D184 F327 V49 A62 V96 M112 E113 Y114 V115 E119 E162 L165 D176 F319 D166 K168 E170 N171 D184 T201 D158 K160 E162 N163 D176 T193 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=1uM remove_due_to_license_issue P00517 23920481 1351 GSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3zo2 A 1.98 BS02 15I A 1 L49 F54 V57 A70 V104 M120 E121 V123 E127 E170 N171 L173 T183 D184 F327 L43 F48 V51 A64 V98 M114 E115 V117 E121 E164 N165 L167 T177 D178 F321 D166 K168 E170 N171 D184 T201 D160 K162 E164 N165 D178 T195 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=80nM remove_due_to_license_issue P00517 23920481 1351 KKGSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3zo4 A 1.65 BS02 QWI A 1 T51 G52 G55 R56 A70 K72 M120 V123 E127 L173 T183 D184 F327 T38 G39 G42 R43 A57 K59 M107 V110 E114 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=149nM remove_due_to_license_issue P00517 23920481 1352 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 3zos A 1.92 BS01 0LI A 1 A653 K655 E672 M676 T701 Y703 M704 V763 H764 R765 L773 I782 A783 D784 F785 A52 K54 E71 M75 T100 Y102 M103 V151 H152 R153 L161 I170 A171 D172 F173 D766 R770 N771 D784 A793 D154 R158 N159 D172 A181 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Q08345 24768818 1000 RVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSLDFPLNVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDAAQGPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNTV 3zos A 1.92 BS02 0LI A 2 V799 C814 I815 L816 G818 F861 V187 C202 I203 L204 G206 F249 D766 R770 N771 D784 A793 D154 R158 N159 D172 A181 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Q08345 24768818 1004 RVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSLDFPLNVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDAAQGPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNTV 3zot A 2.399 BS01 L6C A 1 M149 H150 F153 N154 W157 S201 V204 Y205 W236 H254 M58 H59 F62 N63 W66 S110 V113 Y114 W145 H161 3.4.21.105 0004252,0006508,0016020 remove_due_to_license_issue P09391 23665170 401 RAGPVTWVMMIACVVVFIAMQILGDQEVMLWLAWPFDPTLKFEFWRYFTHALMHFSLMHILFNLLWWWYLGGAVEKRLGSGKLIVITLISALLSGYVQQKFSGPWFGGLSGVVYALMGYVWLRGERDPQSGIYLQRGLIIFALIWIVAGWFDLFGMANGAHIAGLAVGLAMAFVDSLN 3zov A 2.1 BS01 WZV A 1 G72 Q73 G74 Y75 L91 D93 Y132 F169 D289 G291 T293 A396 G16 Q17 G18 Y19 L35 D37 Y76 F113 D221 G223 T225 A321 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 23695257 1447 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 3zp9 A 1.31 BS01 9TH A 1 H94 H96 H119 F131 L198 T199 T200 P202 H92 H94 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 1001 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 3zpl A 2.8 BS01 dna C 0 R32 M61 T62 R72 S76 H77 R90 R98 G99 Q100 R28 M57 T58 R68 S72 H73 R86 R94 G95 Q96 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 PRWLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEAGADLPWLR 3zpl A 2.8 BS02 dna D 0 Y44 S73 R74 H77 R81 D96 K97 R98 Y40 S69 R70 H73 R77 D92 K93 R94 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 PRWLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEAGADLPWLR 3zpl B 2.8 BS01 dna C 0 Y44 S73 R74 H77 R81 D96 K97 R98 Y40 S69 R70 H73 R77 D92 K93 R94 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 PRWLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEAGADLPWLR 3zpl B 2.8 BS02 dna D 0 R32 M61 T62 R72 S76 H77 R90 R98 G99 Q100 R28 M57 T58 R68 S72 H73 R86 R94 G95 Q96 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 PRWLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEAGADLPWLR 3zpl E 2.8 BS01 dna G 0 R32 M61 T62 R72 S76 H77 R90 R98 G99 Q100 R31 M60 T61 R71 S75 H76 R89 R97 G98 Q99 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 NDEPRWLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEADLPWLR 3zpl E 2.8 BS02 dna H 0 Y44 S73 R74 H77 R81 K97 R98 Y43 S72 R73 H76 R80 K96 R97 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 NDEPRWLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEADLPWLR 3zpl F 2.8 BS01 dna G 0 Y44 S73 R74 H77 R81 D96 K97 R98 Y38 S67 R68 H71 R75 D90 K91 R92 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 WLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEDLPWLR 3zpl F 2.8 BS02 dna H 0 R32 M61 T62 R72 S73 S76 H77 R90 R98 G99 Q100 R26 M55 T56 R66 S67 S70 H71 R84 R92 G93 Q94 ? 0003700,0006355,0006950 remove_due_to_license_issue Q9KYU1 23748564 1 ~ 22 WLTAEEQLVWRSYIEAATLLEDHLDRQLQRDAGMPHVYYGLLVKLAESPRRRLRMTELAKYAKITRSRLSHAVARLEKNGWVRREDCPSDKRGQFAILTDEGYEVLRRTAPGHVDAVRQAVFDRLTPEQQKSLGEIMRIVAEGLQPSEDLPWLR 3zpq A 2.8 BS07 XF5 A 1 D121 V122 F201 W303 F306 F307 N329 D90 V91 F170 W232 F235 F236 N258 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 23517028 1359 GAELLSQQWEAGMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVALRVYREAKEQSRVMLMREHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLLA 3zpr A 2.7 BS03 3WC A 1 D121 F201 S211 W303 F307 N310 N329 Y333 D90 F170 S180 W229 F233 N236 N255 Y259 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 23517028 500 GAELLSQQWEAGMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVALRVYREAKEQMLMREHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLL 3zps A 1.55 BS01 EQM B 1 D25 G27 A28 D29 G48 G49 I50 P81 D25 G27 A28 D29 G48 G49 I50 P81 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 24160253 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3zps B 1.55 BS01 EQM B 1 L123 D125 G127 A128 D129 G148 G149 I150 P181 L23 D25 G27 A28 D29 G48 G49 I50 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 24160253 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3zpt A 1.54 BS01 M8Y B 1 D25 G27 A28 D29 G48 G49 I50 P81 T82 D25 G27 A28 D29 G48 G49 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 24160253 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3zpt B 1.54 BS01 M8Y B 1 L123 D125 G127 D129 G148 G149 I150 T182 L23 D25 G27 D29 G48 G49 I50 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.1nM remove_due_to_license_issue P03366 24160253 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3zpu A 1.8 BS01 M8B B 1 D25 G27 A28 D29 G48 I50 P81 T82 D25 G27 A28 D29 G48 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 24160253 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3zpu B 1.8 BS01 M8B B 1 R108 L123 D125 G127 D129 G148 G149 I150 R8 L23 D25 G27 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.2nM remove_due_to_license_issue P03366 24160253 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 3zq9 A 1.86 BS01 NOY A 1 G47 N48 N186 E187 E358 W391 G41 N42 N180 E181 E352 W385 3.2.1.151','3.2.1.4 remove_due_to_license_issue Q1A2D0 21795708 1519 AKTITIKVDTFKDRKPISPYIYGTNQDLAGDENMAARRLGGNRMTGYNWENNMSNAGSDWQQSSDNYLCSNGGLTQAECEKPGAVTTSFHDQSLKLGTYSLVTLPMAGYVAKDGNGSVQESEAAPSARWNQVVNAKNAPFQLQPDLNDNYVYVDEFVHFLVNKYGTASTKAGVKGYALDNEPALWSHTHPRIHGEKVGAKELVDRSVSLSKAVKAIDAGAEVFGPVLYGFGAYKDLQTAPDWDSVKGNYSWFVDYYLDQMRLSSQVEGKRLLDVFDVHWYPEAMGGGIRITNEVGNDETKKARMQAPRTLWDPTYKEDSWIAQWNSEFLPILPRLKQSVDKYYPGTKLAMTEYSYGGENDISGGIAMTDVLGILGKNDVYMANYWKLKDGVNNYVSAAYKLYRNYDGKNSTFGDTSVSAQTSDIVNSSVHASVTNASDKELHLVVMNKSMDSAFDAQFDLSGAKTYISGKVWGFDKNSSQIKEAAPITQISGNRFTYTVPPLTAYHIVLTTG 3zq9 A 1.86 BS02 BGC A 1 R49 D65 W391 R43 D59 W385 3.2.1.151','3.2.1.4 remove_due_to_license_issue Q1A2D0 21795708 1520 AKTITIKVDTFKDRKPISPYIYGTNQDLAGDENMAARRLGGNRMTGYNWENNMSNAGSDWQQSSDNYLCSNGGLTQAECEKPGAVTTSFHDQSLKLGTYSLVTLPMAGYVAKDGNGSVQESEAAPSARWNQVVNAKNAPFQLQPDLNDNYVYVDEFVHFLVNKYGTASTKAGVKGYALDNEPALWSHTHPRIHGEKVGAKELVDRSVSLSKAVKAIDAGAEVFGPVLYGFGAYKDLQTAPDWDSVKGNYSWFVDYYLDQMRLSSQVEGKRLLDVFDVHWYPEAMGGGIRITNEVGNDETKKARMQAPRTLWDPTYKEDSWIAQWNSEFLPILPRLKQSVDKYYPGTKLAMTEYSYGGENDISGGIAMTDVLGILGKNDVYMANYWKLKDGVNNYVSAAYKLYRNYDGKNSTFGDTSVSAQTSDIVNSSVHASVTNASDKELHLVVMNKSMDSAFDAQFDLSGAKTYISGKVWGFDKNSSQIKEAAPITQISGNRFTYTVPPLTAYHIVLTTG 3zqe B 2.19 BS01 DXC B 1 Y47 R232 Y37 R140 ? 0005576,0009986,0015031,0030254,0030257,0042802 Kd=59uM remove_due_to_license_issue P41784,Q56026 21829362 1079 DVSAKFDTGVDNLQTQVTEALDKLAAKPSDPALLAAYQSKLSEYNLYRNAQSNGDSYLGVYENVVAVYTDFYQAFSDILSKMGGWLLPGKDGNTVKLDVTSLKNDLNSLVNKYNQINSNTVLFPAQSGSGVKVATEAEARQWLSELNLPNSCLKSYGSGYVVTVDLTPLQKMVQDIDGLGAPGKDSKLEMDNAKYQAWQSGFKAQEENMKTTLQTLTQKYSNANSLYDNLVKVLSSTISSSLETAKSF 3zqt A 2.29 BS02 30Z A 1 F673 N727 L830 E837 F4 N58 L161 E168 ? remove_due_to_license_issue P10275 22047606 1920 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 3zrc C 2.9 BS01 L8B C 1 W88 Y98 P99 R107 I109 H110 S111 Y112 H115 W117 W26 Y36 P37 R45 I47 H48 S49 Y50 H53 W55 ? remove_due_to_license_issue IC50=4100nM, Kd=5300nM P40337 22369643 1205 LRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQE 3zrk A 2.37 BS02 ZRK A 1 V70 A83 K85 Y134 V135 L188 D200 V35 A48 K50 Y97 V98 L151 D163 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.13uM remove_due_to_license_issue IC50=125.89nM P49841 21764580 1400 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 3zrl A 2.48 BS02 ZRL A 1 F67 V70 K85 Y134 V135 L188 D200 F32 V35 K50 Y97 V98 L151 D163 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.16uM remove_due_to_license_issue IC50=158.49nM P49841 21764580 1390 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 3zrm A 2.49 BS02 ZRM A 1 G63 F67 V70 A83 K85 Y134 V135 L188 D200 G28 F32 V35 A48 K50 Y97 V98 L151 D163 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.13uM remove_due_to_license_issue IC50=125.89nM P49841 21764580 1388 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 3zso A 1.75 BS01 O2N A 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=7.6uM remove_due_to_license_issue P12497 22808106 1219 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 3zso A 1.75 BS02 O2N B 1 Q95 A98 L102 A128 A129 W131 Q39 A42 L46 A72 A73 W75 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=7.6uM remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 3zso B 1.75 BS01 O2N A 1 Q95 A98 L102 A128 A129 W131 Q39 A42 L46 A72 A73 W75 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=7.6uM remove_due_to_license_issue P12497 22808106 1219 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 3zso B 1.75 BS02 O2N B 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=7.6uM remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 3zsq A 1.7 BS01 O4N A 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=10.9uM remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsq A 1.7 BS02 O4N B 1 Q95 A98 Y99 Q39 A42 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=10.9uM remove_due_to_license_issue P12497 22808106 1213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsq B 1.7 BS01 O4N A 1 Q95 A98 Q39 A42 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=10.9uM remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsq B 1.7 BS02 O4N B 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=10.9uM remove_due_to_license_issue P12497 22808106 1213 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsw A 1.8 BS02 ZSW A 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 308 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsw A 1.8 BS03 ZSW B 1 Q95 E96 Y99 Q39 E40 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 307 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsw B 1.8 BS01 ZSW A 1 Q95 E96 Y99 Q39 E40 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 308 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsw B 1.8 BS03 ZSW B 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 307 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsx A 1.95 BS01 N44 A 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsx A 1.95 BS02 N44 B 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsx B 1.95 BS01 N44 A 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsx B 1.95 BS02 N44 B 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsy A 2.2 BS01 OM3 A 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsy B 2.2 BS01 OM3 A 1 Q95 Y99 A129 Q39 Y43 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsy B 2.2 BS02 OM3 B 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsz A 2.0 BS01 OM2 A 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsz A 2.0 BS02 OM2 B 1 Q95 Y99 Q39 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsz B 2.0 BS01 OM2 A 1 Q95 Y99 Q39 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zsz B 2.0 BS02 OM2 B 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt1 A 1.75 BS01 OM1 A 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt1 A 1.75 BS02 OM1 B 1 Q95 A98 Y99 A129 Q39 A42 Y43 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt1 B 1.75 BS01 OM1 A 1 Q95 A98 Y99 A128 A129 Q39 A42 Y43 A72 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt1 B 1.75 BS02 OM1 B 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 A 1.7 BS01 ZT2 A 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 A 1.7 BS02 ZT2 A 2 Y83 H185 R187 S195 G197 Y27 H129 R131 S135 G137 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 A 1.7 BS03 ZT2 B 1 Q95 A129 W132 Q39 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 A 1.7 BS04 ZT2 B 2 R107 P109 I208 R51 P53 I148 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 B 1.7 BS01 ZT2 A 1 Q95 A129 W132 Q39 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 B 1.7 BS02 ZT2 A 2 R107 P109 I208 R51 P53 I148 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 B 1.7 BS03 ZT2 B 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt2 B 1.7 BS04 ZT2 B 2 H185 R187 S195 G197 H129 R131 S135 G137 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt3 A 1.95 BS01 ZT4 A 1 A169 E170 H171 T174 M178 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1435uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt3 A 1.95 BS02 ZT4 B 1 Q95 A129 W132 Q39 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1435uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt3 B 1.95 BS01 ZT4 A 1 Q95 A129 W132 Q39 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1435uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKYSAGERIVDIIATDIQ 3zt3 B 1.95 BS02 ZT4 B 1 A169 E170 H171 T174 M178 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1435uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKYSAGERIVDIIATDIQ 3zt4 A 2.2 BS01 ZT2 A 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQT 3zt4 A 2.2 BS02 ZT2 A 2 Y83 H185 R187 S195 G197 E198 Y27 H129 R131 S136 G138 E139 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQT 3zt4 A 2.2 BS03 ZT2 B 1 Q95 W132 Q39 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQT 3zt4 A 2.2 BS04 ZT2 B 2 R107 W108 P109 R51 W52 P53 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQT 3zt4 B 2.2 BS01 ZT2 A 1 Q95 A129 W132 Q40 A74 W77 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1216 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt4 B 2.2 BS02 ZT2 A 2 R107 W108 P109 R52 W53 P54 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1217 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt4 B 2.2 BS03 ZT2 B 1 Q168 A169 E170 H171 T174 M178 Q113 A114 E115 H116 T119 M123 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1214 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3zt4 B 2.2 BS04 ZT2 B 2 Y83 H185 S195 G197 Y28 H130 S136 G138 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1375uM remove_due_to_license_issue P12497 22808106 1215 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 3ztc C 2.65 BS01 TR0 C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W26 Y36 P37 I47 H48 S49 Y50 H53 W55 ? remove_due_to_license_issue P40337 23102223 1205 LRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQE 3ztd C 2.79 BS01 ZTD C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W26 Y36 P37 I47 H48 S49 Y50 H53 W55 ? remove_due_to_license_issue P40337 23102223 1205 LRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQE 3ztx A 1.95 BS01 ZTX A 1 V107 A120 L154 L170 F172 A173 G176 E177 L223 V21 A34 L68 L84 F86 A87 G90 E91 L137 D216 K218 E220 N221 D234 T252 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q6DE08 21992004 1357 KFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQ 3zuk A 2.6 BS02 RDF A 1 F48 N452 A453 E494 H497 R616 H622 R628 F45 N446 A447 E488 H491 R610 H616 R622 H493 E494 H497 E560 D564 H622 R628 H487 E488 H491 E554 D558 H616 R622 3.4.24.- 0004222,0005886,0006508,0008237,0009274,0016485,0046872 remove_due_to_license_issue O53649 21813647 1665 AIPSGIDLSHIDADARPQDDLFGHVNGRWLAEHEIPADRATDGAFRSLFDRAETQVRDLIIQASQAGAAVGTDAQRIGDLYASFLDEEAVERAGVQPLHDELATIDSAADATELAAALGTLQRAGVGGGIGVYVDTDSKDSTRYLVHFTQSGIGLPDESYYRDEQHAAVLAAYPGHIARMFGLVYGGESRDHAKTADRIVALETKLADAHWDVVKRRDADLGYNLRTFAQLQTEGAGFDWVSWVTALGSAPDAMTELVVRQPDYLVTFASLWASVNVEDWKCWARWRLIRARAPWLTRALVAEDFEFYGRTLTGAQQLRDRWKRGVSLVENLMGDAVGKLYVQRHFAKSRIDTLVDNLQEAYRISISELDWMTPQTRQRALAKLNKFTAKVGYPIKWRDYSKLAIDRDDLYGNVQRGYAVNHDRELAKLFGPVDRDEWFMTPQTVNAYYNPGMNEIVFPAAILQPPFFDPQADEAANYGGIGAVIGHEIGHGFDDQGAKYDGDGNLVDWWTDDDRTEFAARTKALIEQYHAYTPRDLVDHPGPPHVQGAFTIGENIGDLGGLSIALLAYQLSLNGNPAPVIDGLTGMQRVFFGWAQIWRTKSRAAEAIRRLAVDPHSPPEFRCNGVVRNVDAFYQAFDVTEDDALFLDPQRRVRIWN 3zv7 A 2.26 BS01 NHG A 1 W84 G118 G119 S200 F331 H440 W83 G117 G118 S199 F330 H439 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G117 G118 G150 S199 A200 A238 F289 F291 E326 H439 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 22390827 1541 DHSELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 3zvk E 2.5 BS01 dna X 0 N9 G10 Q11 S12 N8 G9 Q10 S11 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 2 ~ 27 NKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEISS 3zvk E 2.5 BS02 dna Y 0 K5 R16 K19 K4 R15 K18 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 1 ~ 26 NKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEISS 3zvk F 2.5 BS01 dna X 0 N9 Q11 S12 K19 N9 Q11 S12 K19 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 2 ~ 27 MNKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEISSDDIFPEGRKDLPPQKRKYFE 3zvk F 2.5 BS02 dna Y 0 K5 R16 P18 K19 R22 K5 R16 P18 K19 R22 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 1 ~ 26 MNKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEISSDDIFPEGRKDLPPQKRKYFE 3zvk G 2.5 BS01 dna X 0 K5 G10 R16 P18 K19 R22 K4 G9 R15 P17 K18 R21 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 2 ~ 27 NKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEISSDDIFPEGRKDLPPQKRKYFE 3zvk G 2.5 BS02 dna Y 0 N9 G10 Q11 S12 N8 G9 Q10 S11 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 1 ~ 26 NKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEISSDDIFPEGRKDLPPQKRKYFE 3zvk H 2.5 BS01 dna X 0 K5 R16 P18 K19 R22 K5 R16 P18 K19 R22 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 2 ~ 27 MNKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEIS 3zvk H 2.5 BS02 dna Y 0 N9 Q11 S12 N9 Q11 S12 ? 0003677 remove_due_to_license_issue Q4UNB3 22140099 1 ~ 26 MNKAKIFMNGQSQAVRLPKEFRFSVKEVSVIPLGKGIVLQPLPNSWKDVFQEMAEIS 3zvt A 3.1 BS01 B07 A 1 A48 S49 Y147 S298 G348 K410 T411 G412 A48 S49 Y147 S298 G348 K410 T411 G412 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue IC50=1300nM, Ki=1500nM P39045 21574608 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAPE 3zvv A 2.5 BS01 XAZ A 1 I831 Y867 I879 E880 V882 M953 F961 I963 I581 Y617 I629 E630 V632 M703 F711 I713 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=915uM remove_due_to_license_issue IC50=915000nM P48736 21925880 1500 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 3zvw B 2.0 BS01 FP5 B 1 A48 S49 S298 N300 G348 L349 K410 T411 G412 T413 A48 S49 S298 N300 G348 L349 K410 T411 G412 T413 3.4.16.4 0000270,0004180,0004185,0005576,0006508,0008360,0009002,0009252,0046677,0071555 remove_due_to_license_issue Ki=125000nM, IC50=320000nM P39045 21574608 500 RLTELREDIDAILEDPALEGAVSGVVVVDTATGEELYSRDGGEQLLPASNMKLFTAAAALEVLGADHSFGTEVAAESAPGRRGEVQDLYLVGRGDPTLSAEDLDAMAAEVAASGVRTVRGDLYADDTWFDSERLVDDWWPEDEPYAYSAQISALTVAHGERFDTGVTEVSVTPAAEGEPADVDLGAAEGYAELDNRAVTGAAGSANTLVIDRPVGTNTIAVTGSLPADAAPVTALRTVDEPAALAGHLFEEALESNGVTVKGDVGLGGVPADWQDAEVLADHTSAELSEILVPFMKFSNNGHAEMLVKSIGQETAGAGTWDAGLVGVEEALSGLGVDTAGLVLNDGSGLSRGNLVTADTVVDLLGQAGSAPWAQTWSASLPVAGESDPFVGGTLANRMRGTAAEGVVEAKTGTMSGVSALSGYVPGPEGELAFSIVNNGHSGPAPLAVQDAIAVRLAEYAGHQAP 3zw3 A 2.8 BS01 ZW3 A 1 W812 K833 I879 V882 A885 M953 I963 D964 W562 K583 I629 V632 A635 M703 I713 D714 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 21925880 2191 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYRVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 3zxe A 1.67 BS01 PGZ A 1 H33 H49 R53 W69 E72 H30 H46 R50 W66 E69 ? 0005515,0005576,0005615,0005634,0005737,0006915,0007157,0030246,0070062 Kd=450uM remove_due_to_license_issue P47929 22059385 1 PHKSSLPEGIRPGTVLRIRGLVPPNASRFHVNLLCGEEQGSDAALHFNPRLDTSEVVFNSKEQGSWGREERGPGVPFQRGQPFEVLIIASDDGFKAVVGDAQYHHFRHRLPLARVRLVEVGGDVQLDSVRIF 3zxh A 1.3 BS07 E41 A 1 L184 L185 A186 H222 E223 H226 H232 P242 I243 Y244 L81 L82 A83 H119 E120 H123 H129 P139 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=3nM P45452 21937229 401 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGFMLPDDDVQGIQSLYGPGDED 3zxh B 1.3 BS06 E41 B 1 L184 A186 H222 E223 H226 H232 P242 I243 Y244 L81 A83 H119 E120 H123 H129 P139 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=3nM P45452 21937229 401 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 3zxr A 2.15 BS01 IQ1 A 1 G131 F232 H278 S280 R364 G128 F229 H275 S277 R361 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E130 E132 E216 E224 H273 R344 E363 R365 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 ic50=0.02uM remove_due_to_license_issue P9WN39 22369127 501 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSIHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 3zxr F 2.15 BS01 IQ1 F 1 G131 F232 H278 S280 R364 G128 F229 H275 S277 R361 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E130 E132 E216 E224 H273 R344 E363 R365 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 ic50=0.02uM remove_due_to_license_issue P9WN39 22369127 501 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSIHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 3zxv A 2.26 BS01 MXI A 1 Y129 G131 F232 H278 S280 K361 R364 Y126 G128 F229 H275 S277 K358 R361 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E130 E132 E216 E224 H273 R344 E363 R365 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 ic50=0.049uM remove_due_to_license_issue P9WN39 22369127 501 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSIHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 3zxv F 2.26 BS01 MXI F 1 Y129 G131 F232 H278 S280 K361 R364 Y126 G128 F229 H275 S277 K358 R361 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E130 E132 E216 E224 H273 R344 E363 R365 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 ic50=0.049uM remove_due_to_license_issue P9WN39 22369127 501 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSIHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 3zxz A 1.8 BS01 KRW A 1 I1084 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 D1231 F1344 I33 A53 Y104 M105 D109 R153 M156 A166 D167 Y175 D176 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.004uM remove_due_to_license_issue IC50=4nM, EC50=0.300000nM, Ki=5nM P08581 22924734 2345 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 3zy2 A 1.54 BS01 GDP A 1 R40 F41 G42 N43 H238 R240 A307 S308 D309 D334 M336 S355 T356 F357 R16 F17 G18 N19 H200 R202 A269 S270 D271 D296 M298 S317 T318 F319 2.4.1.221 0005783,0006004,0006486,0006493,0007219,0008417,0016757,0036066,0046922 Kd=0.35uM remove_due_to_license_issue Q18014 21966509 1381 ATDPNGYIVFCPCMGRFGNQVDQFLGVLAFAKALDRTLVLPNFIEFKHPETKMIPFEFLFQVGTVAKYTRVVTMQEFTKKIMPTVWPPEKRKAFCWTPRQEPGCHSKEGNPFGPYWDQIDVSFVGDEYFGDIPGGFDLKWLEKFPSEEYPVLAFSSAPAPFPSKGKVWSIQKYLRWSSRITEQAKKFISANLAKPFVAVHLRNDADWVRVCEHIDTTTNRPLFASEQCLGEGHHLGTLTKEICSPSKQQILEQIVEKVGSIGAKSVFVASDKDHMIDEINEALKPYEIEAHRQEPDDMYTSLAIMGRADLFVGNCVSTFSHIVKRERDHAGQSPRPSAFFGI 3zy5 A 1.96 BS01 GFB A 1 R40 G42 N43 H238 R240 W245 F261 A307 S308 D309 M336 S355 T356 F357 R18 G20 N21 H213 R215 W220 F236 A282 S283 D284 M311 S330 T331 F332 2.4.1.221 0005783,0006004,0006486,0006493,0007219,0008417,0016757,0036066,0046922 Kd=0.23uM remove_due_to_license_issue Q18014 21966509 1386 AEATDPNGYIVFCPCMGRFGNQVDQFLGVLAFAKALDRTLVLPNFIEFKHPETKMIPFEFLFQVGTVAKYTRVVTMQEFTKKIMPTVWPPEKRKAFCWTPRQAIYAEPGCHSKEGNPFGPYWDQIDVSFVGDEYFGDIPGGFDLNQMGSRKKWLEKFPSEEYPVLAFSSAPAPFPSKGKVWSIQKYLRWSSRITEQAKKFISANLAKPFVAVHLRNDADWVRVCEHIDTTTNRPLFASEQCLGEGHHLGTLTKEICSPSKQQILEQIVEKVGSIGAKSVFVASDKDHMIDEINEALKPYEIEAHRQEPDDMYTSLAIMGRADLFVGNCVSTFSHIVKRERDHAGQSPRPSAFFGIR 3zya A 1.9 BS01 2A8 A 1 Y35 A51 K53 L104 T106 L108 M109 G110 A111 L167 Y40 A56 K58 L109 T111 L113 M114 G115 A116 L172 D150 K152 N155 D168 T185 D155 K157 N160 D173 T178 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=50nM Q16539 22198732 400 SHMLEMSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 3zyf A 1.944 BS02 147 A 1 Y36 H50 D100 T104 N107 Y36 H50 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 Kd=14.1uM remove_due_to_license_issue Q05097 21919164 1001 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 3zyh A 1.501 BS02 G0S A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 21919164 202 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 3zyr A 1.65 BS01 BMA C 1 N145 S146 E230 Q231 N138 S139 E223 Q224 ? 0030246,0046872 remove_due_to_license_issue G1EUI6 22692206 3 STDSLSFSFINFDRDERNLIFQGDAHTSRNNILQLTRTDSNGAPVRSTVGRILHSAQVRLWEKSTNRVANLQTQFSFFLSSPLSNPADGIAFFIAPPDTTIPSGSAGGLLGLFNPRTALNESANQVLAVEFDTFFAQNSNTWDPNYQHIGIDVNSIRSSKVVRWERREGKTLNVLVTYNPSTRTIDVVATYPDGQRYQLSHVVDLTTILPEWVRVGFSAASGEQFQTHNLESWSFTSTLL 3zyr A 1.65 BS02 MAN C 1 D95 G114 G115 F141 N147 G229 E230 Q231 D88 G107 G108 F134 N140 G222 E223 Q224 ? 0030246,0046872 remove_due_to_license_issue G1EUI6 22692206 6 STDSLSFSFINFDRDERNLIFQGDAHTSRNNILQLTRTDSNGAPVRSTVGRILHSAQVRLWEKSTNRVANLQTQFSFFLSSPLSNPADGIAFFIAPPDTTIPSGSAGGLLGLFNPRTALNESANQVLAVEFDTFFAQNSNTWDPNYQHIGIDVNSIRSSKVVRWERREGKTLNVLVTYNPSTRTIDVVATYPDGQRYQLSHVVDLTTILPEWVRVGFSAASGEQFQTHNLESWSFTSTLL 3zyu A 1.5 BS01 1GH A 1 W81 P82 F83 L92 Y139 I146 M149 W40 P41 F42 L51 Y98 I105 M108 ? ic50=0.1uM remove_due_to_license_issue IC50=790nM, Ki=9.0nM, Kd=53nM O60885 21964340 1173 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 3zze A 1.87 BS01 6XP A 1 A1108 M1160 R1208 D1222 A1226 Y1230 F1344 A50 M102 R150 D164 A168 Y172 F286 D1204 A1206 R1208 N1209 D1222 A1243 D146 A148 R150 N151 D164 A185 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.0013uM remove_due_to_license_issue P08581 22924734 2345 NPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 3zzf A 2.2 BS01 NLG A 1 G135 T136 G137 R158 N247 V248 N249 A250 G74 T75 G76 R97 N186 V187 N188 A189 K103 G106 G137 D251 K309 K42 G45 G76 D190 K248 1.2.1.38,2.7.2.8 0005737 Ki=400mM remove_due_to_license_issue Q01217 22529931 1360 NGFSATRSTVIQLLNNISTKREVEQYLKYFTSVSQQQFAVIKVGGAIISDNLHELASCLAFLYHVGLYPIVLHGTGPQVNGRLEAQGIEPDYIDGIRITDEHTMAVVRKCFLEQNLKLVTALEQLGVRARPITSGVFTADYLDKDKYKLVGNIKSVTKEPIEASIKAGALPILTSLAETASGQMLNVNADVAAGELARVFEPLKIVYLNEKGGIINGSTGEKISMINLDEEYDDLMKQSWVKYGTKLKIREIKELLDYLPRSSSVAIINVQDLQKELFTDSGAGTMIRRGY 3zzh C 2.1 BS01 ARG C 1 Y87 K265 S285 E337 L338 T340 D341 S342 G345 M347 Y25 K203 S223 E275 L276 T278 D279 S280 G283 M285 K103 G106 G137 D251 K309 K41 G44 G75 D189 K247 1.2.1.38,2.7.2.8 0005737 remove_due_to_license_issue Q01217 22529931 1362 GFSATRSTVIQLLNNISTKREVEQYLKYFTSVSQQQFAVIKVGGAIISDNLHELASCLAFLYHVGLYPIVLHGTGPQVNGRLEAQGIEPDYIDGIRITDEHTMAVVRKCFLEQNLKLVTALEQLGVRARPITSGVFTADYLDKDKYKLVGNIKSVTKEPIEASIKAGALPILTSLAETASGQMLNVNADVAAGELARVFEPLKIVYLNEKGGIINGSTGEKISMINLDEEYDDLMKQSWVKYGTKLKIREIKELLDYLPRSSSVAIINVQDLQKELFTDSGAGTMIRR 456c A 2.4 BS04 CBP A 1 L184 L185 A186 L218 H222 E223 H226 H232 L239 F241 P242 I243 Y244 T245 L75 L76 A77 L109 H113 E114 H117 H123 L130 F132 P133 I134 Y135 T136 H222 E223 H226 H232 H113 E114 H117 H123 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.17nM remove_due_to_license_issue P45452 10074939 1 TLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 4a12 A 3.15 BS01 dna F 0 D29 R44 R47 E54 L55 R56 D23 R38 R41 E48 L49 R50 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 KLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 A 3.15 BS02 dna G 0 R13 V38 S39 Q41 T42 R7 V32 S33 Q35 T36 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 KLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 B 3.15 BS01 dna F 0 K10 R13 S39 Q41 T42 L45 K7 R10 S36 Q38 T39 L42 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 ETLKLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 B 3.15 BS02 dna G 0 D29 R44 R47 E54 L55 R56 D26 R41 R44 E51 L52 R53 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 ETLKLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 C 3.15 BS01 dna F 0 D29 R44 R47 E54 L55 R56 D26 R41 R44 E51 L52 R53 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 ETLKLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 C 3.15 BS02 dna G 0 K10 R13 V38 S39 Q41 T42 K7 R10 V35 S36 Q38 T39 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 ETLKLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 D 3.15 BS01 dna F 0 R13 V38 S39 Q41 T42 R189 R7 V32 S33 Q35 T36 R183 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 KLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a12 D 3.15 BS02 dna G 0 D29 R44 R47 E54 L55 R56 D23 R38 R41 E48 L49 R50 ? 0003677,0003700,0006633,0045717,0045892,0046872 remove_due_to_license_issue Q2FZ56 23300457 1 ~ 40 KLKKDKRREAIRQQIDSNPFITDHELSDLFQVSIQTIRLDRTYLNIPELRKRIKLVAEKNYDQISSIEEQEFIGDLIQVNPNVKAQSILDITSDSVFHKTGIARGHVLFAQANSLCVALIKQPTVLTHESSIQFIEKVKLNDTVRAEARVVNQTAKHYYVEVKSYVKHTLVFKGNFKMFYDKR 4a16 A 2.65 BS01 H34 A 1 W86 G121 Y124 E202 W286 F295 F297 Y337 F338 Y341 W439 H447 Y449 W83 G118 Y121 E199 W283 F292 F294 Y334 F335 Y338 W436 H444 Y446 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G118 G119 G151 S200 A201 G239 F294 F296 E331 H444 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 22052791 1545 EDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPGGAGGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 4a22 A 1.9 BS01 TD4 A 1 N27 S53 D95 H96 H212 G213 H252 G253 S255 N274 V275 D276 T277 N26 S52 D94 H95 H198 G199 H238 G239 S241 N260 V261 D262 T263 D95 H96 H212 H252 N274 D94 H95 H198 H238 N260 4.1.2.13 0004332,0005576,0005829,0005886,0005975,0006096,0008270,0009274,0016829,0016832,0035375,0046872 Kd=6.8nM remove_due_to_license_issue IC50=3.2nM P9WQA3 21949126 1344 PIATPEVYAEMLGQAKQNSYAFPAINCTSSETVNAAIKGFADAGSDGIIQFSTGGAEFGSGLGVKDMVTGAVALAEFTHVIAAKYPVNVALHTDHCPKDKLDSYVRPLLAISAQRVSKGGNPLFQSHMWDGSAVPIDENLAIAQELLKAAAAAKIILEIEIGVVGGYTSPEDFEKTIEALGAGEHGKYLLAATFGNVHGVYKPGNVKLRPDILAQGQQVAAAKLGLPADAKPFDFVFHGGSGSLKSEIEEALRYGVVKMNVDTDTQYAFTRPIAGHMFTNYDGVLKVDGEVGVKKVYDPRSYLKKAEASMSQRVVQACNDLHCAGKSLT 4a22 B 1.9 BS01 TD4 B 1 N27 S53 G55 D95 H96 H212 G213 G253 S255 N274 V275 D276 T277 N26 S52 G54 D94 H95 H198 G199 G239 S241 N260 V261 D262 T263 D95 H96 H212 H252 N274 D94 H95 H198 H238 N260 4.1.2.13 0004332,0005576,0005829,0005886,0005975,0006096,0008270,0009274,0016829,0016832,0035375,0046872 Kd=6.8nM remove_due_to_license_issue IC50=3.2nM P9WQA3 21949126 1344 PIATPEVYAEMLGQAKQNSYAFPAINCTSSETVNAAIKGFADAGSDGIIQFSTGGAEFGSGLGVKDMVTGAVALAEFTHVIAAKYPVNVALHTDHCPKDKLDSYVRPLLAISAQRVSKGGNPLFQSHMWDGSAVPIDENLAIAQELLKAAAAAKIILEIEIGVVGGYTSPEDFEKTIEALGAGEHGKYLLAATFGNVHGVYKPGNVKLRPDILAQGQQVAAAKLGLPADAKPFDFVFHGGSGSLKSEIEEALRYGVVKMNVDTDTQYAFTRPIAGHMFTNYDGVLKVDGEVGVKKVYDPRSYLKKAEASMSQRVVQACNDLHCAGKSLT 4a23 A 2.4 BS01 C56 A 1 D74 Y124 W286 I294 F295 R296 Y341 D74 Y124 W279 I287 F288 R289 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=1.3uM remove_due_to_license_issue P21836 22140425 1542 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4a4e A -1.00 BS01 2MR A 1 W102 D105 Y109 Y127 Y130 N132 W19 D22 Y26 Y44 Y47 N49 ? 0003723,0005634,0005737,0006397 remove_due_to_license_issue Q16637 22101937 1148 NTAASLQQWKVGDKCSAIWSEDGCIYPATIASIDFKRETCVVVYTGYGNREEQNLSDLLSPICE 4a4f A -1.00 BS01 2MR A 1 W83 Y90 F108 Y111 N113 W19 Y26 F44 Y47 N49 ? 0003723,0005634,0005737,0006397 remove_due_to_license_issue O75940 22101937 201 ASTQPTHSWKVGDKCMAVWSEDGQCYEAEIEEIDEENGTAAITFAGYGNAEVTPLLNLKPVEEG 4a4g A -1.00 BS01 DA2 A 1 W102 Y109 Y127 Y130 N132 W19 Y26 Y44 Y47 N49 ? 0003723,0005634,0005737,0006397 remove_due_to_license_issue Q16637 22101937 1148 NTAASLQQWKVGDKCSAIWSEDGCIYPATIASIDFKRETCVVVYTGYGNREEQNLSDLLSPICE 4a4h A -1.00 BS01 DA2 A 1 W83 Y90 F108 Y111 N113 W19 Y26 F44 Y47 N49 ? 0003723,0005634,0005737,0006397 remove_due_to_license_issue O75940 22101937 1129 ASTQPTHSWKVGDKCMAVWSEDGQCYEAEIEEIDEENGTAAITFAGYGNAEVTPLLNLKPVEEG 4a4l A 2.35 BS02 939 A 1 L59 C67 A80 K82 C133 R134 R136 S137 E140 F183 D194 L21 C29 A42 K44 C95 R96 R98 S99 E102 F145 D156 D176 K178 G180 N181 D194 T214 D138 K140 G142 N143 D156 T176 2.7.11.21 0004672,0005524,0006468 ic50=0.015uM remove_due_to_license_issue IC50=15nM P53350 22154349 1331 EIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKTLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 4a4o A 2.7 BS02 664 A 1 R57 L59 G60 K61 G62 C67 A80 K82 C133 R134 R136 S137 E140 F183 D194 R19 L21 G22 K23 G24 C29 A42 K44 C95 R96 R98 S99 E102 F145 D156 D176 K178 G180 N181 D194 T214 D138 K140 G142 N143 D156 T176 2.7.11.21 0004672,0005524,0006468 remove_due_to_license_issue IC50=9nM P53350 22154349 1332 EIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKTLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIA 4a4q A 1.8 BS01 UX9 A 1 D25 G27 A28 D30 V32 G48 G49 I50 P81 T82 D25 G27 A28 D30 V32 G48 G49 I50 P81 T82 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q8Q3H0 22376008 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4a4q B 1.8 BS01 UX9 A 1 D125 D129 I147 G148 G149 P181 T182 D25 D29 I47 G48 G49 P81 T82 D125 T126 G127 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q8Q3H0 22376008 1100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4a4v A 2.0 BS01 YFD A 1 G284 C285 R288 L330 I341 S342 L353 G71 C72 R75 L117 I128 S129 L140 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=1200nM, Kd=287nM P37231 23286787 999 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKISKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4a4w A 2.0 BS01 YFB A 1 I281 G284 C285 R288 I326 L330 I341 S342 L353 I67 G70 C71 R74 I112 L116 I127 S128 L139 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=19nM, EC50=73nM P37231 23286787 999 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4a4x A 2.4 BS01 JUP A 1 I14 G15 Y19 C22 V35 M86 Y88 C89 F148 G158 D159 F160 I12 G13 Y17 C20 V33 M84 Y86 C87 F139 G149 D150 F151 D141 K143 A145 N146 D159 T179 D132 K134 A136 N137 D150 T156 2.7.11.1 0004672,0005524,0006468 ic50=0.059uM remove_due_to_license_issue IC50=2700nM P51955 22404346 1280 SRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSHRDLKPANVFLDGKQNVKLGDFGLVGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 4a50 A 2.75 BS02 DQ6 A 1 E116 G117 E118 R119 I136 P137 Y211 E215 R221 E100 G101 E102 R103 I120 P121 Y195 E199 R205 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=11.1nM P52732 22248262 1367 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENININQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 4a51 A 2.75 BS03 DQ8 A 1 E116 G117 E118 R119 P137 Y211 A218 R221 E99 G100 E101 R102 P120 Y194 A201 R204 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=185.8nM P52732 22248262 801 NIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKLVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKP 4a6b A 1.8 BS01 QG8 B 1 D25 G27 A28 D30 I50 P81 T82 D25 G27 A28 D30 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 22376008 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4a6b B 1.8 BS01 QG8 B 1 L123 D125 G127 A128 D129 G148 I150 F153 T182 V184 L23 D25 G27 A28 D29 G48 I50 F53 T82 V84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=12nM remove_due_to_license_issue P35963 22376008 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4a6c A 1.5 BS01 QG9 B 1 D25 G27 A28 G48 I50 P81 T82 D25 G27 A28 G48 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P35963 22376008 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4a6c B 1.5 BS01 QG9 B 1 L123 D125 G127 A128 D129 G148 G149 I150 F153 P181 V184 L23 D25 G27 A28 D29 G48 G49 I50 F53 P81 V84 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.2nM remove_due_to_license_issue P35963 22376008 1200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4a6l A 2.05 BS01 P43 A 1 Q105 Y181 I193 D207 S208 C209 Q210 S213 V231 W233 G234 E235 G237 Q87 Y162 I174 D188 S189 C190 Q191 S194 V212 W214 G215 E216 G217 H59 D109 Q210 G211 D212 S213 G214 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=10nM remove_due_to_license_issue P20231 22192588 1263 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 4a6l C 2.05 BS01 P43 C 1 Q105 Y181 I193 D207 S208 C209 Q210 S213 V231 W233 G234 E235 G237 R243 Q87 Y162 I174 D188 S189 C190 Q191 S194 V212 W214 G215 E216 G217 R223 H59 D109 Q210 G211 D212 S213 G214 H44 D91 Q191 G192 D193 S194 G195 3.4.21.59 0004252,0005515,0005576,0005615,0006508,0008233,0008236,0062023 Ki=10nM remove_due_to_license_issue P20231 22192588 1263 IVGGQEAPRSKWPWQVSLRVHGPYWMHFCGGSLIHPQWVLTAAHCVGPDVKDLAALRVQLREQHLYYQDQLLPVSRIIVHPQFYTAQIGADIALLELEEPVKVSSHVHTVTLPPASETFPPGMPCWVTGWGDVDNDERLPPPFPLKQVKVPIMENHICDAKYHLGAYTGDDVRIVRDDMLCAGNTRRDSCQGDSGGPLVCKVNGTWLQAGVVSWGEGCAQPNRPGIYTRVTYYLDWIHHYVP 4a6s A 2.15 BS02 GS9 A 1 Y36 H50 D100 T104 N107 Y36 H50 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 24057051 1123 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4a6v A 1.46 BS03 IKY A 1 C59 Y62 Y65 C70 H79 D97 D108 H171 F177 H178 E204 W221 E235 C58 Y61 Y64 C69 H78 D96 D107 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 0006508,0070006 ic50=1.9uM remove_due_to_license_issue 22489069 1268 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDEA 4a6w A 1.46 BS02 5C1 A 1 C59 Y62 Y65 C70 H79 D97 D108 H171 F177 H178 W221 E235 C58 Y61 Y64 C69 H78 D96 D107 H170 F176 H177 W220 E234 H79 D97 D108 H171 Q175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 Q174 H177 Q181 E203 N207 Q232 E234 0006508,0070006 ic50=1.9uM remove_due_to_license_issue 22489069 1265 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGQGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 4a75 A 1.75 BS01 dna B 0 K38 W39 N41 F46 F48 D64 F66 H68 S93 K95 F97 K14 W15 N17 F22 F24 D40 F42 H44 S69 K71 F73 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 3 ~ 7 GSDPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a75 C 1.75 BS01 dna D 0 W39 N41 V42 M44 G45 F46 F48 D64 F66 H68 Q69 F77 R78 S93 K95 W13 N15 V16 M18 G19 F20 F22 D38 F40 H42 Q43 F51 R52 S67 K69 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 2 ~ 7 DPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a75 E 1.75 BS01 dna F 0 K38 W39 N41 F46 F48 D64 F66 H68 S93 K95 K13 W14 N16 F21 F23 D39 F41 H43 S68 K70 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 3 ~ 7 SDPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a75 G 1.75 BS01 dna H 0 K38 W39 N41 V42 M44 G45 F46 F48 D64 F66 H68 Q69 F77 R78 K95 F97 K13 W14 N16 V17 M19 G20 F21 F23 D39 F41 H43 Q44 F52 R53 K70 F72 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 2 ~ 7 SDPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a76 A 1.92 BS01 dna B 0 W39 N41 V42 M44 G45 F46 F48 D64 F66 H68 Q69 F77 R78 S93 K95 E98 W12 N14 V15 M17 G18 F19 F21 D37 F39 H41 Q42 F50 R51 S66 K68 E71 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 1 ~ 7 PQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a76 C 1.92 BS01 dna D 0 W39 N41 V42 M44 G45 F46 F48 D64 F66 H68 Q69 F77 R78 K95 W11 N13 V14 M16 G17 F18 F20 D36 F38 H40 Q41 F49 R50 K67 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 1 ~ 7 QVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a76 E 1.92 BS01 dna D 0 V42 R43 G45 Q69 F77 R78 V16 R17 G19 Q43 F51 R52 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 1 ~ 7 DPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a76 E 1.92 BS02 dna F 0 W39 N41 M44 F48 D64 F66 H68 S93 K95 W13 N15 M18 F22 D38 F40 H42 S67 K69 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 4 ~ 7 DPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a76 G 1.92 BS01 dna B 0 V42 R43 G45 Q69 F77 R78 V17 R18 G20 Q44 F52 R53 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 1 ~ 7 SDPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a76 G 1.92 BS02 dna H 0 W39 N41 M44 F46 F48 D64 F66 H68 S93 K95 W14 N16 M19 F21 F23 D39 F41 H43 S68 K70 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 3 ~ 7 SDPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4a7b A 2.2 BS01 3W5 A 1 G183 L184 L185 V219 H222 E223 G237 L239 F241 P242 I243 Y244 T245 T247 G80 L81 L82 V116 H119 E120 G134 L136 F138 P139 I140 Y141 T142 T144 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P45452 22153941 1000 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDED 4a7c A 2.3 BS01 E46 A 1 L44 F49 A65 K67 I104 E121 D128 L174 D186 L13 F18 A34 K36 I73 E90 D97 L143 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.006uM remove_due_to_license_issue IC50=6nM, EC50=45nM P11309 22266039 1306 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4a7i B 2.4 BS02 A7I B 1 Y99 A190 Q192 V213 W215 G216 G219 C220 G226 I227 Y228 Y85 A180 Q182 V203 W205 G206 G208 C209 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=0.002uM remove_due_to_license_issue P00742 22190348 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4a95 A 1.55 BS01 9MT A 1 V96 E97 D98 F103 F105 Y211 H213 F226 S319 L330 Y334 N365 V70 E71 D72 F77 F79 Y185 H187 F200 S293 L304 Y308 N339 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=1.73uM remove_due_to_license_issue A5K1A2 22439843 1000 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4a9c B 2.1 BS01 B5F B 1 K541 T563 S564 G565 N566 R611 Y661 T683 N684 K110 T132 S133 G134 N135 R172 Y222 T244 N245 3.1.3.86 0016791,0046856 ic50=24.8uM remove_due_to_license_issue O15357 22330088 1732 DMISVFIGTWNMGSVPPPKNVTSWFTSKGLGKTLDETIPHDIYVFGTQENSVGDREWLDLLRGGLKELTDLDYRPIAMQSLWNIKVAVLVKPEHENRISHVSTSSVKTNKGAVGVSFMFNGTSFGFVNCHLTSGNEKTARRNQNYLDILRLLSLDISLRFTHLFWFGDLNYRLDMDIQEILNYISRKEFEPLLRVDQLNLEREKHKVFLRFSEEEISFPPTYRYERGSRDTYAWHKQKPTGVRTNVPSWCDRILWKSYPETHIICNSYGCTDDIVTSDHSPVFGTFEVGVTS 4a9i A 2.25 BS01 P9I A 1 W97 V103 L108 N156 I162 W23 V29 L34 N82 I88 ? remove_due_to_license_issue P25440 22136404 1185 VTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEE 4a9m A 2.06 BS01 P9M A 1 W97 P98 F99 L108 N156 M165 W23 P24 F25 L34 N82 M91 ? ic50=0.5uM remove_due_to_license_issue IC50=500nM P25440 22136469 1187 VTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQE 4a9n A 1.85 BS01 A9N A 1 W97 P98 F99 L108 N156 M165 W23 P24 F25 L34 N82 M91 ? ic50=1.5uM remove_due_to_license_issue P25440 22136469 1190 VTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQE 4a9r A 2.85 BS01 RU5 A 1 L226 V234 K249 L301 M304 E305 G307 L354 T367 D368 L17 V19 K34 L74 M77 E78 G80 L127 T140 D141 D347 K349 N352 D368 T387 D120 K122 N125 D141 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=15nM O96017 23058106 1514 SVYPKALRDEYIMSKTLEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4a9s A 2.66 BS01 RU9 A 1 L226 K249 M304 E305 G307 L354 T367 D368 L16 K33 M76 E77 G79 L126 T139 D140 D347 K349 N352 D368 T387 D119 K121 N124 D140 T157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=61nM O96017 23058106 1515 VYPKALRDEYIMSKTLEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4a9t A 2.7 BS01 A9T A 1 L226 V234 K249 M304 G307 L354 T367 D368 L512 L18 V23 K38 M81 G84 L131 T144 D145 L289 D347 K349 N352 D368 T387 D124 K126 N129 D145 T164 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23058106 1514 MSVYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4a9u A 2.48 BS01 A9U A 1 L226 V234 K249 L301 M304 G307 L354 T367 D368 L18 V22 K37 L78 M81 G84 L131 T144 D145 D347 K349 N352 D368 T387 D124 K126 N129 D145 T162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=70nM O96017 23058106 1516 MSVYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKDPALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4aa0 A 1.8 BS01 AA0 A 1 S32 V38 A51 K53 E71 L74 I84 T106 M109 H148 L167 D168 F169 P351 S28 V34 A47 K49 E67 L70 I80 T102 M105 H137 L156 D157 F158 P328 D150 K152 N155 D168 T185 D139 K141 N144 D157 T162 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=35nM remove_due_to_license_issue IC50=420nM Q16539 22608965 1353 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 4aa4 A 2.3 BS01 QC0 A 1 V30 S32 V38 A51 K53 E71 L75 T106 L167 D168 F169 L171 V26 S28 V34 A47 K49 E67 L71 T102 L159 D160 F161 L163 D150 K152 N155 D168 T185 D142 K144 N147 D160 T177 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=9nM remove_due_to_license_issue IC50=15.85nM Q16539 22608965 1356 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQ 4aa5 A 2.38 BS01 NQB A 1 V30 S32 A51 K53 E71 L75 T106 L167 D168 F169 V26 S28 A47 K49 E67 L71 T102 L159 D160 F161 D150 K152 N155 D168 T185 D142 K144 N147 D160 T174 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=16nM remove_due_to_license_issue IC50=15.85nM Q16539 22608965 1353 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4aa7 A 2.0 BS01 R82 A 1 C385 Y387 D388 V410 C154 Y156 D157 V179 2.3.1.157,2.7.7.23 0003977,0006048,0016740,0019134 ic50=2uM remove_due_to_license_issue IC50=2000nM P0ACC7 22297115 1454 LSRLERVYQSEQAEKLLLAGVMLRDPARFDLRGTLTHGRDVEIDTNVIIEGNVTLGHRVKIGTGCVIKNSVIGDDCEISPYTVVEDANLAAACTIGPFARLRPGAELLEGAHVGNFVEMKKARLGKGSKAGHLTYLGDAEIGDNVNIGAGTITCNYDGANKFKTIIGDDVFVGSDTQLVAPVTVGKGATIAAGTTVTRNVGENALAISRVPQTQKEGWRRPV 4aa7 B 2.0 BS01 R82 B 1 C385 Y387 D388 V410 C153 Y155 D156 V178 2.3.1.157,2.7.7.23 0003977,0006048,0016740,0019134 ic50=2uM remove_due_to_license_issue IC50=2000nM P0ACC7 22297115 1454 SRLERVYQSEQAEKLLLAGVMLRDPARFDLRGTLTHGRDVEIDTNVIIEGNVTLGHRVKIGTGCVIKNSVIGDDCEISPYTVVEDANLAAACTIGPFARLRPGAELLEGAHVGNFVEMKKARLGKGSKAGHLTYLGDAEIGDNVNIGAGTITCNYDGANKFKTIIGDDVFVGSDTQLVAPVTVGKGATIAAGTTVTRNVGENALAISRVPQTQKEGWRRPV 4aac A 2.5 BS01 AAV A 1 V30 G31 S32 V38 A51 K53 E71 L75 T106 L167 D168 F169 L171 V26 G27 S28 V34 A47 K49 E67 L71 T102 L158 D159 F160 L162 D150 K152 N155 D168 T185 D141 K143 N146 D159 T176 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=6.7nM remove_due_to_license_issue IC50=4.68nM Q16539 22608965 1360 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNILTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQEEME 4aaw A 2.2 BS01 R84 A 1 V384 Y386 D387 I409 V380 Y382 D383 I405 R15 R14 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009058,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=0.5uM remove_due_to_license_issue Q8DQ18 22297115 1460 SNFAIILAAGKGTRMKSDLPKVLHKVAGISMLEHVFRSVGAIQPEKTVTVVGHKAELVEEVLAEQTEFVTQSEQLGTGHAVMMTEPILEGLSGHTLVIAGDTPLITGESLKNLIDFHINHKNVATILTAETDNPFGYGRIVRNDNAEVLRIVEQKDATDFEKQIKEINTGTYVFDNERLFEALKNINTNNEYYITDVIGIFRETGEKVGAYTLKDFDESLGVNDRVALATAESVMRRRINHKHMVNGVSFVNPEATYIDIDVEIAPEVQIEANVILKGQTKIGAETVLTNGTYVVDSTIGAGAVITNSMIEESSVADGVTVGPYAHIRPNSSLGAQVHIGNFVEVKGSSIGENTKAGHLTYIGNCEVGSNVNFGAGTITVNYDGKNKYKTVIGDNVFVGSNSTIIAPVELGDNSLVGAGSTITKDVPADAIAIGRGRQINKDEYATRLPHHPKNQ 4ab8 A 1.6 BS02 VXU A 1 D189 S190 C191 Q192 S195 V213 W215 G216 G219 C220 D171 S172 C173 Q174 S177 V191 W193 G194 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1253 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4ab9 A 1.2 BS02 VXQ A 1 D189 S190 Q192 S195 W215 G219 D171 S172 Q174 S177 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1251 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4aba A 1.25 BS02 SW1 A 1 D189 S190 C191 Q192 W215 D171 S172 C173 Q174 W193 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1256 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abb A 1.25 BS02 K9S A 1 D189 S190 C191 Q192 V213 G219 D171 S172 C173 Q174 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1252 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abd A 1.25 BS02 SW2 A 1 D189 S190 C191 Q192 V213 W215 G219 D171 S172 C173 Q174 V191 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1252 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abe A 1.3 BS02 913 A 1 D189 S190 C191 Q192 V213 W215 C220 D171 S172 C173 Q174 V191 W193 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1254 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abf A 1.3 BS02 513 A 1 D189 S190 Q192 V213 G219 C220 D171 S172 Q174 V191 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1252 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abg A 1.52 BS02 91B A 1 D189 S190 C191 Q192 V213 G219 D171 S172 C173 Q174 V191 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1255 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abh A 1.25 BS02 7Z3 A 1 D189 S190 C191 V213 W215 G216 G219 D171 S172 C173 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 22187139 1253 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 4abk A 1.6 BS01 AR6 A 1 D1235 I1236 S1247 T1248 L1254 G1257 V1258 G1303 G1304 G1332 T1333 G1334 N1335 A1336 F1371 D29 I30 S41 T42 L48 G51 V52 G97 G98 G126 T127 G128 N129 A130 F165 2.4.2.- remove_due_to_license_issue Q460N5 23473667 2389 MFYGTVSSPDSGVYEMKIGSIIFQVASGDITKEEADVIVNSTSNSFNLKAGVSKAILECAGQNVERECSQQAQQRKNDYIITGGGFLRCKNIIHVIGGNDVKSSVSSVLQECEKKNYSSICLPAIGTGNAKQHPDKVAEAIIDAIEDFVQKGSAQSVKKVKVVIFLPQVLDVFYANMKKREG 4abu A 1.86 BS01 FT1 A 1 L17 A108 S117 T118 T119 L8 A99 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.52uM remove_due_to_license_issue Kd=13.9nM, IC50=520nM P02766 22973437 1125 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4abu B 1.86 BS01 FT1 B 1 K15 L17 S117 T119 K6 L8 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.52uM remove_due_to_license_issue Kd=13.9nM, IC50=520nM P02766 22973437 1125 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4abv A 1.8 BS01 FT2 A 1 K15 L17 A108 A109 L110 S117 T118 T119 K6 L8 A99 A100 L101 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.85uM remove_due_to_license_issue Kd=5.7nM, IC50=850nM P02766 22973437 1125 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4abv B 1.8 BS01 FT2 B 1 K15 L17 A108 A109 L110 S117 T118 T119 K6 L8 A99 A100 L101 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 ic50=0.85uM remove_due_to_license_issue Kd=5.7nM, IC50=850nM P02766 22973437 1125 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4ac3 A 2.1 BS01 R83 A 1 V384 Y386 D387 I409 V381 Y383 D384 I406 R15 R14 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009058,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=110uM remove_due_to_license_issue Q8DQ18 22297115 1460 SNFAIILAAGKGTRMKSDLPKVLHKVAGISMLEHVFRSVGAIQPEKTVTVVGHKAELVEEVLAEQTEFVTQSEQLGTGHAVMMTEPILEGLSGHTLVIAGDTPLITGESLKNLIDFHINHKNVATILTAETDNPFGYGRIVRNDNAEVLRIVEQKDATDFEKQIKEINTGTYVFDNERLFEALKNINTNNGEYYITDVIGIFRETGEKVGAYTLKDFDESLGVNDRVALATAESVMRRRINHKHMVNGVSFVNPEATYIDIDVEIAPEVQIEANVILKGQTKIGAETVLTNGTYVVDSTIGAGAVITNSMIEESSVADGVTVGPYAHIRPNSSLGAQVHIGNFVEVKGSSIGENTKAGHLTYIGNCEVGSNVNFGAGTITVNYDGKNKYKTVIGDNVFVGSNSTIIAPVELGDNSLVGAGSTITKDVPADAIAIGRGRQINKDEYATRLPHHPKNQ 4acc A 2.21 BS01 7YG A 1 I62 F67 A83 K85 Y134 V135 R141 L188 D200 I28 F33 A49 K51 Y100 V101 R107 L154 D166 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 Ki=20nM remove_due_to_license_issue Ki=20nM P49841 22489897 1387 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 4acd A 2.6 BS01 GR9 A 1 F67 A83 K85 D133 Y134 V135 P136 T138 R141 L188 D200 F33 A49 K51 D99 Y100 V101 P102 T104 R107 L154 D166 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue Ki=4.9nM P49841 22489897 1385 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 4acf A 2.0 BS01 46B A 1 Y129 F232 H278 Q279 W282 N359 K361 R364 Y126 F229 H275 Q276 W279 N356 K358 R361 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E130 E132 E216 E224 H273 R344 E363 R365 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 remove_due_to_license_issue P9WN39 1479 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSIHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 4acf F 2.0 BS01 46B F 1 Y129 F232 H278 W282 N359 K361 R364 Y126 F229 H275 W279 N356 K358 R361 D54 E133 E135 E219 E227 H276 R347 E366 R368 D51 E130 E132 E216 E224 H273 R344 E363 R365 6.3.1.2 0000287,0001968,0003824,0004356,0005524,0005576,0005737,0005829,0005886,0006542,0009274,0010756,0016020,0016874,0019740,0035375,0046872,0051260 remove_due_to_license_issue P9WN39 1479 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGSSIRGFQSIHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 4acg A 2.6 BS01 6LQ A 1 I62 A83 K85 Y134 V135 P136 R141 Q185 N186 L188 C199 D200 I28 A49 K51 Y100 V101 P102 R107 Q151 N152 L154 C165 D166 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 22489897 1385 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 4ach A 2.6 BS01 KDI A 1 I62 A83 D133 Y134 V135 P136 R141 L188 C199 I28 A49 D99 Y100 V101 P102 R107 L154 C165 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue Ki=22nM P49841 22489897 1386 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 4aci A 1.65 BS01 CIT A 1 N77 G78 L79 V80 R130 N134 M140 E181 R185 N67 G68 L69 V70 R120 N124 M130 E171 R175 ? 0000287,0000976,0003677,0003700,0006355,0046872 remove_due_to_license_issue Q8NQ97 23589369 1189 NSRQEILEGARRCFAEHGYEGATVRRLEEATGKSRGAIFHHFGDKENLFLALAREDAARMAEVVSENGLVEVMRGMLEDPERYDWMSVRLEISKQLRTDPVFRAKWIDHQSVLDEAVRVRLSRNVDKGQMRTDVPIEVLHTFLETVLDGFISRLATGASTEGLSEVLDLVEGTVRK 4acm A 1.63 BS01 7YG A 1 I10 V18 A31 E81 F82 L83 D86 K89 L134 D145 I10 V18 A31 E72 F73 L74 D77 K80 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T144 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=210nM remove_due_to_license_issue P24941 22489897 1302 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4acu A 1.75 BS01 QN7 A 1 G11 G13 L30 D32 S35 Y71 Q73 F108 I110 W115 I118 D228 S229 G230 T231 T232 G15 G17 L34 D36 S39 Y75 Q77 F112 I114 W119 I122 D218 S219 G220 T221 T222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=40.7nM remove_due_to_license_issue IC50=20nM P56817 22325942 1506 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLEDCGY 4acx A 2.0 BS01 S8Z A 1 Q12 G13 L30 D32 S35 N37 Y71 Q73 W76 F108 I110 I118 R128 D228 G230 T232 Q14 G15 L32 D34 S37 N39 Y73 Q75 W78 F110 I112 I120 R130 D216 G218 T220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D216 T219 3.4.23.46 0004190,0006508,0016020 ic50=77.6nM remove_due_to_license_issue P56817 22325942 1504 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLEDCGY 4ad2 A 2.1 BS01 GLC A 1 H63 R295 E333 H335 E336 H29 R261 E299 H301 E302 3.2.1.130 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 22219371 500 TELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 4ad2 A 2.1 BS02 IFM A 1 Y46 W126 H154 E156 Y195 Y252 E333 E336 Y12 W92 H120 E122 Y161 Y218 E299 E302 3.2.1.130 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 22219371 501 TELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 4ad3 A 2.0 BS01 GLC A 1 H63 I294 R295 E333 H335 E336 H29 I260 R261 E299 H301 E302 3.2.1.130 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 22219371 500 TELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 4ad3 A 2.0 BS02 DMJ A 1 Y46 H154 E156 Y195 Y252 E333 E336 Y12 H120 E122 Y161 Y218 E299 E302 3.2.1.130 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 22219371 501 TELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 4ad6 A 1.85 BS01 GSY A 1 T43 A44 V46 F54 N56 D95 F123 T45 A46 V48 F56 N58 D97 F125 R83 R92 D95 D97 R85 R94 D97 D99 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656 Kd=16.7uM remove_due_to_license_issue A0A0H3JKY1 23565155 1159 SHMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRYK 4ad6 A 1.85 BS02 GSY B 1 P109 K110 P111 K112 R83 R92 D95 D97 R85 R94 D97 D99 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656 Kd=16.7uM remove_due_to_license_issue A0A0H3JKY1 23565155 1159 SHMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRYK 4ael A 2.2 BS02 4HN A 1 I692 Y693 F696 P712 M713 E721 V722 G725 Q726 F729 I245 Y246 F249 P265 M266 E274 V275 G278 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=12nM remove_due_to_license_issue IC50=12nM Q9Y233 22321214 1769 ASICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIR 4af3 A 2.75 BS01 VX6 A 1 L83 F88 V91 A104 K106 E155 Y156 A157 P158 G160 L207 L14 F19 V22 A35 K37 E86 Y87 A88 P89 G91 L138 D200 K202 E204 N205 D218 D131 K133 E135 N136 D149 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=18nM, IC50=30nM, Kd=7.4nM Q96GD4 22920039 500 RHFTIDDFEIGRPLGKGKFGNVYLAREKKSHFIVALKVLFKSQIEKEGVEHQLRREIEIQAHLHHPNILRLYNYFYDRRRIYLILEYAPRGELYKELQKSCTFDEQRTATIMEELADALMYCHGKKVIHRDIKPENLLLGLKGELKIADFGLDYLPPEMIEGRMHNEKVDLWCIGVLCYELLVGNPPFESASHNETYRRIVKVDLKFPASVPTGAQDLISKLLRHNPSERLPLAQVSAHPWVRANSRRVLPPS 4afe A 2.597 BS01 GGY A 1 I14 Y19 C22 V35 M86 E87 Y88 C89 F148 D159 F160 I12 Y17 C20 V33 M84 E85 Y86 C87 F139 D150 F151 D141 K143 A145 N146 D159 T179 D132 K134 A136 N137 D150 T156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=800nM P51955 22404346 1280 SRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSHRDLKPANVFLDGKQNVKLGDFGLVGTPYYMSPEQMNRNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 4afg A 2.001 BS01 QMR A 1 W153 V154 Y194 C197 Y201 W152 V153 Y193 C196 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=5nM remove_due_to_license_issue I6L8L2 22619328 1214 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afg A 2.001 BS02 QMR B 1 I118 I128 I117 I127 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=5nM remove_due_to_license_issue I6L8L2 22619328 1214 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afg B 2.001 BS01 QMR A 1 I118 I128 I117 I127 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=5nM remove_due_to_license_issue I6L8L2 22619328 1214 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afg B 2.001 BS02 QMR E 1 W153 Y194 C197 Y201 W152 Y193 C196 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=5nM remove_due_to_license_issue I6L8L2 22619328 1214 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afh A 1.88 BS01 L0B A 1 F102 F150 G151 S152 W153 Y194 C196 C197 Y201 F102 F150 G151 S152 W153 Y194 C196 C197 Y201 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=0.29nM remove_due_to_license_issue I6L8L2 22619328 1216 SNGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afh A 1.88 BS02 L0B E 1 I118 L126 I128 I118 L126 I128 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=0.29nM remove_due_to_license_issue I6L8L2 22619328 1218 SNGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afh B 1.88 BS01 L0B A 1 I118 L126 I128 I118 L126 I128 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=0.29nM remove_due_to_license_issue I6L8L2 22619328 1216 SNGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afh B 1.88 BS02 L0B B 1 F102 F150 G151 S152 W153 Y194 C197 Y201 E203 F102 F150 G151 S152 W153 Y194 C197 Y201 E203 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=0.29nM remove_due_to_license_issue I6L8L2 22619328 1218 SNGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRSE 4afj A 1.98 BS02 SJJ A 1 F67 A83 Y134 V135 P136 L188 D200 F32 A48 Y94 V95 P96 L148 D160 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=398nM remove_due_to_license_issue IC50=1995nM P49841 22310227 1391 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 4aft A 3.2 BS01 QMR A 1 Y91 W145 Y186 C188 Y193 Y91 W145 Y186 C188 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 22553201 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4aft A 3.2 BS02 QMR E 1 V106 I116 V106 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 22553201 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4aft B 3.2 BS01 QMR A 1 M114 I116 M114 I116 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 22553201 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4aft B 3.2 BS02 QMR B 1 Y91 W145 Y186 Y193 Y91 W145 Y186 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 22553201 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4ag8 A 1.95 BS01 AXI A 1 V848 A866 K868 E885 V914 V916 F918 C919 K920 G922 L1035 C1045 D1046 F1047 V33 A51 K53 E70 V99 V101 F103 C104 K105 G107 L163 C173 D174 F175 D1028 A1030 R1032 N1033 D1046 K1055 D1064 D156 A158 R160 N161 D174 K183 D192 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 Ki=1.1nM remove_due_to_license_issue P35968 22988103 2000 HCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 4agc A 2.0 BS01 AXI A 1 V848 A866 K868 E885 V914 V916 E917 F918 C919 K920 G922 L1035 C1045 D1046 F1047 A1168 V41 A59 K61 E78 V107 V109 E110 F111 C112 K113 G115 L171 C181 D182 F183 A304 D1028 A1030 R1032 N1033 D1046 D1064 D164 A166 R168 N169 D182 D200 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 Ki=0.02nM remove_due_to_license_issue P35968 22988103 2000 YLSIVMDPDELPLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 4agd A 2.81 BS01 B49 A 1 L840 K868 V899 F918 C919 K920 G922 L1035 D1046 F1047 A1168 L32 K60 V91 F110 C111 K112 G114 L170 D181 F182 A303 D1028 A1030 R1032 N1033 D1046 D1064 D163 A165 R167 N168 D181 D199 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=18900nM, Kd=1.5nM, Ki=9nM P35968 22988103 2000 LSIVMDPDELPLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 4agl A 1.7 BS01 P84 A 1 L145 V147 T150 P151 C220 E221 P222 P223 T230 L50 V52 T55 P56 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=225uM remove_due_to_license_issue P04637 22439615 400 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 4agm A 1.52 BS01 P86 A 1 L145 V147 D148 T150 C220 E221 P222 P223 T230 L50 V52 D53 T55 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=105uM remove_due_to_license_issue P04637 22439615 400 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 4agn A 1.6 BS02 NXG A 1 L145 V147 D148 T150 P151 P152 P153 C220 P222 P223 T230 L50 V52 D53 T55 P56 P57 P58 C125 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=107uM remove_due_to_license_issue P04637 22439615 1294 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 4ago A 1.45 BS01 P74 A 1 L145 V147 D148 T150 P151 C220 E221 P222 P223 T230 L50 V52 D53 T55 P56 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=15.5uM remove_due_to_license_issue P04637 22439615 1292 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 4agp A 1.5 BS01 P51 A 1 L145 V147 D148 T150 P151 C220 E221 P222 P223 T230 L50 V52 D53 T55 P56 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=20.6uM remove_due_to_license_issue P04637 22439615 1292 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 4agq A 1.42 BS01 P96 A 1 L145 V147 D148 T150 P151 C220 E221 P222 P223 T230 L50 V52 D53 T55 P56 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=9.7uM remove_due_to_license_issue Kd=10000nM P04637 22439615 1291 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 4ah9 A 1.7 BS01 0MB A 1 R107 P109 I204 I208 R52 P54 I147 I151 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 218 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQTK 4ah9 A 1.7 BS02 0MB B 1 Y83 H185 G197 E198 Y28 H130 G140 E141 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 218 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQTK 4ah9 B 1.7 BS01 0MB A 1 Y83 H185 G197 E198 Y28 H130 G138 E139 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 218 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ah9 B 1.7 BS02 0MB B 1 R107 P109 I204 I208 R52 P54 I145 I149 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 218 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ahr A 1.9 BS01 I2E A 1 G106 R107 P109 G51 R52 P54 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1218 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQT 4ahr A 1.9 BS02 I2E B 1 H185 G197 E198 H130 G140 E141 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1217 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQT 4ahr B 1.9 BS01 I2E A 1 H185 G197 E198 H130 G140 E141 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1218 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQT 4ahr B 1.9 BS02 I2E B 1 G106 R107 W108 P109 I208 G51 R52 W53 P54 I151 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1217 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQT 4ahs A 1.75 BS01 AKH A 1 R107 W108 P109 R51 W52 P53 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 4ahs A 1.75 BS02 AKH B 1 H185 G197 E198 V201 H129 G137 E138 V141 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1218 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 4ahs B 1.75 BS01 AKH A 1 H185 G197 V201 H129 G138 V142 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQT 4ahs B 1.75 BS02 AKH B 1 R107 W108 P109 R51 W52 P53 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1218 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQT 4ahu A 1.9 BS01 ICO A 1 H185 G197 E198 H130 G140 E141 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1217 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQT 4ahu A 1.9 BS02 ICO B 1 R107 P109 I208 R52 P54 I151 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1220 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGGYSAGERIVDIIATDIQT 4ahu B 1.9 BS01 ICO A 1 R107 P109 I208 R52 P54 I150 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1217 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQTK 4ahu B 1.9 BS02 ICO B 1 N184 H185 G197 E198 V201 N129 H130 G139 E140 V143 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1220 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDIQTK 4ahv A 1.8 BS01 Z5P A 1 H185 G197 E198 V201 H129 G137 E138 V141 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1219 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ahv A 1.8 BS02 Z5P B 1 G106 R107 W108 P109 I208 G50 R51 W52 P53 I148 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ahv B 1.8 BS01 Z5P A 1 G106 R107 W108 P109 I208 G51 R52 W53 P54 I149 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1219 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ahv B 1.8 BS02 Z5P B 1 H185 G197 E198 V201 H130 G138 E139 V142 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 23139382 1216 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ai5 A 2.22 BS02 ADK A 1 F6 Y13 W21 E38 W46 F8 Y15 W23 E40 W48 0003824,0006281,0006284,0008725 Kd=1.2mM remove_due_to_license_issue 22684054 400 GAMNECAFGTKDPVYLNFHDHVWGQPLYDSKALFKLLALESQHAGLSWLTILKKKEAYEEAFYDFEPEKVAQMTAQDIDRLMTFPNIVHHRKKLEAIVNQAQGYLKIEQAYGSFSKFLWSYVNGKPKDLQYEHASDRITVDDTATQLSKDLKQYGFKFLGPVTVFSFLEAAGLYDAHLKDCPSKPKHN 4ai8 A 2.4 BS01 DZA A 1 Y145 T196 H199 D201 N205 F207 K214 H279 Y135 T186 H189 D191 N195 F197 K204 H269 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50>100uM remove_due_to_license_issue IC50=>100000nM Q9NWT6 22724510 1358 SGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 4aia A 1.8 BS02 ADK A 1 Y13 W21 E38 W46 Y15 W23 E40 W48 0003824,0006281,0006284,0008725 Kd=220uM remove_due_to_license_issue 22684054 400 GAMNECAFGTKDPVYLNYHDHVWGQPLYDSKALFKLLALESQHAGLSWLTILKKKEAYEEAFYDFEPEKVAQMTAQDIDRLMTFPNIVHHRKKLEAIVNQAQGYLKIEQAYGSFSKFLWSYVNGKPKDLQYEHASDRITVDDTATQLSKDLKQYGFKFLGPVTVFSFLEAAGLYDAHLKDCPSKPKHN 4aig A 2.0 BS03 FLX A 1 K106 I107 I108 T139 H142 E143 H146 H152 I165 R167 P168 G169 L170 K105 I106 I107 T138 H141 E142 H145 H151 I164 R166 P167 G168 L169 3.4.24.46 0004222,0005576,0005886,0006508,0008237,0046872 ic50=0.3uM remove_due_to_license_issue P34179 9428736 400 NLPQRYIELVVVADRRVFMKYNSDLNIIRTRVHEIVNIINEFYRSLNIRVSLTDLEIWSGQDFITIQSSSSNTLNSFGEWRERVLLTRKRHDNAQLLTAINFEGKIIGKAYTSSMCNPRSSVGIVKDHSPINLLVAVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTPGRSYEFSDDSMGYYQKFLNQYKPQCILNKP 4aij A 2.05 BS01 dna C 0 S48 Q49 Q60 P61 V64 R86 A87 K88 S46 Q47 Q58 P59 V62 R84 A85 K86 ? 0000976,0001216,0001217,0003677,0003700,0006355,0006950,0032993,0045892,0045893 remove_due_to_license_issue B1JJ73 22936808 1 ~ 21 STLGSDLARLVRVWRALIDHRLKPLELTQTHWVTLYNINRLPPEQSQIQLAKAIGIEQPSLVRTLDQLEEKGLITRHTSANDRRAKRIKLTEQSSPIIEQVDGVISSTRKEILGGISSDEIAVLSGLIDKLEKNIIQLQ 4aij A 2.05 BS02 dna D 0 T32 E59 P61 S62 T30 E57 P59 S60 ? 0000976,0001216,0001217,0003677,0003700,0006355,0006950,0032993,0045892,0045893 remove_due_to_license_issue B1JJ73 22936808 1 ~ 21 STLGSDLARLVRVWRALIDHRLKPLELTQTHWVTLYNINRLPPEQSQIQLAKAIGIEQPSLVRTLDQLEEKGLITRHTSANDRRAKRIKLTEQSSPIIEQVDGVISSTRKEILGGISSDEIAVLSGLIDKLEKNIIQLQ 4aij B 2.05 BS01 dna C 0 T32 P61 S62 R85 T31 P60 S61 R84 ? 0000976,0001216,0001217,0003677,0003700,0006355,0006950,0032993,0045892,0045893 remove_due_to_license_issue B1JJ73 22936808 1 ~ 21 ESTLGSDLARLVRVWRALIDHRLKPLELTQTHWVTLYNINRLPPEQSQIQLAKAIGIEQPSLVRTLDQLEEKGLITRHTSANDRRAKRIKLTEQSSPIIEQVDGVISSTRKEILGGISSDEIAVLSGLIDKLEKNIIQLQTK 4aij B 2.05 BS02 dna D 0 Q49 P61 V64 R78 R86 K88 Q48 P60 V63 R77 R85 K87 ? 0000976,0001216,0001217,0003677,0003700,0006355,0006950,0032993,0045892,0045893 remove_due_to_license_issue B1JJ73 22936808 1 ~ 21 ESTLGSDLARLVRVWRALIDHRLKPLELTQTHWVTLYNINRLPPEQSQIQLAKAIGIEQPSLVRTLDQLEEKGLITRHTSANDRRAKRIKLTEQSSPIIEQVDGVISSTRKEILGGISSDEIAVLSGLIDKLEKNIIQLQTK 4aik A 1.85 BS01 dna C 0 Q49 Q60 V64 R78 R86 K88 Q47 Q58 V62 R76 R84 K86 ? 0000976,0001216,0001217,0003677,0003700,0006355,0006950,0032993,0045892,0045893 remove_due_to_license_issue B1JJ73 22936808 1 ~ 21 STLGSDLARLVRVWRALIDHRLKPLELTQTHWVTLYNINRLPPEQSQIQLAKAIGIEQPSLVRTLDQLEEKGLITRHTSANDRRAKRIKLTEQSSPIIEQVDGVISSTRKEILGGISSDEIAVLSGLIDKLEKNIIQLQ 4aik A 1.85 BS02 dna D 0 T32 P61 S62 D84 R85 R86 T30 P59 S60 D82 R83 R84 ? 0000976,0001216,0001217,0003677,0003700,0006355,0006950,0032993,0045892,0045893 remove_due_to_license_issue B1JJ73 22936808 1 ~ 21 STLGSDLARLVRVWRALIDHRLKPLELTQTHWVTLYNINRLPPEQSQIQLAKAIGIEQPSLVRTLDQLEEKGLITRHTSANDRRAKRIKLTEQSSPIIEQVDGVISSTRKEILGGISSDEIAVLSGLIDKLEKNIIQLQ 4aj1 A 1.87 BS01 AJ1 A 1 D51 V52 A95 G96 I115 D47 V48 A91 G92 I111 R105 D165 R168 H192 R101 D161 R164 H188 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=770uM remove_due_to_license_issue Kd=1.000e+6nM, IC50=>5.00e+5nM P04642 22417091 1333 ALKDQLIVNLLKVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4aj2 A 1.75 BS01 52C A 1 D51 V52 Y82 I115 F118 I119 D47 V48 Y78 I111 F114 I115 R105 D165 R168 H192 R101 D161 R164 H188 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 remove_due_to_license_issue Kd=4.200e+6nM, IC50=>5.00e+5nM P04642 22417091 1333 ALKDQLIVNLLKVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4aj4 A 1.9 BS01 VAB A 1 G28 D51 V52 A95 G96 I115 F118 G27 D50 V51 A94 G95 I114 F117 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=130uM remove_due_to_license_issue Kd=1.30e+5nM, IC50=>5.00e+5nM P04642 22417091 1333 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4aje A 2.35 BS01 2B4 A 1 V30 Q99 R105 V135 N137 L164 R168 H192 T247 V26 Q95 R101 V131 N133 L160 R164 H188 T243 R105 D165 R168 H192 R101 D161 R164 H188 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=210uM remove_due_to_license_issue Kd=4.70e+5nM, IC50=>5.00e+5nM P04642 22417091 1332 ALKDQLIVNLLKVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4aje B 2.35 BS01 2B4 B 1 V30 Q99 R105 V135 S136 N137 R168 H192 A237 T247 V29 Q98 R104 V134 S135 N136 R167 H191 A236 T246 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=210uM remove_due_to_license_issue Kd=4.70e+5nM, IC50=>5.00e+5nM P04642 22417091 1333 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4aji A 1.93 BS01 88R A 1 V30 T94 R98 R105 V135 N137 R168 H192 T247 I251 V26 T90 R94 R101 V131 N133 R164 H188 T243 I247 R105 D165 R168 H192 R101 D161 R164 H188 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=280uM remove_due_to_license_issue Kd=1.000e+6nM, IC50=>5.00e+5nM P04642 22417091 1332 ALKDQLIVNLLKVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4aji B 1.93 BS01 88R B 1 V30 T94 Q99 R105 N137 L164 R168 H192 A237 T247 V29 T93 Q98 R104 N136 L163 R167 H191 A236 T246 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=280uM remove_due_to_license_issue Kd=1.000e+6nM, IC50=>5.00e+5nM P04642 22417091 1332 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajk A 2.03 BS01 88S A 1 G28 D51 V52 T94 A95 G96 I115 I119 G27 D50 V51 T93 A94 G95 I114 I118 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=770uM remove_due_to_license_issue Kd=7.70e+5nM, IC50=>5.00e+5nM P04642 22417091 1332 AALKDQLIVNLLKEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajl A 1.77 BS01 88W A 1 G26 G28 D51 V52 T94 A95 G96 I115 G23 G25 D48 V49 T91 A92 G93 I112 R105 D165 R168 H192 R102 D162 R165 H189 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=160uM remove_due_to_license_issue Kd=1.60e+5nM, IC50=>5.00e+5nM P04642 22417091 1333 ALKDQLIVNLLKQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajn A 2.1 BS01 88V A 1 V30 D51 V52 T94 A95 G96 R105 I115 N137 L164 R168 H192 T247 V28 D49 V50 T92 A93 G94 R103 I113 N135 L162 R166 H190 T245 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.069uM remove_due_to_license_issue Kd=69nM, IC50=1.9e+3nM P04642 22417091 1332 ALKDQLIVNLLKEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajn B 2.1 BS01 88V B 1 V30 D51 V52 T94 A95 G96 R98 Q99 R105 I115 I119 N137 R168 H192 A237 T247 V29 D50 V51 T93 A94 G95 R97 Q98 R104 I114 I118 N136 R167 H191 A236 T246 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.069uM remove_due_to_license_issue Kd=69nM, IC50=1.9e+3nM P04642 22417091 1333 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajo A 1.96 BS01 88N A 1 V30 D51 V52 T94 A95 G96 R105 I115 N137 L164 R168 H192 A237 T247 V29 D50 V51 T93 A94 G95 R104 I114 N136 L163 R167 H191 A236 T246 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.093uM remove_due_to_license_issue P04642 22417091 1332 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajo B 1.96 BS01 88N B 1 V30 D51 V52 T94 A95 G96 R98 Q99 R105 I119 N137 R168 H192 A237 T247 V28 D49 V50 T92 A93 G94 R96 Q97 R103 I117 N135 R166 H190 A235 T245 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.093uM remove_due_to_license_issue P04642 22417091 1333 ALKDQLIVNLLKEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4ajw A 2.8 BS01 VWN A 1 M752 P758 W760 I777 Y813 V828 M511 P517 W519 I536 Y572 V587 2.7.1.137,2.7.1.153 0001782,0002250,0005524,0005737,0005829,0006629,0006935,0006954,0007166,0010628,0016301,0016303,0030154,0036092,0042113,0043491,0045087,0045766,0046854,0046934,0048872,0050832 remove_due_to_license_issue O35904 22524426 2027 KKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNQPFSIELIEGRKVNAVQAGLFHGNEMLCKTDISVCDLPRMARLCFALYADCPIAWANLMLFDYKDQLKTGERCLYMWPSLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLTAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRES 4akn A 1.82 BS01 S5B A 1 W97 F99 L108 N156 I162 W23 F25 L34 N82 I88 ? ic50=0.79uM remove_due_to_license_issue IC50=794.33nM P25440 22437115 1188 VTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQE 4al4 A 1.78 BS01 W7E A 1 V30 D51 V52 T94 A95 G96 R105 I115 I119 V135 N137 R168 H192 A237 T247 I251 V29 D50 V51 T93 A94 G95 R104 I114 I118 V134 N136 R167 H191 A236 T246 I250 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.13uM remove_due_to_license_issue IC50=4.2e+3nM, Kd=1.3e+2nM P04642 22417091 1333 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4al4 A 1.78 BS02 W7E A 2 G28 A29 V52 A97 R98 R111 I115 G27 A28 V51 A96 R97 R110 I114 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.13uM remove_due_to_license_issue IC50=4.2e+3nM, Kd=1.3e+2nM P04642 22417091 1334 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4al4 B 1.78 BS01 W7E B 1 V30 D51 V52 T94 A95 G96 R98 Q99 R105 I115 I119 V135 N137 L164 R168 H192 A237 T247 I251 V29 D50 V51 T93 A94 G95 R97 Q98 R104 I114 I118 V134 N136 L163 R167 H191 A236 T246 I250 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.13uM remove_due_to_license_issue IC50=4.2e+3nM, Kd=1.3e+2nM P04642 22417091 1332 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4al4 B 1.78 BS02 W7E B 2 G28 A29 A97 R98 R111 I115 G27 A28 A96 R97 R110 I114 R105 D165 R168 H192 R104 D164 R167 H191 1.1.1.27 0001666,0001889,0003824,0004457,0004459,0005515,0005737,0005739,0005829,0006089,0006090,0007519,0007584,0009410,0009749,0014070,0016491,0016616,0019661,0019674,0019752,0019900,0035686,0042542,0042802,0042867,0043065,0043627,0051287,0051591,1990204 Kd=0.13uM remove_due_to_license_issue IC50=4.2e+3nM, Kd=1.3e+2nM P04642 22417091 1333 ALKDQLIVNLLKEEQVPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLKTPKIVSSKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPQCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPQLGTDADKEQWKDVHKQVVDSAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGIKEDVFLSVPCILGQNGISDVVKVTLTPDEEARLKKSADTLWGIQKELQF 4alg A 1.6 BS01 1GH A 1 W51 P52 F53 V57 L62 N110 I116 M119 W26 P27 F28 V32 L37 N85 I91 M94 ? ic50=0.5uM remove_due_to_license_issue IC50=501.19nM, Kd=70nM, Ki=50nM P25440 22437115 1146 PGRVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQELVV 4alp A 1.48 BS01 rna E 0 G45 Q69 F77 R78 G19 Q43 F51 R52 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 1 ~ 6 DPQVLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4alp D 1.48 BS01 rna E 0 G45 Q69 F77 R78 G16 Q40 F48 R49 ? 0003676 remove_due_to_license_issue B4F6I0 22570413 1 ~ 6 VLRGSGHCKWFNVRMGFGFISMTSREGSPLENPVDVFVHQSKLYMEGFRSLKEGEPVEFTFKKSSKGFESLRVTGPGGNPCLGN 4alu A 2.6 BS01 79O A 1 G45 S46 S49 V52 A65 K67 R122 L174 I185 D186 G13 S14 S17 V20 A33 K35 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=17nM P11309 22542012 1308 PLESQYQVGPLLGSGGSGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4alv A 2.59 BS01 R9P A 1 G45 F49 A65 K67 L120 R122 D128 F130 D131 E171 L174 I185 D186 G13 F17 A33 K35 L88 R90 D96 F98 D99 E139 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=7.0nM P11309 22542012 1308 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4alw A 1.92 BS01 HY7 A 1 F49 V52 A65 K67 E121 R122 N172 L174 I185 D186 F16 V19 A32 K34 E88 R89 N139 L141 I152 D153 D167 K169 N172 D186 L193 T204 D134 K136 N139 D153 L160 T171 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=27nM remove_due_to_license_issue IC50=27nM P11309 22542012 1308 LESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4alx F 2.3 BS01 IZN F 1 Y89 W143 Y185 C187 Y192 Y89 W143 Y185 C187 Y192 ? 0004888,0005216,0005230,0006811,0016020,0034220 Ki=52nM remove_due_to_license_issue P58154 22927902 400 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4alx F 2.3 BS02 IZN J 1 W53 L112 M114 W53 L112 M114 ? 0004888,0005216,0005230,0006811,0016020,0034220 Ki=52nM remove_due_to_license_issue P58154 22927902 400 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4alx G 2.3 BS01 IZN F 1 W53 R104 L112 M114 W53 R104 L112 M114 ? 0004888,0005216,0005230,0006811,0016020,0034220 Ki=52nM remove_due_to_license_issue P58154 22927902 400 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4alx G 2.3 BS02 IZN G 1 Y89 W143 Y185 C187 Y192 Y89 W143 Y181 C183 Y188 ? 0004888,0005216,0005230,0006811,0016020,0034220 Ki=52nM remove_due_to_license_issue P58154 22927902 400 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4aml A 1.6 BS01 GYU A 1 S62 Y64 Y66 E72 Y73 S62 Y64 Y66 E72 Y73 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1172 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 4aml A 1.6 BS02 GYU A 2 D86 S105 W107 F109 F116 D86 S105 W107 F109 F116 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1173 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 4aml A 1.6 BS03 GYU B 1 S114 E115 S114 E115 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1171 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 4aml A 1.6 BS04 GYU B 2 A71 E72 A71 E72 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1172 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCDG 4aml B 1.6 BS01 GYU A 1 S114 E115 S114 E115 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1172 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCD 4aml B 1.6 BS02 GYU A 2 A71 E72 A71 E72 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1173 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCD 4aml B 1.6 BS03 GYU B 1 S62 Y64 Y66 E72 Y73 S62 Y64 Y66 E72 Y73 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1171 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCD 4aml B 1.6 BS04 GYU B 2 D86 S105 W107 F109 F116 D86 S105 W107 F109 F116 ? 0008061,0030246 remove_due_to_license_issue P10968 20527753 1172 ERCGEQGSNMECPNNLCCSQYGYCGMGGDYCGKGCQNGACWTSKRCGSQAGGATCTNNQCCSQYGYCGFGAEYCGAGCQGGPCRADIKCGSQAGGKLCPNNLCCSQWGFCGLGSEFCGGGCQSGACSTDKPCGKDAGGRVCTNNYCCSKWGSCGIGPGYCGAGCQSGGCD 4amx A 2.1 BS01 5GF A 1 F373 D412 Y513 W551 D553 R649 W662 D665 F698 H731 F360 D399 Y500 W538 D540 R636 W649 D652 F685 H718 4.2.2.13 0003824,0004553,0005975,0016798,0016829,0030246,0047457 remove_due_to_license_issue Q9STC1 23902768 1039 TDNPDGIDYKTYDYVGVWGFSPLSNTNWFAAGSSTPGGITDWTATMNVNFDRIDNPSITVQHPVQVQVTSYNNNSYRVRFNPDGPIRDVTRGPILKQQLDWIRTQELSEGCDPGMTFTSEGFLTFETKDLSVIIYGNFKTRVTRKSDGKVIMENDEVGTASSGNKCRGLMFVDRLYGNAIASVNKNFRNDAVKQEGFYGAGEVNCKYQDTYILERTGIAMTNYNYDNLNYNQWDLRPPHHDGALNPDYYIPMYYAAPWLIVNGCAGTSEQYSYGWFMDNVSQSYMNTGDTTWNSGQEDLAYMGAQYGPFDQHFVYGAGGGMECVVTAFSLLQGKEFENQVLNKRSVMPPKYVFGFFQGVFGTSSLLRAHMPAGENNISVEEIVEGYQNNNFPFEGLAVDVDMQDNLRVFTTKGEFWTANRVGTGGDPNNRSVFEWAHDKGLVCQTNITCFLRNDNEGQDYEVNQTLRERQLYTKNDSLTGTDFGMTDDGPSDAYIGHLDYGGGVECDALFPDWGRPDVAEWWGNNYKKLFSIGLDFVWQDMTVPAMMPHKIGDDINVKPDGNWPNADDPSNGQYNWKTYHPQVLVTDMRYENHGREPMVTQRNIHAYTLCESTRKEGIVENADTLTKFRRSYIISRGGYIGNQHFGGMWVGDNSTTSNYIQMMIANNINMNMSCLPLVGSDIGGFTSYDNENQRTPCTGDLMVRYVQAGCLLPWFRNHYDRWIESKDHGKDYQELYMYPNEMDTLRKFVEFRYRWQEVLYTAMYQNAAFGKPIIKAASMYNNDSNVRRAQNDHFLLGGHDGYRILCAPVVWENSTERELYLPVLTQWYKFGPDFDTKPLEGAMNGGDRIYNYPVPQSESPIFVREGAILPTRYTLNGENKSLNTYTDEDPLVFEVFPLGNNRADGMCYLDDGGVTTNAEDNGKFSVVKVAAEQDGGTETITFTNDCYEYVFGGPFYVRVRGAQSPSNIHVSSGAGSQDMKVSSATSRAALFNDGENGDFWVDQETDSLWLKLPNVVLPDAVITIT 4amy A 2.0 BS01 2P2 A 1 F173 M235 G254 C255 Y473 F476 S554 N555 I591 W595 R643 H680 F173 M235 G254 C255 Y473 F476 S554 N555 I591 W595 R643 H680 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 22484394 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4amz A 2.0 BS01 2P4 A 1 F173 M235 Y473 F476 S554 N555 A594 W595 R643 H680 F173 M235 Y473 F476 S554 N555 A594 W595 R643 H680 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 22484394 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4an0 A 2.2 BS01 2P6 A 1 F173 M235 G254 Y473 F476 S554 N555 A594 W595 R643 V644 F173 M235 G254 Y473 F476 S554 N555 A594 W595 R643 V644 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue IC50=6nM, Ki=0.100000nM P23687 22484394 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4an1 A 1.9 BS01 2P8 A 1 F173 M235 Y473 F476 S554 N555 A594 W595 R643 H680 F173 M235 Y473 F476 S554 N555 A594 W595 R643 H680 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 22484394 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4an2 A 2.5 BS01 EUI A 1 N78 K97 V127 I141 D190 D208 F209 V211 S212 L215 G225 N21 K40 V70 I84 D133 D151 F152 V154 S155 L158 G168 D190 K192 S194 N195 D208 D217 T226 D133 K135 S137 N138 D151 D160 T169 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=4.2nM Q02750 24900486 1382 MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL 4an3 A 2.1 BS03 5Y0 A 1 K97 V127 I141 D208 F209 V211 L215 K40 V70 I84 D151 F152 V154 L158 D190 K192 S194 N195 D208 D217 T226 D133 K135 S137 N138 D151 D160 T167 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue Q02750 24900486 1384 MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL 4an9 A 2.8 BS03 2P7 A 1 K97 L118 V127 I141 M143 D190 D208 F209 G210 V211 L215 K40 L61 V70 I84 M86 D133 D151 F152 G153 V154 L158 D190 K192 S194 N195 D208 D217 T226 D133 K135 S137 N138 D151 D160 T168 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=44nM Q02750 24900486 1384 MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL 4anb A 2.2 BS01 YQY A 1 K97 V127 I141 D208 F209 V211 L215 K40 V70 I84 D151 F152 V154 L158 D190 K192 S194 N195 D208 D217 T226 D133 K135 S137 N138 D151 D160 T169 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=6.6nM Q02750 24900486 501 MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL 4anm A 1.7 BS01 WUL A 1 R47 V53 I66 K68 V116 N161 M163 I174 D175 R42 V48 I61 K63 V111 N156 M158 I169 D170 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=28nM remove_due_to_license_issue P28523 22560567 1334 SSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 4anq A 1.76 BS01 VGH A 1 A1148 M1199 A1200 G1202 R1214 N1254 L1256 A1269 D1270 Y1401 A46 M97 A98 G100 R112 N152 L154 A167 D168 Y293 D1249 A1251 R1253 N1254 D1270 L1291 D147 A149 R151 N152 D168 L183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=605nM remove_due_to_license_issue IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 24432909 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIADFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 4anu A 2.81 BS01 EM7 A 1 W812 I831 Y867 I879 I881 V882 M953 I963 D964 W570 I589 Y625 I637 I639 V640 M711 I721 D722 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=21nM P48736 22548342 2089 SSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 4anv A 2.13 BS01 751 A 1 M804 P810 W812 I831 K833 Y867 I879 E880 V882 T887 M953 I963 D964 M574 P580 W582 I601 K603 Y637 I649 E650 V652 T657 M723 I733 D734 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=441nM remove_due_to_license_issue IC50=441nM P48736 22548342 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEETVSLWDCDRKFRVKIRGIDIPVLPRNLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNYCHPIALPKHQRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPELTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLH 4anw A 2.31 BS01 O92 A 1 M804 S806 W812 I831 K833 Y867 I879 V882 M953 I963 D964 M562 S564 W570 I589 K591 Y625 I637 V640 M711 I721 D722 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=18nM remove_due_to_license_issue IC50=18nM P48736 22548342 1189 SSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 4anx A 2.73 BS01 534 A 1 M804 I831 K833 Y867 I879 E880 I881 V882 T887 D950 M953 I963 D964 M562 I589 K591 Y625 I637 E638 I639 V640 T645 D708 M711 I721 D722 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=18nM P48736 22548342 2088 SSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 4aoc A 2.7 BS03 A1Q A 1 A29 A30 E31 D110 H112 D113 D115 D118 A18 A19 E20 D99 H101 D102 D104 D107 ? 0046872 remove_due_to_license_issue A0A0H2Y045 22763039 1131 EFSIPPNTDFRAIFFANAAEQQHIKLFIGDSQEPAAYHKLTTRDGPREATLNSGNGKIRFEVSVNGKPSATDARLAPINGKKSDGSPFTVNFGIVVSEDGHDSDYNDGIVVLQWPIG 4aoc B 2.7 BS03 A1Q B 1 A30 E31 D110 H112 D113 D115 D118 A22 E23 D102 H104 D105 D107 D110 ? 0046872 remove_due_to_license_issue A0A0H2Y045 22763039 1131 RAGEFSIPPNTDFRAIFFANAAEQQHIKLFIGDSQEPAAYHKLTTRDGPREATLNSGNGKIRFEVSVNGKPSATDARLAPINGKKSDGSPFTVNFGIVVSEDGHDSDYNDGIVVLQWPIG 4aof A 3.3 BS01 7L0 A 1 W812 I831 Y867 E880 V882 M953 I963 D964 W569 I588 Y624 E637 V639 M710 I720 D721 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=79.43nM P48736 22544264 2095 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLGI 4aoi A 1.9 BS01 4K0 A 1 I1084 A1108 L1157 P1158 M1160 D1164 N1167 R1208 M1211 A1221 D1222 Y1230 I33 A53 L102 P103 M105 D109 N112 R153 M156 A166 D167 Y175 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.004uM remove_due_to_license_issue IC50=16nM, Ki=4nM P08581 22924734 2345 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 4ap0 A 2.594 BS02 G7X A 1 E116 G117 E118 R119 W127 I136 P137 L160 Y211 L214 G217 R221 E96 G97 E98 R99 W107 I116 P117 L140 Y191 L194 G197 R201 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=2.3nM, IC50=47nM P52732 22993085 2001 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKEVKIGKLNLVDLAGSENIGRINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 4ap7 A 1.8 BS01 F47 A 1 A1108 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 F1344 A53 M105 D109 R153 M156 A166 D167 Y175 F289 D1204 A1206 R1208 N1209 D1222 A1243 D149 A151 R153 N154 D167 A188 2.7.10.1 0004672,0004713,0005524,0006468 Ki=0.011uM remove_due_to_license_issue Ki=11nM, IC50=7nM P08581 22924734 2345 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 4app A 2.2 BS01 N53 A 1 G330 G333 V335 A348 K350 E396 F397 L398 G401 D405 L447 D458 R586 T590 G32 G35 V37 A50 K52 E98 F99 L100 G103 D107 L149 D160 R288 T292 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 Ki=0.064uM remove_due_to_license_issue Ki=64nM, EC50=810nM O96013 22554206 601 MSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNRT 4aq3 A 2.4 BS01 398 A 1 F63 Y67 D70 M74 E95 L96 F36 Y40 D43 M47 E68 L69 ? 0042981 ic50=37nM remove_due_to_license_issue P10415,Q07817 22608961 1163 YDNREIVMKYIHYKLSQRGYEWDVVHLALRQAGDDFSRRYRGDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 4aq3 A 2.4 BS02 398 E 1 Q58 L160 Y161 G162 Q31 L133 Y134 G135 ? 0042981 ic50=37nM remove_due_to_license_issue P10415,Q07817 22608961 1163 YDNREIVMKYIHYKLSQRGYEWDVVHLALRQAGDDFSRRYRGDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 4aq4 A 1.8 BS01 G3P A 1 Y42 E66 S121 W169 W172 S247 G283 G284 Y323 R374 Y46 E70 S125 W173 W176 S251 G287 G288 Y327 R378 ? 0001407,0015794,0016020,0030288,0042597,0055085,1902517 Kd=0.68uM remove_due_to_license_issue P0AG80 23013274 1415 GSHMVTTIPFWHSMEGELGKEVDSLAQRFNAENPDYKIVPTYKGNYEQNLSAGIAAFRTGNAPAILQVYEVGTATMMASKAIKPVYDVFKEAGIQFDESQFVPTVSGYYSDSKTGHLLSQPFNSSTPVLYYNKDAFKKAGLDPEQPPKTWQDLADYAAKLKASGMKCGYASGWQGWIQLENFSAWNGLPFASKNNGFDGTDAVLEFNKPEQVKHIAMLEEMNKKGDFSYVGRKDESTEKFYNGDCAMTTASSGSLANIREYAKFNYGVGMMPYDADAKDAPQNAIIGGASLWVMQGKDKETYTGVAKFLDFLAKPENAAEWHQKTGYLPITKAAYDLTREQGFYEKNPGADTATRQMLNKPPLPFTKGLRLGNMPQIRVIVDEELESVWTGKKTPQQALDTAVERGNQLLRRFEKSTK 4aq6 A 1.98 BS02 OMD A 1 H288 P291 P328 E337 M339 Y346 H367 H280 P283 P320 E329 M331 Y338 H359 H288 H331 E337 H361 H367 H280 H323 E329 H353 H359 1.13.11.5 0000976,0001217,0004411,0005506,0005737,0006520,0006559,0006570,0006572,0032993,0045892,0046872,0051213 remove_due_to_license_issue Q88E47 23858455 838 LHYLSGFGNEFASEALPGALPVGQNSPQKAPYGLYAELLSGTAFTMARSELRRTWLYRIRPSALHPRFERLARQPLGGPLGGINPNRLRWSPQPIPAEPTDFIEGWLPMAANAGAEKPAGVSIYIYRANRSMERVFFNADGELLLVPEQGRLRIATELGVMEVEPLEIAVIPRGMKFRVELLDGQARGYIAENHGAPLRLPDLGPIGSNGLANPRDFLTPVAHYEEAEGPVQLVQKFLGEHWACELQHSPLDVVAWHGSNVPYKYDLRRFNTIGTVSFDHPDPSIFTVLTSPTSVHGMANMDFVIFPPRWMVAENTFRPPWFHRNLMNEFMGLINGAYDAKAEGFLPGGASLHGVMSAHGPDAETCEKAIAADLAPHKIDNTMAFMFETSQVLRPSLQALECPQLQADYDSCWATLPSTFNPNRR 4aq6 B 1.98 BS02 OMD B 1 H288 P291 P328 M339 Y346 H367 H280 P283 P320 M331 Y338 H359 H288 H331 E337 H361 H367 H280 H323 E329 H353 H359 1.13.11.5 0000976,0001217,0004411,0005506,0005737,0006520,0006559,0006570,0006572,0032993,0045892,0046872,0051213 remove_due_to_license_issue Q88E47 23858455 838 LHYLSGFGNEFASEALPGALPVGQNSPQKAPYGLYAELLSGTAFTMARSELRRTWLYRIRPSALHPRFERLARQPLGGPLGGINPNRLRWSPQPIPAEPTDFIEGWLPMAANAGAEKPAGVSIYIYRANRSMERVFFNADGELLLVPEQGRLRIATELGVMEVEPLEIAVIPRGMKFRVELLDGQARGYIAENHGAPLRLPDLGPIGSNGLANPRDFLTPVAHYEEAEGPVQLVQKFLGEHWACELQHSPLDVVAWHGSNVPYKYDLRRFNTIGTVSFDHPDPSIFTVLTSPTSVHGMANMDFVIFPPRWMVAENTFRPPWFHRNLMNEFMGLINGAYDAKAEGFLPGGASLHGVMSAHGPDAETCEKAIAADLAPHKIDNTMAFMFETSQVLRPSLQALECPQLQADYDSCWATLPSTFNPNRR 4aqc A 1.9 BS01 88A A 1 L855 G856 K857 G858 V863 A880 V911 M929 Y931 L932 G935 L983 G993 L14 G15 K16 G17 V22 A39 V70 M88 Y90 L91 G94 L142 G152 D976 A978 R980 N981 D994 S1016 D135 A137 R139 N140 D153 S175 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.9nM remove_due_to_license_issue IC50=0.9nM O60674 22594690 2001 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4aqh A 2.4 BS01 TB7 A 1 Y37 S41 L75 R76 L78 Y79 T94 D95 F117 R118 Y40 S44 L78 R79 L81 Y82 T97 D98 F120 R121 ? 0001525,0002020,0004867,0005102,0005515,0005576,0005615,0005886,0010469,0010757,0010951,0014912,0030194,0030195,0030336,0031093,0032757,0033629,0035491,0042730,0045766,0048260,0050729,0050829,0051918,0061044,0061045,0062023,0070062,0071222,0090026,0090399,0097180,0097187,1901331,1902042,1904090,2000098,2000352 remove_due_to_license_issue P05121 23155046 1380 SHMVHHPPSYVAHLASDFGVRVFQQVAQASKDRNVVFSPYGVASVLAMLQLTTGGETQQQIQAAMGFKIDDKGMAPALRHLYKELMGPWNKDEISTTDAIFVQRDLKLVQGFMPHFFRLFRSTVKQVDFSEVERARFIINDWVKTHTKGMISNLLGKGAVDQLTRLVLVNALYFNGQWKTPFPDSSTHRRLFHKSDGSTVSVPMMAQTNKFNYTEFTTPDGHYYDILELPYHGDTLSMFIAAPYEKEVPLSALTNILSAQLISHWKGNMTRLPRLLVLPKFSLETEVDLRKPLENLGMTDMFRQFQADFTSLSDQEPLHVAQALQKVKIEVNESGTVASSSTAVIVSARMAPEEIIMDRPFLFVVRHNPTGTVLFMGQVMEP 4aqu A 2.3 BS01 dna C 0 K28 S32 Y33 K34 Q38 Y66 R68 R70 E80 I81 K116 D137 K139 K27 S31 Y32 K33 Q37 Y65 R67 R69 E79 I80 K115 D136 K138 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 22740697 401 ~ 424 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 4aqu A 2.3 BS02 dna D 0 D20 S22 Q26 K28 Q44 T46 Q47 K48 R70 V73 N136 D137 S138 T140 R141 K142 D19 S21 Q25 K27 Q43 T45 Q46 K47 R69 V72 N135 D136 S137 T139 R140 K141 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 22740697 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 4aqu B 2.3 BS01 dna C 0 D220 G221 S222 Q226 K228 Q244 T246 Q247 K248 R270 N336 D337 S338 R341 K342 T343 D19 G20 S21 Q25 K27 Q43 T45 Q46 K47 R69 N135 D136 S137 R140 K141 T142 G219 D220 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 22740697 401 ~ 424 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 4aqu B 2.3 BS02 dna D 0 S232 Y233 K234 Q238 R268 R270 E280 I281 K316 D337 K339 T340 S31 Y32 K33 Q37 R67 R69 E79 I80 K115 D136 K138 T139 G219 D220 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 22740697 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSYKFKHQLSLTFQVTQKTQRRWFLDKLVDEIGVGYVRDRGSVSDYILSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLD 4ara A 2.5 BS01 C56 A 1 D74 W86 Y124 W286 I294 F295 R296 Y337 F338 Y341 D74 W86 Y124 W279 I287 F288 R289 Y330 F331 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd=0.9uM remove_due_to_license_issue P21836 23161758 600 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4arb A 2.25 BS01 C57 A 1 D74 W86 Y124 W286 I294 F295 R296 Y337 F338 Y341 D74 W86 Y124 W279 I287 F288 R289 Y330 F331 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd=1.3uM remove_due_to_license_issue P21836 23161758 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4ark A 2.6 BS03 M3K A 1 K97 V127 M143 D190 D208 F209 V211 L215 M219 K37 V67 M83 D130 D148 F149 V151 L155 M159 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T166 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue Q02750 23474388 1385 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 4aro A 1.59 BS01 IHS A 1 R18 H19 R22 T25 K26 R94 H128 T219 F257 H306 D307 R15 H16 R19 T22 K23 R89 H123 T207 F245 H294 D295 3.1.3.26 0030288,0050308 remove_due_to_license_issue H9TUK5 23741456 501 APAGFQLEKVVILSRHGVRAPTKMTQTMRDVTPHQWPEWPVKLGYITPRGEHLISLMGGFYRERFQQQGLLPKCPTPDAVYVWADVDQRTRKTGEAFLAGLAPQCDLAIHHQQNTQQADPLFHPVKAGICSMDKSQVHAAVEKQAGTPIETLNQRYQASLALMSSVLDFPKSPYCQQHLCDFSQAMPSRLAIGNKVALEGAVGLASTLAEIFLLEHAQGMPKVAWGNIHTEQQWNSLLKLHNAQFDLMSRTPYIAKHNGTPLLQTIAHALGSNITSRPLPDISPDNKILFIAGHDANIANISGMLGMTWTLPGQPDNTPPGGALVFERWVDNAGKPYVSVNMVYQTLAQLHDQAPLTLQHPAGSVRLNIPGCSDQTPDGYCPLSTFSRLVSHSVEPACQLP 4aro A 1.59 BS02 IHS A 2 P43 P51 R52 Q230 M232 P40 P48 R49 Q218 M220 3.1.3.26 0030288,0050308 remove_due_to_license_issue H9TUK5 23741456 502 APAGFQLEKVVILSRHGVRAPTKMTQTMRDVTPHQWPEWPVKLGYITPRGEHLISLMGGFYRERFQQQGLLPKCPTPDAVYVWADVDQRTRKTGEAFLAGLAPQCDLAIHHQQNTQQADPLFHPVKAGICSMDKSQVHAAVEKQAGTPIETLNQRYQASLALMSSVLDFPKSPYCQQHLCDFSQAMPSRLAIGNKVALEGAVGLASTLAEIFLLEHAQGMPKVAWGNIHTEQQWNSLLKLHNAQFDLMSRTPYIAKHNGTPLLQTIAHALGSNITSRPLPDISPDNKILFIAGHDANIANISGMLGMTWTLPGQPDNTPPGGALVFERWVDNAGKPYVSVNMVYQTLAQLHDQAPLTLQHPAGSVRLNIPGCSDQTPDGYCPLSTFSRLVSHSVEPACQLP 4arw A 2.204 BS01 HNR A 1 S41 L45 Y113 Y114 G115 V250 A251 E255 S42 L46 Y114 Y115 G116 V251 A252 E256 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 Kd=0.074uM remove_due_to_license_issue IC50=2.1e+2nM Q9HU22 23138692 400 HHHRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4as9 A 2.71 BS01 4QS A 1 N37 A41 K44 M84 E88 N92 K98 G121 V122 F124 T171 V213 E214 N36 A40 K43 M83 E87 N91 K97 G120 V121 F123 T170 V212 E213 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 23511419 1215 ASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 4asd A 2.03 BS01 BAX A 1 L840 V848 A866 K868 E885 L889 V916 E917 F918 C919 G922 L1019 L1035 I1044 C1045 D1046 F1047 L34 V42 A60 K62 E79 L83 V110 E111 F112 C113 G116 L156 L172 I181 C182 D183 F184 D1028 A1030 R1032 N1033 D1046 D1064 D165 A167 R169 N170 D183 D201 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 Ki=0.52nM remove_due_to_license_issue IC50=90nM, Kd=59nM, Ki=22nM, EC50=500nM P35968 22988103 1500 DPDELPLDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 4ase A 1.83 BS01 AV9 A 1 L840 V848 A866 K868 E885 L889 V916 C919 L1035 C1045 D1046 F1047 N1167 A1168 L34 V42 A60 K62 E79 L83 V110 C113 L172 C182 D183 F184 N304 A305 D1028 A1030 R1032 N1033 D1046 D1064 D165 A167 R169 N170 D183 D201 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 Ki=0.01nM remove_due_to_license_issue P35968 22988103 3169 DPDELPLDEHCERLPYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARDIYKDPDYVRKGDARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 4asj A 2.25 BS01 N6A A 1 S41 L45 Y113 G115 F118 V250 E255 S40 L44 Y112 G114 F117 V249 E254 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 Kd=0.028uM remove_due_to_license_issue IC50=73nM Q9HU22 23138692 1294 KRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4asj C 2.25 BS01 N6A C 1 S41 L45 Y113 H119 V250 E255 S40 L44 Y112 H118 V249 E254 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 Kd=0.028uM remove_due_to_license_issue IC50=73nM Q9HU22 23138692 1294 KRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4ask A 1.86 BS02 K0I A 1 R1246 T1330 N1331 Y1379 K1381 T1387 P1388 H1390 E1392 N1393 N1400 N1480 R70 T124 N125 Y173 K175 T181 P182 H184 E186 N187 N194 N274 1.14.11.68 remove_due_to_license_issue IC50=16nM O15054 22842901 2639 PREKLNPPTPSIYLESKRDAFSPVLLQFCTDPRNPITVIRGLAGSLRLNLGLFSTKTLVEASGEHTVEVRTQVQQPSDENWDLTGTRQIWPCESSRSHTTIAKYAQYQASSFQESLHHIIKFGTNIDLSDAKRWKPQLQELLKLPAFMRVTSTGNMLSHVGHTILGMNTVQLYMKVPGSRTPGHQENNNFCSVNINIGPGDCEWFAVHEHYWETISAFCDRHGVDYLTGSWWPILDDLYASNIPVYRFVQRPGDLVWINAGTVHWVQATGWCNNIAWNVGPLTAYQYQLALERYEWNEVKNVKSIVPMIHVSWNVARTVKISDPDLFKMIKFCLLQSMKHCQVQRESLVRAGKKIAYQGRVKDEPAYYCNECDVEVFNILFVTSENTYLVHCEGCARRRSAGLQGVVVLEQYRTEELAQAYDAFTLAP 4asy A 2.3 BS01 N5Y A 1 S41 T42 L45 Y113 G115 V250 E255 S41 T42 L45 Y113 G115 V250 E255 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 remove_due_to_license_issue IC50=>6.0e+4nM Q9HU22 23138692 1294 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4asy B 2.3 BS01 N5Y B 1 S41 L45 Y113 G115 V250 E255 S40 L44 Y112 G114 V249 E254 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 remove_due_to_license_issue IC50=>6.0e+4nM Q9HU22 23138692 1294 KRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4at3 A 1.77 BS01 LTI A 1 L560 F565 A586 F633 Y635 M636 G639 N697 L699 G709 L21 F26 A43 F88 Y90 M91 G94 N150 L152 G162 D692 A694 R696 N697 D710 S719 L731 D145 A147 R149 N150 D163 S170 L182 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.004uM remove_due_to_license_issue Q16620 22902478 1839 GAMDTFVQHIKRHNIVLKRELGEGAFGKVFLAECYNLCKILVAVKTLASDNARKDFHREAELLTNLQHEHIVKFYGVCVEGDPLIMVFEYMKHGDLNKFLRAHGPDAVLMANPPTELTQSQMLHIAQQIAAGMVYLASQHFVHRDLATRNCLVGENLLVKIGDFGMSRYSTDYYRVGGHTMLPIRWMPPESIMYRKFTTESDVWSLGVVLWEIFTYGKQPWYQLSNNEVIECITQGRVLQRPRTCPQEVYELMLGCWQREPHMRKNIKGIHTLLQNLAKASPVYLDILG 4at4 A 2.36 BS01 T6E A 1 A586 L608 F633 Y635 M636 F688 L699 I708 G709 D710 F711 A43 L65 F90 Y92 M93 F142 L153 I162 G163 D164 F165 D692 A694 R696 N697 D710 S719 L731 D146 A148 R150 N151 D164 S173 L185 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.012uM remove_due_to_license_issue Q16620 22902478 1839 GAMDTFVQHIKRHNIVLKRELGEGAFGKVFLAECYNLCKILVAVKTLKDASDNARKDFHREAELLTNLQHEHIVKFYGVCVEGDPLIMVFEYMKHGDLNKFLRAHGPDAVLMAPPTELTQSQMLHIAQQIAAGMVYLASQHFVHRDLATRNCLVGENLLVKIGDFGMSRDVYSTDYYRVGGHTMLPIRWMPPESIMYRKFTTESDVWSLGVVLWEIFTYGKQPWYQLSNNEVIECITQGRVLQRPRTCPQEVYELMLGCWQREPHMRKNIKGIHTLLQNLAKASPVYLDILG 4at5 A 1.71 BS01 MUJ A 1 A586 L608 V617 F633 Y635 M636 F688 N697 L699 G709 D710 F711 A42 L64 V73 F89 Y91 M92 F144 N153 L155 G165 D166 F167 D692 A694 R696 N697 D710 S719 L731 D148 A150 R152 N153 D166 S175 L187 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.038uM remove_due_to_license_issue Kd=36nM Q16620 22902478 1839 GAMDTFVQHIKRHNIVLKRELGEGAFGKVFLAECYNLKILVAVKTLKDASDNARKDFHREAELLTNLQHEHIVKFYGVCVEGDPLIMVFEYMKHGDLNKFLRAHGPDAVLMAEGNPPTELTQSQMLHIAQQIAAGMVYLASQHFVHRDLATRNCLVGENLLVKIGDFGMSRDVYSTDYYRVGGHTMLPIRWMPPESIMYRKFTTESDVWSLGVVLWEIFTYGKQPWYQLSNNEVIECITQGRVLQRPRTCPQEVYELMLGCWQREPHMRKNIKGIHTLLQNLAKASPVYLDILG 4ati A 2.6 BS01 dna C 0 H209 N210 R217 N221 K243 H1 N2 R9 N13 K31 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 HNLIERRRRFNINDRIKELGTLIPKSMRWNKGTILKASVDYIRKLQREQQRAKDLEN 4ati A 2.6 BS02 dna D 0 H209 I212 E213 R216 H1 I4 E5 R8 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 HNLIERRRRFNINDRIKELGTLIPKSMRWNKGTILKASVDYIRKLQREQQRAKDLEN 4ati B 2.6 BS01 dna C 0 H209 I212 E213 R216 H7 I10 E11 R14 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 RQKKDNHNLIERRRRFNINDRIKELGTLIPKSDPDMRWNKGTILKASVDYIRKLQREQQRAKDLENRQKKL 4ati B 2.6 BS02 dna D 0 K206 H209 N210 E213 R214 R217 N242 K243 K4 H7 N8 E11 R12 R15 N39 K40 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 RQKKDNHNLIERRRRFNINDRIKELGTLIPKSDPDMRWNKGTILKASVDYIRKLQREQQRAKDLENRQKKL 4atk A 2.95 BS01 dna C 0 H209 N210 R240 K243 H3 N4 R32 K35 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 DNHNLIERRRRFNINDRIKELGTLIPKDPDMRWNKGTILKASVDYIRKLQREQQRAKDLE 4atk A 2.95 BS02 dna D 0 H209 I212 E213 R215 H3 I6 E7 R9 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 DNHNLIERRRRFNINDRIKELGTLIPKDPDMRWNKGTILKASVDYIRKLQREQQRAKDLE 4atk B 2.95 BS01 dna C 0 E213 R216 E9 R12 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 KKDNHNLIERRRRFNINDRIKELGTLIPKSNDPDMRWNKGTILKASVDYIRKLQREQQRA 4atk B 2.95 BS02 dna D 0 H209 N210 E213 R214 R217 F218 N242 K243 H5 N6 E9 R10 R13 F14 N38 K39 ? 0046983 remove_due_to_license_issue Q08874 23207919 1 ~ 16 KKDNHNLIERRRRFNINDRIKELGTLIPKSNDPDMRWNKGTILKASVDYIRKLQREQQRA 4att A 1.251 BS01 HNV A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 Y137 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=104.6nM remove_due_to_license_issue P08191 24900609 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4au7 A 2.07 BS02 SAH A 1 H32 Y114 E117 G120 A121 F160 A179 N182 H183 Y217 F222 E230 C231 H29 Y111 E114 G117 A118 F157 A176 N179 H180 Y214 F219 E227 C228 2.1.1.361,2.1.1.362 0042799 remove_due_to_license_issue Q6Q783 24049080 1247 DRVTARELCENDDLATSLVLDPYLGFRTHKMNVSPVPTLRRQHHLRSALEAFLRQRDLEAAFRALTLGGWMAHYFQSRAPRQEAALKTHIFCYLRAFLPESGFTILPCTRYSMETNGAKIVSTRAWKKNEKLELLVGCIAELREEDEDLLRAGENDFSIMYSTRKRSAQLWLGPAAFINHDCKPNCKFVPSDGNTACVKVLRDIEPGDEVTCFYGEGFFGEKNEHCECYTCERKGEGAFRLQP 4au8 A 1.9 BS01 Z3R A 1 I10 V18 F80 C83 D84 Q85 D86 K89 L133 D144 I11 V19 F69 C72 D73 Q74 D75 K78 L122 D133 D126 K128 Q130 N131 D144 T164 D115 K117 Q119 N120 D133 T151 2.7.11.1 0000226,0000307,0001764,0001963,0002039,0004672,0004674,0004676,0004677,0004679,0004693,0004694,0004711,0005176,0005515,0005524,0005634,0005654,0005737,0005829,0005874,0005886,0006338,0006468,0006886,0006915,0007160,0007268,0007399,0007409,0007416,0007519,0008017,0008045,0008306,0008542,0014044,0014069,0016020,0016079,0016241,0016301,0016310,0016477,0016533,0018105,0018107,0019233,0021537,0021549,0021695,0021697,0021766,0021819,0021954,0021987,0022038,0030027,0030036,0030054,0030175,0030182,0030334,0030424,0030425,0030426,0030517,0030549,0030900,0031175,0031397,0031594,0031914,0032801,0035175,0035249,0035402,0035403,0035418,0035979,0042220,0042981,0042995,0043005,0043025,0043113,0043125,0043204,0043525,0044022,0044023,0044024,0044025,0045202,0045786,0045861,0045892,0045956,0046826,0048148,0048156,0048167,0048488,0048489,0048511,0048675,0048709,0048813,0050321,0051301,0051402,0051649,0051726,0051879,0051966,0060078,0060079,0061001,0070509,0072354,0072371,0072518,0090314,0098793,0106310,0140823,0140855,0140857,1901987,1903076,1903421,1904646,1990244 ic50=551nM remove_due_to_license_issue Q00535 22889803 1293 GSQKYEKLEKIGEGTYGTVFKAKNRETHEIVALKRVPSSALREICLLKELKHKNIVRLHDVLHKLTLVFEFCDQDLKKYFDSCNGDLDPEIVKSFLFQLLKGLGFCHSRNVLHRDLKPQNLLINRNGELKLADFGLARAFGIPVRSAEVVTLWYRPPDVLFGAKLYSTSIDMWSAGCIFAELANAGRPLFPGNDVDDQLKRIFRLLGTPTEEQWPSMTKLPDYKPYPMYPATTSLVNVVPKLNATGRDLLQNLLKCNPVQRISAEEALQHPYFSDF 4aua A 2.31 BS01 4AU A 1 I19 A41 E99 H100 V101 D102 Q103 D104 L152 I9 A30 E68 H69 V70 D71 Q72 D73 L121 D145 K147 Q149 N150 D163 T182 D114 K116 Q118 N119 D132 T137 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 ic50=7.2uM remove_due_to_license_issue IC50=7200nM Q00534 24900493 1302 QQYECVAEIGEGAGKVFKARDLKNGGRFVALKRSTIREVAVLRHLETFEHPNVVRLFDVCTKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLATLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPRDVALPRQAFHSKSAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQ 4auj A 1.527 BS01 HNW A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 ? 0007155,0009289 Kd=18.3nM remove_due_to_license_issue P08191 24900609 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4auy A 2.102 BS01 HNW A 1 F1 N46 D54 Q133 N135 D140 F1 N46 D54 Q133 N135 D140 ? 0007155,0009289 Kd=18.3nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4av0 A 2.099 BS01 HNV A 1 F1 N46 Y48 D54 Q133 N135 Y137 D140 F1 N46 Y48 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=104.6nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4av4 A 1.9 BS01 FVQ A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 Y137 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=94.3nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVNLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4av5 A 1.4 BS01 FYZ A 1 F1 I13 N46 Y48 I52 D54 Q133 N135 Y137 D140 F1 I13 N46 Y48 I52 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=61nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4avg A 2.2 BS01 SL6 A 1 H41 E80 D108 E119 Y130 K134 K137 H43 E78 D106 E117 Y128 K132 K135 3.1.-.- 0003723,0039694 ic50=0.06uM remove_due_to_license_issue C3W5S0 22876177 801 MAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVENALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERG 4avh A 2.105 BS01 FK9 A 1 F1 N46 D47 Y48 D54 Q133 N135 Y137 D140 F1 N46 D47 Y48 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=59.5nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4avi A 2.4 BS01 XNS A 1 F1 N46 Y48 I52 D54 Q133 N135 Y137 D140 F1 N46 Y48 I52 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=23.6nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4avj A 2.105 BS01 J73 A 1 F1 N46 D47 Y48 D54 Q133 N135 D140 F1 N46 D47 Y48 D54 Q133 N135 D140 ? 0007155,0009289 Kd=36.5nM remove_due_to_license_issue P08191 22657089 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4avs A 1.399 BS03 N7P A 1 N59 Y64 Y74 E136 D138 Q148 N59 Y64 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 remove_due_to_license_issue P02743 25084341 208 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 4avt C 3.2 BS03 GHE C 1 N59 Y64 E136 D138 Q148 N59 Y64 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 remove_due_to_license_issue P02743 25084341 1207 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 4avu A 2.4 BS02 LDR A 1 H1031 G1032 Y1050 Y1060 S1068 Y1071 I1075 H80 G81 Y99 Y109 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24900770 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4avw A 2.15 BS01 G18 A 1 H1031 G1032 Y1050 Y1060 K1067 S1068 Y1071 H80 G81 Y99 Y109 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24900770 2162 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4aw5 A 2.33 BS01 30K A 1 I97 A121 K123 M172 E173 G175 L223 I15 A39 K41 M90 E91 G93 L141 D216 A218 R220 N221 D234 P259 D134 A136 R138 N139 D152 P156 2.7.10.1 0004672,0004713,0005524,0006468 ic50=765nM remove_due_to_license_issue P54760 22765894 1365 AKEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 4awf A 2.3 BS03 XI7 A 1 H41 R84 D108 E119 K134 H45 R80 D104 E115 K130 3.1.-.- 0003723,0039694 ic50=2.7uM remove_due_to_license_issue C3W5S0 22876177 303 SGMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFISIIVEPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERGE 4awg A 2.6 BS01 CI3 A 1 E23 Y24 A37 I38 H41 E80 R84 D108 E119 K134 E26 Y27 A40 I41 H44 E77 R81 D105 E116 K131 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 22876177 801 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awi A 1.91 BS01 AQ2 A 1 S34 V40 A53 K55 M111 S155 L168 S27 V33 A46 K48 M104 S148 L161 D151 K153 N156 D169 T188 D144 K146 N149 D162 T176 2.7.11.24 0004672,0004707,0005524,0006468 ic50=1uM remove_due_to_license_issue P45983 22801646 1365 NNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 4awj C 2.5 BS01 V6F C 1 W88 Y98 H110 S111 Y112 H115 W117 W27 Y37 H49 S50 Y51 H54 W56 ? Kd~10000uM remove_due_to_license_issue Kd=4900000nM P40337 23102223 1201 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLER 4awk A 1.9 BS01 CI1 A 1 A20 E23 Y24 E26 K34 I38 H41 E80 R84 L106 D108 E119 K134 A21 E24 Y25 E27 K35 I39 H42 E60 R64 L86 D88 E99 K114 3.1.-.- 0003723,0039694 ic50=0.13uM remove_due_to_license_issue C3W5S0 22876177 801 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4awm A 2.6 BS03 KDH A 1 Y24 E26 K34 A37 I38 H41 E80 D108 E119 K134 Y25 E27 K35 A38 I39 H42 E64 D92 E103 K118 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 22876177 911 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 4awm A 2.6 BS04 KDH A 2 D83 I85 D67 I69 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 22876177 921 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 4awo A 1.7 BS01 99B A 1 F22 Q23 N51 M98 L103 N105 N106 L107 F138 Y139 W162 F170 F6 Q7 N35 M82 L87 N89 N90 L91 F119 Y120 W143 F151 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=24nM remove_due_to_license_issue P07900 22877636 1225 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQDISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4awp A 1.82 BS01 99A A 1 F22 Q23 N51 M98 L103 I104 N106 L107 F138 Y139 W162 F170 F6 Q7 N35 M82 L87 I88 N90 L91 F119 Y120 W143 F151 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=81nM remove_due_to_license_issue P07900 22877636 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQDISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4awq A 1.6 BS01 592 A 1 F22 Q23 N51 M98 L103 I104 N106 I110 F138 Y139 W162 F170 T184 V186 F6 Q7 N35 M82 L87 I88 N90 I94 F119 Y120 W143 F151 T165 V167 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=479nM remove_due_to_license_issue IC50=479nM P07900 22877636 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQDISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4ax9 H 1.9 BS03 N5N H 1 H57 Y60A E97A N98 L99 D189 A190 C191 S195 W215 G216 E217 G219 H43 Y47 E94 N95 L96 D192 A193 C194 S198 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.00027uM remove_due_to_license_issue Ki=0.3nM P00734 7966150 1246 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4axa A 1.9 BS02 RKD A 1 G50 T51 G55 R56 V57 A70 K72 E121 Y122 E127 E170 N171 M173 T183 D184 G37 T38 G42 R43 V44 A57 K59 E108 Y109 E114 E157 N158 M160 T170 D171 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 22781553 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4axd A 2.05 BS01 ANP A 1 E18 G19 G20 A21 N22 V24 R40 N147 D148 H149 E166 M372 I406 D407 E18 G19 G20 A21 N22 V24 R40 N147 D148 H149 E166 M372 I405 D406 2.7.1.158 0005524,0005634,0005737,0010264,0016301,0030643,0032942,0035299,0042742,0046872,0048527,0050832,0051607,0055062,0102731 Kd=37uM remove_due_to_license_issue Q93YN9 22745128 600 MEMILEEKDASDWIYRGEGGANLVLAYAGSSPLFVGKVIRIQKARRNDKAIKNSNGVVSVLTSDEQHLWRENNELISSPNKEVLEQRYVQNVIIPLLGPKHVDAGVRVSVSKEFLECVDKKVTKQRPLARVNAANVDTSHDSALILNDHSLFSQGITSGGDCISVEIKPKCGFLPTSRFIGKENMLKTSVSRFKMHQLLKLEYIEISEESEYDPLDLFSGSKERVLEAIKALYSTPQNNFRVFLNGSLILGGSGESTGRTSPEIGYAFEDALKGFIQSEDGHRTECFLQLVSDAVYGSGVLDRLLEIQKLDKLDIEGAIHCYYDIINQPCPICREGRPLEAELSLHALPLDESLKIVKEYLIAATAKDCSIMISFQSRNAWDSEPGDYVSLKPTNQTFDYKVHFIDLSLKPLKRMESYYKLDKKIISFYNRKQ 4axm A 2.8 BS01 V65 A 1 G23 C25 G67 G68 L69 D162 H163 G164 G23 C25 G67 G68 L69 D162 H163 G164 Q19 C25 H163 N187 Q19 C25 H163 N185 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 23658062 1222 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESSDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 4ay5 A 3.15 BS02 UDP A 1 Q839 K842 L866 F868 V895 A896 K898 H901 H920 T921 T922 D925 Q509 K512 L536 F538 V565 A566 K568 H571 H590 T591 T592 D595 2.4.1.255 0006493,0016757 remove_due_to_license_issue IC50=1800nM O15294 23103942 1201 SCPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 4ay6 A 3.3 BS02 12V A 1 H498 P559 T560 G654 P656 Q839 K842 L866 A896 K898 H901 H920 T921 T922 D925 H187 P248 T249 G343 P345 Q509 K512 L536 A566 K568 H571 H590 T591 T592 D595 2.4.1.255 0006493,0016757 remove_due_to_license_issue O15294 23103942 1200 SCPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 4ayq A 1.1 BS01 MVL A 1 D249 L310 R363 P364 E365 Y423 E427 T451 E452 D221 L282 R335 P336 E337 Y395 E399 T423 E424 E121 R125 D249 E365 E93 R97 D221 E337 3.2.1.113 0004559,0004571,0005509,0005975,0016020,0016798,0046872 Kd=47nM remove_due_to_license_issue B0SWV2 23012075 503 TPEDWKALAADVRSEFQWAWQGYVAKAWGKDEINPVSGTSRSFFIEGHDLGLSLVEALDTLWIMGLDAEFQAGVDWVKANLSFDVDGNAQVFETNIRLVGGLLSAHLASGDPVLLAKARDLADRLAKAFEASPHGLPWRYVNLRTGAVSDPETNLAEIGTYLSEFGVLSQLTGERKYFDMAKRAMRHTLDRRSKIGLMAANIHAMTGAFTSRNASIDVYADSFYEYLWDAWALFGDEDCKRWAVECVDAQLAHQAKRYDGRLWFPMVDFETGAVTGTAQSELAAYYAGLLGQVGRKAQGDDYLASFTYLQATFGVIPESIDVTTGQPRRKHTGLRPEYPDACLNLWLIDRDPRYRRLAAIHYREMKATSRAAFGYTALKDITTRPMTQDDNCPGYWWSEQMKYYYLLFSDTPRIDYGQLQLSTEANVLRGFRKV 4ayr A 1.1 BS01 IFL A 1 R363 P364 E365 Y423 E427 T451 E452 R333 P334 E335 Y393 E397 T421 E422 E121 R125 D249 E365 E91 R95 D219 E335 3.2.1.113 0004559,0004571,0005509,0005975,0016020,0016798,0046872 Kd=99nM remove_due_to_license_issue B0SWV2 23012075 503 EDWKALAADVRSEFQWAWQGYVAKAWGKDEINPVSGTSRSFFIEGHDLGLSLVEALDTLWIMGLDAEFQAGVDWVKANLSFDVDGNAQVFETNIRLVGGLLSAHLASGDPVLLAKARDLADRLAKAFEASPHGLPWRYVNLRTGAVSDPETNLAEIGTYLSEFGVLSQLTGERKYFDMAKRAMRHTLDRRSKIGLMAANIHAMTGAFTSRNASIDVYADSFYEYLWDAWALFGDEDCKRWAVECVDAQLAHQAKRYDGRLWFPMVDFETGAVTGTAQSELAAYYAGLLGQVGRKAQGDDYLASFTYLQATFGVIPESIDVTTGQPRRKHTGLRPEYPDACLNLWLIDRDPRYRRLAAIHYREMKATSRAAFGYTALKDITTRPMTQDDNCPGYWWSEQMKYYYLLFSDTPRIDYGQLQLSTEANVLRGFRKV 4ayr A 1.1 BS02 IFL A 2 F120 E185 Y247 D249 F90 E155 Y217 D219 E121 R125 D249 E365 E91 R95 D219 E335 3.2.1.113 0004559,0004571,0005509,0005975,0016020,0016798,0046872 Kd=99nM remove_due_to_license_issue B0SWV2 23012075 504 EDWKALAADVRSEFQWAWQGYVAKAWGKDEINPVSGTSRSFFIEGHDLGLSLVEALDTLWIMGLDAEFQAGVDWVKANLSFDVDGNAQVFETNIRLVGGLLSAHLASGDPVLLAKARDLADRLAKAFEASPHGLPWRYVNLRTGAVSDPETNLAEIGTYLSEFGVLSQLTGERKYFDMAKRAMRHTLDRRSKIGLMAANIHAMTGAFTSRNASIDVYADSFYEYLWDAWALFGDEDCKRWAVECVDAQLAHQAKRYDGRLWFPMVDFETGAVTGTAQSELAAYYAGLLGQVGRKAQGDDYLASFTYLQATFGVIPESIDVTTGQPRRKHTGLRPEYPDACLNLWLIDRDPRYRRLAAIHYREMKATSRAAFGYTALKDITTRPMTQDDNCPGYWWSEQMKYYYLLFSDTPRIDYGQLQLSTEANVLRGFRKV 4ayt A 2.85 BS03 ACP A 1 Y501 A503 G530 G532 K533 S534 T535 Q575 Y348 A350 G377 G379 K380 S381 T382 Q422 ? 0005524,0016020,0016887,0055085,0140359 remove_due_to_license_issue Q9NRK6 23716676 900 LPEARKLLGLAYPERRRLAAAVGFLTMSSVISMSAPFFLGKIIDVIYTNPTVDYSDNLTRLCLGLSAVFLCGAAANAIRVYLMQTSGQRIVNRLRTSLFSSILRQEVAFFDKTRTGELINRLSSDTALLGRSVTENLSDGLRAGAQASVGISMMFFVSPNLATFVLSVVPPVSIIAVIYGRYLRKLTKVTQDSLAQATQLAEERIGNVRTVRAFGKEMTEIEKYASKVDHVMQLARKEAFARAGFFGATGLSGNLIVLSVLYKGGLLMGSAHMTVGELSSFLMYAFWVGISIGGLSSFYSELMKGLGAGGRLWELLEREPKLPFNEGVILNEKSFQGALEFKNVHFAYPARPEVPIFQDFSLSIPSGSVTALVGPSGSGKSTVLSLLLRLYDPASGTISLDGHDIRQLNPVWLRSKIGTVSQEPILFSCSIAENIAYGADDPSSVTAEEIQRVAEVANAVAFIRNFPQGFNTVVGEKGVLLSGGQKQRIAIARALLKNPKILLLDEATSALDAENEYLVQEALDRLMDGRTVLVIAHRLSTIKNANMVAVLDQGKITEYGKHEE 4ayu A 1.5 BS03 N8P A 1 N59 L62 Y64 Y74 E136 Q148 N59 L62 Y64 Y74 E136 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=18.6uM remove_due_to_license_issue P02743 25084341 499 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 4ayv B 2.8 BS02 9MQ B 1 H43 Y47 I179 D199 S205 V225 W227 G228 E229 G230 H43 Y47 I179 D199 S205 V225 W227 G228 E229 G230 H43 D99 E202 G203 D204 S205 G206 H43 D99 E202 G203 D204 S205 G206 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=0.68nM P00734 7966150 1258 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4ayw A 3.3 BS01 ANP A 1 Y501 S529 G530 G532 K533 S534 T535 Y348 S376 G377 G379 K380 S381 T382 ? 0005524,0016020,0016887,0055085,0140359 remove_due_to_license_issue Q9NRK6 23716676 1719 LPEARKLLGLAYPERRRLAAAVGFLTMSSVISMSAPFFLGKIIDVIYTNPTVDYSDNLTRLCLGLSAVFLCGAAANAIRVYLMQTSGQRIVNRLRTSLFSSILRQEVAFFDKTRTGELINRLSSDTALLGRSVTENLSDGLRAGAQASVGISMMFFVSPNLATFVLSVVPPVSIIAVIYGRYLRKLTKVTQDSLAQATQLAEERIGNVRTVRAFGKEMTEIEKYASKVDHVMQLARKEAFARAGFFGATGLSGNLIVLSVLYKGGLLMGSAHMTVGELSSFLMYAFWVGISIGGLSSFYSELMKGLGAGGRLWELLEREPKLPFNEGVILNEKSFQGALEFKNVHFAYPARPEVPIFQDFSLSIPSGSVTALVGPSGSGKSTVLSLLLRLYDPASGTISLDGHDIRQLNPVWLRSKIGTVSQEPILFSCSIAENIAYGADDPSSVTAEEIQRVAEVANAVAFIRNFPQGFNTVVGEKGVLLSGGQKQRIAIARALLKNPKILLLDELDAENEYLVQEALDRLMDGRTVLVIAHHLSTIKNANMVAVLDQGKITEYGKHEE 4ayx A 2.9 BS03 ACP A 1 Y501 S529 G530 G532 K533 S534 T535 Y348 S376 G377 G379 K380 S381 T382 ? 0005524,0016020,0016887,0055085,0140359 remove_due_to_license_issue Q9NRK6 23716676 900 LPEARKLLGLAYPERRRLAAAVGFLTMSSVISMSAPFFLGKIIDVIYTNPTVDYSDNLTRLCLGLSAVFLCGAAANAIRVYLMQTSGQRIVNRLRTSLFSSILRQEVAFFDKTRTGELINRLSSDTALLGRSVTENLSDGLRAGAQASVGISMMFFVSPNLATFVLSVVPPVSIIAVIYGRYLRKLTKVTQDSLAQATQLAEERIGNVRTVRAFGKEMTEIEKYASKVDHVMQLARKEAFARAGFFGATGLSGNLIVLSVLYKGGLLMGSAHMTVGELSSFLMYAFWVGISIGGLSSFYSELMKGLGAGGRLWELLEREPKLPFNEGVILNEKSFQGALEFKNVHFAYPARPEVPIFQDFSLSIPSGSVTALVGPSGSGKSTVLSLLLRLYDPASGTISLDGHDIRQLNPVWLRSKIGTVSQEPILFSCSIAENIAYGADDPSSVTAEEIQRVAEVANAVAFIRNFPQGFNTVVGEKGVLLSGGQKQRIAIARALLKNPKILLLDEATSALDAENEYLVQEALDRLMDGRTVLVIAHRLSTIKNANMVAVLDQGKITEYGKHEELLSKPNG 4ayy B 2.6 BS02 9MX B 1 H43 Y47 W50 L96 D199 C201 W227 G228 G230 H43 Y47 W50 L96 D199 C201 W227 G228 G230 H43 D99 E202 G203 D204 S205 G206 H43 D99 E202 G203 D204 S205 G206 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=6.7nM P00734 7966150 1258 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4az0 A 2.17 BS01 S61 A 1 N55 G56 C60 D64 E149 S150 Y247 N56 G57 C61 D65 E150 S151 Y248 G57 S150 Y151 G58 S151 Y152 3.4.16.5 0004185,0006508 ic50=0.038uM remove_due_to_license_issue IC50=38nM P10619 22861813 1262 RAPDQDEIQRLPGLAKQPSFRQYSGYLKGSGSKHLHYWFVESQKDPENSPVVLWLNGGPGCSSLDGLLTEHGPFLVQPDGVTLEYNPYSWNLIANVLYLESPAGVGFSYSDDKFYATNDTEVAQSNFEALQDFFRLFPEYKNNKLFLTGESYAGIYIPTLAVLVMQDPSMNLQGLAVGNGLSSYEQNDNSLVYFAYYHGLLGNRLWSSLQTHCCSQNKCNFYDNKDLECVTNLQEVARIVGNSGLNIYNLYAPCAGGVPS 4az0 B 2.17 BS01 S61 A 1 P301 M333 C334 N339 H429 P1 M33 C34 N39 H129 D372 H429 D72 H129 3.4.16.5 0004185,0006508 remove_due_to_license_issue IC50=38nM P10619 22861813 1262 PPCTNTTAASTYLNNPYVRKALNIPEQLPQWDMCNFLVNLQYRRLYRSMNSQYLKLLSSQKYQILLYNGDVDMACNFMGDEWFVDSLNQKMEVQRRPWLVKYGDSGEQIAGFVKEFSHIAFLTIKGAGHMVPTDKPLAAFTMFSRFLNKQPYE 4az2 B 2.6 BS02 9MU B 1 L96 D199 S205 W227 G228 G230 L96 D199 S205 W227 G228 G230 H43 D99 E202 G203 D204 S205 G206 H43 D99 E202 G203 D204 S205 G206 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue Ki=32nM P00734 7966150 1258 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4az3 A 2.04 BS01 S35 A 1 N55 G56 G57 C60 D64 E149 S150 Y247 N56 G57 G58 C61 D65 E150 S151 Y248 G57 S150 Y151 G58 S151 Y152 3.4.16.5 0004185,0006508 ic50=0.005uM remove_due_to_license_issue IC50=5nM P10619 22861813 1259 RAPDQDEIQRLPGLAKQPSFRQYSGYLKGSGSKHLHYWFVESQKDPENSPVVLWLNGGPGCSSLDGLLTEHGPFLVQPDGVTLEYNPYSWNLIANVLYLESPAGVGFSYSDDKFYATNDTEVAQSNFEALQDFFRLFPEYKNNKLFLTGESYAGIYIPTLAVLVMQDPSMNLQGLAVGNGLSSYEQNDNSLVYFAYYHGLLGNRLWSSLQTHCCSQNKCNFYDNKDLECVTNLQEVARIVGNSGLNIYNLYAPCAGGVP 4az3 B 2.04 BS01 S35 A 1 P301 C334 N335 N339 R344 H429 P3 C36 N37 N41 R46 H131 D372 H429 D74 H131 3.4.16.5 0004185,0006508 remove_due_to_license_issue IC50=5nM P10619 22861813 1259 MDPPCTNTTAASTYLNNPYVRKALNIPEQLPQWDMCNFLVNLQYRRLYRSMNSQYLKLLSSQKYQILLYNGDVDMACNFMGDEWFVDSLNQKMEVQRRPWLVKYGDSGEQIAGFVKEFSHIAFLTIKGAGHMVPTDKPLAAFTMFSRFLNKQPYE 4az5 A 1.73 BS01 NGW A 1 R196 H297 D360 E361 F415 W439 Y469 Y482 W517 D519 R16 H117 D180 E181 F235 W259 Y289 Y302 W337 D339 3.2.1.52 0004553,0005975 Kd=1.02uM remove_due_to_license_issue P49610 24132305 1615 NEKLAKKKIVSIDAGRKYFSPEQLKEIIDKAKHYGYTDLHLLVGNDGLRFMLDDMSITANGKTYASDDVKRAIEKGTNDYYNDPNGNHLTESQMTDLINYAKDKGIGLIPTVNSPGHMDAILNAMKELGIQNPNFSYFGKKSARTVDLDNEQAVAFTKALIDKYAAYFAKKTEIFNIGLDEYANDATDAKGWSVLQADKYYPNEGYPVKGYEKFIAYANDLARIVKSHGLKPMAFNDGIYYNSDTSFGSFDKDIIVSMWTGGWGGYDVASSKLLAEKGHQILNTNDAWYYVLGRNADGQGWYNLDQGLNGIKNTPITSVPKTEGADIPIIGGMVAAWADTPSARYSPSRLFKLMRHFANANAEYFAADYESAEQALNEVPKDLNRYTAESVTAVKEAEKAIRSLDSNLSRAQQDTIDQAIAKLQETVNNLTLTP 4az6 A 1.36 BS01 OAN A 1 R196 D360 E361 F415 W439 W443 Y469 W481 Y482 W517 D519 R18 D182 E183 F237 W261 W265 Y291 W303 Y304 W339 D341 3.2.1.52 0004553,0005975 Ki=0.8nM remove_due_to_license_issue P49610 24132305 1614 SHNEKLAKKKIVSIDAGRKYFSPEQLKEIIDKAKHYGYTDLHLLVGNDGLRFMLDDMSITANGKTYASDDVKRAIEKGTNDYYNDPNGNHLTESQMTDLINYAKDKGIGLIPTVNSPGHMDAILNAMKELGIQNPNFSYFGKKSARTVDLDNEQAVAFTKALIDKYAAYFAKKTEIFNIGLDEYANDATDAKGWSVLQADKYYPNEGYPVKGYEKFIAYANDLARIVKSHGLKPMAFNDGIYYNSDTSFGSFDKDIIVSMWTGGWGGYDVASSKLLAEKGHQILNTNDAWYYVLGRNADGQGWYNLDQGLNGIKNTPITSVPKTEGADIPIIGGMVAAWADTPSARYSPSRLFKLMRHFANANAEYFAADYESAEQALNEVPKDLNRYTAESVTAVKEAEKAIRSLDSNLSRAQQDTIDQAIAKLQETVNNLTLT 4azb A 2.1 BS01 OAN A 1 R196 D360 E361 F415 W439 D466 Y469 W517 D519 R16 D180 E181 F235 W259 D286 Y289 W337 D339 3.2.1.52 0004553,0005975 Kd=57.69nM remove_due_to_license_issue P49610 24132305 1606 NEKLAKKKIVSIDAGRKYFSPEQLKEIIDKAKHYGYTDLHLLVGNDGLRFMLDDMSITANGKTYASDDVKRAIEKGTNDYYNDPNGNHLTESQMTDLINYAKDKGIGLIPTVNSPGHMDAILNAMKELGIQNPNFSYFGKKSARTVDLDNEQAVAFTKALIDKYAAYFAKKTEIFNIGLDEYANDATDAKGWSVLQADKYYPNEGYPVKGYEKFIAYANDLARIVKSHGLKPMAFNDGIYYNSDTSFGSFDKDIIVSMWTGGWGGYDVASSKLLAEKGHQILNTNDAWYYVLGRNADGQGGGNLDQGLNGIKNTPITSVPKTEGADIPIIGGMVAAWADTPSARYSPSRLFKLMRHFANANAEYFAADYESAEQALNEVPKDAIRSLDSNLSRAQQDTIDQAIAKLQE 4azc A 2.09 BS01 NGW A 1 R641 D804 E805 F849 W872 Y902 I904 W951 D953 R19 D182 E183 F227 W250 Y280 I282 W329 D331 3.2.1.52 0004553,0005975 Kd=1.38uM remove_due_to_license_issue P49610 24132305 2042 GSHMEKLAKNKVISIDAGRKYFTLNQLKRIVDKASELGYSDVHLLLGNDGLRFLLDDMTITANGKTYASDDVKKAIIEGTKAYYDDPNGTALTQAEVTELIEYAKSKDIGLIPAINSPGHMDAMLVAMEKLGIKNPQAHFDKVSKTTMDLKNEEAMNFVKALIGKYMDFFAGKTKIFNFGTDEYANDATSAQGWYYLKWYQLYGKFAEYANTLAAMAKERGLQPMAFNDGFYYEDKDDVQFDKDVLISYWSKGWWGYNLASPQYLASKGYKFLNTNGDWYYILGQKPEDGGGFLKKAIENTGKTPFNQLASTKYPEVDLPTVGSMLSIWADRPSAEYKEEEIFELMTAFADHNKDYFRANYNALREELAKIPTGYSKESLEALDAAKTALNYNLNRNKQAELDTLVANLKAALQGK 4aze A 3.15 BS01 3RA A 1 I165 F170 A186 K188 L241 L294 D307 I34 F39 A55 K57 L110 L163 D176 D287 K289 N292 D307 S324 D156 K158 N161 D176 S193 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=7.6nM Q13627 22998443 700 ERKVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDGKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 4azf A 2.55 BS01 3RA A 1 G156 F160 V163 A176 K178 L230 L231 L282 I294 G102 F106 V109 A122 K124 L176 L177 L228 I240 D275 K277 N280 D295 S312 D221 K223 N226 D241 S258 2.7.12.1 0004672,0004712,0005524,0006468 remove_due_to_license_issue Q92630 22998443 600 HHHSSGVDLGTENLYFQSMGKVKATPMTPEQAMKQYMQKLTAFEHHEIFSYPEIYFLGLNAKKRQGMTGGPNNGGYDDDQGSYVQVPHDHVAYRYEVLKVIGKGSFGQVVKAYDHKVHQHVALKMVRNEKRFHRQAAEEIRILEHLRKQDKDNTMNVIHMLENFTFRNHICMTFELLSMNLYELIKKNKFQGFSLPLVRKFAHSILQCLDALHKNRIIHCDLKPENILLKQQGRSGIKVIDFGSSCYEHQRVYTYIQSRFYRAPEVILGARYGMPIDMWSLGCILAELLTGYPLLPGEDEGDQLACMIELLGMPSQKLLDASKRAKNFVSSKGYPRYCTVTTLSDVVLNGGRSRRGKLRGPPESREWGNALKGCDDPLFLDFLKQCLEWDPAVRMTPGQALRHPWLR 4azg A 2.4 BS01 OAN A 1 R641 D804 E805 W872 W876 Y879 Y902 I904 W951 D953 R20 D183 E184 W251 W255 Y258 Y281 I283 W330 D332 3.2.1.52 0004553,0005975 Kd=79.05nM remove_due_to_license_issue P49610 24132305 2040 RGSHMEKLAKNKVISIDAGRKYFTLNQLKRIVDKASELGYSDVHLLLGNDGLRFLLDDMTITANGKTYASDDVKKAIIEGTKAYYDDPNGTALTQAEVTELIEYAKSKDIGLIPAINSPGHMDAMLVAMEKLGIKNPQAHFDKVSKTTMDLKNEEAMNFVKALIGKYMDFFAGKTKIFNFGTDEYANDATSAQGWYYLKWYQLYGKFAEYANTLAAMAKERGLQPMAFNDGFYYEDKDDVQFDKDVLISYWSKGWWGYNLASPQYLASKGYKFLNTNGDWYYILGQKPEDGGGFLKKAIENTGKTPFNQLASTKYPEVDLPTVGSMLSIWADRPSAEYKEEEIFELMTAFADHNKDYFRANYNALREELAKISKESLEALDAAKTALNYNLNRNKQAELDTLVANLKAALQ 4azi A 1.98 BS01 OAN A 1 R641 D804 E805 F849 W872 Y902 I904 Y914 W951 D953 R19 D182 E183 F227 W250 Y280 I282 Y292 W329 D331 3.2.1.52 0004553,0005975 Kd=35.56nM remove_due_to_license_issue P49610 24132305 2038 GSHMEKLAKNKVISIDAGRKYFTLNQLKRIVDKASELGYSDVHLLLGNDGLRFLLDDMTITANGKTYASDDVKKAIIEGTKAYYDDPNGTALTQAEVTELIEYAKSKDIGLIPAINSPGHMDAMLVAMEKLGIKNPQAHFDKVSKTTMDLKNEEAMNFVKALIGKYMDFFAGKTKIFNFGTDEYANDATSAQGWYYLKWYQLYGKFAEYANTLAAMAKERGLQPMAFNDGFYYEDKDDVQFDKDVLISYWSKGWWGYNLASPQYLASKGYKFLNTNGDWYYILGQKPEDGWYFLKKAIENTGKTPFNQLASTKYPEVDLPTVGSMLSIWADRPSAEYKEEEIFELMTAFADHNKDYFRANYNALREELAKIPYSKESLEALDAAKTALNYNLNRNKQAELDTLVANLKAA 4azp A 2.1 BS01 A9M A 1 M23 T56 V60 K61 A78 D79 R129 Y131 M22 T55 V59 K60 A77 D78 R128 Y130 ? 0001972,0005324,0005504,0005576,0005615,0005634,0005737,0006006,0006629,0006656,0006869,0008289,0010829,0014069,0015909,0031392,0035360,0042593,0042802,0045202,0051930,0098921,0098978,0099092,0099178,0099524,0120162,1990379 Ki=1.26uM remove_due_to_license_issue Q05816 24531463 1136 ASLKDLEGKWRLMESHGFEEYMKELGVGLALRKMAAMAKPDCIITCDGNNITVKTESTVKTTVFSCNLGEKFDETTADGRKTETVCTFQDGALVQHQQWDGKESTITRKLKDGKMIVECVMNNATCTRVYEKVQ 4azt A 2.34 BS02 LY2 A 1 Y243 F245 V250 L311 M358 Y229 F231 V236 L297 M344 2.1.1.294,2.7.1.181 0004672,0005524,0006468 ic50=68uM remove_due_to_license_issue Q47592 22970759 1483 DLNTLVSELPEIYQTIFGHPEWDGDAARDCNQRLDLITEQYDNLSRALGRPLNVLDLGCAQGFFSLSLASKGATIVGIDFQQENINVCRALAEENPDFAAEFRVGRIEEVIAALEEGEFDLAIGLSVFHHIVHLHGIDEVKRLLSRLADVTQAVILELAVKEEPFYWGVSQPDDPRELIEQCAFYRLIGEFDTHLSPVPRPMYLVSNHRVLINDFNQPFQHWQNRSRRYFFGEDYVCKFFYYDMPHGILTAEESQRNKYELHNEIKFLTQPPAGFDAPAVLAHGENAQSGWLVMEKLPGRLLSDMLAAGEEIDREKILGSLLRSLAALEKQGFWHDDVRPWNVMVDARQHARLIDFGSIVTTSWPTNLVQSFFVFVNELFNLPQPWSNWLYAVWQEPVERWNFVLLLALFEKKAKLPSAEQQRGATEQWIIAQET 4azy A 1.79 BS01 7F3 A 1 G11 Q12 D32 S35 Y71 Q73 W76 F108 I110 W115 I118 D228 G230 G15 Q16 D36 S39 Y75 Q77 W80 F112 I114 W119 I122 D219 G221 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=125nM remove_due_to_license_issue P56817 22924815 1507 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b00 A 1.83 BS01 I6X A 1 S10 Q12 G13 D32 S35 Y71 W76 F108 I110 I118 D228 S229 G230 T231 S14 Q16 G17 D36 S39 Y75 W80 F112 I114 I122 D219 S220 G221 T222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=2.44nM remove_due_to_license_issue P56817 22924815 1507 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b05 A 1.8 BS01 32D A 1 G13 L30 D32 S35 N37 Y71 W76 F108 I110 I118 D228 G230 G18 L35 D37 S40 N42 Y76 W80 F112 I114 I122 D218 G220 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D218 T221 3.4.23.46 0004190,0006508,0016020 Ki=26.1nM remove_due_to_license_issue IC50=0.600000nM, Ki=26nM P56817 23048024 1391 KGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHDEFRTAAVEGPFVTLMEDCGY 4b0b A 1.9 BS01 54F A 1 W87 Q88 G103 R104 A105 W86 Q87 G102 R103 A104 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 1172 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4b0b A 1.9 BS02 54F B 1 V76 M77 V75 M76 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 1172 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4b0b B 1.9 BS01 54F A 1 F71 V76 M77 F69 V74 M75 H70 V76 G79 C80 D84 H68 V74 G77 C78 D82 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 1172 KQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4b0b B 1.9 BS02 54F B 1 W87 Q88 G103 R104 A105 W85 Q86 G101 R102 A103 H70 V76 G79 C80 D84 H68 V74 G77 C78 D82 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 1172 KQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4b0c A 2.7 BS01 C9H A 1 H70 P78 G79 H69 P77 G78 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTF 4b0c A 2.7 BS02 C9H B 1 G103 R104 A105 G102 R103 A104 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTF 4b0c B 2.7 BS01 C9H A 1 W87 A105 F171 W86 A104 F170 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 remove_due_to_license_issue O33877 23174186 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4b0g A 2.5 BS01 VEK A 1 L139 G140 K141 G142 K143 G145 N146 V147 K162 Y212 A213 G216 L263 L14 G15 K16 G17 K18 G20 N21 V22 K37 Y83 A84 G87 L134 D256 K258 E260 N261 D274 T292 D127 K129 E131 N132 D145 T151 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=0.015uM remove_due_to_license_issue IC50=15nM O14965 23043539 1392 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVTLDYLPPEMIEHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 4b11 A 1.59 BS01 7I1 A 1 V96 E97 D98 F103 F105 Y107 Y211 Y334 L367 L388 L410 V71 E72 D73 F78 F80 Y82 Y186 Y309 L342 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 ic50=2.3uM remove_due_to_license_issue A5K1A2 23035716 999 MDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4b12 A 1.79 BS01 C23 A 1 E97 D98 F103 F105 Y211 Y315 S319 Y334 L367 L388 L410 E72 D73 F78 F80 Y186 Y290 S294 Y309 L342 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 ic50=10.2uM remove_due_to_license_issue A5K1A2 23035716 1411 MDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4b13 A 1.58 BS01 X25 A 1 V96 E97 D98 F103 F105 Y211 Y315 S319 Y334 L367 L388 L410 V71 E72 D73 F78 F80 Y186 Y290 S294 Y309 L342 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 ic50=2uM remove_due_to_license_issue A5K1A2 23035716 1411 MDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4b14 A 1.5 BS01 4XB A 1 E97 D98 F103 F105 Y107 Y211 S319 Y334 L367 L388 L410 E72 D73 F78 F80 Y82 Y186 S294 Y309 L342 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 ic50=0.6uM remove_due_to_license_issue A5K1A2 23035716 1001 MDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4b1c A 1.95 BS01 1B1 A 1 S10 Q12 G13 D32 Y71 F108 I118 D228 S229 G230 S16 Q18 G19 D38 Y77 F114 I124 D220 S221 G222 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.079uM remove_due_to_license_issue P56817 23017051 1504 KKGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLEDCGYN 4b1d A 1.95 BS01 6TG A 1 Q12 D32 W76 F108 I110 I118 D228 G230 Q16 D36 W80 F112 I114 I122 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.012uM remove_due_to_license_issue P56817 23017051 1505 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b1j A 2.08 BS01 A1R A 1 I726 E727 F738 N740 V753 Q754 E755 E756 Y795 N869 G871 G873 A874 F875 F902 I271 E272 F283 N285 V298 Q299 E300 E301 Y340 N414 G416 G418 A419 F420 F447 3.2.1.143 0004649,0005975,0006282 remove_due_to_license_issue IC50=120nM Q86W56 23251397 1966 KKWLGTPIEEMRRMPRCGIRLPLLRPSANHTVTIRVDLLRAGEVPKPFPTHYKDLWDNKHVKMPCSEQNLYPVERTAGSRWELIQTALLNKFTRPQNLKDAILKYNVAYSKKWDFTALIDFWDKVLEEAEAQHLYQSILPDMVKIALCLPNICTQPIPLLAAAMNHSITMSQEQIASLLANAFFCTFPRRNAKMKSEYSSYPDINFNRLFEGRSSRKPEKLKTLFCYFRRVTAAAPTGLVTFTRQSLEDFPEWERCEKPLTRLHVTYEGTIEENGQGMLQVDFANRFVGGGVTSAGLVQEEIRFLINPELIISRLFTEVLDHNECLIITGTEQYSEYTGYAETYRWSRSHEDGSERDDWQRRCTEIVAIDALHFRRYLDQFVPEKMRRELNKAYCGFLRPGVSSENLSAVATGNWGCGAFGGDARLKALIQILAAAAAERDVVYFTFGDSELMRDIYSMHIFLTERKLTVGDVYKLLLRYYNEECRNCSTPGPDIKLYPFIYHAVESC 4b20 A 2.75 BS01 dna C 0 Y80 G83 L85 D110 Q112 I122 A138 K139 S140 R141 L142 Y80 G83 L85 D110 Q112 I122 A138 K139 S140 R141 L142 3.1.21.7 0000287,0003727,0004519,0005737,0006281,0016891,0043737,0046872 remove_due_to_license_issue Q9X2H9 23313664 2 ~ 7 MDYRQLHRWDLPPEEAIKVQNELRKKIKLTPYEGEPEYVAGVDLSFPGKEEGLAVIVVLEYPSFKILEVVSERGEITFPYIPGLLAFREGPLFLKAWEKLRTKPDVVVFDGQGLAHPRKLGIASHMGLFIEIPTIGVAKSRLYGTFKMPEDKRCSWSYLYDGEEIIGCVIRTKEGSAPIFVSPGHLMDVESSKRLIKAFTLPGRRIPEPTRLAHIYTQRLKKG 4b20 A 2.75 BS02 dna D 0 Q218 K221 Q218 K221 3.1.21.7 0000287,0003727,0004519,0005737,0006281,0016891,0043737,0046872 remove_due_to_license_issue Q9X2H9 23313664 8 ~ 16 MDYRQLHRWDLPPEEAIKVQNELRKKIKLTPYEGEPEYVAGVDLSFPGKEEGLAVIVVLEYPSFKILEVVSERGEITFPYIPGLLAFREGPLFLKAWEKLRTKPDVVVFDGQGLAHPRKLGIASHMGLFIEIPTIGVAKSRLYGTFKMPEDKRCSWSYLYDGEEIIGCVIRTKEGSAPIFVSPGHLMDVESSKRLIKAFTLPGRRIPEPTRLAHIYTQRLKKG 4b20 B 2.75 BS01 dna C 0 L220 K222 G223 L220 K222 G223 3.1.21.7 0000287,0003727,0004519,0005737,0006281,0016891,0043737,0046872 remove_due_to_license_issue Q9X2H9 23313664 2 ~ 7 MDYRQLHRWDLPPEEAIKVQNELRKKIKLTPYEGEPEYVAGVDLSFPGKEEGLAVIVVLEYPSFKILEVVSERGEITFPYIPGLLAFREGPLFLKAWEKLRTKPDVVVFDGQGLAHPRKLGIASHMGLFIEIPTIGVAKSRLYGTFKMPEDKRCSWSYLYDGEEIIGCVIRTKEGSAPIFVSPGHLMDVESSKRLIKAFTLPGRRIPEPTRLAHIYTQRLKKG 4b20 B 2.75 BS02 dna F 0 Y80 G83 L85 D110 Q112 H116 G121 I122 A138 K139 S140 R141 L142 Y80 G83 L85 D110 Q112 H116 G121 I122 A138 K139 S140 R141 L142 3.1.21.7 0000287,0003727,0004519,0005737,0006281,0016891,0043737,0046872 remove_due_to_license_issue Q9X2H9 23313664 2 ~ 7 MDYRQLHRWDLPPEEAIKVQNELRKKIKLTPYEGEPEYVAGVDLSFPGKEEGLAVIVVLEYPSFKILEVVSERGEITFPYIPGLLAFREGPLFLKAWEKLRTKPDVVVFDGQGLAHPRKLGIASHMGLFIEIPTIGVAKSRLYGTFKMPEDKRCSWSYLYDGEEIIGCVIRTKEGSAPIFVSPGHLMDVESSKRLIKAFTLPGRRIPEPTRLAHIYTQRLKKG 4b20 B 2.75 BS03 dna G 0 F46 K221 F46 K221 3.1.21.7 0000287,0003727,0004519,0005737,0006281,0016891,0043737,0046872 remove_due_to_license_issue Q9X2H9 23313664 8 ~ 17 MDYRQLHRWDLPPEEAIKVQNELRKKIKLTPYEGEPEYVAGVDLSFPGKEEGLAVIVVLEYPSFKILEVVSERGEITFPYIPGLLAFREGPLFLKAWEKLRTKPDVVVFDGQGLAHPRKLGIASHMGLFIEIPTIGVAKSRLYGTFKMPEDKRCSWSYLYDGEEIIGCVIRTKEGSAPIFVSPGHLMDVESSKRLIKAFTLPGRRIPEPTRLAHIYTQRLKKG 4b2d A 2.3 BS01 SER A 1 R43 N70 H464 I469 F470 R30 N57 H451 I456 F457 R73 R120 K270 T328 R60 R107 K257 T315 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 Kd=200uM remove_due_to_license_issue P14618 23064226 1532 QTQQLHAAMADTFLEHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 4b2i A 1.3 BS01 LZ1 A 1 M169 I171 A201 A203 Q217 A218 M62 I64 A94 A96 Q110 A111 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=1mM remove_due_to_license_issue Kd=1000000nM O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVSATLRVYLRKGKGGKRIARLIDAPHLPEGEAVFSITEKGIED 4b2l A 1.5 BS01 TR7 A 1 M169 I171 A201 A203 L214 Q217 A218 M221 M62 I64 A94 A96 L107 Q110 A111 M114 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=0.57mM remove_due_to_license_issue Kd=570000nM O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVSATLRVYLRKGKGGKRIARLIDAPHLPEGEAVFSITEKGIED 4b32 A 1.5 BS01 03V A 1 M169 I171 A201 A203 Q217 M62 I64 A94 A96 Q110 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=0.46mM remove_due_to_license_issue Kd=460000nM O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVSATLRVYLRKGKGGKRIARLIDAPHLPEGEAVFSITEKGIED 4b33 A 1.499 BS01 1NP A 1 M169 I171 A201 A203 L214 Q217 A218 M62 I64 A94 A96 L107 Q110 A111 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=0.43mM remove_due_to_license_issue Kd=430000nM O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVSATLRVYLRKGKGGKRIARLIDAPHLPEGEAVFSITEKGIED 4b34 A 1.55 BS01 ABV A 1 M169 A201 Y202 A203 L214 Q217 A218 M62 A94 Y95 A96 L107 Q110 A111 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=0.73mM remove_due_to_license_issue Kd=730000nM O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVSATLRVYLRKGKGGKRIARLIDAPHLPEGEAVFSITEKGIED 4b35 A 1.4 BS01 4ME A 1 M169 A201 Y202 A203 L214 M62 A94 Y95 A96 L107 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=1.3mM remove_due_to_license_issue O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVSATLRVYLRKGKGGKRIARLIDAPHLPEGEAVFSITEKGIED 4b3d A 1.589 BS01 5MI A 1 M169 I171 A203 M62 I64 A96 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=2.1mM remove_due_to_license_issue Kd=2100000nM O74036 23344974 1351 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVATLRVYLRKGKGGKRIARLIDGEAVFSITEKGIED 4b3d A 1.589 BS02 5MI A 2 R204 F206 R97 F99 ? 0003677,0003684,0005524,0006259,0006281,0006310,0008094,0016887,0140664 Kd=2.1mM remove_due_to_license_issue Kd=2100000nM O74036 23344974 1352 ATIGRISTGSKSLDKLLGGGIETQAITEVFGEFGSGKTQLAHTLAVMVQLPPEEGGLNGSVMWIDTENTFRPERIREIAQNRGLDPDEVLKHIAYARAFNSNHQMLLVQQAEDMIKELLNTDRPVKLLIVDSLTSHFRSEYIGRGALAERQQKLAKHLADLHRLANLYDIAVFVTNQVATLRVYLRKGKGGKRIARLIDGEAVFSITEKGIED 4b3u A 1.8 BS01 NWL A 1 L45 E255 I256 R259 Q260 L51 E261 I262 R265 Q266 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=4.7uM remove_due_to_license_issue IC50=4.7e+3nM Q9HU22 23138692 400 HHHHHHMKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b3u C 1.8 BS01 NWL C 1 L45 E255 I256 R259 L50 E260 I261 R264 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=4.7uM remove_due_to_license_issue IC50=4.7e+3nM Q9HU22 23138692 400 HHHHHMKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b4g A 2.5 BS01 KKT A 1 L45 Y113 G115 F118 V250 A251 E255 I256 R259 L45 Y113 G115 F118 V250 A251 E255 I256 R259 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=0.175uM remove_due_to_license_issue IC50=175nM Q9HU22 23138692 400 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b4g B 2.5 BS01 KKT B 1 S41 T42 Y113 G115 F118 V250 E255 S41 T42 Y113 G115 F118 V247 E252 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=0.175uM remove_due_to_license_issue IC50=175nM Q9HU22 23138692 400 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPLEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b4m A 2.35 BS01 JWT A 1 S41 T42 L45 Y113 G115 V250 A251 E255 I256 R259 S44 T45 L48 Y116 G118 V253 A254 E258 I259 R262 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=0.205uM remove_due_to_license_issue IC50=205nM Q9HU22 23138692 400 HHHMKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b4m C 2.35 BS01 JWT C 1 S41 T42 L45 Y113 G115 V250 A251 E255 S41 T42 L45 Y113 G115 V250 A251 E255 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=0.205uM remove_due_to_license_issue IC50=205nM Q9HU22 23138692 400 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b4q A 2.0 BS01 GLC C 1 S90 K114 R117 S71 K95 R98 ? remove_due_to_license_issue Q47212 22812428 1 SAQVTGTLLGTGKTNTTQMPALYTWQHQIYNVNFIPSSSGTLTCQAGTILVWKNGRETQYALECRVSIHHSSGSINESQWGQQSQVGFGTACGNKKCRFTGFEISLRIPPNAQTYPLSSGDLKGSFSLTNKEVNWSASIYVP 4b4q A 2.0 BS02 GAL C 1 S90 R117 S71 R98 ? remove_due_to_license_issue Q47212 22812428 2 SAQVTGTLLGTGKTNTTQMPALYTWQHQIYNVNFIPSSSGTLTCQAGTILVWKNGRETQYALECRVSIHHSSGSINESQWGQQSQVGFGTACGNKKCRFTGFEISLRIPPNAQTYPLSSGDLKGSFSLTNKEVNWSASIYVP 4b4q A 2.0 BS03 FUC C 1 Y49 N50 H88 T119 G120 Y30 N31 H69 T100 G101 ? remove_due_to_license_issue Q47212 22812428 5 SAQVTGTLLGTGKTNTTQMPALYTWQHQIYNVNFIPSSSGTLTCQAGTILVWKNGRETQYALECRVSIHHSSGSINESQWGQQSQVGFGTACGNKKCRFTGFEISLRIPPNAQTYPLSSGDLKGSFSLTNKEVNWSASIYVP 4b5b A 2.055 BS01 BBE A 1 S41 L45 Y113 G115 V250 A251 E255 I256 S41 L45 Y113 G115 V250 A251 E255 I256 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=0.387uM remove_due_to_license_issue IC50=387nM Q9HU22 23138692 400 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b5b C 2.055 BS01 BBE C 1 S41 L45 Y113 G115 H119 V250 E255 R259 S41 L45 Y113 G115 H119 V248 E253 R257 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 ic50=0.387uM remove_due_to_license_issue IC50=387nM Q9HU22 23138692 400 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4b5d A 2.195 BS01 SW4 A 1 W153 V154 C197 E198 Y201 W152 V153 C196 E197 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=12.8nM remove_due_to_license_issue I6L8L2 22928944 1213 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRS 4b5d A 2.195 BS02 SW4 E 1 I118 F120 I117 F119 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=12.8nM remove_due_to_license_issue I6L8L2 22928944 1213 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRS 4b5d B 2.195 BS01 SW4 A 1 I118 I128 I117 I127 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=12.8nM remove_due_to_license_issue I6L8L2 22928944 1213 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRS 4b5d B 2.195 BS02 SW4 B 1 W153 Y194 C197 Y201 W152 Y193 C196 Y200 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802,0098794 Ki=12.8nM remove_due_to_license_issue I6L8L2 22928944 1213 NGLMAKRLRRELLNTYEQLGKSGLPFLDDIGKVDVKFGLSLQLLKSIEQRGMGFNSIGTFKAIVKLSWVDTILRWDPEPPFDFQKIEISPDEIWTPDIKLFNSVDLDMTLDRTTQAIVFSNGTVLWIPPAVLKVLCVSQDDVDSCHFQFGSWVYSVDEVDIHFMDDKAEVLLDFYQDSLEILENSAQRQEVVYPCCESAYVEMKYLLALRS 4b5s A 1.68 BS02 PYR A 1 E149 F170 G172 P173 A174 D175 E149 F170 G172 P173 A174 D175 H45 R70 D84 E149 D175 H45 R70 D84 E149 D175 4.1.2.52 0003824,0005737,0009056,0010124,0016829,0016832,0043863,0046872,0061677,1901023 remove_due_to_license_issue B1IS70 22908224 1256 MENSFKAALKAGRPQIGLWLGLSSSYSAELLAGAGFDWLLIDGEHAPNNVQTVLTQLQAIAPYPSQPVVRPSWNDPVQIKQLLDVGTQTLLVPMVQNADEAREAVRATRYPPAGIRGVGSALARASRWNRIPDYLQKANDQMCVLVQIETREAMKNLPQILDVEGVDGVFIGPADLSADMGYAGNPQHPEVQAAIEQAIVQIRESGKAPGILIANEQLAKRYLELGALFVAVGVDTTLLARAAEALAARFG 4b5t A 1.923 BS03 2KT A 1 W19 R70 F170 G172 P173 A174 D175 L212 W19 R70 F170 G172 P173 A174 D175 L212 H45 R70 D84 E149 D175 H45 R70 D84 E149 D175 4.1.2.52 0003824,0005737,0009056,0010124,0016829,0016832,0043863,0046872,0061677,1901023 remove_due_to_license_issue B1IS70 22908224 4000 MENSFKAALKAGRPQIGLWLGLSSSYSAELLAGAGFDWLLIDGEHAPNNVQTVLTQLQAIAPYPSQPVVRPSWNDPVQIKQLLDVGTQTLLVPMVQNADEAREAVRATRYPPAGIRGVGSALARASRWNRIPDYLQKANDQMCVLVQIETREAMKNLPQILDVEGVDGVFIGPADLSADMGYAGNPQHPEVQAAIEQAIVQIRESGKAPGILIANEQLAKRYLELGALFVAVGVDTTLLARAAEALAARFG 4b5w A 1.792 BS02 PYR A 1 Q147 E149 G172 P173 A174 D175 Q147 E149 G172 P173 A174 D175 H45 A70 D84 E149 D175 H45 A70 D84 E149 D175 4.1.2.52 0003824,0005737,0009056,0010124,0016829,0016832,0043863,0046872,0061677,1901023 Kd=26.9mM remove_due_to_license_issue B1IS70 22908224 1259 MENSFKAALKAGRPQIGLWLGLSSSYSAELLAGAGFDWLLIDGEHAPNNVQTVLTQLQAIAPYPSQPVVAPSWNDPVQIKQLLDVGTQTLLVPMVQNADEAREAVRATRYPPAGIRGVGSALARASRWNRIPDYLQKANDQMCVLVQIETREAMKNLPQILDVEGVDGVFIGPADLSADMGYAGNPQHPEVQAAIEQAIVQIRESGKAPGILIANEQLAKRYLELGALFVAVGVDTTLLARAAEALAARFGAQATA 4b5w B 1.792 BS02 PYR B 1 Q147 E149 F170 G172 P173 A174 D175 Q147 E149 F170 G172 P173 A174 D175 H45 A70 D84 E149 D175 H45 A70 D84 E149 D175 4.1.2.52 0003824,0005737,0009056,0010124,0016829,0016832,0043863,0046872,0061677,1901023 Kd=26.9mM remove_due_to_license_issue B1IS70 22908224 1255 MENSFKAALKAGRPQIGLWLGLSSSYSAELLAGAGFDWLLIDGEHAPNNVQTVLTQLQAIAPYPSQPVVAPSWNDPVQIKQLLDVGTQTLLVPMVQNADEAREAVRATRYPPAGIRGVGSALARASRWNRIPDYLQKANDQMCVLVQIETREAMKNLPQILDVEGVDGVFIGPADLSADMGYAGNPQHPEVQAAIEQAIVQIRESGKAPGILIANEQLAKRYLELGALFVAVGVDTTLLARAAEALAARFGAQ 4b6c A 2.2 BS01 B5U A 1 N52 E56 R82 G83 I84 P85 Q102 V123 S126 T169 N17 E21 R47 G48 I49 P50 Q60 V61 S64 T107 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.69uM remove_due_to_license_issue P0C559 23268609 1256 STGERGLHHLIWEVVDNAVDEAMAGFATRVDVKIHADGSVEVRDDGRGIPVPTIDVVMTQVGVSVVNALSTRLEATVLRDGYEWFQYYDRSVPGKLKQGGETKETGTTIRFWADPEIFETTDYNFETVARRLQEMAFLNKGLTIELTDERDGKHRVFHYPG 4b6e B 2.46 BS01 10L B 1 D81 V524 C525 Q526 D79 V522 C523 Q524 T10 C16 H57 D81 G137 S139 T8 C14 H55 D79 G135 S137 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0004386,0005524,0006508,0008236,0019087 remove_due_to_license_issue P26663 23023261 1722 ITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGIDPNIRTGVRTITTGAPVTYSTYGKFLADGGCSGGAYDIIICDECHSTDSTTILGIGTVLDQAETAGARLVVLATATPPGSVTVPHPNIEEVALSNTGEIPFYGKAIPIEAIRGGRHLIFCHSKKKCDELAAKLSGLGINAVAYYRGLDVSVIPTIGDVVVVATDALMTGYTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTVPQDAVSRSQRRGRTGRGRRGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETSVRLRAYLNTPGLPVCQDHLEFWESVFTGLTHIDAHFLSQTKQAGDNFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMACMSADLEVVTGSVVIVGRIILSS 4b6f A 2.89 BS01 20L A 1 D79 D81 R155 M485 V524 Q526 V630 D77 D79 R153 M483 V522 Q524 V628 T10 C16 H57 D81 G137 S139 T8 C14 H55 D79 G135 S137 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0004386,0005524,0006508,0008236,0019087 remove_due_to_license_issue P26663 23023261 1722 ITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGIDPNIRTGVRTITTGAPVTYSTYGKFLADGGCSGGAYDIIICDECHSTDSTTILGIGTVLDQAETAGARLVVLATATPPGSVTVPHPNIEEVALSNTGEIPFYGKAIPIEAIRGGRHLIFCHSKKKCDELAAKLSGLGINAVAYYRGLDVSVIPTIGDVVVVATDALMTGYTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTVPQDAVSRSQRRGRTGRGRRGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETSVRLRAYLNTPGLPVCQDHLEFWESVFTGLTHIDAHFLSQTKQAGDNFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMACMSADLEVVTGSVVIVGRIILSGSGS 4b6o A 2.0 BS01 3DQ A 1 N12 N75 G77 G78 H81 H101 I102 S103 R112 N11 N74 G76 G77 H80 H100 I101 S102 R111 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P10 N11 R18 Y23 N74 G77 E98 H100 R107 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=100nM remove_due_to_license_issue P9WPX7 23198883 1144 ELIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4b6p A 2.3 BS01 2HN A 1 N12 L16 R19 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N10 L14 R17 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=74nM remove_due_to_license_issue P9WPX7 23198883 1145 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEHV 4b6q A 1.54 BS01 BZ5 A 1 L13 R15 L16 N75 G77 G78 H81 H101 I102 S103 R112 L11 R13 L14 N66 G68 G69 H72 H92 I93 S94 R103 P11 N12 N75 G78 E99 H101 R108 P9 N10 N66 G69 E90 H92 R99 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=28nM remove_due_to_license_issue P9WPX7 23198883 1145 LIVNVINGPNLGRLGRGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEHV 4b6r A 2.0 BS01 3DQ A 1 Y22 N76 G78 A79 H82 H102 L103 T104 R113 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=1420nM remove_due_to_license_issue Q48255 23198883 1158 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKN 4b6r A 2.0 BS02 3DQ B 1 D89 L93 D89 L93 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=1420nM remove_due_to_license_issue Q48255 23198883 1158 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKN 4b6r C 2.0 BS01 3DQ A 1 D89 L93 D89 L93 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=1420nM remove_due_to_license_issue Q48255 23198883 1158 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKN 4b6r C 2.0 BS02 3DQ C 1 Y22 N76 G78 A79 H82 H102 L103 T104 R113 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=1420nM remove_due_to_license_issue Q48255 23198883 1158 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKN 4b6s A 1.9 BS01 2HN A 1 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=970nM remove_due_to_license_issue Q48255 23198883 200 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQKNN 4b6s C 1.9 BS01 2HN A 1 D89 L93 D89 L93 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=970nM remove_due_to_license_issue Q48255 23198883 200 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQ 4b6s C 1.9 BS02 2HN C 1 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 N10 L14 Y22 N76 G78 A79 H82 H102 L103 T104 R113 P9 N10 R17 Y22 N76 A79 E100 H102 R109 P9 N10 R17 Y22 N76 A79 E100 H102 R109 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0019631 Ki=970nM remove_due_to_license_issue Q48255 23198883 200 MKILVIQGPNLNMLGHRDPRLYGMVTLDQIHEIMQTFVKQGNLDVELEFFQTNFEGEIIDKIQESVGSDYEGIIINPGAFSHTSIAIADAIMLAGKPVIEVHLTNIQAREEFRKNSYTGAACGGVIMGFGPLGYNMALMAMVNILAEMKAFQEAQ 4b6u A -1.00 BS01 M7G A 1 S43 P45 C52 L97 W98 R152 S43 P45 C52 L97 W98 R152 ? 0003723,0003743,0006412,0006413,0006417 remove_due_to_license_issue Q9DBB5 23431134 208 MALPPAAAPPGANEPLDKALSALPPEPGGVPLHSPWTFWLDRSLPGATAAECASNLKKIYTVQTVQIFWSVYNNIPPVTSLPLRCSYHLMRGERRPLWEEESNAKGGVWKMKVPKDSTSTVWKELLLATIGEQFTDCAAADDEIIGVSVSVRDREDVVQVWNVNASLVGEATVLEKIHQLLPHIAFKAVFYKPHEEHHAFEGGRGKH 4b70 A 1.6 BS01 WM9 A 1 G11 Q12 G13 D32 Y71 F108 I110 I118 D228 G230 G12 Q13 G14 D33 Y72 F109 I111 I119 D216 G218 D32 S35 N37 A39 Y71 D228 T231 D33 S36 N38 A40 Y72 D216 T219 3.4.23.46 0004190,0006508,0016020 ic50=6.3uM remove_due_to_license_issue IC50=6300nM P56817 23126626 1503 VEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b71 A 2.5 BS01 DJL A 1 V78 D79 D81 R155 M485 F486 V524 C525 Q526 V92 D93 D95 R169 M499 F500 V538 C539 Q540 T10 C16 H57 D81 G137 S139 T24 C30 H71 D95 G151 S153 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0004386,0005524,0006508,0008236,0019087 remove_due_to_license_issue P26663 23023261 1721 GSVVIVGRIILSGSGSITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGIDPNIRTGVRTITTGAPVTYSTYGKFLADGGCSGGAYDIIICDECHSTDSTTILGIGTVLDQAETAGARLVVLATATPPGSVTVPHPNIEEVALSNTGEIPFYGKAIPIEAIRGGRHLIFCHSKKKCDELAAKLSGLGINAVAYYRGLDVSVIPTIGDVVVVATDALMTGYTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTVPQDAVSRSQRRGRTGRGRRGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETSVRLRAYLNTPGLPVCQDHLEFWESVFTGLTHIDAHFLSQTKQAGDNFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMACMSADLEVVT 4b72 A 1.6 BS01 2FB A 1 Q12 D32 S35 Y71 Q73 W76 F108 I110 I118 D228 G230 Q16 D36 S39 Y75 Q77 W80 F112 I114 I122 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.63uM remove_due_to_license_issue IC50=32nM P56817 23126626 1503 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b73 A 2.5 BS01 4VA A 1 V78 D79 D81 R155 M485 L517 V524 C525 Q526 V92 D93 D95 R169 M499 L531 V538 C539 Q540 T10 C16 H57 D81 G137 S139 T24 C30 H71 D95 G151 S153 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0004386,0005524,0006508,0008236,0019087 Kd=0.062uM remove_due_to_license_issue P26663 23023261 1721 GSVVIVGRIILSGSGSITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGIDPNIRTGVRTITTGAPVTYSTYGKFLADGGCSGGAYDIIICDECHSTDSTTILGIGTVLDQAETAGARLVVLATATPPGSVTVPHPNIEEVALSNTGEIPFYGKAIPIEAIRGGRHLIFCHSKKKCDELAAKLSGLGINAVAYYRGLDVSVIPTIGDVVVVATDALMTGYTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTVPQDAVSRSQRRGRTGRGRRGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETSVRLRAYLNTPGLPVCQDHLEFWESVFTGLTHIDAHFLSQTKQAGDNFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMACMSADLEVVT 4b74 A 2.18 BS01 1LH A 1 V78 D79 D81 R155 M485 F486 Y516 L517 T519 L522 P523 V524 C525 Q526 V92 D93 D95 R169 M499 F500 Y530 L531 T533 L536 P537 V538 C539 Q540 T10 C16 H57 D81 G137 S139 T24 C30 H71 D95 G151 S153 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0004386,0005524,0006508,0008236,0019087 Kd=0.022uM remove_due_to_license_issue P26663 23023261 1721 GSVVIVGRIILSGSGSITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGIDPNIRTGVRTITTGAPVTYSTYGKFLADGGCSGGAYDIIICDECHSTDSTTILGIGTVLDQAETAGARLVVLATATPPGSVTVPHPNIEEVALSNTGEIPFYGKAIPIEAIRGGRHLIFCHSKKKCDELAAKLSGLGINAVAYYRGLDVSVIPTIGDVVVVATDALMTGYTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTVPQDAVSRSQRRGRTGRGRRGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETSVRLRAYLNTPGLPVCQDHLEFWESVFTGLTHIDAHFLSQTKQAGDNFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMACMSADLEVVT 4b76 A 2.14 BS01 PW1 A 1 V78 D81 R155 M485 F486 V524 C525 E628 V630 V92 D95 R169 M499 F500 V538 C539 E642 V644 T10 C16 H57 D81 G137 S139 T24 C30 H71 D95 G151 S153 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0004386,0005524,0006508,0008236,0019087 Kd=29uM remove_due_to_license_issue P26663 23023261 1721 GSVVIVGRIILSGSGSITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGIDPNIRTGVRTITTGAPVTYSTYGKFLADGGCSGGAYDIIICDECHSTDSTTILGIGTVLDQAETAGARLVVLATATPPGSVTVPHPNIEEVALSNTGEIPFYGKAIPIEAIRGGRHLIFCHSKKKCDELAAKLSGLGINAVAYYRGLDVSVIPTIGDVVVVATDALMTGYTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTVPQDAVSRSQRRGRTGRGRRGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETSVRLRAYLNTPGLPVCQDHLEFWESVFTGLTHIDAHFLSQTKQAGDNFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMACMSADLEVVT 4b77 A 1.8 BS01 54M A 1 Q12 D32 S35 Y71 W76 F108 I110 I118 D228 G230 Q16 D36 S39 Y75 W80 F112 I114 I122 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=7.9uM remove_due_to_license_issue IC50=7900nM P56817 23126626 1504 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b78 A 1.5 BS01 KGG A 1 G11 Q12 D32 S35 W76 F108 I110 I118 D228 G230 G11 Q12 D32 S35 W76 F108 I110 I118 D216 G218 D32 S35 N37 A39 Y71 D228 T231 D32 S35 N37 A39 Y71 D216 T219 3.4.23.46 0004190,0006508,0016020 ic50=3.2uM remove_due_to_license_issue IC50=40000nM P56817 23126626 1385 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 4b7j A 2.417 BS02 G39 A 1 D151 R225 E277 R293 R368 Y402 D69 R143 E195 R211 R286 Y320 D151 E278 R293 R368 Y402 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 Ki=11.1nM remove_due_to_license_issue F8UU09 23028314 1470 VKLAGNSSLCPVSGWAIYSKDNSIRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNRLRTQESECACVNGSCFTVMTDGPSDGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNDFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTIDK 4b7n A 2.84 BS01 ZMR A 1 R118 E119 D151 R152 W179 R225 E228 S247 E277 R293 R368 Y402 R36 E37 D69 R70 W97 R143 E146 S165 E195 R211 R286 Y320 D151 E278 R293 R368 Y402 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 remove_due_to_license_issue F8UU09 23028314 601 VKLAGNSSLCPVSGWAIYSKDNSIRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNRLRTQESECACVNGSCFTVMTDGPSDGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNDFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 4b7p A 1.7 BS01 9UN A 1 N51 A55 K58 D93 I96 G97 M98 D102 N106 L107 T184 N40 A44 K47 D82 I85 G86 M87 D91 N95 L96 T173 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.346nM remove_due_to_license_issue Kd=0.35nM P07900 23674492 1226 MEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 4b7q A 2.728 BS01 ZMR A 1 E119 D151 W179 R225 S247 E277 R293 R368 Y402 E37 D69 W97 R143 S165 E195 R211 R286 Y320 D151 E278 R293 R368 Y402 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 remove_due_to_license_issue C7FH46 23028314 601 VKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTIDK 4b7r A 1.9 BS03 G39 A 1 R118 E119 D151 R152 R225 R293 R368 Y402 R36 E37 D69 R70 R143 R211 R286 Y320 D151 E278 R293 R368 Y402 D69 E196 R211 R286 Y320 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=0.23nM remove_due_to_license_issue C7FH46 23028314 801 VKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTIDK 4b7z A 2.3 BS01 Q4Q A 1 W86 G121 Y124 Y337 F338 Y341 H447 W86 G121 Y124 Y330 F331 Y334 H440 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=49uM remove_due_to_license_issue IC50=49000nM P21836 23984975 600 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b80 A 2.5 BS01 A36 A 1 W86 Y124 Y337 F338 Y341 W86 Y124 Y333 F334 Y337 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F293 F295 E330 H443 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=40uM remove_due_to_license_issue IC50=40000nM P21836 23984975 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPGGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b81 A 2.8 BS01 ZN4 A 1 W86 G121 Y124 W286 Y337 Y341 H447 W86 G121 Y124 W279 Y330 Y334 H440 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue IC50=12000nM, Kd=11100nM P21836 23984975 600 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b82 A 2.1 BS01 B3Z A 1 W86 G121 Y124 E202 Y337 F338 Y341 H447 W86 G121 Y124 E202 Y330 F331 Y334 H440 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=41uM remove_due_to_license_issue IC50=41000nM P21836 23984975 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b83 A 2.4 BS01 B3V A 1 W86 G121 Y124 W286 F297 Y337 F338 Y341 H447 W86 G121 Y124 W280 F291 Y331 F332 Y335 H441 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue IC50=7000nM P21836 23984975 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b83 A 2.4 BS02 B3V A 2 R219 F222 F321 D323 R219 F222 F315 D317 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue IC50=7000nM P21836 23984975 1553 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b84 A 2.6 BS01 Z5K A 1 W86 G121 Y124 Y337 Y341 H447 W86 G121 Y124 Y332 Y336 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Kd=14800nM, IC50=22000nM P21836 23984975 1546 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPANDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 4b85 A 2.1 BS01 B3W A 1 W86 G121 G122 Y124 F297 Y337 F338 Y341 H447 W86 G121 G122 Y124 F291 Y331 F332 Y335 H441 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F291 F293 E328 H441 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=88uM remove_due_to_license_issue IC50=88000nM P21836 23984975 600 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4b95 C 2.8 BS01 UCK C 1 W88 F91 Y98 P99 R107 I109 H110 Y112 H115 W117 W27 F30 Y37 P38 R46 I48 H49 Y51 H54 W56 ? remove_due_to_license_issue P40337 23065727 1206 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQ 4b9k C 2.0 BS01 TG0 C 1 W88 F91 Y98 P99 R107 I109 H110 S111 Y112 H115 W117 W27 F30 Y37 P38 R46 I48 H49 S50 Y51 H54 W56 ? Ki=0.67uM remove_due_to_license_issue IC50=900nM P40337 23065727 1203 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4bae A 2.35 BS01 RWX A 1 N52 E56 D79 R82 G83 I84 P85 V125 R141 T169 N31 E35 D58 R61 G62 I63 P64 V87 R103 T131 5.6.2.2 0003677,0003918,0005524,0006265 ic50=3nM remove_due_to_license_issue P0C559 24126580 1256 GLEAVRKRPGMYIGSTGERGLHHLIWEVVDNAVDEAMAGFATRVDVKIHADGSVEVRDDGRGIPVEMHATGMPTIDVVMTQLHGVGVSVVNALSTRLEATVLRDGYEWFQYYDRSVPGKLKQGGETKETGTTIRFWADPEIFETTDYNFETVARRLQEMAFLNKGLTIELTDERDGKHRVFHYP 4bah B 1.94 BS03 MEL B 1 H79 Y83 W86 I209 D229 A230 S235 W257 G258 E259 G260 H43 Y47 W50 I172 D192 A193 S198 W220 G221 E222 G223 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=2.01nM remove_due_to_license_issue IC50=69nM, Ki=1.2nM P00734 23290007 1291 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4bak B 1.94 BS03 M67 B 1 H79 Y83 W86 I209 D229 A230 E232 S235 W257 G258 E259 G260 C261 H43 Y47 W50 I172 D192 A193 E195 S198 W220 G221 E222 G223 C224 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=1.22nM remove_due_to_license_issue P00734 23290007 1287 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 4bam B 1.88 BS03 MM9 B 1 H79 Y83 W86 L132 I209 D229 A230 C231 S235 V255 W257 G258 G260 C261 H43 Y47 W50 L96 I172 D192 A193 C194 S198 V218 W220 G221 G223 C224 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=1.14nM remove_due_to_license_issue P00734 23290007 1287 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 4ban B 1.87 BS03 M6S B 1 H79 Y83 W86 L132 I209 D229 A230 E232 S235 W257 G258 G260 C261 H43 Y47 W50 L96 I172 D192 A193 E195 S198 W220 G221 G223 C224 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=2.43nM remove_due_to_license_issue P00734 23290007 1287 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 4bao B 1.87 BS03 MVF B 1 H79 Y83 W86 I209 D229 A230 E232 S235 W257 G258 E259 G260 H43 Y47 W50 I172 D192 A193 E195 S198 W220 G221 E222 G223 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=4.29nM remove_due_to_license_issue P00734 23290007 1287 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 4baq B 1.89 BS03 M4Z B 1 H79 Y83 W86 I209 D229 A230 E232 S235 W257 G258 E259 G260 C261 H43 Y47 W50 I172 D192 A193 E195 S198 W220 G221 E222 G223 C224 H79 D135 E232 G233 D234 S235 G236 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=0.98nM remove_due_to_license_issue P00734 23290007 1287 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 4bb2 A 2.48 BS02 STR B 1 S19 R260 N264 S7 R243 N247 ? 0004867,0005615 remove_due_to_license_issue Ki=42nM P08185 23300763 1384 HHRGLASANVDFAFSLYKHLVALSPKKNIFISPVSISMALAMLSLGTCGHTRAQLLQGLGFNLTERSETEIHQGFQHLHQLFALEMTMGNALFLDGSLELLESFSADIAHYYESEVLAMNFQDWATASRQINSYVKNKTQGKIVDLFSGLDSPAILVLVNYIFFKGTWTQPFDLASTREENFYVDETTVVKVPMMLQSSTISYLHDSELPCQLVQMNYVGNGTVFFILPDKGKMNTVIAALSRDTINRWSAGLTSSQVDLYIPKVTISGVYDLGDVLEEMGIADLFTNQANFSRITQDAQLKSSKVVHKAVLQLNEEGVDTAGSTGVTLNLT 4bb2 B 2.48 BS01 STR B 1 F366 H368 W371 F16 H18 W21 ? remove_due_to_license_issue Ki=42nM P08185 23300763 1384 KPIILRFNQPFIIMIFDHFTWSSLFLARVMNPV 4bb4 A 1.65 BS01 32W A 1 I621 A645 K647 E664 M668 T693 M696 G699 L747 I16 A40 K42 E56 M60 T85 M88 G91 L139 D740 A742 R744 N745 D758 K781 P783 D132 A134 R136 N137 D150 K158 P160 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P54760 23398453 1889 FAKEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFGKIPIRWTAPEAIAFRKFTSASDAWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQVVSALDKMIRNPASLKIVA 4bb9 A 1.47 BS01 F1P A 1 G107 G108 S110 E153 S179 V180 G181 E348 H351 N512 K514 G97 G98 S100 E143 S169 V170 G171 E338 H341 N502 K504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 23621087 702 RFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQESTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLETTGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIGDHSDMFNQKAELTNQGPQFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4bbe A 1.9 BS01 3O4 A 1 L855 F860 V863 K882 E930 Y931 L932 G935 L983 D994 L15 F20 V23 K42 E90 Y91 L92 G95 L143 D154 N976 A978 R980 N981 D994 S1016 N136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0005524,0006468 ic50=3.6nM remove_due_to_license_issue IC50=974.7nM O60674 23127890 2229 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRNLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRD 4bbf A 2.0 BS01 O19 A 1 L855 G858 G861 V863 A880 Y931 L932 G935 D994 L15 G18 G21 V23 A40 Y91 L92 G95 D154 N976 A978 R980 N981 D994 S1016 N136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0005524,0006468 ic50=2.2nM remove_due_to_license_issue IC50=2.2nM O60674 23127890 2229 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRNLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRD 4bbg A 2.75 BS02 V02 A 1 E116 G117 E118 R119 A133 P137 E100 G101 E102 R103 A117 P121 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=4.8nM P52732 23394180 1370 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENININQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 4bbh A 1.63 BS02 YBN A 1 F105 Y211 H213 Y315 Y334 S335 N365 A366 L367 L388 V408 L409 L410 F79 Y185 H187 Y289 Y308 S309 N339 A340 L341 L362 V382 L383 L384 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=0.08uM remove_due_to_license_issue A5K1A2 23170970 1001 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4bc5 A 1.98 BS01 5FX A 1 Q97 Q98 H99 W137 R170 D280 N281 Q91 Q92 H93 W131 R164 D274 N275 2.7.1.17 0004856,0005524,0005829,0005975,0005997,0005998,0006091,0016301,0019640,0042732,0046835 Ki=25uM remove_due_to_license_issue O75191 23179721 1531 RRCCLGWDFSTQQVKVVAVDAELNVFYEESVHFDRDLPEFGTQGGVHVHKDGLTVTSPVLMWVQALDIILEKMKASGFDFSQVLALSGAGQQHGSIYWKAGAQQALTSLSPDLRLHQQLQDCFSISDCPVWMDSSTTAQCRQLEAAVGGAQALSCLTGSRAYERFTGNQIAKIYQQNPEAYSHTERISLVSSFAASLFLGSYSPIDYSDGSGMNLLQIQDKVWSQACLGACAPHLEEKLSPPVPSCSVVGAISSYYVQRYGFPPGCKVVAFTGDNPASLAGMRLEEGDIAVSLGTSDTLFLWLQEPMPALEGHIFCNPVDSQHYMALLCFKNGSLMREKIRNESVSRSWSDFSKALQSTEMGNGGNLGFYFDVMEITPEIIGRHRFNTENHKVAAFPGDVEVRALIEGQFMAKRIHAEGLGYRVMSKTKILATGGASHNREILQVLADVFDAPVYVIDTANSACVGSAYRAFHGLAGGTDVPFSEVVKLAPNPRLAATPSPGASQVYEALLPQYAKLEQRILSQ 4bcb A 1.7 BS01 4I4 A 1 F173 M235 G254 Y473 F476 S554 N555 A594 W595 R643 V644 F173 M235 G254 Y473 F476 S554 N555 A594 W595 R643 V644 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 23121075 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4bcc A 1.65 BS01 JKT A 1 F173 M235 G254 Y473 F476 S554 N555 W595 R643 F173 M235 G254 Y473 F476 S554 N555 W595 R643 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 remove_due_to_license_issue P23687 23121075 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4bcd A 1.5 BS01 TDV A 1 F173 M235 G254 F476 I478 S554 A594 W595 R643 V644 F173 M235 G254 F476 I478 S554 A594 W595 R643 V644 Y473 S554 D641 H680 Y473 S554 D641 H680 3.4.21.26 0004252,0005737,0005829,0006508,0008236,0070012 ic50=0.033uM remove_due_to_license_issue IC50=33nM P23687 23121075 791 MLSFQYPDVYRDETAIQDYHGHKVCDPYAWLEDPDSEQTKAFVEAQNKITVPFLEQCPIRGLYKERMTELYDYPKYSCHFKKGKRYFYFYNTGLQNQRVLYVQDSLEGEARVFLDPNILSDDGTVALRGYAFSEDGEYFAYGLSASGSDWVTIKFMKVDGAKELPDVLERVKFSCMAWTHDGKGMFYNAYPQQDGKSDGTETSTNLHQKLYYHVLGTDQSEDILCAEFPDEPKWMGGAELSDDGRYVLLSIREGCDPVNRLWYCDLQQESNGITGILKWVKLIDNFEGEYDYVTNEGTVFTFKTNRHSPNYRLINIDFTDPEESKWKVLVPEHEKDVLEWVACVRSNFLVLCYLHDVKNTLQLHDLATGALLKIFPLEVGSVVGYSGQKKDTEIFYQFTSFLSPGIIYHCDLTKEELEPRVFREVTVKGIDASDYQTVQIFYPSKDGTKIPMFIVHKKGIKLDGSHPAFLYGYGGFNISITPNYSVSRLIFVRHMGGVLAVANIRGGGEYGETWHKGGILANKQNCFDDFQCAAEYLIKEGYTSPKRLTINGGSNGGLLVATCANQRPDLFGCVIAQVGVMDMLKFHKYTIGHAWTTDYGCSDSKQHFEWLIKYSPLHNVKLPEADDIQYPSMLLLTADHDDRVVPLHSLKFIATLQYIVGRSRKQNNPLLIHVDTKAGHGAGKPTAKVIEEVSDMFAFIARCLNIDWIP 4bcf A 3.011 BS01 T6Q A 1 F30 A46 V79 F103 C106 D109 A153 L156 D167 F25 A41 V74 F90 C93 D96 A140 L143 D154 D149 K151 A153 N154 D167 T191 D136 K138 A140 N141 D154 T173 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 23252711 1327 DSVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKASIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKG 4bcg A 3.085 BS01 T3C A 1 I25 T29 V33 A46 V79 F103 C106 D109 L156 D167 I19 T23 V27 A40 V73 F89 C92 D95 L142 D153 D149 K151 A153 N154 D167 S180 T191 D135 K137 A139 N140 D153 S166 T177 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 23301767 1328 SVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAKNSQPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKGM 4bch A 2.958 BS01 T7Z A 1 A46 V79 F103 C106 D109 L156 D167 A40 V73 F90 C93 D96 L143 D154 D149 K151 A153 N154 D167 T191 D136 K138 A140 N141 D154 T173 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 23252711 1328 SVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKAGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKGM 4bci A 3.1 BS01 T3E A 1 I25 F30 V79 F103 C106 E107 L156 I21 F26 V75 F90 C93 E94 L143 D149 K151 A153 N154 D167 T191 D136 K138 A140 N141 D154 T174 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 23252711 1327 YDSVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKG 4bcj A 3.162 BS01 T9N A 1 F30 A46 V79 F103 C106 E107 H108 D109 L156 F25 A41 V74 F91 C94 E95 H96 D97 L144 D149 K151 A153 N154 D167 T191 D137 K139 A141 N142 D155 T175 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 23252711 1327 DSVECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKKGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKG 4bck A 2.052 BS01 T3E A 1 I10 V18 L83 H84 Q85 D86 K89 L134 I12 V20 L85 H86 Q87 D88 K91 L136 D127 K129 Q131 N132 D145 T158 T165 D129 K131 Q133 N134 D147 T160 T167 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.004uM remove_due_to_license_issue P24941 23252711 1298 GSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 4bcm A 2.45 BS01 T7Z A 1 I10 E12 V18 V64 F80 F82 L83 H84 D86 K89 L134 I13 E15 V21 V64 F80 F82 L83 H84 D86 K89 L134 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.123uM remove_due_to_license_issue P24941 23252711 1297 PGSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 4bcn C 2.1 BS01 T9N C 1 I10 A31 V64 F80 F82 L83 H84 D86 L134 D145 I12 A33 V66 F82 F84 L85 H86 D88 L136 D147 D127 K129 Q131 N132 D145 T158 T165 D129 K131 Q133 N134 D147 T160 T167 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.012uM remove_due_to_license_issue P24941 23252711 1296 GSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVP 4bco A 2.05 BS01 T6Q A 1 E8 K20 A31 V64 F80 F82 L83 H84 L134 D145 E9 K21 A32 V65 F81 F83 L84 H85 L135 D146 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.131uM remove_due_to_license_issue P24941 23252711 1299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4bcp A 2.26 BS01 T3C A 1 I10 V18 V64 F80 L83 H84 Q85 D86 K89 L134 D145 I11 V19 V65 F81 L84 H85 Q86 D87 K90 L135 D146 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=568nM remove_due_to_license_issue P24941 23301767 1299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4bcq C 2.4 BS01 TJF C 1 I10 V18 F80 L83 L134 I11 V17 F79 L82 L133 D127 K129 Q131 N132 D145 T158 T165 D126 K128 Q130 N131 D144 T157 T164 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=0.147uM remove_due_to_license_issue Ki=199nM P24941 23252711 1295 SMENFQKVEKIGEYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVP 4bcs A 1.8 BS01 BTN A 1 D12 L14 S16 Y33 T35 V37 A38 W68 F70 S71 T75 W95 N116 D10 L12 S14 Y31 T33 V35 A36 W66 F68 S69 T73 W93 N114 ? 0005576,0009374 Kd=103nM remove_due_to_license_issue P56734 24632863 1128 KCSLTGKWTDDLGSNMTIGAVNSRGEFTGTYITAVADNPGNITLSPLLGIQHKRASQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDISDDWIATRVGINIFTRQRTQK 4bcw A 1.5 BS02 TU0 A 1 Q92 H94 H119 F131 L198 Q89 H91 H116 F127 L194 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 23241068 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4bda A 2.6 BS01 VFB A 1 L226 A247 E302 M304 L354 L18 A35 E75 M77 L127 D347 K349 N352 D368 T387 D120 K122 N125 D141 T159 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1515 MSVYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdb A 2.5 BS01 ODO A 1 V234 L301 E302 M304 L354 V20 L73 E74 M76 L126 D347 K349 N352 D368 T387 D119 K121 N124 D140 T158 2.7.11.1 0004672,0005524,0006468 ic50=85.6uM remove_due_to_license_issue O96017 23776527 1515 MSVYPKALRDEYIMSKTLEVKLAFERKTCKKVAIKIISKLNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdc A 3.0 BS01 ODH A 1 L226 V234 M304 E305 G307 L354 L17 V21 M76 E77 G79 L126 D347 K349 N352 D368 T387 D119 K121 N124 D140 T158 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1513 SVYPKALRDEYIMSKTLGSEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdd A 2.67 BS01 Z0O A 1 V234 M304 G307 L354 V20 M75 G78 L125 D347 K349 N352 D368 T387 D118 K120 N123 D139 T156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1514 MSVYPKALRDEYIMSKTLEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bde A 2.55 BS01 CWS A 1 L226 V234 M304 L354 L18 V20 M77 L127 D347 K349 N352 D368 T387 D120 K122 N125 D141 T158 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1515 MSVYPKALRDEYIMSKTLEVKLAFERKTCKKVAIKIISKALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdf A 2.7 BS01 H3R A 1 A247 M304 G307 L354 A35 M77 G80 L127 D347 K349 N352 D368 T387 D120 K122 N125 D141 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1513 MSVYPKALRDEYIMSKTLGGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdg A 2.84 BS01 P3J A 1 L226 A247 L301 E302 M304 G307 L354 L18 A36 L75 E76 M78 G81 L128 D347 K349 N352 D368 T387 D121 K123 N126 D142 T161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1513 MSVYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdh A 2.7 BS01 WVI A 1 V234 A247 M304 V19 A32 M74 D347 K349 N352 D368 T387 D117 K119 N122 D138 T157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1514 SVYPKALRDEYIMSKTLEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL 4bdi A 2.32 BS01 HAU A 1 L226 A247 M304 E305 G307 L354 L18 A35 M79 E80 G82 L129 D347 K349 N352 D368 T387 D122 K124 N127 D143 T162 2.7.11.1 0004672,0005524,0006468 ic50=227.7uM remove_due_to_license_issue O96017 23776527 1516 MSVYPKALRDEYIMSKTLGGEVKLAFERKTCKKVAIKIISKALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVLAQP 4bdj A 3.01 BS01 Z2M A 1 L226 V234 A247 E302 M304 L354 L16 V19 A32 E72 M74 L124 D347 K349 N352 D368 T387 D117 K119 N122 D138 T156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1514 VYPKALRDEYIMSKTLGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVLA 4bdk A 3.3 BS01 RQQ A 1 L226 M304 E305 G307 L354 L16 M77 E78 G80 L127 D347 K349 N352 D368 T387 D120 K122 N125 D141 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96017 23776527 1514 VYPKALRDEYIMSKTLGGEVKLAFERKTCKKVAIKIISKALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVLA 4bds A 2.1 BS03 THA A 1 W82 E197 A328 W430 H438 W79 E194 A325 W425 H433 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G113 G114 G146 S195 A196 Y234 V285 F287 E322 H433 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 Ki=25nM remove_due_to_license_issue IC50=23nM, Ki=7nM P06276 23679855 701 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 4bdt A 3.104 BS01 HUW A 1 W86 G121 G122 S203 Y337 W439 H447 W82 G117 G118 S199 Y333 W435 H443 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G117 G118 G150 S199 A200 G238 F293 F295 E330 H443 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P22303 23679855 701 DAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPGGTGGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDPKAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSATDTLDEAERQWKAEFHRWSSYMVHW 4bek A 2.39 BS01 XK0 A 1 D93 Y132 D289 D37 Y76 D221 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=41.2uM remove_due_to_license_issue P56817 23735744 1447 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4bf1 A 1.35 BS02 9FK A 1 H94 H119 V121 F131 L198 T199 P202 H91 H116 V118 F127 L194 T195 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.4nM remove_due_to_license_issue Ki=2.4nM P00918 23859774 271 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4bf6 A 1.82 BS02 X0Q A 1 Q92 H94 H119 F131 L198 T199 T200 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=4.5nM remove_due_to_license_issue Ki=4.5nM P00918 23859774 1263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4bfd A 2.3 BS01 8T3 A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 D221 G223 T225 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.096uM remove_due_to_license_issue P56817 23735744 1447 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4bfp A 2.4 BS01 SWY A 1 H1031 S1033 P1034 F1035 A1038 I1039 G1043 F1044 D1045 H1048 I1051 I1059 Y1060 Y1071 G1074 I1075 H80 S82 P83 F84 A87 I88 G92 F93 D94 H97 I100 I108 Y109 Y120 G123 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 23762361 2162 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4bfr A 2.8 BS01 J82 A 1 Y772 M773 W781 I797 Y833 I845 E846 V847 V848 M920 I930 D931 Y575 M576 W584 I600 Y636 I648 E649 V650 V651 M723 I733 D734 2.7.11.1,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue Q8BTI9 24387221 2000 DSKIGVLIGKGLHEFDALKDPEVNEFRRKMRKFSEAKIQSLVGLSWIDWLKHTYPPEHEPSVLENLEDKLYGGKLVVAVHFENSQDVFSFQVSPNLNPIKINELAIQKRLTIASPCDYVLQVSGRVEYVFGDHPLIQFQYIRNCVMNRTLPHFILVECCKIKKMYEQEMIAIEAAIIWDNNNPFQITLVKGNKLNHVRAGLFHGTELLCKTVVSSEIIWNEQLEFDINICDLPRMARLCFAVYYPVAWVNTMVFDFKGQLRSGDVILHSWSSFPDELEEMLNPMGTVQTNPYAENATALHITFPENKKQPCYYPPFDKIIEKAAELASKKFLAVLKEILDRDPLSQLCENEMDLIWTLRQDCRENFPQSLPKLLLSIKWNKLEDVAQLQALLQIWPKLPPREALELLDFNYPDQYVREYAVGCLRQMSDEELSQYLLQLVQVLKYEPFLDCALSRFLLERALDNRRIGQFLFWHLRSEVHTPAVSVQFGVILEAYCRGSVGHMKVLSKQVEALNKLKTLNSLIKLNAVKLSRAKGKEAMHTCLKQSAYREALSDLQSPLNPCVILSELYVEKCKYMDSKMKPLWLVYSSRAFGEDSVGVIFKNGDDLRQDMLTLQMLRLMDLLWKEAGLDLRMLPYGCLATGDRSGLIEVVSTSETIADIQLNSSNVAATAAFNKDALLNWLKEYNSGDDLDRAIEEFTLSCAGYCVASYVLGIGDRHSDNIMVKKTGQLFHIDFGHILGNFRVPFILTYDFIHVIQQGKTGNTEKFGRFRQCCEDAYLILRRHGNLFITLFALMLTAGLPELTSVKDIQYLKDSLALGKSEEEALKQFKQKFDEALRESWTTKVNWMAHTVRKD 4bfy A 2.3 BS01 ZVY A 1 M144 H145 K147 G148 Y182 Y235 R238 M242 F254 I272 I276 N277 M138 H139 K141 G142 Y176 Y229 R232 M236 F248 I266 I270 N271 2.7.1.33 0004594,0005515,0005524,0005737,0005886,0015937,0016301 ic50=0.12uM remove_due_to_license_issue P9WPA7 23661699 501 PSPYVEFDRRQWRALRMSTPLALTEEELVGLRGLGEQIDLLEVEEVYLPLARLIHLQVAARQRLFAATAEFLGEPQQNPDRPVPFIIGVAGSVAVGKSTTARVLQALLARWDHHPRVDLVTTDGFLYPNAELQRRNLMHRKGFPESYNRRALMRFVTSVKSGSDYACAPVYSHLHYDIIPGAEQVVRHPDILILEGLNVLQTGPTLMVSDLFDFSLYVDARIEDIEQWYVSRFLAMRTTAFADPESHFHHYAAFSDSQAVVAAREIWRTINRPNLVENILPTRPRATLVLRKDADHSINRLRLRKL 4bfz A 2.1 BS01 ZVZ A 1 D129 L132 M144 H145 K147 G148 Y182 Y235 M242 F254 I276 N277 D123 L126 M138 H139 K141 G142 Y176 Y229 M236 F248 I270 N271 2.7.1.33 0004594,0005515,0005524,0005737,0005886,0015937,0016301 ic50=0.55uM remove_due_to_license_issue P9WPA7 23661699 501 PSPYVEFDRRQWRALRMSTPLALTEEELVGLRGLGEQIDLLEVEEVYLPLARLIHLQVAARQRLFAATAEFLGEPQQNPDRPVPFIIGVAGSVAVGKSTTARVLQALLARWDHHPRVDLVTTDGFLYPNAELQRRNLMHRKGFPESYNRRALMRFVTSVKSGSDYACAPVYSHLHYDIIPGAEQVVRHPDILILEGLNVLQTGPTLMVSDLFDFSLYVDARIEDIEQWYVSRFLAMRTTAFADPESHFHHYAAFSDSQAVVAAREIWRTINRPNLVENILPTRPRATLVLRKDADHSINRLRLRKL 4bg1 A 1.89 BS01 IVL A 1 Y177 W181 N191 A193 Y194 D204 Y205 N292 Y366 Y177 W181 N191 A193 Y194 D204 Y205 N292 Y366 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 ic50=0.49uM remove_due_to_license_issue O75936 24571165 901 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVEN 4bgg A 2.56 BS01 844 A 1 V214 A233 K235 T283 Y285 H286 G289 D293 L343 V12 A31 K33 T81 Y83 H84 G87 D91 L141 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=15nM Q04771 25101911 1000 TVARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSRHSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKI 4bgh A 1.95 BS01 3I6 A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 D145 I10 A31 F71 F73 L74 H75 Q76 D77 K80 L125 D136 D127 K129 Q131 N132 D145 T165 D118 K120 Q122 N123 D136 T142 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=4nM remove_due_to_license_issue P24941 23671017 1001 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4bgk A 2.18 BS01 RTK A 1 Y177 W181 N191 Y194 D204 Y205 N292 Y366 Y177 W181 N191 Y194 D204 Y205 N292 Y366 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 ic50=0.52uM remove_due_to_license_issue O75936 24571165 401 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVEN 4bgm A 2.4 BS01 DLT A 1 Y177 W181 N191 Y194 D204 Y205 N292 Y366 Y177 W181 N191 Y194 D204 Y205 N292 Y366 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 ic50=0.61uM remove_due_to_license_issue O75936 24571165 401 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVE 4bgx A 2.48 BS01 SIA C 1 Y91 V131 S132 S133 W149 H179 E186 L190 Q222 Y91 V131 S132 S133 W149 H179 E186 L190 Q222 ? 0019031,0019064,0046789 remove_due_to_license_issue Q6DQ34 23615615 2 DQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKTHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPVNDLCYPGDFNDYEELKHLLSRINHFEKIQIIPKSSWSSHEASLGVSSACPYQGKSSFFRNVVWLIKKNSTYPTIKRSYNNTNQEDLLVLWGIHHPNDAAEQTKLYQNPTTYISVGTSTLNQRLVPRIATRSKVNGQSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSTIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNSP 4bgy A 2.68 BS01 SIA E 1 Y91 V131 S132 S133 H179 E186 L190 Q222 Y91 V131 S132 S133 H179 E186 L190 Q222 ? 0019031,0019064,0046789 remove_due_to_license_issue Q6DQ34 23615615 3 DQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKTHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPVNDLCYPGDFNDYEELKHLLSRINHFEKIQIIPKSSWSSHEASLGVSSACPYQGKSSFFRNVVWLIKKNSTYPTIKRSYNNTNQEDLLVLWGIHHPNDAAEQTKLYQNPTTYISVGTSTLNQRLVPRIATRSKVNGQSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSTIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNSP 4bh3 A 2.0 BS01 SIA D 1 Y91 V131 S132 S133 W149 H179 E186 L190 Y93 V133 S134 S135 W151 H181 E188 L192 ? 0019031,0019064,0046789 remove_due_to_license_issue Q5EP31 23615615 3 DPDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKKHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPVNDLCYPGDFNDYEELKHLLSRINHFEKIQIIPKSSWSSHEASLGVSSACPYQGKSSFFRNVVWLIKKDSTYPTIKRSYNNTNQEDLLVLWGIHHPNDAAEQTKLYQNPTTYISVGTSTLNQRLVPRIATRSKVKGLSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSTIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLAIGLRNSPQ 4bh4 A 1.9 BS01 SIA D 1 Y91 V131 S132 S133 H179 E186 L190 Y93 V133 S134 S135 H181 E188 L192 ? 0019031,0019064,0046789 remove_due_to_license_issue Q5EP31 23615615 3 DPDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKKHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPVNDLCYPGDFNDYEELKHLLSRINHFEKIQIIPKSSWSSHEASLGVSSACPYQGKSSFFRNVVWLIKKDSTYPTIKRSYNNTNQEDLLVLWGIHHPNDAAEQTKLYQNPTTYISVGTSTLNQRLVPRIATRSKVKGLSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSTIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLAIGLRNSPQ 4bhf A 2.05 BS01 MZT A 1 Y177 W181 N191 Y194 D204 Y205 N292 Y366 Y177 W181 N191 Y194 D204 Y205 N292 Y366 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 Kd=4.1uM remove_due_to_license_issue O75936 24571165 401 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVE 4bhi A 2.15 BS01 RUJ A 1 Y177 W181 N191 Y194 D204 Y205 N292 Y366 Y177 W181 N191 Y194 D204 Y205 N292 Y366 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 Kd=9.3uM remove_due_to_license_issue O75936 24571165 401 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVEN 4bhn A 2.3 BS01 BH9 A 1 L686 V694 A707 K709 M754 Q756 V757 G759 G760 L810 L17 V25 A38 K40 M78 Q80 V81 G83 G84 L134 D803 K805 D807 N808 D822 T842 D127 K129 D131 N132 D146 T158 2.7.11.25 0004672,0005524,0006468 ic50=13nM remove_due_to_license_issue Q99683 23776076 1 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPEPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLEFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 4bhz A 2.85 BS01 Z0B A 1 I531 G605 L654 I16 G87 L136 D647 K649 N652 D664 T686 D129 K131 N134 D146 T156 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 23672464 1797 QSMSVKGRIYSILKQIGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4bi0 A 2.84 BS01 Z0W A 1 I531 A551 E603 G605 L654 I16 A36 E88 G90 L139 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 23672464 1797 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4bi1 A 2.7 BS01 ZO6 A 1 I531 G605 L654 I16 G89 L138 D647 K649 N652 D664 T686 D131 K133 N136 D148 T157 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 23672464 1797 QSMSVKGRIYSILKQIGSGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4bi2 A 3.11 BS01 ZO8 A 1 I531 M602 G605 L654 I16 M87 G90 L139 D647 K649 N652 D664 T686 D132 K134 N137 D149 T158 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 23672464 1797 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4bi6 A 1.45 BS01 PGA A 1 K13 H96 E170 I175 G176 G215 S216 L235 G237 G238 K12 H95 E169 I174 G175 G214 S215 L234 G236 G237 N11 K13 H96 E98 E170 G176 S216 N10 K12 H95 E97 E169 G175 S215 4.2.3.3,5.3.1.1 0004807,0005737,0005829,0006094,0006096,0008929,0016829,0016853,0019563,0046166 Kd=113.3uM remove_due_to_license_issue P36186 23894402 401 PARRPFIGGNFKCNGSLDFIKSHVAAIAAHKIPDSVDVVIAPSAVHLSTAIAANTSKQLRIAAQNVYLEGNGAWTGETSVEMLQDMGLKHVIVGHSERRRIMGETDEQSAKKAKRALEKGMTVIFCVGETLDERKANRTMEVNIAQLEALGKELGESKMLWKEVVIAYEPVWSIGTGVVATPEQAEEVHVGLRKWFVEKVAAEGAQHIRIIYGGSANGSNNEKLGQCPNIDGFLVGGASLKPEFMTMIDILTKTR 4bi7 A 1.6 BS01 PGA A 1 K13 H96 E170 I175 G176 S216 G237 G238 K12 H95 E169 I174 G175 S215 G236 G237 N11 K13 H96 E98 E170 G176 S216 N10 K12 H95 E97 E169 G175 S215 4.2.3.3,5.3.1.1 0004807,0005737,0005829,0006094,0006096,0008929,0016829,0016853,0019563,0046166 Kd=26.4uM remove_due_to_license_issue P36186 23894402 401 PARRPFIGGNFKCNGSLDFIKSHVAAIAAHKIPDSVDVVIAPSAVHLSTAIAANTSKQLRIAAQNVYLEGNGAWTGETSVEMLQDMGLKHVIVGHSERRRIMGETDEQSAKKAKRALEKGMTVIFCVGETLDERKANRTMEVNIAQLEALGKELGESKMLWKEVVIAYEPVWSIGTGVVATPEQAEEVHVGLRKWFAEKVAAEGAQHIRIIYGGSANGSNCEKLGQCPNIDGFLVGGASLKPEFMTMIDILTKTRT 4bib A 2.43 BS01 IEO A 1 V694 A707 M754 Q756 V757 L810 S821 D822 V25 A38 M77 Q79 V80 L133 S144 D145 D803 K805 D807 N808 D822 T842 D126 K128 D130 N131 D145 T157 2.7.11.25 0004672,0005524,0006468 ic50=0.63uM remove_due_to_license_issue Q99683 23776076 1940 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPELHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKREEFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 4bic A 2.62 BS01 IE4 A 1 G687 K688 V694 A707 Q756 V757 D807 L810 G18 K19 V25 A38 Q82 V83 D133 L136 D803 K805 D807 N808 D822 T842 D129 K131 D133 N134 D148 T162 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue Q99683 23776076 1 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPESQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGEFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 4bid A 2.8 BS01 IE8 A 1 L686 G687 V694 A707 K709 V738 I752 M754 E755 V757 D807 N808 L810 D822 L17 G18 V25 A38 K40 V61 I75 M77 E78 V80 D130 N131 L133 D145 D803 K805 D807 N808 D822 T842 D126 K128 D130 N131 D145 T157 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue Q99683 23776076 4000 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPELHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKREEFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 4bie A 2.36 BS01 IE6 A 1 G687 K688 G689 V694 A707 K709 Q756 V757 N808 L810 D822 G18 K19 G20 V25 A38 K40 Q79 V80 N131 L133 D145 D803 K805 D807 N808 D822 T842 D126 K128 D130 N131 D145 T159 2.7.11.25 0004672,0005524,0006468 ic50=0.79uM remove_due_to_license_issue Q99683 23776076 1942 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPELHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGEFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 4bio A 2.45 BS02 8XQ A 1 Y102 Y145 L188 T196 H199 F207 K214 H279 I281 Y92 Y135 L178 T186 H189 F197 K204 H269 I271 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 remove_due_to_license_issue Q9NWT6 26682036 601 SGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 4bis A 2.493 BS02 8HQ A 1 Y132 Y177 F185 H188 E190 K206 W208 Y125 Y170 F178 H181 E183 K199 W201 G170 Y177 H188 E190 H276 S288 G163 Y170 H181 E183 H269 S281 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=1700nM O75164 26682036 601 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 4bj8 E 2.4 BS01 BTN E 1 L16 S18 Y33 T35 S39 A43 W70 S74 W78 W96 D117 L13 S15 Y30 T32 S36 A40 W67 S71 W75 W93 D114 ? 0005576,0009374 Kd=5.13nM remove_due_to_license_issue E7F650 24204770 1123 SSCNVTGVWRNELGSTLRVKAEGSEVRGVYQTAVESTRGAAGHHRSARIIGMVSDGTQPTVSFSVLWEKGSCSAWVGQCFILDDGAQVLKTFWMLRSVADNLASAWGSTRMGEDIFFKT 4bj8 F 2.4 BS01 BTN F 1 S18 Y33 T35 V37 S39 A43 W70 S74 W78 W96 D117 S14 Y29 T31 V33 S35 A39 W66 S70 W74 W92 D113 ? 0005576,0009374 Kd=5.13nM remove_due_to_license_issue E7F650 24204770 1123 SCNVTGVWRNELGSTLRVKAEGSEVRGVYQTAVESTRGAAGHHRSARIIGMVSDGTQPTVSFSVLWEKGSCSAWVGQCFILDDGAQVLKTFWMLRSVADNLASAWGSTRMGEDIFFKT 4bj9 A 2.05 BS02 UHB A 1 H1031 G1032 S1033 F1035 I1039 H1048 A1049 I1051 G1058 Y1060 S1068 Y1071 H80 G81 S82 F84 I88 H97 A98 I100 G107 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=45nM remove_due_to_license_issue Q9H2K2 24900770 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4bjb A 2.3 BS02 P34 A 1 G1032 Y1060 A1062 K1067 S1068 Y1071 I1075 G81 Y102 A104 K109 S110 Y113 I117 2.4.2.-,2.4.2.30 0003950 ic50=219nM remove_due_to_license_issue IC50=2951nM Q9H2K2 24900770 2166 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDEMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4bjc A 2.2 BS01 RPB A 1 H1031 G1032 Y1060 F1061 A1062 K1067 S1068 Y1071 E1138 H80 G81 Y101 F102 A103 K108 S109 Y112 E174 2.4.2.-,2.4.2.30 0003950 ic50=14nM remove_due_to_license_issue IC50=890nM Q9H2K2 24900770 2162 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4bjx A 1.59 BS01 73B A 1 W81 P82 N140 I146 M149 W40 P41 N99 I105 M108 ? ic50=22nM remove_due_to_license_issue IC50=0.398107nM, Kd=4.4nM O60885 24009722 1169 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4bkj A 1.7 BS01 STI A 1 A653 K655 E672 M676 T701 Y703 M704 V763 H764 L773 A783 D784 F785 A54 K56 E73 M77 T102 Y104 M105 V149 H150 L159 A169 D170 F171 D766 R770 N771 D784 A793 D152 R156 N157 D170 A179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd=1.9nM remove_due_to_license_issue IC50=337nM, Kd=0.700000nM Q08345 24768818 1000 MPRVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSLDFPLNVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNTV 4bks C 2.2 BS01 X6C C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=150uM remove_due_to_license_issue Kd=150000nM P40337 24436777 1203 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4bkt C 2.35 BS01 QD0 C 1 W88 F91 Y98 H110 S111 Y112 H115 W117 W27 F30 Y37 H49 S50 Y51 H54 W56 ? Kd=240uM remove_due_to_license_issue Kd=240000nM P40337 24436777 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERL 4bky A 1.83 BS01 82B A 1 G18 T19 G20 A23 V25 A38 L86 E87 Y88 C89 G92 E136 L139 I149 G16 T17 G18 A21 V23 A36 L82 E83 Y84 C85 G88 E132 L135 I145 D132 K134 E136 N137 D150 S171 D128 K130 E132 N133 D146 S152 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.012uM remove_due_to_license_issue Q14680 23914841 1334 DYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCASLAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4bkz A 2.2 BS01 1WS A 1 I17 A38 L86 E87 Y88 C89 P90 N137 L139 I149 I16 A35 L80 E81 Y82 C83 P84 N131 L133 I143 D132 K134 E136 N137 D150 S171 D126 K128 E130 N131 D144 S150 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.027uM remove_due_to_license_issue Q14680 23914841 1335 KDYDELLKYYELHETIGTGAKVKLACHILTGEMVAIKIMDKNTLLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCASLAYAAPELIQGGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLRL 4bnt B 2.3 BS01 36E B 1 F107 N111 L114 F94 N98 L101 G16 S141 Y154 K158 G17 S128 Y137 K141 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=137.69uM remove_due_to_license_issue O54438 24015914 1248 SMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bnu A 2.0 BS01 9KQ B 1 W106 V110 L114 A156 G160 G163 W98 V102 L106 A148 G152 G155 G16 S141 Y154 K158 G18 S133 Y146 K150 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNRMKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bnu B 2.0 BS01 9KQ B 1 F107 V110 N111 L114 G160 G163 F100 V103 N104 L107 G153 G156 G16 S141 Y154 K158 G22 S134 Y147 K151 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.02uM remove_due_to_license_issue O54438 24015914 1248 NLYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNADEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bnv A 2.5 BS01 Q7U B 1 F107 V110 N111 L114 F164 F96 V99 N100 L103 F148 G16 S141 Y154 K158 G17 S130 Y138 K142 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1247 SMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGIEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYM 4bnv B 2.5 BS01 Q7U B 1 W106 F107 L114 G160 G163 W94 F95 L102 G143 G146 G16 S141 Y154 K158 G16 S129 Y137 K141 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.03uM remove_due_to_license_issue O54438 24015914 1247 MSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGIEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYM 4bnx A 2.3 BS01 O74 A 1 V110 N111 L114 A156 G160 G163 F164 V103 N104 L107 A149 G153 G156 F157 G16 S141 Y154 K158 G18 S134 Y147 K151 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.02uM remove_due_to_license_issue O54438 24015914 1247 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNARMKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYM 4bnx B 2.3 BS01 O74 A 1 F107 V110 N111 L114 G163 F164 F102 V105 N106 L109 G158 F159 G16 S141 Y154 K158 G21 S136 Y149 K153 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1247 LYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAMKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYM 4bny A 1.8 BS01 36I B 1 W106 L114 A156 G163 F164 W98 L106 A148 G155 F156 G16 S141 Y154 K158 G17 S133 Y146 K150 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNARMKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bny B 1.8 BS01 36I B 1 W106 F107 V110 L114 G163 F164 W92 F93 V96 L100 G149 F150 G16 S141 Y154 K158 G16 S127 Y140 K144 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.08uM remove_due_to_license_issue O54438 24015914 1248 MSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bnz A 2.5 BS01 8M5 A 1 F107 V110 L114 A156 G160 F164 F101 V104 L108 A150 G154 F158 G16 S141 Y154 K158 G18 S135 Y148 K152 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.26uM remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGRMKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bnz B 2.5 BS01 8M5 A 1 V110 L114 G163 V108 L112 G156 G16 S141 Y154 K158 G22 S139 Y147 K151 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 NLYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGITRDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo0 A 2.4 BS01 FXE A 1 W106 V110 L114 A156 G160 W94 V98 L102 A144 G148 G16 S141 Y154 K158 G17 S129 Y142 K146 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.2uM remove_due_to_license_issue O54438 24015914 1248 SMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo0 B 2.4 BS01 FXE A 1 F107 L114 A156 G160 G163 F164 F97 L104 A146 G150 G153 F154 G16 S141 Y154 K158 G17 S131 Y144 K148 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGIDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo1 A 2.2 BS01 NKH B 1 W106 V110 N111 L114 A156 G160 W100 V104 N105 L108 A146 G150 G16 S141 Y154 K158 G21 S135 Y144 K148 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 LYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo1 B 2.2 BS01 NKH B 1 F107 V110 L114 G160 G163 F94 V97 L101 G142 G145 G16 S141 Y154 K158 G15 S128 Y136 K140 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.05uM remove_due_to_license_issue O54438 24015914 1248 SLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo2 A 1.9 BS01 36K A 1 W106 V110 N111 L114 A156 G163 F164 W97 V101 N102 L105 A147 G154 F155 G16 S141 Y154 K158 G20 S132 Y145 K149 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.05uM remove_due_to_license_issue O54438 24015914 1248 YFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo2 B 1.9 BS01 36K A 1 F107 L114 A156 G160 G163 F164 F95 L102 A144 G148 G151 F152 G16 S141 Y154 K158 G15 S129 Y142 K146 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGIDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo3 A 2.5 BS01 U98 A 1 W106 F107 V110 N111 L114 A156 G160 F164 W94 F95 V98 N99 L102 A142 G146 F150 G16 S141 Y154 K158 G16 S129 Y140 K144 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 ic50=0.3uM remove_due_to_license_issue O54438 24015914 1248 MSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo3 B 2.5 BS01 U98 A 1 L114 G163 F164 L100 G145 F146 G16 S141 Y154 K158 G15 S127 Y136 K140 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo4 A 2.7 BS01 36G A 1 F107 L114 G160 F95 L102 G148 G16 S141 Y154 K158 G18 S129 Y142 K146 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo4 B 2.7 BS01 36G A 1 F107 V110 N111 G160 F100 V103 N104 G153 G16 S141 Y154 K158 G22 S134 Y147 K151 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 NLYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNADEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo5 A 2.6 BS01 WI4 B 1 W106 F107 V110 A156 A159 G160 W104 F105 V108 A154 A157 G158 G16 S141 Y154 K158 G21 S139 Y152 K156 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 LYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGITRDNDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo5 B 2.6 BS01 WI4 B 1 W106 V110 L114 A159 G160 G163 W95 V99 L103 A148 G149 G152 G16 S141 Y154 K158 G15 S130 Y143 K147 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo6 A 2.8 BS01 36P A 1 F107 V110 N111 L114 G163 F164 F96 V99 N100 L103 G149 F150 G16 S141 Y154 K158 G18 S130 Y140 K144 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo6 B 2.8 BS01 36P A 1 V110 N111 L114 F164 V105 N106 L109 F154 G16 S141 Y154 K158 G21 S136 Y144 K148 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 LYFQSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGITDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo7 A 2.6 BS01 J2T A 1 F107 V110 L114 F164 F98 V101 L105 F155 G16 S141 Y154 K158 G18 S132 Y145 K149 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAKDDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo7 B 2.6 BS01 J2T A 1 F107 V110 L114 F94 V97 L101 G16 S141 Y154 K158 G15 S128 Y136 K140 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGIEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo8 A 2.7 BS01 34X B 1 W106 V110 N111 L114 A156 G163 F164 W95 V99 N100 L103 A145 G152 F153 G16 S141 Y154 K158 G18 S130 Y143 K147 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo8 B 2.7 BS01 34X B 1 W106 V110 N111 G163 F164 W96 V100 N101 G147 F148 G16 S141 Y154 K158 G17 S131 Y138 K142 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 SMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGIDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo9 A 2.9 BS01 3X3 A 1 V110 N111 L114 G160 G163 F164 V98 N99 L102 G148 G151 F152 G16 S141 Y154 K158 G18 S129 Y142 K146 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGAMGNAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bo9 B 2.9 BS01 3X3 A 1 V110 N111 G160 G163 F164 V100 N101 G148 G151 F152 G16 S141 Y154 K158 G18 S131 Y142 K146 1.1.1.100 0004316,0006633,0016491,0016616,0030497,0050661,0051287 remove_due_to_license_issue O54438 24015914 1248 QSMSLQGKVALVTGASRGIGQAIALELGRLGAVVIGTATSASGAEKIAETLKANGVEGAGLVLDVSSDESVAATLEHIQQHLGQPLIVVNNAGDEWFDVVNTNLNSLYRLSKAVLRGMTKARWGRIINIGSVVGANAGQTNYAAAKAGLEGFTRALAREVGSRAITVNAVAPGFIDTDMTRELPEAQREALLGQIPLGRLGQAEEIAKVVGFLASDGAAYVTGATVPVNGGMYMS 4bps A 1.081 BS01 3EB A 1 Y155 R162 A179 T180 G181 Y215 F226 A244 I248 E338 Y142 R149 A166 T167 G168 Y202 F213 A231 I235 E325 3.3.2.13 0016787,0016803 Ki=1.02mM remove_due_to_license_issue Q9KID9 24036425 1345 SISVTAPYCRFEKTGSPDLEGDETVLGLIEHGTGHTDVSLVDGAPRTAVHTTTRDDEAFTEVWHAQRPVESGMDNGIAWARTDAYLFGVVRTGESGRYADATAALYTNVFQLTRSLGYPLLARTWNYVSGINTTNADGLEVYRDFCVGRAQALDEGGIDPATMPAATGIGAHGGGITCVFLAARGGVRINIENPAVLTAHHYPTTYGPRPPVFARATWLGPPEGGRLFISATAGILGHRTVHHGDVTGQCEVALDNMARVIGAENLRRHGVQRGHVLADVDHLKVYVRRREDLDTVRRVCAARLSSTAAVALLHTDIAREDLLVEIEGMVA 4bqa A 2.5 BS01 dna B 0 Y414 R419 R422 Y423 Y425 K432 R437 Y438 Y86 R91 R94 Y95 Y97 K104 R109 Y110 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P15036 25670864 1 ~ 10 MSFKDYIQERSDPVEQGKPVIPAAVLAGFTGSGPIQLWQFLLELLSDKSCQSFISWTGDGWEFKLADPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTSGKRYVYRFVCDLQNLLGFTPEELHAI 4bqa A 2.5 BS02 dna C 0 Q364 L365 W403 K407 K409 M412 K416 R419 Y423 Y424 K427 Q36 L37 W75 K79 K81 M84 K88 R91 Y95 Y96 K99 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P15036 25670864 1 ~ 10 MSFKDYIQERSDPVEQGKPVIPAAVLAGFTGSGPIQLWQFLLELLSDKSCQSFISWTGDGWEFKLADPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTSGKRYVYRFVCDLQNLLGFTPEELHAI 4bqa D 2.5 BS01 dna E 0 Y414 R419 R422 Y423 Y425 K432 R437 Y438 Y54 R59 R62 Y63 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P15036 25670864 1 ~ 10 GPIQLWQFLLELLSDKSCQSFISWTGDGWEFKLADPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTSGKRYVYRFVC 4bqa D 2.5 BS02 dna F 0 Q364 L365 W403 K407 M412 K416 Y423 Y424 Q4 L5 W43 K47 M52 K56 Y63 Y64 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P15036 25670864 1 ~ 10 GPIQLWQFLLELLSDKSCQSFISWTGDGWEFKLADPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTSGKRYVYRFVC 4bqa G 2.5 BS01 dna H 0 Y414 R419 R422 Y423 Y425 K432 R437 Y438 Y54 R59 R62 Y63 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P15036 25670864 1 ~ 10 GPIQLWQFLLELLSDKSCQSFISWTGDGWEFKLADPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTSGKRYVYRFVCD 4bqa G 2.5 BS02 dna I 0 Q364 W403 K407 M412 Y423 Y424 Q4 W43 K47 M52 Y63 Y64 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P15036 25670864 1 ~ 10 GPIQLWQFLLELLSDKSCQSFISWTGDGWEFKLADPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTSGKRYVYRFVCD 4bqg A 1.9 BS01 50Q A 1 N51 D93 M98 F138 W162 N36 D78 M83 F123 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 24100158 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4bqh A 1.75 BS01 9VU A 1 G44 V45 D46 F50 V209 G232 A236 A239 M370 K371 Y376 G48 V49 D50 F54 V208 G231 A235 A238 M363 K364 Y369 2.7.7.23 0003977,0005737,0006011,0006048,0016772,0016779,0020015,0070569 Kd=2.58uM remove_due_to_license_issue Q386Q8 23834437 1539 PLGSMSDRDVCIQRLTGANQDHILTALEHGSEAERASLTAQITNELAGVDFRHFNDVLRESLEISKSLAEPPAKDSFFDISSVDRRRGQAKRIKNLEAVGYKAIQKGQIAFLILAGGSGTRLGFDKPKGFFTCDGLQQRKSLFMMHCEKIRRRQEIAESISGSGRKARVQLLVMTSGQNDAETQRFFEENSYFGLEREQVHFFAQSSVPCYDENTGRIIMENRGRICAAPGGNGAVFAALAAPRATKTLQVKESLLQHLRKLGIAYVQIGNIDNLLANVADPVFIGYAIEEEAHVVVKTCPKRGPDERVGVFVRASGKWGVVEYTEIRAKEIDDATGELKFNCANISSNLCSLHFMSLAAERMKSFTQYHAARKKIPTIKGPVMGIKLEAFLFDLFRFVDECDHPPKDSGAFRIMQVDRDDEFGPVKNADGAASDTPADAVRLLLSQHTRWLITALETAAMGVDVTEAKEAVAVMRSCSIKAEISPLVSVGGEGLRQHLPRVIHQLLRNPPPVIFIRRDDE 4bqs A 2.15 BS02 K2Q A 1 D34 R136 D33 R135 2.7.1.71 0000287,0004765,0005524,0005737,0005829,0008652,0009073,0009423,0016301,0019632,0019752,0046872 Ki=62uM remove_due_to_license_issue P9WPY3 23889343 1172 APKAVLVGLPGSGKSTIGRRLAKALGVGLLDTDVAIEQRTGRSIADIFATDGEQEFRRIEEDVVRAALADHDGVLSLGGGAVTSPGVRAALAGHTVVYLEISAAEGVRRTGGNTVRPLLAGPDRAEKYRALMAKRAPLYRRVATMRVDTNRRNPGAVVRHILSRLQVPS 4bqt A 2.88 BS01 C5E A 1 Y91 W145 V146 C188 Y193 Y91 W145 V146 C188 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 22553201 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4bqt B 2.88 BS01 C5E B 1 Y91 W145 V146 Y186 C188 Y193 Y91 W145 V146 Y186 C188 Y193 ? 0004888,0005216,0005230,0005515,0006811,0016020,0034220,0042802,0046872,0098794 remove_due_to_license_issue Q8WSF8 22553201 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4bqw A 1.79 BS02 QNM A 1 D254 M299 Y303 Y310 H313 Y329 L343 H374 V376 R383 D67 M112 Y116 Y123 H126 Y142 L156 H187 V189 R196 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue Q9GZT9 23683440 901 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKY 4bqx A 1.79 BS02 UN9 A 1 D254 M299 Y303 Y310 H313 Y329 L343 H374 V376 R383 D67 M112 Y116 Y123 H126 Y142 L156 H187 V189 R196 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=300nM, EC50=79000nM, Kd=80nM Q9GZT9 23683440 601 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYL 4bqy A 1.53 BS02 FNT A 1 D254 M299 Y303 Y310 H313 I327 Y329 L343 H374 V376 R383 D67 M112 Y116 Y123 H126 I140 Y142 L156 H187 V189 R196 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue IC50=512nM Q9GZT9 23683440 601 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYLVRVE 4br3 A 2.2 BS01 U85 A 1 R117 D306 Q308 Y333 Y354 W420 W423 F435 Y440 R38 D203 Q205 Y230 Y251 W317 W320 F332 Y337 2.7.1.32,2.7.1.82 Kd=1.9uM remove_due_to_license_issue P35790 23813777 1458 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 4brx A 2.05 BS01 KGW A 1 I428 L501 C502 G505 E506 N551 L553 D564 L567 I16 L89 C90 G93 E94 N139 L141 D152 L155 D546 A548 R550 N551 D564 D134 A136 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.32uM remove_due_to_license_issue Q00944 23845217 1685 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRYMLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEK 4bs0 A 1.09 BS01 6NT A 1 W44 G83 C84 D127 L236 M237 T265 W41 G80 C81 D124 L233 M234 T262 E131 M172 H209 M237 D239 E128 M169 H206 M234 D236 3.2.1.8 0004553,0005975,0016798,0031176,0045493 Ki=2uM remove_due_to_license_issue P23360 24132235 1305 QSIDQLIKARGKVYFGVATDQNRLTTGKNAAIIKADFGMVWPENSMQWDATEPSQGNFNFAGADYLVNWAQQNGKLIGAGCLVWHNFLPSWVSSITDKNTLINVMKNHITTLMTRYKGKIRTWDVVGEAFNEDGSLRQNVFLNVIGEDYIPIAFQTARAADPNAKLYIMDYNLDSASYPKTQAIVNRVKQWRAAGVPIDGIGSQMHLSAGQGAGVLQALPLLASAGTPEVSILMLDVAGASPTDYVNVVNACLNVQSCVGITVMGVADPDSAFASSTPLLFDGNFNPKPAYNAIVQDLQ 4bs2 A -1.00 BS01 rna B 0 D105 I107 L109 G110 W113 K136 K145 F147 F149 D174 K176 P178 N179 K181 F194 R197 F221 R227 A228 F229 F231 S254 S258 N259 A260 E261 K263 D10 I12 L14 G15 W18 K41 K50 F52 F54 D79 K81 P83 N84 K86 F99 R102 F126 R132 A133 F134 F136 S159 S163 N164 A165 E166 K168 ? 0003676,0003723 remove_due_to_license_issue Q13148 24240615 1 ~ 12 GSHMASKTSDLIVLGLPWKTTEQDLKEYFSTFGEVLMVQVKKDLKTGHSKGFGFVRFTEYETQVKVMSQRHMIDGRWCDCKLPNSKQSQDEPLRSRKVFVGRCTEDMTEDELREFFSQYGDVMDVFIPKPFRAFAFVTFADDQIAQSLCGEDLIIKGISVHISNAEPKHNSNRQ 4bs4 A 1.89 BS02 A64 A 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 H80 G81 Y99 Y109 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=72nM remove_due_to_license_issue Q9H2K2 24116873 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4bs5 A 1.25 BS01 MG2 A 1 G145 C147 G191 G192 Y193 M194 G260 V285 N286 H287 Y334 G24 C26 G70 G71 Y72 M73 G139 V164 N165 H166 Y213 Q141 C147 H287 N307 Q20 C26 H166 N186 3.4.22.27 0006508,0008234 remove_due_to_license_issue O70370 24224654 1341 TLPDTVDWREKGCVTEVKYQGSCGACWAFSAVGALEGQLKLKTGKLISLSAQNLVDCSNEEKYGNKGCGGGYMTEAFQYIIDNGGIEADASYPYKAMDEKCHYNSKNRAATCSRYIQLPFGDEDALKEAVATKGPVSVGIDASHSSFFFYKSGVYDDPSCTGNVNHGVLVVGYGTLDGKDYWLVKNSWGLNFGDQGYIRMARNNKNHCGIASYCSYPEI 4bsq A 1.96 BS01 QQV A 1 G145 C147 K187 G191 G192 Y193 V285 N286 H287 Y334 G24 C26 K66 G70 G71 Y72 V164 N165 H166 Y213 Q141 C147 H287 N307 Q20 C26 H166 N186 3.4.22.27 0006508,0008234 remove_due_to_license_issue O70370 24224654 1341 TLPDTVDWREKGCVTEVKYQGSCGACWAFSAVGALEGQLKLKTGKLISLSAQNLVDCSNEEKYGNKGCGGGYMTEAFQYIIDNGGIEADASYPYKAMDEKCHYNSKNRAATCSRYIQLPFGDEDALKEAVATKGPVSVGIDASHSSFFFYKSGVYDDPSCTGNVNHGVLVVGYGTLDGKDYWLVKNSWGLNFGDQGYIRMARNNKNHCGIASYCSYPEI 4bt3 A 1.1 BS02 WTZ A 1 G57 T58 E65 R145 H194 H196 H207 E253 G38 T39 E46 R126 H175 H177 H188 E234 4.1.1.5 0016831,0045151,0047605 Ki=0.76mM remove_due_to_license_issue P23616 23985082 302 APKNVLFQYSTINALMLGQFEGDLTLKDLKLRGDMGLGTINDLDGEMIQMGTKFYQIDSTGKLSELPESVKTPFAVTTHFEPKEKTTLTNVQDYNQLTKMLEEKFENKNVFYAVKLTGTFKMVKARTVPKQTRPYPQLTEVTKKQSEFEFKNVKGTLIGFYTPNYAAALNVPGFHLHFITEDKTSGGHVLNLQFDNANLEISPIHEFDVQLPHTDDFAHSDLTQVTTSQVHQAESE 4bt4 A 1.6 BS02 QFH A 1 E65 R145 H194 H196 H207 E253 E46 R126 H175 H177 H188 E234 4.1.1.5 0016831,0045151,0047605 Ki=0.46mM remove_due_to_license_issue P23616 23985082 302 APKNVLFQYSTINALMLGQFEGDLTLKDLKLRGDMGLGTINDLDGEMIQMGTKFYQIDSTGKLSELPESVKTPFAVTTHFEPKEKTTLTNVQDYNQLTKMLEEKFENKNVFYAVKLTGTFKMVKARTVPKQTRPYPQLTEVTKKQSEFEFKNVKGTLIGFYTPNYAAALNVPGFHLHFITEDKTSGGHVLNLQFDNANLEISPIHEFDVQLPHTDDFAHSDLTQVTTSQVHQAESE 4bt5 A 1.1 BS02 23B A 1 T58 E65 R145 H194 H196 H207 E253 T39 E46 R126 H175 H177 H188 E234 4.1.1.5 0016831,0045151,0047605 Ki=1.72mM remove_due_to_license_issue P23616 23985082 302 APKNVLFQYSTINALMLGQFEGDLTLKDLKLRGDMGLGTINDLDGEMIQMGTKFYQIDSTGKLSELPESVKTPFAVTTHFEPKEKTTLTNVQDYNQLTKMLEEKFENKNVFYAVKLTGTFKMVKARTVPKQTRPYPQLTEVTKKQSEFEFKNVKGTLIGFYTPNYAAALNVPGFHLHFITEDKTSGGHVLNLQFDNANLEISPIHEFDVQLPHTDDFAHSDLTQVTTSQVHQAESE 4bti F 2.3 BS02 7R9 F 1 Q61 Y99 F174 A190 Q192 W215 G216 E217 G219 C220 G226 I227 Y228 Q46 Y85 F162 A180 Q182 W205 G206 E207 G208 C209 G216 I217 Y218 G193 S195 G196 G183 S185 G186 3.4.21.6 0004252,0006508 ic50=0.2nM remove_due_to_license_issue IC50=0.200000nM P00742 24175584 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4btk A 2.0 BS01 DTQ A 1 I72 K87 E101 C115 M131 L133 Q134 D200 I24 K39 E53 C67 M83 L85 Q86 D152 2.7.11.1 0004672,0005524,0006468 Kd=0.24uM remove_due_to_license_issue Kd=240nM Q5TCY1 24039150 1337 DILPANYVVKDRWKVLKKIGGGEIYEAMDLLTRENVALKVESAQQPKQVLKMEVAVLKKLQGKDHVCRFIGCGRNEKFNYVVMQLQGRNLADLRRSQPRGTFTLSTTLRLGKQILESIEAIHSVGFLHRDIKPSNFAMGRLPSTYRKCYMLDFGLARQYTNTTGDVRPPRNVAGFRGTVRYASVNAHKNREMGRHDDLWSLFYMLVEFAVGQLPWRKIKDKEQVGMIKEKYEHRMLLKHMPSEFHLFLDHIASLDYFTKPDYQLIMSVFENSMKERGIAENEAFDWE 4btl A 2.5 BS01 5GZ A 1 W86 G121 Y124 W286 Y337 F338 Y341 H447 W86 G121 Y124 W279 Y330 F331 Y334 H440 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=2.5uM remove_due_to_license_issue IC50=2500nM P21836 23984975 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4btl A 2.5 BS02 5GZ A 2 W286 H287 L289 S293 W279 H280 L282 S286 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=2.5uM remove_due_to_license_issue IC50=2500nM P21836 23984975 1549 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 4btm A 2.54 BS01 F8E A 1 I64 A85 C115 M131 L133 Q134 L199 I20 A41 C71 M87 L89 Q90 L155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=4100nM Q5TCY1 24039150 1340 ADILPANYVVKDRWKVLKKIGGGGFGEIYEAMDLLTRENVALKVESAQQPKQVLKMEVAVLKKLQGKDHVCRFIGCGRNEKFNYVVMQLQGRNLADLRRSQPRGTFTLSTTLRLGKQILESIEAIHSVGFLHRDIKPSNFAMGRLPSTYRKCYMLDFGLARQYTNTTGDVRPPRNVAGFRGTVRYASVNAHKNREMGRHDDLWSLFYMLVEFAVGQLPWRKIKDKEQVGMIKEKYEHRMLLKHMPSEFHLFLDHIASLDYFTKPDYQLIMSVFENSMKERGIAENEAFDWEK 4btt F 2.59 BS02 VYR F 1 Q61 T98 Y99 F174 A190 Q192 V213 S214 W215 G216 G226 Y228 Q46 T84 Y85 F162 A180 Q182 V203 S204 W205 G206 G216 Y218 G193 S195 G196 G183 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue IC50=2.6nM P00742 24175584 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4btu B 2.37 BS02 6XS B 1 Y99 F174 A190 Q192 V213 W215 G216 G219 C220 Y228 Y85 F162 A180 Q182 V203 W205 G206 G208 C209 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 ic50=0.5nM remove_due_to_license_issue IC50=0.500000nM P00742 24175584 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4btw A 2.8 BS04 JW7 A 1 Y176 L177 D180 T210 T212 F389 Y394 L469 Y125 L126 D129 T159 T161 F338 Y343 L418 Y372 D386 Y471 H520 H522 H684 Y321 D335 Y420 H469 H471 H633 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Q16853 24304424 2000 THPGQSQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFSH 4btw B 2.8 BS01 JW7 A 1 L447 Y448 L391 Y392 Y372 D386 Y471 H520 H522 H684 Y316 D330 Y415 H464 H466 H628 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Q16853 24304424 2000 SQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFS 4btw B 2.8 BS05 JW7 B 1 Y176 D180 T210 F389 Y394 L469 Y120 D124 T154 F333 Y338 L413 Y372 D386 Y471 H520 H522 H684 Y316 D330 Y415 H464 H466 H628 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Q16853 24304424 2000 SQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFS 4btx A 2.78 BS04 WF8 A 1 F173 Y176 T210 F389 Y394 L469 F120 Y123 T157 F336 Y341 L416 Y372 D386 Y471 H520 H522 H684 Y319 D333 Y418 H467 H469 H631 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Kd=200nM, IC50=290nM Q16853 24304424 2000 PGQSQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFSH 4btx B 2.78 BS01 WF8 A 1 L447 Y448 L391 Y392 Y372 D386 Y471 H520 H522 H684 Y316 D330 Y415 H464 H466 H628 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Kd=200nM, IC50=290nM Q16853 24304424 2000 SQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFSH 4btx B 2.78 BS05 WF8 B 1 Y176 T210 F389 Y394 L469 Y120 T154 F333 Y338 L413 Y372 D386 Y471 H520 H522 H684 Y316 D330 Y415 H464 H466 H628 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Kd=200nM, IC50=290nM Q16853 24304424 2000 SQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFSH 4bty A 3.1 BS04 JWF A 1 F173 Y176 L177 F389 Y394 L469 H762 F121 Y124 L125 F337 Y342 L417 H710 Y372 D386 Y471 H520 H522 H684 Y320 D334 Y419 H468 H470 H632 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Q16853 24304424 2000 HPGQSQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFSHN 4bty B 3.1 BS04 JWF B 1 F173 Y176 L177 D180 T210 T212 F389 Y394 L469 H762 F117 Y120 L121 D124 T154 T156 F333 Y338 L413 H706 Y372 D386 Y471 H520 H522 H684 Y316 D330 Y415 H464 H466 H628 1.4.3.21 0005507,0005509,0005515,0005737,0005769,0005783,0005794,0005886,0005902,0006954,0007155,0008131,0009308,0009986,0016020,0016491,0016641,0042802,0046872,0046982,0048038,0052595 remove_due_to_license_issue Q16853 24304424 2000 SQLFADLSREELTAVMRFLTQRLGPGLVDAAQARPSDNCVFSVELQLPPKAAALAHLDRGSPPPAREALAIVFFGRQPQPNVSELVVGPLPHPSYMRDVTVERHGGPLPYHRRPVLFQEYLDIDQMIFNRELPQASGLLHHCCFYKHRGRNLVTMTTAPRGLQSGDRATWFGLYYNISGAGFFLHHVGLELLVNHKALDPARWTIQKVFYQGRYYDSLAQLEAQFEAGLVNVVLIPDNGTGGSWSLKSPVPPGPAPPLQFYPQGPRFSVQGSRVASSLWTFSFGLGAFSGPRIFDVRFQGERLVYEISLQEALAIYGGNSPAAMTTRYVDGGFGMGKYTTPLTRGVDCPYLATYVDWHFLLESQAPKTIRDAFCVFEQNQGLPLRRHHSDLYSHYFGGLAETVLVVRSMSTLLNYDYVWDTVFHPSGAIEIRFYATGYISSAFLFGATGKYGNQVSEHTLGTVHTHSAHFKVDLDVAGLENWVWAEDMVFVPMAVPWSPEHQLQRLQVTRKLLEMEEQAAFLVGSATPRYLYLASNHSNKWGHPRGYRIQMLSFAGEPLPQNSSMARGFSWERYQLAVTQRKEEEPSSSSVFNQNDPWAPTVDFSDFINNETIAGKDLVAWVTAGFLHIPHAEDIPNTVTVGNGVGFFLRPYNFFDEDPSFYSADSIYFRGDQDAGACEVNPLACLPQAAACAPDLPAFSHGGFSHN 4bup A 2.166 BS02 SAM A 1 H90 Y195 S197 E198 G201 A202 F242 A261 F262 N264 H265 Y299 F304 E312 H34 Y101 S103 E104 G107 A108 F148 A167 F168 N170 H171 Y205 F210 E218 2.1.1.361,2.1.1.362 0042799 Kd=11.2uM remove_due_to_license_issue Q3U8K7 24049080 500 GSHMSSGMSAKELCENDDLATSLVLDPYLGFQTHKMNTRQEELKEVIERFKKDEHLEKAFKCLTSLNKNKMQEKLFKEHVFIYLRMFATDSGFEILPCNRYSSEQNGAKIVATKEWKRNDKIELLVGCIAELSEIEENMLLRHGENDFSVMYSTRKNCAQLWLGPAAFINHDCRPNCKFVSTGRDTACVKALRDIEPGEEISCYYGDGFFGENNEFCECYTCERRGTGAFKS 4buq A 2.199 BS01 KGM A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 ? 0007155,0009289 Kd=7.3nM remove_due_to_license_issue A2IC68 24900609 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4bvb A 2.0 BS01 OCZ A 1 I154 F157 F180 L199 Q228 N229 I230 D231 H248 I291 I33 F36 F59 L78 Q107 N108 I109 D110 H127 I170 P155 D156 F157 R158 N229 D231 H248 P34 D35 F36 R37 N108 D110 H127 2.3.1.286 0017136,0051287,0070403 remove_due_to_license_issue IC50=>50000nM Q9NTG7 23840057 1395 KLSLQDVAELIRARACQRVVVMVGAGISTPSGIPDFRSPGSGLYSNLQQYDLPYPEAIFELPFFFHNPKPFFTLAKELYPGNYKPNVTHYFLRLLHDKGLLLRLYTQNIDGLERVSGIPASKLVEAHGTFASATCTVCQRPFPGEDIRADVMADRVPRCPVCTGVVKPDIVFFGEPLPQRFLLHVVDFPMADLLLILGTSLEVEPFASLTEAVRSSVPRLLINRDLVGPLAWHPRSRDVAQLGDVVHGVESLVELLGWTEEMRDLVQRETGKL 4bw0 B 2.33 BS01 rna A 0 K30 G31 T32 N33 E34 K37 R41 D54 I88 E89 V90 P91 C92 A93 K30 G31 T32 N33 E34 K37 R41 D54 I88 E89 V90 P91 C92 A93 ? 0001682,0003723,0003735,0004526,0005737,0005840,0006412,0008033,0019843,0042254,1990904 remove_due_to_license_issue O29494 24149842 1 ~ 26 SYVRFEVPEDMQNEALSLLEKVRESGKVKKGTNETTKAVERGLAKLVYIAEDVDPPEIVAHLPLLCEEKNVPYIYVKSKNDLGRAVGIEVPCASAAIINEGELRKELGSLVEKIKGL 4bw1 A 1.4 BS01 S5B A 1 W81 P82 F83 L92 N140 I146 W40 P41 F42 L51 N99 I105 ? ic50=1.26uM remove_due_to_license_issue IC50=1258.93nM O60885 24000170 1172 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4bw2 A 1.92 BS01 UTH A 1 W81 F83 L92 N140 I146 W40 F42 L51 N99 I105 ? ic50=6.31uM remove_due_to_license_issue O60885 24000170 1170 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4bw3 A 1.5 BS01 9BM A 1 W81 P82 F83 L92 Y139 W40 P41 F42 L51 Y98 ? ic50=501nM remove_due_to_license_issue O60885 24000170 1172 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4bw4 A 1.67 BS01 9B6 A 1 W81 P82 F83 L92 N140 I146 M149 W40 P41 F42 L51 N99 I105 M108 ? ic50=631nM remove_due_to_license_issue O60885 24000170 1169 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4bxk A 2.2 BS01 1IU A 1 Q259 H331 A332 S333 A334 H361 E362 H365 Y369 H388 E389 K489 F490 H491 T496 Y498 Y501 Q256 H328 A329 S330 A331 H358 E359 H362 Y366 H385 E386 K486 F487 H488 T493 Y495 Y498 H331 A332 H361 E362 H365 E389 H491 Y501 H328 A329 H358 E359 H362 E386 H488 Y498 3.4.15.1 0006508,0008237,0008241,0016020 Ki=11.21nM remove_due_to_license_issue P12821 24015848 1001 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 4bxn A 2.793 BS02 6LX A 1 E116 G117 E118 R119 A133 P137 Y211 L214 E215 K216 G217 A218 R221 E99 G100 E101 R102 A116 P120 Y194 L197 E198 K199 G200 A201 R204 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=0.140000nM, Ki=0.500000nM, Kd=>10.0nM P52732 23875972 1375 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENIGRSGAVDKRAREAGNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 4bxo B 2.15 BS01 dna H 0 K173 V199 G200 V203 K155 V181 G182 V185 ? 0000785,0003677,0003682,0005515,0005634,0005654,0005829,0006281,0036297,0043231,0043240,0071821 remove_due_to_license_issue Q9BTP7 23932590 1 ~ 11 VHVPLGHIVANEKWRGSQLAEEMQGKIKLIFEDGLTPDFYLSNRCCILYVTEADLVAGNGYRKRLVRVRNSNNLKGIVVVEKTRMSEQYFPALQKFTVLDLGMVLLPVASQMEASCLVIQLVQEQTKEPSKNPLLLSEPSLLRTVQQIPGVGKVKAPLLLQKFPSIQQLSNASIGELEQVVGQAVAQQIHAFFTQP 4bxo B 2.15 BS02 dna I 0 G168 G170 V172 K173 G150 G152 V154 K155 ? 0000785,0003677,0003682,0005515,0005634,0005654,0005829,0006281,0036297,0043231,0043240,0071821 remove_due_to_license_issue Q9BTP7 23932590 1 ~ 11 VHVPLGHIVANEKWRGSQLAEEMQGKIKLIFEDGLTPDFYLSNRCCILYVTEADLVAGNGYRKRLVRVRNSNNLKGIVVVEKTRMSEQYFPALQKFTVLDLGMVLLPVASQMEASCLVIQLVQEQTKEPSKNPLLLSEPSLLRTVQQIPGVGKVKAPLLLQKFPSIQQLSNASIGELEQVVGQAVAQQIHAFFTQP 4byi A 2.6 BS01 FH3 A 1 R137 L139 V147 Y212 A213 P214 G216 L263 R12 L14 V22 Y87 A88 P89 G91 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 24195668 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4byj A 2.75 BS01 FH5 A 1 L139 V147 K162 Y212 A213 P214 G216 L263 L14 V22 K37 Y87 A88 P89 G91 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T150 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 24195668 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4bzn A 1.9 BS01 UGX A 1 G45 F49 V52 A65 K67 L120 R122 D128 L174 I185 D186 G13 F17 V20 A33 K35 L88 R90 D96 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=1.441uM remove_due_to_license_issue IC50=1441nM P11309 24139169 1306 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4bzo A 2.1 BS01 676 A 1 L44 F49 A65 K67 R122 L174 I185 D186 L12 F17 A33 K35 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.013uM remove_due_to_license_issue IC50=13nM P11309 24139169 1306 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4bzr A 1.84 BS02 K26 A 1 A354 S355 A356 W357 D358 Y360 H383 E384 H387 F391 H410 E411 F512 V518 Y523 A315 S316 A317 W318 D319 Y321 H344 E345 H348 F352 H371 E372 F469 V475 Y480 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H470 Y480 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=11nM, IC50=110nM P12821 24900839 1627 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPN 4bzs A 2.1 BS02 K26 A 1 S333 A334 W335 D336 Y338 H361 E362 H365 Y369 H388 E389 F490 Y501 S333 A334 W335 D336 Y338 H361 E362 H365 Y369 H388 E389 F490 Y501 H331 A332 H361 E362 H365 E389 H491 Y501 H331 A332 H361 E362 H365 E389 H491 Y501 3.4.15.1 0006508,0008237,0008241,0016020 Ki=75nM remove_due_to_license_issue Ki=11nM, IC50=110nM P12821 24900839 1001 LDPGLQPGNFSADEAGAQLFAQSYNSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQNFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSNMSRIYSTAKVCLPNKTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWNATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLQAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEGID 4c0r A 1.547 BS01 GDS A 1 V10 T12 T13 W51 N68 N69 I70 S71 R76 V115 N118 T119 S142 D144 Q148 K160 F162 E163 V10 T12 T13 W51 N68 N69 I70 S71 R76 V115 N118 T119 S142 D144 Q148 K160 F162 E163 ? Kd=12.2uM remove_due_to_license_issue Q93DA5 23701283 500 MDKTVTLATVGTTNPFSYEKKGKLTGYDIEVAKEVFKASDKYDVKYQKTEWTSIFSGLDSDKYQIGANNISYTKERANKYLYSNPTASNPLVLVVPKDSDIKSYNDIAGHSTQVVQGNTTVPMLQKFNKNHENNQVKLNFTSEDLAHQIRNVSDGKYDFKIFEKISAETIIKEQGLDNLKVIDLPSDQKPYVYFIFAQDQKDLQKFVNKRLKKLYENGTLEKLSKKYLGGSYLPDKKDM 4c1c A 1.18 BS01 MCO A 1 H118 D120 H179 C198 K201 G209 N210 H240 H79 D81 H140 C159 K162 G170 N171 H201 H116 H118 D120 H179 C198 K201 N210 H240 H77 H79 D81 H140 C159 K162 N171 H201 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P04190 26482303 1261 KTVIKNETGTISISQLNKNVWVHTELGSAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 4c1d A 1.198 BS01 X8Z A 1 F62 Y67 W87 H116 D118 H179 N210 F31 Y36 W56 H85 D87 H148 N179 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue Q9K2N0 26482303 350 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4c1e A 1.399 BS01 MCO A 1 F62 Y67 W87 H116 D118 H179 R205 G209 N210 H240 F31 Y36 W56 H85 D87 H148 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue Q9K2N0 26482303 350 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4c1f A 2.01 BS01 X8Z A 1 W46 D99 H157 K179 H215 W26 D79 H137 K159 H195 H95 H97 D99 H157 C176 K179 N185 H215 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P52699 26482303 300 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESK 4c1g A 1.714 BS03 MCO A 1 W46 V49 D99 H157 K179 G184 W26 V29 D79 H137 K159 G164 H95 H97 D99 H157 C176 K179 N185 H215 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P52699 26482303 305 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESK 4c1h A 1.1 BS01 X8Z A 1 W89 H118 D120 H179 C198 G209 N210 H240 W53 H82 D84 H143 C162 G173 N174 H204 H116 H118 D120 H179 C198 K201 N210 H240 H80 H82 D84 H143 C162 K165 N174 H204 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P04190 26482303 305 TVIKNETGTISISQLNKNVWVHTELGSFNGEAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 4c1m B 2.0 BS02 NIH B 1 Q91 H95 Q91 H95 Q91 D94 H95 D96 Q91 D94 H95 D96 1.11.2.2 0004601,0006979,0020037 Kd=15.8nM remove_due_to_license_issue Kd=15.8nM, IC50=5.01nM P05164 24194519 606 CPEQDKYRTITGMCNNRRSPTLGASNRAFVRWLPAEYEDGFSLPYGWTPGVKRNGFPVALARAVSNEIVRFPTDQLTPDQERSLMFMQWGQLLDHDLDFTPEPA 4c1m D 2.0 BS03 NIH B 1 P220 T238 R239 E242 F366 P108 T126 R127 E130 F254 T168 F170 D172 S174 R239 E242 H336 T56 F58 D60 S62 R127 E130 H224 1.11.2.2 0004601,0006979,0020037 remove_due_to_license_issue Kd=15.8nM, IC50=5.01nM P05164 24194519 606 VNCETSCVQQPPCFPLKIPPNDPRIKNQADCIPFFRSCPACPGSNITIRNQINALTSFVDASMVYGSEEPLARNLRNMSNQLGLLAVNQRFQDNGRALLPFDNLHDDPCLLTNRSARIPCFLAGDTRSSEMPELTSMHTLLLREHNRLATELKSLNPRWDGERLYQEARKIVGAMVQIITYRDYLPLVLGPTAMRKYLPTYRSYNDSVDPRIANVFTNAFRYGHTLIQPFMFRLDNRYQPMEPNPRVPLSRVFFASWRVVLEGGIDPILRGLMATPAKLNRQNQIAVDEIRERLFEQVMRIGLDLPALNMQRSRDHGLPGYNAWRRFCGLPQPETVGQLGTVLRNLKLARKLMEQYGTPNNIDIWMGGVSEPLKRKGRVGPLLACIIGTQFRKLRDGDRFWWENEGVFSMQQRQALAQISLPRIICDNTGITTVSKNNIFMSNSYPRDFVNCSTLPALNLASWREA 4c1t A 2.39 BS01 XYP B 1 A40 S41 Q254 W277 F350 A11 S12 Q225 W248 F321 remove_due_to_license_issue 24279727 1 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1t A 2.39 BS02 XYP B 2 N39 N72 W195 Q254 W277 N10 N43 W166 Q225 W248 remove_due_to_license_issue 24279727 2 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1t A 2.39 BS03 XYP B 3 W195 H199 W384 D386 W166 H170 W355 D357 remove_due_to_license_issue 24279727 3 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1t A 2.39 BS04 AHR B 1 N72 A76 L96 N43 A47 L67 remove_due_to_license_issue 24279727 4 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1u A 2.0 BS01 XYP B 1 W195 H199 W384 D386 W166 H170 W355 D357 remove_due_to_license_issue 24279727 1 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1u A 2.0 BS02 XYP B 2 N72 W195 Q254 W277 N43 W166 Q225 W248 remove_due_to_license_issue 24279727 2 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1u A 2.0 BS03 AHR B 1 N39 S144 E146 T318 Y346 N10 S115 E117 T289 Y317 remove_due_to_license_issue 24279727 3 DDKTITFWHNASAGEGRQYWENLAKSFEEANPGTKVEIQAIQNEDFAGKLQTAMQDPASGPDVFMSLGGAKTKEMIDAGQVMDLTDKISDTVKTDMKTTLSAATFDGKVYGVPVSVEPGGMWYSKDLFKKAGVSDVPATYEELLADAKKLKDSGTDAIALGAKDAWPAAHWYYWLVLRECSPEVYDKSVQDHDFSNACWVNAGKKLQELKDLKVFNDGFLTTTAQQGANSSAGLLANHKAAMELMGAWEPGVLKDLTPDQKPMADLGFFAFPEVAGGEGEPGALMGGVTYFCVNPKASQTSIDFVNYMGEKKNQEDYAKAFSTIPASEPARAVVTDESLKQVIEYLDKAPSMQLWMDTALGTNIGNALNAAVVNMLSGQGSPEDIVKAMQDAAQKG 4c1y A 2.23 BS01 MFB A 1 R25 E37 L69 Y88 W94 R24 E36 L68 Y87 W93 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 910 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4c1y A 2.23 BS02 MFB A 2 R126 E138 M140 T150 Y192 W198 R125 E137 M139 T149 Y191 W197 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 930 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4c1y A 2.23 BS03 MFB A 3 L24 Y40 W44 R282 E296 L23 Y39 W43 R281 E295 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 960 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4c2t A 3.997 BS01 dna M 0 F65 H93 R142 Y261 F263 R264 R362 T363 R422 G424 G426 T428 R459 L544 S546 T569 H571 N572 F633 F61 H89 R138 Y257 F259 R260 R358 T359 R418 G420 G422 T424 R455 L540 S542 T557 H559 N560 F621 K38 T39 D227 E228 Q258 R617 K34 T35 D223 E224 Q254 R605 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 2 ~ 26 AGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPGAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPARIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILDRGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEGQEGQVRLENLEELVSAAEEWSQDEANVGGSIADFLDDAALLSSDMRTKAEDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQPI 4c2t A 3.997 BS02 dna N 0 R393 F633 G634 R389 F621 G622 K38 T39 D227 E228 Q258 R617 K34 T35 D223 E224 Q254 R605 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 1 ~ 25 AGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPGAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPARIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILDRGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEGQEGQVRLENLEELVSAAEEWSQDEANVGGSIADFLDDAALLSSDMRTKAEDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQPI 4c2t B 3.997 BS01 dna M 0 R393 F633 R389 F616 K38 T39 D227 E228 Q258 R617 K34 T35 D223 E224 Q254 R600 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 2 ~ 26 AGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPGAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPARIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEGQEGQVRLENLEELVSAAEEWSQDEANVGGSIADFLDDAALLSSDMREDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQPI 4c2t B 3.997 BS02 dna N 0 F65 T91 R142 Y261 F263 R264 R362 T363 N364 A365 R422 G424 I425 G426 T428 L544 S546 H571 N572 F633 F61 T87 R138 Y257 F259 R260 R358 T359 N360 A361 R418 G420 I421 G422 T424 L538 S540 H554 N555 F616 K38 T39 D227 E228 Q258 R617 K34 T35 D223 E224 Q254 R600 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 1 ~ 25 AGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPGAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPARIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEGQEGQVRLENLEELVSAAEEWSQDEANVGGSIADFLDDAALLSSDMREDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQPI 4c2t C 3.997 BS01 dna O 0 H93 Q140 R142 Y261 F263 R362 T363 R422 G424 I425 G426 R459 S546 S547 H571 S593 F633 H92 Q139 R141 Y260 F262 R361 T362 R420 G422 I423 G424 R457 S539 S540 H560 S582 F622 K38 T39 D227 E228 Q258 R617 K37 T38 D226 E227 Q257 R606 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 1 ~ 26 TSSAGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPGAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPRIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILDRGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEEGQVRLENLEELVSAAEEWSQDEANSIADFLDDAALLSSVDDMRTKAEPEDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQPI 4c2t C 3.997 BS02 dna P 0 F633 G634 F622 G623 K38 T39 D227 E228 Q258 R617 K37 T38 D226 E227 Q257 R606 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 1 ~ 26 TSSAGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPGAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPRIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILDRGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEEGQVRLENLEELVSAAEEWSQDEANSIADFLDDAALLSSVDDMRTKAEPEDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQPI 4c2t D 3.997 BS01 dna O 0 R368 H462 M631 F633 R364 H457 M615 F617 K38 T39 D227 E228 Q258 R617 K35 T36 D223 E224 Q254 R601 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 1 ~ 26 SAGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPRIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILDRGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEGQEGQVRLENLEELVSAAEEWSQDEANVSIADFLDDAALLSSDMRTAEDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQP 4c2t D 3.997 BS02 dna P 0 R142 Y261 F263 R362 N364 A365 R422 G424 I425 S546 H571 N572 R138 Y257 F259 R358 N360 A361 R417 G419 I420 S539 H555 N556 K38 T39 D227 E228 Q258 R617 K35 T36 D223 E224 Q254 R601 5.6.2.4 0000725,0003677,0003678,0003689,0004386,0005524,0005829,0006338,0009378,0016787,0016853,0016887,0032508,0033202,0036121,0043138,0046872,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q9RTI9 24143224 1 ~ 26 SAGPDLLQALNPTQAQAADHFTGPALVIAGAGSGKTRTLIYRIAHLIGHYGVHPGEILAVTFTNKAAAEMRERAGHLVPAGDLWMSTFHSAGVRILRTYGEHIGLRRGFVIYDDDDQLDIIKEVMGSIPGIGAETQPRVIRGIIDRAKSNLWTPDDLDRSREPFISGLPRDAAAEAYRRYEVRKKGQNAIDFGDLITETVRLFKEVPGVLDKVQNKAKFIHVDEYQDTNRAQYELTRLLASRDRNLLVVGDPDQSIYKFRGADIQNILDFQKDYPDAKVYMLEHNYRSSARVLEAANKLIENNTERLDKTLKPVKEAGQPVTFHRATDHRAEGDYVADWLTRLHGEGRAWSEMAILYRTNAQSRVIEESLRRVQIPRIVGGVGFYDRREIRDILAYARLALNPADDVALRRIIGRPRRGIGDTALQKLMEWARTHHTSVLTACANAAEQNILDRGAHKATEFAGLMEAMSEAADNYEPAAFLRFVMETSGYLDLLRQEGQEGQVRLENLEELVSAAEEWSQDEANVSIADFLDDAALLSSDMRTAEDAVTLMTLHNAKGLEFPVVFIVGVEQGLLPSKGAIAEGPSGIEEERRLFYVGITRAMERLLMTAAQNRMQFGKTNAAEDSAFLEDIEGLFDTVDPYGQP 4c2v A 1.49 BS01 YJA A 1 K122 L138 E141 I142 Q145 M156 L168 L170 F172 A173 P174 G176 L223 A233 K36 L52 E55 I56 Q59 M70 L82 L84 F86 A87 P88 G90 L137 A147 D216 K218 E220 N221 D234 T252 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Ki=1nM remove_due_to_license_issue Q6DE08 24598913 1357 KFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQS 4c35 A 2.19 BS02 NU3 A 1 V57 A70 K72 E91 L95 V104 L120 Y122 L123 M173 T183 D184 F327 V48 A61 K63 E82 L86 V95 L111 Y113 L114 M164 T174 D175 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=0.56uM remove_due_to_license_issue P00517 24072592 1351 SEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSYGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVLEYLPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4c36 A 1.98 BS02 ZO9 A 1 L49 V57 A70 E121 Y122 M173 D184 F327 L37 V45 A58 E109 Y110 M161 D172 F315 D166 K168 E170 N171 D184 T201 D154 K156 E158 N159 D172 T189 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=19.8nM remove_due_to_license_issue P00517 24072592 1351 ESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSYGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVLEYLPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4c37 A 1.7 BS02 Z21 A 1 Y54 V57 A70 K72 L120 E121 Y122 M173 T183 D184 F327 Y42 V45 A58 K60 L108 E109 Y110 M161 T171 D172 F315 D166 K168 E170 N171 D184 T201 D154 K156 E158 N159 D172 T189 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=19.7nM remove_due_to_license_issue P00517 24072592 1351 ESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSYGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVLEYLPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4c38 A 1.58 BS02 VUP A 1 Y54 V57 A70 K72 L120 E121 Y122 M173 T183 D184 F327 Y41 V44 A57 K59 L107 E108 Y109 M160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=17.4nM remove_due_to_license_issue P00517 24072592 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSYGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVLEYLPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4c3k D 3.099 BS01 ADP D 1 G35 F36 G37 K58 I86 G87 K90 F92 G35 F36 G37 K44 I72 G73 K76 F78 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 remove_due_to_license_issue P0A3F4 24519945 1116 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGRVEFLQKLKLEIVVEDAQVDTVIDKIVAAARTGEIGDGKIFVSPVDQTIRIRTGEKNADAISAW 4c3k D 3.099 BS02 ADP F 1 G27 M28 T29 E62 V64 R101 R103 G27 M28 T29 E48 V50 R87 R89 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 remove_due_to_license_issue P0A3F4 24519945 1115 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGRVEFLQKLKLEIVVEDAQVDTVIDKIVAAARTGEIGDGKIFVSPVDQTIRIRTGEKNADAISAW 4c3k E 3.099 BS01 ADP D 1 G27 M28 T29 V64 R101 R103 G27 M28 T29 V49 R86 R88 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 remove_due_to_license_issue P0A3F4 24519945 1116 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGREFLQKLKLEIVVEDAQVDTVIDKIVAAARTGEIGDGKIFVSPVDQTIRIRTGEKNADA 4c3k E 3.099 BS02 ADP E 1 I7 G35 F36 G37 R38 K58 I86 G87 K90 F92 I7 G35 F36 G37 R38 K43 I71 G72 K75 F77 ? 0000166,0005515,0005524,0005829,0006808,0030234,0042802 remove_due_to_license_issue P0A3F4 24519945 1112 MKKIEAIIRPFKLDEVKIALVNAGIVGMTVSEVRGFGREFLQKLKLEIVVEDAQVDTVIDKIVAAARTGEIGDGKIFVSPVDQTIRIRTGEKNADA 4c4e A 2.6 BS01 4T9 A 1 I531 A551 K553 I586 E603 G605 L654 I16 A36 K38 I71 E88 G90 L139 D647 K649 N652 D664 T686 D132 K134 N137 D149 T162 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=25nM P33981 24256217 1796 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4c4f A 2.36 BS01 7CE A 1 I531 A551 K553 I586 M602 C604 G605 D608 L654 I17 A37 K39 I72 M88 C90 G91 D94 L140 D647 K649 N652 D664 T686 D133 K135 N138 D150 T160 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=26nM P33981 24256217 1799 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4c4g A 2.65 BS01 7RO A 1 I531 A551 K553 I586 M602 C604 G605 S611 L654 I663 I17 A37 K39 I72 M88 C90 G91 S97 L140 I149 D647 K649 N652 D664 T686 D133 K135 N138 D150 T157 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=6.0nM P33981 24256217 1796 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIAVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4c4h A 2.8 BS01 7RO A 1 I531 Q541 A551 K553 M602 C604 G605 I607 D608 S611 L654 I663 I16 Q25 A35 K37 M86 C88 G89 I91 D92 S95 L138 I147 D647 K649 N652 D664 T686 D131 K133 N136 D148 T153 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=6.0nM P33981 24256217 1795 QSMSVKGRIYSILKQIGSGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIATVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4c4i A 2.65 BS01 X20 A 1 I531 A551 K553 M602 C604 G605 I607 D608 L654 I663 I16 A36 K38 M87 C89 G90 I92 D93 L139 I148 D647 K649 N652 D664 T686 D132 K134 N137 D149 T157 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=5600nM P33981 24256217 1795 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4c4j A 2.5 BS01 X21 A 1 I531 A551 K553 E571 M602 C604 G605 I607 D608 S611 L654 I663 M671 I16 A36 K38 E56 M87 C89 G90 I92 D93 S96 L139 I148 M156 D647 K649 N652 D664 T686 D132 K134 N137 D149 T163 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=3.0nM P33981 24256217 1795 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTVGTVNYMPPEAIKDMSSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 4c4n A 2.36 BS01 IDS C 1 K88 R124 R154 K49 R85 R115 3.1.-.- 0007267,0007275 remove_due_to_license_issue Q62226 24062467 5 LTPLAYKQFIPNVAEKTLGASGRYEGKITRNSERFKELTPNYNPDIIFKDEENTGADRLMTQRCKDKLNALAISVMNQWPGVKLRVTEGWDEDGHHSEESLHYEGRAVDITTSDRDRSKYGMLARLAVEAGFDWVYYESKAHIHCSVKAEN 4c4n A 2.36 BS02 SGN C 1 K88 R124 K49 R85 3.1.-.- 0007267,0007275 remove_due_to_license_issue Q62226 24062467 6 LTPLAYKQFIPNVAEKTLGASGRYEGKITRNSERFKELTPNYNPDIIFKDEENTGADRLMTQRCKDKLNALAISVMNQWPGVKLRVTEGWDEDGHHSEESLHYEGRAVDITTSDRDRSKYGMLARLAVEAGFDWVYYESKAHIHCSVKAEN 4c52 A 2.049 BS01 X0D A 1 F97 Y101 L112 F123 V127 L130 F143 F146 G147 L150 F46 Y50 L61 F72 V76 L79 F92 F95 G96 L99 ? 0042981 Kd=2.1uM remove_due_to_license_issue IC50=22000nM Q07817 24456288 300 GPLGSMSQSNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 4c52 B 2.049 BS01 X0D B 1 Y101 Q111 L112 F123 L130 F143 F146 G147 M170 Y48 Q58 L59 F70 L77 F90 F93 G94 M117 ? 0042981 Kd=2.1uM remove_due_to_license_issue IC50=22000nM Q07817 24456288 300 LGSMSQSNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGNN 4c5d A 2.3 BS01 X0R A 1 F97 Y101 Q111 L112 F123 V127 R139 F143 F146 G147 L150 F46 Y50 Q60 L61 F72 V76 R88 F92 F95 G96 L99 ? 0042981 Kd=4uM remove_due_to_license_issue IC50=13000nM Q07817 24456288 2000 GPLGSMSQSNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 4c5d B 2.3 BS01 X0R B 1 F97 Y101 R103 A104 Q111 F123 L130 R139 F143 F146 G147 M170 F44 Y48 R50 A51 Q58 F70 L77 R86 F90 F93 G94 M117 ? 0042981 Kd=4uM remove_due_to_license_issue IC50=13000nM Q07817 24456288 2000 LGSMSQSNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYGNN 4c5w A 1.7 BS01 NM3 A 1 W181 N191 Y194 D204 Y205 N292 Y366 W181 N191 Y194 D204 Y205 N292 Y366 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 ic50=3.3uM remove_due_to_license_issue O75936 24571165 401 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVE 4c61 A 2.45 BS01 LMM A 1 L855 A880 M929 Y931 L932 P933 G935 N981 L983 G993 L12 A33 M77 Y79 L80 P81 G83 N129 L131 G141 D976 A978 R980 N981 D994 S1016 D124 A126 R128 N129 D142 S160 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.004uM remove_due_to_license_issue IC50=4.0nM O60674 24359159 2133 FEERHLKFLQQLGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYNLKLIMEYLPYGSLRDYLQAHAERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQM 4c66 A 1.87 BS01 H4C A 1 W81 P82 F83 V87 L92 N140 I146 W40 P41 F42 V46 L51 N99 I105 ? remove_due_to_license_issue O60885 24015967 1168 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 4c68 A 1.38 BS01 EN5 A 1 V96 D98 F105 T197 Y211 H213 S215 F226 Y242 G382 G384 D385 G386 V70 D72 F79 T171 Y185 H187 S189 F200 Y216 G356 G358 D359 G360 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0046872 remove_due_to_license_issue A5K1A2 25230674 1000 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4c6u A 2.4 BS01 TLG A 1 C171 F237 V278 A279 P280 H311 T313 H345 F402 G403 F404 G406 C169 F235 V276 A277 P278 H309 T311 H343 F400 G401 F402 G404 0016746 Kd=25.6uM remove_due_to_license_issue 24108128 1421 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSACSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c6v A 2.7 BS01 TLG A 1 C171 F237 V278 A279 P280 H311 T313 H345 F402 G403 F404 G406 C170 F236 V277 A278 P279 H310 T312 H344 F401 G402 F403 G405 0016746 remove_due_to_license_issue 24108128 1419 SQPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSACSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c6x A 1.95 BS01 TLM A 1 Q171 V278 A279 P280 H311 T313 H345 F402 G403 F404 G406 Q170 V277 A278 P279 H310 T312 H344 F401 G402 F403 G405 0016746 Ki=175.4uM remove_due_to_license_issue 24108128 1419 SQPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c6x B 1.95 BS02 TLM B 1 Q171 F237 A279 P280 H311 T313 H345 F402 G403 F404 G406 Q170 F236 A278 P279 H310 T312 H344 F401 G402 F403 G405 0016746 Ki=175.4uM remove_due_to_license_issue 24108128 1418 SQPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c6z A 1.8 BS01 TLE A 1 Q171 F237 V278 A279 P280 H311 T313 H345 F402 G403 F404 G406 Q169 F235 V276 A277 P278 H309 T311 H343 F400 G401 F402 G404 0016746 Ki=357uM remove_due_to_license_issue 24108128 1420 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c6z B 1.8 BS01 TLE B 1 Q171 F237 V278 A279 P280 H311 T313 H345 F402 F404 G406 Q169 F235 V276 A277 P278 H309 T311 H343 F400 F402 G404 0016746 Ki=357uM remove_due_to_license_issue 24108128 1421 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c70 A 1.75 BS01 TLJ A 1 Q171 F237 V278 A279 P280 H311 T313 H345 F402 G403 F404 G406 Q170 F236 V277 A278 P279 H310 T312 H344 F401 G402 F403 G405 0016746 Ki=305uM remove_due_to_license_issue 24108128 1423 SQPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c70 B 1.75 BS01 TLJ B 1 Q171 F237 V278 A279 P280 H311 T313 H345 F402 F404 G406 Q169 F235 V276 A277 P278 H309 T311 H343 F400 F402 G404 0016746 Ki=305uM remove_due_to_license_issue 24108128 1420 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c71 A 1.8 BS01 7RD A 1 Q171 F210 F237 V278 A279 P280 H311 T313 H345 I347 F402 G403 F404 G406 Q170 F209 F236 V277 A278 P279 H310 T312 H344 I346 F401 G402 F403 G405 0016746 Ki=384uM remove_due_to_license_issue 24108128 1423 SQPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c71 B 1.8 BS01 7RD B 1 Q171 F237 A279 P280 H311 T313 H345 I347 F402 G403 F404 G406 Q170 F236 A278 P279 H310 T312 H344 I346 F401 G402 F403 G405 0016746 Ki=384uM remove_due_to_license_issue 24108128 1419 SQPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c72 A 1.5 BS01 TLG A 1 Q171 A279 P280 H311 T313 H345 F402 G403 F404 G406 Q168 A276 P277 H308 T310 H342 F399 G400 F401 G403 0016746 Ki=8.2uM remove_due_to_license_issue 24108128 1429 PSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c72 B 1.5 BS01 TLG B 1 Q171 A279 P280 H311 T313 H345 F402 G403 F404 G406 Q168 A276 P277 H308 T310 H342 F399 G400 F401 G403 0016746 Ki=8.2uM remove_due_to_license_issue 24108128 1425 PSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c73 A 1.8 BS01 TLH A 1 Q171 F237 A279 P280 H311 T313 T315 H345 F402 G403 F404 G406 Q169 F235 A277 P278 H309 T311 T313 H343 F400 G401 F402 G404 0016746 Ki=12.1uM remove_due_to_license_issue 24108128 1427 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c73 B 1.8 BS01 TLH B 1 Q171 F237 A279 P280 H311 T313 T315 H345 F402 G403 F404 G406 Q169 F235 A277 P278 H309 T311 T313 H343 F400 G401 F402 G404 0016746 Ki=12.1uM remove_due_to_license_issue 24108128 1421 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSAQSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 4c7o A 2.6 BS01 rna E 0 E277 K278 E274 K275 3.6.5.4 0003924,0005525,0006614,0016887,0048500 remove_due_to_license_issue P0AGD7 24211265 0 ~ 47 NLTDRLSRTLRNISGRGRLTEDNVKDTLREVRMALLEADVALPVVREFINRVKEKAVGHEVNKSLTPGQEFVKIVRNELVAAMGEENQTLNLAAQPPAVVLMAGLQGAGKTTSVGKLGKFLREKHKKKVLVVSADVYRPAAIKQLETLAEQVGVDFFPSDVGQKPVDIVNAALKEAKLKFYDVLLVDTAGRLHVDEAMMDEIKQVHASINPVETLFVVDAMTGQDAANTAKAFNEALPLTGVVLTKVDGDARGGAALSIRHITGKPIKFLGVGEKTEALEPFHPDRIASRILG 4c7o B 2.6 BS01 rna E 0 F138 A159 Q160 D165 S168 F171 D172 Q175 A176 A179 R180 H198 L199 E202 K205 R208 V209 K212 F109 A130 Q131 D136 S139 F142 D143 Q146 A147 A150 R151 H169 L170 E173 K176 R179 V180 K183 3.6.5.4 0005525,0006614,0016887 remove_due_to_license_issue P10121 24211265 0 ~ 47 DDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFA 4c7o D 2.6 BS01 rna E 0 D165 A167 S168 F171 D172 K205 R208 V209 K212 D140 A142 S143 F146 D147 K180 R183 V184 K187 3.6.5.4 0005525,0006614,0016887 remove_due_to_license_issue P10121 24211265 0 ~ 47 GKKIDDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFARE 4c7t A 2.05 BS01 5RI A 1 I428 V436 L501 C502 G505 N551 L553 D564 L567 I15 V23 L88 C89 G92 N138 L140 D151 L154 D546 A548 R550 N551 D564 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.4uM remove_due_to_license_issue Q00944 24657306 1685 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRYMLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEK 4c8r A 2.82 BS02 6YT A 1 L199 H202 D204 L217 S229 F340 H347 R360 L199 H202 D204 L217 S229 F340 H347 R360 1.14.11.1 0005506,0005515,0005737,0005739,0005829,0008270,0008336,0016491,0016706,0042802,0045329,0046872,0051213,0070062 remove_due_to_license_issue O75936 26682037 601 MACTIQKAEALDGAHLMQILWYDEEESLYPAVWLRDNCPCSDCYLDSAKARKLLVEALDVNIGIKGLIFDRKKVYITWPDEHYSEFQADWLKKRCFSKQARAKLQRELFFPECQYWGSELQLPTLDFEDVLRYDEHAYKWLSTLKKVGIVRLTGASDKPGEVSKLGKRMGFLYLTFYGHTWQVQDKIDANNVAYTTGKLSFHTDYPALHHPPGVQLLHCIKQTVTGGDSEIVDGFNVCQKLKKNNPQAFQILSSTFVDFTDIGVDYCDFSVQSKHKIIELDDKGQVVRINFNNATRDTIFDVPVERVQPFYAALKEFVDLMNSKESKFTFKMNPGDVITFDNWRLLHGRRSYEAGTEISRHLEGAYADWDVVMSRLRILRQRVE 4c8z A 2.503 BS01 rna C 0 R22 Y26 H37 Q39 G40 F128 R129 R130 V133 H134 L142 E145 R149 E186 V187 D188 A225 K226 S228 R22 Y26 H37 Q39 G40 F128 R129 R130 V133 H134 L142 E145 R149 E186 V187 D188 A225 K226 S228 ? 0004519,0016788,0051607 remove_due_to_license_issue Q5SM65 24150936 14 ~ 28 MVLAALVLVLEGEGLPEPLGLRGFFYGLLREVAPEVHDQGENPFALGFGGREGAAWARVSLLVEGLYARLAPRLYALEGEEVRLGPPFRVRAVLQEGHPWAGVSTYPRLFQGPPSRDLALRFASPTFFRRKGVHYPVPEPRLVLESLLRRLEAFGPLKAPEGVREALLERTTVRSLEGRTLPARTEVDTAGFVGRVVYHLPRATEEEALWLSALGRFAFYSGVGAKTSLGYGRARAES 4c8z B 2.503 BS01 rna C 0 R174 H199 R202 R167 H192 R195 ? 0004519,0016788,0051607 remove_due_to_license_issue Q5SM65 24150936 14 ~ 28 MVLAALVLVLEGEGLPEPLGLRGFFYGLLREVAENPFALGFGGREGAAWARVSLLVEGLYARLAPRLYALEGEEVRLGPPFRVRAVLQEGHPWAGVSTYPRLFQGPPSRDLALRFASPTFFRRKGVHYPVPEPRLVLESLLRRLEAFGPLKAPEGVREALLERTTVRSLEGRTLPARTEVDTAGFVGRVVYHLPRATEEEALWLSALGRFAFYSGVGAKTSLGYGRARAES 4c94 A 3.0 BS01 KXN A 1 L59 S63 H70 R139 L61 S65 H72 R141 ? 0004864,0005634,0005737,0006952,0009738,0009813,0010427,0038023 remove_due_to_license_issue D0E0C7 24133217 160 AMAGVFTYESEFTSVIPPPKLFKAFVLDADNLIPKIAPQAVKSAEIIEGDGGVGTIKKIHLGEGSEYSYVKHKIDGIDKDNFVYSYSIIEGDAIGDKIEKISYEIKLVASGGGSIIKSTSHYHTKGEVEIKEEHVKAGKERAAGLFKIIENHLLAHPEEYN 4c9d A 3.0 BS01 rna C 0 H23 H42 P45 K47 A145 T146 S147 K148 P149 T153 Y155 R162 L163 S167 R208 K213 G251 A252 K253 Y256 H23 H42 P45 K47 A143 T144 S145 K146 P147 T151 Y153 R160 L161 S165 R206 K211 G249 A250 K251 Y254 ? 0004519,0016788,0046872,0051607 remove_due_to_license_issue Q53VU8 24150936 16 ~ 28 MPQAVVLELVGEKPPLYPARYAHGLFFALLSRVSPELAQKLHEAPRKPFTLAPLPGPEGATLKGTLRLRLTTLDDGLFAPFLRALLEAAPDGLPLGDSSYRLARVLATREGHPLAGATSWEELKEAPKREKATFRFLTPTVFATSKPGGRTRYTPLPDPRLIAGSLLDKWQAHSPFPYNPKEEAALRELFELDLEVAGFRNLRFHRVQAGKGFFPGFTGEATLRLWSQSLEAQEALGRLHALAFFSGVGAKTPYGMGLAVPL 4c9d A 3.0 BS02 rna D 0 E197 W228 E195 W226 ? 0004519,0016788,0046872,0051607 remove_due_to_license_issue Q53VU8 24150936 15 ~ 28 MPQAVVLELVGEKPPLYPARYAHGLFFALLSRVSPELAQKLHEAPRKPFTLAPLPGPEGATLKGTLRLRLTTLDDGLFAPFLRALLEAAPDGLPLGDSSYRLARVLATREGHPLAGATSWEELKEAPKREKATFRFLTPTVFATSKPGGRTRYTPLPDPRLIAGSLLDKWQAHSPFPYNPKEEAALRELFELDLEVAGFRNLRFHRVQAGKGFFPGFTGEATLRLWSQSLEAQEALGRLHALAFFSGVGAKTPYGMGLAVPL 4c9d B 3.0 BS01 rna C 0 E197 W228 E193 W224 ? 0004519,0016788,0046872,0051607 remove_due_to_license_issue Q53VU8 24150936 16 ~ 28 ASMPQAVVLELVGEKPPLYPARYAHGLFFALLSRVSPELAQKLHEAPRKPFTLAPLPRTLKGTLRLRLTTLDDGLFAPFLRALLEAAPDGLPLGDSSYRLARVLATREGHPLAGATSWEELKEAPKREKATFRFLTPTVFATSKPGGRTRYTPLPDPRLIAGSLLDKWQAHSPFPYNPKEEAALRELFELDLEVAGFRNLRFHRVQAGKGFFPGFTGEATLRLWSQSLEAQEALGRLHALAFFSGVGAKTPYGMGLAVPL 4c9d B 3.0 BS02 rna D 0 H23 H42 P45 K47 F144 A145 T146 S147 K148 P149 T153 Y155 R162 L163 R208 K213 G214 G251 A252 K253 P255 Y256 H25 H44 P47 K49 F140 A141 T142 S143 K144 P145 T149 Y151 R158 L159 R204 K209 G210 G247 A248 K249 P251 Y252 ? 0004519,0016788,0046872,0051607 remove_due_to_license_issue Q53VU8 24150936 15 ~ 28 ASMPQAVVLELVGEKPPLYPARYAHGLFFALLSRVSPELAQKLHEAPRKPFTLAPLPRTLKGTLRLRLTTLDDGLFAPFLRALLEAAPDGLPLGDSSYRLARVLATREGHPLAGATSWEELKEAPKREKATFRFLTPTVFATSKPGGRTRYTPLPDPRLIAGSLLDKWQAHSPFPYNPKEEAALRELFELDLEVAGFRNLRFHRVQAGKGFFPGFTGEATLRLWSQSLEAQEALGRLHALAFFSGVGAKTPYGMGLAVPL 4c9w A 1.65 BS01 VGH A 1 Y7 N33 F72 F74 M81 W117 D119 Y5 N31 F70 F72 M79 W115 D117 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=781nM remove_due_to_license_issue P36639 24695225 1158 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 4c9x A 1.2 BS01 VHS A 1 Y7 F27 F72 F74 E77 M81 W117 D119 Y5 F25 F70 F72 E75 M79 W115 D117 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=48nM remove_due_to_license_issue IC50=330nM P36639 24695225 1157 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 4ca4 A 2.84 BS01 KGM A 1 F1 N46 D47 D54 Q133 N135 Y137 D140 F1 N46 D47 D54 Q133 N135 Y137 D140 ? 0007155,0009289 remove_due_to_license_issue A2IC68 28250938 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDAPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4ca5 A 1.85 BS03 3EF A 1 Q281 H353 A354 S355 A356 E376 V380 H383 E384 H387 F391 H410 F457 K511 F512 H513 V518 Y520 Y523 F527 Q242 H314 A315 S316 A317 E337 V341 H344 E345 H348 F352 H371 F418 K472 F473 H474 V479 Y481 Y484 F488 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H474 Y484 3.4.15.1 0006508,0008237,0008241,0016020 Ki=0.41nM remove_due_to_license_issue Ki=0.41nM P12821 24289879 1700 DEAEASKFVEEYDRTSQVVWNEYAEANWNYNTNITTETSKILLQKNMQIANHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPNGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWNKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPNMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPNS 4ca6 A 1.91 BS02 3EF A 1 Q259 H331 A332 S333 S357 T358 H361 E362 H365 Y369 H388 E389 D393 E431 F435 K489 F490 H491 T496 Y498 Y501 F505 Q257 H329 A330 S331 S355 T356 H359 E360 H363 Y367 H386 E387 D391 E429 F433 K487 F488 H489 T494 Y496 Y499 F503 H331 A332 H361 E362 H365 E389 H491 Y501 H329 A330 H359 E360 H363 E387 H489 Y499 3.4.15.1 0006508,0008237,0008241,0016020 Ki=180nM remove_due_to_license_issue Ki=0.41nM P12821 24289879 1630 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLKTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 4ca7 A 1.82 BS02 3EF A 1 Q265 Q266 H337 A338 S339 A340 D360 F363 T364 H367 E368 H371 F375 H394 D399 K495 H497 V502 Y504 Y507 F511 Q247 Q248 H319 A320 S321 A322 D342 F345 T346 H349 E350 H353 F357 H376 D381 K477 H479 V484 Y486 Y489 F493 H337 A338 H367 E368 H371 E395 H497 Y507 H319 A320 H349 E350 H353 E377 H479 Y489 3.4.15.1 0006508,0008237,0008241,0016020 Ki=24nM remove_due_to_license_issue Q10714 24289879 1715 VKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 4ca8 A 1.99 BS01 3ES A 1 Q266 H337 A338 S339 T364 H367 E368 H371 F375 H394 D399 K495 H497 V502 Y504 Y507 F511 Q250 H321 A322 S323 T348 H351 E352 H355 F359 H378 D383 K479 H481 V486 Y488 Y491 F495 H337 A338 H367 E368 H371 E395 H497 Y507 H321 A322 H351 E352 H355 E379 H481 Y491 3.4.15.1 0006508,0008237,0008241,0016020 Ki=120nM remove_due_to_license_issue Q10714 24289879 1615 ALVKEEIQAKEYLENLNKELAKRTNVETEAAWAYGSNITDENEKKKNEISAELAKFMKEVASDTTKFQWRSYQSEDLKRQFKALTKLGYAALPEDDYAELLDTLSAMESNFAKVKVCDYKDSTKCDLALDPEIEEVISKSRDHEELAYYWREFYDKAGTAVRSQFERYVELNTKAAKLNNFTSGAEAWLDEYEDDTFEQQLEDIFADIRPLYQQIHGYVRFRLRKHYGDAVVSETGPIPMHLLGNMWAQQWSEIADIVSPFPEKPLVDVSAEMEKQGYTPLKMFQMGDDFFTSMNLTKLPQDFWDKSIIEKPTDGRDLVCHASAWDFYLTDDVRIKQCTRVTQDQLFTVHHELGHIQYFLQYQHQPFVYRTGANPGFHEAVGDVLSLSVSTPKHLEKIGLLKDYVRDDEARINQLFLTALDKIVFLPFAFTMDKYRWSLFRGEVDKANWNCAFWKLRDEYSGIEPPVVRSEKDFDAPAKYHISADVEYLRYLVSFIIQFQFYKSACIKAGQYDPDNVELPLDNCDIYGSAAAGAAFHNMLSMGASKPWPDALEAFNGERIMSGKAIAEYFEPLRVWLEAENIKNNVHIGWTTSNKCVS 4cae A 1.46 BS02 3F3 A 1 V96 E97 D98 F105 Y107 Y211 Y315 S319 Y334 N365 A366 L367 L388 L409 L410 V70 E71 D72 F79 Y81 Y185 Y289 S293 Y308 N339 A340 L341 L362 L383 L384 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=18nM remove_due_to_license_issue A5K1A2 24641010 1414 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4caf A 1.7 BS01 370 A 1 F105 Y107 Y211 Y315 Y334 S335 N365 A366 L367 L388 L409 L410 F79 Y81 Y185 Y289 Y308 S309 N339 A340 L341 L362 L383 L384 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=75nM remove_due_to_license_issue A5K1A2 24641010 1411 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4cbt A 3.03 BS01 9F4 A 1 H802 H803 F812 D840 H842 F871 D934 G974 H124 H125 F134 D162 H164 F193 D256 G296 3.5.1.98 remove_due_to_license_issue IC50=60.0nM P56524 24261862 2035 PRFTTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPLSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELLQQRPNANAVRSMEKVMEIHSKYWRCLQRH 4cby A 2.72 BS01 KEE A 1 R681 H802 H803 F812 D840 H842 F871 D934 R29 H150 H151 F160 D188 H190 F219 D282 3.5.1.98 remove_due_to_license_issue IC50=20.0nM P56524 24261862 2033 TTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPANRQKLDSKKLLGSLASVFVRLPCGGVGVDSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELDPLPEKVLQQRPNANAVRSMEKVMEIHSKYWRCLQ 4cc5 A 1.88 BS01 L5V A 1 L82 E110 Y219 K283 L81 E109 Y218 K282 E110 K112 D114 Y219 K307 E109 K111 D113 Y218 K306 6.5.1.2 0003911 Kd=38uM remove_due_to_license_issue Q9AIU7 24900632 1311 ADLSSRVNELHDLLNQYSYEYYVEDNPSVPDSEYDKLLHELIKIEEEHPEYKTVDSPTVRVGGEAQASFNKVNHDTPMLSLGNAFNEDDLRKFDQRIREQIGNVEYMCELKIDGLAVSLKYVDGYFVQGLTRGDGTTGEDITENLKTIHAIPLKMKEPLNVEVRGEAYMPRRSFLRLNEEKEKNDEQLFANPRNAAAGSLRQLDSKLTAKRKLSVFIYSVNDFTDFNARSQSEALDELDKLGFTTNKNRARVNNIDGVLEYIEKWTSQRESLPYDIDGIVIKVNDLDQQDEMGFTQKSPRWAIAYKFP 4cc6 A 2.01 BS01 L5Y A 1 L80 L82 E110 L111 K112 I113 Y219 K283 L79 L81 E109 L110 K111 I112 Y218 K282 E110 K112 D114 Y219 K307 E109 K111 D113 Y218 K306 6.5.1.2 0003911 ic50=0.23uM remove_due_to_license_issue IC50=230nM Q9AIU7 24900632 1311 ADLSSRVNELHDLLNQYSYEYYVEDNPSVPDSEYDKLLHELIKIEEEHPEYKTVDSPTVRVGGEAQASFNKVNHDTPMLSLGNAFNEDDLRKFDQRIREQIGNVEYMCELKIDGLAVSLKYVDGYFVQGLTRGDGTTGEDITENLKTIHAIPLKMKEPLNVEVRGEAYMPRRSFLRLNEEKEKNDEQLFANPRNAAAGSLRQLDSKLTAKRKLSVFIYSVNDFTDFNARSQSEALDELDKLGFTTNKNRARVNNIDGVLEYIEKWTSQRESLPYDIDGIVIKVNDLDQQDEMGFTQKSPRWAIAYKFP 4ccd A 1.97 BS01 2DG A 1 G48 T93 Y238 E258 S261 W291 Y303 G24 T69 Y214 E234 S237 W267 Y279 3.2.1.46 0004336,0006683 remove_due_to_license_issue P54818 24297913 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4cd0 A 2.23 BS01 AWJ A 1 L1122 V1130 A1148 M1199 G1202 D1203 L1256 G1269 D1270 Y1401 L29 V37 A48 M99 G102 D103 L156 G169 D170 Y295 D1249 A1251 R1253 N1254 D1270 L1291 D149 A151 R153 N154 D170 L185 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.2nM remove_due_to_license_issue Q9UM73 24432909 1500 PNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILMELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 4cd1 A 2.0 BS01 8E9 A 1 H50 R245 L249 K392 T393 R394 Y398 H13 R208 L212 K347 T348 R349 Y353 3.6.1.- 0016787 remove_due_to_license_issue O35795 24462745 1452 LKYGIVLDAGSSHTSMFVYKWPADKENDTGIVGQHSSCDVQGGGISSYANDPSKAGQSLVRCLEQALRDVPRDRHASTPLYLGATAGMRLLNLTSPEATARVLEAVTQTLTQYPFDFRGARILSGQDEGVFGWVTANYLLENFIKYGWVGRWIRPRKGTLGAMDLGGASTQITFETTSPSEDPGNEVHLRLYGQHYRVYTHSFLCYGRDQILLRLLASALQIHRFHPCWPKGYSTQVLLQEVYQSPCTMGQAIVSLSGTSNATLCRDLVSRLFNISSCPFSQCSFNGVFQPPVAGNFIAFSAFYYTVDFLTTVMGLPVGTLKQLEEATEITCNQTWTELQARVPGQKTRLADYCAVAMFIHQLLSRGYHFDERSFREVVFQKKAADTAVGWALGYMLNLTNLIPAD 4cd1 A 2.0 BS02 8E9 A 2 D76 S346 Y350 Y398 D39 S301 Y305 Y353 3.6.1.- 0016787 remove_due_to_license_issue O35795 24462745 1453 LKYGIVLDAGSSHTSMFVYKWPADKENDTGIVGQHSSCDVQGGGISSYANDPSKAGQSLVRCLEQALRDVPRDRHASTPLYLGATAGMRLLNLTSPEATARVLEAVTQTLTQYPFDFRGARILSGQDEGVFGWVTANYLLENFIKYGWVGRWIRPRKGTLGAMDLGGASTQITFETTSPSEDPGNEVHLRLYGQHYRVYTHSFLCYGRDQILLRLLASALQIHRFHPCWPKGYSTQVLLQEVYQSPCTMGQAIVSLSGTSNATLCRDLVSRLFNISSCPFSQCSFNGVFQPPVAGNFIAFSAFYYTVDFLTTVMGLPVGTLKQLEEATEITCNQTWTELQARVPGQKTRLADYCAVAMFIHQLLSRGYHFDERSFREVVFQKKAADTAVGWALGYMLNLTNLIPAD 4cd4 A 1.2 BS01 BMA A 1 D130 W373 R374 Q385 D78 W321 R322 Q333 3.2.1.78 0004553,0006080,0016985 remove_due_to_license_issue B3PGI1 24339341 1422 LPALIDTQATAETRALYRNLAKLRYKHLLFGHEDSLAYGVHWEGDMDRSDVRDVTGANPAVYGWELGGLELGHTANLDAVNFEKMQHWIKAGYSRGGVITISWHVFNPVSGGNSWDKTPAVHELIPGGARHATLKAYLDTFVAFNEGLADVDAQGNKHYPPIIFRPWHEHNGDWFWWGKGHASEQDYIALWRFTVHYLRDEKKLRNLIYAYSPDRSRIDMANFEAGYLYGYPGDAYVDIIGLDNYWDVGHEANTASADEQKAALTASLKQLVQIARSKGKIAALTETGNNRLTIDNFWTERLLGPISADADASEIAYVMVWRNANLAREKSEQFFAPFPGQATADDFKRFYQSEVVLFEDELPPLYR 4cd4 A 1.2 BS02 IFM A 1 H156 E221 Y297 E338 W373 H104 E169 Y245 E286 W321 3.2.1.78 0004553,0006080,0016985 remove_due_to_license_issue B3PGI1 24339341 1423 LPALIDTQATAETRALYRNLAKLRYKHLLFGHEDSLAYGVHWEGDMDRSDVRDVTGANPAVYGWELGGLELGHTANLDAVNFEKMQHWIKAGYSRGGVITISWHVFNPVSGGNSWDKTPAVHELIPGGARHATLKAYLDTFVAFNEGLADVDAQGNKHYPPIIFRPWHEHNGDWFWWGKGHASEQDYIALWRFTVHYLRDEKKLRNLIYAYSPDRSRIDMANFEAGYLYGYPGDAYVDIIGLDNYWDVGHEANTASADEQKAALTASLKQLVQIARSKGKIAALTETGNNRLTIDNFWTERLLGPISADADASEIAYVMVWRNANLAREKSEQFFAPFPGQATADDFKRFYQSEVVLFEDELPPLYR 4cd5 A 1.1 BS01 BMA A 1 D130 W373 R374 Q385 D78 W321 R322 Q333 3.2.1.78 0004553,0006080,0016985 remove_due_to_license_issue B3PGI1 24339341 1422 LPALIDTQATAETRALYRNLAKLRYKHLLFGHEDSLAYGVHWEGDMDRSDVRDVTGANPAVYGWELGGLELGHTANLDAVNFEKMQHWIKAGYSRGGVITISWHVFNPVSGGNSWDKTPAVHELIPGGARHATLKAYLDTFVAFNEGLADVDAQGNKHYPPIIFRPWHEHNGDWFWWGKGHASEQDYIALWRFTVHYLRDEKKLRNLIYAYSPDRSRIDMANFEAGYLYGYPGDAYVDIIGLDNYWDVGHEANTASADEQKAALTASLKQLVQIARSKGKIAALTETGNNRLTIDNFWTERLLGPISADADASEIAYVMVWRNANLAREKSEQFFAPFPGQATADDFKRFYQSEVVLFEDELPPLYR 4cd5 A 1.1 BS02 MVL A 1 H156 H220 E221 Y297 E338 W373 H104 H168 E169 Y245 E286 W321 3.2.1.78 0004553,0006080,0016985 remove_due_to_license_issue B3PGI1 24339341 1423 LPALIDTQATAETRALYRNLAKLRYKHLLFGHEDSLAYGVHWEGDMDRSDVRDVTGANPAVYGWELGGLELGHTANLDAVNFEKMQHWIKAGYSRGGVITISWHVFNPVSGGNSWDKTPAVHELIPGGARHATLKAYLDTFVAFNEGLADVDAQGNKHYPPIIFRPWHEHNGDWFWWGKGHASEQDYIALWRFTVHYLRDEKKLRNLIYAYSPDRSRIDMANFEAGYLYGYPGDAYVDIIGLDNYWDVGHEANTASADEQKAALTASLKQLVQIARSKGKIAALTETGNNRLTIDNFWTERLLGPISADADASEIAYVMVWRNANLAREKSEQFFAPFPGQATADDFKRFYQSEVVLFEDELPPLYR 4cd6 A 1.64 BS01 IFM A 1 R104 E151 Y203 E231 W245 Y247 W281 Y299 R99 E146 Y198 E226 W240 Y242 W276 Y294 3.2.1.78 remove_due_to_license_issue A5H1I6 24339341 500 SAFDLGFIRGMTFGFVGQHGTWGTDEARASMRALAEQPFNWVTLAFAGLMEHPGDPAIAYGPPVTVSDDEIASMAELAHALGLKVCLKPTVNCRDGTWRGEIRFEKEHGPDLESWEAWFGSYSDMMAHYAHVAKRTGCEMFCVGCEMTTAEPHEAMWRETIARVRTEYDGLVTYNCNHGREEHVRFWDAVDLISSSAYYPIDRWRDRVPVLREVAEAHEKPLFFMEVGCPSRSGSGACPWDYRHPGAVCLDEQARFYEAMFAAMPDEPWFKGYMLWEWPWKLYPREAASEDGSYCIYGKPAEDVVARAFSAIANR 4cd6 A 1.64 BS02 BMA A 1 F20 N97 Y247 W281 E282 F15 N92 Y242 W276 E277 3.2.1.78 remove_due_to_license_issue A5H1I6 24339341 501 SAFDLGFIRGMTFGFVGQHGTWGTDEARASMRALAEQPFNWVTLAFAGLMEHPGDPAIAYGPPVTVSDDEIASMAELAHALGLKVCLKPTVNCRDGTWRGEIRFEKEHGPDLESWEAWFGSYSDMMAHYAHVAKRTGCEMFCVGCEMTTAEPHEAMWRETIARVRTEYDGLVTYNCNHGREEHVRFWDAVDLISSSAYYPIDRWRDRVPVLREVAEAHEKPLFFMEVGCPSRSGSGACPWDYRHPGAVCLDEQARFYEAMFAAMPDEPWFKGYMLWEWPWKLYPREAASEDGSYCIYGKPAEDVVARAFSAIANR 4cd8 A 1.47 BS01 MVL A 1 R104 E151 Y203 E231 W245 Y247 W281 Y299 R99 E146 Y198 E226 W240 Y242 W276 Y294 3.2.1.78 remove_due_to_license_issue A5H1I6 24339341 400 SAFDLGFIRGMTFGFVGQHGTWGTDEARASMRALAEQPFNWVTLAFAGLMEHPGDPAIAYGPPVTVSDDEIASMAELAHALGLKVCLKPTVNCRDGTWRGEIRFEKEHGPDLESWEAWFGSYSDMMAHYAHVAKRTGCEMFCVGCEMTTAEPHEAMWRETIARVRTEYDGLVTYNCNHGREEHVRFWDAVDLISSSAYYPIDRWRDRVPVLREVAEAHEKPLFFMEVGCPSRSGSGACPWDYRHPGAVCLDEQARFYEAMFAAMPDEPWFKGYMLWEWPWKLYPREAASEDGSYCIYGKPAEDVVARAFSAIA 4cd8 A 1.47 BS02 BMA A 1 F20 N97 Y247 W281 E282 F15 N92 Y242 W276 E277 3.2.1.78 remove_due_to_license_issue A5H1I6 24339341 401 SAFDLGFIRGMTFGFVGQHGTWGTDEARASMRALAEQPFNWVTLAFAGLMEHPGDPAIAYGPPVTVSDDEIASMAELAHALGLKVCLKPTVNCRDGTWRGEIRFEKEHGPDLESWEAWFGSYSDMMAHYAHVAKRTGCEMFCVGCEMTTAEPHEAMWRETIARVRTEYDGLVTYNCNHGREEHVRFWDAVDLISSSAYYPIDRWRDRVPVLREVAEAHEKPLFFMEVGCPSRSGSGACPWDYRHPGAVCLDEQARFYEAMFAAMPDEPWFKGYMLWEWPWKLYPREAASEDGSYCIYGKPAEDVVARAFSAIA 4ce1 A 2.01 BS01 7FK A 1 N37 A41 D79 M84 N92 F124 T171 L173 N37 A41 D79 M84 N92 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 24435512 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 4ce2 A 2.38 BS01 BO5 A 1 N37 A41 D79 M84 N92 F124 T171 L173 N37 A41 D79 M84 N92 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 24435512 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 4ce3 A 2.31 BS01 L4V A 1 N37 A41 D79 N92 F124 T171 L173 N37 A41 D79 N92 F124 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P02829 24435512 1215 MASETFEFQAEITQLMSLIINTVYSNKEIFLRELISNASDALDKIRYKSLSDPKQLETEPDLFIRITPKPEQKVLEIRDSGIGMTKAELINNLGTIAKSGTKAFMEALSAGADVSMIGQFGVGFYSLFLVADRVQVISKSNDDEQYIWESNAGGSFTVTLDEVNERIGRGTILRLFLKDDQLEYLEEKRIKEVIKRHSEFVAYPIQLVVTKEVE 4ceb A 1.75 BS01 ZSV B 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ceb A 1.75 BS02 ZSV B 2 Q95 E96 A98 Y99 Q39 E40 A42 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ceb B 1.75 BS01 ZSV B 1 Q95 E96 A98 Y99 Q39 E40 A42 Y43 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1080uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ceb B 1.75 BS02 ZSV B 2 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=1080uM remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4cfe C 3.023 BS02 992 C 1 K29 K31 I46 N48 D88 K20 K22 I37 N39 D79 D139 K141 E143 N144 D157 S176 D130 K132 E134 N135 D148 S167 2.7.11.1,2.7.11.31 0003682,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005524,0005634,0005654,0005737,0005794,0005829,0006325,0006338,0006468,0006633,0006695,0006914,0007165,0008610,0010468,0010494,0010508,0010629,0014850,0016055,0016239,0016241,0016607,0030424,0030425,0031588,0031669,0032007,0034599,0035175,0035402,0035403,0035979,0042149,0042593,0042752,0043025,0043066,0044022,0044023,0044024,0044025,0045821,0046872,0047322,0048511,0055089,0062028,0070507,0071277,0071333,0071380,0071466,0072354,0072371,0072518,0097009,0106310,0140823,0140855,0140857,1903829,1903944,1904262,1904428,1905691,1990044,1990244,2000758 remove_due_to_license_issue P54646 24352254 1553 RVKIGHYVLGDTLGVGTFGKVKIGEHQLTGHKVAVKILNRQKIRSLDVVGKIKREIQNLKLFRHPHIIKLYQVISTPTDFFMVMEYVSGGELFDYICKHGRVEEMEARRLFQQILSAVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSCGVILYALLCGTLPFDDEHVPTLFKKIRGGVFYIPEYLNRSVATLLMHMLQVDPLKRATIKDIREHEWFKQDLPSYLFPEDPSYDIIDNRRIMNQASEFYLASSPLKPHPERMPPLAVKKAKWHLGIRSQSKPYDIMAEVYRAMKQLDFEWKVVNAYHLRVRRKNPVTGNYVKMSLQLYLVDNRSYLLDFKSIDLGSHTMDFFEMCASLITTLA 4cfe D 3.023 BS01 992 C 1 R83 R107 S108 N111 V113 R6 R30 S31 N34 V36 ? 0005515,0005634,0005654,0005737,0005829,0006633,0007165,0019901,0031588,0031669,0032991,0035878,0120162 remove_due_to_license_issue EC50=2.0nM Q9Y478 24352254 1553 RPTVFRWTGGGKEVYLSGSFNNWSKLPLTRSHNNFVAILDLPEGEHQYKFFVDGQWTHDPSEPIVTSQLGTVNNIIQVKKTDFEVFDALMVDSQEPYVCPPILPPHLLQVILNKDTGISCDPALLPEPNHVMLNHLYALSIKDGVMVLSATHRYKKKYVTTLLYKPI 4cff C 3.924 BS02 C1V C 1 G19 K29 K31 I46 D88 G10 K20 K22 I37 D79 D139 K141 E143 N144 D157 S176 D130 K132 E134 N135 D148 S167 2.7.11.1,2.7.11.31 0003682,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005524,0005634,0005654,0005737,0005794,0005829,0006325,0006338,0006468,0006633,0006695,0006914,0007165,0008610,0010468,0010494,0010508,0010629,0014850,0016055,0016239,0016241,0016607,0030424,0030425,0031588,0031669,0032007,0034599,0035175,0035402,0035403,0035979,0042149,0042593,0042752,0043025,0043066,0044022,0044023,0044024,0044025,0045821,0046872,0047322,0048511,0055089,0062028,0070507,0071277,0071333,0071380,0071466,0072354,0072371,0072518,0097009,0106310,0140823,0140855,0140857,1903829,1903944,1904262,1904428,1905691,1990044,1990244,2000758 remove_due_to_license_issue P54646 24352254 1553 RVKIGHYVLGDTLGVGTFGKVKIGEHQLTGHKVAVKILNRQKIRSLDVVGKIKREIQNLKLFRHPHIIKLYQVISTPTDFFMVMEYVSGGELFDYICKHGRVEEMEARRLFQQILSAVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSCGVILYALLCGTLPFDDEHVPTLFKKIRGGVFYIPEYLNRSVATLLMHMLQVDPLKRATIKDIREHEWFKQDLPSYLFPEDPSYDANVIDDEAVKEVAYHLIIDNRRIMNQASEFYLASSPLKPHPERMPPLIADAVKKAKWHLGIRSQSKPYDIMAEVYRAMKQLDFEWKVVNAYHLRVRRKNPVTGNYVKMSLQLYLVDNRSYLLDFKSIDLGSHTMDFFEMCASLITTLA 4cff D 3.924 BS01 C1V C 1 S108 V113 S31 V36 ? 0005515,0005634,0005654,0005737,0005829,0006633,0007165,0019901,0031588,0031669,0032991,0035878,0120162 remove_due_to_license_issue Kd=487nM, EC50=390nM Q9Y478 24352254 1553 RPTVFRWTGGGKEVYLSGSFNNWSKLPLTRSHNNFVAILDLPEGEHQYKFFVDGQWTHDPSEPIVTSQLGTVNNIIQVKKTDFEVFDALMVDSQKCQEPYVCKPPPILPPHLLQVILNKDTGISCDPALLPEPNHVMLNHLYALSIKDGVMVLSATHRYKKKYVTTLLYKPI 4cfl A 1.32 BS01 8DQ A 1 P82 V87 L92 L94 N140 I146 P41 V46 L51 L53 N99 I105 ? Kd=1.33uM remove_due_to_license_issue IC50=9050nM O60885 24533473 1169 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4cfm A 2.85 BS01 4QE A 1 I10 A31 E81 L83 H84 L134 D145 I11 A32 E82 L84 H85 L135 D146 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=18200nM P24941 24304238 1297 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 4cft A 1.79 BS03 M48 A 1 V338 W358 E363 V261 W281 E286 C186 R189 W358 E363 C109 R112 W281 E286 1.14.13.39 0004517,0006809 Ki=11.16uM remove_due_to_license_issue Ki=11160nM P29473 24472039 801 GPKFPRVKNWELGSITYDTLCAQSQQDGPCTPRRCLGSLVLPRPAEQLLSQARDFINQYYSSIKRSGSQAHEERLQEVEAEVASTGTYHLRESELVFGAKQAWRNAPRCVGRIQWGKLQVFDARDCSSAQEMFTYICNHIKYATNRGNLRSAITVFPQRAPGRGDFRIWNSQLVRYAGYRQQDGSVRGDPANVEITELCIQHGWTPGNGRFDVLPLLLQAPDEAPELFVLPPELVLEVPLEHPTLEWFAALGLRWYALPAVSNMLLEIGGLEFSAAPFSGWYMSTEIGTRNLCDPHRYNILEDVAVCMDLDTRTTSSLWKDKAAVEINLAVLHSFQLAKVTIVDHHAATVSFMKHLDNEQKARGGCPADWAWIVPPISGSLTPVFHQEMVNYILSPAFRYQPDPW 4cft B 1.79 BS05 M48 B 1 V338 W358 E363 Y477 V259 W279 E284 Y398 C186 R189 W358 E363 C107 R110 W279 E284 1.14.13.39 0004517,0006809 Ki=11.16uM remove_due_to_license_issue Ki=11160nM P29473 24472039 801 KFPRVKNWELGSITYDTLCAQSQQDGPCTPRRCLGSLVLPRPAEQLLSQARDFINQYYSSIKRSGSQAHEERLQEVEAEVASTGTYHLRESELVFGAKQAWRNAPRCVGRIQWGKLQVFDARDCSSAQEMFTYICNHIKYATNRGNLRSAITVFPQRAPGRGDFRIWNSQLVRYAGYRQQDGSVRGDPANVEITELCIQHGWTPGNGRFDVLPLLLQAPDEAPELFVLPPELVLEVPLEHPTLEWFAALGLRWYALPAVSNMLLEIGGLEFSAAPFSGWYMSTEIGTRNLCDPHRYNILEDVAVCMDLDTRTTSSLWKDKAAVEINLAVLHSFQLAKVTIVDHHAATVSFMKHLDNEQKARGGCPADWAWIVPPISGSLTPVFHQEMVNYILSPAFRYQPDPW 4cfu A 2.2 BS01 2WC A 1 I10 A31 E81 F82 L83 H84 D86 K89 N132 L134 I14 A35 E83 F84 L85 H86 D88 K91 N134 L136 D127 K129 Q131 N132 D145 T158 T165 D129 K131 Q133 N134 D147 T160 T167 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 24304238 1299 PPGSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4cfv C 2.0 BS01 75X C 1 I10 E12 A31 E81 L83 H84 Q85 D86 K89 N132 L134 I11 E13 A30 E80 L82 H83 Q84 D85 K88 N131 L133 D127 K129 Q131 N132 D145 T158 T165 D126 K128 Q130 N131 D144 T157 T164 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=23.5uM remove_due_to_license_issue P24941 24304238 1297 SMENFQKVEKIGEYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 4cfw C 2.45 BS01 SQ9 C 1 I10 A31 E81 L83 Q85 D86 K89 L134 I12 A33 E83 L85 Q87 D88 K91 L136 D127 K129 Q131 N132 D145 T158 T165 D129 K131 Q133 N134 D147 T160 T167 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=0.51uM remove_due_to_license_issue P24941 24304238 1297 GSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 4cfx C 3.5 BS01 G6T C 1 I10 A31 L83 H84 K89 L134 D145 I11 A32 L84 H85 K90 L135 D146 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 24304238 1299 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4cg8 A 1.75 BS01 G8S A 1 T252 Y256 D306 Y333 Y354 L419 W420 W423 I433 Y440 T148 Y152 D202 Y229 Y250 L315 W316 W319 I329 Y336 2.7.1.32,2.7.1.82 Kd=0.11uM remove_due_to_license_issue P35790 24387243 1458 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 4cg9 A 1.83 BS01 GQG A 1 D306 Y333 Y354 W420 W423 F435 Y440 D202 Y229 Y250 W316 W319 F331 Y336 2.7.1.32,2.7.1.82 remove_due_to_license_issue P35790 24387243 0 EQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 4cga A 1.74 BS01 QLW A 1 D306 Q308 Y333 Y354 W420 W423 F435 Y440 D203 Q205 Y230 Y251 W317 W320 F332 Y337 2.7.1.32,2.7.1.82 remove_due_to_license_issue P35790 24387243 0 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 4cgi A 2.07 BS01 NZL A 1 D167 Q168 E170 H171 T174 M178 D111 Q112 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=752uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 4cgi A 2.07 BS02 NZL B 1 A129 W132 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=752uM remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQT 4cgi B 2.07 BS01 NZL A 1 A129 W132 A73 W76 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=752uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4cgi B 2.07 BS02 NZL B 1 D167 Q168 E170 H171 T174 M178 D111 Q112 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=752uM remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4cgj A 2.15 BS01 NZL A 1 D167 Q168 E170 H171 T174 M178 D111 Q112 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4cgj A 2.15 BS02 NZL B 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4cgj B 2.15 BS01 NZL A 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4cgj B 2.15 BS02 NZL B 1 Q168 E170 H171 T174 M178 Q112 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDIQ 4ch1 A -1.00 BS01 dna B 0 K36 F38 L42 Y44 V65 I67 G77 Y78 F80 R103 N106 A110 G113 A114 K115 K12 F14 L18 Y20 V41 I43 G53 Y54 F56 R79 N82 A86 G89 A90 K91 ? 0003676,0003723 remove_due_to_license_issue H2L051 25183497 1 ~ 7 GAMGSRDTMFTKIFVGGLPYHTSDKTLHEYFEQFGDIEEAVVITDRNTQKSRGYGFVTMKDRASAERACKDPNPIIDGRKANVNLAYLGAKPRTNVQ 4chu A 2.489 BS01 dna C 0 R2 S5 K6 Y9 S38 S40 Y41 Q44 R59 G60 P61 R3 S6 K7 Y10 S39 S41 Y42 Q45 R60 G61 P62 ? 0003677,0003690,0003700,0005506,0005829,0006355,0046872,0051537 remove_due_to_license_issue C3SZN7 24847070 1 ~ 27 MGRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDESVDKSLTHALWRDLSDRLTGFLNNITLGELVNNQEVLDVS 4chu A 2.489 BS02 dna D 0 P27 E43 R50 S57 R59 P61 G64 Y65 P28 E44 R51 S58 R60 P62 G65 Y66 ? 0003677,0003690,0003700,0005506,0005829,0006355,0046872,0051537 remove_due_to_license_issue C3SZN7 24847070 1 ~ 27 MGRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDESVDKSLTHALWRDLSDRLTGFLNNITLGELVNNQEVLDVS 4chu B 2.489 BS01 dna C 0 P27 L28 E43 R50 S57 R59 G60 G64 Y65 P27 L28 E43 R50 S57 R59 G60 G64 Y65 ? 0003677,0003690,0003700,0005506,0005829,0006355,0046872,0051537 remove_due_to_license_issue C3SZN7 24847070 1 ~ 27 GRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDQGKGGSQGGDKSLTHALWRDLSDRLTGFLNNITLGELVNNQEV 4chu B 2.489 BS02 dna D 0 S5 K6 Y9 S38 S40 Y41 Q44 R59 G60 P61 S5 K6 Y9 S38 S40 Y41 Q44 R59 G60 P61 ? 0003677,0003690,0003700,0005506,0005829,0006355,0046872,0051537 remove_due_to_license_issue C3SZN7 24847070 1 ~ 27 GRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDQGKGGSQGGDKSLTHALWRDLSDRLTGFLNNITLGELVNNQEV 4ci1 B 2.98 BS02 EF2 B 1 N353 P354 H355 H380 S381 W382 W388 W402 F404 N296 P297 H298 H323 S324 W325 W331 W345 F347 ? 0005634,0005737,0016567,0031464,0043161,0046872 remove_due_to_license_issue P0CF65 25043012 1429 MINFDTSLPTSHMYLGSDMEEFHGRTLHDDDSCQVIPVLPHVMVMLIPGQTLPLQLFHPQEVSMVRNLIQKDRTFAVLAYSNVREREAHFGTTAEIYAYREEQEYGIETVKVKAIGRQRFKVLEIRTQSDGIQQAKVQILPERVLPSTMSAVQLQSLSRRHIRAFRQWWQKYQKRKFHCASLTSWPPWLYSLYDAETLMERVKRQLHEWDENLKDESLPTNPIDFSYRVAACLPIDDALRIQLLKIGSAIQRLRCELDIMNKCTSLCCKQCQDTEITTKNEIFSLSLCGPMAAYVNPHGYIHETLTVYKACNLNLSGRPSTEHSWFPGYAWTIAQCRICGNHMGWKFTATKKDMSPQKFWGLTRSALLPR 4ci2 B 2.95 BS02 LVY B 1 N353 P354 H355 H380 S381 W382 W388 W402 F404 N296 P297 H298 H323 S324 W325 W331 W345 F347 ? 0005634,0005737,0016567,0031464,0043161,0046872 remove_due_to_license_issue P0CF65 25043012 1429 MINFDTSLPTSHMYLGSDMEEFHGRTLHDDDSCQVIPVLPHVMVMLIPGQTLPLQLFHPQEVSMVRNLIQKDRTFAVLAYSNVREREAHFGTTAEIYAYREEQEYGIETVKVKAIGRQRFKVLEIRTQSDGIQQAKVQILPERVLPSTMSAVQLQSLSRRHIRAFRQWWQKYQKRKFHCASLTSWPPWLYSLYDAETLMERVKRQLHEWDENLKDESLPTNPIDFSYRVAACLPIDDALRIQLLKIGSAIQRLRCELDIMNKCTSLCCKQCQDTEITTKNEIFSLSLCGPMAAYVNPHGYIHETLTVYKACNLNLSGRPSTEHSWFPGYAWTIAQCRICGNHMGWKFTATKKDMSPQKFWGLTRSALLPR 4ci3 B 3.5 BS02 Y70 B 1 N353 P354 H355 H380 S381 W382 W388 W402 F404 N296 P297 H298 H323 S324 W325 W331 W345 F347 ? 0005634,0005737,0016567,0031464,0043161,0046872 remove_due_to_license_issue P0CF65 25043012 1429 MINFDTSLPTSHMYLGSDMEEFHGRTLHDDDSCQVIPVLPHVMVMLIPGQTLPLQLFHPQEVSMVRNLIQKDRTFAVLAYSNVREREAHFGTTAEIYAYREEQEYGIETVKVKAIGRQRFKVLEIRTQSDGIQQAKVQILPERVLPSTMSAVQLQSLSRRHIRAFRQWWQKYQKRKFHCASLTSWPPWLYSLYDAETLMERVKRQLHEWDENLKDESLPTNPIDFSYRVAACLPIDDALRIQLLKIGSAIQRLRCELDIMNKCTSLCCKQCQDTEITTKNEIFSLSLCGPMAAYVNPHGYIHETLTVYKACNLNLSGRPSTEHSWFPGYAWTIAQCRICGNHMGWKFTATKKDMSPQKFWGLTRSALLPR 4cig A 1.7 BS01 X0P A 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=214uM remove_due_to_license_issue P12497 24532034 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDI 4cig A 1.7 BS02 X0P B 1 Q95 T125 A128 Q39 T69 A72 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=214uM remove_due_to_license_issue P12497 24532034 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDI 4cig B 1.7 BS01 X0P A 1 Q95 A128 Q39 A72 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=214uM remove_due_to_license_issue P12497 24532034 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDI 4cig B 1.7 BS02 X0P B 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=214uM remove_due_to_license_issue P12497 24532034 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDI 4cik A 1.78 BS01 XO3 A 1 R35 D55 D57 W62 Y64 R71 Y72 R36 D56 D58 W63 Y65 R72 Y73 3.4.21.7 remove_due_to_license_issue IC50=950nM P00747 24900876 1081 SECKTGNGKNYRGTMSKTKNGITCQKWSSTSPHRPRFSPATHPSEGLEENYCRNPDNDPQGPWCYTTDPEKRYDYCDILEC 4cio A -1.00 BS01 rna B 0 K36 F38 L42 P43 Y44 V65 I67 Y78 F80 R103 N106 A110 G113 K12 F14 L18 P19 Y20 V41 I43 Y54 F56 R79 N82 A86 G89 ? 0003676,0003723 remove_due_to_license_issue O45189 25183497 1 ~ 7 GAMGSRDTMFTKIFVGGLPYHTSDKTLHEYFEQFGDIEEAVVITDRNTQKSRGYGFVTMKDRASAERACKDPNPIIDGRKANVNLAYLGAKPRTNVQ 4civ A 2.9 BS01 48P A 1 R19 G77 G78 H101 I102 S103 R112 R17 G70 G71 H94 I95 S96 R105 P11 N12 R19 N75 G78 E99 H101 R108 P9 N10 R17 N68 G71 E92 H94 R101 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 24689821 201 LIVNVINGPNLGRLGRRGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEHV 4ciw A 2.2 BS01 XH2 A 1 Y24 N75 G77 G78 H81 H101 I102 S103 R112 Y22 N73 G75 G76 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=15uM remove_due_to_license_issue P9WPX7 24689821 1148 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4cix A 2.9 BS01 W4N A 1 L16 R18 N75 G77 G78 H101 I102 S103 R112 L14 R16 N66 G68 G69 H92 I93 S94 R103 P11 N12 N75 G78 E99 H101 R108 P9 N10 N66 G69 E90 H92 R99 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 24689821 1143 LIVNVINGPNLGRLGRGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAE 4ciy A 2.1 BS01 NDY A 1 N12 Y24 N75 G77 G78 H81 H101 I102 S103 R112 N10 Y17 N68 G70 G71 H74 H94 I95 S96 R105 P11 N12 Y24 N75 G78 E99 H101 R108 P9 N10 Y17 N68 G71 E92 H94 R101 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 Ki=27uM remove_due_to_license_issue P9WPX7 24689821 1144 LIVNVINGPNLGRLGRYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4ciz A 3.403 BS01 RET A 1 F204 M223 V224 V254 F182 M201 V202 V232 ? 0005502,0005515,0005654,0005737,0005813,0005829,0006776,0007601,0019841,0044297,1902936 remove_due_to_license_issue P12271 24328211 1307 EQLTTKDHGPVFGPCSQLPRHTLQKAKDELNEREETREEAVRELQEMVQAQAASGEELAVAVAERVQEKDSGFFLRFIRARKFNVGRAYELLRGYVNFRLQYPELFDSLSPEAVRCTIEAGYPGVLSSRDKYGRVVMLFNIENWQSQEITFDEILQAYCFILEKLLENEETQINGFCIIENFKGFTMQQAASLRTSDLRKMVDMLQDSFPARFKAIHFIHQPWYFTTTYNVVKPFLKSKLLERVFVHGDDLSGFYQEIDENILPSDFGGTLPKYDGKAVAEQLF 4cj4 A 1.8 BS01 S3G A 1 A169 E170 H171 T174 M178 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=432uM remove_due_to_license_issue P12497 24532034 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cj4 A 1.8 BS02 S3G B 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=432uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cj4 B 1.8 BS01 S3G A 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=432uM remove_due_to_license_issue P12497 24532034 1217 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cj4 B 1.8 BS02 S3G B 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=432uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cja A 2.651 BS01 dna B 0 Y29 D61 C62 H65 I94 G95 Q98 Q164 T193 G194 Q197 G227 Q230 I259 I292 Q296 N325 G326 Q329 Q362 I391 Q395 I424 G425 Q428 T457 G458 Q461 Q494 S523 G524 Q527 D556 G557 Q560 N589 G590 Q593 G622 G655 Q659 S688 G689 Q692 Q724 R753 Y15 D47 C48 H51 I80 G81 Q84 Q150 T179 G180 Q183 G213 Q216 I245 I278 Q282 N311 G312 Q315 Q348 I377 Q381 I410 G411 Q414 T443 G444 Q447 Q480 S509 G510 Q513 D542 G543 Q546 N575 G576 Q579 G608 G641 Q645 S674 G675 Q678 Q710 R739 remove_due_to_license_issue 25004980 -1 ~ 21 LNLSPLERSKIEKQYGGATTLAFISNKQQELAQILSRADILKIASYDCAAHALQAVLDCGPMLGKRGFSQSDIVKIAGNIGGAQALQAVLDLESMLGKRGFSRDDIAKMAGNIGGAQTLQAVLDLESAFRERGFSQADIVKIAGNNGGAQALYSVLDVEPTLGKRGFSRADIVKIAGNTGGAQALHTVLDLEPALGKRGFSRIDIVKIAANNGGAQALHAVLDLGPTLRECGFSQATIAKIAGNIGGAQALQMVLDLGPALGKRGFSQATIAKIAGNIGGAQALQTVLDLEPALCERGFSQATIAKMAGNNGGAQALQTVLDLEPALRKRDFRQADIIKIAGNDGGAQALQAVIEHGPTLRQHGFNLADIVKMAGNIGGAQALQAVLDLKPVLDEHGFSQPDIVKMAGNIGGAQALQAVLSLGPALRERGFSQPDIVKIAGNTGGAQALQAVLDLELTLVEHGFSQPDIVRITGNRGGAQALQAVLALELTLRERGFSQPDIVKIAGNSGGAQALQAVLDLELTFRERGFSQADIVKIAGNDGGTQALHAVLDLERMLGDRGFSRADIVNVAGNNGGAQALKAVLEHEATLNERGFSRADIVKIAGNGGGAQALKAVLEHEATLDERGFSRADIVRIAGNGGGAQALKAVLEHGPTLNERGFNLTDIVEMAANSGGAQALKAVLEHGPTLRQRGLSLIDIVEIASNGGAQALKAVLKYGPVLMQAGRSNEEIVHVAARRGGAGRIRKMVAPLL 4cja A 2.651 BS02 dna C 0 K155 K353 R490 K141 K339 R476 remove_due_to_license_issue 25004980 -1 ~ 21 LNLSPLERSKIEKQYGGATTLAFISNKQQELAQILSRADILKIASYDCAAHALQAVLDCGPMLGKRGFSQSDIVKIAGNIGGAQALQAVLDLESMLGKRGFSRDDIAKMAGNIGGAQTLQAVLDLESAFRERGFSQADIVKIAGNNGGAQALYSVLDVEPTLGKRGFSRADIVKIAGNTGGAQALHTVLDLEPALGKRGFSRIDIVKIAANNGGAQALHAVLDLGPTLRECGFSQATIAKIAGNIGGAQALQMVLDLGPALGKRGFSQATIAKIAGNIGGAQALQTVLDLEPALCERGFSQATIAKMAGNNGGAQALQTVLDLEPALRKRDFRQADIIKIAGNDGGAQALQAVIEHGPTLRQHGFNLADIVKMAGNIGGAQALQAVLDLKPVLDEHGFSQPDIVKMAGNIGGAQALQAVLSLGPALRERGFSQPDIVKIAGNTGGAQALQAVLDLELTLVEHGFSQPDIVRITGNRGGAQALQAVLALELTLRERGFSQPDIVKIAGNSGGAQALQAVLDLELTFRERGFSQADIVKIAGNDGGTQALHAVLDLERMLGDRGFSRADIVNVAGNNGGAQALKAVLEHEATLNERGFSRADIVKIAGNGGGAQALKAVLEHEATLDERGFSRADIVRIAGNGGGAQALKAVLEHGPTLNERGFNLTDIVEMAANSGGAQALKAVLEHGPTLRQRGLSLIDIVEIASNGGAQALKAVLKYGPVLMQAGRSNEEIVHVAARRGGAGRIRKMVAPLL 4cjn B 1.947 BS01 QNZ B 1 N104 Y105 N146 K273 E294 Y297 K316 N78 Y79 N120 K247 E268 Y271 K290 3.4.16.4 0005886,0008658,0009002,0016020,0046677,0071555,0071972 Kd=17.5uM remove_due_to_license_issue A0A0J9X1X5 25629446 1673 DKEINNTIDAIEDKNFKQVYKDSSYISKSDNGEVEMTERPIKIYNSLGVKDINIQDRKIKKVSKNKKRVDAQYKIKTNYGNIDRNVQFNFVKEDGMWKLDWDHSVIIPGMQKDQSIHIENLKSERGKILDRNNVELANTGTAYEIGIVPKNVSKKDYKAIAKELSISEDYIKQQMDQNWVQDDTFVPLKTVKKMDEYLSDFAKKFHLTTNETESRNYPLGKATSHLLGYVGPINSEELKQKEYKGYKDDAVIGKKGLEKLYDKKLQHEDGYRVTIVDDNSNTIAHTLIEKKKKDGKDIQLTIDAKVQKSIYNNMKNDYGSGTAIHPQTGELLALVSTPSYDVYPFMYGMSNEEYNKLTEDKKEPLLNKFQITTSPGSTQKILTAMIGLNNKTLDDKTSYKIDGKGWQKDKSWGGYNVTRYEVVNGNIDLKQAIESSDNIFFARVALELGSKKFEKGMKKLGVGEDIPSDYPFYNAQISNKNLDNEILLADSGYGQGEILINPVQILSIYSALENNGNINAPHLLKDTKNKVWKKNIISKENINLLTDGMQQVVNKTHKEDIYRSYANLIGKSGTAELKMKQGETGRQIGWFISYDKDNPNMMMAINVKDVQDKGMASYNAKISGKVYDELYENGNKKYDIDE 4cjp A 2.0 BS01 4D2 A 1 Q168 E170 H171 T174 M178 Q112 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjp B 2.0 BS01 4D2 A 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjp B 2.0 BS02 4D2 B 1 Q168 E170 H171 T174 M178 Q112 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjq A 1.7 BS01 VXO A 1 D167 A169 E170 H171 T174 M178 D111 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=256uM remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjq B 1.7 BS01 VXO A 1 Q95 A129 Q39 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=256uM remove_due_to_license_issue P12497 24532034 1214 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjq B 1.7 BS02 VXO B 1 D167 A169 E170 H171 T174 M178 D111 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=256uM remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjr A 1.8 BS01 FYM A 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=793uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjr A 1.8 BS02 FYM B 1 Q95 A128 A129 Q39 A72 A73 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=793uM remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjr B 1.8 BS01 FYM A 1 Q95 A128 Q39 A72 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=793uM remove_due_to_license_issue P12497 24532034 1215 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4cjr B 1.8 BS02 FYM B 1 Q168 A169 E170 H171 T174 Q112 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=793uM remove_due_to_license_issue P12497 24532034 1216 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDIQ 4ck3 A 1.79 BS01 K1T A 1 A169 E170 H171 T174 M178 A114 E115 H116 T119 M123 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=268uM remove_due_to_license_issue P12497 24532034 1213 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDI 4ck3 A 1.79 BS02 K1T B 1 Q95 A129 Q40 A74 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=268uM remove_due_to_license_issue P12497 24532034 1216 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDI 4ck3 B 1.79 BS01 K1T A 1 Q95 A129 Q40 A74 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=268uM remove_due_to_license_issue P12497 24532034 1213 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDI 4ck3 B 1.79 BS02 K1T B 1 A169 E170 H171 T174 M178 A114 E115 H116 T119 M123 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=268uM remove_due_to_license_issue P12497 24532034 1216 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIPYNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGYSAGERIVDIIATDI 4cki A 2.116 BS01 ADN A 1 L730 G731 E732 V738 A756 E805 A807 S811 L881 L31 G32 E33 V39 A57 E106 A108 S112 L163 D850 D874 A876 R878 N879 D892 D132 D156 A158 R160 N161 D174 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P07949 24560924 2022 GPLSLSVDAFKILEDPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVDERALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWTAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKRR 4ckj A 1.65 BS01 ADN A 1 G731 V738 A756 Y806 A807 L881 G32 V39 A57 Y107 A108 L161 D850 D874 A876 R878 N879 D892 D130 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P07949 24560924 2014 GPLSLSVDAFKILEDPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVRALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKRR 4ckr A 2.2 BS01 DI1 A 1 A653 K655 E672 M676 T701 Y703 M704 V763 H764 R765 L773 I782 A783 D784 F785 A54 K56 E73 M77 T102 Y104 M105 V149 H150 R151 L159 I168 A169 D170 F171 D766 R770 N771 D784 A793 D152 R156 N157 D170 A179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=105nM remove_due_to_license_issue IC50=105nM, EC50=86nM Q08345 23899692 1000 MPRVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSLDFPLNVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNTV 4cku A 1.85 BS01 P2F A 1 I32 D34 G36 Y77 V78 S79 F111 I123 Y192 D214 G216 T217 S218 I290 I300 I30 D32 G34 Y75 V76 S77 F109 I121 Y190 D212 G214 T215 S216 I284 I294 D34 S37 N39 W41 Y77 D214 T217 D32 S35 N37 W39 Y75 D212 T215 3.4.23.39 0004190,0006508 ic50=0.15uM remove_due_to_license_issue IC50=150nM P46925 24900843 400 NDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 4cku B 1.85 BS01 P2F B 1 I14 I32 D34 G36 Y77 V78 F111 I123 Y192 D214 G216 T217 S218 F294 I300 I12 I30 D32 G34 Y75 V76 F109 I121 Y190 D212 G214 T215 S216 F292 I298 D34 S37 N39 W41 Y77 D214 T217 D32 S35 N37 W39 Y75 D212 T215 3.4.23.39 0004190,0006508 ic50=0.15uM remove_due_to_license_issue IC50=150nM P46925 24900843 400 NDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 4cku F 1.85 BS01 P2F F 1 M15 I32 D34 G36 V78 S79 F111 I123 Y192 D214 G216 T217 S218 I290 L292 M15 I32 D34 G36 V78 S79 F111 I123 Y192 D214 G216 T217 S218 I290 L292 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 ic50=0.15uM remove_due_to_license_issue IC50=150nM P46925 24900843 400 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 4cl6 A 2.41 BS01 7SB A 1 H70 F71 G115 H69 F70 G114 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 Ka=247000M^-1 remove_due_to_license_issue O33877 26562505 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4cl6 A 2.41 BS02 7SB B 1 Q27 L28 Q88 G91 F92 G103 R104 A105 Q26 L27 Q87 G90 F91 G102 R103 A104 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 Ka=247000M^-1 remove_due_to_license_issue O33877 26562505 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4cl6 B 2.41 BS01 7SB A 1 Q27 L28 Q88 G91 F92 G103 R104 A105 Q26 L27 Q87 G90 F91 G102 R103 A104 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 Ka=247000M^-1 remove_due_to_license_issue O33877 26562505 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4cl6 B 2.41 BS02 7SB B 1 H70 F71 H69 F70 H70 V76 G79 C80 D84 H69 V75 G78 C79 D83 4.2.1.59,5.3.3.14 0005737,0006633,0006636,0016829,0016853,0019171,0034017 Ka=247000M^-1 remove_due_to_license_issue O33877 26562505 501 TKQHAFTREDLLRCSRGELFGPGNAQLPAPNMLMIDRIVHISDVGGKYGKGELVAELDINPDLWFFACHFEGDPVMPGCLGLDAMWQLVGFYLGWQGNPGRGRALGSGEVKFFGQVLPTAKKVTYNIHIKRTINRSLVLAIADGTVSVDGREIYSAEGLRVGLFTSTDSF 4cl9 A 1.4 BS01 IES A 1 W81 P82 Q84 Q85 K91 L92 N140 I146 M149 W40 P41 Q43 Q44 K50 L51 N99 I105 M108 ? remove_due_to_license_issue O60885 1170 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4clb A 1.6 BS01 83T A 1 W81 L92 N140 I146 W40 L51 N99 I105 ? remove_due_to_license_issue O60885 1170 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4cli A 2.05 BS01 5P8 A 1 L1122 A1148 L1196 E1197 M1199 N1254 L1256 G1269 D1270 I1399 E1400 L30 A48 L96 E97 M99 N154 L156 G169 D170 I293 E294 D1249 A1251 R1253 N1254 D1270 D149 A151 R153 N154 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki<0.07nM remove_due_to_license_issue Q9UM73 24819116 2401 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 4clj A 1.66 BS01 5P8 A 1 L1122 A1148 M1196 E1197 M1199 G1202 N1254 L1256 G1269 D1270 Y1401 L29 A48 M96 E97 M99 G102 N154 L156 G169 D170 Y295 D1249 A1251 R1253 N1254 D1270 L1291 D149 A151 R153 N154 D170 L185 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.7nM remove_due_to_license_issue Q9UM73 24819116 2402 PNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILMELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 4clp A 1.9 BS01 CMP A 1 R199 I202 E203 I204 E205 S206 R192 I195 E196 I197 E198 S199 4.6.1.1 0009190,0035556 Kd=54.2mM remove_due_to_license_issue Q96PN6 24567411 1473 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFELDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTE 4clp A 1.9 BS02 CMP A 2 A97 G98 F336 F338 L345 V411 N412 R416 A97 G98 F329 F331 L338 V404 N405 R409 4.6.1.1 0009190,0035556 Kd=54.2mM remove_due_to_license_issue Q96PN6 24567411 1474 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFELDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTE 4clz A 1.9 BS01 4DS A 1 F8 D10 V14 R15 A252 C253 Q276 I277 N279 Q283 T399 F8 D10 V14 R15 A242 C243 Q266 I267 N269 Q273 T389 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24567411 1479 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4clz A 1.9 BS02 4DS A 2 F45 K95 A97 L101 L102 R176 F336 F338 D339 R416 M419 Y420 F45 K95 A97 L101 L102 R166 F326 F328 D329 R406 M409 Y410 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24567411 1480 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4clz A 1.9 BS03 4DS A 3 F51 M54 K57 F58 M62 Y63 H78 F51 M54 K57 F58 M62 Y63 H78 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24567411 1481 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4cmo A 2.05 BS01 YPW A 1 V1130 A1148 E1197 M1199 G1202 R1214 N1254 L1256 G1269 D1270 Y1401 V38 A48 E97 M99 G102 R114 N154 L156 G169 D170 Y295 D1249 A1251 R1253 N1254 D1270 D149 A151 R153 N154 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.85nM remove_due_to_license_issue Ki=0.850000nM, IC50=16nM Q9UM73 24819116 2402 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 4cmt A 1.73 BS01 GWH A 1 R1120 L1122 G1123 V1130 A1148 L1196 E1197 M1199 G1202 N1254 L1256 G1269 D1270 E1400 R28 L30 G31 V35 A45 L93 E94 M96 G99 N148 L150 G163 D164 E284 D1249 A1251 R1253 N1254 D1270 D143 A145 R147 N148 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki<0.2nM remove_due_to_license_issue Q9UM73 24819116 2401 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 4cmu A 1.8 BS01 IV7 A 1 L1122 A1148 L1196 E1197 M1199 G1202 N1254 L1256 G1269 D1270 I1399 E1400 L30 A48 L96 E97 M99 G102 N154 L156 G169 D170 I293 E294 D1249 A1251 R1253 N1254 D1270 D149 A151 R153 N154 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki<0.2nM remove_due_to_license_issue IC50=0.700000nM, Ki=0.290000nM Q9UM73 24819116 2401 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 4cn2 C 2.069 BS01 dna A 0 K145 H146 Y147 K156 R164 Q206 E208 R209 K17 H18 Y19 K28 R36 Q78 E80 R81 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 MFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cn2 C 2.069 BS02 dna B 0 E153 G154 R161 R184 N185 Q188 R191 E25 G26 R33 R56 N57 Q60 R63 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 MFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cn2 D 2.069 BS01 dna A 0 K145 H146 Y147 K160 R164 Q206 E208 R209 R211 G212 K14 H15 Y16 K29 R33 Q75 E77 R78 R80 G81 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQRG 4cn2 D 2.069 BS02 dna B 0 E153 G154 F158 R161 R184 N185 Q188 R191 E22 G23 F27 R30 R53 N54 Q57 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQRG 4cn3 A 2.35 BS01 dna E 0 Y147 K156 R164 Q206 E208 Y17 K26 R34 Q76 E78 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEE 4cn3 A 2.35 BS02 dna F 0 E153 G154 F158 R161 R184 N185 Q188 R191 E23 G24 F28 R31 R54 N55 Q58 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEE 4cn3 B 2.35 BS01 dna G 0 H146 Y147 K160 R164 A204 Q206 H14 Y15 K28 R32 A72 Q74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 HICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEE 4cn3 B 2.35 BS02 dna H 0 E153 G154 F158 R161 R184 N185 R191 E21 G22 F26 R29 R52 N53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 HICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEE 4cn3 C 2.35 BS01 dna G 0 Y147 K156 R164 Q206 E208 R209 Y22 K31 R39 Q81 E83 R84 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 GSHMFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn3 C 2.35 BS02 dna H 0 E153 G154 R161 R184 N185 Q188 R191 R209 E28 G29 R36 R59 N60 Q63 R66 R84 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 GSHMFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn3 D 2.35 BS01 dna E 0 K145 H146 Y147 R164 Q206 E208 R209 K14 H15 Y16 R33 Q75 E77 R78 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDDKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn3 D 2.35 BS02 dna F 0 E153 G154 R161 R184 N185 Q188 R191 R209 E22 G23 R30 R53 N54 Q57 R60 R78 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDDKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn5 A 2.0 BS01 dna C 0 K145 H146 Y147 R164 Q206 E208 R209 K17 H18 Y19 R36 Q78 E80 R81 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 MFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn5 A 2.0 BS02 dna D 0 E153 G154 R161 R184 N185 Q188 R191 E25 G26 R33 R56 N57 Q60 R63 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 MFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn5 B 2.0 BS01 dna C 0 K145 H146 Y147 K156 R164 Q206 E208 R209 K14 H15 Y16 K25 R33 Q72 E74 R75 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn5 B 2.0 BS02 dna D 0 E153 G154 R161 R184 N185 Q188 R191 E22 G23 R30 R50 N51 Q54 R57 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 17 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEER 4cn7 A 2.34 BS01 dna C 0 K145 H146 Y147 K156 K160 R202 K20 H21 Y22 K31 K35 R77 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 GSHMFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREA 4cn7 A 2.34 BS02 dna D 0 E153 G154 R161 R184 N185 R191 E28 G29 R36 R59 N60 R66 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 GSHMFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREA 4cn7 B 2.34 BS01 dna C 0 K145 H146 Y147 K156 K160 R164 V205 Q206 E208 R209 K14 H15 Y16 K25 K29 R33 V74 Q75 E77 R78 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cn7 B 2.34 BS02 dna D 0 E153 G154 F158 R161 K165 R184 N185 Q188 R191 R209 E22 G23 F27 R30 K34 R53 N54 Q57 R60 R78 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cn7 B 2.34 BS03 dna H 0 Y169 Q188 Y38 Q57 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 KHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cn7 E 2.34 BS01 dna G 0 G144 K145 H146 Y147 K156 R164 V205 Q206 G14 K15 H16 Y17 K26 R34 V75 Q76 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQE 4cn7 E 2.34 BS02 dna H 0 E153 G154 R161 R184 N185 Q188 R191 E23 G24 R31 R54 N55 Q58 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQE 4cn7 F 2.34 BS01 dna G 0 K145 H146 Y147 K156 K160 R164 Q206 E208 R209 K15 H16 Y17 K26 K30 R34 Q76 E78 R79 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cn7 F 2.34 BS02 dna H 0 E153 G154 R161 R184 N185 Q188 R191 R209 E23 G24 R31 R54 N55 Q58 R61 R79 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P19793 25645674 1 ~ 16 TKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNKDCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQ 4cnh A 1.9 BS01 3U9 A 1 L1122 A1148 M1199 N1254 L1256 G1269 L29 A42 M93 N148 L150 G163 D1249 A1251 R1253 N1254 D1270 D143 A145 R147 N148 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=4nM remove_due_to_license_issue IC50=95nM, Ki=4.0nM Q9UM73 24819116 2402 PNYCFAGKTSSISDLKEVPRKNITLIRGLEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 4cp5 D 2.32 BS01 EOI D 1 K16 H59 F64 L68 R92 T98 R109 V116 K12 H55 F60 L64 R88 T94 R105 V112 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM remove_due_to_license_issue P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp5 F 2.32 BS01 EOI F 1 K16 H59 F64 R92 T98 R109 V116 N119 K12 H55 F60 R88 T94 R105 V112 N115 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM remove_due_to_license_issue P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp7 A 1.8 BS01 9MW A 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 T82 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=7.8nM remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cp7 B 1.8 BS01 9MW A 1 L123 D125 G127 A128 D129 G148 G149 F153 T182 L23 D25 G27 A28 D29 G48 G49 F53 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpq A 2.35 BS01 9MW A 1 D25 G27 D29 G48 I50 P81 T82 D25 G27 D29 G48 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpq B 2.35 BS01 9MW A 1 L123 D125 G127 A128 D129 G148 G149 F153 T182 L23 D25 G27 A28 D29 G48 G49 F53 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpr A 1.8 BS01 378 A 1 D25 G27 A28 D29 D30 G48 G49 I50 P81 T82 D25 G27 A28 D29 D30 G48 G49 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=35nM remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpr B 1.8 BS01 378 A 1 R108 D125 G127 A128 D129 G148 G149 F153 P181 T182 R8 D25 G27 A28 D29 G48 G49 F53 P81 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cps A 1.55 BS01 1T8 B 1 D25 G27 A28 D29 D30 G48 G49 P81 T82 D25 G27 A28 D29 D30 G48 G49 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cps B 1.55 BS01 1T8 B 1 L123 D125 G127 A128 D129 G148 G149 F153 L23 D25 G27 A28 D29 G48 G49 F53 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpt A 1.7 BS01 1T8 B 1 D25 G27 A28 D29 G48 G49 I50 P81 T82 D25 G27 A28 D29 G48 G49 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpt B 1.7 BS01 1T8 B 1 L123 D125 G127 A128 D129 G148 G149 F153 L23 D25 G27 A28 D29 G48 G49 F53 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=20nM remove_due_to_license_issue P03366 25054811 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpu A 1.82 BS01 V78 B 1 D25 G27 A28 D29 G48 I50 P81 D25 G27 A28 D29 G48 I50 P81 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpu B 1.82 BS01 V78 B 1 L123 D125 G127 A128 D129 G148 G149 I150 F153 P181 L23 D25 G27 A28 D29 G48 G49 I50 F53 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=29.5nM remove_due_to_license_issue P03366 25054811 1202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpw A 1.7 BS01 V78 A 1 D25 G27 A28 D29 G48 G49 I50 P81 T82 D25 G27 A28 D29 G48 G49 I50 P81 T82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpw B 1.7 BS01 V78 A 1 L123 D125 G127 A128 D129 G148 G149 F153 T182 L23 D25 G27 A28 D29 G48 G49 F53 T82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25054811 1101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 4cpy A 1.8 BS02 G39 A 1 R115 E116 D148 R149 A244 E274 R291 N293 R373 Y408 R40 E41 D73 R74 A169 E199 R216 N218 R298 Y333 D148 E275 R291 R373 Y408 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046872,0055036 Ki=491.35nM remove_due_to_license_issue U5XBU0 24795482 1470 EPEWTYPRLSCPGSTFQKALLISPHRFGETKGNSAPLIIREPFIACGPNECKHFALTHYAAQPGGYYNGTRGDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGKEWTYIGVDGPDNDALLKVKYGEAYTDTYHSYANKLLRTQESACNCIGGNCYLMITDGSASGVSECRFLKIREGRIIKEIFPTGRVKHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTDTYLDTPRPDDGSITGPCESNGDKGSGGIKGGFVHQRMESKIGRWYSRTMSKTERMGMGLYVKYDGDPWADSDALAFSGVMVSMKEPGWYSFGFEIKDKECDVPCIGIEMVHDGGKETWHSAATAIYCLMGSGQLLWDTVTGVDMAL 4cpz A 2.2 BS02 ZMR A 1 R115 E116 D148 R149 W176 E225 E274 E275 R291 N293 R373 Y408 R40 E41 D73 R74 W101 E150 E199 E200 R216 N218 R298 Y333 D148 E275 R291 R373 Y408 D73 E200 R216 R298 Y333 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046872,0055036 Ki=20.85nM remove_due_to_license_issue U5XBU0 24795482 1471 EPEWTYPRLSCPGSTFQKALLISPHRFGETKGNSAPLIIREPFIACGPNECKHFALTHYAAQPGGYYNGTRGDRNKLRHLISVKLGKIPTVENSIFHMAAWSGSACHDGKEWTYIGVDGPDNDALLKVKYGEAYTDTYHSYANKLLRTQESACNCIGGNCYLMITDGSASGVSECRFLKIREGRIIKEIFPTGRVKHTEECTCGFASNKTIECACRDNSYTAKRPFVKLNVETDTAEIRLMCTDTYLDTPRPDDGSITGPCESNGDKGSGGIKGGFVHQRMESKIGRWYSRTMSKTERMGMGLYVKYDGDPWADSDALAFSGVMVSMKEPGWYSFGFEIKDKECDVPCIGIEMVHDGGKETWHSAATAIYCLMGSGQLLWDTVTGVDMAL 4cq0 A 1.45 BS02 SXS A 1 H94 H96 H119 V121 F131 L198 T199 T200 H90 H92 H115 V117 F126 L193 T194 T195 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>50000nM, IC50=49000nM P00918 24689792 1264 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4cqe A 2.3 BS01 CQE A 1 A481 K483 L505 L514 F516 I527 T529 W531 C532 F583 G593 D594 F595 G596 A31 K33 L55 L64 F66 I77 T79 W81 C82 F133 G143 D144 F145 G146 D576 K578 N580 N581 D594 S616 D126 K128 N130 N131 D144 S148 2.7.11.1 0004672,0005524,0006468 Kd<3nM remove_due_to_license_issue P15056 25430902 1721 DWEIPDGQITVGQRIGSGGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRMQNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 4cqf A 2.3 BS02 9Z8 A 1 Y99 D100 H142 F151 D186 H188 F216 G339 Y341 Y98 D99 H141 F150 D176 H178 F206 G310 Y312 3.5.1.98 0004407,0005634,0006325,0031507,0046872 remove_due_to_license_issue IC50=50119nM A5H660 24657767 700 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 4cqg A 2.57 BS01 OT5 A 1 I17 G18 V25 A38 K40 L86 E87 Y88 C89 E93 L139 I149 D150 I16 G17 V24 A37 K39 L85 E86 Y87 C88 E92 L138 I148 D149 D132 K134 E136 N137 D150 S171 D131 K133 E135 N136 D149 S158 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q61846 24657156 1332 KDYDELLKYYELYETIGTGGFAKVKLACHVLTGEMVAIKIMDKNALGSDLPRVKTEIDALKSLRHQHICQLYHVLETKNKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQILSAVAYVHSQGYAHRDLKPENLLFDENHKLKLIDFGLCAKCGSLAYAAPELIQGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYEVPKWLSPSSILLLQQMLQVDPKKRISMRNLLNHPWVMQDYSCPVEWQSKTPLTHLDEDCVTELSVHHRSSRQTMEDLISSWQYDHLTATYLLLLAKKARLEHHH 4cr5 A 2.0 BS01 0TU A 1 D189 A190 T213 W215 G216 G218 C219 G226 V227 Y228 D182 A183 T206 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=70uM remove_due_to_license_issue Ki=70000nM, IC50=140000nM P03951 25629509 1489 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4cr9 A 1.7 BS01 OTW A 1 D189 A190 K192 W215 G216 G218 C219 D182 A183 K185 W208 G209 G211 C212 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=80uM remove_due_to_license_issue P03951 25629509 1489 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4cra A 1.8 BS01 XJ8 A 1 H38 L39 H57 Y143 I151 D189 A190 K192 G193 S195 W215 G216 G218 H27 L28 H44 Y134 I141 D182 A183 K185 G186 S188 W208 G209 G211 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.06uM remove_due_to_license_issue P03951 25629509 1491 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4crb A 1.85 BS01 7P0 A 1 H38 L39 H57 Y143 I151 D189 A190 C191 K192 G193 S195 W215 G218 C219 V227 H27 L28 H44 Y134 I141 D182 A183 C184 K185 G186 S188 W208 G211 C212 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.027uM remove_due_to_license_issue Ki=1.6nM P03951 25629509 1485 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4crc A 1.6 BS01 OTM A 1 L39 C40 H57 Y143 I151 A190 C191 K192 G193 S195 W215 G216 G218 C219 G226 V227 L28 C29 H44 Y134 I141 A183 C184 K185 G186 S188 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.0019uM remove_due_to_license_issue Ki=1.4nM P03951 25629509 1245 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGERNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQA 4crd A 2.1 BS01 OTJ A 1 R37D H38 L39 I151 D189 A190 C191 K192 G193 S195 T213 S214 W215 G216 G218 C219 G226 V227 Y228 R26 H27 L28 I141 D182 A183 C184 K185 G186 S188 T206 S207 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.08uM remove_due_to_license_issue P03951 25629509 1244 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQ 4crf A 2.3 BS01 R9B A 1 H38 L39 H57 Y143 I151 D189 A190 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 H27 L28 H44 Y134 I141 D182 A183 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.0005uM remove_due_to_license_issue IC50=1.000000nM, Ki=0.500000nM P03951 25629509 1438 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQAEIAEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYADSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4crj A 2.0 BS04 YH5 A 1 T43 A44 P45 V46 G47 F54 N56 R121 F123 T44 A45 P46 V47 G48 F55 N57 R122 F124 0003848,0009396 Kd=1.1uM remove_due_to_license_issue 25357262 1163 HMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRYK 4crl A 2.4 BS01 C1I A 1 V27 Y32 V35 A50 I79 A100 W105 H106 A155 L158 V30 Y35 V38 A53 I82 A103 W108 H109 A152 L155 D151 K153 N156 D173 N181 T196 D148 K150 N153 D170 N178 T183 2.7.11.22,2.7.11.23 0004672,0005524,0006468 Kd=195pM remove_due_to_license_issue Kd=17nM, IC50=12nM P49336 26416749 1360 DDKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4cs9 A 2.01 BS02 AMP A 1 C7 K8 Y9 F23 C5 K6 Y7 F21 ? 0000166,0005198,0030430,0042025,0044423,0046782,0046872 remove_due_to_license_issue Q8QN58 24842877 1172 RKAPCKYEVRGKCNRGSECKFNHNYWSWPDRYLLIRSNYLLNQLLRNTDRGREDRTQDFVLGSTNVVQGYIDDNQSITKAAACYSLHNIIKQLQEVEVRQARDNKLSDSKHVALHNLVLSYMEMSKTPASLINNLKRLPREKLKKLAKLIIDLSAGAE 4cs9 C 2.01 BS02 AMP C 1 C7 K8 Y9 F23 C6 K7 Y8 F22 ? 0000166,0005198,0030430,0042025,0044423,0046782,0046872 remove_due_to_license_issue Q8QN58 24842877 1174 SRKAPCKYEVRGKCNRGSECKFNHNYWSWPDRYLLIRSNYLLNQLLRDTDRADGAGREDRTQDFVLGSTNVVQGYIDDNQSITKAAACYSLHNIIKQLQEVEVRQARDNKLSDSKHVALHNLVLSYMEMSKTPASLINNLKRLPREKLKKLAKLIIDLSAGAEND 4cs9 C 2.01 BS03 AMP C 2 Y9 C15 N16 R17 Y8 C14 N15 R16 ? 0000166,0005198,0030430,0042025,0044423,0046782,0046872 remove_due_to_license_issue Q8QN58 24842877 1175 SRKAPCKYEVRGKCNRGSECKFNHNYWSWPDRYLLIRSNYLLNQLLRDTDRADGAGREDRTQDFVLGSTNVVQGYIDDNQSITKAAACYSLHNIIKQLQEVEVRQARDNKLSDSKHVALHNLVLSYMEMSKTPASLINNLKRLPREKLKKLAKLIIDLSAGAEND 4csd A 1.35 BS01 MFU A 1 R108 E119 G130 A131 W167 W172 R104 E115 G126 A127 W162 W167 ? Kd=1.23uM remove_due_to_license_issue Q8XXK6 25044646 301 MSSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTEWCWDGNGWTKGAYTSSTVPGDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 4csd A 1.35 BS02 MFU A 2 R153 E164 A176 W213 W218 R149 E159 A171 W208 W213 ? Kd=1.23uM remove_due_to_license_issue Q8XXK6 25044646 302 MSSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTEWCWDGNGWTKGAYTSSTVPGDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 4csd A 1.35 BS03 MFU A 3 R199 E210 G221 A222 W258 W263 R194 E205 G216 A217 W253 W258 ? Kd=1.23uM remove_due_to_license_issue Q8XXK6 25044646 303 MSSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTEWCWDGNGWTKGAYTSSTVPGDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 4csd A 1.35 BS04 MFU A 4 I16 W31 W36 R244 E255 A267 I17 W32 W37 R239 E250 A262 ? Kd=1.23uM remove_due_to_license_issue Q8XXK6 25044646 304 MSSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTEWCWDGNGWTKGAYTSSTVPGDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 4csd A 1.35 BS05 MFU A 5 R17 E28 G39 A40 W76 W81 R18 E29 G40 A41 W77 W82 ? Kd=1.23uM remove_due_to_license_issue Q8XXK6 25044646 305 MSSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTEWCWDGNGWTKGAYTSSTVPGDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 4csd A 1.35 BS06 MFU A 6 R62 E73 A85 I107 W122 W127 R63 E74 A86 I103 W118 W123 ? Kd=1.23uM remove_due_to_license_issue Q8XXK6 25044646 306 MSSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTSDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTEWCWDGNGWTKGAYTSSTVPGDQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 4csf A 2.598 BS01 rna a 0 Y32 F35 N71 G100 N101 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y29 F32 N68 G97 N98 P99 S107 R108 T182 I183 P185 R188 T198 K201 P202 M204 A205 A206 S208 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf B 2.598 BS01 rna a 0 Y32 K204 P205 Y29 K201 P202 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf B 2.598 BS02 rna c 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf C 2.598 BS01 rna c 0 Y32 F35 N71 G100 N101 P102 S110 R111 T185 I186 R191 T201 K204 P205 M207 A208 A209 S211 Y30 F33 N69 G98 N99 P100 S108 R109 T183 I184 R189 T199 K202 P203 M205 A206 A207 S209 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 DENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGKDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf D 2.598 BS01 rna c 0 Y32 K204 Y29 K201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf D 2.598 BS02 rna e 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf E 2.598 BS01 rna e 0 Y32 F35 N71 G100 N101 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y29 F32 N68 G97 N98 P99 S107 R108 T182 I183 P185 R188 T198 K201 P202 M204 A205 A206 S208 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYEGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf F 2.598 BS01 rna a 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf F 2.598 BS02 rna e 0 Y32 K204 Y29 K201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf G 2.598 BS01 rna g 0 Y32 F35 N71 G100 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y29 F32 N68 G97 P99 S107 R108 T182 I183 P185 R188 T198 K201 P202 M204 A205 A206 S208 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf H 2.598 BS01 rna g 0 Y32 N101 K204 P205 Y29 N98 K201 P202 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf H 2.598 BS02 rna i 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf I 2.598 BS01 rna i 0 Y32 F35 N71 K72 G100 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y29 F32 N68 K69 G97 P99 S107 R108 T182 I183 P185 R188 T198 K201 P202 M204 A205 A206 S208 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf J 2.598 BS01 rna i 0 Y32 N101 K204 Y29 N98 K201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf J 2.598 BS02 rna k 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf K 2.598 BS01 rna k 0 Y32 F35 N71 K72 G100 N101 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y31 F34 N70 K71 G99 N100 P101 S109 R110 T184 I185 P187 R190 T200 K203 P204 M206 A207 A208 S210 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 SDENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf L 2.598 BS01 rna g 0 K79 T185 I186 K77 T183 I184 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 DENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf L 2.598 BS02 rna k 0 Y32 N101 P205 Y30 N99 P203 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 DENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf M 2.598 BS01 rna m 0 Y32 F35 N71 K72 G100 P102 S110 R111 F182 T185 I186 T201 K204 P205 M207 A208 A209 S211 Y28 F31 N67 K68 G96 P98 S106 R107 F178 T181 I182 T197 K200 P201 M203 A204 A205 S207 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 NYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf N 2.598 BS01 rna m 0 Y32 K204 Y29 K201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf N 2.598 BS02 rna o 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf O 2.598 BS01 rna o 0 Y32 F35 N71 K72 G100 N101 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y28 F31 N67 K68 G96 N97 P98 S106 R107 T181 I182 P184 R187 T197 K200 P201 M203 A204 A205 S207 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 NYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf P 2.598 BS01 rna o 0 Y32 N101 K204 Y29 N98 K201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf Q 2.598 BS01 rna q 0 Y32 F35 N71 K72 G100 P102 S110 R111 T185 I186 R191 T201 K204 P205 M207 A208 A209 S211 Y29 F32 N68 K69 G97 P99 S107 R108 T182 I183 R188 T198 K201 P202 M204 A205 A206 S208 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf R 2.598 BS01 rna m 0 K79 T185 I186 K75 T181 I182 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 NYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf R 2.598 BS02 rna q 0 Y32 N101 P205 Y28 N97 P201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 NYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf S 2.598 BS01 rna s 0 Y32 F35 N71 K72 G100 P102 S110 R111 T185 I186 R191 T201 K204 P205 M207 A208 A209 S211 Y29 F32 N68 K69 G97 P99 S107 R108 T182 I183 R188 T198 K201 P202 M204 A205 A206 S208 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf T 2.598 BS01 rna s 0 Y32 K204 P205 Y30 K202 P203 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 DENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf T 2.598 BS02 rna u 0 K79 T185 I186 K77 T183 I184 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 DENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf U 2.598 BS01 rna u 0 Y32 F35 N71 P102 S110 R111 T185 I186 R191 T201 K204 P205 M207 A208 A209 S211 Y28 F31 N67 P98 S106 R107 T181 I182 R187 T197 K200 P201 M203 A204 A205 S207 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 NYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKV 4csf V 2.598 BS01 rna u 0 Y32 K204 Y29 K201 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf V 2.598 BS02 rna w 0 K79 T185 I186 K76 T182 I183 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf W 2.598 BS01 rna w 0 Y32 F35 N71 K72 G100 N101 P102 S110 R111 T185 I186 P188 R191 T201 K204 P205 M207 A208 A209 S211 Y30 F33 N69 K70 G98 N99 P100 S108 R109 T183 I184 P186 R189 T199 K202 P203 M205 A206 A207 S209 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 DENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGRDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf X 2.598 BS01 rna s 0 K79 T185 K76 T182 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGKDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csf X 2.598 BS02 rna w 0 Y32 N101 Y29 N98 ? 0003723,0019013,0019029,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue P21701 24688060 1 ~ 9 ENYRDIALAFLDESADSGTINAWVNEFAYQGFDPKRIVQLVKERGTAKGKDWKKDVKMMIVLNLVRGNKPEAMMKKMSEKGASIVANLISVYQLKEGNPGRDTITLSRVSAAFVPWTVQALRVLSESLPVSGTTMDAIAGVTYPRAMMHPSFAGIIDLDLPNGAGATIADAHGLFMIEFSKTINPSLRTKQANEVAATFEKPNMAAMSGRFFTREDKKKLLIAVGIIDEDLVLASAVVRSAEKYRAKVG 4csj A 2.3 BS02 NN7 A 1 M560 L563 N564 L566 G567 Q570 M604 A607 L608 R611 F623 Q642 C736 M31 L34 N35 L37 G38 Q41 M75 A78 L79 R82 F94 Q113 C207 ? ic50=4.9nM remove_due_to_license_issue IC50=1.5nM P04150 24755427 1778 PTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQMIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 4css A 1.069 BS01 CWX A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 I52 D54 Q130 N132 D137 ? 0007155,0009289 Kd=3.5nM remove_due_to_license_issue P08191 25666045 1159 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4cst A 1.1 BS01 CWK A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 ? 0007155,0009289 Kd=1.3nM remove_due_to_license_issue P08191 25666045 1160 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPTG 4ctj A 1.47 BS02 3A9 A 1 L237 R241 M244 R247 L231 R235 M238 R241 3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue A9LIE0 24704437 1264 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 4ctk A 1.53 BS02 SVN A 1 L17 L20 F25 L11 L14 F19 3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue A9LIE0 24704437 1264 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 4cts A 2.9 BS01 OAA A 1 H238 N242 H274 R329 H238 N242 H274 R329 S244 H274 H320 R329 D375 S244 H274 H320 R329 D375 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 remove_due_to_license_issue P00889 6716477 438 ASSTNLKDILADLIPKEQARIKTFRQQHGNTVVGQITVDMMYGGMRGMKGLVYETSVLDPDEGIRFRGYSIPECQKMLPKAKGGEEPLPEGLFWLLVTGQIPTEEQVSWLSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGIHRTKYWELIYEDCMDLIAKLPCVAAKIYRNLYREGSSIGAIDSKLDWSHNFTNMLGYTDAQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLVWLTQLQKEVGKDVSDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPHDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTDGLIKLVDSK 4cts B 2.9 BS01 OAA B 1 H238 N242 H274 H320 R329 R401 H238 N242 H274 H320 R329 R401 S244 H274 H320 R329 D375 S244 H274 H320 R329 D375 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 remove_due_to_license_issue P00889 6716477 438 ASSTNLKDILADLIPKEQARIKTFRQQHGNTVVGQITVDMMYGGMRGMKGLVYETSVLDPDEGIRFRGYSIPECQKMLPKAKGGEEPLPEGLFWLLVTGQIPTEEQVSWLSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGIHRTKYWELIYEDCMDLIAKLPCVAAKIYRNLYREGSSIGAIDSKLDWSHNFTNMLGYTDAQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLVWLTQLQKEVGKDVSDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPHDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTDGLIKLVDSK 4cu1 A 1.89 BS03 71S A 1 Q249 P336 V338 N340 F355 W358 E363 W449 Y477 Q172 P259 V261 N263 F278 W281 E286 W372 Y400 C186 R189 W358 E363 C109 R112 W281 E286 1.14.13.39 0004517,0006809 Ki=19417nM remove_due_to_license_issue Ki=16000nM P29473 24758147 800 GPKFPRVKNWELGSITYDTLCAQSQQDGPCTPRRCLGSLVLPRPAEQLLSQARDFINQYYSSIKRSGSQAHEERLQEVEAEVASTGTYHLRESELVFGAKQAWRNAPRCVGRIQWGKLQVFDARDCSSAQEMFTYICNHIKYATNRGNLRSAITVFPQRAPGRGDFRIWNSQLVRYAGYRQQDGSVRGDPANVEITELCIQHGWTPGNGRFDVLPLLLQAPDEAPELFVLPPELVLEVPLEHPTLEWFAALGLRWYALPAVSNMLLEIGGLEFSAAPFSGWYMSTEIGTRNLCDPHRYNILEDVAVCMDLDTRTTSSLWKDKAAVEINLAVLHSFQLAKVTIVDHHAATVSFMKHLDNEQKARGGCPADWAWIVPPISGSLTPVFHQEMVNYILSPAFRYQPDPW 4cu1 B 1.89 BS04 71S B 1 L107 Q249 P336 V338 N340 F355 W358 E363 W449 L39 Q171 P258 V260 N262 F277 W280 E285 W371 C186 R189 W358 E363 C108 R111 W280 E285 1.14.13.39 0004517,0006809 Ki=19417nM remove_due_to_license_issue Ki=16000nM P29473 24758147 800 KFPRVKNWELGSITYDTLCAQSQQDGPCTPRRCLGSLVLPRKPAEQLLSQARDFINQYYSSIKRSGSQAHEERLQEVEAEVASTGTYHLRESELVFGAKQAWRNAPRCVGRIQWGKLQVFDARDCSSAQEMFTYICNHIKYATNRGNLRSAITVFPQRAPGRGDFRIWNSQLVRYAGYRQQDGSVRGDPANVEITELCIQHGWTPGNGRFDVLPLLLQAPDEAPELFVLPPELVLEVPLEHPTLEWFAALGLRWYALPAVSNMLLEIGGLEFSAAPFSGWYMSTEIGTRNLCDPHRYNILEDVAVCMDLDTRTTSSLWKDKAAVEINLAVLHSFQLAKVTIVDHHAATVSFMKHLDNEQKARGGCPADWAWIVPPISGSLTPVFHQEMVNYILSPAFRYQPDPW 4cu7 A 2.2 BS01 GIF A 1 R288 H484 E564 E645 S648 W685 W708 E716 F733 R152 H348 E428 E509 S512 W549 W572 E580 F597 R288 H450 H484 T509 Y511 E564 Y629 E645 S730 F733 R152 H314 H348 T373 Y375 E428 Y493 E509 S594 F597 3.2.1.23 0004553,0005975 Kd=26nM remove_due_to_license_issue A0A0H2UP19 25210925 1985 AVTNEEVNQMIEDRKVDFNQNWYFKLNANSKEAIKPDADVSTWKKLDLPYDWSIFNDFDHESPAQNEGGQLNGGEAWYRKTFKLDEKDLKKNVRLTFDGVYMDSQVYVNGQLVGHYPNGYNQFSYDITKYLQKDGRENVIAVHAVNKQPSSRWYSGSGIYRDVTLQVTDKVHVEKNGTTILTPKLEEQQHGKVETHVTSKIVNTDDKDHELVAEYQIVERGGHAVTGLVRTASRTLKAHESTSLDAILEVERPKLWTVLNDKPALYELITRVYRDGQLVDAKKDLFGYRYYHWTPNEGFSLNGERIKFHGVSLHHDHGALGAEENYKAEYRRLKQMKEMGVNSIRTTHNPASEQTLQIAAELGLLVQEEAFDTWYGGKKPYDYGRFFEKDATHPEARKGEKWSDFDLRTMVERGKNNPAIFMWSIGNEIGEANGDAHSLATVKRLVKVIKDVDKTRYVTMGADKFRFGNGSGGHEKIADELDAVGFNYSEDNYKALRAKHPKWLIYGSETSSATRTRGSYYRPERELKHSNGPERNYEQSDYGNDRVGWGKTATASWTFDRDNAGYAGQFIWTGTDYIGEPTPWHNQNQTPVKSSYFGIVDTAGIPKHDFYLYQSQWVSVKKKPMVHLLPHWNWENKELASKVADSEGKIPVRAYSNASSVELFLNGKSLGLKTFNKKQTSDGRTYQEGANANELYLEWKVAYQPGTLEAIARDESGKEIARDKITTAGKPAAVRLIKEDHAIAADGKDLTYIYYEIVDSQGNVVPTANNLVRFQLHGQGQLVGVDNGEQASRERYKAQADGSWIRKAFNGKGVAIVKSTEQAGKFTLTAHSDLLKSNQVTVFTGKKE 4cu8 A 2.5 BS01 DGJ A 1 R288 H484 N563 E564 E645 S648 W685 W708 E716 F733 R152 H348 N427 E428 E509 S512 W549 W572 E580 F597 R288 H450 H484 T509 Y511 E564 Y629 E645 S730 F733 R152 H314 H348 T373 Y375 E428 Y493 E509 S594 F597 3.2.1.23 0004553,0005975 Ki=33.9uM remove_due_to_license_issue A0A0H2UP19 25210925 1985 AVTNEEVNQMIEDRKVDFNQNWYFKLNANSKEAIKPDADVSTWKKLDLPYDWSIFNDFDHESPAQNEGGQLNGGEAWYRKTFKLDEKDLKKNVRLTFDGVYMDSQVYVNGQLVGHYPNGYNQFSYDITKYLQKDGRENVIAVHAVNKQPSSRWYSGSGIYRDVTLQVTDKVHVEKNGTTILTPKLEEQQHGKVETHVTSKIVNTDDKDHELVAEYQIVERGGHAVTGLVRTASRTLKAHESTSLDAILEVERPKLWTVLNDKPALYELITRVYRDGQLVDAKKDLFGYRYYHWTPNEGFSLNGERIKFHGVSLHHDHGALGAEENYKAEYRRLKQMKEMGVNSIRTTHNPASEQTLQIAAELGLLVQEEAFDTWYGGKKPYDYGRFFEKDATHPEARKGEKWSDFDLRTMVERGKNNPAIFMWSIGNEIGEANGDAHSLATVKRLVKVIKDVDKTRYVTMGADKFRFGNGSGGHEKIADELDAVGFNYSEDNYKALRAKHPKWLIYGSETSSATRTRGSYYRPERELKHSNGPERNYEQSDYGNDRVGWGKTATASWTFDRDNAGYAGQFIWTGTDYIGEPTPWHNQNQTPVKSSYFGIVDTAGIPKHDFYLYQSQWVSVKKKPMVHLLPHWNWENKELASKVADSEGKIPVRAYSNASSVELFLNGKSLGLKTFNKKQTSDGRTYQEGANANELYLEWKVAYQPGTLEAIARDESGKEIARDKITTAGKPAAVRLIKEDHAIAADGKDLTYIYYEIVDSQGNVVPTANNLVRFQLHGQGQLVGVDNGEQASRERYKAQADGSWIRKAFNGKGVAIVKSTEQAGKFTLTAHSDLLKSNQVTVFTGKKE 4cwb A 1.56 BS04 X6L A 1 T43 P45 V46 G47 F54 N56 R88 R92 R121 F123 T44 P46 V47 G48 F55 N57 R89 R93 R122 F124 0003848,0009396 Kd=0.81uM remove_due_to_license_issue 25357262 1163 HMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRYK 4cwf A 2.0 BS01 H05 A 1 N51 M98 L107 F138 Y139 W162 N36 M83 L92 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=32.4uM remove_due_to_license_issue P07900 24980703 1224 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4cwn A 1.8 BS01 6LV A 1 N51 I96 G97 M98 L107 F138 Y139 V150 W162 T184 N35 I80 G81 M82 L91 F122 Y123 V134 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=2.6uM remove_due_to_license_issue P07900 24980703 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4cwo A 2.31 BS01 T62 A 1 N51 D93 M98 L107 F138 W162 T184 N36 D78 M83 L92 F123 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=6.1uM remove_due_to_license_issue P07900 24980703 1226 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 4cwp A 1.95 BS01 TV2 A 1 N51 I96 M98 L107 F138 V150 W162 T184 N35 I80 M82 L91 F122 V134 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.17uM remove_due_to_license_issue P07900 24980703 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4cwq A 2.0 BS01 W2D A 1 N51 A55 K58 G97 M98 D102 L107 F138 W162 T184 N35 A39 K42 G81 M82 D86 L91 F122 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.088uM remove_due_to_license_issue P07900 24980703 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4cwr A 2.0 BS01 HAJ A 1 N51 A55 I96 G97 M98 L107 F138 W162 T184 N35 A39 I80 G81 M82 L91 F122 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.005uM remove_due_to_license_issue P07900 24980703 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4cws A 2.3 BS01 G3R A 1 N51 A55 K58 G97 M98 D102 L107 F138 V150 W162 T184 N35 A39 K42 G81 M82 D86 L91 F122 V134 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.012uM remove_due_to_license_issue P07900 24980703 1224 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4cwt A 1.9 BS01 IK9 A 1 N51 K58 M98 L103 L107 F138 Y139 V150 W162 F170 N36 K43 M83 L88 L92 F123 Y124 V135 W147 F155 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.179uM remove_due_to_license_issue P07900 24980703 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4cxw A 3.1 BS01 6MK A 1 Y106 Y108 V228 H231 D233 E234 Y295 H307 R316 S318 R322 Y80 Y82 V168 H171 D173 E174 Y224 H236 R245 S247 R251 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 28553460 1504 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGTEAEIAAACETFLKLNDYLQIETIQALEELAAKEKDEVDIKSRAAYNVTLLNFMDPQKLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLE 4cxx A 2.76 BS01 640 A 1 R96 Y106 L109 H231 D233 E234 Y295 H307 V309 R316 S318 R322 R70 Y80 L83 H176 D178 E179 Y229 H241 V243 R250 S252 R256 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 28553460 1505 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGEAEIAAACETFLKLNDYLQIETIQALEELAAKEKANEDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4cxy A 2.65 BS01 DGR A 1 Y108 H231 D233 E234 Y295 H307 V309 R316 S318 R322 Y82 H177 D179 E180 Y230 H242 V244 R251 S253 R257 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 28553460 1503 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNITEAEIAAACETFLKLNDYLQIETIQALEELAAKEKDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLE 4czs A 1.73 BS04 8LR E 1 Y12 G98 L99 Y100 A207 D208 G227 R228 Y12 G98 L99 Y100 A207 D208 G227 R228 ? 0005515,0005537,0030246,0046872 remove_due_to_license_issue P81461 25860443 101 ADTIVAVELDTYPNTDIGDPSYPHIGIDIKSVRSKKTAKWNMQNGKVGTAHIIYNSVDKRLSAVVSYPNADSATVSYDVDLDNVLPEWVRVGLSASTGLYKETNTILSWSFTSKLKSNSTHETNALHFMFNQFSKDQKDLILQGDATTGTDGNLELTRVSSNGSPQGSSVGRALFYAPVHIWESSAVVASFEATFTFLIKSPDSHPADGIAFFISNIDSSIPSGSTGRLLGLFPDAN 4d08 A 1.9 BS02 Q2T A 1 T768 D808 F830 M847 M848 Q859 F862 T190 D230 F252 M269 M270 Q281 F284 3.1.4.17 0004114,0007165,0008081 ic50=10nM remove_due_to_license_issue IC50=10.0nM O00408 25221665 1918 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 4d09 A 2.5 BS01 788 A 1 L770 L774 L809 I826 M847 F862 L192 L196 L231 I248 M269 F284 3.1.4.17 0004114,0007165,0008081 ic50=1.7nM remove_due_to_license_issue O00408 25221665 1 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLDE 4d0w A 1.77 BS01 VVQ A 1 L855 G856 G861 V863 A880 Y931 L932 L983 D994 L17 G18 G22 V24 A41 Y92 L93 L144 D155 D976 A978 R980 N981 D994 S1016 D137 A139 R141 N142 D155 S177 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.02uM remove_due_to_license_issue IC50=20nM O60674 25009002 2132 RDPTQFEERHLKFLQQLGKGFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4d0x A 1.82 BS01 953 A 1 L855 G856 K857 G858 A880 Y931 L932 N981 L983 D994 L17 G18 K19 G20 A42 Y93 L94 N143 L145 D156 D976 A978 R980 N981 D994 S1016 D138 A140 R142 N143 D156 S178 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.008uM remove_due_to_license_issue IC50=8.0nM O60674 25009002 2132 RDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 4d1a A 3.4 BS01 I5H A 1 Q42 A44 W117 G219 W220 N318 Q32 A34 W107 G209 W210 N308 ? 0005886,0015205,0015851,0016020,0022857,0046872,0055085 remove_due_to_license_issue D6R8X8 24952894 1467 SLLNPSNAPTRYAERSVGPFSLAAIWFAMAIQVAIFIAAGQMTSSFQVWQVIVAIAAGCTIAVILLFFTQSAAIRWGINFTVAARMPFGIRGSLIPITLKALLSLFWFGFQTWLGALALDEITRLLTGFTNLPLWIVIFGAIQVVTTFYGITFIRWMNVFASPVLLAMGVYMVYLMLDGADVSLGEVMSMGGENPGMPFSTAIMIFVGGWIAVVVSIHDIVKECKVDPNASREGQTKADARYATAQWLGMVPASIIFGFIGAASMVLVGEWNPVIAITEVVGGVSIPMAILFQVFVLLATWSTNPAANLLSPAYTLCSTFPRVFTFKTGVIVSAVVGLLMMPWQFAGVLNTFLNLLASALGPLAGIMISDYFLVRRRRISLHDLYRTKGIYTYWRGVNWVALAVYAVALAVSFLTPDLMFVTGLIAALLLHIPAMRWVAKTFPLFSEAESRNEDYL 4d1b A 3.8 BS01 5FH A 1 Q42 A44 W117 G219 W220 N318 Q32 A34 W107 G209 W210 N308 ? 0005886,0015205,0015851,0016020,0022857,0046872,0055085 remove_due_to_license_issue D6R8X8 24952894 1467 SLLNPSNAPTRYAERSVGPFSLAAIWFAMAIQVAIFIAAGQMTSSFQVWQVIVAIAAGCTIAVILLFFTQSAAIRWGINFTVAARMPFGIRGSLIPITLKALLSLFWFGFQTWLGALALDEITRLLTGFTNLPLWIVIFGAIQVVTTFYGITFIRWMNVFASPVLLAMGVYMVYLMLDGADVSLGEVMSMGGENPGMPFSTAIMIFVGGWIAVVVSIHDIVKECKVDPNASREGQTKADARYATAQWLGMVPASIIFGFIGAASMVLVGEWNPVIAITEVVGGVSIPMAILFQVFVLLATWSTNPAANLLSPAYTLCSTFPRVFTFKTGVIVSAVVGLLMMPWQFAGVLNTFLNLLASALGPLAGIMISDYFLVRRRRISLHDLYRTKGIYTYWRGVNWVALAVYAVALAVSFLTPDLMFVTGLIAALLLHIPAMRWVAKTFPLFSEAESRNEDYL 4d1c A 3.7 BS01 B5H A 1 Q42 A44 I45 W117 G219 W220 N318 Q32 A34 I35 W107 G209 W210 N308 ? 0005886,0015205,0015851,0016020,0022857,0046872,0055085 remove_due_to_license_issue D6R8X8 24952894 1467 SLLNPSNAPTRYAERSVGPFSLAAIWFAMAIQVAIFIAAGQMTSSFQVWQVIVAIAAGCTIAVILLFFTQSAAIRWGINFTVAARMPFGIRGSLIPITLKALLSLFWFGFQTWLGALALDEITRLLTGFTNLPLWIVIFGAIQVVTTFYGITFIRWMNVFASPVLLAMGVYMVYLMLDGADVSLGEVMSMGGENPGMPFSTAIMIFVGGWIAVVVSIHDIVKECKVDPNASREGQTKADARYATAQWLGMVPASIIFGFIGAASMVLVGEWNPVIAITEVVGGVSIPMAILFQVFVLLATWSTNPAANLLSPAYTLCSTFPRVFTFKTGVIVSAVVGLLMMPWQFAGVLNTFLNLLASALGPLAGIMISDYFLVRRRRISLHDLYRTKGIYTYWRGVNWVALAVYAVALAVSFLTPDLMFVTGLIAALLLHIPAMRWVAKTFPLFSEAESRNEDYL 4d1d A 3.7 BS02 5ND A 1 Q42 A48 W117 Q121 F216 G219 W220 N318 Q32 A38 W107 Q111 F206 G209 W210 N308 ? 0005886,0015205,0015851,0016020,0022857,0046872,0055085 remove_due_to_license_issue D6R8X8 24952894 1468 SLLNPSNAPTRYAERSVGPFSLAAIWFAMAIQVAIFIAAGQMTSSFQVWQVIVAIAAGCTIAVILLFFTQSAAIRWGINFTVAARMPFGIRGSLIPITLKALLSLFWFGFQTWLGALALDEITRLLTGFTNLPLWIVIFGAIQVVTTFYGITFIRWMNVFASPVLLAMGVYMVYLMLDGADVSLGEVMSMGGENPGMPFSTAIMIFVGGWIAVVVSIHDIVKECKVDPNASREGQTKADARYATAQWLGMVPASIIFGFIGAASMVLVGEWNPVIAITEVVGGVSIPMAILFQVFVLLATWSTNPAANLLSPAYTLCSTFPRVFTFKTGVIVSAVVGLLMMPWQFAGVLNTFLNLLASALGPLAGIMISDYFLVRRRRISLHDLYRTKGIYTYWRGVNWVALAVYAVALAVSFLTPDLMFVTGLIAALLLHIPAMRWVAKTFPLFSEAESRNEDYL 4d1j A 1.8 BS01 DGJ A 1 N67 K134 N135 N204 E205 E349 F374 N383 N31 K98 N99 N168 E169 E313 F338 N347 3.2.1.23 0004565,0005975,0009341 Kd=485nM remove_due_to_license_issue B3PBE0 25171165 600 APLPELLSNNGKHALMVDGAPYIILGSQTNNSSNYPDALKDVWPSMEKMGANTLSIPVAWEQIEPVEGQFDFSFVDVLLKEARQRKVRLVLLWFATWKNNAPHYAPAWVKLDNARFPRVVKEDGDTLNSLSPLGQNTLAADKKAFVELMKYLAKRDKDHTVIMVQVQNEVGTYGAVRDYSPMAQAVFNAAVPDDLIQKLQLKPGTWSQVFGRDADEFFHAYQIARYCDEVTVAGKAIKNLPMYVNVALRNPFNPGLPGQYSSGGGTDNVLHIWKAAAPNIDLIAPDIYFRDYKTVSKVLELYTRPDNALFVAEIGNDQPFARYLFPTLGKGGIGFSPFGMDDTDYTNYPLGAKVYNDETIEQFAQVYRLVNPMMREWARLSYQGQVWGVAEPLDSTTETQKIWNAEATPEEKEQHKKDRASALTQQLDLGLWDAEVTYGRPMFWVTPPEGNTPAAGGALIAQLDDNEYLVTAYKARVEFKPSQELAGKKFMIERVEEGRFEKGKWVMERVWNGDQTDWGLNFTDRPHLLRVKMASYSVQ 4d1s A 1.66 BS01 BJG A 1 L855 G856 K857 V863 A880 Y931 L932 G935 L983 D994 L14 G15 K16 V21 A38 Y89 L90 G93 L141 D152 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S169 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.022uM remove_due_to_license_issue IC50=22nM O60674 25009002 1141 TQFEERHLKFLQQLGKGFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVSPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIESKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4d1y A 2.6 BS01 RBF A 1 N161 W164 N161 W164 ? 0000166,0005737,0046872 remove_due_to_license_issue Q8A8A4 25263158 1176 MAKKVAVLAVNPVNGCGLFQYLEAFFENGISYKVFAVSDTKEIKTNSGMVLIVDDVIANLKGHEDEFDALVFSCGDAVPVFQQYANQPYNVDLMEVIKTFGEKGKMMIGHCAGAMMFDFTGITKGKKVAVHPLAKPAIQNGIATDEKSEIDGNFFTAQDENTIWTMLPKVIEALK 4d2p B 2.55 BS01 6Z7 B 1 L27 A38 K40 E57 L61 C70 Y88 C89 P90 L139 I149 D150 L27 A38 K40 E57 L61 C70 Y88 C89 P90 L139 I149 D150 D132 K134 E136 N137 D150 A171 D132 K134 E136 N137 D150 A165 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKDCGALAYAAPELIQGGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2p C 2.55 BS01 6Z7 C 1 L27 A38 K40 E57 L61 C70 Y88 C89 P90 L139 I149 D150 L28 A39 K41 E55 L59 C68 Y86 C87 P88 L137 I147 D148 D132 K134 E136 N137 D150 A171 D130 K132 E134 N135 D148 A156 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589925 1334 HMKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKGALAYAAPELIQGKSGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2r A 2.1 BS01 DYK A 1 L1005 G1006 V1013 A1031 L1081 M1082 T1083 G1085 M1142 M1156 L21 G22 V29 A47 L97 M98 T99 G101 M158 M172 D1135 R1139 N1140 D1153 E1162 D151 R155 N156 D169 E178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=3.3uM remove_due_to_license_issue IC50=3300nM P08069 25738750 2288 DVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 4d2s A 2.5 BS01 DYK A 1 I531 V539 K553 G605 N606 I607 D608 S611 L654 I663 I19 V27 K41 G93 N94 I95 D96 S99 L140 I149 D647 K649 N652 D664 T686 D133 K135 N138 D150 T155 2.7.12.1 0004672,0005524,0006468 ic50=0.02uM remove_due_to_license_issue IC50=20nM P33981 25738750 1794 AANECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIATVNYMPPEAIKDMSPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQI 4d2t A 2.7 BS01 3I7 A 1 A38 K40 E57 C70 E87 Y88 C89 P90 I149 A38 K40 E54 C67 E84 Y85 C86 P87 I146 D132 K134 E136 N137 D150 A171 D129 K131 E133 N134 D147 A156 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCACCGALAYAAPELIQGKSGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2v B 2.45 BS01 45R B 1 I17 L27 K40 E57 L86 C89 P90 I149 D150 I16 L26 K39 E56 L85 C88 P89 I148 D149 D132 K134 E136 N137 D150 A171 D131 K133 E135 N136 D149 A164 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589925 1334 KDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKDCGALAYAAPELIQGGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2v C 2.45 BS01 45R C 1 I17 V25 L27 A38 L86 E87 Y88 C89 P90 I17 V25 L27 A38 L82 E83 Y84 C85 P86 D132 K134 E136 N137 D150 A171 D128 K130 E132 N133 D146 A154 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKGALAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2w A 1.92 BS01 NF5 A 1 I17 A38 C89 P90 L139 I17 A38 C86 P87 L136 D132 K134 E136 N137 D150 A171 D129 K131 E133 N134 D147 A155 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=31000nM Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCACGALAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2w D 1.92 BS01 NF5 A 1 T16 I17 T16 I17 D132 K134 E136 N137 D150 A171 D132 K134 E136 N137 D150 A164 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=31000nM Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKCGALAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d2w D 1.92 BS02 NF5 D 1 L27 A38 Y88 C89 P90 L139 L27 A38 Y88 C89 P90 L139 D132 K134 E136 N137 D150 A171 D132 K134 E136 N137 D150 A164 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=31000nM Q14680 25589925 1334 MKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKCGALAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4d3h A 2.0 BS01 2BA A 1 R26 A27 T28 G47 Q108 R35 A36 T37 G56 Q102 ? Kd=0.37uM remove_due_to_license_issue Q2G229 25505271 110 SGLVPRGSHMKMIIAIVQDQDSQELADQLVKNNFRATKLATTGGFLRAGNTTFLCGVNDDRVDEILSVINQTCGNREQLVSPVEVEVGGATVFVMPVDAFHQF 4d3h A 2.0 BS02 2BA C 1 I7 G34 F36 L37 T97 F99 I16 G43 F45 L46 T91 F93 ? Kd=0.37uM remove_due_to_license_issue Q2G229 25505271 110 SGLVPRGSHMKMIIAIVQDQDSQELADQLVKNNFRATKLATTGGFLRAGNTTFLCGVNDDRVDEILSVINQTCGNREQLVSPVEVEVGGATVFVMPVDAFHQF 4d3h B 2.0 BS01 2BA A 1 I7 G34 F36 L37 T97 F99 I15 G42 F44 L45 T92 F94 ? Kd=0.37uM remove_due_to_license_issue Q2G229 25505271 110 GLVPRGSHMKMIIAIVQDQDSQELADQLVKNNFRATKLATTGGFLRAGNTTFLCGVNDDRVDEILSVINQTCGNREQLVSPIPVEVEVGGATVFVMPVDAFHQF 4d3h B 2.0 BS02 2BA B 1 R26 A27 T28 G47 Q108 R34 A35 T36 G55 Q103 ? Kd=0.37uM remove_due_to_license_issue Q2G229 25505271 110 GLVPRGSHMKMIIAIVQDQDSQELADQLVKNNFRATKLATTGGFLRAGNTTFLCGVNDDRVDEILSVINQTCGNREQLVSPIPVEVEVGGATVFVMPVDAFHQF 4d4d A 1.4 BS01 IFM A 1 W73 D124 D125 Y243 D294 W35 D86 D87 Y205 D256 3.2.1.101 0005975 remove_due_to_license_issue Q9Z4P9 25772148 400 SDGDTAMKAFNDTFWDPNAKMFWKDSKREKHQDFWVEAELWELVMDAYQHTSDPALKAELKTQIDDVYDGTVAKYGQDWTNNPFNDDIMWWAMGSARAYQITGNPRYLEAARDHFDFVYDTQWDEEFANGGIWWLNSDHNTKNACINFPAAQAALYLYDITKDEHYLNAATKIFRWGKTMLTDGNGKVFDRIEIEHGAVPDATHYNQGTYIGSAVGLYKATGNAVYLDDAVKAAKFTKNHLVDSNGVLNYEGPNGDLKGGKTILMRNLAHLQKTLDETGQYPEFSAEFDEWLAFNIEMAWSHQNSDHIVDGNWAGQGTYESWSSAAAVQALNG 4d4d A 1.4 BS02 MAN A 1 W172 C183 D228 Y243 L295 W134 C145 D190 Y205 L257 3.2.1.101 0005975 remove_due_to_license_issue Q9Z4P9 25772148 401 SDGDTAMKAFNDTFWDPNAKMFWKDSKREKHQDFWVEAELWELVMDAYQHTSDPALKAELKTQIDDVYDGTVAKYGQDWTNNPFNDDIMWWAMGSARAYQITGNPRYLEAARDHFDFVYDTQWDEEFANGGIWWLNSDHNTKNACINFPAAQAALYLYDITKDEHYLNAATKIFRWGKTMLTDGNGKVFDRIEIEHGAVPDATHYNQGTYIGSAVGLYKATGNAVYLDDAVKAAKFTKNHLVDSNGVLNYEGPNGDLKGGKTILMRNLAHLQKTLDETGQYPEFSAEFDEWLAFNIEMAWSHQNSDHIVDGNWAGQGTYESWSSAAAVQALNG 4d52 A 1.76 BS01 GXL A 1 R25 E37 L69 Y88 R24 E36 L68 Y87 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 1316 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d52 A 1.76 BS02 GIV A 1 R25 E37 L69 Y88 R24 E36 L68 Y87 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 2316 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d52 A 1.76 BS03 GXL A 2 R73 E85 G98 L125 W141 W146 R72 E84 G97 L124 W140 W145 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 1318 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d52 A 1.76 BS04 GXL A 3 R126 E138 T150 I176 Y192 W198 R125 E137 T149 I175 Y191 W197 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 1319 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d52 A 1.76 BS05 GXL A 4 Y40 R282 E296 Y39 R281 E295 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 1322 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d52 A 1.76 BS06 GIV A 2 R126 E138 M140 T150 I176 Y192 W198 R125 E137 M139 T149 I175 Y191 W197 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 2319 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d52 A 1.76 BS07 GIV A 3 Y40 R282 E296 Y39 R281 E295 ? 0008150,0030246,0046872 remove_due_to_license_issue Q4WW81 25760594 2322 STPGAQQVLFRTGIAAVNSTNHLRVYFQDVYGSIRESLYEGSWANGTEKNVIGNAKLGSPVAATSKELKHIRVYTLTEGNTLQEFAYDSGTGWYNGGLGGAKFQVAPYSCIAAVFLAGTDALQLRIYAQKPDNTIQEYMWNGDGWKEGTNLGGALPGTGIGATSFRYTDYNGPSIRIWFQTDDLKLVQRAYDPHKGWYPDLVTIFDRAPPRTAIAATSFGAGNSSIYMRIYFVNSDNTIWQVCWDHGKGYHDKGTITPVIQGSEVAIISWGSFANNGPDLRLYFQNGTYISAVSEWVWNRAHGSQLGRSALPPA 4d62 A 2.5 BS01 SIA A 1 E392 V420 K421 N422 E76 V104 K105 N106 Kd=3.64mM remove_due_to_license_issue 26418008 1455 GRATNGQFVTKTAKVLRYKFVRWDALLIIQFIDNIGVMENPTFYRNKSIELRSADFLSPMLNNTYIVPLNGGVRVESPTIPVQLEVILENNSSFIQVGFVRLTVKNGNPHMIIQCNPVPGNIKMIKIKSVMLFTCLIG 4d63 A 2.2 BS01 SIA A 1 E392 V420 K421 N422 E76 V104 K105 N106 Kd~7mM remove_due_to_license_issue 26418008 1455 GRATNGQFVTKTAKVLRYKFVRWDALLIIQFIDNIGVMENPTFYRNKSIELRSADFLSPMLNNTYIVPLNGGVRVESPTIPVQLEVILENNSSFIQVGFVRLTVKNGNPHMIIQCNPVPGNIKMIKIKSVMLFTCLIG 4d7b A 1.15 BS01 TCW B 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=21nM remove_due_to_license_issue Kd=56nM P02766 26902880 1126 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4d7b B 1.15 BS01 TCW A 1 K15 L17 A108 S117 K6 L8 A99 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=21nM remove_due_to_license_issue Kd=56nM P02766 26902880 1126 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4d83 A 2.4 BS01 0GT A 1 L30 D32 G34 S35 P70 Y71 T72 F108 I110 W115 Y187 D217 G219 T220 R224 L33 D35 G37 S38 P73 Y74 T75 F111 I113 W118 Y190 D220 G222 T223 R227 D32 S35 N37 A39 Y71 D217 T220 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.055uM remove_due_to_license_issue P56817 22380629 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4d85 A 2.65 BS01 0GU A 1 G13 D34 G36 S37 Y73 T74 Q75 G76 F110 I112 R130 Y190 D220 G222 G15 D36 G38 S39 Y75 T76 Q77 G78 F112 I114 R132 Y192 D222 G224 D34 S37 N39 A41 Y73 D220 T223 D36 S39 N41 A43 Y75 D222 T225 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 22380629 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4d88 A 1.7 BS01 BXQ A 1 G11 Q12 G13 D32 G34 S35 Y71 T72 F108 I110 Y185 D215 G217 T218 G14 Q15 G16 D35 G37 S38 Y74 T75 F111 I113 Y188 D218 G220 T221 D32 S35 N37 A39 Y71 D215 T218 D35 S38 N40 A42 Y74 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=0.049uM remove_due_to_license_issue P56817 22380629 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4d89 A 1.65 BS01 BXD A 1 Q60 G61 L78 D80 G82 S83 P118 Y119 T120 Q121 F156 Y246 D276 G278 T279 Q15 G16 L33 D35 G37 S38 P73 Y74 T75 Q76 F111 Y188 D218 G220 T221 D80 S83 N85 A87 Y119 D276 T279 D35 S38 N40 A42 Y74 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=0.002uM remove_due_to_license_issue P56817 22380629 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4d8a A 2.183 BS02 0HY A 1 I25 D101 N120 I122 M145 D184 F189 G216 K220 R254 I24 D91 N110 I112 M135 D174 F179 G206 K210 R244 D54 K220 R254 D53 K210 R244 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue Q81VW8 22416048 305 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIG 4d8c A 2.07 BS01 BXD A 1 Q12 G13 L30 D32 G34 S35 Y71 T72 Q73 F108 I110 Y187 D217 G219 T220 Q15 G16 L33 D35 G37 S38 Y74 T75 Q76 F111 I113 Y190 D220 G222 T223 D32 S35 N37 A39 Y71 D217 T220 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.002uM remove_due_to_license_issue P56817 22380629 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4d8e A 1.497 BS01 E64 A 1 Q162 C192 V193 G281 S282 G339 H340 Q17 C47 V48 G136 S137 G194 H195 0006508,0008234 remove_due_to_license_issue 22645124 501 QPVVKSLLNSKGIHYNQGNPYNLLTPVIEKVKPGEQSFVGQHAATGCVATATAQIMKYHNYPNKGLKDYTYTLSSNNPYFNHPKNLFAAISTRQYNWNNILPTYSGRESNVQKMAISELMADVGISVDMDYGPSSGSAGSSRVQRALKENFGYNQSVHQINRSDFSKQDWEAQIDKELSQNQPVYYQGVGKVGGHAFVIDGADGRNFYHVNWGWGGVSDGFFRLDALNPSALGTGGGAGGFNGYQSAVVGIKPL 4d8n A 1.68 BS01 0HM A 1 H57 H99 D189 S190 C191 Q192 G193 S195 W215 G216 H41 H82 D170 S171 C172 Q173 G174 S176 W192 G193 H57 D102 Q192 G193 D194 S195 G196 H41 D85 Q173 G174 D175 S176 G177 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 ic50=1.8uM remove_due_to_license_issue Q92876 22386244 301 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNIPCGSKEKPGVYTNVCRYTNWIQKTIQA 4d8s A 2.398 BS02 0HX A 1 E119 D151 R152 W178 E276 R292 R371 Y406 E37 D69 R70 W97 E195 R211 R288 Y322 D151 E277 R292 R371 Y406 D69 E196 R211 R288 Y322 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=0.32uM remove_due_to_license_issue Q07599 23017008 502 TYMNNTEAICDAKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVEVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVVNSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQTDISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDTQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQIRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEVADWSWHDGAILPFDID 4d8z A 2.198 BS01 0J2 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D90 N109 I111 M134 D173 F178 G205 K209 R243 D54 K220 R254 D52 K209 R243 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 Kd=0.51uM remove_due_to_license_issue Q81VW8 22416048 305 KWDYDLRCGEYTLNLNEKTLIMGILNTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4d9p A 2.26 BS01 Z17 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D91 N110 I112 M135 D174 F179 G206 K210 R244 V28 D54 K220 R254 V27 D53 K210 R244 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=145uM remove_due_to_license_issue Q81VW8 22416048 306 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4da5 A 2.4 BS01 0H7 A 1 D306 Q308 Y354 W420 W423 F435 Y437 D201 Q203 Y249 W315 W318 F330 Y332 2.7.1.32,2.7.1.82 0004103,0004104,0004305,0004713,0005524,0005737,0005811,0005829,0006338,0006629,0006646,0006656,0006657,0006869,0008654,0035401,0042802,0042803,0140801 Ki=0.36uM remove_due_to_license_issue P35790 23416529 502 EQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 4daf A 2.501 BS01 0J4 A 1 D101 N120 M145 D184 G216 K220 R254 D79 N98 M123 D162 G194 K198 R232 D54 K220 R254 D43 K198 R232 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 Kd=0.076uM remove_due_to_license_issue Q81VW8 22416048 301 KWDYDLRCGEYTLNLNEKTLIMGILNSYNEVDAAVRHAKEMRDEGAHIIDIGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4dai A 2.5 BS01 0J5 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D89 N108 I110 M133 D172 F177 G204 K208 R242 V28 D54 K220 R254 V27 D53 K208 R242 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 Kd=110nM remove_due_to_license_issue Q81VW8 22416048 301 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4daw A 2.0 BS01 0H2 A 1 I276 S281 G282 V284 A297 R299 M344 E345 Y346 L396 D407 I28 S33 G34 V36 A49 R51 M96 E97 Y98 L148 D159 D389 K391 D393 N394 D407 P416 T427 D141 K143 D145 N146 D159 P168 T179 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13153 22383326 601 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 4db7 A 2.5 BS01 Z25 A 1 D101 N120 I122 M145 D184 G216 K220 R254 D86 N105 I107 M130 D169 G201 K205 R239 D54 K220 R254 D50 K205 R239 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 Kd=0.273uM remove_due_to_license_issue Q81VW8 22416048 301 KWDYDLRCGEYTLNLNEKTLIMGILNDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4dbm A 2.3 BS01 0J0 A 1 Y93 W147 Y97 W151 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=24nM remove_due_to_license_issue Q8WSF8 22394239 302 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4dbm A 2.3 BS02 0J0 B 1 Q57 V108 M116 I118 Q61 V112 M120 I122 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=24nM remove_due_to_license_issue Q8WSF8 22394239 300 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4dbm E 2.3 BS01 0J0 A 1 Q57 V108 M116 I118 Q59 V110 M118 I120 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=24nM remove_due_to_license_issue Q8WSF8 22394239 302 DKLHSQANLMRLKSDLFNRSMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4dbm E 2.3 BS02 0J0 E 1 W147 Y188 C190 C191 E193 Y195 W149 Y190 C192 C193 E195 Y197 ? 0004888,0005216,0005230,0006811,0016020,0034220 Kd=24nM remove_due_to_license_issue Q8WSF8 22394239 306 DKLHSQANLMRLKSDLFNRSMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4dbn A 3.15 BS01 0JA A 1 A480 K482 E500 L504 T507 L513 I526 T528 W530 C531 G533 F582 G592 D593 F594 A34 K36 E54 L58 T61 L67 I80 T82 W84 C85 G87 F136 G146 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22376051 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 4dbn B 3.15 BS01 0JA B 1 A480 K482 E500 V503 L504 L513 I526 T528 W530 C531 F582 G592 D593 F594 A34 K36 E54 V57 L58 L67 I80 T82 W84 C85 F136 G146 D147 F148 D575 K577 N579 N580 D593 W603 S615 D129 K131 N133 N134 D147 W157 S159 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22376051 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 4dcd A 1.69 BS01 K36 A 1 H40 L127 G128 T142 R143 C147 H161 V162 G163 G164 N165 H44 L131 G132 T146 R147 C151 H165 V166 G167 G168 N169 H40 E71 G145 C147 H44 E75 G149 C151 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue P03300 22915796 202 HHHHGPGFDYAVAMAKRNIVTATTSKGEFTMLGVHDNVAILPTHASPGESIVIDGKEVEILDAKALEDQAGTNLEITIITLKRNEKFRDIRPHIPTQITETNDGVLIVNTSKYPNMYVPVGAVTEQGYLNLGGRQTARTLMYNFPTRAGQCGGVITCTGKVIGMHVGGNGSHGFAAALKRSYFT 4dce A 2.03 BS01 0JF A 1 A1148 K1150 I1171 F1174 V1180 L1196 M1199 G1202 L1256 G1269 D1270 F1271 A48 K50 I71 F74 V80 L96 M99 G102 L156 G169 D170 F171 D1249 A1251 R1253 N1254 D1270 D149 A151 R153 N154 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.174uM remove_due_to_license_issue IC50=384nM Q9UM73 22263917 1501 NPNYSFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVSPSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYG 4dcs A 2.25 BS01 GDP A 1 N185 V186 G187 K188 S189 S190 K236 N294 K295 D297 S329 L331 N162 V163 G164 K165 S166 S167 K207 N265 K266 D268 S300 L302 F20 E26 F18 E24 ? 0005525,0042254,0043022 Kd=8uM remove_due_to_license_issue P50743 23056455 501 KPVVAIVGRPNVGKSTIFNRIAGERISRIYSSAEWLNYDFNLIDTGGPFLAQIRQQAEIAMDEADVIIFMVNGREGVTAADEEVAKILYRTKKPVVLAVNKLMRANIYDFYSLGFGEPYPISGTHGLGLGDLLDAVAEHFKNIPETKYNEEVIQFCLIGRPNVGKSSLVNAMLGEERVIVSNDAVDTSFTYNQQEFVIVDTAGMRKKGKVYETTEKYSVLRALKAIDRSEVVAVVLDGEEGIIEQDKRIAGYAHEAGKAVVIVVNKWDAVDKDESTMKEFEENIRDHFQFLDYAPILFMSALTKKRIHTLMPAIIKASENHSLRVQTNVLNDVIMDAVAMNPTPTHNGSRLKIYYATQVSVKPPSFVVFVNDPELMHFSYERFLENRIRDAFGFEGTPIKIFARAR 4dcx A 2.0 BS01 L2D A 1 Y22 M27 W100 R137 W398 Y402 H416 Y20 M25 W98 R135 W396 Y400 H414 ? 0005515,0015675,0015833,0016020,0016151,0020037,0030288,0042597,0043190,0046914,0050919,0051540,0055052,0055085,0098716,1904680 remove_due_to_license_issue P33590 22526565 630 PDEITTAWPVNVGPLNPHLYTPNQMFAQSMVYEPLVKYQADGSVIPWLAKSWTHSEDGKTWTFTLRDDVKFSNGEPFDAEAAAENFRAVLDNRQRHAWLELANQIVDVKALSKTELQITLKSAYYPFLQELALPRPFRFIAPSQFKNHETMNGIKAPIGTGPWILQESKLNQYDVFVRNENYWGEKPAIKKITFNVIPDPTTRAVAFETGDIDLLYGNEGLLPLDTFARFSQNPAYHTQLSQPIETVMLALNTAKAPTNELAVREALNYAVNKKSLIDNALYGTQQVADTLFAPSVPYANLGLKPSQYDPQKAKALLEKAGWTLPAGKDIREKNGQPLRIELSFIGTDALSKSMAEIIQADMRQIGADVSLIGEEESSIYARQRDGRFGMIFHRTWGAPYDPHAFLSSMRVPSHADFQAQQGLADKPLIDKEIGEVLATHDETQRQALYRDILTRLHDEAVYLPISYISMMVVSKPELGNIPYAPIATEIPFEQIKP 4dcy A 2.0 BS01 L2M A 1 W100 R137 W398 Y402 W98 R135 W396 Y400 ? 0005515,0015675,0015833,0016020,0016151,0020037,0030288,0042597,0043190,0046914,0050919,0051540,0055052,0055085,0098716,1904680 remove_due_to_license_issue P33590 22526565 629 PDEITTAWPVNVGPLNPHLYTPNQMFAQSMVYEPLVKYQADGSVIPWLAKSWTHSEDGKTWTFTLRDDVKFSNGEPFDAEAAAENFRAVLDNRQRHAWLELANQIVDVKALSKTELQITLKSAYYPFLQELALPRPFRFIAPSQFKNHETMNGIKAPIGTGPWILQESKLNQYDVFVRNENYWGEKPAIKKITFNVIPDPTTRAVAFETGDIDLLYGNEGLLPLDTFARFSQNPAYHTQLSQPIETVMLALNTAKAPTNELAVREALNYAVNKKSLIDNALYGTQQVADTLFAPSVPYANLGLKPSQYDPQKAKALLEKAGWTLPAGKDIREKNGQPLRIELSFIGTDALSKSMAEIIQADMRQIGADVSLIGEEESSIYARQRDGRFGMIFHRTWGAPYDPHAFLSSMRVPSHADFQAQQGLADKPLIDKEIGEVLATHDETQRQALYRDILTRLHDEAVYLPISYISMMVVSKPELGNIPYAPIATEIPFEQIKPV 4ddh A 2.07 BS01 MS0 A 1 H44 G46 H47 K160 V187 M195 S196 S197 H42 G44 H45 K158 V185 M193 S194 S195 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=0.48mM remove_due_to_license_issue P9WIL5 23872845 403 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4ddk A 1.75 BS01 0HN A 1 H44 G46 L50 G158 P185 T186 V187 H42 G44 L48 G156 P183 T184 V185 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=5.13mM remove_due_to_license_issue P9WIL5 23872845 401 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4ddl A 2.07 BS02 0JQ A 1 L625 L665 I682 F686 Q716 F719 L184 L224 I241 F245 Q275 F278 3.1.4.17 0004114,0007165,0008081 ic50=4.9nM remove_due_to_license_issue IC50=4.9nM Q9Y233 22365755 1010 TSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4ddm A 1.83 BS01 0HO A 1 P38 T39 M40 H47 Q164 P36 T37 M38 H45 Q162 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=3.48mM remove_due_to_license_issue P9WIL5 23872845 406 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4dds A 1.36 BS01 0J7 A 1 S70 N104 Y105 S130 N132 P167 T168 N170 T171 T235 G236 S237 G238 S42 N76 Y77 S102 N104 P139 T140 N142 T143 T207 G208 S209 G210 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=9.7uM remove_due_to_license_issue Q9L5C8 22296601 301 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4dds A 1.36 BS02 0J7 A 2 G143 G146 G115 G118 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=9.7uM remove_due_to_license_issue Q9L5C8 22296601 302 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4dds A 1.36 BS03 0J7 A 3 N104 Y105 T216 N76 Y77 T188 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=9.7uM remove_due_to_license_issue Q9L5C8 22296601 303 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4ddy A 1.36 BS01 DN6 A 1 N104 Y105 S130 N132 P167 N170 T171 T235 G236 S237 D240 N76 Y77 S102 N104 P139 N142 T143 T207 G208 S209 D211 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=2.4uM remove_due_to_license_issue Q9L5C8 22296601 301 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4ddy A 1.36 BS02 DN6 A 2 N104 Y105 T216 S237 N76 Y77 T188 S209 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=2.4uM remove_due_to_license_issue Q9L5C8 22296601 302 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4ddy A 1.36 BS03 DN6 A 3 T51 N54 R191 Q192 G196 T24 N27 R163 Q164 G168 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=2.4uM remove_due_to_license_issue Q9L5C8 22296601 303 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de0 A 1.12 BS01 0JB A 1 N104 Y105 S130 N132 N170 T235 G236 S237 G238 D240 N79 Y80 S105 N107 N145 T210 G211 S212 G213 D214 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.3uM remove_due_to_license_issue Q9L5C8 22296601 300 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de1 A 1.26 BS01 0J6 A 1 N104 Y105 S130 N132 P167 N170 T235 G236 S237 D240 N79 Y80 S105 N107 P142 N145 T210 G211 S212 D214 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.1uM remove_due_to_license_issue Q9L5C8 22296601 301 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de2 A 1.4 BS01 DN3 A 1 N104 Y105 S130 N132 P167 N170 T235 G236 S237 D240 N76 Y77 S102 N104 P139 N142 T207 G208 S209 D211 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=76uM remove_due_to_license_issue Q9L5C8 22296601 301 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de2 A 1.4 BS02 DN3 A 2 K82 Q83 L142 G147 A154 K54 Q55 L114 G119 A126 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=76uM remove_due_to_license_issue Q9L5C8 22296601 302 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de3 A 1.44 BS01 DN8 A 1 N104 Y105 S130 N132 P167 N170 T235 G236 S237 G238 D240 N76 Y77 S102 N104 P139 N142 T207 G208 S209 G210 D211 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3uM remove_due_to_license_issue Q9L5C8 22296601 301 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de3 A 1.44 BS02 DN8 A 2 N104 Y105 S237 N76 Y77 S209 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3uM remove_due_to_license_issue Q9L5C8 22296601 302 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de3 A 1.44 BS03 DN8 A 3 A79 A150 F151 A154 A51 A122 F123 A126 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3uM remove_due_to_license_issue Q9L5C8 22296601 303 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de3 A 1.44 BS04 DN8 A 4 I173 D176 I145 D148 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3uM remove_due_to_license_issue Q9L5C8 22296601 304 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de3 A 1.44 BS05 DN8 A 5 R191 Q192 R163 Q164 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3uM remove_due_to_license_issue Q9L5C8 22296601 305 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de3 A 1.44 BS06 DN8 A 6 S274 R276 S244 R246 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=3uM remove_due_to_license_issue Q9L5C8 22296601 306 AVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4de5 A 2.25 BS01 0JD A 1 P38 T39 M40 H47 Q164 P36 T37 M38 H45 Q162 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=670uM remove_due_to_license_issue P9WIL5 23872845 401 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4de7 A 3.0 BS01 UDP A 1 P50 A51 L52 E54 S81 K114 P30 A31 L32 E34 S61 K94 2.4.1.266 0000287,0006011,0016757,0016758,0042803,0046872 remove_due_to_license_issue P9WMW9 22637481 401 PLDTTWHRPGWTIGELEAAKAGRTISVVLPALNEEATIESVIDSISPLVDGLVDELIVLDSGSTDDTEIRAIASGARVVSREQALPEVPVRPGKGEALWRSLAATSGDIVVFIDSDLINPHPLFVPWLVGPLLTGEGIQLVKSFYRGGRVTELVARPLLAALRPELGCVLQPLSGEYAASRELLTSLPFAPGYGVEIGLLIDTFDRLGLDAIAQVNLGVRAHRNRPLDELGAMSRQVIATLLSRCGIPDSGVGLTQFLPGDYTRHTWPVSLVDRPPMKVMR 4dea A 2.45 BS01 NHI A 1 R137 L139 G140 V147 A213 G216 R220 L263 R14 L16 G17 V24 A90 G93 R97 L140 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=256nM remove_due_to_license_issue IC50=256nM O14965 22803810 504 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 4deb A 3.05 BS01 NHJ A 1 R137 L139 V147 A213 G216 R220 L263 R13 L15 V23 A89 G92 R96 L139 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=226.0nM O14965 22803810 501 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4ded A 3.05 BS01 NHU A 1 R137 L139 G140 V147 A160 K162 A213 G216 R220 L263 R14 L16 G17 V24 A37 K39 A90 G93 R97 L140 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=38.2nM O14965 22803810 501 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4deg A 2.0 BS01 0JJ A 1 I1084 A1108 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I33 A51 M100 D104 R148 M151 A161 D162 Y170 D1204 A1206 R1208 N1209 D1222 A1243 D144 A146 R148 N149 D162 A183 2.7.10.1 0004672,0004713,0005524,0006468 ic50=6nM remove_due_to_license_issue IC50=3nM, Ki=3.2nM P08581 22595176 1401 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4deh A 2.0 BS01 0JK A 1 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 A50 Y99 M100 D104 R148 M151 A161 D162 Y170 D1204 A1206 R1208 N1209 D1222 A1243 D144 A146 R148 N149 D162 A183 2.7.10.1 0004672,0004713,0005524,0006468 ic50=612nM remove_due_to_license_issue IC50=612nM P08581 22595176 1401 IDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4dei A 2.05 BS01 0JL A 1 I1084 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I32 A52 Y100 M101 D105 R149 M152 A162 D163 Y171 D1204 A1206 R1208 N1209 D1222 A1243 D145 A147 R149 N150 D163 A184 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=2nM P08581 22595176 1401 IDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDKIHCAVKSLNRIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4del A 1.58 BS03 PGH A 1 D95 H96 H212 G213 H252 G253 S255 N274 D276 T277 D94 H95 H211 G212 H251 G252 S254 N273 D275 T276 D95 H96 E169 H212 H252 N274 D94 H95 E168 H211 H251 N273 4.1.2.13 0004332,0005576,0005829,0005886,0005975,0006096,0008270,0009274,0016829,0016832,0035375,0046872 Kd=21.1nM remove_due_to_license_issue P9WQA3 23298222 404 PIATPEVYAEMLGQAKQNSYAFPAINCTSSETVNAAIKGFADAGSDGIIQFSTGGAEFGSGLGVKDMVTGAVALAEFTHVIAAKYPVNVALHTDHCPKDKLDSYVRPLLAISAQRVSKGGNPLFQSHMWDGSAVPIDENLAIAQELLKAAAAAKIILEIEIGVVGGEEDGVANEINEKLYTSPEDFEKTIEALGAGEHGKYLLAATFGNVHGVYKPGNVKLRPDILAQGQQVAAAKLGLPADAKPFDFVFHGGSGSLKSEIEEALRYGVVKMNVDTDTQYAFTRPIAGHMFTNYDGVLKVDGEVGVKKVYDPRSYLKKAEASMSQRVVQACNDLHCAGKSLTHHH 4dem F 1.85 BS01 YS4 F 1 F113 D117 R126 T181 E182 Q185 K214 D257 K271 F92 D96 R105 T160 E161 Q164 K193 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=28nM remove_due_to_license_issue IC50=28nM P14324 22390415 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4der A 1.9 BS01 AGI A 1 K15 A108 L110 K6 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.49uM remove_due_to_license_issue IC50=653nM, Kd=250nM P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4der B 1.9 BS01 AGI B 1 K15 L17 L110 K6 L8 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.49uM remove_due_to_license_issue IC50=653nM, Kd=250nM P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4des A 1.75 BS01 57D A 1 K15 A108 L110 T119 V121 K6 A99 L101 T110 V112 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=1.4uM remove_due_to_license_issue P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4des B 1.75 BS01 57D B 1 K15 A108 L110 V121 K6 A99 L101 V112 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=1.4uM remove_due_to_license_issue P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4det B 2.05 BS01 KMP B 1 L17 L110 L8 L96 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=2.1uM remove_due_to_license_issue P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANRYTIAALLSPYSYSTTAVVT 4deu A 1.599 BS01 NAR A 1 K15 L17 A108 S117 T119 K7 L9 A100 S109 T111 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=2.29uM remove_due_to_license_issue P02766 22842046 205 ACPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4deu B 1.599 BS01 NAR B 1 K15 A108 L110 K6 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=2.29uM remove_due_to_license_issue P02766 22842046 202 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4dew A 1.899 BS01 LU2 A 1 K15 L17 S117 K6 L8 S108 ? Kd=0.1uM remove_due_to_license_issue IC50=7000nM, Kd=70nM P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4dew B 1.899 BS01 LU2 B 1 K15 L17 K6 L8 ? Kd=0.1uM remove_due_to_license_issue IC50=7000nM, Kd=70nM P02766 22842046 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDPRRYTIAALLSPYSYSTTAVVTN 4dfb A 1.95 BS01 KAN A 1 D197 D220 E235 W271 D197 D220 E235 W269 ? 0000166,0016301,0046872 remove_due_to_license_issue O68183 22195561 401 MRTYTFDQVEKAIEQLYPDFTINTIEISGEGNDCIAYEINRDFIFKFPKHSRGSTNLFNEVNILKRIHNKLPLPIPEVVFTGMPSETYQMSFAGFTKIKGVPLTPLLLNNLPKQSQNQAAKDLARFLSELHSINISGFKSNLVLDFREKINEDNKKIKKLLSRELKGPQMKKVDDFYRDILENEIYFKYYPCLIHNDFSSDHILFDTEKNTICGIIDFGDAAISDPDNDFISLMEEEYGMEFVSKILNHYKHKDIPTVLEKYRMKEKYWSFEKIIYGKEYGYMDWYEEGLNEIRSIK 4dff B 2.11 BS01 0JP B 1 F696 M713 Q726 F729 F213 M222 Q234 F237 3.1.4.17 0004114,0007165,0008081 Ki=35nM remove_due_to_license_issue Ki=35nM Q9Y233 22377514 801 EIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDPIPMMDRKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4dfg A 1.23 BS01 0JV B 1 R8 D25 A28 D30 V82 R8 D25 A28 D30 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 22364812 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4dfg B 1.23 BS01 0JV B 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.8pM remove_due_to_license_issue P03367 22364812 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4dfl A 1.98 BS01 0K0 A 1 L377 A400 M448 M450 A451 G454 N499 L501 D512 L15 A33 M75 M77 A78 G81 N126 L128 D139 D494 A496 R498 N499 D512 K533 D121 A123 R125 N126 D139 K160 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.67uM remove_due_to_license_issue P43405 22425453 701 VYLDRKLLTLEDKELGSGTVKKGYYQMVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNE 4dfn A 2.48 BS01 0K1 A 1 L377 F382 V385 A400 M448 A451 P455 K458 L501 D512 L15 F20 V23 A38 M81 A84 P88 K91 L134 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.02uM remove_due_to_license_issue IC50=20nM P43405 22425453 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNE 4dfu A 1.98 BS02 QUE A 1 I44 K46 K97 I98 G100 P102 I216 D217 I42 K44 K95 I96 G98 P100 I214 D215 ? 0000166,0016301,0046872 Ki=25.1uM remove_due_to_license_issue O68183 22195561 402 TYTFDQVEKAIEQLYPDFTINTIEISGEGNDCIAYEINRDFIFKFPKHSRGSTNLFNEVNILKRIHNKLPLPIPEVVFTGMPSETYQMSFAGFTKIKGVPLTPLLLNNLPKQSQNQAAKDLARFLSELHSINISGFKSNLVLDFREKINEDNKKIKKLLSRELKGPQMKKVDDFYRDILENEIYFKYYPCLIHNDFSSDHILFDTEKNTICGIIDFGDAAISDPDNDFISLMEDDEEYGMEFVSKILNHYKHKDIPTVLEKYRMKEKYWSFEKIIYGKEYGYMDWYEEGLNEIRSI 4dfu A 1.98 BS03 QUE B 1 R52 T55 T87 Y88 Q89 R50 T53 T85 Y86 Q87 ? 0000166,0016301,0046872 Ki=25.1uM remove_due_to_license_issue O68183 22195561 401 TYTFDQVEKAIEQLYPDFTINTIEISGEGNDCIAYEINRDFIFKFPKHSRGSTNLFNEVNILKRIHNKLPLPIPEVVFTGMPSETYQMSFAGFTKIKGVPLTPLLLNNLPKQSQNQAAKDLARFLSELHSINISGFKSNLVLDFREKINEDNKKIKKLLSRELKGPQMKKVDDFYRDILENEIYFKYYPCLIHNDFSSDHILFDTEKNTICGIIDFGDAAISDPDNDFISLMEDDEEYGMEFVSKILNHYKHKDIPTVLEKYRMKEKYWSFEKIIYGKEYGYMDWYEEGLNEIRSI 4dgg A 2.65 BS01 I76 A 1 V281 A293 F307 A311 T338 M341 L393 D404 V26 A38 F52 A56 T83 M86 L138 D149 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F152 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 23143416 601 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4dgm A 1.65 BS01 AGI A 1 V45 I66 K68 F113 V116 N118 M163 I174 D175 V39 I60 K62 F107 V110 N112 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=1.2uM remove_due_to_license_issue P28523 22794353 406 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLMGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAEN 4dgn A 1.75 BS01 LU2 A 1 V45 I66 K68 F113 V116 N118 M163 I174 D175 V39 I60 K62 F107 V110 N112 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=0.35uM remove_due_to_license_issue P28523 22794353 401 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAEN 4dgr A 1.551 BS04 3LV A 1 R118 E119 D151 R152 W178 I222 R224 E227 E277 R292 R371 Y406 R38 E39 D71 R72 W99 I143 R145 E148 E198 R213 R291 Y325 D151 E277 R292 R371 Y406 D71 E198 R213 R291 Y325 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=9.1uM remove_due_to_license_issue P03472 22559154 488 IRDFNNLTKGLCTINSWHIYGKDNAVRIGEDSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKTRMSICISGPNNNASAVIWYNRRPVTEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPAETRIYYFKEGKILKWEPLAGTAKHIEECSCYGERAEITCTCRDNWQGSNRPVIRIDPVAMTHTSQYICSPVLTDNPRPNDPTVGKCNDPYPGNNNNGVKGFSYLDGVNTWLGRTISIASRSGYEMLKVPNALTDDKSKPTQGQTIVLNTDWSGYSGSFMDYWAEGECYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWDWPDGAKIEYFL 4dh6 A 2.5 BS01 0KN A 1 L30 D32 G34 P70 Y71 T72 F108 W115 D228 G230 T329 V332 L32 D34 G36 P72 Y73 T74 F110 W117 D219 G221 T311 V314 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=16.8nM remove_due_to_license_issue IC50=26nM P56817 22468639 411 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQATPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4dhf A 2.8 BS01 0K6 A 1 R137 L139 G140 V147 A213 L215 G216 T217 L263 R10 L12 G13 V20 A86 L88 G89 T90 L136 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T161 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=28nM O14965 22607669 401 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 4dhl A 2.3 BS03 0K7 A 1 D164 N201 H202 H295 H296 H323 H325 Y365 D157 N194 H195 H288 H289 H316 H318 Y358 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D128 D157 Y160 N194 H195 H279 H288 H289 H316 H318 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 Ki=33uM remove_due_to_license_issue P80366 22943065 503 NRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDDS 4dhl D 2.3 BS03 0K7 D 1 N201 H202 H296 H323 H325 N194 H195 H289 H316 H318 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D128 D157 Y160 N194 H195 H279 H288 H289 H316 H318 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 Ki=33uM remove_due_to_license_issue P80366 22943065 503 NRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDD 4dhm A 1.7 BS02 0KB A 1 G53 R56 A57 R60 R129 Y130 L174 N175 G57 R60 A61 R64 R126 Y127 L171 N172 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 308 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dhn A 1.8 BS02 0KC A 1 R56 R60 R129 Y130 L174 N175 V178 R60 R64 R126 Y127 L171 N172 V175 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 307 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dho A 1.7 BS02 Y09 A 1 G53 R56 R60 R129 Y130 L174 N175 V178 G57 R60 R64 R126 Y127 L171 N172 V175 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 308 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dhp A 1.75 BS02 Y07 A 1 G53 R56 R60 R129 Y130 L174 N175 V178 G57 R60 R64 R126 Y127 L171 N172 V175 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 309 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dhq A 1.75 BS02 Y06 A 1 G53 R56 A57 R60 R129 Y130 L174 N175 V178 G57 R60 A61 R64 R129 Y130 L174 N175 V178 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 309 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNEEKGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dhr A 1.4 BS02 Y04 A 1 G53 R56 R60 R129 Y130 L174 N175 G57 R60 R64 R126 Y127 L171 N172 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 309 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dhs A 1.74 BS02 Y03 A 1 G53 R56 A57 R60 R129 Y130 L174 N175 V178 G57 R60 A61 R64 R126 Y127 L171 N172 V175 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 307 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dht A 1.8 BS02 0KG A 1 R56 R60 R129 Y130 L174 N175 R60 R64 R126 Y127 L171 N172 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 23939230 306 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4dhu A 1.67 BS02 0KH A 1 G53 R56 A57 R60 R129 Y130 L174 N175 G57 R60 A61 R64 R126 Y127 L171 N172 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue IC50=5000nM P31947 23939230 309 AMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 4di2 A 2.0 BS01 0K9 A 1 G11 Q12 G13 L30 D32 G34 P70 Y71 T72 F108 I110 Y198 D228 G230 T329 V332 G17 Q18 G19 L36 D38 G40 P76 Y77 T78 F114 I116 Y194 D224 G226 T319 V322 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=5.5nM remove_due_to_license_issue P56817 22468684 501 KKGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4dij A 1.9 BS01 BLF A 1 L54 G58 I61 F86 V93 H96 I99 Y100 L37 G41 I44 F69 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 ic50=0.03uM remove_due_to_license_issue Q00987 22507962 201 QIPASEQETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4dij A 1.9 BS02 BLF B 1 M62 Y67 M45 Y50 2.3.2.27 0005634,0043066,0051726 ic50=0.03uM remove_due_to_license_issue Q00987 22507962 201 QIPASEQETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4dj7 A 2.81 BS01 GAL H 1 E181 Q217 E181 Q217 ? 0019031,0019064,0046789 remove_due_to_license_issue Q6VMK1 22674977 2 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNVPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKETMGFTYSGIRTNGTTSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKDPALIIWGIHHSGSTTEQTKLYGSGNKLITVGSSNYQQSFVPSPGARPQVNGQSGRIDFHWLILNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSEVQVDANCEGDCYHSGGTIISNLPFQNINSRAVGKCPRYVKQESLLLATGMKNVPE 4dj7 A 2.81 BS02 SIA H 1 Y88 T125 T126 S127 W142 H174 E181 Q217 Y88 T125 T126 S127 W142 H174 E181 Q217 ? 0019031,0019064,0046789 remove_due_to_license_issue Q6VMK1 22674977 3 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNVPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKETMGFTYSGIRTNGTTSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKDPALIIWGIHHSGSTTEQTKLYGSGNKLITVGSSNYQQSFVPSPGARPQVNGQSGRIDFHWLILNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSEVQVDANCEGDCYHSGGTIISNLPFQNINSRAVGKCPRYVKQESLLLATGMKNVPE 4djh A 2.9 BS01 JDC A 1 Q115 V134 D138 M142 V230 W287 I294 G319 Y320 Q61 V80 D84 M88 V176 W392 I399 G419 Y420 E1011 D1020 E217 D226 ?,3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P41145 22437504 1300 SPAIPVIITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTVYLMNSWPFGDVLCKIVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFPDDDYSWWDLFMKICVFIFAFVIPVLIIIVCYTLMILRLKSVRLLSGNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYREKDRNLRRITRLVLVVVAVFVVCWTPIHIFILVEALGSAALSSYYFCIALGYTNSSLNPILYAFLDENFKRCFRDFCFP 4djo A 1.78 BS01 MK5 A 1 D25 G27 A28 D29 I47 G48 I50 D25 G27 A28 D29 I47 G48 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.003nM remove_due_to_license_issue Q90K99 22708897 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djo B 1.78 BS01 MK5 A 1 D25 A28 D30 I50 P81 V82 D25 A28 D30 I50 P81 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 22708897 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djp A 1.4 BS01 M73 A 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 D25 G27 A28 D29 D30 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.028nM remove_due_to_license_issue Q90K99 22708897 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djp B 1.4 BS01 M73 A 1 D25 A28 D30 I50 P81 V82 I84 D25 A28 D30 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 22708897 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djq A 1.4 BS01 M86 A 1 D25 G27 A28 D29 G48 I50 D25 G27 A28 D29 G48 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.048nM remove_due_to_license_issue Q90K99 22708897 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djq B 1.4 BS01 M86 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 22708897 200 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djr A 1.55 BS01 0KJ A 1 D25 G27 D29 G48 I50 V82 D25 G27 D29 G48 I50 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.003nM remove_due_to_license_issue Q90K99 22708897 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4djr B 1.55 BS01 0KJ A 1 D25 A28 D30 G48 P81 V82 D25 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90K99 22708897 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4dju A 1.8 BS01 0KK A 1 L91 D93 Y132 F169 I179 D289 G291 L34 D36 Y75 F112 I122 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=3.6uM remove_due_to_license_issue P56817 22390835 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4djv A 1.73 BS01 0KM A 1 Q73 G74 L91 D93 S96 Y132 W137 F169 I171 W176 I179 D289 S290 G291 T292 Q16 G17 L34 D36 S39 Y75 W80 F112 I114 W119 I122 D232 S233 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=0.19uM remove_due_to_license_issue IC50=392nM P56817 22390835 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4djw A 1.9 BS01 0KP A 1 G72 G74 L91 D93 S96 Y132 F169 I171 W176 I179 D289 G291 G15 G17 L34 D36 S39 Y75 F112 I114 W119 I122 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=0.53uM remove_due_to_license_issue IC50=1680nM P56817 22390835 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4djx A 1.5 BS01 0KQ A 1 G72 Q73 G74 D93 S96 Y132 F169 W176 D289 G291 T292 G15 Q16 G17 D36 S39 Y75 F112 W119 D232 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=59nM remove_due_to_license_issue P56817 22390835 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4djy A 1.86 BS01 0KR A 1 S71 Q73 G74 D93 S96 Y132 F169 I179 D289 S290 G291 T292 S14 Q16 G17 D36 S39 Y75 F112 I122 D232 S233 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=5.4nM remove_due_to_license_issue P56817 22390835 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4dk5 A 2.95 BS01 0KO A 1 K802 M804 A805 K833 D841 Y867 V882 K890 M953 I963 D964 K560 M562 A563 K591 D599 Y625 V640 K648 M711 I721 D722 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=8nM P48736 22548365 1204 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNPIALPKHMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 4dk7 A 2.45 BS02 0KS A 1 L274 A275 S278 T316 F329 F340 H435 L449 W457 L50 A51 S54 T92 F105 F116 H211 L225 W233 ? 0003677,0004879,0006629 ic50=0.02uM remove_due_to_license_issue P55055 22406115 501 HMQLTAAQELMIQQLVAAQLQCNKRSFSKVTPWPLSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 4dk8 A 2.75 BS02 0KT A 1 F271 M312 T316 F329 H435 W457 F46 M87 T91 F104 H210 W232 ? 0003677,0004879,0006629 remove_due_to_license_issue P55055 22406115 501 MQLTAAQELMIQQLVAAQLQCNKRSFSKVTPWPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWD 4dko A 1.981 BS01 0LM A 1 S256 T257 E370 S375 F376 F382 N425 W427 G429 G473 S140 T141 E231 S236 F237 F243 N272 W274 G276 G320 ? 0019031 Kd=0.3uM remove_due_to_license_issue Q0ED31 22497421 513 VWKDADTTLFCASDAKAHETEVHNVWATHACVPTDPNPQEIHLENVTENFNMWKNNMVEQMQEDVISLWDQSLQPCVKLTGGSVIKQACPKISFDPIPIHYCTPAGYVILKCNDKNFNGTGPCKNVSSVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNKSVEINCTRPSNGDIRKAYCEINGTKWNKVLKQVTEKLKEHFNNKTIIFQPPSGGDLEITMHSFNCRGEFFYCNTTQLFNNTCINGTITLPCKIKQIINMWQGTGQAMYAPPIDGKINCVSNITGILLTRDGGANNTSNETFRPGGGNIKDNWRSELYKYKVVQIE 4dkp A 1.7978 BS01 0LL A 1 S256 T257 E370 S375 F376 F382 I424 N425 W427 S140 T141 E231 S236 F237 F243 I271 N272 W274 ? 0019031 Kd=1.9uM remove_due_to_license_issue Q0ED31 22497421 513 VWKDADTTLFCASDAKAHETEVHNVWATHACVPTDPNPQEIHLENVTENFNMWKNNMVEQMQEDVISLWDQSLQPCVKLTGGSVIKQACPKISFDPIPIHYCTPAGYVILKCNDKNFNGTGPCKNVSSVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNKSVEINCTRPSNGDIRKAYCEINGTKWNKVLKQVTEKLKEHFNNKTIIFQPPSGGDLEITMHSFNCRGEFFYCNTTQLFNNTCINGTITLPCKIKQIINMWQGTGQAMYAPPIDGKINCVSNITGILLTRDGGANNTSNETFRPGGGNIKDNWRSELYKYKVVQIE 4dkq A 1.888 BS01 0LK A 1 V255 S256 E370 S375 F376 F382 I424 N425 W427 G473 N474 V139 S140 E231 S236 F237 F243 I271 N272 W274 G320 N321 ? 0019031 Kd=0.25uM remove_due_to_license_issue Q0ED31 22497421 613 VWKDADTTLFCASDAKAHETEVHNVWATHACVPTDPNPQEIHLENVTENFNMWKNNMVEQMQEDVISLWDQSLQPCVKLTGGSVIKQACPKISFDPIPIHYCTPAGYVILKCNDKNFNGTGPCKNVSSVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNKSVEINCTRPSNGDIRKAYCEINGTKWNKVLKQVTEKLKEHFNNKTIIFQPPSGGDLEITMHSFNCRGEFFYCNTTQLFNNTCINGTITLPCKIKQIINMWQGTGQAMYAPPIDGKINCVSNITGILLTRDGGANNTSNETFRPGGGNIKDNWRSELYKYKVVQIE 4dkr A 1.8 BS01 0LJ A 1 S256 T257 D368 E370 I371 S375 F376 N425 W427 G429 G473 S140 T141 D229 E231 I232 S236 F237 N272 W274 G276 G320 ? 0019031 Kd=0.3uM remove_due_to_license_issue Q0ED31 22497421 513 VWKDADTTLFCASDAKAHETEVHNVWATHACVPTDPNPQEIHLENVTENFNMWKNNMVEQMQEDVISLWDQSLQPCVKLTGGSVIKQACPKISFDPIPIHYCTPAGYVILKCNDKNFNGTGPCKNVSSVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNKSVEINCTRPSNGDIRKAYCEINGTKWNKVLKQVTEKLKEHFNNKTIIFQPPSGGDLEITMHSFNCRGEFFYCNTTQLFNNTCINGTITLPCKIKQIINMWQGTGQAMYAPPIDGKINCVSNITGILLTRDGGANNTSNETFRPGGGNIKDNWRSELYKYKVVQIE 4dld A 2.0 BS01 TZG A 1 Y16 Y61 P88 L89 T90 R95 S141 T142 S173 E190 S193 Y216 Y14 Y59 P86 L87 T88 R93 S139 T140 S171 E188 S191 Y214 ? 0015276,0016020 Ki=1.5uM remove_due_to_license_issue Ki=3000nM P22756 22407805 301 NRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 4dli A 1.91 BS01 IRG A 1 E192 L195 W197 L246 I250 S252 A255 D294 E172 L175 W177 L226 I230 S232 A235 D274 D150 K152 N155 D168 T185 D142 K144 N147 D160 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=2.4uM remove_due_to_license_issue Q16539 22768308 401 RPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4dli A 1.91 BS02 IRG A 2 M194 L195 H228 S254 A255 Y258 M174 L175 H208 S234 A235 Y238 D150 K152 N155 D168 T185 D142 K144 N147 D160 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=2.4uM remove_due_to_license_issue Q16539 22768308 402 RPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4dlj A 2.6 BS01 6RG A 1 E192 L195 W197 L246 I250 S252 A255 I259 L291 D294 E174 L177 W179 L228 I232 S234 A237 I241 L273 D276 D150 K152 N155 D168 T185 D146 K148 N151 D164 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 22768308 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4dlj A 2.6 BS02 6RG A 2 A51 K53 T106 M109 L167 D168 A48 K50 T103 M106 L163 D164 D150 K152 N155 D168 T185 D146 K148 N151 D164 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 22768308 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4dmn A 2.45 BS01 0L9 A 1 T124 A128 W132 T70 A74 W78 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=2.3uM remove_due_to_license_issue IC50=4e+2nM P12497 22437836 305 DCSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGIGGYSAGERIVDIIATDIQ 4dmw A 2.5 BS02 UDP A 1 V100 W101 I102 L264 S268 D285 S517 V99 W100 I101 L261 S265 D282 S514 2.4.1.-,3.4.22.- 0016757 remove_due_to_license_issue P16154 22747490 602 SLISKEELIKLAYSIRPRENEYKTILTNLDEYNKLTTNNNENKYLQLKKLNESIDVFMNKYKTSSRNRALSNLKKDILKEVILIKNSNTSPVEKNLHFVWIGGEVSDIALEYIKQWADINAEYNIKLWYDSEAFLVNTLKKAIVESSTTEALQLLEEEIQNPQFDNMKFYKKRMEFIYDRQKRFINYYKSQINKVPTIDDIIKSHLVSEYNRDETVLESYRTNSLRKINSNHGIDIRANSLFTEQELLNIYSQELLNRGNLAAASDIVRLLALKNFGGVYLDVDMLPGIHSDLFKTISRPSSIGLDRWEMIKLEAIMKYKKYINNYTSENFDKLDQQLKDNFKLIIESKSEKSEIFSKLENLNVSDLEIKIAFALGSVINQALISKQGSYLTNLVIEQVKNRYQFLNQHLNPAIESDNNFTDTTKIFHDSLFNSATAENSMFLTKIAPYLQVGFMPEARSTISLSGPGAYASAYYDFINLQENTIEKTLKASDLIEFKFPENNLSQLTEQEINSLWSFDQASAKYQFEKYVRDYT 4dmy A 1.63 BS01 0LC A 1 G23 C25 N60 G64 G65 G66 Y67 N161 H162 G23 C25 N60 G64 G65 G66 Y67 N161 H162 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 22742641 301 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 4dn0 A 2.3 BS01 C2E A 1 R161 R367 D370 G395 G398 Y399 R402 R4 R191 D194 G219 G222 Y223 R226 ? Kd=1.9uM (22605337) Kd=1.9uM remove_due_to_license_issue A0A0H2ZD98 22605337 501 QSLRSSLLGLRQLLRELPGDEAPLDALAETVLALLAQYGSLRIAGLYRVRHDRTPEPQPLATLGEMPVLDADDLLVRTCLERGELVSVRQELALQVCVPLVDTDGRILALLAVEQMPFFVFNERTFSLLAILAGHIADLLQDIDAQRFSQYLKRSLLDARDHGLPACLYAFELTDARYGEEVQRLLEGSQRGLDVQLRLRNDEGRRVLLVLLPLTSAEGSQGYLQRLRILFAERFGQARELESLGVRIRQYELDAGNDRQALGHFLFNECGLNDQQVAV 4dn0 A 2.3 BS02 C2E A 2 R161 L165 Q366 R367 G368 R402 R4 L8 Q190 R191 G192 R226 ? Kd=1.9uM (22605337) Kd=1.9uM remove_due_to_license_issue A0A0H2ZD98 22605337 502 QSLRSSLLGLRQLLRELPGDEAPLDALAETVLALLAQYGSLRIAGLYRVRHDRTPEPQPLATLGEMPVLDADDLLVRTCLERGELVSVRQELALQVCVPLVDTDGRILALLAVEQMPFFVFNERTFSLLAILAGHIADLLQDIDAQRFSQYLKRSLLDARDHGLPACLYAFELTDARYGEEVQRLLEGSQRGLDVQLRLRNDEGRRVLLVLLPLTSAEGSQGYLQRLRILFAERFGQARELESLGVRIRQYELDAGNDRQALGHFLFNECGLNDQQVAV 4do3 A 2.25 BS02 0LA A 1 L192 F381 F432 M436 T488 W531 L160 F349 F400 M404 T456 W499 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 ic50=74uM remove_due_to_license_issue IC50=32000nM P97612 23240907 602 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMLSFDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSAGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNSMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAISYTVLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQ 4do4 A 1.4 BS01 DJN A 1 W33 D78 D79 C127 K154 D156 S188 R213 D217 W16 D61 D62 C110 K137 D139 S171 R196 D200 D156 D217 D139 D200 3.2.1.49 0004553,0004557,0005737,0005764,0005975,0006629,0008456,0009311,0016020,0016052,0016139,0016798,0019377,0042803,0070062 remove_due_to_license_issue P17050 23045655 510 LDNGLLQTPPMGWLAWERFRCNINCDEDPKNCISEQLFMEMADRMAQDGWRDMGYTYLNIDDCWIGGRDASGRLMPDPKRFPHGIPFLADYVHSLGLKLGIYADMGNFTCMGYPGTTLDKVVQDAQTFAEWKVDMLKLDGCFSTPEERAQGYPKMAAALNATGRPIAFSCSWPAYEGGLPPRVQYSLLADICNLWRNYDDIQDSWWSVLSILNWFVEHQDILQPVAGPGHWNDPDMLLIGNFGLSLEQSRAQMALWTVLAAPLLMSTDLRTISAQNMDILQNPLMIKINQDPLGIQGRRIHKEKSLIEVYMRPLSNKASALVFFSCRTDMPYRYHSSLGQLNFTGSVIYEAQDVYSGDIISGLRDETNFTVIINPSGVVMWYLYPIK 4do5 A 1.51 BS01 DGJ A 1 W33 D78 D79 C127 K154 D156 R213 D217 W16 D61 D62 C110 K137 D139 R196 D200 D156 D217 D139 D200 3.2.1.49 0004553,0004557,0005737,0005764,0005975,0006629,0008456,0009311,0016020,0016052,0016139,0016798,0019377,0042803,0070062 remove_due_to_license_issue P17050 23045655 509 LDNGLLQTPPMGWLAWERFRCNINCDEDPKNCISEQLFMEMADRMAQDGWRDMGYTYLNIDDCWIGGRDASGRLMPDPKRFPHGIPFLADYVHSLGLKLGIYADMGNFTCMGYPGTTLDKVVQDAQTFAEWKVDMLKLDGCFSTPEERAQGYPKMAAALNATGRPIAFSCSWPAYEGGLPPRVQYSLLADICNLWRNYDDIQDSWWSVLSILNWFVEHQDILQPVAGPGHWNDPDMLLIGNFGLSLEQSRAQMALWTVLAAPLLMSTDLRTISAQNMDILQNPLMIKINQDPLGIQGRRIHKEKSLIEVYMRPLSNKASALVFFSCRTDMPYRYHSSLGQLNFTGSVIYEAQDVYSGDIISGLRDETNFTVIINPSGVVMWYLYPIK 4dpf A 1.8 BS01 0LG A 1 G59 Q60 L78 D80 G82 Y119 T120 Q121 I158 D276 G278 T279 T280 N281 R283 G13 Q14 L32 D34 G36 Y73 T74 Q75 I112 D218 G220 T221 T222 N223 R225 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=400nM remove_due_to_license_issue P56817 22698785 500 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4dpi A 1.9 BS01 0N1 A 1 G59 Q60 G61 L78 D80 G82 Y119 T120 Q121 D276 G278 T279 T280 A383 G13 Q14 G15 L32 D34 G36 Y73 T74 Q75 D217 G219 T220 T221 A324 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=78nM remove_due_to_license_issue P56817 22698785 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHHDEFRTAAVEGPFVTLDMEDCGYN 4dpt B 2.191 BS01 FM0 B 1 A14 Y18 K21 S139 G140 S141 R144 R193 M196 D283 A13 Y17 K20 S138 G139 S140 R143 R188 M191 D278 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 remove_due_to_license_issue Q9FD73 22734632 401 VKSGKARAHTNIALIKYWGKADETYIIPMNNSLSVTLDRFYTETKVTFDPDFTEDCLILNGNEVNAKEKEKIQNYMNIVRDLAGNRLHARIESENYVPTAAGLASSASAYAALAAACNEALSLNLSDTDLSRLARRGSGSASRSIFGGFAEWEKGHDDLTSYAHGINSNGWEKDLSMIFVVINNVSSRSGMSLTRDTSRFYQYWLDHVDEDLNEAKEAVKNQDFQRLGEVIEANGLRMHATNLGAQPPFTYLVQESYDAMAIVEQCRKANLPCYFTMDAGPNVKVLVEKKNKQAVMEQFLKVFDESKIIASDIISSGVEIIK 4dpu A 1.9 BS01 FM0 A 1 A14 Y18 K21 S139 G140 S141 R144 R193 D283 A284 A17 Y21 K24 S142 G143 S144 R147 R196 D286 A287 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 remove_due_to_license_issue Q9FD73 22734632 401 TGSMVKSGKARAHTNIALIKYWGKADETYIIPMNNSLSVTLDRFYTETKVTFDPDFTEDCLILNGNEVNAKEKEKIQNYMNIVRDLAGNRLHARIESENYVPTAAGLASSASAYAALAAACNEALSLNLSDTDLSRLARRGSGSASRSIFGGFAEWEKGHDDLTSYAHGINSNGWEKDLSMIFVVINNQSKKVSARSGMSLTRDTSRFYQYWLDHVDEDLNEAKEAVKNQDFQRLGEVIEANGLRMHATNLGAQPPFTYLVQESYDAMAIVEQCRKANLPCYFTMDAGPNVKVLVEKKNKQAVMEQFLKVFDESKIIASDIISSGVEIIK 4dpy A 2.14 BS01 2P0 A 1 A14 K17 Y18 K21 S139 G140 S141 R144 A192 R193 D283 A17 K20 Y21 K24 S142 G143 S144 R147 A195 R196 D286 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 remove_due_to_license_issue Q9FD73 22734632 401 TGSMVKSGKARAHTNIALIKYWGKADETYIIPMNNSLSVTLDRFYTETKVTFDPDFTEDCLILNGNEVNAKEKEKIQNYMNIVRDLAGNRLHARIESENYVPTAAGLASSASAYAALAAACNEALSLNLSDTDLSRLARRGSGSASRSIFGGFAEWEKGHDDLTSYAHGINSNGWEKDLSMIFVVINNQSKKVSARSGMSLTRDTSRFYQYWLDHVDEDLNEAKEAVKNQDFQRLGEVIEANGLRMHATNLGAQPPFTYLVQESYDAMAIVEQCRKANLPCYFTMDAGPNVKVLVEKKNKQAVMEQFLKVFDESKIIASDIISSGVEIIK 4dq2 A 2.5 BS01 BTX A 1 S93 T94 Q116 R120 G121 R122 R125 H126 W127 S128 M137 K187 G190 G208 I209 N212 I224 S92 T93 Q115 R119 G120 R121 R124 H125 W126 S127 M136 K186 G189 G207 I208 N211 I223 0004077,0006355,0036211 Ki=0.03uM remove_due_to_license_issue 22437830 500 SKYSQDVLQLLYKNKPNYISGQSIAESLNISRTAVKKVIDQLKLEGCKIDSVNHKGHLLQQLPDIWYQGIIDQYTKSSALFDFSEVYDSIDSTQLAAKKSLVGNQSSFFILSDEQTKGRGRFNRHWSSSKGQGLWMSVVLRPNVAFSMISKFNLFIALGIRDAIQHFSQDEVKVKWPNDIYIDNGKVCGFLTEMVANNDGIEAIICGIGINLTQQLENFDESIRHRATSIQLHDKNKLDRYQFLERLLQEIEKRYNQFLTLPFSEIREEYIAASNIWNRTLLFTENDKQFKGQAIDLDYDGYLIVRDEAGESHRLISADIDF 4dr9 A 1.9 BS02 BB2 A 1 G59 I60 G61 Q66 E107 G108 C109 L110 H151 E152 H155 G58 I59 G60 Q65 E101 G102 C103 L104 H145 E146 H149 G61 Q66 C109 L110 H151 E152 H155 G60 Q65 C103 L104 H145 E146 H149 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=10nM remove_due_to_license_issue A0A0H3JZJ4 23407310 203 TAAVAIRVAKKKLAKPPLDLHYLGDRVLRQPAKRVSRIDDELRQTIRQMLQTMYSADGIGLAAPQVGINKQLIVIDLELPPLVLINPKIERTAGDLEQCQEGCLSIPGVYLDVERPEIVEVSYKDENGRPQRLVADGLLARCIQHEMDHLNGVLFVDRVENRLELNEALDKKGFAVQAVRPV 4drk A 1.5 BS01 I63 A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 ic50=8.36uM remove_due_to_license_issue Ki=2700nM, IC50=8360nM Q13451 22455444 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4drm A 1.48 BS01 0MC A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 I122 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 I110 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 ic50=5.8uM remove_due_to_license_issue IC50=5800nM Q13451 22455444 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4drn A 1.069 BS01 0MC A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 S118 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 S106 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 ic50=5.8uM remove_due_to_license_issue IC50=5800nM Q13451 22455444 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4dro A 1.1 BS01 0MD A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 ic50=3.9uM remove_due_to_license_issue IC50=3900nM Q13451 22455444 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4drp A 1.8 BS01 0MD A 1 Y57 F67 F77 Q85 V86 I87 W90 Y113 I122 Y45 F55 F65 Q73 V74 I75 W78 Y101 I110 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 ic50=3.9uM remove_due_to_license_issue IC50=3900nM Q13451 22455444 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4dru A 2.1 BS01 0LN A 1 V37 A395 A396 H428 L492 V494 P495 W500 R503 V27 A381 A382 H414 L478 V480 P481 W486 R489 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=2.4nM remove_due_to_license_issue O92972 22473861 601 SMSYTWTGALITPCAAEESKLPHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4dst A 2.3 BS01 9LI A 1 S39 D54 I55 L56 T74 G75 S39 D54 I55 L56 T74 G75 3.6.5.2 0000139,0000165,0001934,0003924,0003925,0005515,0005525,0005737,0005741,0005789,0005829,0005886,0005925,0007165,0007265,0008283,0008542,0009898,0010467,0010628,0012505,0014009,0016020,0016601,0016787,0019003,0021897,0030036,0030857,0032228,0035022,0035914,0043495,0043524,0044877,0048169,0048873,0051146,0051402,0060252,0060441,0060509 remove_due_to_license_issue IC50=155000nM P01116 22431598 201 STEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEKMSKDGKKKKKK 4dsu A 1.7 BS02 BZI A 1 K5 V7 D54 L56 T74 K5 V7 D54 L56 T71 3.6.5.2 0000139,0000165,0001934,0003924,0003925,0005515,0005525,0005737,0005741,0005789,0005829,0005886,0005925,0007165,0007265,0008283,0008542,0009898,0010467,0010628,0012505,0014009,0016020,0016601,0016787,0019003,0021897,0030036,0030857,0032228,0035022,0035914,0043495,0043524,0044877,0048169,0048873,0051146,0051402,0060252,0060441,0060509 remove_due_to_license_issue P01116 22431598 203 STEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEKMSKDGKKKKKK 4dsy A 2.3 BS03 0LO A 1 N201 H202 H295 H296 H323 H325 Y365 N195 H196 H289 H290 H317 H319 Y359 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D129 D158 Y161 N195 H196 H280 H289 H290 H317 H319 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 Ki=37uM remove_due_to_license_issue P80366 22943065 503 KNRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDDS 4dt2 A 2.7 BS03 0LV A 1 N201 H202 H296 H323 H325 Y365 N195 H196 H290 H317 H319 Y359 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D129 D158 Y161 N195 H196 H280 H289 H290 H317 H319 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 remove_due_to_license_issue P80366 22943065 504 KNRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDDST 4dt2 D 2.7 BS03 0LV D 1 N201 H202 H296 H323 H325 Y365 N195 H196 H290 H317 H319 Y359 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D129 D158 Y161 N195 H196 H280 H289 H290 H317 H319 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 remove_due_to_license_issue P80366 22943065 511 KNRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDDST 4dt6 A 2.6 BS01 6LI A 1 F48 W56 L60 D90 S92 P100 M101 W102 E103 F22 W30 L34 D64 S66 P74 M75 W76 E77 ? 0000082,0000339,0000340,0000932,0001662,0003723,0003743,0005515,0005634,0005737,0005829,0006406,0006412,0006413,0006417,0010494,0010507,0016281,0016442,0016604,0016607,0017148,0019827,0019899,0030182,0031370,0033391,0036464,0045665,0045931,0048471,0051028,0051168,0070062,0071549,0098794,0098808,0098978,0099578,0140297 remove_due_to_license_issue P06730 22458568 1001 EVANPEHYIKHPLQNRWALWFFKNDKSKTWQANLRLISKFDTVEDFWALYNHIQLSSNLMPGCDYSLFKDGIEPMWEDEKNKRGGRWLITLNKQQRRSDLDRFWLETLLCLIGESFDDYSDDVCGAVVNVRAKGDKIAIWTTECENREAVTHIGRVYKERLGLPPKIVIGYQSHADTATKSKNRFVV 4dtk A 1.86 BS01 7LI A 1 L44 A65 K67 L120 V126 L174 I185 D186 L12 A33 K35 L88 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50<0.004uM remove_due_to_license_issue P11309 22727640 408 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4dtm A 1.95 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 K878 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtm A 1.95 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtn A 1.96 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 G568 N572 W574 K705 K706 R707 P799 K800 F803 K844 K874 S360 P361 I362 Y391 P392 G393 A394 G568 N572 W574 K705 K706 R707 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 4dtn A 1.96 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 4dtr A 2.04 BS01 dna T 0 E219 I253 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 K878 E219 I253 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtr A 2.04 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dts A 1.96 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 K878 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dts A 1.96 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtt A 3.22 BS02 I41 A 1 S138 N139 A140 E189 Y831 S96 N97 A98 E147 Y789 E111 E69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 24735644 1102 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLEHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDINLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4dtt A 3.22 BS03 I41 A 2 E341 V360 G361 K364 E299 V318 G319 K322 E111 E69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 24735644 1103 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLEHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDINLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4dtu A 1.86 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtu A 1.86 BS02 dna P 0 N284 D621 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtx A 1.84 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4dtx A 1.84 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22630605 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4du1 A 2.15 BS01 dna T 0 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 G571 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 G571 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22571765 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4du1 A 2.15 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22571765 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4du3 A 2.02 BS01 dna T 0 E219 I253 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 G571 N572 K705 K706 R707 S784 K800 F803 G827 K844 K874 E219 I253 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 L561 S565 G568 G571 N572 K705 K706 R707 S784 K800 F803 G827 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22571765 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4du3 A 2.02 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22571765 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4du4 A 2.28 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 S565 G568 G571 N572 W574 K705 K706 R707 P799 K800 C801 F803 K844 K874 S360 P361 I362 Y391 P392 G393 A394 S565 G568 G571 N572 W574 K705 K706 R707 P799 K800 C801 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22571765 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 4du4 A 2.28 BS02 dna P 0 N284 D621 T622 K706 Y708 M728 G729 Q733 K734 S735 S783 S784 N786 H804 N284 D621 T622 K706 Y708 M728 G729 Q733 K734 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 22571765 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKLLINSLYGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFD 4du8 A 2.1 BS01 2P0 A 1 A14 K17 Y18 K21 S139 G140 S141 R144 S192 R193 A283 A17 K20 Y21 K24 S142 G143 S144 R147 S195 R196 A286 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 remove_due_to_license_issue Q9FD73 22734632 401 TGSMVKSGKARAHTNIALIKYWGKADETYIIPMNNSLSVTLDRFYTETKVTFDPDFTEDCLILNGNEVNAKEKEKIQNYMNIVRDLAGNRLHARIESENYVPTAAGLASSASAYAALAAACNEALSLNLSDTDLSRLARRGSGSASRSIFGGFAEWEKGHDDLTSYAHGINSNGWEKDLSMIFVVINNQSKKVSSRSGMSLTRDTSRFYQYWLDHVDEDLNEAKEAVKNQDFQRLGEVIEANGLRMHATNLGAQPPFTYLVQESYDAMAIVEQCRKANLPCYFTMAAGPNVKVLVEKKNKQAVMEQFLKVFDESKIIASDIISSGVEIIK 4duh A 1.5 BS01 RLI A 1 N46 E50 D73 R76 I78 P79 G101 K103 R136 V167 N32 E36 D59 R62 I64 P65 G87 K89 R114 V145 5.6.2.2 0003677,0003918,0005524,0006265 Kd=6.6uM remove_due_to_license_issue P0AES6 22731783 301 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLHAGGKFDDNSGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFH 4dum A 2.95 BS01 HLI A 1 F48 W56 L60 D90 S92 P100 M101 W102 E103 W166 F22 W30 L34 D64 S66 P74 M75 W76 E77 W140 ? 0000082,0000339,0000340,0000932,0001662,0003723,0003743,0005515,0005634,0005737,0005829,0006406,0006412,0006413,0006417,0010494,0010507,0016281,0016442,0016604,0016607,0017148,0019827,0019899,0030182,0031370,0033391,0036464,0045665,0045931,0048471,0051028,0051168,0070062,0071549,0098794,0098808,0098978,0099578,0140297 remove_due_to_license_issue IC50=95nM P06730 22458568 1001 EVANPEHYIKHPLQNRWALWFFKNDKSKTWQANLRLISKFDTVEDFWALYNHIQLSSNLMPGCDYSLFKDGIEPMWEDEKNKRGGRWLITLNKQQRRSDLDRFWLETLLCLIGESFDDYSDDVCGAVVNVRAKGDKIAIWTTECENREAVTHIGRVYKERLGLPPKIVIGYQSHADTATKSKNRFVV 4dus A 2.5 BS01 0MP A 1 D32 G34 P70 Y71 T72 F108 D228 G230 V332 D34 G36 P72 Y73 T74 F110 D219 G221 V312 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 24900403 410 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4dv8 A 1.632 BS02 0LX A 1 Q646 V653 S655 G657 L658 E676 L677 H686 E687 H690 Y728 E735 E739 Q382 V389 S391 G393 L394 E412 L413 H422 E423 H426 Y464 E471 E475 H686 E687 H690 Y728 E735 H422 E423 H426 Y464 E471 3.4.24.83 0008237 Ki=0.58nM remove_due_to_license_issue Ki=0.58nM P15917 22342144 802 LSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEEEKELLNRIQVDSSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4dve A 2.09 BS01 BTN A 1 P37 I38 I39 N42 S89 Y92 R93 F159 D163 K166 P38 I39 I40 N43 S90 Y93 R94 F160 D164 K167 ? 0005886,0015225,0015878 Kd=0.3nM remove_due_to_license_issue A2RMJ9 22891302 201 AMTNNQKVKTLTYSAFMTAFIIILGFLPGIPIGFIPVPIILQNMGIMMAGGLLGPKYGTISVGAFLALALIGLPVLTGGNGGAASFLGPSGGYRIAWLFTPFLIGFFLKKLKITTSQNWFGELIIVLLFGVIFVDFVGAIWLSFQSNIPLLTSLISNLVFIPGDCIKAILTVVIVRRLRKQGGFELYFR 4dvi A 1.9 BS02 2IW A 1 S1186 F1188 A1191 K1195 G1196 D1198 H1201 Y1203 F1208 Y1213 I1228 S82 F84 A87 K91 G92 D94 H97 Y99 F101 Y106 I121 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 22438990 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVGLAYAEYVIYRGEQAYPEYLITYQIMKPE 4dwb A 2.1 BS04 0M7 A 1 Y94 D98 R107 T163 Q167 K207 Y211 D250 K264 Y94 D98 R107 T163 Q167 K207 Y211 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=1840nM remove_due_to_license_issue Q95WL3 22715997 509 MASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKRK 4dwg A 2.01 BS03 0M8 A 1 Y94 D98 R107 Q167 K207 D250 K264 Y94 D98 R107 Q167 K207 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=58nM remove_due_to_license_issue Q95WL3 22715997 404 MASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKRK 4dwk A 3.0 BS01 MGK A 1 H332 G339 E341 L359 G361 H291 G298 E300 L318 G320 Q111 Q70 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 24735644 1101 MNNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMNLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4dxg A 2.5 BS01 GAL B 1 E173 Q179 R182 E167 Q173 R176 ? 0005576 remove_due_to_license_issue A0A0H3K6A3 22949551 2 EINPKFKDLRAYYTKPSLEFKNEIGIILKKWTTIRFMNVVPDYFIYKIALVGKDDKKYGEGVHRNVDVFVVLEENNYNLEKYSVGGITKSNSKKVDHKAGVRITKEDNKGTISHDVSEFKITKEQISLKELDFKLRKQLIEKNNLYGNVGSGKIVIKMKNGGKYTFELHKKLQENRMADVIDGTNIDNIEVNIK 4dxg A 2.5 BS02 SIA B 1 K169 Y170 T171 R182 D185 K163 Y164 T165 R176 D179 ? 0005576 remove_due_to_license_issue A0A0H3K6A3 22949551 3 EINPKFKDLRAYYTKPSLEFKNEIGIILKKWTTIRFMNVVPDYFIYKIALVGKDDKKYGEGVHRNVDVFVVLEENNYNLEKYSVGGITKSNSKKVDHKAGVRITKEDNKGTISHDVSEFKITKEQISLKELDFKLRKQLIEKNNLYGNVGSGKIVIKMKNGGKYTFELHKKLQENRMADVIDGTNIDNIEVNIK 4dxg A 2.5 BS03 FUC B 1 E173 K176 Q179 E167 K170 Q173 ? 0005576 remove_due_to_license_issue A0A0H3K6A3 22949551 4 EINPKFKDLRAYYTKPSLEFKNEIGIILKKWTTIRFMNVVPDYFIYKIALVGKDDKKYGEGVHRNVDVFVVLEENNYNLEKYSVGGITKSNSKKVDHKAGVRITKEDNKGTISHDVSEFKITKEQISLKELDFKLRKQLIEKNNLYGNVGSGKIVIKMKNGGKYTFELHKKLQENRMADVIDGTNIDNIEVNIK 4dxj A 2.35 BS03 0M9 A 1 D98 R107 Q167 K207 Y211 D250 K264 D98 R107 Q167 K207 Y211 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=38nM remove_due_to_license_issue Q95WL3 22715997 404 MASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKRKK 4dxj B 2.35 BS03 0M9 B 1 D98 R107 Q167 K207 Y211 D250 K264 D98 R107 Q167 K207 Y211 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=38nM remove_due_to_license_issue Q95WL3 22715997 404 MASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKRKK 4dy6 A 2.2 BS01 A22 A 1 D45 G46 H71 F74 N122 E123 T161 A162 Y163 S166 D45 G46 H71 F74 N117 E118 T156 A157 Y158 S161 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 17686780 301 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIE 4dzw A 3.05 BS01 0MQ A 1 R107 Q167 K207 Y211 Q247 D250 K273 R107 Q167 K207 Y211 Q247 D250 K273 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 remove_due_to_license_issue Q95WL3 22715997 401 MASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKR 4dzy A 2.101 BS02 WJ1 A 1 I72 Y99 L128 H132 R167 I170 R171 I34 Y61 L90 H94 R129 I132 R133 Y241 E245 K248 N249 Y203 E207 K210 N211 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 404 RLTPTMMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYHFTTAGFGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHIDG 4e0w A 2.3501 BS01 KAI A 1 E15 Y63 P90 T92 R97 G142 A143 T144 E191 E11 Y59 P86 T88 R93 G138 A139 T140 E187 ? 0015276,0016020 remove_due_to_license_issue Ki=32.8nM P42264 22425692 301 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 4e0x A 2.0 BS01 KAI A 1 E13 Y61 P88 T90 R95 G140 S141 T142 E190 E10 Y58 P85 T87 R92 G137 S138 T139 E187 ? 0015276,0016020 remove_due_to_license_issue IC50=77nM, Ki=75.9nM, EC50=37000nM P22756 22425692 301 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWR 4e1e A 2.65 BS03 0MW A 1 Y94 D98 R107 Q167 K207 D250 K264 Y93 D97 R106 Q166 K206 D249 K263 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K47 H92 D97 D101 R106 D169 K206 F245 D249 D250 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 remove_due_to_license_issue Q95WL3 22715997 404 ASMERFLSVYDEVQAFLLDQLQSKYEIDPNRARYLRIMMDTTCLGGKYFRGMTVVNVAEGFLAVTQHDEATKERILHDACVGGWMIEFLQAHYLVEDDIMDGSVMRRGKPCWYRFPGVTTQCAINDGIILKSWTQIMAWHYFADRPFLKDLLCLFQKVDYATAVGQMYDVTSMCDSNKLDPEVAQPMTTDFAEFTPAIYKRIVKYKTTFYTYLLPLVMGLFVSEAAASVEMNLVERVAHLIGEYFQVQDDVMDCFTPPEQLGKVGTDIEDAKCSWLAVTFLGKANAAQVAEFKANYGDKDPAKVAVVKRLYSEANLQADFAAYEAEVVREVESLIEQLKVKSPTFAESVAVVWEKTHKRKK 4e1k A 2.0 BS01 0N5 A 1 L11 A12 A13 G14 T82 Y103 D105 Y139 V223 E224 L8 A9 A10 G11 T79 Y100 D102 Y136 V220 E221 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 Kd=0.5uM remove_due_to_license_issue P43889 22721802 505 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 4e1m A 1.9 BS01 TQ2 A 1 A169 E170 H171 T174 A113 E114 H115 T118 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=215nM remove_due_to_license_issue P12497 22535962 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSATVKAACWWAGIKQEFGIPNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGYSAGERIVDIIATD 4e1n A 2.0 BS01 TQX A 1 Q168 A169 E170 H171 T174 M178 Q112 A113 E114 H115 T118 M122 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=19nM remove_due_to_license_issue P12497 22535962 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSATVKAACWWAGIKQEFGIPNPQSQGVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKYSAGERIVDIIATD 4e1z A 2.5 BS01 0MX A 1 R897 L899 G900 E901 G902 G905 K906 V907 A924 E975 Y976 V977 P978 G980 R1023 N1024 L1026 D1037 R15 L17 G18 E19 G20 G23 K24 V25 A42 E90 Y91 V92 P93 G95 R138 N139 L141 D152 A1019 A1021 R1023 N1024 D1037 S1059 A134 A136 R138 N139 D152 S174 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue Q9R117 22995073 1201 SDPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKEGCGPQLRSGWQREIEILRTLYHEHIVKYKGCCEDKSVQLVMEYVPLGSLRDYLPRHCVGLAQLLLFAQQICEGMAYLHAQHYIHRALAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKECKFYYASDVWSFGVTLYELLTYCDSNQSPHTKFTELIGHTQGQMTVLRLTELLERGERLPRPDRCPCEIYHLMKNCWETEASFRPTFQNLVPILQTAQEKYQ 4e20 A 2.6 BS01 0MY A 1 L899 G900 E901 G902 G905 K906 V907 A924 K926 Y976 V977 R1023 N1024 L1026 D1037 L16 G17 E18 G19 G22 K23 V24 A41 K43 Y89 V90 R136 N137 L139 D150 A1019 A1021 R1023 N1024 D1037 S1059 A132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue Q9R117 22995073 1201 DPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKEGCGPQLRSGWQREIEILRTLYHEHIVKYKGCCEDSVQLVMEYVPLGSLRDYLPRHCVGLAQLLLFAQQICEGMAYLHAQHYIHRALAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKECKFYYASDVWSFGVTLYELLTYCDSNQSPHTKFTELIGQMTVLRLTELLERGERLPRPDRCPCEIYHLMKNCWETEASFRPTFQNLVPILQTAQEKYQ 4e26 A 2.55 BS01 734 A 1 A481 L514 W531 C532 S535 S536 F583 A34 L67 W84 C85 S88 S89 F136 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S163 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=800nM P15056 22537109 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRFEQLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4e3d A 1.6 BS02 GTQ A 1 H94 L198 T200 H91 L194 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=5mM remove_due_to_license_issue IC50=5000000nM, Ki=4100nM P00918 22531842 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3d A 1.6 BS03 GTQ A 2 G6 Y7 G8 F231 E239 G3 Y4 G5 F227 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=5mM remove_due_to_license_issue IC50=5000000nM, Ki=4100nM P00918 22531842 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3f A 1.5 BS02 GRE A 1 L198 T199 T200 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=3mM remove_due_to_license_issue Ki=5200nM P00918 22531842 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3f A 1.5 BS03 GRE A 2 Y7 G8 F231 E239 Y4 G5 F227 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=3mM remove_due_to_license_issue Ki=5200nM P00918 22531842 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3f A 1.5 BS04 GRE A 3 D130 F131 G132 D126 F127 G128 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=3mM remove_due_to_license_issue Ki=5200nM P00918 22531842 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3h A 1.5 BS02 HQE A 1 V121 F131 V143 L198 V118 F127 V139 L194 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=90nM remove_due_to_license_issue Ki=90nM P00918 22531842 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3i A 1.6 BS01 0N3 A 1 S64 Y150 V211 S212 Y221 G317 A318 G320 S61 Y147 V208 S209 Y218 G314 A315 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3j A 1.7999 BS01 0N4 A 1 S64 Y150 V211 S212 Y221 A318 S61 Y147 V208 S209 Y218 A308 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K305 A308 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3k A 1.4299 BS01 0NA A 1 S64 Y150 V211 Y221 A318 T319 S61 Y147 V208 Y218 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3l A 1.43 BS01 0NB A 1 S64 Y150 V211 S212 Y221 G317 A318 T319 G320 S61 Y147 V208 S209 Y218 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3l A 1.43 BS02 0NB B 1 L85 Q250 L254 Y259 P304 L82 Q247 L251 Y256 P301 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3m A 1.44 BS01 0ND A 1 S64 Y150 V211 S212 Y221 A318 T319 G320 S61 Y147 V208 S209 Y218 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3m A 1.44 BS02 0ND A 2 L85 Q250 Q253 L254 Y259 P304 L82 Q247 Q250 L251 Y256 P301 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 402 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3n A 1.49 BS01 0NE A 1 S64 Y150 V211 Y221 A318 T319 G320 S61 Y147 V208 Y218 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue Ki=50nM P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e3o A 1.6 BS01 0NG A 1 S64 Q120 Y150 N152 Y221 G317 A318 S61 Q117 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 23043117 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4e49 A 1.45 BS02 RCO A 1 L141 V143 L198 V207 L137 V139 L194 V203 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.7uM remove_due_to_license_issue Ki=7700nM P00918 22531842 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e49 A 1.45 BS03 RCO A 2 N67 E69 I91 Q92 N64 E66 I88 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.7uM remove_due_to_license_issue Ki=7700nM P00918 22531842 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e49 A 1.45 BS04 RCO A 3 F70 D72 I91 F67 D69 I88 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.7uM remove_due_to_license_issue Ki=7700nM P00918 22531842 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e4a A 1.45 BS02 JKE A 1 H94 L198 T200 H91 L194 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=9mM remove_due_to_license_issue P00918 22531842 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e4l A 2.0 BS01 0NH A 1 G882 E883 V889 A906 M956 F958 L959 R1007 N1008 L1010 D1021 G18 E19 V25 A42 M81 F83 L84 R132 N133 L135 D146 D1003 A1005 R1007 N1008 D1021 D1040 D128 A130 R132 N133 D146 D165 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.7nM remove_due_to_license_issue EC50=210nM, Ki=1.7nM P23458 22591402 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4e4n A 1.9 BS01 0NL A 1 L881 E883 G887 K888 V889 A906 M956 F958 L959 L1010 L29 E31 G35 K36 V37 A54 M95 F97 L98 L149 D1003 A1005 R1007 N1008 D1021 D1040 D142 A144 R146 N147 D160 D179 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.9nM remove_due_to_license_issue EC50=91nM, Ki=0.9nM P23458 22591402 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4e4x A 3.6 BS01 T1Q A 1 A481 K483 L505 L514 T529 C532 F583 D594 F595 G596 A34 K36 L58 L67 T82 C85 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=41nM P15056 22534450 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 4e5d A 2.201 BS01 0NJ A 1 H245 G246 F247 G315 G341 L342 T343 S347 A348 H238 G239 F240 G308 G331 L332 T333 S337 A338 S198 R218 H245 T343 E344 S196 R211 H238 T333 E334 1.13.12.7 0004497,0005524,0005777,0008218,0016405,0046872,0047077,0051087 remove_due_to_license_issue IC50=600nM P08659 22921073 601 DAKNIKKGPAPFYPLEDGTAGEQLHKAMKRYALVPGTIAFTDAHIEVNITYAEYFEMSVRLAEAMKRYGLNTNHRIVVCSENSLQFFMPVLGALFIGVAVAPANDIYNERELLNSMNISQPTVVFVSKKGLQKILNVQKKLPIIQKIIIMDSKTDYQGFQSMYTFVTSHLPPGFNEYDFVPESFDRDKTIALIMNSLPKGVALPHRTACVRFSHARDPIFGNQIIPDTAILSVVPFHHGFGMFTTLGYLICGFRVVLMYRFEEELFLRSLQDYKIQSALLVPTLFSFFAKSTLIDKYDLSNLHEIASGLSKEVGEAVAKRFHLPGIRQGYGLTETTSAILITPEGDDKPGAVGKVVPFFEAKVVDLDTGKTLGVNQRGELCVRGPMIMSGYVNNPEATNALIDKDGWLHSGDIAYWDEDEHFFIV 4e5f A 2.392 BS03 0N7 A 1 H41 E80 D108 E119 K134 H41 E61 D89 E100 K115 3.1.-.- 0003723,0039694 ic50=15uM remove_due_to_license_issue Q5EP34 22876176 305 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRTMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHTYYLEKANKIKSEETHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSERAAA 4e5g A 2.647 BS03 XI7 A 1 H41 E80 E119 K134 H41 E61 E100 K115 3.1.-.- 0003723,0039694 remove_due_to_license_issue Q5EP34 22876176 305 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRTMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHTYYLEKANKIKSEETHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSERAAAE 4e5g A 2.647 BS04 XI7 A 2 A20 Y24 I38 H41 A20 Y24 I38 H41 3.1.-.- 0003723,0039694 remove_due_to_license_issue Q5EP34 22876176 306 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRTMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHTYYLEKANKIKSEETHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSERAAAE 4e5h D 2.158 BS03 0N8 D 1 Y24 H41 R84 W88 F105 L106 D108 E119 Y24 H41 R65 W69 F86 L87 D89 E100 3.1.-.- 0003723,0039694 ic50=0.43uM remove_due_to_license_issue Q5EP34 22876176 305 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRTMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHTYYLEKANKIKSEETHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSERAAAELA 4e5j A 2.35 BS01 581 A 1 H41 E80 D108 E119 Y130 K134 H41 E61 D89 E100 Y111 K115 3.1.-.- 0003723,0039694 Ki=18.7uM remove_due_to_license_issue Q5EP34 22876176 303 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRTMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHTYYLEKANKIKSEETHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSERAAAE 4e5j A 2.35 BS02 581 A 2 K34 A37 I38 H41 V122 R124 A198 K34 A37 I38 H41 V103 R105 A179 3.1.-.- 0003723,0039694 Ki=18.7uM remove_due_to_license_issue Q5EP34 22876176 304 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRTMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHTYYLEKANKIKSEETHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSERAAAE 4e5w A 1.86 BS01 0NT A 1 L881 G882 E883 V889 A906 M956 F958 L959 R1007 N1008 L1010 D1021 L29 G30 E31 V37 A54 M96 F98 L99 R147 N148 L150 D161 D1003 A1005 R1007 N1008 D1021 D1040 D143 A145 R147 N148 D161 D180 2.7.10.2 0004672,0004713,0005524,0006468 Ki=22nM remove_due_to_license_issue Ki=22nM, EC50=>8800nM P23458 22591402 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKNHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4e6c A 2.39 BS01 0O8 A 1 L195 N196 W197 A255 L174 N175 W176 A234 D150 K152 N155 D168 T185 D144 K146 N149 D162 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd~15uM remove_due_to_license_issue Q16539 23079240 500 ERPTFYRQELNKTIWEVPERYQNLSPVGSGYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPP 4e6d A 2.22 BS01 0NU A 1 L855 G856 K857 G861 S862 V863 A880 M929 E930 F931 L932 L983 D994 L16 G17 K18 G22 S23 V24 A41 M85 E86 F87 L88 L139 D150 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.2nM remove_due_to_license_issue Ki=1.2nM O60674 22591402 1201 DPTQFEERHLKFLRQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYNLKLIMEFLPYGSLREYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4e6q A 1.948 BS01 0NV A 1 K857 G858 V863 A880 E930 L932 R980 L983 K23 G24 V29 A46 E96 L98 R146 L149 D976 A978 R980 N981 D994 S1016 D142 A144 R146 N147 D160 S182 2.7.10.2 0004672,0004713,0005524,0006468 Ki=4.4nM remove_due_to_license_issue Ki=4.4nM O60674 22591402 1201 AFEDRDPTQFEERHLKFLRQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEFLPYGSLREYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4e70 A 1.6093 BS01 N7I A 1 L118 S122 M179 W268 D272 L325 F326 L112 S116 M173 W262 D266 L316 F317 D272 D302 L334 D266 D293 L325 ? 0008168,0008171,0032259,0046983 Kd=2.94uM remove_due_to_license_issue A6XNE6 23633600 403 MDAATAVELLDAQPQVWHHFLGYINSMTLQCALELDIADVIHRHGHPIPLNQLAAALEIPQTKAPFLSRLMRMLVHLGYFTQVITKPVLPSYWLAPLSRLLLKQNPYNARSLTFCSVHEHLVDPWRQMSAWLRTGKEDGKDTPNAFAFAHEGKKVYEVCSEDANFSQLFSEGMAGDSWLFSRALVSKCRDAFEGLSSLVDVGGGTGNTSKVIAETFPNIHCTVFDLPHVVSGPKQTHPNLDYESGNMFTDEIPHADAVLFKWVLCDWPDEPVLKMLKQCKKALTKKGKLMIADHVLDHESCNDSNSMGTSLILDMLFMSFLEGSLRTEKQWAKLFAEAGFKDYKITPVGGLRVLIEVYP 4e70 B 1.6093 BS01 N7I B 1 L1118 S1122 M1179 W1268 D1272 L1325 F1326 L117 S121 M175 W260 D264 L313 F314 C1271 D1272 D1302 L1334 C263 D264 D290 L322 ? 0008168,0008171,0032259,0046983 Kd=2.94uM remove_due_to_license_issue A6XNE6 23633600 1402 GLVPHMDAATAVELLDAQPQVWHHFLGYINSMTLQCALELDIADVIHRHGHPIPLNQLAAALEIPQTKAPFLSRLMRMLVHLGYFTQVITKPVLPSYWLAPLSRLLLKQNPYNARSLTFCSVHEHLVDPWRQMSAWLRTGKKDTPNAFAFAHEGKKVYEVCSEDANFSQLFSEGMAGDSWLFSRALVSKCRDAFEGLSSLVDVGGGTGNTSKVIAETFPNIHCTVFDLPGPKQTHPNLDYESGNMFTDEIPHADAVLFKWVLCDWPDEPVLKMLKQCKKALTKGKLMIADHVLDHESCNDSNSMGTSLILDMLFMSFLEGSLRTEKQWAKLFAEAGFKDYKITPVGGLRVLIEVYP 4e7r H 2.25 BS03 0NW H 1 H57 Y60A W60D N98 L99 D189 A190 C191 E192 S195 V213 W215 G216 G219 H43 Y47 W50 N95 L96 D191 A192 C193 E194 S197 V217 W219 G220 G222 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 302 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4e8w A 2.8654 BS01 IHA A 1 N202 T238 S240 G243 A257 V265 A268 G269 N294 V301 N193 T229 S231 G234 A248 V251 A254 G255 N280 V287 ? 0003824,0005829,0005975,0016301,0016773,0016779,0033785,0033786,0046835 remove_due_to_license_issue IC50=810nM B4EB35 23256532 501 VPREQLARSRVLVVGDVMLDRYWFGNVDRISPEAPVPVVHVQRQEERLGGAANVARNAVTLGGQAGLLCVVGCDEPGERIVELLGSSGVTPHLERDPALPTTIKLRVLARQQQLLRVDFEAMPTHEVLLAGLARFDVLLPQHDVVLMSDYAKGGLTHVTTMIEKARAAGKAVLVDPKGDDWARYRGASLITPNRAELREVVGQWKSEDDLRARVANLRAELDIDALLLTRSEEGMTLFSAGGELHAPALAVSGAGDTVIATVATMLGAGVPLVDAVVLANRAAGIVVGKTATVDYDELF 4e8y A 2.6 BS01 IHA A 1 N202 T238 S240 G243 A257 A259 V262 A268 N294 N196 T232 S234 G237 A251 A253 V256 A262 N288 ? 0003824,0005829,0005975,0016301,0016773,0016779,0033785,0033786,0046835 remove_due_to_license_issue IC50=810nM B4EB35 23256532 501 VVPVPREQLARSRVLVVGDVMLDRYWFGNVDRISPEAPVPVVHVQRQEERLGGAANVARNAVTLGGQAGLLCVVGCDEPGERIVELLGSSGVTPHLERDPALPTTIKLRVLARQQQLLRVDFEAMPTHEVLLAGLARFDVLLPQHDVVLMSDYAKGGLTHVTTMIEKARAAGKAVLVDPKGDDWARYRGASLITPNRAELREVVGQWKSEDDLRARVANLRAELDIDALLLTRSEEGMTLFSAGGELHAPALAREVFDVSGAGDTVIATVATMLGAGVPLVDAVVLANRAAGIVVGKLGTATVDYDEL 4e8y B 2.6 BS01 IHA B 1 T238 S240 E241 G243 M244 R260 A268 G269 N294 T230 S232 E233 G235 M236 R252 A260 G261 N286 ? 0003824,0005829,0005975,0016301,0016773,0016779,0033785,0033786,0046835 remove_due_to_license_issue IC50=810nM B4EB35 23256532 501 PVPREQLARSRVLVVGDVMLDRYWFGNVDRISPEAPVPVVHVQRQEERLGGAANVARNAVTLGGQAGLLCVVGCDEPGERIVELLGSSGVTPHLERDPALPTTIKLRVLARQQQLLRVDFEAMPTHEVLLAGLARFDVLLPQHDVVLMSDYAKGGLTHVTTMIEKARAAGKAVLVDPKGDDWARYRGASLITPNRAELREVVGQWKSEDDLRARVANLRAELDIDALLLTRSEEGMTLFSAGGELHAPALAREVFDVSGAGDTVIATVATMLGAGVPLVDAVVLANRAAGIVVGKLGTATVDYDELF 4e8z A 3.05 BS01 IHC A 1 N202 T238 S240 E241 G243 A268 G269 N294 G298 N196 T232 S234 E235 G237 A262 G263 N288 G292 ? 0003824,0005829,0005975,0016301,0016773,0016779,0033785,0033786,0046835 remove_due_to_license_issue IC50=230nM B4EB35 23256532 501 VVPVPREQLARSRVLVVGDVMLDRYWFGNVDRISPEAPVPVVHVQRQEERLGGAANVARNAVTLGGQAGLLCVVGCDEPGERIVELLGSSGVTPHLERDPALPTTIKLRVLARQQQLLRVDFEAMPTHEVLLAGLARFDVLLPQHDVVLMSDYAKGGLTHVTTMIEKARAAGKAVLVDPKGDDWARYRGASLITPNRAELREVVGQWKSEDDLRARVANLRAELDIDALLLTRSEEGMTLFSAGGELHAPALAREVFDVSGAGDTVIATVATMLGAGVPLVDAVVLANRAAGIVVGKLGTATVDYDEL 4e90 A 2.5 BS02 7RG A 1 L420 Y424 F441 Q453 F456 L243 Y247 F264 Q276 F279 3.1.4.35 0004114,0007165,0008081 ic50=8nM remove_due_to_license_issue IC50=70.0nM O76083 23025719 903 GSHMTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 4e93 A 1.84 BS01 GUI A 1 I567 R569 V575 A588 K590 M636 V639 G642 L690 I120 R122 V128 A141 K143 M189 V192 G195 L243 D683 A685 R687 N688 D701 D236 A238 R240 N241 D254 2.7.10.2 0004672,0004713,0005524,0006468 ic50=45.8nM remove_due_to_license_issue P07332 22520759 901 SMIPEVQKPLHEQLWYHGAIPRAEVAELLVHSGDFLVRESQQEYVLSVLWDGLPRHFIIQSLDNLYRLEGEGFPSIPLLIDHLLSTQQPLTKKSGVVLHRAVPKDKWVLNHEDLVLGEQIGRGNFGEVFSGRLRADNTLVAVKSCRETLPPDLKAKFLQEARILKQYSHPNIVRLIGVCTQKQPIYIVMELVQGGDFLTFLRTEGARLRVKTLLQMVGDAAAGMEYLESKCCIHRDLAARNCLVTEKNVLKISDFGMSREVPVKWTAPEALNYGRYSSESDVWSFGILLWETFSLGASPYPNLSNQQTREFVEKGGRLPCPELCPDAVFRLMEQCWAYEPGQRPSFSTIYQELQSIRKRHR 4e96 A 1.92 BS01 0NS A 1 W81 L94 N140 I146 W40 L53 N99 I105 ? ic50=0.22uM remove_due_to_license_issue IC50=220nM, Kd=136nM O60885 23095041 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 4e9u A 2.1 BS01 RWY A 1 F22 A134 V137 G138 A157 G161 L164 N168 Y248 F22 A134 V137 G138 A157 G161 L164 N168 Y248 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=1.5uM remove_due_to_license_issue Ki=1500nM A9JQL9 22486710 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDVYGDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 4ea1 A 2.46 BS01 3RX A 1 D48 V111 Y129 V133 Q165 D48 V107 Y125 V129 Q161 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=0.36uM remove_due_to_license_issue IC50=100000nM, Ki=360nM A9JQL9 22486710 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 4ea2 A 2.05 BS01 RWZ A 1 F22 C44 R45 D48 V133 A134 V137 L160 L164 F22 C44 R45 D48 V130 A131 V134 L157 L161 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 Ki=0.36uM remove_due_to_license_issue A9JQL9 22486710 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 4ea3 A 3.013 BS01 0NN A 1 Q107 I127 D130 Y131 M134 I219 S223 W276 Q280 V283 T305 Y309 Q61 I81 D84 Y85 M88 I166 S170 W223 Q227 V230 T252 Y256 ? 0001626,0004930,0004985,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41146 22596163 1501 PLGLKVTIVGLYLAVCVGGLLGNCLVMYVILRHTKMKTATNIYIFNLALADTLVLLTLPFQGTDILLGFWPFGNALCKTVIAIDYYNMFTSTFTLTAMSVDRYVAICHPTSSKAQAVNVAIWALASVVGVPVAIMGSAQVEDEEIECLVEIPTPQDYWGPVFAICIFLFSFIVPVLVISVCYSLMIRRLRGVRLLSGSREKDRNLRRITRLVLVVVAVFVGCWTPVQVFVLAQGLGVQPSSETAVAILRFCTALGYVNSCLNPILYAFLDENFKACFR 4ear A 1.7 BS01 IM5 A 1 Y88 A116 A117 G118 F200 E201 V217 M219 N243 X257 Y85 A113 A114 G115 F197 E198 V214 M216 N240 X254 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 W257 S30 H61 H83 Y85 E86 A113 M216 S217 N240 V242 W254 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=7nM P00491 23438750 301 GYTYEDYKNTAEYLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLYKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTYKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANWEEVLAAGKQAAQKLEQFVSILMASIPLPD 4ear C 1.7 BS01 IM5 C 1 S33 Y88 A116 A117 G118 F200 E201 M219 N243 X257 S30 Y85 A113 A114 G115 F197 E198 M216 N240 X254 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 W257 S30 H61 H83 Y85 E86 A113 M216 S217 N240 V242 W254 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=7nM P00491 23438750 301 GYTYEDYKNTAEYLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLYKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTYKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANWEEVLAAGKQAAQKLEQFVSILMASIPLPDKA 4eb8 A 2.3 BS02 IM5 A 1 Y88 A116 A117 G118 F200 E201 V217 M219 N243 W257 V260 Y90 A118 A119 G120 F202 E203 V219 M221 N245 W259 V262 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 W257 S35 H66 H88 Y90 E91 A118 M221 S222 N245 V247 W259 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=7nM P00491 23438750 302 TLMENGYTYEDYKNTAEYLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLYKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTYKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANWEEVLAAGKQAAQKLEQFVSILMASIPLPD 4eb8 C 2.3 BS02 IM5 C 1 Y88 A116 A117 G118 F200 E201 V217 M219 N243 W257 Y85 A113 A114 G115 F197 E198 V214 M216 N240 W254 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 W257 S30 H61 H83 Y85 E86 A113 M216 S217 N240 V242 W254 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 remove_due_to_license_issue Ki=7nM P00491 23438750 302 GYTYEDYKNTAEYLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLYKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTYKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANWEEVLAAGKQAAQKLEQFVSILMASIPLPD 4eb9 A 2.6 BS02 0O6 C 1 D297 G306 L307 R308 C309 D314 W323 L353 L354 D44 G53 L54 R55 C56 D61 W70 L100 L101 2.3.2.27 remove_due_to_license_issue IC50=5.4nM Q13490 23166698 402 SISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRYPHLLEQLLS 4eb9 C 2.6 BS02 0O6 C 1 D297 G306 L307 R308 C309 W310 E311 D314 E319 W323 D43 G52 L53 R54 C55 W56 E57 D60 E65 W69 2.3.2.27 remove_due_to_license_issue IC50=5.4nM Q13490 23166698 402 ISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRYPHLLEQLLST 4ebv A 1.67 BS01 0O7 A 1 L534 L537 H544 R550 N551 L562 G563 D604 M607 C611 L125 L128 H135 R141 N142 L153 G154 D180 M183 C187 D546 A548 R550 N551 D564 K583 D137 A139 R141 N142 D155 K159 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.99uM remove_due_to_license_issue IC50=4200nM Q05397 22819505 700 SSTRDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4ebw A 2.65 BS01 0PF A 1 L534 L537 H544 R550 N551 L562 G563 D604 M607 L122 L125 H132 R138 N139 L150 G151 D177 M180 D546 A548 R550 N551 D564 K583 D134 A136 R138 N139 D152 K156 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>30000nM Q05397 22819505 700 STRDYEIQRERIELGRCIGEGQFGDVHQGIYMSNPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4ec0 A 1.85 BS02 7PQ A 1 Y8 M11 G13 R14 M99 W104 Y152 T159 L199 Y8 M11 G13 R14 M99 W104 Y152 T159 L199 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 remove_due_to_license_issue IC50=845nM O60760 22546671 203 MPNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4ec4 A 3.3 BS02 0O6 A 1 N249 K297 G306 L307 T308 D309 W310 E314 Q319 W323 N4 K52 G61 L62 T63 D64 W65 E69 Q74 W78 2.3.2.27 remove_due_to_license_issue IC50=25.4nM P98170 23166698 402 SDRNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 4ec4 F 3.3 BS01 0O6 A 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 K50 G59 L60 T61 D62 W63 E67 Q72 W76 2.3.2.27 remove_due_to_license_issue IC50=25.4nM P98170 23166698 402 RNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECL 4ed5 A 2.0 BS01 rna D 0 I23 N25 Y26 Q29 I52 H59 L61 Y63 F65 K89 T90 K92 A96 R97 S99 I103 K104 Y109 I133 N134 R136 L138 R147 F151 R153 K182 A185 I6 N8 Y9 Q12 I35 H42 L44 Y46 F48 K72 T73 K75 A79 R80 S82 I86 K87 Y92 I116 N117 R119 L121 R130 F134 R136 K165 A168 ? 0003676,0003723,1990904 remove_due_to_license_issue Q15717 23519412 2 ~ 11 GRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPITVKFAA 4ed5 B 2.0 BS01 rna C 0 I23 N25 Y26 K50 I52 S60 L61 Y63 F65 K89 T90 K92 A96 R97 S99 I103 K104 Y109 I133 R136 R147 F151 R153 A185 I6 N8 Y9 K33 I35 S43 L44 Y46 F48 K72 T73 K75 A79 R80 S82 I86 K87 Y92 I116 R119 R130 F134 R136 A168 ? 0003676,0003723,1990904 remove_due_to_license_issue Q15717 23519412 2 ~ 11 GRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPITVKFAAN 4ede B 1.4 BS01 RET B 1 W33 Q38 C53 S55 W58 N59 Y60 W106 K108 W33 Q38 C53 S55 W58 N59 Y60 W106 K108 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 23224553 202 TRDQNGTWEMESNENFEGWMKALDIDFALRKIWVRLTQTLVIDQDGDNFKVKCTSTFWNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 4edy A 1.72 BS02 9PQ A 1 Y8 F9 M11 G13 R14 Q36 M99 W104 Y152 T159 L199 Y7 F8 M10 G12 R13 Q35 M98 W103 Y151 T158 L198 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 remove_due_to_license_issue IC50=1480nM O60760 22546671 203 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4edz A 2.0 BS02 0O5 A 1 M11 G13 R14 D96 M99 W104 M10 G12 R13 D95 M98 W103 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 remove_due_to_license_issue IC50=8.26nM O60760 22546671 202 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4ee0 A 1.75 BS01 0O4 A 1 F9 M11 G13 R14 D96 M99 W104 F8 M10 G12 R13 D91 M94 W99 Y8 R14 R19 W104 Y7 R13 R18 W99 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 remove_due_to_license_issue IC50=2.34nM O60760 22546671 202 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 4eeh A 1.6 BS01 HH6 A 1 N51 A55 D93 I96 G97 M98 T184 N35 A39 D77 I80 G81 M82 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=45uM remove_due_to_license_issue P07900 22632933 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4eej A 1.501 BS01 RET A 1 F16 W19 A33 Q38 W58 L77 W106 K108 L117 F16 W19 A33 Q38 W58 L77 W106 K108 L117 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 23224553 201 TRDRNGTWEMESNENFEGWMKALDIDFALRKIAVRLTQTLVIDQDGDNFKVKCTSTFWNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 4eev A 1.8 BS01 L1X A 1 I1084 A1108 E1127 M1131 L1157 Y1159 M1160 M1211 V1220 A1221 D1222 F1223 I40 A64 E83 M87 L113 Y115 M116 M167 V176 A177 D178 F179 D1204 A1206 R1208 N1209 D1222 D160 A162 R164 N165 D178 2.7.10.1 0004672,0004713,0005524,0006468 ic50=4.7nM remove_due_to_license_issue IC50=4.7nM P08581 23275061 1401 PLLQNTVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4ef4 A 2.147 BS01 C2E A 1 Y167 T263 P264 Y16 T103 P104 ? 0002218,0032481 Kd=4.42uM (22579474) Kd=4.42uM remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22579474 401 NFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPFSLSQEVLRHLRQEEKEEVTV 4ef4 B 2.147 BS01 C2E A 1 Y167 T263 P264 Y16 T100 P101 ? 0002218,0032481 Kd=4.42uM (22579474) remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22579474 401 NFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPASFSLSQEVLRHLRQEEKEEVTV 4ef6 A 1.94 BS01 I2E A 1 H44 G46 L50 G158 K160 V187 M195 S196 S197 H43 G45 L49 G157 K159 V186 M194 S195 S196 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M39 H43 H46 D87 D88 Q91 K159 S195 S196 R197 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1.18mM remove_due_to_license_issue P9WIL5 23872845 404 AIPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4efg A 1.58 BS01 RET A 1 W19 A33 Q38 C53 W58 N59 W106 K108 L117 W19 A33 Q38 C53 W58 N59 W106 K108 L117 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 23224553 201 TRDQNGTWEMESNENFEGWMKALDIDFALRKIAVRLTQTLVIDQDGDNFKVKCTSTFWNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 4efk A 1.7 BS01 0OC A 1 P38 M40 F67 V142 V143 Q164 P35 M37 F64 V132 V133 Q154 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D78 D79 Q82 K150 S186 S187 R188 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=3.18mM remove_due_to_license_issue P9WIL5 23872845 401 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPLNGSGRLLVAARLGTTRLLDNIAIEIGTFAG 4efs A 1.63 BS06 E37 A 1 I180 L181 A182 L214 H218 E219 H222 H228 P232 A234 V235 P238 T239 Y240 K241 I76 L77 A78 L110 H114 E115 H118 H124 P128 A130 V131 P134 T135 Y136 K137 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=2.5nM remove_due_to_license_issue Ki=2.5nM P39900 22689580 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 4eft A 2.12 BS01 EFT A 1 N51 A55 D93 M98 L103 F138 W162 T184 N35 A39 D77 M82 L87 F122 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=85uM remove_due_to_license_issue P07900 22632933 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4efu A 2.0 BS01 EFU A 1 N51 A55 D93 G97 M98 L107 F138 W162 T184 N35 A39 D77 G81 M82 L91 F122 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.25uM remove_due_to_license_issue P07900 22632933 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4egh A 1.6 BS01 0OY A 1 N51 K58 D93 M98 T184 N36 K43 D78 M83 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=550uM remove_due_to_license_issue P07900 22573733 302 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4egi A 1.79 BS01 B2J A 1 A55 G97 T184 A46 G88 T175 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=150uM remove_due_to_license_issue Kd=42000nM P07900 22573733 301 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKER 4egk A 1.69 BS01 RDC A 1 N51 D54 A55 K58 D93 M98 T184 N41 D44 A45 K48 D83 M88 T174 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=19nM remove_due_to_license_issue Kd=1.2nM P07900 22573733 301 PMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4egy A 2.301 BS01 dna T 0 P3 K4 Y5 S40 H42 T43 Q61 G62 G63 P16 K17 Y18 S53 H55 T56 Q74 G75 G76 ? 0003700,0006355 remove_due_to_license_issue P96711 23109551 1 ~ 21 LEVLFQGPLGSEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 4egy A 2.301 BS02 dna U 0 T29 E30 R41 R45 Q61 G62 G64 T42 E43 R54 R58 Q74 G75 G77 ? 0003700,0006355 remove_due_to_license_issue P96711 23109551 22 ~ 42 LEVLFQGPLGSEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 4egy B 2.301 BS01 dna T 0 T29 E30 R41 R45 Q61 G62 G64 T31 E32 R43 R47 Q63 G64 G66 ? 0003700,0006355 remove_due_to_license_issue P96711 23109551 1 ~ 21 EFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 4egy B 2.301 BS02 dna U 0 P3 K4 Y5 S40 H42 T43 Q61 G62 G63 P5 K6 Y7 S42 H44 T45 Q63 G64 G65 ? 0003700,0006355 remove_due_to_license_issue P96711 23109551 22 ~ 42 EFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 4eh2 A 2.0 BS02 0OK A 1 A51 T106 A46 T101 D150 K152 N155 D168 T185 D145 K147 N150 D163 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh3 A 2.4 BS01 NAR A 1 K53 I84 T106 L108 M109 L171 K48 I79 T101 L103 M104 L166 D150 K152 N155 D168 T185 D145 K147 N150 D163 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh4 A 2.5 BS02 0OL A 1 A51 K53 I84 L104 T106 L167 A46 K48 I79 L99 T101 L160 D150 K152 N155 D168 T185 D143 K145 N148 D161 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh5 A 2.0 BS02 0OM A 1 V38 A51 K53 L104 T106 L108 M109 V33 A46 K48 L99 T101 L103 M104 D150 K152 N155 D168 T185 D140 K142 N145 D158 T160 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh6 A 2.1 BS02 0ON A 1 A51 K53 L104 T106 M109 A46 K48 L99 T101 M104 D150 K152 N155 D168 T185 D145 K147 N150 D163 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh7 A 2.1 BS02 0OO A 1 A51 I84 T106 L167 A46 I79 T101 L162 D150 K152 N155 D168 T185 D145 K147 N150 D163 T168 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh8 A 2.2 BS02 0OP A 1 E71 V83 I141 H148 D168 F169 E66 V78 I136 H143 D163 F164 D150 K152 N155 D168 T185 D145 K147 N150 D163 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh8 A 2.2 BS03 0OP A 2 V38 A51 K53 I84 T106 L108 M109 V33 A46 K48 I79 T101 L103 M104 D150 K152 N155 D168 T185 D145 K147 N150 D163 T167 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 403 ERPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4eh9 A 2.1 BS02 0OQ A 1 R70 E71 L74 L75 D168 R64 E65 L68 L69 D159 D150 K152 N155 D168 T185 D141 K143 N146 D159 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 RPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4ehe A 3.3 BS01 RI8 A 1 V471 A481 K483 L505 L514 T529 W531 C532 F583 D594 F595 G596 V24 A34 K36 L58 L67 T82 W84 C85 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S159 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22335519 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4ehe B 3.3 BS01 RI8 B 1 V471 A481 K483 L514 I527 T529 W531 C532 F583 D594 F595 G596 V24 A34 K36 L67 I80 T82 W84 C85 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S169 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22335519 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSGSHQFEQLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4ehg A 3.5 BS01 RI9 A 1 A481 L505 L514 I527 W531 C532 G534 F583 D594 F595 A34 L58 L67 I80 W84 C85 G87 F136 D147 F148 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22335519 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATEGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4ehg B 3.5 BS01 RI9 B 1 A481 K483 L505 L514 I527 T529 W531 C532 G534 F583 D594 F595 G596 A34 K36 L58 L67 I80 T82 W84 C85 G87 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S153 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22335519 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4ehm B 2.2 BS01 PJA A 1 R144 G192 Q193 W244 F289 R138 G186 Q187 W238 F283 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H184 R226 K229 D232 C234 Y235 D274 D281 H284 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 remove_due_to_license_issue Q08603 22480322 401 QKDVTIKSDAPDTLLLEKHADYIASYGSDDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 4ehr A 2.09 BS01 0Q5 A 1 F97 R100 Y101 A104 F105 L108 E129 L130 G138 R139 F40 R43 Y44 A47 F48 L51 E72 L73 G81 R82 ? 0042981 ic50=0.013uM remove_due_to_license_issue IC50=13nM Q07817 22608393 301 SQSNRELVVDFLSYKLSQKGYSWSQSEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 4ehv A 1.6 BS01 0SJ A 1 Y35 R67 R70 E71 L74 H148 D168 Y31 R63 R66 E67 L70 H144 D164 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4ehv A 1.6 BS02 0SJ A 2 R149 R189 I193 W197 Y200 V204 R145 R174 I178 W182 Y185 V189 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 402 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4ehv A 1.6 BS04 0SJ A 3 M194 N196 W197 S252 S254 A255 Y258 M179 N181 W182 S237 S239 A240 Y243 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Q16539 23247173 404 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4ehz A 2.174 BS01 JAK A 1 V889 A906 M956 F958 L959 E966 L1010 V32 A49 M94 F96 L97 E104 L148 D1003 A1005 R1007 N1008 D1021 D1040 D141 A143 R145 N146 D159 D178 2.7.10.2 0004672,0004713,0005524,0006468 Ki=10nM remove_due_to_license_issue EC50=250nM, Ki=10.0nM P23458 22698084 1201 EKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4ei4 A 2.22 BS01 0Q2 A 1 V889 A906 M956 F958 L959 R1007 N1008 L1010 V37 A54 M93 F95 L96 R144 N145 L147 D1003 A1005 R1007 N1008 D1021 D1040 D140 A142 R144 N145 D158 D177 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.8nM remove_due_to_license_issue P23458 22698084 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4ej2 A 2.65 BS01 D1F A 1 G135 L136 D283 D339 T340 H377 A383 L384 E385 N484 E672 A673 S674 G675 G124 L125 D266 D313 T314 H351 A357 L358 E359 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue IC50=6100000nM P00489 22770609 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4ej8 A 2.347 BS01 1F1 A 1 W42 P44 K45 K55 W42 P44 K45 K55 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=4.1uM remove_due_to_license_issue P12499 23540839 106 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMNLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4ejl A 2.445 BS01 IOP A 1 P44 K45 K55 V56 P44 K45 K55 V56 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=7.2uM remove_due_to_license_issue P12499 23540839 106 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMNLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4ejn A 2.19 BS01 0R4 A 1 N53 N54 Q59 Q79 W80 I84 L210 T211 V270 Y272 R273 I290 D292 N43 N44 Q49 Q69 W70 I74 L153 T154 V213 Y215 R216 I233 D235 D274 K276 N279 D292 T312 D217 K219 N222 D235 T250 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 ic50=0.005uM remove_due_to_license_issue IC50=44nM P31749 22533986 501 VAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYF 4ejy A 2.0 BS01 dna C 0 Q125 N126 R128 N216 G217 G219 P220 K221 V222 D240 V241 W242 Q125 N126 R128 N216 G217 G219 P220 K221 V222 D240 V241 W242 K221 D240 K221 D240 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 11 ~ 26 MKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMGK 4ejy A 2.0 BS02 dna D 0 N126 Q131 R175 G177 F178 R179 N126 Q131 R175 G177 F178 R179 K221 D240 K221 D240 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 2 ~ 16 MKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMGK 4ejy B 2.0 BS01 dna E 0 Q125 N126 R128 F178 N216 G217 G219 P220 K221 V222 D240 V241 Q126 N127 R129 F179 N217 G218 G220 P221 K222 V223 D241 V242 K221 D240 K222 D241 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 11 ~ 26 RMKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMG 4ejy B 2.0 BS02 dna F 0 N126 R175 G177 F178 R179 N127 R176 G178 F179 R180 K221 D240 K222 D241 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 2 ~ 16 RMKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMG 4ejz A 3.05 BS01 dna C 0 Q125 N126 R128 F178 N216 G217 V218 G219 P220 K221 V222 D240 V241 W242 Q125 N126 R128 F178 N216 G217 V218 G219 P220 K221 V222 D240 V241 W242 K221 D240 K221 D240 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 11 ~ 26 MKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMGK 4ejz A 3.05 BS02 dna D 0 R175 G177 F178 R179 R175 G177 F178 R179 K221 D240 K221 D240 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 2 ~ 16 MKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMGK 4ejz B 3.05 BS01 dna E 0 Q125 N126 R128 F178 N216 G217 V218 G219 P220 K221 V222 D240 V241 Q125 N126 R128 F178 N216 G217 V218 G219 P220 K221 V222 D240 V241 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 11 ~ 26 MKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMGK 4ejz B 3.05 BS02 dna F 0 R175 G177 F178 R179 R175 G177 F178 R179 4.2.99.18 0003684,0003824,0006281,0006284,0006289,0008534,0016798,0016829,0140097 remove_due_to_license_issue Q8R5T9 23246782 2 ~ 16 MKYNVEEKGTKVIVRGIADFNLKETFESGQCFRWNEEEDGSYTGVAYDRVVNVKLEGDTLIIDNTNLTDFYDIWFDYFDLGRDYGQIKESLSKDPVLKEAIKFGQGIRILRQDTWETLVSFIVSQNNRIPQIKKVIENLATSFGNPIEYKGKIYYTFPKPEELVMYDVETIAKTRCGFRAKYIFDAASKVFSGEINLLKLHEYSTSEIRDILMTINGVGPKVADCVILYSIGRYDTFPTDVWIKRIVEHLYLKREGTPVEIQLFAIDKFGDLSGFAQQYLFYYGREMGK 4ek9 A 2.5 BS01 EP4 A 1 P133 G137 G163 E186 K187 G221 D222 F223 P126 G130 G156 E179 K180 G214 D215 F216 2.1.1.360 0031151,0051726 Ki=38000nM remove_due_to_license_issue Ki=9000nM Q8TEK3 22978415 501 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLKNP 4eke A 2.6 BS01 D1I A 1 G135 L136 D283 F285 H377 N484 E672 S674 G675 G124 L125 D266 F268 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue Ki=33400nM P00489 22770609 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4ekg A 2.8 BS01 0QJ A 1 V135 Y136 D161 G163 E186 K187 D222 F223 F239 N241 S268 Y312 V123 Y124 D149 G151 E174 K175 D210 F211 F227 N229 S256 Y300 2.1.1.360 0031151,0051726 remove_due_to_license_issue Ki=13nM Q8TEK3 22978415 500 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLKN 4eki A 2.85 BS01 0QK A 1 L143 D161 G163 S164 V169 E186 K187 D222 F223 N241 L132 D150 G152 S153 V158 E175 K176 D211 F212 N230 2.1.1.360 0031151,0051726 remove_due_to_license_issue Ki=0.300000nM, IC50=0.400000nM, EC50=9.0nM, Kd=0.250000nM Q8TEK3 22978415 501 KLELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLK 4eky A 2.45 BS01 D1J A 1 G135 L136 D283 N284 D339 H341 H377 T378 N484 E672 A673 S674 G675 G124 L125 D266 N267 D313 H315 H351 T352 N458 E646 A647 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=303uM remove_due_to_license_issue Ki=303000nM P00489 22770609 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4el0 A 2.4 BS01 D1K A 1 G135 L136 D339 H377 N484 E672 S674 G675 G124 L125 D313 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=32.4uM remove_due_to_license_issue Ki=32400nM P00489 22770609 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4el5 A 2.0 BS01 D1M A 1 G135 L136 D283 N284 D339 H377 T378 N484 E672 S674 G675 G124 L125 D266 N267 D313 H351 T352 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.7uM remove_due_to_license_issue Ki=4700nM P00489 22770609 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4el9 A 1.55 BS01 AFE A 1 F79 K100 V131 L147 D148 L155 E197 L200 L214 F31 K52 V78 L94 D95 L102 E144 L147 L161 D193 K195 E197 N198 D211 T231 D140 K142 E144 N145 D158 T175 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P18654 22846040 400 EIAITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKESEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKP 4elb A 2.6 BS01 34S A 1 M6 V7 A8 L21 E28 L29 Q30 V32 I51 L55 P56 F96 M6 V7 A8 L21 E28 L29 Q30 V32 I51 L55 P56 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 remove_due_to_license_issue Q81R22 22999981 203 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 4ele A 2.35 BS02 31I A 1 M6 V7 A8 L21 E28 L29 V32 K33 R53 L55 P56 R58 F96 M6 V7 A8 L21 E28 L29 V32 K33 R53 L55 P56 R58 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 Ki=13.2nM remove_due_to_license_issue Q81R22 22999981 203 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 4elf A 2.3 BS02 35I A 1 M6 V7 A8 L21 E28 L29 V32 K33 I51 P56 R58 F96 M6 V7 A8 L21 E28 L29 V32 K33 I51 P56 R58 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 Ki=9.4nM remove_due_to_license_issue Q81R22 22999981 203 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 4elg A 2.101 BS01 52J A 1 M6 V7 A8 N20 L21 E28 L29 Q30 V32 K33 I51 L55 P56 R58 F96 M6 V7 A8 N20 L21 E28 L29 Q30 V32 K33 I51 L55 P56 R58 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 Ki=6.9nM remove_due_to_license_issue Q81R22 22999981 201 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 4elh A 2.103 BS02 53I A 1 M6 V7 A8 N20 L21 E28 L29 V32 K33 A50 I51 R53 L55 F96 M6 V7 A8 N20 L21 E28 L29 V32 K33 A50 I51 R53 L55 F96 M6 L21 W23 E28 L29 V32 L55 I93 T115 M6 L21 W23 E28 L29 V32 L55 I93 T115 1.5.1.3 0000166,0004146,0005829,0006730,0016491,0046452,0046654,0046655,0046872,0050661 Ki=8.2nM remove_due_to_license_issue Q81R22 22999981 202 MIVSFMVAMDENRVIGKDNNLPWRLPSELQYVKKTTMGHPLIMGRKNYEAIGRPLPGRRNIIVTRNEGYHVEGCEVAHSVEEVFELCKNEEEIFIFGGAQIYDLFLPYVDKLYITKIHHAFEGDTFFPEMDMTNWKEVFVEKGLTDEKNPYTYYYHVYEKQQLVPR 4em7 A 1.9 BS01 0RA A 1 N51 E55 R81 G82 M83 R140 N35 E39 R65 G66 M67 R107 0003677,0003918,0005524,0006265 ic50=7.7uM remove_due_to_license_issue 22814212 301 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHAVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4emf A 1.77 BS01 M7G A 1 Y70 E85 G109 N110 Y111 I155 E160 R163 E189 Y70 E85 G109 N110 Y111 I155 E160 R163 E189 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 23280611 304 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 4emr A 1.75 BS01 MGP A 1 Y70 E85 G109 N110 Y111 E160 R163 E189 S193 Y70 E85 G109 N110 Y111 E160 R163 E189 S193 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 23280611 301 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 4emt A 1.5 BS01 C2E A 1 Y163 Y167 R238 T263 P264 Y10 Y14 R76 T101 P102 ? 0002218,0032481 Kd=5uM (22728658) Kd=4.63uM remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22728658 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEE 4emt B 1.5 BS01 C2E A 1 Y167 T263 P264 Y14 T101 P102 ? 0002218,0032481 Kd=5uM (22728658) remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22728658 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEE 4emv A 1.7 BS01 0R9 A 1 N51 E55 D78 R81 M83 P84 I98 R140 T172 N35 E39 D62 R65 M67 P68 I82 R110 T142 0003677,0003918,0005524,0006265 ic50=0.005uM remove_due_to_license_issue 22814212 301 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHGLHGVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4en4 A 2.15 BS02 GT0 A 1 S12 T47 Y84 D235 S10 T45 Y82 D233 2.7.1.35 0000287,0005524,0005576,0005634,0005654,0005737,0005829,0008270,0008478,0009443,0016301,0016773,0030170,0030955,0031402,0031403,0034774,0035580,0042803,0042816,0042817,0042818,0042822,0046872,0070062 Ki=3uM remove_due_to_license_issue O00764 22879864 405 EECRVLSIQSHVIRGYVGNRAATFPLQVLGFEIDAVNSVQFSNHTGYAHWKGQVLNSDELQELYEGLRLNNMNKYDYVLTGYTRDKSFLAMVVDIVQELKQQNPRLVYVCDPVLGDKWDGEGSMYVPEDLLPVYKEKVVPLADIITPNQFEAELLSGRKIHSQEEALRVMDMLHSMGPDTVVITSSDLPSPQGSNYLIVLGSQRRRNPAGSVVMERIRMDIRKVDAVFVGTGDLFAAMLLAWTHKHPNNLKVACEKTVSTLHHVLQRTIQCAKAQAGEGVRPSPMQLELRMVQSKRDIEDPEIVVQATVL 4enj A 3.0989 BS01 dna B 0 Y25 G26 R39 M45 K46 W56 N61 S62 S67 R69 D70 I71 Y25 G26 R39 M45 K46 W56 N61 S62 S67 R69 D70 I71 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enj A 3.0989 BS02 dna C 0 M3 S36 Y37 R39 Q40 M3 S36 Y37 R39 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 14 ~ 26 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enk A 3.0445 BS01 dna B 0 Y25 G26 R39 M45 K46 W56 N61 S62 S67 R69 Y25 G26 R39 M45 K46 W56 N61 S62 S67 R69 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enk A 3.0445 BS02 dna C 0 M3 S36 Y37 R39 Q40 M3 S36 Y37 R39 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 14 ~ 26 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enm A 2.8402 BS01 dna B 0 Y25 G26 R39 M45 K46 P50 W56 V59 N61 S62 R69 D70 I71 R77 Y25 G26 R39 M45 K46 P50 W56 V59 N61 S62 R69 D70 I71 R77 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enm A 2.8402 BS02 dna C 0 M3 S36 Y37 R39 Q40 Q43 M3 S36 Y37 R39 Q40 Q43 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 14 ~ 26 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enn A 2.8448 BS01 dna C 0 Y25 G26 A38 R39 Q43 M45 K46 W56 S62 S67 R69 Y25 G26 A38 R39 Q43 M45 K46 W56 S62 S67 R69 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enn A 2.8448 BS02 dna D 0 S36 Y37 R39 Q40 S36 Y37 R39 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enn B 2.8448 BS01 dna E 0 Y25 G26 A38 R39 Q43 M45 K46 W56 N61 S62 S67 R69 Y25 G26 A38 R39 Q43 M45 K46 W56 N61 S62 S67 R69 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enn B 2.8448 BS02 dna F 0 M3 S36 Y37 R39 Q40 M3 S36 Y37 R39 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 22658721 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4enx A 2.8 BS01 Z20 A 1 L44 G45 S46 F49 G50 S51 V52 A65 K67 L120 E121 L174 I185 D186 L8 G9 S10 F13 G14 S15 V16 A29 K31 L81 E82 L135 I146 D147 D167 K169 N172 D186 L193 T204 D128 K130 N133 D147 L154 T165 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 22869110 402 QYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4eny A 2.801 BS01 J19 A 1 G45 S46 G50 S51 V52 A65 K67 L120 L174 D186 G9 S10 G13 S14 V15 A28 K30 L76 L130 D142 D167 K169 N172 D186 L193 T204 D123 K125 N128 D142 L149 T160 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 22869110 404 QYQVGPLLGSGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGRVPMEVVLLKKVSSFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4eo4 A 2.87 BS01 SSA A 1 M131 R162 T173 R174 L175 F178 Q180 D182 Q287 V288 Q292 G324 S325 R328 M92 R123 T134 R135 L136 F139 Q141 D143 Q242 V243 Q247 G279 S280 R283 C133 R162 Q180 D182 H184 K273 H319 C94 R123 Q141 D143 H145 K228 H274 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0005739,0005759,0006412,0006418,0006435,0008270,0070159,0140101 remove_due_to_license_issue P07236 22773845 1001 ATMTSMVSQRQDLFMTDPLSPGSMFFLPNGAKIFNKLIEFMKLQQKFKFGFNEVVTPLIYKKTLWEKSGHWENYADDMFKVETKEEYGLKPMNCPGHCLIFGKKDRSYNELPLRFSDFSPLHRNEASGALSGLTRLRKFHQDDGHIFCTPSQVKSEIFNSLKLIDIVYNKIFPFAESNYFINFSTRPDHFIGDLKVWNHAEQVLKEILEESGKPWKLNPGDGAFYGPKLDIMVTDHLRKTHQVATIQLDFQLPERFDLKFKDQDNSYKRPIMIHRATFGSIERFMALLIDSNEGRWPFWLNPYQAVIIPVNTKNVQQLDMCTALQKKLRNELEADDMEPVPLNDWHFNVDLDIRNEPVGYRIKSAILKNYSYLIIVGDEEVQLQKYNIRERDNRKSFEKLTMSQIWEKFIELEKNYK 4eo4 A 2.87 BS02 SSA A 2 I407 K408 I411 R434 R439 I362 K363 I366 R389 R394 C133 R162 Q180 D182 H184 K273 H319 C94 R123 Q141 D143 H145 K228 H274 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0005739,0005759,0006412,0006418,0006435,0008270,0070159,0140101 remove_due_to_license_issue P07236 22773845 1002 ATMTSMVSQRQDLFMTDPLSPGSMFFLPNGAKIFNKLIEFMKLQQKFKFGFNEVVTPLIYKKTLWEKSGHWENYADDMFKVETKEEYGLKPMNCPGHCLIFGKKDRSYNELPLRFSDFSPLHRNEASGALSGLTRLRKFHQDDGHIFCTPSQVKSEIFNSLKLIDIVYNKIFPFAESNYFINFSTRPDHFIGDLKVWNHAEQVLKEILEESGKPWKLNPGDGAFYGPKLDIMVTDHLRKTHQVATIQLDFQLPERFDLKFKDQDNSYKRPIMIHRATFGSIERFMALLIDSNEGRWPFWLNPYQAVIIPVNTKNVQQLDMCTALQKKLRNELEADDMEPVPLNDWHFNVDLDIRNEPVGYRIKSAILKNYSYLIIVGDEEVQLQKYNIRERDNRKSFEKLTMSQIWEKFIELEKNYK 4eo6 A 1.791 BS01 0S2 A 1 L419 R422 H475 S476 Y477 I482 W528 L414 R417 H470 S471 Y472 I477 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.002uM remove_due_to_license_issue P26663 22664130 600 HHSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 4eo8 A 1.798 BS01 0S3 A 1 L419 R422 H475 S476 Y477 I482 W528 L414 R417 H470 S471 Y472 I477 W523 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=0.007uM remove_due_to_license_issue P26663 22664130 600 HHSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASQLDLSGWFVAGYSGGDIYH 4eoh A 2.1 BS01 TEP A 1 S12 G20 V231 D235 S9 G17 V222 D226 2.7.1.35 0000287,0005524,0005576,0005634,0005654,0005737,0005829,0008270,0008478,0009443,0016301,0016773,0030170,0030955,0031402,0031403,0034774,0035580,0042803,0042816,0042817,0042818,0042822,0046872,0070062 Ki=50uM remove_due_to_license_issue O00764 22879864 402 ECRVLSIQSHVIRGYVGNRAATFPLQVLGFEIDAVNSVQFSNHTGYAHWKGQVLNSDELQELYEGLRLNNMNKYDYVLTGYTRDKSFLAMVVDIVQELKQQNPRLVYVCDPVLGDKWDGEGSMYVPEDLLPVYKEKVVPLADIITPNQFEAELLSGRKIHSQEEALRVMDMLHSMGPDTVVITSSDLPSPQGSNYLIVLGSQRRVVMERIRMDIRKVDAVFVGTGDLFAAMLLAWTHKHPNNLKVACEKTVSTLHHVLQRTIQCAKAQAGEGVRPSPMQLELRMVQSKRDIEDPEIVVQATVL 4eoi A 2.0 BS01 1RO A 1 E12 G13 V18 A31 K33 E81 F82 L83 E131 L134 D145 E13 G14 V19 A32 K34 E78 F79 L80 E128 L131 D142 D127 K129 E131 N132 D145 T158 T165 D124 K126 E128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=253nM, Ki=340nM P24941 22921070 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKDFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPENLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4eok A 2.57 BS01 4SP A 1 G11 E12 A31 V64 F80 L83 M85 D86 D89 L134 G12 E13 A32 V61 F77 L80 M82 D83 D86 L131 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=6.0nM, Ki=6.0nM, Kd=1310nM P24941 22921070 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLSMDLKDFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 4eol A 2.4 BS01 1RO A 1 E12 G13 V18 A31 K33 E81 F82 L83 L134 D145 E13 G14 V19 A32 K34 E80 F81 L82 L132 D143 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=253nM, Ki=340nM P24941 22921070 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLSMDLKDFMDASLTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 4eon A 2.4 BS01 1RO A 1 I10 E12 V18 A31 K33 F82 L83 L134 D145 I12 E14 V20 A33 K35 F84 L85 L136 D147 D127 K129 E131 N132 D145 T158 T165 D129 K131 E133 N134 D147 T160 T167 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=253nM, Ki=340nM P24941 22921070 301 GSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLSMDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPENLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4eop A 1.99 BS01 1RO A 1 E12 G13 V18 A31 K33 E81 F82 L83 H84 E131 L134 D145 E15 G16 V21 A34 K36 E82 F83 L84 H85 E132 L135 D146 D127 K129 E131 N132 D145 T158 T165 D128 K130 E132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=253nM, Ki=340nM P24941 22921070 301 PGSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPENLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 4eor A 2.2 BS01 4SP A 1 I10 A31 V64 F80 E81 L83 H84 Q85 D86 K89 L134 I11 A32 V61 F77 E78 L80 H81 Q82 D83 K86 L131 D127 K129 Q131 N132 D145 T158 T165 D124 K126 Q128 N129 D142 T155 T162 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Ki=500nM remove_due_to_license_issue IC50=6.0nM, Ki=6.0nM, Kd=1310nM P24941 22921070 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 4eos A 2.57 BS01 1RO A 1 G11 E12 V18 A31 K33 E81 F82 L83 Q131 L134 D145 G14 E15 V21 A34 K36 E81 F82 L83 Q131 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=253nM, Ki=340nM P24941 22921070 301 PGSMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 4eot A 2.855 BS01 dna C 0 V237 R259 R260 Y267 V12 R34 R35 Y42 ? 0003677,0003700,0006355 remove_due_to_license_issue Q8NHW3 23148532 1 ~ 19 RFSDDQLVSMSVRELNRQLRGFSKEEVIRLKQKRRTLKNRGYAQSCRFKRVQQRHILESEKCQLQSQVEQLKLEVGRLAKERDLYKEKYEKL 4eot A 2.855 BS02 dna D 0 T261 R265 Q269 R272 T36 R40 Q44 R47 ? 0003677,0003700,0006355 remove_due_to_license_issue Q8NHW3 23148532 1 ~ 19 RFSDDQLVSMSVRELNRQLRGFSKEEVIRLKQKRRTLKNRGYAQSCRFKRVQQRHILESEKCQLQSQVEQLKLEVGRLAKERDLYKEKYEKL 4eot B 2.855 BS01 dna C 0 T261 R265 R272 T35 R39 R46 ? 0003677,0003700,0006355 remove_due_to_license_issue Q8NHW3 23148532 1 ~ 19 FSDDQLVSMSVRELNRQLRGFSKEEVIRLKQKRRTLKNRGYAQSCRFKRVQQRHILESEKCQLQSQVEQLKLEVGRLAKERDLYKEKYEKLA 4eot B 2.855 BS02 dna D 0 R259 R260 Y267 C271 R33 R34 Y41 C45 ? 0003677,0003700,0006355 remove_due_to_license_issue Q8NHW3 23148532 1 ~ 19 FSDDQLVSMSVRELNRQLRGFSKEEVIRLKQKRRTLKNRGYAQSCRFKRVQQRHILESEKCQLQSQVEQLKLEVGRLAKERDLYKEKYEKLA 4eox P 1.783 BS01 0S5 P 1 G69 G70 V71 G72 Q77 G129 C130 L131 V170 H173 E174 H177 G68 G69 V70 G71 Q76 G119 C120 L121 V160 H163 E164 H167 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=0.28nM remove_due_to_license_issue Q8DP79 22579486 302 SAIERITKAAHLIDMNDIIREGNPTLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNIAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLIL 4epy A 1.801 BS02 0QY A 1 K5 L6 V7 E37 D38 S39 D54 L56 T74 K6 L7 V8 E38 D39 S40 D55 L57 T75 3.6.5.2 0003924,0005525,0007165,0016020 Kd=340uM remove_due_to_license_issue P01116 22566140 203 GMTEYKLVVVGAVGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEK 4eqc A 2.01 BS01 XR1 A 1 A297 R299 E315 V342 M344 Y346 L347 G350 L396 T541 A53 R55 E71 V98 M100 Y102 L103 G106 L152 T297 D389 K391 D393 N394 D407 P416 T427 D145 K147 D149 N150 D163 P172 T183 2.7.11.1 0004672,0005524,0006468 ic50=8nM remove_due_to_license_issue IC50=2.8nM Q13153 23960073 601 DPFTSDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT 4er1 E 2.0 BS01 0ZP E 1 D12 A13 D30 D32 G34 Y75 G76 D77 F189 I213 D215 G217 T218 T219 L220 Y222 I299 D15 A16 D33 D35 G37 Y79 G80 D81 F194 I217 D219 G221 T222 T223 L224 Y226 I302 3.4.23.22 0004190,0006508 Ki=0.24uM remove_due_to_license_issue P11838 6381096 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4erd A 2.589 BS01 rna C 0 F525 K528 F101 K104 ? 0003723 remove_due_to_license_issue W7X6T2 22705372 117 ~ 150 NCLIKIINIPQGTLKAEVVLAVRHLGYEFYCDYIDGQAMIRFQNSDEQRLAIQKLLNHNNNKLQIEIRGQICDVISTIPEDEEKNYWNYIKFKKNEFRKFFFMKKQQK 4erd A 2.589 BS02 rna D 0 F406 Y407 D409 R465 Q467 I514 K517 K518 F521 R522 F29 Y30 D32 R41 Q43 I90 K93 K94 F97 R98 ? 0003723 remove_due_to_license_issue W7X6T2 22705372 117 ~ 150 NCLIKIINIPQGTLKAEVVLAVRHLGYEFYCDYIDGQAMIRFQNSDEQRLAIQKLLNHNNNKLQIEIRGQICDVISTIPEDEEKNYWNYIKFKKNEFRKFFFMKKQQK 4erd B 2.589 BS01 rna C 0 F406 Y407 D409 R465 Q467 I514 K518 R522 F29 Y30 D32 R41 Q43 I90 K94 R98 ? 0003723 remove_due_to_license_issue W7X6T2 22705372 117 ~ 150 NCLIKIINIPQGTLKAEVVLAVRHLGYEFYCDYIDGQAMIRFQNSDEQRLAIQKLLNHNNNKLQIEIRGQICDVISTIPEDEEKNYWNYIKFKKNEFRKFFFMKKQQK 4erd B 2.589 BS02 rna D 0 K392 A393 F525 K528 K15 A16 F101 K104 ? 0003723 remove_due_to_license_issue W7X6T2 22705372 117 ~ 150 NCLIKIINIPQGTLKAEVVLAVRHLGYEFYCDYIDGQAMIRFQNSDEQRLAIQKLLNHNNNKLQIEIRGQICDVISTIPEDEEKNYWNYIKFKKNEFRKFFFMKKQQK 4ere A 1.8 BS01 0R2 A 1 L54 I61 V93 K94 H96 I99 L33 I40 V67 K68 H70 I73 2.3.2.27 0005634,0043066,0051726 ic50=4.2nM remove_due_to_license_issue Q00987 22524527 201 SEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 4erf A 2.0 BS01 0R3 A 1 L54 I61 Y67 V93 K94 H96 I99 Y100 L36 I43 Y49 V75 K76 H78 I81 Y82 2.3.2.27 0005634,0043066,0051726 Kd=0.4nM remove_due_to_license_issue Kd=0.4nM, IC50=4.1nM Q00987 22524527 201 IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4erk A 2.2 BS01 OLO A 1 I29 A50 Q103 L105 M106 E107 K112 L154 I24 A45 Q98 L100 M101 E102 K107 L149 D147 K149 S151 N152 D165 T188 D142 K144 S146 N147 D160 T183 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 ic50=27uM remove_due_to_license_issue IC50=27000nM P63086 9753691 800 AAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 4erw A 2.0 BS01 STU A 1 I10 V18 A31 K33 F80 E81 F82 L83 Q131 L134 D145 I10 V18 A31 K33 F75 E76 F77 L78 Q126 L129 D140 D127 K129 Q131 N132 D145 T158 T165 D122 K124 Q126 N127 D140 T153 T160 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 22893598 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4esi A 1.87 BS01 0RB A 1 Y80 V81 G121 N122 Y123 I172 R180 Y76 V77 G117 N118 Y119 I168 R176 V81 E177 R180 V77 E173 R176 3.2.2.22 0017148,0030598 ic50=70uM remove_due_to_license_issue P02879 23050058 301 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSS 4etz A 2.05 BS01 C2E A 1 Q158 R367 D370 G395 G398 Y399 R402 Q1 R198 D201 G226 G229 Y230 R233 ? Kd=0.5uM (22810222) Kd~0.5uM remove_due_to_license_issue Q9HZE7 22810222 501 QSLRSSLLGLRQLLRELPGDEAPLDALAETVLALLAQYGSLRIAGLYRVRYDRTPEPQPLATLGEMPALDADDLLVRTCLERGELVSVRQALQVCVPLVDTDGRILALLAVEQMPFFVFNERTFSLLAILAGHIADLLQSDRRALQLADIDAQRFSQYLKRSLLDARDHGLPACLYAFELTDARYGEEVQRLLEGSQRGLDVQLRLRNDEGRRVLLVLLPLTSAEGSQGYLQRLRILFAERFGQARELESLGVRIRQYELDAGNDRQALGHFLFNECGLNDQQVA 4eu0 A 1.7 BS01 C2E A 1 R367 D370 G395 G398 Y399 R402 R197 D200 G225 G228 Y229 R232 ? Kd=0.5uM (22810222) Kd=0.4uM remove_due_to_license_issue Q9HZE7 22810222 501 QSLRSSLLGLRQLLRELPGDEAPLDALAETVLALLAQYGSLRIAGLYRVRYDRTPEPQPLATLGEMPALDADDLLVRTCLERGELVSVRQAAVCVPLVDTDGRILALLAVEQMPFFVFNERTFSLLAILAGHIADLLQSDRRALQLADIDAQRFSQYLKRSLLDARDHGLPACLYAFELTDARYGEEVQRLLEGSQRGLDVQLRLRNDEGRRVLLVLLPLTSAEGSQGYLQRLRILFAERFGQARELESLGVRIRQYELDAGNDRQALGHFLFNECGLNDQQVAI 4eu3 B 1.58 BS01 CIT B 1 T36 S71 T94 R228 P231 T35 S70 T93 R227 P230 2.8.3.18 0003986,0006083,0006084,0006085,0008410,0008775,0016740,0019427,0045733,1901289 remove_due_to_license_issue B3EY95 23030530 2502 TERIRNVALRSKVCPAETASELIKHGDVVGTSGFTGAGYPKEVPKALAQRMEAAHDRGEKYQISLITGASTGPQLDGELAKANGVYFRSPFNTDATMRNRINAGETEYFDNHLGQVAGRAVQGNYGKFNIALVEATAITEDGGIVPTSSVGNSQTFLNLAEKVIIEVNEWQNPMLEGIHDIWDGNVSGVPTRDIVPIVRADQRVGGPVLRVNPDKIAAIVRTNDRDRNAPFAAPDETAKAIAGYLLDFFGHEVKQNRLPPSLLPLQSGVGNVANAVLEGLKEGPFENLVGYSEVIQDGMLAMLDSGRMRIASASSFSLSPEAAEEINNRMDFFRSKIILRQQDVSNSPGIIRRLGCIAMNGMIEADIYGNVNSTRVMGSKMMNGIGGSGDFARSSYLSIFLSPSTAKGGKISAIVPMAAHVDHIMQDAQIFVTEQGLADLRGLSPVQRAREIISKCAHPDYRPMLQDYFDRALKNSFGKHTPHLLTEALSWHQRFIDTGTMLPS 4euc A 2.644 BS01 0RQ A 1 G269 V270 G271 N272 V273 N361 M363 I364 M383 N384 G385 G387 G388 S389 A407 K408 I412 G268 V269 G270 N271 V272 N360 M362 I363 M382 N383 G384 G386 G387 S388 A406 K407 I411 2.8.3.18 0003986,0006083,0006084,0006085,0008410,0008775,0016740,0019427,0045733,1901289 remove_due_to_license_issue B3EY95 23030530 601 TERIRNVALRSKVCPAETASELIKHGDVVGTSGFTGAGYPKEVPKALAQRMEAAHDRGEKYQISLITGASTGPQLDGELAKANGVYFRSPFNTDATMRNRINAGETEYFDNHLGQVAGRAVQGNYGKFNIALVEATAITEDGGIVPTSSVGNSQTFLNLAEKVIIEVNEWQNPMLEGIHDIWDGNVSGVPTRDIVPIVRADQRVGGPVLRVNPDKIAAIVRTNDRDRNAPFAAPDETAKAIAGYLLDFFGHEVKQNRLPPSLLPLQSGVGNVANAVLEGLKEGPFENLVGYSAVIQDGMLAMLDSGRMRIASASSFSLSPEAAEEINNRMDFFRSKIILRQQDVSNSPGIIRRLGCIAMNGMIEADIYGNVNSTRVMGSKMMNGIGGSGDFARSSYLSIFLSPSTAKGGKISAIVPMAAHVDHIMQDAQIFVTEQGLADLRGLSPVQRAREIISKCAHPDYRPMLQDYFDRALKNSFGKHTPHLLTEALSWHQRFIDTGTMLPS 4euc B 2.644 BS01 0RQ B 1 G269 V270 G271 N272 V273 N361 M363 I364 M383 N384 G385 G387 G388 S389 A407 K408 I412 G268 V269 G270 N271 V272 N360 M362 I363 M382 N383 G384 G386 G387 S388 A406 K407 I411 2.8.3.18 0003986,0006083,0006084,0006085,0008410,0008775,0016740,0019427,0045733,1901289 remove_due_to_license_issue B3EY95 23030530 601 TERIRNVALRSKVCPAETASELIKHGDVVGTSGFTGAGYPKEVPKALAQRMEAAHDRGEKYQISLITGASTGPQLDGELAKANGVYFRSPFNTDATMRNRINAGETEYFDNHLGQVAGRAVQGNYGKFNIALVEATAITEDGGIVPTSSVGNSQTFLNLAEKVIIEVNEWQNPMLEGIHDIWDGNVSGVPTRDIVPIVRADQRVGGPVLRVNPDKIAAIVRTNDRDRNAPFAAPDETAKAIAGYLLDFFGHEVKQNRLPPSLLPLQSGVGNVANAVLEGLKEGPFENLVGYSAVIQDGMLAMLDSGRMRIASASSFSLSPEAAEEINNRMDFFRSKIILRQQDVSNSPGIIRRLGCIAMNGMIEADIYGNVNSTRVMGSKMMNGIGGSGDFARSSYLSIFLSPSTAKGGKISAIVPMAAHVDHIMQDAQIFVTEQGLADLRGLSPVQRAREIISKCAHPDYRPMLQDYFDRALKNSFGKHTPHLLTEALSWHQRFIDTGTMLPS 4euo A 1.28 BS01 ABU A 1 T34 F121 W222 R225 D248 Y284 T11 F98 W199 R202 D225 Y261 ? 0042597 remove_due_to_license_issue A9CGA5 23043322 404 DLVFSSWGGTTQDAQKAAWAEKFMVETGINVLQDGPTDYGKLKAMVEANGVTWDVVDVEGDYAAQAGPKGLLEKLDFSVIDKTKLDPRFVTDYSVGSFYYSFVIGCNVDSVSACPKSWADLFDTAKFPGKRTFYKWSAPGVIEAALLADGVTADKLYPLDLDRAFKKLDTIKSDIIWWSGGAQSQQLIASAEAPFGSVWNGRMTALEQSGVKVETSWAQNITAADSLVVPKGTKNKDAAMKFIALATSAQAQADMATATGYAPVNIESAKLMDPKIAKSLPDQQTESQVNADMNYWAQHRDEIGERWYAWQAK 4euv A 2.0 BS01 C2E A 1 R367 D370 L388 G395 G398 Y399 R402 R199 D202 L220 G227 G230 Y231 R234 ? Kd=0.5uM (22810222) Kd~0.5uM remove_due_to_license_issue Q9HZE7 22810222 501 QSLRSSLLGLRQLLRELPGDEAPLDALAETVLALLAQYGSLRIAGLYRVRYDRTPEPQPLATLGEMPALDADDLLVRTCLERGELVSVRQELAAVCVPLVDTDGRILALLAVEQMPFFVFNERTFSLLAILAGHIADLLQSDRRALQLADIDAQRFSQYLKRSLLDARDHGLPACLYAFELTDARYGEEVQRLLEGSQRGLDVQLRLRNDEGRRVLLVLLPLTSAEGSQGYLQRLRILFAERFGQARELESLGVRIRQYELDAGNDRQALGHFLFNECGLNDQQVA 4ew2 A 1.602 BS01 DXY A 1 R64 M89 R90 I91 L92 V139 A140 R64 M89 R90 I91 L92 V139 A140 N106 H108 T135 D144 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 remove_due_to_license_issue P22102 23869564 304 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWVKEEHH 4ew3 A 1.702 BS01 DXZ A 1 R64 M89 R90 I91 L92 V139 A140 R64 M89 R90 I91 L92 V139 A140 N106 H108 T135 D144 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=0.18uM remove_due_to_license_issue P22102 23869564 304 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWVKEEHH 4ewh A 2.5 BS01 T77 A 1 L132 G133 A156 A208 P209 G211 L259 G269 L16 G17 A40 A92 P93 G95 L143 G153 D252 A254 R256 N257 D270 V292 D136 A138 R140 N141 D154 V176 2.7.10.2,2.7.11.1 0004672,0004713,0005524,0006468 Ki=0.0003uM remove_due_to_license_issue Ki=0.3nM Q07912 22929232 401 LTCLIGEKDLRLLEKLGDGSFGVVRRGEWDAPSGKTVSVAVKCLKPDVLSQPEAMDDFIREVNAMHSLDHRNLIRLYGVVLTPPMKMVTELAPLGSLLDRLRKHQGHFLLGTLSRYAVQVAEGMGYLESKRFIHRDLAARNLLLATRDLVKIGDFGLMRALPQNDDHYVMQEHRKVPFAWCAPESLKTRTFSHASDTWMFGVTLWEMFTYGQEPWIGLNGSQILHKIDKEGERLPRPEDCPQDIYNVMVQCWAHKPEDRPTFVALRDFLLEAQPT 4ewn D 1.903 BS01 0VR D 1 V130 G177 S201 G202 G203 L222 A223 A224 S225 V123 G170 S194 G195 G196 L215 A216 A217 S218 4.3.2.10 0000105,0000107,0005515,0005737,0016829 Kd=0.2uM remove_due_to_license_issue Q9X0C6 23109729 400 LAKRIIACLDVKDGRVVKGTNFENLRDSGDPVELGKFYSEIGIDELVFLDITKTMLELVEKVAEQIDIPFTVGGGIHDFETASELILRGADKVSINTAAVENPSLITQIAQTFGSQAVVVAIVAKRVDGEFMVFTYSGKKNTGILLRDWVVEVEKRGAGEILLTSIDRVGTKSGYDTEMIRFVRPLTTLPIIASGGAGKMEHFLEAFLAGADAALAASVFHFREIDVRELKEYLKKHGVNVRL 4ewo A 1.8 BS01 996 A 1 L78 D80 G82 Y119 T120 F156 W163 Y246 D276 G278 L31 D33 G35 Y72 T73 F109 W116 Y190 D220 G222 D80 S83 N85 A87 Y119 D276 T279 D33 S36 N38 A40 Y72 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=44nM remove_due_to_license_issue P56817 23010268 501 VEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4exg A 1.8 BS01 916 A 1 L78 D80 G82 Y119 T120 F156 W163 Y246 D276 G278 L31 D33 G35 Y72 T73 F109 W116 Y190 D220 G222 D80 S83 N85 A87 Y119 D276 T279 D33 S36 N38 A40 Y72 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=8.5nM remove_due_to_license_issue P56817 23010268 500 VEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4exs B 2.4 BS01 X8Z B 1 V73 H122 D124 H189 N220 H250 V32 H81 D83 H148 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 Ki=39uM remove_due_to_license_issue Kd=14000nM, IC50=50119nM C7C422 22713171 301 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLRLV 4exz A 1.608 BS01 RET A 1 F16 M20 Y60 L77 W106 K108 F16 M20 Y60 L77 W106 K108 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 23224553 202 TRDQNGTWEMESNENFEGYMKALDIDFATRKIAVRLTQTLVIDQDGDNFKTKTTSTFRNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGNKLYLELTCGDQVCRQVFKKK 4eyj A 2.102 BS01 N61 A 1 V39 A52 E72 I85 M107 M110 L167 D168 F169 V38 A51 E71 I84 M106 M109 L166 D167 F168 D150 K152 N155 D168 T185 D149 K151 N154 D167 T172 2.7.11.24 0000165,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005737,0005829,0006468,0006970,0007254,0018105,0032755,0033554,0034644,0035556,0050729,0051403,0070301,0071347,0072709,0072740,0106310,1903936 remove_due_to_license_issue IC50=619.5nM O15264 23187130 401 SLIRKKGFYKQDVNKTAWELPKTYVSPTHVGSGAYGSVCSAIDKRSGEKVAIKKLSRPFQSEIFAKRAYRELLLLKHMQHENVIGLLDVFTPASSLRNFYDFYLVMPFMQTDLQKIMGMEFSEEKIQYLVYQMLKGLKYIHSAGVVHRDLKPGNLAVNEDCELKILDFGLVTRWYRAPEVILSWMHYNQTVDIWSVGCIMAEMLTGKTLFKGKDYLDQLTQILKVTGVPGTEFVQKLNDKAAKSYIQSLPQTPRKDFTQLFPRASPQAADLLEKMLELDVDKRLTAAQALTHPFFEPFRDPEEETEAQQPFDDSLEHEKLTVDEWKQHIYKEIVNFSP 4eym A 2.353 BS01 0RX A 1 A52 K54 R68 E72 M107 D168 F169 A51 K53 R67 E71 M106 D167 F168 D150 K152 N155 D168 T185 D149 K151 N154 D167 T174 2.7.11.24 0000165,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005737,0005829,0006468,0006970,0007254,0018105,0032755,0033554,0034644,0035556,0050729,0051403,0070301,0071347,0072709,0072740,0106310,1903936 remove_due_to_license_issue IC50=14884nM O15264 23187130 401 SLIRKKGFYKQDVNKTAWELPKTYVSPTHVGSGAYGSVCSAIDKRSGEKVAIKKLSRPFQSEIFAKRAYRELLLLKHMQHENVIGLLDVFTPASSLRNFYDFYLVMPFMQTDLQKIMGMEFSEEKIQYLVYQMLKGLKYIHSAGVVHRDLKPGNLAVNEDCELKILDFGLYVVTRWYRAPEVILSWMHYNQTVDIWSVGCIMAEMLTGKTLFKGKDYLDQLTQILKVTGVPGTEFVQKLNDKAAKSYIQSLPQTPRKDFTQLFPRASPQAADLLEKMLELDVDKRLTAAQALTHPFFEPFRDPEEETEAQQPFDDSLEHEKLTVDEWKQHIYKEIVNFSP 4eyr A 1.8 BS01 RIT B 1 L23 N25 G27 A28 D29 D30 T82 L23 N25 G27 A28 D29 D30 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q000H7 23313846 301 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 4eyr B 1.8 BS01 RIT B 1 R8 N25 G27 A28 D29 D30 T82 R8 N25 G27 A28 D29 D30 T82 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=237nM remove_due_to_license_issue Q000H7 23313846 301 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 4ez3 A 2.0 BS01 0S0 A 1 I10 A31 F80 F82 L83 H84 Q85 D86 K89 L134 I10 A31 F76 F78 L79 H80 Q81 D82 K85 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 22893598 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4ez5 A 2.7 BS01 0RS A 1 I19 V27 A41 K43 V77 E99 H100 V101 Q149 N150 L152 A162 D163 I9 V16 A30 K32 V57 E71 H72 V73 Q121 N122 L124 A134 D135 D145 K147 Q149 N150 D163 T182 D117 K119 Q121 N122 D135 T141 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue IC50=300nM Q00534 24900493 900 QQYECVAEIGEGAGKVFKARDLKNGGRFVALKRVPLSTIREVAVLRHLETFEHPNVVRLFDVCTKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLAVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPRDVALPRQAFHSAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQ 4ezj A 2.67 BS01 0SC A 1 M804 W812 I831 K833 D841 Y867 I879 E880 I881 V882 M953 I963 D964 M559 W567 I586 K588 D596 Y622 I634 E635 I636 V637 M708 I718 D719 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=1585nM P48736 22672799 1201 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCTVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLG 4ezk A 2.803 BS01 0SD A 1 W812 I831 Y867 E880 I881 V882 K890 M953 I963 D964 W575 I594 Y630 E643 I644 V645 K653 M716 I726 D727 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 22672799 4000 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCTVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 4ezl A 2.94 BS01 0SE A 1 M804 I831 I879 I881 V882 T887 M953 I963 D964 M559 I586 I634 I636 V637 T642 M708 I718 D719 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 22672799 1201 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCTVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVLG 4f08 A 2.82 BS01 1RS A 1 L855 A880 Y931 L932 L983 L13 A38 Y89 L90 L141 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S174 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=250nM, EC50=>8800nM O60674 22698084 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4f09 A 2.4 BS01 JAK A 1 V863 A880 M929 Y931 L932 L983 V21 A38 M87 Y89 L90 L141 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S174 2.7.10.2 0004672,0004713,0005524,0006468 Ki=200nM remove_due_to_license_issue Ki=200nM, EC50=>8200nM O60674 22698084 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4f0c A 1.901 BS01 GDS A 1 G15 P16 N17 H44 R57 I58 E73 S74 G114 P115 W122 W176 G14 P15 N16 H43 R56 I57 E72 S73 G113 P114 W121 W175 G15 G14 ? 0016740 remove_due_to_license_issue I7B368 26348000 301 SHGKQFTLFNHQVGPNGWKVDMLLRELGLSFETVYVNLGQREHKSPSFTKYNPNGRIPALIDHYYNDFVVWESDAILLYIVEKYDPEHKFSVSTFDDKIIMTQWLFFQASGQGPYFGQAGWFLAVAPPEERNPTIAERYQKEILRVFGVLESVLSQRQWLVADKLTIADISFVIWNATAVNLLVKGYKGFDFEKDFPSVHRWHTALITRPAIAESLKTKAEAIAQMNR 4f1l A 1.9 BS01 0RY A 1 H1601 G1602 N1624 Y1633 F1634 A1635 Y1640 S1641 Y1646 H68 G69 N91 Y100 F101 A102 Y107 S108 Y113 2.4.2.- 0003950 remove_due_to_license_issue IC50=>20000nM, Kd=7600nM Q460N5 22823910 1801 QNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4f1q A 2.8 BS01 0RZ A 1 H1601 G1602 Y1633 Y1640 S1641 Y1646 H70 G71 Y98 Y105 S106 Y111 2.4.2.- 0003950 remove_due_to_license_issue IC50=>20000nM, Kd=11200nM Q460N5 22823910 1801 KQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4f1s A 3.0 BS01 F1S A 1 M804 I831 K833 Y867 I879 E880 V882 M953 I963 D964 M562 I589 K591 Y625 I637 E638 V640 M709 I719 D720 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 22832322 1207 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEWVSLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNPIALPKHQAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 4f2j C 2.64 BS01 dna A 0 Y484 K511 T512 R515 Y14 K41 T42 R45 ? remove_due_to_license_issue O75362 23436653 0 ~ 19 RECSYCGKFFRSNYYLNIHLRTHTGEKPYKCEFCEYAAAQKTSLRYHLERHH 4f2w A 2.0 BS01 TDI A 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 0003824,0008782,0008930,0009116,0009164,0019509 Ki=5pM remove_due_to_license_issue 23685211 301 MKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLAH 4f2w B 2.0 BS01 TDI B 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I57 S83 A84 G85 F158 I159 E179 M180 E181 D204 F214 0003824,0008782,0008930,0009116,0009164,0019509 Ki=5pM remove_due_to_license_issue 23685211 301 LVPRGSHMKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLA 4f39 A 1.834 BS01 KAI A 1 Y61 P89 T91 R96 L138 G141 S142 T143 E193 Y58 P86 T88 R93 L135 G138 S139 T140 E190 ? 0015276,0016020 Ki=3.44uM remove_due_to_license_issue EC50=40000nM, Ki=5780nM P19492 22512472 301 RTIVVTTILESPYVMYKKNHEQLEGNERYEGYCVDLAYEIAKHVRIKYKLSIVGDGKYGARDPETKIWNGMVGELVYGRADIAVAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLAKQTEIAYGTLDSGSTKEFFRRSKIAVYEKMWSYMKSAEPSVFTKTTADGVARVRKSKGKFAFLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGVATPKGSALGTPVNLAVLKLSEQGILDKLKNKWWYDKGEC 4f3c A 1.93 BS01 BIG A 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 0003824,0008782,0008930,0009116,0009164,0019509 Ki=1.5pM remove_due_to_license_issue 23685211 301 MKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLA 4f3c B 1.93 BS01 BIG B 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 0003824,0008782,0008930,0009116,0009164,0019509 Ki=1.5pM remove_due_to_license_issue 23685211 301 MKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLA 4f3h A 2.5 BS01 C2E A 1 Q26 F42 L43 R44 S53 P54 N55 D71 R97 E216 F217 Q236 G237 D238 Q26 F42 L43 R44 S53 P54 N55 D71 R97 E216 F217 Q236 G237 D238 ? 0071111 remove_due_to_license_issue Q8P8F1 22993092 501 EEERIERWVEQLREALIGDGFLLHYQPVLNLQGEPLELYQAFLRLERNGEMMSPNAFMAIAEEHDLITEIDRWVVARAIRQLGERQRAGHKTHLLVRIGPNSFSDPQMIDTIREQLAVYGVPGERLWLQTPESKVFTHLRNAQQFLASVSAMGCKVGLEQFGSGLDSFQLLAHFQPAFLKLDRSITGDIASARESQEKIREITSRAQPTGILTVAEFVADAQSMSSFFTAGVDYVQGDFVAPTGPLM 4f3i A 1.4 BS01 0S6 A 1 W81 P82 L92 L94 N140 I146 M149 W40 P41 L51 L53 N99 I105 M108 ? Kd=36.1nM remove_due_to_license_issue Ki=17nM, IC50=18.2nM O60885 22645123 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4f3k A 1.85 BS01 HCE A 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 0003824,0008782,0008930,0009116,0009164,0019509 Ki=69pM remove_due_to_license_issue 23685211 301 MKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLA 4f3k A 1.85 BS02 HCE B 1 F105 Y107 F105 Y107 0003824,0008782,0008930,0009116,0009164,0019509 Ki=69pM remove_due_to_license_issue 23685211 301 MKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLA 4f3k B 1.85 BS01 HCE B 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 0003824,0008782,0008930,0009116,0009164,0019509 Ki=69pM remove_due_to_license_issue 23685211 301 MKIGIIGAMEEEVTLLRDKIDNRQTITLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLASTLKVGDIVVSDETRYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAESCIRELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPDAVAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSTLMVETLVQKLA 4f49 A 2.25 BS01 K36 A 1 H41 F139 I140 C144 H162 L164 E165 Q187 H42 F140 I141 C145 H163 L165 E166 Q188 H41 G142 C144 H42 G143 C145 3.4.19.12,3.4.22.- 0008233,0019082 remove_due_to_license_issue P0C6V2 22915796 401 HSGLRKMAQPSGLVEPCIVRVSYGNNVLNGLWLGDEVICPRHVIASDTTRVINYENEMSSVRLHNFSVSKNNVFLGVVSARYKGVNLVLKVNQVNPNTPEHKFKSIKAGESFNILACYEGCPGSVYGVNMRSQGTIKGSFIAGTCGSVGYVLENGILYFVYMHHLELGNGSHVGSNFEGEMYGGYEDQPSMQLEGTNVMSSDNVVAFLYAALINGERWFVTNTSMSLESYNTWAKTNSFTELSSTDAFSMLAAKTGQSVEKLLDSIVRLNKGFGGRTILSYGSLCDEFTPTEVIRQMYGV 4f4p A 2.37 BS01 0SB A 1 L377 V385 A400 M448 A451 G454 P455 N499 L501 S511 L13 V21 A30 M73 A76 G79 P80 N124 L126 S136 D494 A496 R498 N499 D512 K533 D119 A121 R123 N124 D137 K158 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM remove_due_to_license_issue P43405 22877633 701 LDRKLLTLEDKELGSGNFGTVKKGYVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEG 4f5y A 2.396 BS02 C2E A 1 S162 Y167 R238 V239 T263 S12 Y17 R88 V89 T113 ? 0002218,0032481 Kd=3.7uM (22728660) remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22728660 402 GNFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEKEEVTV 4f5y B 2.396 BS01 C2E A 1 S162 Y167 T263 P264 S12 Y17 T113 P114 ? 0002218,0032481 Kd=3.7uM (22728660) remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22728660 402 GNFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEKEEVTV 4f63 A 2.55 BS01 0S7 A 1 L484 A512 Y563 A564 S565 G567 L630 L21 A40 Y91 A92 S93 G95 L146 D623 A625 R627 N628 D641 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue IC50=501.19nM P11362 22612866 801 ELPEDPRWELPRDRLVLGKPLGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS 4f64 A 2.05 BS01 0S8 A 1 L484 A512 V561 A564 S565 G567 L630 L21 A40 V89 A92 S93 G95 L146 D623 A625 R627 N628 D641 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=63nM remove_due_to_license_issue IC50=794.33nM P11362 22612866 801 ELPEDPRWELPRDRLVLGKPLGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS 4f65 A 2.26 BS01 0S9 A 1 L484 E486 V492 A512 K514 E531 V561 Y563 A564 S565 G567 L630 L21 E23 V29 A47 K49 E66 V96 Y98 A99 S100 G102 L154 D623 A625 R627 N628 D641 D147 A149 R151 N152 D165 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=2.5nM remove_due_to_license_issue IC50=63.1nM P11362 22612866 808 ELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4f6n A 2.8 BS01 dna D 0 R501 Y503 V504 S508 R511 E535 Y536 Q563 Y597 A598 R21 Y23 V24 S28 R31 E55 Y56 Q83 Y117 A118 ? remove_due_to_license_issue Q86T24 22949637 1 ~ 19 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAEYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQYAYL 4f6n A 2.8 BS02 dna E 0 R511 K520 E535 T538 R549 Y550 Y562 S578 Y584 L586 R595 Y597 R31 K40 E55 T58 R69 Y70 Y82 S98 Y104 L106 R115 Y117 ? remove_due_to_license_issue Q86T24 22949637 21 ~ 38 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAEYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQYAYL 4f6s A 2.6 BS01 0SQ A 1 Y32 S62 E66 A172 D173 Y33 S63 E67 A165 D166 D151 K153 N156 D173 T196 D144 K146 N149 D166 T172 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 KMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFAVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4f6u A 2.1 BS01 0SR A 1 Y32 A50 S62 R65 E66 I79 F97 A100 I171 A172 D173 Y34 A52 S64 R67 E68 I81 F99 A102 I168 A169 D170 D151 K153 N156 D173 T196 D148 K150 N153 D170 T176 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 DKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQENPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4f6v A 2.3 BS01 ZYM A 1 F22 Y41 C44 R45 D48 V133 V137 N168 F22 Y41 C44 R45 D48 V130 V134 N165 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 ic50=24uM remove_due_to_license_issue IC50=24000nM, Ki=250nM A9JQL9 22662288 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 4f6w A 2.39 BS01 0SS A 1 V27 Y32 S62 E66 F97 W105 A172 D173 M174 R356 V27 Y32 S62 E66 F97 W105 A167 D168 M169 R327 D151 K153 N156 D173 T196 D146 K148 N151 D168 T173 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 MDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFATFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4f6x A 1.98 BS01 ZYL A 1 H18 F22 A134 V137 L164 Q165 N168 F233 Y248 H18 F22 A131 V134 L161 Q162 N165 F230 Y245 2.5.1.96 0003824,0004311,0009058,0016117,0016740,0016765,0046872,0051996 ic50=45.3uM remove_due_to_license_issue IC50=45300nM, Ki=450nM A9JQL9 22662288 301 MTMMDMNFKYCHKIMKKHSKSFSYAFDLLPEDQRKAVWAIYAVCRKIDDSIDDIQFLNQIKEDIQSIEKYPYEYHHFQSDRRIMMALQHVAQHKNIAFQSFYNLIDTVYKDQHFTMFETDAELFGYCYGVAGTVGEVLTPILSDHETHQTYDVARRLGESLQLINILRDVGEDFENERIYFSKQRLKQYEVDIAEVYQNGVNNHYIDLWEYYAAIAEKDFRDVMDQIKVFSIEAQPIIELAARIYIEILDEVRQANYTLHERVFVEKRKKAKLFHEINSKY 4f70 A 3.0 BS01 0ST A 1 S62 R65 E66 F97 D173 M174 S63 R66 E67 F98 D168 M169 D151 K153 N156 D173 T196 D146 K148 N151 D168 T171 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 KMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKALPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4f7j A 2.6 BS01 0SU A 1 Y32 K52 S62 R65 E66 A172 D173 Y32 K52 S62 R65 E66 A163 D164 D151 K153 N156 D173 T196 D142 K144 N147 D164 T169 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 MDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4f7l A 2.9 BS01 0SO A 1 Y32 V35 A50 S62 E66 F97 I171 A172 D173 R356 Y34 V37 A52 S64 E68 F99 I166 A167 D168 R325 D151 K153 N156 D173 T196 D146 K148 N151 D168 T171 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 DKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 4f7n A 2.65 BS01 0SV A 1 A50 S62 R65 E66 L70 I79 F97 L158 A172 D173 A51 S63 R66 E67 L71 I80 F98 L153 A167 D168 D151 K153 N156 D173 T196 D146 K148 N151 D168 T174 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 23630251 501 KMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQENPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTE 4f7v A 1.73 BS01 J1D A 1 T42 L45 Y53 N55 L70 Q74 E77 W89 R92 D95 L96 D97 I98 R110 L111 T112 Y116 F123 T42 L45 Y53 N55 L70 Q74 E77 W89 R92 D95 L96 D97 I98 R110 L111 T112 Y116 F123 R82 R92 D95 D97 R82 R92 D95 D97 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=4.16uM remove_due_to_license_issue IC50=9530nM, Kd=4160nM P26281 22727779 201 TVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4f8h A 2.99 BS01 RKE A 1 Y23 N152 D153 D154 Y19 N148 D149 D150 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 22958642 401 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 4f8h A 2.99 BS03 RKE E 1 F174 L176 K183 F170 L172 K179 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 22958642 401 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 4f8h B 2.99 BS01 RKE A 1 F174 L176 K183 F170 L172 K179 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 22958642 401 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 4f8h B 2.99 BS02 RKE B 1 Y23 N152 D153 D154 Y19 N148 D149 D150 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 22958642 401 VSPPPPIADEPLTVNTGIYLIECYSLDDKAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNLPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 4f9g A 2.95 BS01 C2E A 1 Y167 T263 P264 Y14 T97 P98 ? 0002218,0032481 Km=2.4+-0.5mM (22705373) remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22705373 401 NVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPNNCRLIAYQEPSFSLSQEVLRHLRQEEKEEVTV 4f9g C 2.95 BS01 C2E A 1 Y167 T263 P264 Y14 T97 P98 ? 0002218,0032481 Km=2.4+-0.5mM (22705373) remove_due_to_license_issue EC50=4500nM, Kd=1210nM Q86WV6 22705373 401 NVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPNNCRLIAYQEPFSLSQEVLRHLRQEEKEEVTV 4f9u A 1.8 BS02 PBD A 1 D131 E170 E171 W176 D218 V270 D271 F292 H297 D99 E138 E139 W144 D179 V231 D232 F253 H258 2.3.2.5 0005576,0008270,0016603,0016746,0046872 Ki=3139nM remove_due_to_license_issue Q9VRQ9 22897232 402 QWRDDEVHFNRTLDSILVPRVVGSRGHQQVREYLVQSLNGLGFQTEVDEFKQRVPVFGELTFANVVGTINPQAQNFLALACHYDSKYFPNDPGFVGATDSAVPCAILLNTAKTLGAYLQKEFRNRSDVGLMLIFFDGEEAFKEWTDADSVYGSKHLAAKLASKRSPRNIDRIEVLVLLDLIGARNPKFSSFYENTDGLHSSLVQIEKSLRTAGQLEGNNNMFLSRVSGGLVDDDHRPFLDENVPVLHLVATPFPDVWHTPRDNAANLHWPSIRNFNRVFRNFVYQYLKRHTSPVNLRF 4f9v A 2.1 BS02 PBD A 1 D131 E170 E171 W176 D218 D271 F292 W296 H297 D102 E141 E142 W147 D189 D242 F263 W267 H268 2.3.2.5 0005576,0008270,0016603,0016746,0046872 remove_due_to_license_issue Q9VRQ9 22897232 402 IGSQWRDDEVHFNRTLDSILVPRVVGSRGHQQVREYLVQSLNGLGFQTEVDEFKQRVPVFGELTFANVVGTINPQAQNFLALAAHYDSKYFPNDPGFVGATDSAVPAAILLNTAKTLGAYLQKEFRNRSDVGLMLIFFDGEEAFKEWTDADSVYGSKHLAAKLASKRSGSQAQLAPRNIDRIEVLVLLDLIGARNPKFSSFYENTDGLHSSLVQIEKSLRTAGQLEGNNNMFLSRVSGGLVDDDHRPFLDENVPVLHLVATPFPDVWHTPRDNAANLHWPSIRNFNRVFRNFVYQYLKRHTSPVNLR 4f9v A 2.1 BS03 PBD B 1 V88 F89 V59 F60 2.3.2.5 0005576,0008270,0016603,0016746,0046872 remove_due_to_license_issue Q9VRQ9 22897232 402 IGSQWRDDEVHFNRTLDSILVPRVVGSRGHQQVREYLVQSLNGLGFQTEVDEFKQRVPVFGELTFANVVGTINPQAQNFLALAAHYDSKYFPNDPGFVGATDSAVPAAILLNTAKTLGAYLQKEFRNRSDVGLMLIFFDGEEAFKEWTDADSVYGSKHLAAKLASKRSGSQAQLAPRNIDRIEVLVLLDLIGARNPKFSSFYENTDGLHSSLVQIEKSLRTAGQLEGNNNMFLSRVSGGLVDDDHRPFLDENVPVLHLVATPFPDVWHTPRDNAANLHWPSIRNFNRVFRNFVYQYLKRHTSPVNLR 4f9w A 2.0 BS03 LM4 A 1 V38 A51 K53 L104 V105 T106 M109 L167 V34 A47 K49 L100 V101 T102 M105 L163 D150 K152 N155 D168 T185 D146 K148 N151 D164 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=114nM remove_due_to_license_issue IC50=210nM, Ki=110nM Q16539 23840427 403 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4f9y A 1.85 BS03 LM3 A 1 V38 A51 V52 K53 I84 L104 T106 M109 L167 V34 A47 V48 K49 I80 L100 T102 M105 L163 D150 K152 N155 D168 T185 D146 K148 N151 D164 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Ki=184nM remove_due_to_license_issue IC50=190nM, Ki=180nM Q16539 23840427 403 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 4fab H 2.7 BS01 FLU H 1 W33 Y102 Y103 W33 Y102 Y103 ? remove_due_to_license_issue P01865 2508085 218 EVKLDETGGGLVQPGRPMKLSCVASGFTFSDYWMNWVRQSPEKGLEWVAQIRNKPYNYETYYSDSVKGRFTISRDDSKSSVYLQMNNLRVEDMGIYYCTGSYYGMDYWGQGTSVTVSSAKTTAPSVYPLAPVCGDTTGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIE 4fab L 2.7 BS01 FLU H 1 H31 Y37 S96 W101 H31 Y37 S96 W101 remove_due_to_license_issue 2508085 218 DVVMTQTPLSLPVSLGDQASISCRSSQSLVHSQGNTYLRWYLQKPGQSPKVLIYKVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYFCSQSTHVPWTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 4fai A 1.65 BS02 PBD A 1 D153 E190 E191 W196 D228 E292 F313 W317 H318 D121 E158 E159 W164 D196 E245 F266 W270 H271 2.3.2.5 0005576,0005739,0008270,0016603,0016746,0046872 remove_due_to_license_issue Q86PD7 22897232 402 ELVDIPKISYNPSELSEPRFLEYSNLSDKLHLREAIDKILIPRVVGTTNHSIVREYIVQSLRDLDWDVEVNSFHDHAPIKGKLHFHNIIATLNPNAERYLVLSCHYDSKYMPGVEFLGATDSAVPCAMLLNLAQVLQEQLKPLKKSKLSLMLLFFDGEEAFEEWGPKDSIYGARHLAKKWHHEGKLDRIDMLVLLDLLGAPDPAFYSFFENTESWYMRIQSVETRLAKLQLRYFQSQAMRSSFIEDDHIPFLRRNVPILHLIPVPFPSVWHTPDDNASVIDYATTDNLALIIRLFALEYLLA 4fak A 1.7 BS01 SAM A 1 L76 E77 I78 I107 G108 S110 G112 S126 F127 S128 F132 M137 L80 E81 I82 I111 G112 S114 G116 S130 F131 S132 F136 M141 2.1.1.177 0005737,0006364,0008168,0031167,0032259,0070038 remove_due_to_license_issue P0C1V0 23150671 201 AAEFMKITILAVGKLKEKYWKQAIAEYEKRLGPYTKIDIIEVPDEKAPENMSDKEIEQVKEKEGQRILAKIKPQSTVITLEIQGKMLSSEGLAQELNQRMTQGQSDFVFVIGGSNGLHKDVLQRSNYALSFSKMTFPHQMMRVVLIEQVYRAFKIMRGEAYHK 4fb3 A 3.79 BS01 dna C 0 N307 T309 K355 H356 R357 A360 N18 T20 K66 H67 R68 A71 3.6.4.- 0003688,0006260 remove_due_to_license_issue P0DOJ4 24109229 1 ~ 26 SDFPSSLTGYLSHAIYSNKTFPAFLVYSTKEKCKQLYDTIGKFRPEFKCLVHYEEGGMLFFLTMTKHRVSAVKNYCSKLCSVSFLMCKAVTKPMECYQVVTAAPFQLITENKPGL 4fb3 A 3.79 BS02 dna W 0 S301 H302 A303 I304 Y305 S306 N307 K308 S12 H13 A14 I15 Y16 S17 N18 K19 3.6.4.- 0003688,0006260 remove_due_to_license_issue P0DOJ4 24109229 1 ~ 26 SDFPSSLTGYLSHAIYSNKTFPAFLVYSTKEKCKQLYDTIGKFRPEFKCLVHYEEGGMLFFLTMTKHRVSAVKNYCSKLCSVSFLMCKAVTKPMECYQVVTAAPFQLITENKPGL 4fb3 B 3.79 BS01 dna C 0 S301 Y305 S306 N307 K308 S12 Y16 S17 N18 K19 3.6.4.- 0003688,0006260 remove_due_to_license_issue P0DOJ4 24109229 1 ~ 26 SDFPSSLTGYLSHAIYSNKTFPAFLVYSTKEKCKQLYDTIGKFRPEFKCLVHYEEGGMLFFLTMTKHRVSAVKNYCSKLCSVSFLMCKAVTKPMECYQVVTAAPFQLITENKPG 4fb3 B 3.79 BS02 dna W 0 N307 T309 K355 H356 R357 A360 N18 T20 K66 H67 R68 A71 3.6.4.- 0003688,0006260 remove_due_to_license_issue P0DOJ4 24109229 1 ~ 26 SDFPSSLTGYLSHAIYSNKTFPAFLVYSTKEKCKQLYDTIGKFRPEFKCLVHYEEGGMLFFLTMTKHRVSAVKNYCSKLCSVSFLMCKAVTKPMECYQVVTAAPFQLITENKPG 4fb3 E 3.79 BS01 dna C 0 N307 T309 K355 H356 R357 A360 N363 N18 T20 K66 H67 R68 A71 N74 3.6.4.- 0003688,0006260 remove_due_to_license_issue P0DOJ4 24109229 1 ~ 26 SDFPSSLTGYLSHAIYSNKTFPAFLVYSTKEKCKQLYDTIGKFRPEFKCLVHYEEGGMLFFLTMTKHRVSAVKNYCSKLCSVSFLMCKAVTKPMECYQVVTAAPFQLITENKPG 4fb3 E 3.79 BS02 dna W 0 S301 H302 A303 I304 Y305 S306 N307 K308 T380 S12 H13 A14 I15 Y16 S17 N18 K19 T91 3.6.4.- 0003688,0006260 remove_due_to_license_issue P0DOJ4 24109229 1 ~ 26 SDFPSSLTGYLSHAIYSNKTFPAFLVYSTKEKCKQLYDTIGKFRPEFKCLVHYEEGGMLFFLTMTKHRVSAVKNYCSKLCSVSFLMCKAVTKPMECYQVVTAAPFQLITENKPG 4fbe A 1.88 BS01 PBD A 1 D153 E190 E191 W196 D228 E292 F313 H318 D121 E158 E159 W164 D196 E247 F268 H273 2.3.2.5 0005576,0005739,0008270,0016603,0016746,0046872 remove_due_to_license_issue Q86PD7 22897232 401 ELVDIPKISYNPSELSEPRFLEYSNLSDKLHLREAIDKILIPRVVGTTNHSIVREYIVQSLRDLDWDVEVNSFHDHAPIKGKLHFHNIIATLNPNAERYLVLSAHYDSKYMPGVEFLGATDSAVPAAMLLNLAQVLQEQLKPLKKSKLSLMLLFFDGEEAFEEWGPKDSIYGARHLAKKWHHEGKLDRIDMLVLLDLLGAPDPAFYSFFENTESWYMRIQSVETRLAKLQLLERYFQSQAMRSSFIEDDHIPFLRRNVPILHLIPVPFPSVWHTPDDNASVIDYATTDNLALIIRLFALEYLL 4fc0 A 2.95 BS01 0T2 A 1 A480 K482 E500 V503 L504 L513 I526 T528 W530 C531 G533 G592 D593 F594 A34 K36 E54 V57 L58 L67 I80 T82 W84 C85 G87 G146 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S151 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=69nM P15056 22883026 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGGSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP 4fcb A 2.1 BS02 0T7 A 1 L665 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 L228 I245 Y246 F249 P265 M266 E274 V275 G278 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=2.9nM remove_due_to_license_issue Q9Y233 22902656 803 MSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4fcd A 2.02 BS02 0T6 A 1 H515 I682 F686 M703 Q716 F719 H78 I245 F249 M266 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=0.28nM remove_due_to_license_issue IC50=0.28nM Q9Y233 22902656 803 MSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4fcf A 1.09 BS01 MA4 A 1 V224 P226 I246 A248 V261 A284 E288 V199 P201 I220 A222 V234 A257 E261 S70 K73 S130 E166 R234 A237 S45 K48 S105 E141 R209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 23252553 301 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADRTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 4fci A 1.82 BS03 GPA A 1 H126 D128 N130 S137 H141 D183 H122 D124 N126 S133 H137 D179 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue P05089 22869115 403 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDY 4fck A 1.9 BS01 GPA A 1 H126 D128 S137 D183 T246 H121 D123 S132 D178 T241 H101 D124 H126 D128 H141 D232 D234 E277 H96 D119 H121 D123 H136 D227 D229 E272 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue P05089 22869115 401 RTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 4fcq A 2.151 BS01 2N6 A 1 N51 S52 A55 D93 G97 M98 L107 T109 F138 T184 N36 S37 A40 D78 G82 M83 L92 T94 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.156uM remove_due_to_license_issue P07900 23018093 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4fcr A 1.698 BS01 0TM A 1 N51 S52 A55 K58 D93 G97 M98 N106 L107 F138 T184 N36 S37 A40 K43 D78 G82 M83 N91 L92 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.4nM remove_due_to_license_issue P07900 23018093 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIASGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4fe6 A 2.0 BS01 0TQ A 1 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki<0.1nM remove_due_to_license_issue P03367 22749283 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4fea A 3.79 BS01 0TE B 1 V292 M294 V159 M161 H144 C186 H74 C105 3.4.22.60 0004197,0006508,0008234 remove_due_to_license_issue P55210 22795132 701 TYQYNMNFEKLGKCIIINNKDKDAEALFKCFRSLGFDVIVYNDCSCAKMQDLLKKASEEDHTNAACFACILLSHVTPIKDLTAHFRGDRCKTLLEKPKLFFIQACPVEADFLFAYSTVRGSWFVQALCSILEEHGKDLEIMQILTRVNDRVARHIPCVVSMLTKELYFSQ 4fea B 3.79 BS01 0TE A 1 E216 F221 E133 F138 G85 V86 H144 G145 C186 G29 V30 H88 G89 C130 3.4.22.60 0004197,0006508,0008234 remove_due_to_license_issue P55210 22795132 701 TYQYNMNFEKLGKCIIINNKNFDKVTGMGVRNGTDKDAEALFKCFRSLGFDVIVYNDCSCAKMQDLLKKASEEDHTNAACFACILLSHGEENVIYGKDGVTPIKDLTAHFRGDRCKTLLEKPKLFFIQACPVEADFLFAYSPGRGSWFVQALCSILEEHGKDLEIMQILTRVNDRVARHFIPCVVSMLTKELYFSQ 4feq A 2.2 BS01 0T8 A 1 L514 A538 L593 F595 M596 K597 H598 M652 D663 L10 A29 L61 F63 M64 K65 H66 M113 D124 D645 A647 R649 N650 D663 D106 A108 R110 N111 D124 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1.1uM remove_due_to_license_issue P55144 23312472 901 EQQFTLGRMLGKGSVREAQLKDGSFVKVAVKMLFLREAACMKEFDHPHVAKLVGVSPMVILPFMKHGDLHAFLLASRIPLQTLVRFMVDIACGMEYLSSRNFIHRDLAARNCMLAEDMTVCVADFGVKWLALESLADNLYTVHSDVWAFGVTMWEIMTRGQTPYAGIENAEIYNYLIGGNRLKQPPECMEEVYDLMYQCWSADPKQRPSFTCLRMELENILGHL 4fev A 1.89 BS02 PP1 A 1 F53 I101 Q108 I215 F45 I93 Q100 I207 K55 D198 N203 D216 K47 D190 N195 D208 0005524,0016773,0046677 remove_due_to_license_issue 23758273 302 QRETSCSRPNLDADLYGYRWARDNVGQSGATIYRLYGKPNAPELFLKHGKGSVANDVTDEMVRLNWLTAFMPLPTIKHFIRTPDDAWLLTTAIPGKTAFQVLEEYPDSGENIVDALAVFLRRLHSIPVCNCPFNSDRVFRLAQAQSRMNNGLVDASDFDDERNGWPVEQVWKEMHKLLPFSPDSVVTHGDFSLDNLIFDEGKLIGCIDVGRVGIADRYQDLAILWNCLGEFSPSLQKRLFQKYGIDNPDMNKLQFHLMLDEFF 4few A 1.98 BS02 PP2 A 1 F53 A100 I101 Q108 I215 F48 A95 I96 Q103 I210 K55 D198 N203 D216 K50 D193 N198 D211 0005524,0016773,0046677 remove_due_to_license_issue 23758273 302 RETSCSRPRLNSNLDADLYGYRWARDNVGQSGATIYRLYGKPNAPELFLKHGKGSVANDVTDEMVRLNWLTAFMPLPTIKHFIRTPDDAWLLTTAIPGKTAFQVLEEYPDSGENIVDALAVFLRRLHSIPVCNCPFNSDRVFRLAQAQSRMNNGLVDASDFDDERNGWPVEQVWKEMHKLLPFSPDSVVTHGDFSLDNLIFDEGKLIGCIDVGRVGIADRYQDLAILWNCLGEFSPSLQKRLFQKYGIDNPDMNKLQFHLMLDEFF 4ff8 A 2.4 BS01 14S A 1 A571 L593 P594 F595 M596 K597 G599 D600 M652 A662 A9 L14 P15 F16 M17 K18 G20 D21 M66 A76 D645 A647 R649 N650 D59 A61 R63 N64 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.4uM remove_due_to_license_issue P55144 23312472 901 KEFDHPHVAKLVILPFMKHGDLHAFLLASRIPLQTLVRFMVDIACGMEYLSSRNFIHRDLAARNCMLAEDMTVCVAVKWLALESLADNLYTVHSDVWAFGVTMWEIMTRGQTPYAGIENAEIYNYLIGGNRLKQPPECMVYDLMYQCWSADPKQRPSFTCLRMELENIL 4ffs A 1.9 BS01 BIG A 1 M10 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 M12 I54 V80 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=36pM remove_due_to_license_issue Q9ZMY2 22891633 301 EFMQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4fgn A 3.2 BS01 dna Z 0 N153 T155 R202 H203 R204 A207 N210 N21 T23 R70 H71 R72 A75 N78 3.6.4.- 0003688,0006260 remove_due_to_license_issue P03070 23269808 1 ~ 23 EDPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDFN 4fgn A 3.2 BS02 dna Y 0 S147 A149 V150 F151 S152 N153 R154 N227 K228 S15 A17 V18 F19 S20 N21 R22 N95 K96 3.6.4.- 0003688,0006260 remove_due_to_license_issue P03070 23269808 1 ~ 23 EDPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDFN 4fgn B 3.2 BS01 dna Z 0 N153 R202 H203 R204 A207 N210 N20 R69 H70 R71 A74 N77 3.6.4.- 0003688,0006260 remove_due_to_license_issue P03070 23269808 1 ~ 23 DPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDF 4fgn B 3.2 BS02 dna Y 0 S147 A149 F151 S152 N153 R154 N227 S14 A16 F18 S19 N20 R21 N94 3.6.4.- 0003688,0006260 remove_due_to_license_issue P03070 23269808 1 ~ 23 DPKDFPSELLSFLSHAVFSNRTLACFAIYTTKEKAALLYKKIMEKYSVTFISRHNSYNHNILFFLTPHRHRVSAINNYAQKLCTFSFLICKGVNKEYLMYSALTRDPFSVIEESLPGGLKEHDF 4fgz A 1.994 BS01 CQA A 1 I30 F31 G32 G39 E42 L213 V216 E217 Y220 I22 F23 G24 G31 E34 L205 V208 E209 Y212 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 ic50=1350uM remove_due_to_license_issue IC50=1350000nM Q8IDQ9 22771008 301 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fgz A 1.994 BS02 CQA A 2 E171 Y175 G243 R246 K247 E163 Y167 G235 R238 K239 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 ic50=1350uM remove_due_to_license_issue IC50=1350000nM Q8IDQ9 22771008 302 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRDAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4fhh A 2.33 BS02 0U3 A 1 Y175 L261 S265 I299 M300 R302 S303 W314 Y323 V328 H333 Y22 L48 S52 I86 M87 R89 S90 W101 Y110 V115 H120 ? 0003677,0004879,0005634,0006355 ic50=35nM remove_due_to_license_issue Q9PTN2 22921063 501 HMLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV 4fhi A 2.4 BS02 0S4 A 1 Y175 L261 V262 Y264 S265 I299 R302 S303 W314 Y323 V328 H333 H423 Y427 Y21 L47 V48 Y50 S51 I85 R88 S89 W100 Y109 V114 H119 H209 Y213 ? 0003677,0004879,0005634,0006355 ic50=100nM remove_due_to_license_issue Q9PTN2 22921063 501 MLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV 4fic A 2.5 BS01 0UL A 1 A293 Y340 M341 G344 L393 A36 Y75 M76 G79 L128 D386 R388 A390 N391 D404 F424 D121 R123 A125 N126 D139 F142 2.7.10.2 0004672,0004713,0005524,0006468 ic50=20uM remove_due_to_license_issue IC50=2.0e+4nM P00523 23534475 601 LAKDAWEIPRESLRLEVKLGQGEVWMGTWNGTTRVAIKTLKPLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4fil A 2.4 BS01 0UE A 1 Y110 Y130 F186 Y191 Y193 W197 R199 W225 W279 Y280 Y64 Y84 F140 Y145 Y147 W151 R153 W179 W233 Y234 ? 0030288,0030313,0046872,1901678 Kd=0.034uM remove_due_to_license_issue A0A0H3JWU6 24606332 401 PKRIAVVAPTYAGGLKKLGANIVAVNQQVDQSKVLKDKFKGVTKIGDGDVEKVAKEKPDLIIVYSTDKDIAAYQAVAPTVVVDYNKHKYLEQQEMLGKIVGKEDKVKAWKKDWEETTAKDGKEIKKAIGQDATVSLFDEFDKKLYTYGDNWGRGGEVLYQAFGLKMQPEQQKLTAKAGWAEVKQEEIEKYAGDYIVSTSEGKPTPGYESTNMWKNLKATKEGHIVKVDAGTYWYNDPYTLDFMRKDLKEKLIKAAK 4fiv A 1.8 BS01 LP1 A 1 R13 D30 G32 A33 D34 M56 I57 R10 D27 G29 A30 D31 M53 I54 3.1.13.2,3.1.26.13 0004190,0006508 Ki=300nM remove_due_to_license_issue Q66972 9827997 201 VGTTTTLEKRPEILIFVNGYPIKFLLDTGADITILNRRDFQVKNSIENGRQNMIGVGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLIQPLLGRDNMIKFNIRLVM 4fj5 A 2.05 BS01 dna T 0 E219 I253 E254 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 E219 I253 E254 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj5 A 2.05 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj7 A 1.9 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj7 A 1.9 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj8 A 2.19 BS01 dna T 0 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 K878 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj8 A 2.19 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj9 A 1.97 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fj9 A 1.97 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjg A 2.02 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 G571 N572 K705 K706 R707 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 G571 N572 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjg A 2.02 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjh A 2.11 BS01 dna T 0 E219 I253 E254 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 E219 I253 E254 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 S784 N786 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjh A 2.11 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fji A 2.2 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 4fji A 2.2 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 K734 S735 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 K734 S735 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMFDF 4fjj A 1.99 BS01 dna T 0 E219 I253 E254 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 N255 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjj A 1.99 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjk A 2.0 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 K878 S360 P361 I362 Y391 P392 G393 A394 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjk A 2.0 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjl A 1.87 BS01 dna T 0 S360 P361 I362 Y391 P392 G393 A394 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 S360 P361 I362 Y391 P392 G393 A394 G568 N572 W574 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjl A 1.87 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjm A 2.02 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjm A 2.02 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSLYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjn A 1.98 BS01 dna T 0 D275 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 N572 K705 K706 R707 K800 F803 K844 K874 D275 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 N572 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 3 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDM 4fjn A 1.98 BS02 dna P 0 N284 D621 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDM 4fjx A 2.11 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 S784 N786 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 1 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjx A 2.11 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fjz A 3.0 BS01 4FJ A 1 M804 P810 W812 K833 E880 I881 V882 T887 K890 I963 D964 M553 P559 W561 K582 E629 I630 V631 T636 K639 I709 D710 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=509nM P48736 22876881 1205 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNIALPKAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSADVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 4fk0 A 2.18 BS01 dna T 0 E219 I253 D275 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 E219 I253 D275 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 N572 K705 K706 R707 P799 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDM 4fk0 A 2.18 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDM 4fk2 A 1.98 BS01 dna T 0 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 A569 N572 K705 K706 R707 P799 K800 F803 K844 K874 K878 E219 I253 E254 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 N564 G565 G568 A569 N572 K705 K706 R707 P799 K800 F803 K844 K874 K878 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fk2 A 1.98 BS02 dna P 0 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 D621 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fk4 A 1.9 BS01 dna T 0 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 K800 F803 K844 K874 E219 I253 R260 D275 F359 S360 P361 I362 Y391 P392 G393 A394 G568 N572 K705 K706 R707 K800 F803 K844 K874 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 2 ~ 18 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fk4 A 1.9 BS02 dna P 0 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 N284 T622 K706 Y708 M728 G729 K734 S735 S783 S784 N786 Y791 H804 2.7.7.7,3.1.11.- 0000166,0003676,0003677,0003887,0004527,0006260,0006261,0008408,0034061,0039686,0039693,0046872 remove_due_to_license_issue Q38087 23214497 103 ~ 115 MKEFYLTVEQIGDSIFERYIDSNGRERTREVEYKPSLFAHCPESQATKYFDIYGKPCTRKLFANMRDASQWIKRMEDIGLEALGMDDFKLAYLSDTYNYEIKYDHTKIRVANFDIEVTSPDGFPEPSQAKHPIDAITHYDSIDDRFYVFDLLNSPYGNVEEWSIEIAAKLQEQGGDEVPSEIIDKIIYMPFDNEKELLMEYLNFWQQKTPVILTGWNVESFAIPYVYNRIKNIFGESTAKRLSPHRKTRVKVIENMYGSREIITLFGISVLDYIDLYKKFSFTNQPSYSLDYISEFELNVGKLKYDGPISKLRESNHQRYISYNIIAVYRVLQIDAKRQFINLSLDMGYYAKIQIQSVFSPIKTWDAIIFNSLKEQNKVIPQGRSHPVQPYPGAFVKEPIPNRYKYVMSFDLTSAYPSIIRQVNISPETIAGTFKVAPLHDYINAVAERPSDVYSCSPNGMMYYKDRDGVVPTEITKVFNQRKEHKGYMLAAQRNGEIIKEALHNPNLSVDEPLDVDYRFDFSDEIKEKIKKLSAKSLNEMLFRAQRTEVAGMTAQINRKALINGLAGALGNVWFRYYDLRNATAITTFGQMALQWIERKVNEYLNEVCGTEGEAFVLYGDTDSIYVSADKIIDKVGESKFRDTNHWVDFLDKFARERMEPAIDRGFREMCEYMNNKQHLMFMDREAIAGPPLGSKGIGGFWTGKKRYALNVWDMEGTRYAEPKLKIMGLETQKSSTPKAVQKALKECIRRMLQEGEESLQEYFKEFEKEFRQLNYISIASVSSANNIAKYDVGGFPGPKCPFHIRGILTYNRAIKGNIDAPQVVEGEKVYVLPLREGNPFGDKCIAWPSGTEITDLIKDDVLHWMDYTVLLEKTFIKPLEGFTSAAKLDYEKKASLFDMF 4fk6 A 2.2 BS01 0UJ A 1 R879 L881 V889 A906 F958 L959 E966 R1007 N1008 L1010 R17 L19 V25 A42 F91 L92 E99 R140 N141 L143 D1003 A1005 R1007 N1008 D1021 D1040 D136 A138 R140 N141 D154 D173 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.2nM remove_due_to_license_issue Ki=3.2nM, EC50=355nM, IC50=1.000nM P23458 23107482 1201 TEVDPTHFEKRFLKRIRDLGEFGKVELCRYDPEGDNTGEQVAVKSLKPENHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4fk7 A 1.78 BS01 P34 A 1 R341 R342 S387 T388 S389 Y398 Q429 E431 R81 R82 S127 T128 S129 Y138 Q169 E171 S387 E431 S127 E171 2.4.2.- 0005576 Kd=5.8uM remove_due_to_license_issue Q4MV79 22992735 1001 VLDFKWYTRKAESWGVQTFKNWKENLTISEKDIITGYTGSKYDPINEYLRKKALEKIENQIKNLDAALQKSKITENLIVYRRVSELQFGKKYEDYNLRQNGIINEEKVMELESNFKGQTFIQHNYMSTSLVQDPHQSYSNDRYPILLEITIPEGVHGAYIADMSEYPGQYEMLINRGYTFKYDKFSIVKPGKEYLKVNLSIYL 4fkk A 2.6 BS01 BES A 1 A346 A348 M349 E350 H383 E384 H387 E406 Y472 A284 A286 M287 E288 H321 E322 H325 E344 Y410 E350 H383 E384 H387 E406 S464 Y472 E288 H321 E322 H325 E344 S402 Y410 3.4.11.2 0001525,0001618,0004177,0005615,0005737,0005886,0006508,0008237,0008270,0030154,0042277,0043171,0046718,0046872,0070006 remove_due_to_license_issue Ki=4100nM, IC50=9400nM P15145 23071329 1024 QSKPWNRYRLPTTLLPDSYNVTLRPYLTPNADGLYIFKGKSIVRFLCQEPTDVIIIHSKKLNYTTQGHMVVLRGVGDSQVPEIDRTELVELTEYLVVHLKGSLQPGHMYEMESEFQGELADDLAGFYRSEYMEGNVKKVLATTQMQSTDARKSFPCFDEPAMKATFNITLIHPNNLTALSNMPPKGSSTPLAEDPNWSVTEFETTPVMSTYLLAYIVSEFQSVNETAQNGVLIRIWARPNAIAEGHGMYALNVTGPILNFFANHYNTSYPLPKSDQIALPDFNAGAMENWGLVTYRENALLFDPQSSSISNKERVVTVIAHELAHQWFGNLVTLAWWNDLWLNEGFASYVEYLGADHAEPTWNLKDLIVPGDVYRVMAVDALASSHPLTTPAEEVNTPAQISEMFDSISYSKGASVIRMLSNFLTEDLFKEGLASYLHAFAYQNTTYLDLWEHLQKAVDAQTSIRLPDTVRAIMDRWTLQMGFPVITVDTKTGNISQKHFLLDSESNVTRSSAFDYLWIVPISSIKNGVMQDHYWLRDVSQAQNDLFKTASDDWVLLNVNVTGYFQVNYDEDNWRMIQHQLQTNLSVIPVINRAQVIYDSFNLATAHMVPVTLALDNTLFLNGEKEYMPWQAALSSLSYFSLMFDRSEVYGPMKKYLRKQVEPLFQHFETLTKNWTERPENLMDQYSEINAISTACSNGLPQCENLAKTLFDQWMSDPENNPIHPNLRSTIYCNAIAQGGQDQWDFAWGQLQQAQLVNEADKLRSALACSNEVWLLNRYLGYTLNPDLIRKQDATSTINSIASNVIGQPLAWDFVQSNWKKLFQDYGGGSFSFSNLIQGVTRRFSSEFELQQLEQFKKNNMDVGFGSGTRALEQALEKTKANIKWVKENKEVVLNWFIEHSS 4fl1 A 1.79 BS01 ANP A 1 G378 S379 G380 V385 A400 K402 M448 E449 M450 A451 L501 G16 S17 G18 V23 A38 K40 M81 E82 M83 A84 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K166 2.7.10.2 0004672,0004713,0005524,0006468 Kd=520uM remove_due_to_license_issue P43405 23154170 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 4fl2 A 2.19 BS02 ANP A 1 S379 G380 N381 V385 A400 K402 A451 P455 R498 L501 K533 S299 G300 N301 V305 A320 K322 A371 P375 R418 L421 K453 D494 A496 R498 N499 D512 K533 D414 A416 R418 N419 D432 K453 2.7.10.2 0001525,0001775,0001784,0001819,0001820,0001945,0002092,0002223,0002250,0002281,0002283,0002366,0002554,0002684,0002752,0002862,0004672,0004674,0004713,0004715,0005102,0005178,0005515,0005524,0005634,0005737,0005829,0005886,0006338,0006468,0006606,0007159,0007166,0007167,0007169,0007229,0009887,0010543,0010803,0016170,0016301,0018108,0019370,0019722,0019815,0019901,0019902,0030154,0030168,0030183,0030593,0031334,0031623,0032009,0032481,0032725,0032733,0032735,0032752,0032753,0032755,0032757,0032760,0032765,0032928,0032930,0032991,0033630,0035325,0035401,0035556,0038063,0038095,0038096,0038156,0042101,0042169,0042492,0042742,0043274,0043303,0043306,0043313,0043366,0043410,0045087,0045579,0045588,0045780,0046638,0046641,0048514,0050731,0050764,0050776,0050850,0050853,0051090,0051649,0070372,0071226,0071396,0071404,0071639,0090237,0090330,0097110,0097190,0097242,0120162,0140801,1904263,1904646,1990858 Kd=220uM remove_due_to_license_issue P43405 23154170 702 SANHLPFFFGNITREEAEDYLVQGGMSDGLYLLRQSRNYLGGFALSVAHGRKAHHYTIERELNGTYAIAGGRTHASPADLCHYHSQESDGLVCLLKKPFNRPQGVQPKTGPFEDLKENLIREYVKQTWNLQGQALEQAIISQKPQLEKLIATTAHEKMPWFHGKISREESEQIVLIGSKTNGKFLIRARDNNGSYALCLLHEGKVLHYRIDKDKTGKLSIPEGKKFDTLWQLVEHYSYKADGLLRVLTVPCQKIGTQREALPMDTEVYESPYADPEEIRPKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 4fl3 A 1.9 BS01 ANP A 1 S379 G380 N381 V385 A400 K402 A451 P455 R498 L501 S295 G296 N297 V301 A316 K318 A367 P371 R414 L417 D494 A496 R498 N499 D512 D410 A412 R414 N415 D428 2.7.10.2 0001525,0001775,0001784,0001819,0001820,0001945,0002092,0002223,0002250,0002281,0002283,0002366,0002554,0002684,0002752,0002862,0004672,0004674,0004713,0004715,0005102,0005178,0005515,0005524,0005634,0005737,0005829,0005886,0006338,0006468,0006606,0007159,0007166,0007167,0007169,0007229,0009887,0010543,0010803,0016170,0016301,0018108,0019370,0019722,0019815,0019901,0019902,0030154,0030168,0030183,0030593,0031334,0031623,0032009,0032481,0032725,0032733,0032735,0032752,0032753,0032755,0032757,0032760,0032765,0032928,0032930,0032991,0033630,0035325,0035401,0035556,0038063,0038095,0038096,0038156,0042101,0042169,0042492,0042742,0043274,0043303,0043306,0043313,0043366,0043410,0045087,0045579,0045588,0045780,0046638,0046641,0048514,0050731,0050764,0050776,0050850,0050853,0051090,0051649,0070372,0071226,0071396,0071404,0071639,0090237,0090330,0097110,0097190,0097242,0120162,0140801,1904263,1904646,1990858 Kd=150uM remove_due_to_license_issue P43405 23154170 701 SANHLPFFFGNITREEAEDYLVQGGMSDGLYLLRQSRNYLGGFALSVAHGRKAHHYTIERELNGTYAIAGGRTHASPADLCHYHSQESDGLVCLLKKPFNRPQGVQPKTGPFEDLKENLIREYVKQTWNLQGQALEQAIISQKPQLEKLIATTAHEKMPWFHGKISREESEQIVLIGSKTNGKFLIRARDNNGSYALCLLHEGKVLHYRIDKDKTGKLSIPEGKKFDTLWQLVEHYSYKADGLLRVLTVPCQKREALPMDTEVFESPFADPEEIRPKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRAPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 4flh A 2.6 BS01 14K A 1 K802 M804 I831 K833 D841 Y867 E880 V882 T887 M953 I963 D964 K561 M563 I590 K592 D600 Y626 E639 V641 T646 M712 I722 D723 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=1nM P48736 22897589 1205 EESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDPIALPKHQEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 4fli A 1.55 BS03 Y16 A 1 P192 Y195 H212 D229 D240 Y300 C301 H303 H310 E336 E367 P103 Y106 H123 D140 D151 Y211 C212 H214 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=3.59uM remove_due_to_license_issue IC50=3590nM P53582 22913487 503 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4flj A 1.74 BS03 Y08 A 1 Y195 H212 D229 D240 C301 H303 F309 H310 E336 E367 Y106 H123 D140 D151 C212 H214 F220 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=7.45uM remove_due_to_license_issue P53582 22913487 503 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4flk A 1.47 BS03 Y10 A 1 Y195 H212 D229 D240 C301 H303 F309 H310 E336 E367 Y106 H123 D140 D151 C212 H214 F220 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=5.58uM remove_due_to_license_issue IC50=5580nM P53582 22913487 503 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4fll A 1.5 BS03 YZ6 A 1 Y195 H212 D229 D240 C301 H303 F309 H310 T311 E336 E367 Y106 H123 D140 D151 C212 H214 F220 H221 T222 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=5.14uM remove_due_to_license_issue P53582 22913487 503 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4flp A 2.23 BS01 JQ1 A 1 P51 L61 L63 N109 I115 M118 P23 L33 L35 N81 I87 M90 ? Kd=190.1nM remove_due_to_license_issue Q58F21 22901802 201 TNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMP 4fm7 A 1.56 BS01 0UP A 1 Q12 G13 L30 D32 Y71 T72 Q73 G74 F108 I110 G230 Q14 G15 L32 D34 Y73 T74 Q75 G76 F110 I112 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.1uM remove_due_to_license_issue P56817 22984865 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4fm8 A 1.9 BS01 0UQ A 1 Q12 G13 L30 D32 Y71 Q73 G74 F108 I110 W115 G230 Q14 G15 L32 D34 Y73 Q75 G76 F110 I112 W117 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=2.4uM remove_due_to_license_issue P56817 22984865 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4fmu A 2.1 BS04 0UM A 1 K1560 G1561 W1562 Y1579 H1603 Y1604 Y1605 R1625 F1626 M1627 N1628 H1629 F1664 Y1666 Q1676 C1678 F1679 L1689 K104 G105 W106 Y123 H147 Y148 Y149 R169 F170 M171 N172 H173 F208 Y210 Q220 C222 F223 L233 Y1579 Y1666 Y123 Y210 2.1.1.-,2.1.1.359 0005634,0016279,0042054,0046975 Kd=360nM remove_due_to_license_issue IC50=800nM Q9BYW2 23043551 1804 LVGPSCVMDDFRDPQRWKECAKQGKMPCYFDLIEENVYLTMQCECTPLSKDERAQGEIACGEDCLNRLLMIECSSRCPNGDYCSNRRFQRKQHADVEVILTEKKGWGLRAAKDLPSNTFVLEYCGEVLDHKEFKARVKEYARNKNIHYYFMALKNDEIIDATQKGNCSRFMNHSCEPNCETQKWTVNGQLRVGFFTTKLVPSGSELTFDYQFQRYGKEAQKCFCGSANCRGYLGG 4fnn A 2.24 BS01 STE B 1 A129 V132 A129 V132 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 23149273 201 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 4fnn B 2.24 BS01 STE B 1 D2 P4 C6 D2 P4 C6 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 23149273 201 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 4fnn D 2.24 BS01 STE B 1 R31 R138 R31 R138 Y71 T152 Y71 T152 ? 0001818,0005576,0008270,0008745,0009253,0016019,0016045,0042742,0042834,0045087,0050830 remove_due_to_license_issue Q9GK12 23149273 201 EDPPACGSIVPRREWRALASECRERLTRPVRYVVVSHTAGSHCDTPASCAQQAQNVQSYHVRNLGWCDVGYNFLIGEDGLVYEGRGWNIKGAHAGPTWNPISIGISFMGNYMNRVPPPRALRAAQNLLACGVALGALRSNYEVKGHRDVQPTLSPGDRLYEIIQTWSHYRA 4fns A 2.6 BS01 DGJ A 1 W336 D366 D367 W411 R443 K476 D478 N480 C526 G528 W545 D548 W327 D357 D358 W402 R434 K467 D469 N471 C517 G519 W536 D539 3.2.1.22 0004553,0004557,0005975,0016052,0016798,0033531,0034484,0051289 remove_due_to_license_issue Q9ALJ4 23012371 801 KQFHLRAGKASYVMQLFRSGYLAHVYWGKAVRDVRGARAFPRLDRAFSPNPDPSDRTFSLDTLLQEYPAYGNTDFRAPAYQVQLENGSTVTDLRYKTHRIYKGKPRLNGLPATYVEHEQEAETLEIVLGDALIGLEVTLQYTAYEKWNVITRSARFENKGGERLKLLRALSMSVDFPTADYDWIHLPGAWGRERWIERRPLVTGVQAAESRRGASSHQQNPFIALVAKNADEHQGEVYGFSFVYSGNFLAQIEVDQFGTARVSMGINPFDFTWLLQPGESFQTPEVVMVYSDQGLNGMSQTYHELYRTRLARGAFRDRERPILINNWEATYFDFNEEKIVNIARTEAELGIELVVLDDGWFGERDDDRRSLGDWIVNRRKLPNGLDGLAKQVNELGLQFGLWVEPEMVSPNSELYRKHPDWCLHVPNRPRSEGRNQLVLDYSREDVCDYIIETISNVLASAPITYVKWDMNRHMTEIGSSALPPERQRETAHRYMLGLYRVMDEITSRLPHILFESCSGGGGRFDPGMLYYMPQTWTSDNTDAVSRLKIQYGTSLVYPISAMGAHVSAVPNHQVGRVASLKTRGHVAMSGNFGYELDITKLTETEKQMMKQQVAFYKDVRRLVQFGTFYRLLSPFEGNEAAWMFVSADRSEALVAYFRVLAEANAPLSYLRLKGLDSNQDYEIEGLGVYGGDELVYAGVALPYRSSDFISMMWRLKAV 4fns D 2.6 BS01 DGJ D 1 W336 D366 D367 W411 R443 K476 D478 N480 C526 G528 D548 W327 D357 D358 W402 R434 K467 D469 N471 C517 G519 D539 3.2.1.22 0004553,0004557,0005975,0016052,0016798,0033531,0034484,0051289 remove_due_to_license_issue Q9ALJ4 23012371 801 KQFHLRAGKASYVMQLFRSGYLAHVYWGKAVRDVRGARAFPRLDRAFSPNPDPSDRTFSLDTLLQEYPAYGNTDFRAPAYQVQLENGSTVTDLRYKTHRIYKGKPRLNGLPATYVEHEQEAETLEIVLGDALIGLEVTLQYTAYEKWNVITRSARFENKGGERLKLLRALSMSVDFPTADYDWIHLPGAWGRERWIERRPLVTGVQAAESRRGASSHQQNPFIALVAKNADEHQGEVYGFSFVYSGNFLAQIEVDQFGTARVSMGINPFDFTWLLQPGESFQTPEVVMVYSDQGLNGMSQTYHELYRTRLARGAFRDRERPILINNWEATYFDFNEEKIVNIARTEAELGIELVVLDDGWFGERDDDRRSLGDWIVNRRKLPNGLDGLAKQVNELGLQFGLWVEPEMVSPNSELYRKHPDWCLHVPNRPRSEGRNQLVLDYSREDVCDYIIETISNVLASAPITYVKWDMNRHMTEIGSSALPPERQRETAHRYMLGLYRVMDEITSRLPHILFESCSGGGGRFDPGMLYYMPQTWTSDNTDAVSRLKIQYGTSLVYPISAMGAHVSAVPNHQVGRVASLKTRGHVAMSGNFGYELDITKLTETEKQMMKQQVAFYKDVRRLVQFGTFYRLLSPFEGNEAAWMFVSADRSEALVAYFRVLAEANAPLSYLRLKGLDSNQDYEIEGLGVYGGDELVYAGVALPYRSSDFISMMWRLKAV 4fny A 2.45 BS01 I3K A 1 A1148 E1167 I1171 L1196 M1199 L1256 G1269 D1270 F1271 A37 E56 I60 L85 M88 L141 G154 D155 F156 D1249 A1251 R1253 N1254 D1270 D134 A136 R138 N139 D155 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.016uM remove_due_to_license_issue Q9UM73 22932897 1501 SSISDLKEVPRKNITLIRGLGHGEVYEGQVSGPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYGPL 4fnz A 2.6 BS01 NZF A 1 L1122 A1148 K1150 I1171 V1180 M1199 A1200 G1202 H1247 L1256 I1268 G1269 D1270 F1271 L30 A48 K50 I71 V80 M99 A100 G102 H147 L156 I168 G169 D170 F171 D1249 A1251 R1253 N1254 D1270 D149 A151 R153 N154 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=16nM Q9UM73 22932897 1501 NPNYSFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVSGSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYG 4fob A 1.9 BS01 0US A 1 L1122 V1130 A1148 L1196 E1197 M1199 G1201 G1202 L1256 G1269 L30 V38 A50 L98 E99 M101 G103 G104 L155 G168 D1249 A1251 R1253 N1254 D1270 R1279 D148 A150 R152 N153 D169 R178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.005uM remove_due_to_license_issue IC50=5nM Q9UM73 22734674 1501 NPNYSFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRAGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYG 4foc A 1.7 BS01 0UU A 1 L1122 V1130 A1148 L1196 E1197 M1199 G1202 L1256 L30 V38 A50 L98 E99 M101 G104 L158 D1249 A1251 R1253 N1254 D1270 R1279 D151 A153 R155 N156 D172 R181 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.003uM remove_due_to_license_issue IC50=3nM Q9UM73 22734674 1501 NPNYSFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYG 4fod A 2.0 BS01 0UV A 1 L1122 H1124 A1148 L1196 E1197 M1199 A1200 G1201 G1202 E1210 L1256 L38 H40 A58 L106 E107 M109 A110 G111 G112 E120 L166 D1249 A1251 R1253 N1254 D1270 R1279 D159 A161 R163 N164 D180 R189 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.0012uM remove_due_to_license_issue Q9UM73 22734674 1501 TSTIMTDYNPNYSFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRACAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYGPLV 4fp1 A 1.68 BS02 BFM A 1 V22 K166 H297 L298 V20 K164 H295 L296 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=0.027mM remove_due_to_license_issue P11444 24472022 402 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 4fp1 B 1.68 BS02 BFM B 1 F52 K166 E247 H297 F50 K164 E245 H295 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=0.027mM remove_due_to_license_issue P11444 24472022 402 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 4fpf A 2.23 BS01 JKK A 1 R245 D270 I326 M346 G351 N352 Y489 R557 R619 Y653 R207 D232 I288 M308 G313 N314 Y451 R519 R581 Y615 D270 E541 Y653 D232 E503 Y615 3.2.1.18 0004308,0005975 ic50=38.9uM remove_due_to_license_issue Q54727 23070966 701 ISPIFQGGSYQLNNKSIDISSLLLDKLSGESQTVVMKFKADKPNSLQALFGLSNSKAGFKNNYFSIFMRDSGEIGVEIRDAQKGINYLFSRPASLWGKHKGQAVENTLVFVSDSKDKTYTMYVNGIEVFSETVDTFLPISNINGIDKATLGAVNREGKEHYLAKGSIDEISLFNKAISDQEVSTIPLSNPFQLIFQSGDSTQANYFRIPTLYTLSSGRVLSSIDARYGGTHDSKSKINIATSYSDDNGKTWSEPIFAMKFNDYEEQLVYWPRDNKLKNSQISGSASFIDSSIVEDKKSGKTILLADVMPAGIGNNNANKADSGFKEINGHYYLKLKKNGDNDFRYTVRENGVVYNETTNKPTNYTINDKYEVLEGGKSLTVEQYSVDFDSGSLRERHNGKQVPMNVFYKDSLFKVTPTNYIAMTTSQNRGESWEQFKLLPPFLGEKHNGTYLCPGQGLALKSSNRLIFATYTSGELTYLISDDSGQTWKKSSASIPFKNATAEAQMVELRDGVIRTFFRTTTGKIAYMTSRDSGETWSKVSYIDGIQQTSYGTQVSAIKYSQLIDGKEAVILSTPNSRSGRKGGQLVVGLVNKEDDSIDWKYHYDIDLPSYGYAYSAITELPNHHIGVLFEKYDSWSRNELHLSNVVQYIDLEINDLT 4fpk A 2.4 BS01 IJ1 A 1 R245 D270 I326 N352 Y489 R557 R619 Y653 W674 R207 D232 I288 N314 Y451 R519 R581 Y615 W636 D270 E541 Y653 D232 E503 Y615 3.2.1.18 0004308,0005975 ic50=57.4uM remove_due_to_license_issue Q54727 23070966 701 ISPIFQGGSYQLNNKSIDISSLLLDKLSGESQTVVMKFKADKPNSLQALFGLSNSKAGFKNNYFSIFMRDSGEIGVEIRDAQKGINYLFSRPASLWGKHKGQAVENTLVFVSDSKDKTYTMYVNGIEVFSETVDTFLPISNINGIDKATLGAVNREGKEHYLAKGSIDEISLFNKAISDQEVSTIPLSNPFQLIFQSGDSTQANYFRIPTLYTLSSGRVLSSIDARYGGTHDSKSKINIATSYSDDNGKTWSEPIFAMKFNDYEEQLVYWPRDNKLKNSQISGSASFIDSSIVEDKKSGKTILLADVMPAGIGNNNANKADSGFKEINGHYYLKLKKNGDNDFRYTVRENGVVYNETTNKPTNYTINDKYEVLEGGKSLTVEQYSVDFDSGSLRERHNGKQVPMNVFYKDSLFKVTPTNYIAMTTSQNRGESWEQFKLLPPFLGEKHNGTYLCPGQGLALKSSNRLIFATYTSGELTYLISDDSGQTWKKSSASIPFKNATAEAQMVELRDGVIRTFFRTTTGKIAYMTSRDSGETWSKVSYIDGIQQTSYGTQVSAIKYSQLIDGKEAVILSTPNSRSGRKGGQLVVGLVNKEDDSIDWKYHYDIDLPSYGYAYSAITELPNHHIGVLFEKYDSWSRNELHLSNVVQYIDLEINDLT 4fqo A 1.65 BS03 AZ3 A 1 H42 F43 C84 H85 F87 F88 H43 F44 C85 H86 F88 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 remove_due_to_license_issue P02638 23264854 103 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFF 4fri A 2.3 BS01 DWA A 1 G11 G13 L30 D32 S35 Y71 W76 F108 I118 D228 G230 G13 G15 L32 D34 S37 Y73 W78 F110 I120 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=2.85uM remove_due_to_license_issue P56817 22928914 404 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4frj A 1.95 BS01 DWB A 1 G11 G13 L30 D32 Y71 F108 I110 R128 D228 G230 G13 G15 L32 D34 Y73 F110 I112 R130 D222 G224 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.28uM remove_due_to_license_issue P56817 22928914 403 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4frk A 2.1 BS01 DWD A 1 G11 Q12 G13 L30 D32 Y71 F108 D228 G230 G13 Q14 G15 L32 D34 Y73 F110 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.008uM remove_due_to_license_issue IC50=36nM P56817 22928914 405 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4frs A 1.7 BS01 0V6 A 1 S71 Q73 G74 L91 D93 Y132 Q134 G135 F169 W176 D289 S290 G291 T292 S14 Q16 G17 L34 D36 Y75 Q77 G78 F112 W119 D232 S233 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 23412139 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4fs3 A 1.8 BS02 0WE A 1 F96 A97 M99 L102 Y147 N156 Y157 S197 V201 F96 A97 M99 L102 Y147 N156 Y157 S197 V201 Y147 Y157 M160 K164 K199 Y147 Y157 M160 K164 K199 1.3.1.39 0000166,0004318,0006633,0016491,0030497,0042802,0050661,0141148 Ki=12.8nM remove_due_to_license_issue Q6GI75 22948878 302 MLNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIKERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4fs4 A 1.74 BS01 H24 A 1 Q73 G74 D93 Y132 F169 I171 W176 D289 S290 G291 Q16 G17 D36 Y75 F112 I114 W119 D232 S233 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=91000nM P56817 24900403 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4fse A 2.65 BS01 0VA A 1 D80 Y119 Q121 G122 F156 W163 Y246 I274 D276 G278 T279 R283 T377 D34 Y73 Q75 G76 F110 W117 Y200 I228 D230 G232 T233 R237 T331 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 23030502 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4fsl A 2.5 BS01 0VB A 1 D80 G82 Y119 Q121 G122 K155 F156 I158 W163 I274 D276 T279 R283 T377 V380 D34 G36 Y73 Q75 G76 K109 F110 I112 W117 I228 D230 T233 R237 T331 V334 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 23030502 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4fth A 3.004 BS01 dna C 0 I60 D61 N64 R67 K68 I50 D51 N54 R57 K58 ? 0043565 remove_due_to_license_issue O66551 25158097 1 ~ 21 LKEKSWRDLSYLLKIKELKEAKKEFEKIFIEEKLREYDYDLKRTAEEIGIDLSNLYRKIKSLNIRVKS 4fth A 3.004 BS02 dna D 0 K29 Y66 R67 K19 Y56 R57 ? 0043565 remove_due_to_license_issue O66551 25158097 1 ~ 21 LKEKSWRDLSYLLKIKELKEAKKEFEKIFIEEKLREYDYDLKRTAEEIGIDLSNLYRKIKSLNIRVKS 4fth B 3.004 BS01 dna C 0 Y66 R67 Y50 R51 ? 0043565 remove_due_to_license_issue O66551 25158097 1 ~ 21 RDLSYLLKIKELKEAKKEFEKIFIEEKLREYDYDLKRTAEEIGIDLSNLYRKIKSLNIRVK 4fth B 3.004 BS02 dna D 0 D61 S63 N64 K68 D45 S47 N48 K52 ? 0043565 remove_due_to_license_issue O66551 25158097 1 ~ 21 RDLSYLLKIKELKEAKKEFEKIFIEEKLREYDYDLKRTAEEIGIDLSNLYRKIKSLNIRVK 4fut A 2.0 BS01 ATP A 1 T163 S164 G165 T166 T167 S277 A278 P279 E298 M302 T303 D382 R397 T163 S164 G165 T166 T167 S277 A278 P279 E298 M302 T303 D382 R397 T163 N183 H207 T303 E304 I403 N408 A488 T163 N183 H207 T303 E304 I403 N408 A488 6.2.1.- 0005524,0006631,0016874,0031956 Kd=0.31uM remove_due_to_license_issue Q6ND88 22773649 608 MNANLFARLFDKLDDPHKLAIETAAGDKISYAELVARAGRVANVLVARGLQVGDRVAAQTEKSVEALVLYLATVRAGGVYLPLNTAYTLHELDYFITDAEPKIVVCDPSKRDGIAAIAAKVGATVETLGPDGRGSLTDAAAGASEAFATIDRGADDLAAILYTSGTTGRSKGAMLSHDNLASNSLTLVDYWRFTPDDVLIHALPIYHTHGLFVASNVTLFARGSMIFLPKFDPDKILDLMARATVLMGVPTFYTRLLQSPRLTKETTGHMRLFISGSAPLLADTHREWSAKTGHAVLERYGMTETNMNTSNPYDGDRVPGAVGPALPGVSARVTDPETGKELPRGDIGMIEVKGPNVFKGYWRMPEKTKSEFRDDGFFITGDLGKIDERGYVHILGRGKDLVITGGFNVYPKEIESEIDAMPGVVESAVIGVPHADFGEGVTAVVVRDKGATIDEAQVLHGLDGQLAKFKMPKKVIFVDDLPRNTMGAVQKNVLRETYKDIYK 4fvq A 1.75 BS01 ATP A 1 G554 T555 T557 I559 L579 K581 Q626 F628 V629 S633 K677 N678 L680 G19 T20 T22 I24 L44 K46 Q91 F93 V94 S98 K142 N143 L145 N673 K677 N678 D699 N138 K142 N143 D164 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue O60674 22820988 901 VFHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSLF 4fvr A 2.0 BS01 ATP A 1 G554 T555 T557 I559 L579 K581 Q626 F628 V629 S633 N673 K677 N678 L680 G19 T20 T22 I24 L44 K46 Q91 F93 V94 S98 N138 K142 N143 L145 N673 K677 N678 D699 N138 K142 N143 D164 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue O60674 22820988 901 VFHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCFCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAWAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSLF 4fxf A 2.55 BS03 FBP A 1 T432 K433 S434 S437 W482 G514 R516 P517 G518 S519 G520 F521 T522 T402 K403 S404 S407 W452 G484 R486 P487 G488 S489 G490 F491 T492 R73 R120 K270 T328 R43 R90 K240 T298 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 23530218 604 CRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQNLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 4fxj A 2.9 BS03 PHE A 1 R43 N44 N70 R106 H464 G468 I469 F470 R16 N17 N43 R79 H431 G435 I436 F437 R73 R120 K270 T328 R46 R93 K240 T298 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 23530218 603 EHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQNLIAREAEAAIYHLQLFEELRRLAPDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 4fxp A 1.954 BS01 ADX A 1 D138 R141 F150 R155 N158 L180 I181 S182 F232 D54 R57 F66 R71 N74 L96 I97 S98 F148 2.7.1.25 0000103,0004020,0005524 remove_due_to_license_issue Q43295 22810229 301 ECSVEKVDRQRLLDQKGCVIWVTGLSGSGKSTLACALNQMLYQKGKLCYILDGDNVRHGLNRDLSFKAEDRAENIRRVGEVAKLFADAGIICIASLISPYRTDRDACRSLLPEGDFVEVFMDVPLSVCEARDPKGLYKLARAGKIKGFTGIDDPYEPPLNCEISLGREGGTSPIEMAEKVVGYLDNKGYLQA 4fxq A 1.9599 BS01 G9L A 1 G281 Y284 R341 R342 S387 T388 S389 Y398 Q429 E431 G263 Y266 R323 R324 S369 T370 S371 Y380 Q411 E413 S387 E431 S369 E413 2.4.2.- 0000166,0003824,0005576,0008237,0016757,0016779,0035821,0046872,0090729 Kd=1.7uM remove_due_to_license_issue Q4MV79 22992735 501 ENSKKTQELVEKLPHEVLELYKNVGGEIYITDKRLTQHEELSDSSHKDMFIVSSEGKSFPLREHFVFAKGGKEPSLIIHAEDYASHLSSVEVYYELGKAIIRDTFPLNQKELGNPKFINAINEVNQQKEGKGVNAKADEDGRDLLFGKELKKNLEHGQLVDLDLISGNLSEFQHVFAKSFALYYEPHYKEALKSYAPALFNYMLELDQMRFKEISDDVKEKNKNVLDFKWYTRKAESWGVQTFKNWKENLTISEKDIITGYTGSKYDPINEYLRKYDGEIIPNIGGDLDKKSKKALEKIENQIKNLDAALQKSKITENLIVYRRVSELQFGKKYEDYNLRQNGIINEEKVMELESNFKGQTFIQHNYMSTSLVQDPHQSYSNDRYPILLEITIPEGVHGAYIADMSEYPGQYEMLINRGYTFKYDKFSIVKPGKEYLKVNLSIYL 4fxy P 2.8 BS01 0W2 P 1 Y49 I72 E73 Y76 R80 D110 M113 S114 S146 Y35 I58 E59 Y62 R66 D96 M99 S100 S132 H474 E475 H478 H460 E461 H464 3.4.24.16 0004222,0005737,0005739,0005758,0005829,0005886,0006111,0006508,0006518,0008233,0008237,0030163,0042277,0043171,0046872,0070012,1902809 remove_due_to_license_issue P42676 25378390 701 SSYTAAGRNVLRWDLSPEQIKTRTEQLIAQTKQVYDTVGTIALKEVTYENCLQVLADIEVTYIVERTMLDFPQHVSSDREVRAASTEADKKLSRFDIEMSMREDVFQRIVHLQETCDLEKIKPEARRYLEKSIKMGKRNGLHLSEAIRNEIKSMKKRMSELCIDFNKNLNEDDTSLVFSKAELGALPDDFIDSLEKTDEDKYKVTLKYPHYFPVMKKCCVPETRRKMEMAFHTRCKQENTAILQQLLPLRAQVAKLLGYNTHADFVLELNTAKSTSRVAAFLDDLSQKLKPLGEAEREFILSLKKKECEERGFEYDGKINAWDLHYYMTQTEELKYSVDQESLKEYFPIEVVTEGLLSIYQELLGLSFEQVPDAHVWNKSVSLYTVKDKATGEVLGQFYLDLYPREGKYNHAACFGLQPGCLLPDGSRMMSVAALVVNFSQPVAGRPSLLRHDEVRTYFHEFGHVMHQICAQTDFARFSGTNVETDFVEVPSQMLENWVWDVDSLRKLSKHYKDGHPITDELLEKLVASRLVNTGLLTLRQIVLSKVDQSLHTNATLDAASEYAKYCTEILGVAATPGTNMPATFGHLAGGYDGQYYGYLWSEVFSMDMFHSCFKKEGIMNPEVGMKYRNLILKPGGSLDGMDMLQNFLQREPNQKAFLMSRGL 4fxz A 2.601 BS01 LEU A 1 A22 G24 G26 A253 T254 S256 F259 I359 A18 G20 G22 A246 T247 S249 F252 I352 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 22836580 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFATLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRN 4fyh A 2.44 BS01 TR5 A 1 C15 G16 S17 I18 R19 I65 N69 S87 G89 E93 C7 G8 S9 I10 R11 I42 N46 S64 G66 E70 3.2.2.- 0009159,0070694 remove_due_to_license_issue O35820 23385460 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAY 4fyh A 2.44 BS02 TR5 B 1 S117 A118 M119 S94 A95 M96 3.2.2.- 0009159,0070694 remove_due_to_license_issue O35820 23385460 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAY 4fyh B 2.44 BS01 TR5 A 1 S117 A118 M119 S92 A93 M94 3.2.2.- 0009159,0070694 remove_due_to_license_issue O35820 23385460 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAY 4fyh B 2.44 BS02 TR5 B 1 C15 G16 S17 I18 R19 N69 S87 G89 E93 C7 G8 S9 I10 R11 N44 S62 G64 E68 3.2.2.- 0009159,0070694 remove_due_to_license_issue O35820 23385460 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAY 4fyo A 1.4 BS01 0VF A 1 L377 G378 S379 V385 A400 M448 A451 E452 G454 P455 K458 R498 L501 L15 G16 S17 V23 A38 M80 A83 E84 G86 P87 K90 R130 L133 D494 A496 R498 N499 D512 K533 D126 A128 R130 N131 D144 K161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=47nM remove_due_to_license_issue IC50=47nM P43405 23151054 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 4fz6 A 1.85 BS01 0VG A 1 V385 A400 M450 A451 E452 G454 L501 V21 A36 M81 A82 E83 G85 L132 D494 A496 R498 N499 D512 K533 D125 A127 R129 N130 D143 K160 2.7.10.2 0004672,0004713,0005524,0006468 ic50=127nM remove_due_to_license_issue IC50=127nM P43405 23151054 701 VYLDRKLLTLEDKELGSFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 4fzj A 1.63 BS01 0W1 A 1 R188 T218 I283 R186 T216 I281 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=0.74mM remove_due_to_license_issue P9WIL5 23872845 405 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 4g0c A 2.0 BS02 AZM A 1 Q92 H94 F131 L198 T199 T200 Q89 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=12nM, Kd=17nM, IC50=10nM P00918 22928733 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4g0k A 2.557 BS01 0VS A 1 W65 W96 R130 T132 V133 E148 S149 F199 W64 W95 R129 T131 V132 E147 S148 F198 1.8.5.7 0004364,0005737,0016491,0016672,0042803 remove_due_to_license_issue P42620 22955277 411 GQLIDGVWHDTWYDTKSTGGKFQRSASAFRNWLTADGAPGPTGTGGFIAEKDRYHLYVSLACPWAHRTLIMRKLKGLEPFISVSVVNPLMLENGWTFDDSFPGATGDTLYQNEFLYQLYLHADPHYSGRVTVPVLWDKKNHTIVSNESAEIIRMFNTAFDALGAKAGDYYPPALQTKIDELNGWIYDTVNNGVYKAGFATSQEAYDEAVAKVFESLARLEQILGQHRYLTGNQLTEADIRLWTTLVRFDPVYVTHFKCDKHRISDYLNLYGFLRDIYQMPGIAETVNFDHIRNHYFRSHKTINPTGIISIGPWQDLDEPHGRDVRFG 4g0l A 2.62 BS01 GSH A 1 C63 W65 W96 R130 T132 V133 E148 S149 C62 W64 W95 R129 T131 V132 E147 S148 1.8.5.7 0004364,0005737,0016491,0016672,0042803 remove_due_to_license_issue P42620 22955277 401 GQLIDGVWHDTWYDTKSTGGKFQRSASAFRNWLTADGAPGPTGTGGFIAEKDRYHLYVSLACPWAHRTLIMRKLKGLEPFISVSVVNPLMLENGWTFDDSFPGATGDTLYQNEFLYQLYLHADPHYSGRVTVPVLWDKKNHTIVSNESAEIIRMFNTAFDALGAKAGDYYPPALQTKIDELNGWIYDTVNNGVYKAGFATSQEAYDEAVAKVFESLARLEQILGQHRYLTGNQLTEADIRLWTTLVRFDPVYVTHFKCDKHRISDYLNLYGFLRDIYQMPGIAETVNFDHIRNHYFRSHKTINPTGIISIGPWQDLDEPHGRDVRFG 4g0p A 1.8 BS01 U5P A 1 Y691 K695 Q707 C708 K728 K732 Y98 K102 Q114 C115 K135 K139 ? 0003676 Kd=0.98mM remove_due_to_license_issue O04379 22850669 801 SNKKMINGGTVNNWICINFSRQVQDNLARTFCQELAQMCYVSGMAFNPEPVLPPVSARPEQVEKVLKTRYHDATSKLSQGKEIDLLIVILPDNNGSLYGDLKRICETELGIVSQCCLTKHVFKMSKQYMANVALKINVKVGGRNTVL 4g0q A 1.8 BS01 C5P A 1 Y691 K695 Q707 C708 K728 K732 Y98 K102 Q114 C115 K135 K139 ? 0003676 Kd=3mM remove_due_to_license_issue O04379 22850669 801 SNKKMINGGTVNNWICINFSRQVQDNLARTFCQELAQMCYVSGMAFNPEPVLPPVSARPEQVEKVLKTRYHDATSKLSQGKEIDLLIVILPDNNGSLYGDLKRICETELGIVSQCCLTKHVFKMSKQYMANVALKINVKVGGRNTVL 4g0y A 1.65 BS01 AMP A 1 N687 Y691 K695 Q707 C708 L710 K728 K732 N94 Y98 K102 Q114 C115 L117 K135 K139 ? 0003676 Kd=4.99mM remove_due_to_license_issue O04379 22850669 801 SNKKMINGGTVNNWICINFSRQVQDNLARTFCQELAQMCYVSGMAFNPEPVLPPVSARPEQVEKVLKTRYHDATSKLSQGKEIDLLIVILPDNNGSLYGDLKRICETELGIVSQCCLTKHVFKMSKQYMANVALKINVKVGGRNTVL 4g0z A 1.75 BS01 5GP A 1 N687 Y691 K695 Q707 C708 L710 K728 K732 N94 Y98 K102 Q114 C115 L117 K135 K139 ? 0003676 Kd=6.13mM remove_due_to_license_issue O04379 22850669 801 SNKKMINGGTVNNWICINFSRQVQDNLARTFCQELAQMCYVSGMAFNPEPVLPPVSARPEQVEKVLKTRYHDATSKLSQGKEIDLLIVILPDNNGSLYGDLKRICETELGIVSQCCLTKHVFKMSKQYMANVALKINVKVGGRNTVL 4g11 A 3.4 BS01 0W7 A 1 M804 P810 W812 Y867 V882 M953 I963 D964 M566 P572 W574 Y629 V644 M714 I724 D725 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=>10000nM P48736 22981333 1201 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 4g16 A 2.3 BS01 0VM A 1 I49 A70 L116 L118 L119 G120 D125 L169 P331 P333 I17 A38 L84 L86 L87 G88 D93 L137 P299 P301 D162 K164 T212 D130 K132 T180 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.14uM remove_due_to_license_issue Q9Y6M4 22877629 401 GSGVLMVGPNFRVGKKIGCGNFGELRLGKNLYTNEYVAIKLEPMKSRAPQLHLEYRFYKQLGSGDGIPQVYYFGPCGKYNAMVLELLGPSLEDLFDLCDRTFSLKTVLMIAIQLISRMEYVHSKNLIYRDVKPENFLIGRPGNKTQQVIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGHMFMYFLRGSLPWQGLKADTLKERYQKIGDTKRATPIEVLCENFPEMATYLRYVRRLDFFEKPDYDYLRKLFTDLFDRKGYMFDYEYDWIGKQLPTPV 4g17 A 2.1 BS01 0VN A 1 G50 A70 L116 L118 L119 G120 P121 L169 P333 G18 A38 L84 L86 L87 G88 P89 L137 P301 D162 K164 T212 D130 K132 T180 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.029uM remove_due_to_license_issue Q9Y6M4 22877629 401 GSGVLMVGPNFRVGKKIGCGNFGELRLGKNLYTNEYVAIKLEPMKSRAPQLHLEYRFYKQLGSGDGIPQVYYFGPCGKYNAMVLELLGPSLEDLFDLCDRTFSLKTVLMIAIQLISRMEYVHSKNLIYRDVKPENFLIGRPGNKTQQVIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGHMFMYFLRGSLPWQGLKADTLKERYQKIGDTKRATPIEVLCENFPEMATYLRYVRRLDFFEKPDYDYLRKLFTDLFDRKGYMFDYEYDWIGKQLPTPV 4g19 A 2.0 BS01 GSH A 1 S22 N24 Y46 H70 T72 L73 D87 S88 Y148 R153 S21 N23 Y45 H69 T71 L72 D86 S87 Y147 R152 ? 0016740 ic50=261.5uM remove_due_to_license_issue I6ZUH3 23007392 302 AQPIVFYDIPSNERIKHSPWSPNTWKIRYALNYKGLKYKTEWVEYPDIAGVVQKLGGKPTEKTPDGRDHYTLPVIYDPNTKKVVEDSAAIAKYLDETYPDTPKLFPAGTDAFQAAFLDFAWPVLGFPVFMLVILDTANSLLPRSHDYFRSTREQKFGKKLEELATEEEWAKVEAGLAKLKGYLDANGKGNDLLLMGAQGGITYSDIQIASFFVWAKIIWGEGSEKWKRLISLHDGKWAQFYAQFTKFEQVD 4g1f A 2.9 BS01 0WG A 1 E206 Y547 S630 Y631 Y662 Y666 H740 E164 Y505 S588 Y589 Y620 Y624 H698 Y547 S630 Y631 D708 H740 Y505 S588 Y589 D666 H698 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=17nM P27487 23025999 800 KTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 4g2f A 1.699 BS01 C07 A 1 A651 K653 E670 T699 E700 M702 L753 S763 D764 A43 K45 E62 T91 E92 M94 L145 S155 D156 D746 A748 R750 N751 D764 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P29320 24900387 1001 VHEFAKELDATNISIDKVVGAGEFGEVCSGRLKLPSKKEISVAIKTLKVGYTEKQRRDFLGEASIMGQFDHPNIIRLEGVVTKSKPVMIVTEYMENGSLDSFLRKHDAQFTVIQLVGMLRGIASGMKYLSDMGYVHRDLAARNILINSNLVCKVSDFGLSRVLPIRWTSPEAIAYRKFTSASDVWSYGIVLWEVMSYGERPYWEMSNQDVIKAVDEGYRLPPPMDCPAALYQLMLDCWQKDRNNRPKFEQIVSILDKLIRNPGSLKIITPSNLLL 4g2j A 2.4 BS02 0WF A 1 M365 L420 Y424 F441 Q453 F456 V460 M188 L243 Y247 F264 Q276 F279 V283 3.1.4.35 0004114,0007165,0008081 ic50=11nM remove_due_to_license_issue IC50=45nM O76083 23025719 903 GSHMTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 4g2l A 3.0 BS02 0WL A 1 L420 Y424 F441 Q453 F456 L243 Y247 F264 Q276 F279 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue IC50=32nM O76083 23025719 903 GSHMTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQK 4g2r A 2.28 BS01 H1L A 1 G98 A99 F115 G137 G138 Y141 G86 A87 F103 G125 G126 Y129 A99 G137 G138 Y326 G366 A367 A87 G125 G126 Y300 G340 A341 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 501 LDPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r A 2.28 BS02 H1L A 2 A140 V157 H184 H185 S188 V190 A128 V145 H159 H160 S163 V165 A99 G137 G138 Y326 G366 A367 A87 G125 G126 Y300 G340 A341 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 502 LDPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r A 2.28 BS03 H1L B 1 L295 Y326 V337 G366 L270 Y300 V311 G340 A99 G137 G138 Y326 G366 A367 A87 G125 G126 Y300 G340 A341 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 501 LDPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r A 2.28 BS04 H1L B 2 E333 W334 V338 E307 W308 V312 A99 G137 G138 Y326 G366 A367 A87 G125 G126 Y300 G340 A341 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 502 LDPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r B 2.28 BS01 H1L A 1 L295 Y326 G366 L270 Y301 G341 A99 G137 G138 Y326 G366 A367 A86 G124 G125 Y301 G341 A342 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 501 DPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPMASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAEKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r B 2.28 BS02 H1L A 2 E333 W334 G335 V338 E308 W309 G310 V313 A99 G137 G138 Y326 G366 A367 A86 G124 G125 Y301 G341 A342 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 502 DPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPMASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAEKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r B 2.28 BS03 H1L B 1 A99 F115 G137 G138 Y141 A86 F102 G124 G125 Y128 A99 G137 G138 Y326 G366 A367 A86 G124 G125 Y301 G341 A342 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 501 DPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPMASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAEKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2r B 2.28 BS04 H1L B 2 A140 V159 H184 H185 S188 V190 A127 V146 H159 H160 S163 V165 A99 G137 G138 Y326 G366 A367 A86 G124 G125 Y301 G341 A342 2.1.3.-,2.1.3.15 0003989,0004658,0005515,0006633,0009274,0009317,0016740,0016874,0019367 Kd=35.8uM remove_due_to_license_issue P9WQH5 25092705 502 DPRDPLLRLSNFFDDGSVELLHERDRSGVLAAAGTVNGVRTIAFCTDGTVMGGAMGVEGCTHIVNAYDTAIEDQSPIVGIWHSGGARLAEGVRALHAVGQVFEAMIRASGYIPQISVVVGFAAGGAAYGPALTDVVVMAPESRVFVTGPMASLGGPETHHKKSGVCHIVADDELDAYDRGRRLVGLFCQQGHFDRSKAEAGDTDIHALLPESSRRAYDVRPIVTAILDADTPFDEFQANWAPSMVVGLGRLSGRTVGVLANNPLRLGGCLNSESAEKAARFVRLCDAFGIPLVVVVDVPGYLPGVDQEWGGVVRRGAKLLHAFGECTVPRVTLVTRKTYGGAYIAMNSRSLNATKVFAWPDAEVAVMGAKAAVGILHKKKLAAAPEHEREALHDQLAAEHERIAGGVDSALDIGVVDEKIDPAHTRSKLTEALAQAPARRG 4g2w A 2.28 BS01 NI0 A 1 Y612 L765 V782 F786 Q817 F820 Y76 L214 V231 F235 Q245 F248 3.1.4.35 0004114,0007165,0008081 ic50=1.6nM remove_due_to_license_issue IC50=1.6nM, Kd=1.3nM O76074 23137303 901 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 4g2y A 2.4 BS02 NI5 A 1 F786 Q817 F820 F246 Q256 F259 3.1.4.35 0004114,0007165,0008081 ic50>1000nM remove_due_to_license_issue O76074 23137303 904 MEETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 4g31 A 2.28 BS01 0WH A 1 A619 L642 A643 V651 Y653 I885 M887 C890 F943 D954 F955 A32 L55 A56 V64 Y66 I80 M82 C85 F138 D149 F150 D936 K938 N941 D954 T986 D131 K133 N136 D149 T155 2.7.11.1 0004672,0005524,0006468 ic50=0.4nM remove_due_to_license_issue IC50=0.400000nM Q9NZJ5 22827572 1102 GRYLTDFEPIQCLGRGGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEKNKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRDLKPSNIFFTMDDVVKVGDFGLVGTKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDL 4g34 A 2.7 BS01 924 A 1 A619 L642 Y653 M887 C890 D954 A34 L57 Y68 M84 C87 D151 D936 K938 N941 D954 T986 D133 K135 N138 D151 T156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=>300nM Q9NZJ5 22827572 1101 GRYLTDFEPIQCLGRGGFGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEKNKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRDLKPSNIFFTMDDVVKVGDFGLGTKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFED 4g3e A 2.5 BS01 0WC A 1 G411 V416 A429 V455 I469 M471 L474 L524 C535 D536 G64 V69 A82 V108 I122 M124 L127 L177 C188 D189 D517 K519 N522 D536 T561 D170 K172 N175 D189 T201 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 22921830 703 PVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 4g3f A 1.642 BS01 0WB A 1 V408 V416 A429 V430 K431 E442 I469 M471 L473 L524 C535 D536 V56 V64 A77 V78 K79 E90 I117 M119 L121 L172 C183 D184 D517 K519 N522 D536 T561 D165 K167 N170 D184 T197 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 22921830 701 SGSVSSGQAHSLASLAKTWSGPETEDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPRG 4g3g A 2.5 BS01 0WA A 1 L408 V416 A429 V430 K431 E442 I469 M471 L524 C535 D536 L56 V64 A77 V78 K79 E90 I117 M119 L172 C183 D184 D517 K519 N522 D536 T561 D165 K167 N170 D184 T197 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 22921830 701 SGSVSSGQAHSLASLAKTWSGPETEDNEGVLLTEKLKPVDYEYREEVHWMTHQPRLGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPRG 4g4p A 1.5 BS01 GLN A 1 F33 F71 A88 G89 M90 S91 R96 K136 T139 E140 D180 F24 F62 A79 G80 M81 S82 R87 K127 T130 E131 D171 ? 0015276,0016020 Kd=0.13uM remove_due_to_license_issue Q837S0 23994008 302 HHGENLYFQGMEGKKYTIGTDLTFAPFEFQDSKGKYIGIDVDLLDAIAKDQDFEVDLKPLGFDSAVQAIQSKQIDGMIAGMSITDERKKSFDFSDPYFDSGLQLAVKKGNDKIKSYDDLKGKTVAAKVGTESANFLEKNKEKYDYTIKNFDDATGLYKALENGEADAIVDDYPVLGYAVKNGQKLQLVGDKETGSSYGFAVKKGQNPELIKKFNAGLKNLKDNGTYDKILNNYLA 4g55 A 1.69 BS01 VH2 A 1 V50 I52 R64 I80 F91 K96 K98 V51 I53 R65 I81 F92 K97 K99 ? 0005198,0006886,0016192,0030130,0030132 remove_due_to_license_issue Q00610 21816279 418 FMAQILPIRFQEHLQLQNLGINPANIGFSTLTMESDKFICIREKVGEQAQVVIIDMNDPSNPIRRPISADSAIMNPASKVIALKAGKTLQIFNIEMKSKMKAHTMTDDVTFWKWISLNTVALVTDNAVYHWSMEGESQPVKMFDRHSSLAGCQIINYRTDAKQKWLLLTGISAQQNRVVGAMQLYSVDRKVSQPIEGHAASFAQFKMEGNAEESTLFCFAVRGQAGGKLHIIEVGTPPTGNQPFPKKAVDVFFPPEAQNDFPVAMQISEKHDVVFLITKYGYIHLYDLETGTCIYMNRISGETIFVTAPHEATAGIIGVNRKGQVLSVCVEEENIIPYITNVLQNPDLALRMAVRNNL 4g5f A 2.33 BS01 0JD A 1 P38 T39 M40 H47 Q164 P35 T36 M37 H44 Q157 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D81 D82 Q85 K153 S189 S190 R191 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=0.7mM remove_due_to_license_issue P9WIL5 23872845 402 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 4g5y A 1.8 BS02 0OC A 1 P38 T39 M40 F67 N69 Q72 V142 P35 T36 M37 F64 N66 Q69 V139 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D85 D86 Q89 K157 S193 S194 R195 6.3.2.1 0000287,0004592,0005515,0005524,0005737,0005829,0015940,0016874,0019482,0030145,0046872 Kd=1.69mM remove_due_to_license_issue P9WIL5 23872845 403 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 4g8l A 2.8 BS01 25A A 1 E55 E57 G58 W60 Q68 K89 Y124 F126 E131 Y135 R155 E40 E42 G43 W45 Q53 K74 Y109 F111 E116 Y120 R140 3.1.26.- remove_due_to_license_issue IC50=20nM, EC50=0.210000nM Q05823 23084743 401 SSGRRAAVEDNHLLIKAVQNEDVDLVQQLLEGGANVNFQEEEGGWTPLHNAVQMSREDIVELLLRHGADPVLRKKNGATPFILAAIAGSVKLLKLFLSKGADVNECDFYGFTAFMEAAVYGKVKALKFLYKRGANVNLRRKTKEDQERLRGATALMDAAEKGHVEVLKILLDEMGADVNACDNMGRNALIHALLSSDDSDVEAITHLLLDHGADVNVRGERGKTPLILAVEKKHLGLVQRLLEQEHIEINDTDSDGKTALLLAVELKLKKIAELLCKRGASTCGDLVMTARRNYDHSLVKVLLSHGA 4g8l A 2.8 BS02 25A B 1 M306 R309 R310 Y312 M288 R291 R292 Y294 3.1.26.- remove_due_to_license_issue IC50=20nM, EC50=0.210000nM Q05823 23084743 401 SSGRRAAVEDNHLLIKAVQNEDVDLVQQLLEGGANVNFQEEEGGWTPLHNAVQMSREDIVELLLRHGADPVLRKKNGATPFILAAIAGSVKLLKLFLSKGADVNECDFYGFTAFMEAAVYGKVKALKFLYKRGANVNLRRKTKEDQERLRGATALMDAAEKGHVEVLKILLDEMGADVNACDNMGRNALIHALLSSDDSDVEAITHLLLDHGADVNVRGERGKTPLILAVEKKHLGLVQRLLEQEHIEINDTDSDGKTALLLAVELKLKKIAELLCKRGASTCGDLVMTARRNYDHSLVKVLLSHGA 4g8m A 2.05 BS01 G8M A 1 Y58 T88 R93 L135 G138 S139 T140 E190 Y60 T90 R95 L137 G140 S141 T142 E192 ? 0015276,0016020 Kd=12.8nM remove_due_to_license_issue P19491 22789682 301 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4g8n A 2.3 BS01 G8M A 1 Y63 T92 R97 G142 A143 T144 E191 Y60 T89 R94 G139 A140 T141 E188 ? 0015276,0016020 Kd=63nM remove_due_to_license_issue P42264 22789682 301 TNRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 4g8o D 2.71 BS01 96P D 1 W175 K176 T177 Q204 N206 F208 L226 P227 D231 R268 W172 K173 T174 Q201 N203 F205 L223 P224 D228 R265 ? 0001525,0002020,0004867,0005102,0005515,0005576,0005615,0005886,0010469,0010757,0010951,0014912,0030194,0030195,0030336,0031093,0032757,0033629,0035491,0042730,0045766,0048260,0050729,0050829,0051918,0061044,0061045,0062023,0070062,0071222,0090026,0090399,0097180,0097187,1901331,1902042,1904090,2000098,2000352 remove_due_to_license_issue P05121 24297881 403 APSYVAHLASDFGVRVFQQVAQASKDRNVVFSPYGVASVLAMLQLTTGGETQQQIQAAMGFKIDDKGMAPALRHLYKELMGPWNKDEISTTDAIFVQRDLKLVQGFMPHFFRLFRSTVKQVDFSEVERARFIINDWVKTHTKGMISHLLGTGAVDQLTRLVLVNALYFNGQWKTPFPDSSTHRRLFHKSDGSTVSVPMMAQTNKFNYTEFTTPDGHYYDILELPYHGDTLSMFIAAPYEKEVPLSALTNILSAQLISHWKGNMTRLPRLLVLPKFSLETEVDLRKPLENLGMTDMFRQFQADFTSLSDQEPLHVALALQKVKIEVNESVIVSARMAPEEIIIDRPFLFVVRHNPTGTVLFMGQVMEP 4g8r B 2.19 BS01 96P B 1 S6 Y7 H10 S3 Y4 H7 ? 0001525,0002020,0004867,0005102,0005515,0005576,0005615,0005886,0010469,0010757,0010951,0014912,0030194,0030195,0030336,0031093,0032757,0033629,0035491,0042730,0045766,0048260,0050729,0050829,0051918,0061044,0061045,0062023,0070062,0071222,0090026,0090399,0097180,0097187,1901331,1902042,1904090,2000098,2000352 Kd=22nM remove_due_to_license_issue P05121 24297881 402 APSYVAHLASDFGVRVFQQVAQASKDRNVVFSPYGVASVLAMLQLTTGGETQQQIQAAMGFKIDDKGMAPALRHLYKELMGPWNKDEISTTDAIFVQRDLKLVQGFMPHFFRLFRSTVKQVDFSEVERARFIINDWVKTHTKGMISHLLGTGAVDQLTRLVLVNALYFNGQWKTPFPDSSTHRRLFHKSDGSTVSVPMMAQTNKFNYTEFTTPDGHYYDILELPYHGDTLSMFIAAPYEKEVPLSALTNILSAQLISHWKGNMTRLPRLLVLPKFSLETEVDLRKPLENLGMTDMFRQFQADFTSLSDQEPLHVALALQKVKIEVNESAVIVSARMAPEEIIIDRPFLFVVRHNPTGTVLFMGQVMEP 4g8r B 2.19 BS02 96P B 2 S41 M45 L75 R76 Y79 F117 R118 S38 M42 L72 R73 Y76 F114 R115 ? 0001525,0002020,0004867,0005102,0005515,0005576,0005615,0005886,0010469,0010757,0010951,0014912,0030194,0030195,0030336,0031093,0032757,0033629,0035491,0042730,0045766,0048260,0050729,0050829,0051918,0061044,0061045,0062023,0070062,0071222,0090026,0090399,0097180,0097187,1901331,1902042,1904090,2000098,2000352 Kd=22nM remove_due_to_license_issue P05121 24297881 403 APSYVAHLASDFGVRVFQQVAQASKDRNVVFSPYGVASVLAMLQLTTGGETQQQIQAAMGFKIDDKGMAPALRHLYKELMGPWNKDEISTTDAIFVQRDLKLVQGFMPHFFRLFRSTVKQVDFSEVERARFIINDWVKTHTKGMISHLLGTGAVDQLTRLVLVNALYFNGQWKTPFPDSSTHRRLFHKSDGSTVSVPMMAQTNKFNYTEFTTPDGHYYDILELPYHGDTLSMFIAAPYEKEVPLSALTNILSAQLISHWKGNMTRLPRLLVLPKFSLETEVDLRKPLENLGMTDMFRQFQADFTSLSDQEPLHVALALQKVKIEVNESAVIVSARMAPEEIIIDRPFLFVVRHNPTGTVLFMGQVMEP 4g8v A 1.7 BS01 0EY A 1 K7 Q11 H12 K41 N44 T45 H119 F120 K7 Q11 H12 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=1.6uM remove_due_to_license_issue P61823 23122937 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 4g8y A 1.8 BS01 0FT A 1 Q11 H12 K41 N44 T45 H119 F120 Q11 H12 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=25.8uM remove_due_to_license_issue P61823 23122937 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 4g90 A 1.9 BS01 0G0 A 1 K7 Q11 H12 K41 N44 T45 H119 F120 K7 Q11 H12 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=30.8uM remove_due_to_license_issue P61823 23122937 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 4g92 A 1.8 BS01 dna D 0 Y268 L269 H270 R273 H274 M278 R282 P284 G285 G286 F288 Y37 L38 H39 R42 H43 M47 R51 P53 G54 G55 F57 ? 0003700,0006355 remove_due_to_license_issue P87249 22902862 1 ~ 25 SPLYVNAKQFHRILKRRVARQKLEEQLRLTSKGRKPYLHESRHNHAMRRPRGPGGRFLTAD 4g92 A 1.8 BS02 dna E 0 H270 S272 R273 H276 R280 R287 F288 T290 A291 H39 S41 R42 H45 R49 R56 F57 T59 A60 ? 0003700,0006355 remove_due_to_license_issue P87249 22902862 1 ~ 25 SPLYVNAKQFHRILKRRVARQKLEEQLRLTSKGRKPYLHESRHNHAMRRPRGPGGRFLTAD 4g92 B 1.8 BS01 dna D 0 P49 I50 A51 N52 R55 P9 I10 A11 N12 R15 ? 0001228,0005634,0006355,0016602,0043565,0046982 remove_due_to_license_issue Q5B5Z6 22902862 1 ~ 25 MKEQDRWLPIANVARIMKLALPENAKIAKEAKECMQECVSEFISFITSEASEKCQQEKRKTVNGEDILFAMTSLGFENYAEALKIYLSKYRE 4g92 B 1.8 BS02 dna E 0 K42 Q44 K66 I67 A68 K69 K2 Q4 K26 I27 A28 K29 ? 0001228,0005634,0006355,0016602,0043565,0046982 remove_due_to_license_issue Q5B5Z6 22902862 1 ~ 25 MKEQDRWLPIANVARIMKLALPENAKIAKEAKECMQECVSEFISFITSEASEKCQQEKRKTVNGEDILFAMTSLGFENYAEALKIYLSKYRE 4g92 C 1.8 BS01 dna D 0 K93 M104 I105 S106 A107 K47 M58 I59 S60 A61 ? 0003677,0046982 remove_due_to_license_issue C8V0B5 22902862 1 ~ 25 GTWANVNQGLQGTARDILTTYWQHVINHLESDNHDYKIHQLPLARIKKVMKADPEVKMISAEAPILFAKGCDVFITELTMRAWIHAEDNKRRTLQRSDIAAALSKSDMFDFLIDIVP 4g92 C 1.8 BS02 dna E 0 P88 L89 A90 R91 K94 P42 L43 A44 R45 K48 ? 0003677,0046982 remove_due_to_license_issue C8V0B5 22902862 1 ~ 25 GTWANVNQGLQGTARDILTTYWQHVINHLESDNHDYKIHQLPLARIKKVMKADPEVKMISAEAPILFAKGCDVFITELTMRAWIHAEDNKRRTLQRSDIAAALSKSDMFDFLIDIVP 4g93 B 4.2 BS01 0YP B 1 P25 D29 L30 T33 W102 S106 P25 D29 L30 T33 W102 S106 ? 0005198 remove_due_to_license_issue P03147 23871485 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHASPHHTALRQAILAWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISALTFGRETVLEYLVSFGVWIRTPPAYRPPNAPIL 4g93 C 4.2 BS01 0YP B 1 R127 T128 R127 T128 ? 0005198 remove_due_to_license_issue P03147 23871485 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHASPHHTALRQAILAWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISALTFGRETVLEYLVSFGVWIRTPPAYRPPNAPI 4g93 C 4.2 BS02 0YP C 1 P25 L30 W102 Y118 P25 L30 W102 Y118 ? 0005198 remove_due_to_license_issue P03147 23871485 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHASPHHTALRQAILAWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISALTFGRETVLEYLVSFGVWIRTPPAYRPPNAPI 4g95 A 1.35 BS01 OAG A 1 I7 V8 A9 L22 E30 F31 F34 S59 I7 V8 A9 L22 E30 F31 F34 S59 L22 E30 L22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=24.4nM remove_due_to_license_issue Ki=24nM P00374 23545530 201 VGSLNCIVAVSQNMGIGKNGDLPWPPLRNEFRYFQRMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 4g9c A 3.5 BS01 0WP A 1 I463 A481 K483 E501 L505 L514 I527 T529 W531 C532 H574 F583 G593 D594 F595 I16 A34 K36 E54 L58 L67 I80 T82 W84 C85 H127 F136 G146 D147 F148 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S158 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 22954737 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4ga3 A 2.39 BS01 4GA A 1 F99 D103 D107 R112 Q171 K200 D243 K257 F92 D96 D100 R105 Q164 K193 D236 K250 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K193 F232 D236 D237 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 23610597 1001 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4gah A 2.3 BS01 0ET A 1 D161 M176 T177 A178 R206 K207 L229 I231 D95 M110 T111 A112 R140 K141 L163 I165 3.1.2.2 Ki=0.8uM remove_due_to_license_issue Q5T1C6 22871024 301 LKDCSVPNPSWNKDLRLLFDQFMKKCEDGSWKRLPSYKRSQAQLFTRSFDDGLGFEYVMFYNDIEKRMVCLFQGGPYLEGPPGFIHGGAIATMIDATVGMCAMMAGGIVMTANLNINYKRPIPLCSVVMINSQLDKVEGRKFFVSCNVQSVDEKTLYSEATSLFIKLNPAKS 4gah A 2.3 BS02 0ET B 1 G146 P147 H152 G153 N183 Y184 K185 R186 P187 G80 P81 H86 G87 N117 Y118 K119 R120 P121 3.1.2.2 Ki=0.8uM remove_due_to_license_issue Q5T1C6 22871024 601 LKDCSVPNPSWNKDLRLLFDQFMKKCEDGSWKRLPSYKRSQAQLFTRSFDDGLGFEYVMFYNDIEKRMVCLFQGGPYLEGPPGFIHGGAIATMIDATVGMCAMMAGGIVMTANLNINYKRPIPLCSVVMINSQLDKVEGRKFFVSCNVQSVDEKTLYSEATSLFIKLNPAKS 4gah B 2.3 BS01 0ET A 1 P147 H152 G153 N183 Y184 K185 R186 P187 P98 H103 G104 N134 Y135 K136 R137 P138 3.1.2.2 Ki=0.8uM remove_due_to_license_issue Q5T1C6 22871024 301 LKDCSVPNPSWNKDLRLLFDQFMKKCEDGSWKRLPSYKRTPTEWIQDFKTHFLDPKSQAQLFTRSFDDGLGFEYVMFYNDIEKRMVCLFQGGPYLEGPPGFIHGGAIATMIDATVGMCAMMAGGIVMTANLNINYKRPIPLCSVVMINSQLDKVEGRKFFVSCNVQSVDEKTLYSEATSLFIKLNPAKSLTLEHH 4gah B 2.3 BS02 0ET B 1 M176 T177 A178 R206 K207 L229 I231 H244 M127 T128 A129 R157 K158 L180 I182 H195 3.1.2.2 Ki=0.8uM remove_due_to_license_issue Q5T1C6 22871024 601 LKDCSVPNPSWNKDLRLLFDQFMKKCEDGSWKRLPSYKRTPTEWIQDFKTHFLDPKSQAQLFTRSFDDGLGFEYVMFYNDIEKRMVCLFQGGPYLEGPPGFIHGGAIATMIDATVGMCAMMAGGIVMTANLNINYKRPIPLCSVVMINSQLDKVEGRKFFVSCNVQSVDEKTLYSEATSLFIKLNPAKSLTLEHH 4gah B 2.3 BS03 0ET B 2 W86 M169 W44 M120 3.1.2.2 Ki=0.8uM remove_due_to_license_issue Q5T1C6 22871024 602 LKDCSVPNPSWNKDLRLLFDQFMKKCEDGSWKRLPSYKRTPTEWIQDFKTHFLDPKSQAQLFTRSFDDGLGFEYVMFYNDIEKRMVCLFQGGPYLEGPPGFIHGGAIATMIDATVGMCAMMAGGIVMTANLNINYKRPIPLCSVVMINSQLDKVEGRKFFVSCNVQSVDEKTLYSEATSLFIKLNPAKSLTLEHH 4gb9 A 2.438 BS01 0WR A 1 K802 W812 I831 K833 Y867 I879 E880 I881 V882 K890 M953 I963 D964 K564 W574 I593 K595 Y629 I641 E642 I643 V644 K652 M715 I725 D726 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=540nM P48736 22877085 1201 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIAAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 4gbd A 1.975 BS01 MCF A 1 H74 M77 L89 W92 E101 M132 F134 P155 H194 H221 E224 H258 D309 H69 M72 L84 W87 E96 M127 F129 P150 H189 H216 E219 H253 D304 ? 0004000,0016787,0016810,0046872,0090614 Ki=0.0048nM remove_due_to_license_issue Q9HZ64 23050701 501 NPFDLLLLPTWIVPVEPAGVVLRDHALGIRDGQIALVAPREQAMRHGATEIRELPGMLLAPGLVNAHGHSAMSLFRGLADDLPLMTWLQDHIWPAEGQWVSEDFIRDGTELAIAEQVKGGITCFSDMYFYPQAICGVVHDSGVRAQVAIPVLDFPIPGARDSAEAIRQGMALFDDLKHHPRIRIAFGPHAPYTVSDDKLEQILVLTEELDASIQMHVHETAFEVEQAMERNGERPLARLHRLGLLGPRFQAVHMTQVDNDDLAMLVETNSSVIHCPESNLKLASGFCPVEKLWQAGVNVAIGTDGAASNNDLDLLGETRTAALLAKAVYGQATALDAHRALRMATLNGARALGLERLIGSLEAGKAADLVAFDLSGLAQQPVYDPVSQLIYASGRDCVRHVWVGGRQLLDDGRLLRHDEQRLIARAREWGAKIAA 4gcj A 1.42 BS01 X64 A 1 I10 V18 A31 K33 F80 L83 H84 Q85 D86 K89 N132 L134 D145 I16 V24 A37 K39 F86 L89 H90 Q91 D92 K95 N138 L140 D151 D127 K129 Q131 N132 D145 T158 T165 D133 K135 Q137 N138 D151 T164 T171 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=1.1nM P24941 23600925 305 LGSPEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4gck A 2.05 BS01 dna W 0 R11 V43 S44 A46 A47 R50 R3 V35 S36 A38 A39 R42 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue B5XTG2 23754405 2 ~ 13 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLILGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEVQLRQVMREKKMREGEGYTLDETLLASQLLAFCEGMLSRFVRSEFKYRPTDDFEARWPLVAAQLQ 4gck A 2.05 BS02 dna Z 0 R31 T33 T34 E45 Y49 S54 K55 R23 T25 T26 E37 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue B5XTG2 23754405 23 ~ 34 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLILGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEVQLRQVMREKKMREGEGYTLDETLLASQLLAFCEGMLSRFVRSEFKYRPTDDFEARWPLVAAQLQ 4gck B 2.05 BS01 dna W 0 R31 T33 T34 E45 Y49 S54 K55 R22 T24 T25 E36 Y40 S45 K46 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue B5XTG2 23754405 2 ~ 13 NRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLILGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEVQLRQVMREKKMREGEGYTLDETLLASQLLAFCEGMLSRFVRSEFKYRPTDDFEARWPLVAAQLQ 4gck C 2.05 BS01 dna W 0 R31 T33 T34 E45 Y49 S54 K55 R23 T25 T26 E37 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue B5XTG2 23754405 2 ~ 13 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLILGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEVQLRQVMREKKMREGEGYTLDETLLASQLLAFCEGMLSRFVRSEFKYRPTDDFEARWPLVAAQLQ 4gck C 2.05 BS02 dna Z 0 V43 S44 A46 A47 R50 V35 S36 A38 A39 R42 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue B5XTG2 23754405 23 ~ 34 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLILGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEVQLRQVMREKKMREGEGYTLDETLLASQLLAFCEGMLSRFVRSEFKYRPTDDFEARWPLVAAQLQ 4gck D 2.05 BS01 dna Z 0 R31 T33 T34 E45 Y49 S54 K55 R22 T24 T25 E36 Y40 S45 K46 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue B5XTG2 23754405 23 ~ 34 NRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLILGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEVQLRQVMREKKMREGEGYTLDETLLASQLLAFCEGMLSRFVRSEFKYRPTDDFEARWPLVAAQLQ 4gcl A 2.65 BS01 dna W 0 S44 A46 A47 R50 H51 S36 A38 A39 R42 H43 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 1 ~ 14 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl A 2.65 BS02 dna Z 0 R31 T33 T34 Y49 K55 R23 T25 T26 Y41 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 22 ~ 35 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl B 2.65 BS01 dna W 0 R31 T33 T34 E45 Y49 S54 K55 R29 T31 T32 E43 Y47 S52 K53 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 1 ~ 14 AEKQAKRNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl C 2.65 BS01 dna W 0 R31 T33 T34 A46 Y49 S54 K55 R23 T25 T26 A38 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 1 ~ 14 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl C 2.65 BS02 dna Z 0 R11 S44 A46 A47 R50 H51 R3 S36 A38 A39 R42 H43 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 22 ~ 35 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl D 2.65 BS01 dna Z 0 R31 T33 T34 E45 Y49 K55 R22 T24 T25 E36 Y40 K46 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 22 ~ 35 NRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl E 2.65 BS01 dna R 0 R31 T33 T34 E45 A46 Y49 S54 K55 R23 T25 T26 E37 A38 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 1 ~ 14 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl E 2.65 BS02 dna T 0 R9 R11 S44 A46 A47 R50 H51 R1 R3 S36 A38 A39 R42 H43 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 22 ~ 35 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl F 2.65 BS01 dna T 0 R31 T33 T34 E45 Y49 S54 K55 R22 T24 T25 E36 Y40 S45 K46 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 22 ~ 35 NRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl G 2.65 BS01 dna R 0 R11 S44 A46 A47 R50 H51 R3 S36 A38 A39 R42 H43 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 1 ~ 14 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl G 2.65 BS02 dna T 0 R31 T33 T34 E45 Y49 S54 K55 R23 T25 T26 E37 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 22 ~ 35 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gcl H 2.65 BS01 dna R 0 R31 T33 T34 E45 Y49 S54 K55 R23 T25 T26 E37 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q1R4V1 23754405 1 ~ 14 RNRREEILQSLALMLESSDGSQRITTAKLAASVGVSEAALYRHFPSKTRMFDSLIEFIEDSLITRINLILKDEKDTTARLRLIVLLLLGFGERNPGLTRILTGHALMFEQDRLQGRINQLFERIEAQLRQVLREKRMREGEGYATDETLLASQILAFCEGMLSRFVRSEFKYRPTDDFDARWPLIAAQLQ 4gct A 2.45 BS01 dna W 0 R9 V41 S42 A44 A45 R48 R3 V35 S36 A38 A39 R42 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 1 ~ 20 INRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gct A 2.45 BS02 dna Z 0 R29 T31 T32 E43 Y47 S52 K53 R23 T25 T26 E37 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 19 ~ 38 INRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gct B 2.45 BS01 dna W 0 R29 T31 T32 E43 Y47 S52 K53 R22 T24 T25 E36 Y40 S45 K46 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 1 ~ 20 NRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKLREGKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gct C 2.45 BS01 dna W 0 T31 T32 E43 Y47 S52 K53 T25 T26 E37 Y41 S46 K47 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 1 ~ 20 INRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKLREGKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gct C 2.45 BS02 dna Z 0 R9 S42 A44 A45 R48 R3 S36 A38 A39 R42 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 19 ~ 38 INRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKLREGKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gct D 2.45 BS01 dna W 0 S42 R48 S35 R41 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 1 ~ 20 NRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKLREGKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gct D 2.45 BS02 dna Z 0 R29 T31 T32 E43 Y47 K53 R22 T24 T25 E36 Y40 K46 ? 0000976,0003677,0003700,0005737,0006355,0009295,0010974,0043565,0043590,0051301,0051302 remove_due_to_license_issue Q9KVD2 23754405 19 ~ 38 NRREEILQALAEMLESNEGASRITTAKLAKQVGVSEAALYRHFPSKTRMFEGLIEFIEESLMSRINRIFDEEKDTLNRIRLVMQLLLAFAERNPGLTRILSGHALMFENERLRDRINQLFERIETSLRQILRERKLREGKSFPVDENILAAQLLGQVEGSLNRFVRSDFKYLPTANFDEYWALLSAQIK 4gd6 A 1.53 BS01 17K A 1 S70 S130 L220 T235 G236 A237 R244 N276 S45 S105 L195 T210 G211 A212 R218 N249 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 23145056 301 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 4gdy A 2.89 BS01 0X1 A 1 G116 S117 Q118 Y142 N202 D230 P232 S260 S262 R270 R399 G109 S110 Q111 Y135 N195 D223 P225 S253 S255 R263 R386 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gdy A 2.89 BS02 0X1 B 1 R20 G39 Y74 S75 L293 R20 G32 Y67 S68 L286 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gdy B 2.89 BS01 0X1 A 1 I19 M33 G39 Y74 S75 I19 M33 G39 Y74 S75 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gdy B 2.89 BS02 0X1 B 1 G116 S117 Q118 Y142 N202 D230 P232 S260 S262 R270 R399 G116 S117 Q118 Y142 N202 D230 P232 S260 S262 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge1 A 2.15 BS01 TSS A 1 I25 F59 D72 V109 V124 I24 F58 D71 V108 V123 ? 0051381,0070026 remove_due_to_license_issue Q86PT9 23275168 201 SGCSTVDTVKDFNKDNFFTGSWYITHYKLGDSTLEVGDKNCTKFLHQKTADGKIKEVFSNYNPNAKTYSYDISFAKVSDFDGNNGKYTAKNVIVEKDGRKIDERTLQVSYIDTDYSKYSVVHVCDPAAPDYYLYAVQSRTENVKEDVKSKVEAALGKVGLKLSGLFDATTLGNKCQYDDETLQKLLKQSFPNYEK 4ge2 A 1.8 BS01 75A A 1 Y333 D335 C515 S516 A517 I519 G520 R521 F556 Q559 Y57 D59 C230 S231 A232 I234 G235 R236 F271 Q274 D470 C515 R521 T522 Q559 D194 C230 R236 T237 Q274 3.1.3.48 0004725,0006470,0016311 ic50=0.9uM remove_due_to_license_issue P43378 23075115 601 SVHVPGPHAMTIQELVDYVNARQKQGIYEEYEDIRRENPVGTFHCSMSPGNLEKNRYGDVPCLDQTRVKLTKRSGHTQTDYINASFMDGYKQKNAYIGTQGPLENTYRDFWLMVWEQKVLVIVMTTRFEEGGRRKCGQYWPLEKDSRIRFGFLTVTNLGVENMNHYKKTTLEIHNTEERQKRQVTHFQFLSWPDYGVPSSAASLIDFLRVVRNQQSLAVSNMEPPIVVHCSAGIGRTGTFCSLDICLAQLEELGTLNVFQTVSRMRTQRAFSIQTPEQYYFCYKAILEFAEKEGMVSA 4ge4 A 2.41 BS01 0KE A 1 G116 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 K263 R270 R399 G110 S111 Q112 Y136 N196 D224 P226 Y227 S254 S256 K257 R264 R393 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSSMISLAGGLPNPNMFPFKTAVITVGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge4 A 2.41 BS02 0KE B 1 I19 G38 G39 L40 Y74 I19 G34 G35 L36 Y68 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSSMISLAGGLPNPNMFPFKTAVITVGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge4 B 2.41 BS01 0KE A 1 I19 G38 G39 L40 Y74 I19 G38 G39 L40 Y74 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge4 B 2.41 BS02 0KE B 1 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 K263 R270 R399 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 K263 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge5 A 2.0 BS01 A89 A 1 R311 Y333 D335 C515 S516 A517 I519 G520 R521 F556 Q559 R35 Y57 D59 C230 S231 A232 I234 G235 R236 F271 Q274 D470 C515 R521 T522 Q559 D194 C230 R236 T237 Q274 3.1.3.48 0004725,0006470,0016311 ic50=0.27uM remove_due_to_license_issue P43378 23075115 601 SVHVPGPHAMTIQELVDYVNARQKQGIYEEYEDIRRENPVGTFHCSMSPGNLEKNRYGDVPCLDQTRVKLTKRSGHTQTDYINASFMDGYKQKNAYIGTQGPLENTYRDFWLMVWEQKVLVIVMTTRFEEGGRRKCGQYWPLEKDSRIRFGFLTVTNLGVENMNHYKKTTLEIHNTEERQKRQVTHFQFLSWPDYGVPSSAASLIDFLRVVRNQQSLAVSNMEPPIVVHCSAGIGRTGTFCSLDICLAQLEELGTLNVFQTVSRMRTQRAFSIQTPEQYYFCYKAILEFAEKEGMVSA 4ge6 A 1.4 BS01 B26 A 1 P315 Y333 D335 C515 S516 A517 I519 G520 R521 F556 Q559 P561 P39 Y57 D59 C235 S236 A237 I239 G240 R241 F276 Q279 P281 D470 C515 R521 T522 Q559 D194 C235 R241 T242 Q279 3.1.3.48 0004725,0006470,0016311 Ki=34nM remove_due_to_license_issue P43378 23075115 601 SVHVPGPHAMTIQELVDYVNARQKQGIYEEYEDIRRENPVGTFHCSMSPGNLEKNRYGDVPCLDQTRVKLTKRSGHTQTDYINASFMDGYKQKNAYIGTQGPLENTYRDFWLMVWEQKVLVIVMTTRFEEGGRRKCGQYWPLEKDSRIRFGFLTVTNLGVENMNHYKKTTLEIHNTEERQKRQVTHFQFLSWPDYGVPSSAASLIDFLRVVRNQQSLAVSNMGARCPEPPIVVHCSAGIGRTGTFCSLDICLAQLEELGTLNVFQTVSRMRTQRAFSIQTPEQYYFCYKAILEFAEKEGMVSA 4ge7 A 2.1 BS01 0K5 A 1 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge7 A 2.1 BS02 0K5 B 1 I19 G39 Y74 S75 S77 L293 I19 G39 Y74 S75 S77 L293 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge7 B 2.1 BS01 0K5 A 1 G39 Y74 S75 S77 G39 Y74 S75 S77 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge7 B 2.1 BS02 0K5 B 1 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 501 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge9 A 2.43 BS01 0L0 A 1 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 4000 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge9 A 2.43 BS02 0L0 B 1 I19 R20 T23 G39 L40 Y74 S75 S77 L293 I19 R20 T23 G39 L40 Y74 S75 S77 L293 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 4000 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge9 B 2.43 BS01 0L0 A 1 I19 R20 T23 G39 Y74 S75 S77 I19 R20 T23 G39 Y74 S75 S77 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 4000 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4ge9 B 2.43 BS02 0L0 B 1 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 S117 Q118 Y142 N202 D230 P232 Y233 S260 S262 R270 R399 2.6.1.39,2.6.1.4,2.6.1.63,2.6.1.7,2.6.1.73 0005739,0005759,0006103,0006536,0008483,0009058,0016212,0030170,0033512,0042803,0047315,0047536,0047958,0050094,0070189,1901605 remove_due_to_license_issue Q8N5Z0 24900560 4000 MNYARFITAASAARNPSPIRTMTDILSRGPKSMISLAGGLPNPNMFPFKTAVITVENGKTIQFGEEMMKRALQYSPSAGIPELLSWLKQLQIKLHNPPTIHYPPSQGQMDLCVTSGSQQGLCKVFEMIINPGDNVLLDEPAYSGTLQSLHPLGCNIINVASDESGIVPDSLRDILSRWKPEDAKNPQKNTPKFLYTVPNGNNPTGNSLTSERKKEIYELARKYDFLIIEDDPYYFLQFNSGRVPTFLSMDVDGRVIRADSFSKIISSGLRIGFLTGPKPLIERVILHIQVSTLHPSTFNQLMISQLLHEWGEEGFMAHVDRVIDFYSNQKDAILAAADKWLTGLAEWHVPAAGMFLWIKVKGINDVKELIEEKAVKMGVLMLPGNAFYVDSSAPSPYLRASFSSASPEQMDVAFQVLAQLIKESLLVP 4gee A 1.7 BS01 0WT A 1 N48 S49 E52 D75 R78 G79 I80 P81 T167 V169 N31 S32 E35 D58 R61 G62 I63 P64 T133 V135 5.6.2.2 0003677,0003918,0005524,0006265 Ki<1nM remove_due_to_license_issue Q839Z1 23352267 301 GLEAVRKRPGMYIGSTSGEGLHHLVWEIVDNSIDEALAGFAKSIQVIIEPDDSITVIDDGRGIPVGIQAKTGRPAVETVFTVLHGVGSSVVNALSTSLDVRVYKDGKVYYQEYRRGAVVDDLKVIEETDRHGTTVHFIPDPEIFTETTVYDFDKLATRVRELAFLNRGLHISIEDRREGQEDKKEYHYEGLEH 4gfd A 1.8 BS01 0YB A 1 E37 R48 L52 F66 R70 R92 S97 Y100 Q101 E36 R47 L51 F63 R67 R89 S94 Y97 Q98 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 Ki=330pM remove_due_to_license_issue P65248 22908966 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIDQEDLKFHEKVIEGYQEIIHQRFKSVNADQPLENVVEDTYQTIIKYLEK 4gfm A 2.3 BS01 0X2 A 1 G856 K857 V863 A880 M929 E930 Y931 R980 N981 L983 G993 D994 G17 K18 V24 A41 M90 E91 Y92 R141 N142 L144 G154 D155 D976 A978 R980 N981 D994 S1016 D137 A139 R141 N142 D155 S177 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.06uM remove_due_to_license_issue O60674 23867602 1201 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4gfn A 1.9 BS01 SUY A 1 N48 S49 E52 D75 R78 G79 I80 P81 T167 N31 S32 E35 D58 R61 G62 I63 P64 T133 5.6.2.2 0003677,0003918,0005524,0006265 Ki=5nM remove_due_to_license_issue Q839Z1 23352267 301 GLEAVRKRPGMYIGSTSGEGLHHLVWEIVDNSIDEALAGFAKSIQVIIEPDDSITVIDDGRGIPVGIQAKTGRPAVETVFTVLHGVGSSVVNALSTSLDVRVYKDGKVYYQEYRRGAVVDDLKVIEETDRHGTTVHFIPDPEIFTETTVYDFDKLATRVRELAFLNRGLHISIEDRREGQEDKKEYHYEGLEH 4gfo A 2.3 BS01 0X2 A 1 L903 G904 E905 G906 V911 A928 E979 Y980 V981 N1028 L1030 L14 G15 E16 G17 V22 A39 E73 Y74 V75 N122 L124 N1023 A1025 R1027 N1028 D1041 P1064 N117 A119 R121 N122 D135 P158 2.7.10.2 0004672,0005524,0006468 Ki=0.24uM remove_due_to_license_issue P29597 23867602 1206 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALWKQEIDILRTLYHEHIIKYKGCCELQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHSQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPCEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYRH 4gg5 A 2.423 BS01 0J3 A 1 I1084 L1157 Y1159 M1160 R1208 N1209 M1211 A1221 D1222 Y1230 I21 L87 Y89 M90 R138 N139 M141 A151 D152 Y160 D1204 A1206 R1208 N1209 D1222 A1243 D134 A136 R138 N139 D152 A173 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.93nM remove_due_to_license_issue IC50=0.930000nM P08581 22985853 1401 QAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 4gg7 A 2.27 BS01 0J8 A 1 I1084 L1157 M1160 K1161 G1163 R1208 M1211 A1221 D1222 Y1230 I21 L91 M94 K95 G97 R142 M145 A155 D156 Y164 D1204 A1206 R1208 N1209 D1222 A1243 D138 A140 R142 N143 D156 A177 2.7.10.1 0004672,0004713,0005524,0006468 ic50=6.5nM remove_due_to_license_issue IC50=6.5nM P08581 22985853 1401 QAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 4ggl A 1.69 BS01 CJC A 1 N48 S49 E52 D75 R78 G79 I80 P81 T167 N31 S32 E35 D58 R61 G62 I63 P64 T133 5.6.2.2 0003677,0003918,0005524,0006265 Ki<1nM remove_due_to_license_issue Q839Z1 23352267 301 GLEAVRKRPGMYIGSTSGEGLHHLVWEIVDNSIDEALAGFAKSIQVIIEPDDSITVIDDGRGIPVGIQAKTGRPAVETVFTVLHGVGSSVVNALSTSLDVRVYKDGKVYYQEYRRGAVVDDLKVIEETDRHGTTVHFIPDPEIFTETTVYDFDKLATRVRELAFLNRGLHISIEDRREGQEDKKEYHYEGLEH 4ggz A 1.75 BS01 BTN A 1 R17 S19 N37 A39 F42 A43 F66 C69 S71 T73 W75 W88 R11 S13 N31 A33 F36 A37 F60 C63 S65 T67 W69 W82 ? 0009374 Kd=0.066nM remove_due_to_license_issue Q89U61 23661323 900 LPAPSYWKNERGSELLIWSANSGTIQGTFTNHAQGFACQGIPYPAAGSVSPTGLYFVVTFAQCNSFTRWVGTIKGSQMPTSWTLFYVDNKGKPSRLKGGDIFTRVW 4gh6 A 2.7 BS01 LUO A 1 H252 M365 L420 A452 Q453 F456 H72 M185 L240 A272 Q273 F276 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76083 22985069 601 PTYPKYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQKK 4gha A 2.5 BS01 rna I 0 G223 T226 P295 G16 T19 P88 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4gha A 2.5 BS02 rna J 0 F228 N261 Q263 A264 T267 I329 F21 N54 Q56 A57 T60 I122 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4gha C 2.5 BS01 rna J 0 F228 N261 T267 I329 F21 N54 T60 I122 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4gha E 2.5 BS01 rna I 0 G223 P295 K298 G16 P88 K91 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4gha E 2.5 BS02 rna J 0 F228 N261 Q263 T267 I329 F21 N54 Q56 T60 I122 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4gha G 2.5 BS01 rna I 0 T226 P295 T19 P88 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4gha G 2.5 BS02 rna J 0 N261 Q263 T267 I329 N54 Q56 T60 I122 ? remove_due_to_license_issue P35259 23028316 1 ~ 12 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFLGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4ghi A 1.5 BS01 0X3 A 1 F244 H248 M252 F254 Y281 S292 L296 S304 Y307 M309 T321 C339 N341 F9 H13 M17 F19 Y46 S57 L61 S69 Y72 M74 T86 C98 N100 ? Kd=81nM remove_due_to_license_issue Kd=90nM, IC50=490nM Q99814 23434853 401 FKGLDSKTFLSEHSMDMKFTYCDDRITELIGYHPEELLGRSAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGGYVWLETQGTVIYPQCIMCVNYVLSEIE 4ghl D 2.02 BS01 rna E 0 N261 Q263 A264 T267 R271 I329 N54 Q56 A57 T60 R64 I122 ? remove_due_to_license_issue Q03039 23185024 1 ~ 18 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFMGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4ghl D 2.02 BS02 rna F 0 T226 P295 K298 T19 P88 K91 ? remove_due_to_license_issue Q03039 23185024 1 ~ 18 LSAKDLALLLFTHLPGNNTPFHILAQVLSKIAYKSGKSGAFLDAFHQILSEGENAQAALTRLSRTFDAFMGVVPPVIRVKNFQTVPRPCQKSLRAVPPNPTIDKGWVCVYSSEQGETRALKI 4ght A 1.96 BS01 AG7 A 1 R39 H40 E71 L125 N126 L127 S128 K130 T142 K143 A144 C147 H161 I162 G163 G164 N165 F170 R40 H41 E72 L126 N127 L128 S129 K131 T143 K144 A145 C148 H162 I163 G164 G165 N166 F171 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 23633597 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 4gid A 2.0 BS01 0GH A 1 G59 Q60 G61 L78 D80 G82 Y119 T120 Q121 F156 D276 G278 T279 T280 N281 R283 G13 Q14 G15 L32 D34 G36 Y73 T74 Q75 F110 D230 G232 T233 T234 N235 R237 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D230 T233 3.4.23.46 0004190,0006508,0016020 Ki=0.017nM remove_due_to_license_issue P56817 22954357 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4gih A 2.0 BS01 0X5 A 1 L903 G904 E905 V911 I960 Y980 V981 G984 L1030 L14 G15 E16 V22 I71 Y91 V92 G95 L141 N1023 A1025 R1027 N1028 D1041 E1050 P1064 N134 A136 R138 N139 D152 E161 P175 2.7.10.2 0004672,0005524,0006468 Ki=0.0048uM remove_due_to_license_issue Ki=4.8nM P29597 23867602 1201 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYR 4gii A 2.31 BS01 0X6 A 1 L903 G904 E905 V911 Y980 V981 G984 R1027 L1030 G1040 L14 G15 E16 V22 Y91 V92 G95 R138 L141 G151 N1023 A1025 R1027 N1028 D1041 E1050 P1064 N134 A136 R138 N139 D152 E161 P175 2.7.10.2 0004672,0005524,0006468 Ki=1.8nM remove_due_to_license_issue P29597 23668484 1201 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYRH 4giu A 1.667 BS04 636 A 1 G137 N138 A179 H183 Y186 R193 G206 G114 N115 A156 H160 Y163 R170 G183 V106 V83 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 Ki=4.7uM remove_due_to_license_issue P9WFX5 24623674 404 VPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQ 4gj2 A 2.4 BS01 0XH A 1 R901 L903 G904 E905 V911 Y980 V981 P982 G984 L1030 G1040 D1041 R12 L14 G15 E16 V22 Y91 V92 P93 G95 L141 G151 D152 N1023 A1025 R1027 N1028 D1041 E1050 P1064 N134 A136 R138 N139 D152 E161 P175 2.7.10.2 0004672,0005524,0006468 Ki=2.5nM remove_due_to_license_issue P29597 23668484 1201 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYR 4gj3 A 2.5 BS01 0XP A 1 R901 L903 G904 E905 V911 Y980 V981 P982 G984 R1027 N1028 L1030 G1040 D1041 R12 L14 G15 E16 V22 Y91 V92 P93 G95 R138 N139 L141 G151 D152 N1023 A1025 R1027 N1028 D1041 E1050 P1064 N134 A136 R138 N139 D152 E161 P175 2.7.10.2 0004672,0005524,0006468 Ki=1.4nM remove_due_to_license_issue P29597 23668484 1201 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYR 4gj6 A 2.58 BS01 0LS A 1 D32 G34 F117 V120 D215 G217 S219 Y220 I291 D37 G39 F120 V123 D219 G221 S223 Y224 I298 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y79 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=14000nM P00797 23425156 1001 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gj6 A 2.58 BS02 0LS A 2 T12 Q13 P111 A115 F117 Y220 F242 T17 Q18 P114 A118 F120 Y224 F246 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y79 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=14000nM P00797 23425156 1002 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gj6 A 2.58 BS03 0LS B 2 L110 F242 L113 F246 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y79 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=14000nM P00797 23425156 1002 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gj7 A 2.8 BS01 0LT A 1 T12 Q13 Y14 V30 D32 G34 Y75 T77 L114 A115 F117 V120 L213 D215 G217 A218 S219 T17 Q18 Y19 V35 D37 G39 Y82 T84 L120 A121 F123 V126 L219 D221 G223 A224 S225 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y82 D221 A224 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=170nM P00797 23425156 1001 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gj8 A 2.5 BS01 0LU A 1 Y75 T77 P111 F112 A115 F117 S219 Y220 Y80 T82 P115 F116 A119 F121 S224 Y225 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y80 D220 A223 3.4.23.15 0004190,0006508 remove_due_to_license_issue Kd=>500000nM P00797 23360239 1001 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gj8 A 2.5 BS02 0LU A 2 M10 L114 Y220 F276 M16 L118 Y225 F280 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y80 D220 A223 3.4.23.15 0004190,0006508 remove_due_to_license_issue Kd=>500000nM P00797 23360239 1002 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gj9 A 2.6 BS01 0M2 A 1 Q13 Y14 V30 Y75 T77 P111 F112 A115 F117 T216 G217 S219 Q17 Y18 V34 Y78 T80 P113 F114 A117 F119 T220 G221 S223 D32 S35 N37 W39 Y75 D215 A218 D36 S39 N41 W43 Y78 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 23360239 1001 LGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gja A 2.6 BS01 0M3 A 1 Q13 D32 G34 Y75 S76 P111 V120 D215 G217 I291 P292 Q19 D38 G40 Y83 S84 P118 V127 D223 G225 I302 P303 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y83 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=500nM P00797 23360239 1001 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gjb A 2.75 BS01 0ME A 1 D32 G34 Y75 S76 F117 V120 D215 G217 D38 G40 Y80 S81 F121 V124 D221 G223 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y80 D221 A224 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 23360239 1001 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gjc A 2.4 BS01 0MJ A 1 D32 G34 Y75 S76 T77 P111 F117 V120 D215 G217 I291 P292 D38 G40 Y83 S84 T85 P118 F124 V127 D223 G225 I302 P303 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y83 D223 A226 3.4.23.15 0004190,0006508 ic50=0.09uM remove_due_to_license_issue IC50=90nM P00797 23360239 1001 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gjd A 2.65 BS01 0N0 A 1 Y14 V30 D32 G34 Y75 S76 T77 P111 F117 V120 D215 G217 I291 Y19 V35 D37 G39 Y82 S83 T84 P117 F123 V126 D221 G223 I300 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y82 D221 A224 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=3.0nM P00797 23360239 1001 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4gk2 A 2.195 BS01 L66 A 1 V635 A651 K653 E670 T699 Y701 M702 G705 L753 D764 V27 A43 K45 E62 T91 Y93 M94 G97 L145 D156 D746 A748 R750 N751 D764 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=40nM P29320 23253074 1001 VHEFAKELDATNISIDKVVGAGEFGEVCSGRLKLPSKKEISVAIKTLKVGYTEKQRRDFLGEASIMGQFDHPNIIRLEGVVTKSKPVMIVTEYMENGSLDSFLRKHDAQFTVIQLVGMLRGIASGMKYLSDMGYVHRDLAARNILINSNLVCKVSDFGLPIRWTSPEAIAYRKFTSASDVWSYGIVLWEVMSYGERPYWEMSNQDVIKAVDEGYRLPPPMDCPAALYQLMLDCWQKDRNNRPKFEQIVSILDKLIRLKIITNLLL 4gk3 A 1.898 BS01 L87 A 1 A651 K653 E670 M674 T699 Y701 M702 G705 L753 S763 A43 K45 E62 M66 T91 Y93 M94 G97 L145 S155 D746 A748 R750 N751 D764 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P29320 23253074 1001 VHEFAKELDATNISIDKVVGAGEFGEVCSGRLKLPSKKEISVAIKTLKVGYTEKQRRDFLGEASIMGQFDHPNIIRLEGVVTKSKPVMIVTEYMENGSLDSFLRKHDAQFTVIQLVGMLRGIASGMKYLSDMGYVHRDLAARNILINSNLVCKVSDFGLSRVLIPIRWTSPEAIAYRKFTSASDVWSYGIVLWEVMSYGERPYWEMSNQDVIKAVDEGYRLPPPMDCPAALYQLMLDCWQKDRNNRPKFEQIVSILDKLIRNPGSLKIITSNLLL 4gk4 A 2.1 BS01 L90 A 1 A651 K653 E670 M674 I697 T699 Y701 M702 L753 S763 D764 A43 K45 E62 M66 I89 T91 Y93 M94 L145 S155 D156 D746 A748 R750 N751 D764 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P29320 23253074 1001 VHEFAKELDATNISIDKVVGAGEFGEVCSGRLKLPSKKEISVAIKTLKVGYTEKQRRDFLGEASIMGQFDHPNIIRLEGVVTKSKPVMIVTEYMENGSLDSFLRKHDAQFTVIQLVGMLRGIASGMKYLSDMGYVHRDLAARNILINSNLVCKVSDFGLSRVLKIPIRWTSPEAIAYRKFTSASDVWSYGIVLWEVMSYGERPYWEMSNQDVIKAVDEGYRLPPPMDCPAALYQLMLDCWQKDRNNRPKFEQIVSILDKLIRNPGSLKIITNLLL 4gkc A 1.3 BS01 RET A 1 W19 A33 Q38 C53 W58 Y60 L77 W106 K108 L117 W19 A33 Q38 C53 W58 Y60 L77 W106 K108 L117 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 23224553 201 TRDANGTWEMESNENFEGWMKALDIDFALRKIAVRLTQTLVIDQDGDNFKVKCTSTFWNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 4gkh A 1.863 BS02 0J9 A 1 V33 F53 I101 I215 V16 F36 I84 I198 K55 D198 N203 D216 K38 D181 N186 D199 0005524,0016773,0046677 remove_due_to_license_issue 23758273 302 NLDADLYGYRWARDNVGQSGATIYRLYGKPNAPELFLKHGKGSVANDVTDEMVRLNWLTAFMPLPTIKHFIRTPDDAWLLTTAIPGKTAFQVLEEYPDSGENIVDALAVFLRRLHSIPVCNCPFNSDRVFRLAQAQSRMNNGLVDASDFDDERNGWPVEQVWKEMHKLLPFSPDSVVTHGDFSLDNLIFDEGKLIGCIDVGRVGIADRYQDLAILWNCLGEFSPSLQKRLFQKYGIDNPDMNKLQFHLMLDEFF 4gki A 1.88 BS02 0JN A 1 D31 F53 A100 I101 I215 D32 F54 A101 I102 I216 K55 D198 N203 D216 K56 D199 N204 D217 0005524,0016773,0046677 remove_due_to_license_issue 23758273 302 GMSHIQRETSCSRPRLNSNLDADLYGYRWARDNVGQSGATIYRLYGKPNAPELFLKHGKGSVANDVTDEMVRLNWLTAFMPLPTIKHFIRTPDDAWLLTTAIPGKTAFQVLEEYPDSGENIVDALAVFLRRLHSIPVCNCPFNSDRVFRLAQAQSRMNNGLVDASDFDDERNGWPVEQVWKEMHKLLPFSPDSVVTHGDFSLDNLIFDEGKLIGCIDVGRVGIADRYQDLAILWNCLGEFSPSLQKRLFQKYGIDNPDMNKLQFHLMLDEFF 4gkm A 1.6683 BS04 683 A 1 N138 A179 P180 Y186 R187 A190 R193 R194 N114 A155 P156 Y162 R163 A166 R169 R170 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 Ki=6.8uM remove_due_to_license_issue P9WFX5 24623674 404 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4glw A 2.0 BS01 0XT A 1 Y77 L79 E107 Y216 Q217 K278 W297 Y47 L49 E77 Y186 Q187 K248 W267 E107 K109 D111 Y216 K302 E77 K79 D81 Y186 K272 6.5.1.2 0003911 Kd=0.8uM remove_due_to_license_issue C1CKI0 23006603 402 NKRMNERELVELETAYPEQVLADSPTHRVGGKVLDGFEKYSHQYPLYSLQDAFSREELDAFDARVRKEVAHPTYICELKIDGLSISLTYEKGILVAGVTRGDGSIGENITENLKRVKDIPLTLPEELDITVRGECYMPRASFDQVNQARQENGEPEFANPRNAAAGTLRQLDTAVVAKRNLATFLYQEASPSTRDSQEKGLKYLEQLGFVVNPKRILAENIDEIWNFIQEVGQERENLPYDIDGVVIKVNDLASQEELGFTVKAPKWAVAYKFPA 4glx A 1.9 BS05 0XS A 1 L80 L114 K115 L116 E173 Y225 V288 K290 W309 L74 L101 K102 L103 E160 Y212 V275 K277 W296 Y225 T427 Y212 T414 6.5.1.2 0003677,0003911,0006260,0006281 remove_due_to_license_issue P15042 23006603 603 SIEQQLTELRTTLRHHEYLYHVMDAPEIPDAEYDRLMRELRELETKHPELITPDSPTQRPLAAFSQIRHEVPMLSLDNVFDEESFLAFNKRVQDRTWCCELKLDGLAVSILYENGVLVSAATRGDGTTGEDITSNVRTIRAIPLKLHGENIPARLEVRGEVFLPQAGFEKINEDARRTGGKVFANPRNAAAGSLRQLDPRITAKRPLTFFCYGVGVLEGGELPDTHLGRLLQFKKWGLPVSDRVTLCESAEEVLAFYHKVEEDRPTLGFDIDGVVIKVNSLAQQEQLGFVARAPRWAVAFKFPAQEQMTFVRDVEFQVGRTGAITPVARLEPVHVAGVLVSNATLHNADEIERLGLRIGDKVVIRRAGDVIPQVVNVVLSERPEDTREVVFPTHCPVCGSDVERVEGEAVARCTGGLICGAQRKESLKHFVSRRAMDVDGMGDKIIDQLVEKEYVHTPADLFKLTAGKLTGLERMGPKSAQNVVNALEKAKETTFARFLYALGIREVGEATAAGLAAYFGTLEALEAASIEELQKVPDVGIVVASHVHNFFAEESNRNVISELLAEGVHWPAP 4gmc B 2.7 BS01 1BI B 1 A396 H428 L492 G493 V494 P495 R503 A374 H406 L470 G471 V472 P473 R481 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 601 SMSYTWTGALITPCAAEMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4gmy A 2.403 BS01 0X5 A 1 V863 Y931 L932 P933 G935 L983 V31 Y99 L100 P101 G103 L151 D976 A978 R980 N981 D994 S1016 D144 A146 R148 N149 D162 S184 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.028uM remove_due_to_license_issue Ki=28nM, EC50=1700nM O60674 23867602 1201 SGAFEDRDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4gny A 1.6367 BS01 SDS A 1 L54 K69 I71 I84 F105 M107 L53 K68 I70 I83 F104 M106 ? 0005515,0005576,0019841,0036041,0036094,0042802 remove_due_to_license_issue P02754 23334914 201 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 4gq4 A 1.27 BS01 0RT A 1 S155 L177 S178 H181 F238 C241 Y276 M278 N282 Y319 Y323 S134 L156 S157 H160 F217 C220 Y255 M257 N261 Y298 Y302 ? 0005634 remove_due_to_license_issue IC50=190nM O00255 22936661 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 4gql A 1.15 BS06 R47 A 1 G178 G179 I180 L181 H183 T215 H218 E219 H222 H228 P232 K233 A234 V235 F237 T239 Y240 G74 G75 I76 L77 H79 T111 H114 E115 H118 H124 P128 K129 A130 V131 F133 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=0.26nM remove_due_to_license_issue Ki=0.260000nM P39900 23343195 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 4gqp H 2.0 BS01 B40 H 1 Y33 S35 Y47 Y50 F95 E101 Y1034 Y1036 H1089 W1091 F1096 Y33 S35 Y47 Y50 F98 E106 Y156 Y158 H211 W213 F218 Kd=0.79nM remove_due_to_license_issue 24419156 1201 EVQLQESGPSLVKPSQTLSLTCSVTGDSVTSGYWSWIRQFPGNKLDYMGYISYRGSTYYNPSLKSRISITRDTSKNQVYLQLKSVSSEDTATYYCTYFDSDDYAMEYWGQGTSVTVSGGGSQIVLTQSPAIMSASPGEKVTLTCSASSSVSSSHLYWYQQKPGSSPKLWIYSTSNLASGVPARFSGSGSGTSYSLTISSMEAEDAASYFCHQWSSFPFTFGSGTKLEIK 4gqq A 1.35 BS01 0XR A 1 D236 S244 K257 G285 F286 V287 P288 D236 S244 K257 G285 F286 V287 P288 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 23050660 502 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 4gqq A 1.35 BS02 0XR A 2 D23 L26 V370 T371 I372 D23 L26 V370 T371 I372 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 23050660 503 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 4gqq A 1.35 BS03 0XR A 3 D77 N81 R85 D77 N81 R85 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 remove_due_to_license_issue P04746 23050660 504 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 4gqr A 1.2 BS02 MYC A 1 W59 Y62 Q63 H101 T163 D197 A198 W59 Y62 Q63 H101 T163 D197 A198 D197 S226 D300 D197 S226 D300 3.2.1.1 0003824,0004556,0005509,0005576,0005615,0005975,0016052,0016160,0016798,0031404,0043169,0044245,0046872,0070062 Ki=110uM remove_due_to_license_issue P04746 23050660 504 QYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL 4gr0 A 1.497 BS06 R4B A 1 G179 I180 L181 A182 H183 T215 H218 E219 H222 H228 K233 A234 V235 F237 T239 Y240 K241 V243 F248 G75 I76 L77 A78 H79 T111 H114 E115 H118 H124 K129 A130 V131 F133 T135 Y136 K137 V139 F144 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=0.28nM remove_due_to_license_issue Ki=0.280000nM P39900 23343195 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 4gr3 A 1.494 BS06 R45 A 1 H172 G179 I180 L181 A182 H183 T215 H218 E219 H222 H228 V235 F237 T239 Y240 H68 G75 I76 L77 A78 H79 T111 H114 E115 H118 H124 V131 F133 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=15.5nM remove_due_to_license_issue Ki=16nM P39900 23343195 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 4gr8 A 1.299 BS06 R4C A 1 G179 L181 A182 H183 T215 H218 E219 H222 H228 V235 F237 T239 Y240 G69 L71 A72 H73 T105 H108 E109 H112 H118 V125 F127 T129 Y130 H218 E219 H222 H228 H108 E109 H112 H118 3.4.24.65 0004222,0006508,0008237,0008270,0031012 Ki=14.7nM remove_due_to_license_issue Ki=15nM P39900 23343195 306 KHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLY 4gs6 A 2.2 BS01 1FM A 1 V42 R44 G45 V50 A61 M104 Y106 A107 G110 P160 N161 L163 C174 D175 V17 R19 G20 V25 A36 M79 Y81 A82 G85 P135 N136 L138 C149 D150 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 23272696 611 GSLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 4gs8 A 2.99 BS01 MGJ A 1 G339 L359 V360 G361 G297 L317 V318 G319 Q111 Q69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue IC50=100nM, EC50=530nM P14735 24735644 1101 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMNLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4gsc A 2.81 BS02 MGW A 1 H332 G339 L359 V360 G361 H291 G298 L318 V319 G320 Q111 Q70 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 24735644 1102 MNNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4gsy A 1.71 BS01 0Y5 A 1 E37 R48 V51 L52 F66 S69 R70 R92 S97 Y100 Q101 E36 R47 V50 L51 F65 S68 R69 R91 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=120nM remove_due_to_license_issue Q6GJI9 23043329 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIDQEDLKFHEKVIEGYQEIIHQRFKSVNADQPLENVVEDTYQTIIKYLEK 4gtm B 2.2 BS03 7TM B 1 L96 A98 S99 W102 A151 P152 D297 D359 Y361 H362 L78 A80 S81 W84 A133 P134 D279 D341 Y343 H344 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H230 R273 K276 D279 C281 Y282 D334 D341 H344 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=9.2nM remove_due_to_license_issue Q02293 22963166 503 WSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 4gto B 2.15 BS02 7TO B 1 W102 R202 C206 C254 D297 W303 Y361 H362 W85 R185 C189 C237 D280 W286 Y344 H345 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H231 R274 K277 D280 C282 Y283 D335 D342 H345 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 ic50=10.5nM remove_due_to_license_issue Q02293 22963166 502 VWSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 4gtp B 2.75 BS03 7TP B 1 Y93 L96 D297 D359 F360 Y361 H362 Y73 L76 D277 D339 F340 Y341 H342 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H228 R271 K274 D277 C279 Y280 D332 D339 H342 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 22963166 503 EPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 4gtq B 2.6 BS03 7TQ B 1 L96 A98 S99 W102 A151 P152 D297 D359 Y361 H362 L78 A80 S81 W84 A133 P134 D279 D341 Y343 H344 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H230 R273 K276 D279 C281 Y282 D334 D341 H344 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 22963166 503 WSEPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 4gtr B 2.2 BS02 7TR B 1 L96 W102 Y105 W106 D297 D359 Y361 H362 Y365 L76 W82 Y85 W86 D277 D339 Y341 H342 Y345 H248 R291 K294 D297 C299 Y300 D352 D359 H362 H228 R271 K274 D277 C279 Y280 D332 D339 H342 2.5.1.58 0003824,0004311,0004659,0004660,0005515,0005875,0005965,0006629,0008270,0008283,0008284,0008285,0008318,0014070,0018343,0034097,0042060,0042277,0045787,0046872,0048144,0048145,0048146,0051770 remove_due_to_license_issue Q02293 22963166 502 EPLYSLRPEHARERLQDDSVETVTSIEQAKVEEKIQEVFSSYKFNHLVPRLVLQREKHFHYLKRGLRQLTDAYECLDASRPWLCYWILHSLELLDEPIPQIVATDVCQFLELCQSPDGGFGGGPGQYPHLAPTYAAVNALCIIGTEEAYNVINREKLLQYLYSLKQPDGSFLMHVGGEVDVRSAYCAASVASLTNIITPDLFEGTAEWIARCQNWEGGIGGVPGMEAHGGYTFCGLAALVILKKERSLNLKSLLQWVTSRQMRFEGGFQGRCNKLVDGCYSFWQAGLLPLLHRALHAQGDPALSMSHWMFHQQALQEYILMCCQCPAGGLLDKPGKSRDFYHTCYCLSGLSIAQHFGSGAMLHDVVMGVPENVLQPTHPVYNIGPDKVIQATTHFLQKPVPGF 4gts B 2.45 BS03 7TP B 1 Y44 L45 W52 D238 F289 Y37 L38 W45 D231 F282 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=12.8nM remove_due_to_license_issue Q08603 22963166 403 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 4gtt B 2.05 BS03 7TQ B 1 Y44 L96 Q103 F147 Y195 D287 F289 Y37 L89 Q96 F140 Y188 D280 F282 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=6nM remove_due_to_license_issue Q08603 22963166 403 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 4gtv B 1.95 BS03 7TR B 1 Y44 L45 C196 D238 W244 F289 H290 Y37 L38 C189 D231 W237 F282 H283 H190 R232 K235 D238 C240 Y241 D280 D287 H290 H183 R225 K228 D231 C233 Y234 D273 D280 H283 2.5.1.60 0003824,0004659,0004661,0004663,0005515,0005968,0006888,0008270,0008318,0018344,0019840,0031267,0046872 ic50=38nM remove_due_to_license_issue Q08603 22963166 403 QKDVTIKSDAPDTLLLEKHADYIASYGSDYEYCMSEYLRMSGVYWGLTVMDLMGQLHRMNKEEILVFIKSCQHECGGVSASIGHDPHLLYTLSAVQILTLYDSIHVINVDKVVAYVQSLQKEDGSFAGDIWGEIDTRFSFCAVATLALLGKLDAINVEKAIEFVLSCMNFDGGFGCRPGSESHAGQIYCCTGFLAITSQLHQVNSDLLGWWLCERQLPSGGLNGRPEKLPDVCYSWWVLASLKIIGRLHWIDREKLRSFILACQDEETGGFADRPGDMVDPFHTLFGIAGLSLLGEEQIKPVSPVFCMPEEVLQRVNVQPELVS 4gu6 A 1.95 BS01 10N A 1 E430 L501 C502 G505 N551 L553 D564 E17 L86 C87 G90 N136 L138 D149 D546 A548 R550 N551 D564 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 Kd=44nM remove_due_to_license_issue IC50=195nM, Kd=44nM Q05397 23294348 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSNPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSRYMEDSTYYKASKGKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4gu9 A 2.4 BS01 4GU A 1 I428 A452 M499 E500 C502 L553 I15 A37 M84 E85 C87 L138 D546 A548 R550 N551 D564 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 Kd=43uM remove_due_to_license_issue Q05397 23294348 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKA 4gue A 1.8 BS01 QCT A 1 F79 K100 V131 L147 D148 L155 E197 L200 L214 F32 K53 V76 L92 D93 L100 E142 L145 L159 D193 K195 E197 N198 D211 T231 D138 K140 E142 N143 D156 T171 2.7.11.1 0004672,0004674,0005524,0006468 Kd=5.8uM remove_due_to_license_issue P18654 23385462 401 KEIAITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVLVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKP 4gui A 1.78 BS01 QIC A 1 E46 R48 R82 H143 K170 M205 R213 F225 A233 Q236 E45 R47 R81 H142 K169 M204 R212 F224 A232 Q235 E86 H143 K170 E85 H142 K169 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0046279 remove_due_to_license_issue P58687 24437575 301 KTVTVRDLVVGEGAPKIIVSLMGKTITDVKSEALAYREADFDILEWRVDHFANVTTAESVLEAAGAIREIITDKPLLFTFRSAKEGGEQALTTGQYIDLNRAAVDSGLVDMIDLELFTGDDEVKATVGYAHQHNVAVIMSNHDFHKTPAAEEIVQRLRKMQELGADIPKIAVMPQTKADVLTLLTATVEMQERYADRPIITMSMSKTGVISRLAGEVFGSAATFGAVKKASAPGQISVADLRTVLTILHQA 4guj A 1.5 BS01 SKM A 1 E46 R48 R82 H143 R213 F225 S232 A233 Q236 E45 R47 R81 H142 R212 F224 S231 A232 Q235 E86 H143 K170 E85 H142 K169 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0046279 remove_due_to_license_issue P58687 24437575 301 KTVTVRDLVVGEGAPKIIVSLMGKTITDVKSEALAYREADFDILEWRVDHFANVTTAESVLEAAGAIREIITDKPLLFTFRSAKEGGEQALTTGQYIDLNRAAVDSGLVDMIDLELFTGDDEVKATVGYAHQHNVAVIMSNHDFHKTPAAEEIVQRLRKMQELGADIPKIAVMPQTKADVLTLLTATVEMQERYADRPIITMSMSKTGVISRLAGEVFGSAATFGAVKKASAPGQISVADLRTVLTILHQA 4guq A 3.7 BS01 dna E 0 K138 R268 K26 R156 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue O15350 23892287 400 ~ 409 EFIPSNTDYPGPHHFEVTFQQSSTAKFATWTYSPLLKKLYCQIAKTCPIQIKVSTPPPPGTAIRAMPVYKKAEHVTDVVKRCPNHELGRDFNEGQSAPASHLIRVEGNNLSQYVDDPVTGRQSVVVPYEPPQVGTEFTTILYNFMCNSSCVGGMNRRPILIIITLEMRDGQVLGRRSFEGRICACPGRDRKADEDHYREQ 4guq A 3.7 BS02 dna F 0 S261 R293 C295 A296 R300 S149 R181 C183 A184 R188 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue O15350 23892287 410 ~ 419 EFIPSNTDYPGPHHFEVTFQQSSTAKFATWTYSPLLKKLYCQIAKTCPIQIKVSTPPPPGTAIRAMPVYKKAEHVTDVVKRCPNHELGRDFNEGQSAPASHLIRVEGNNLSQYVDDPVTGRQSVVVPYEPPQVGTEFTTILYNFMCNSSCVGGMNRRPILIIITLEMRDGQVLGRRSFEGRICACPGRDRKADEDHYREQ 4guq B 3.7 BS01 dna E 0 S261 R293 A296 S148 R180 A183 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue O15350 23892287 400 ~ 409 EFIPSNTDYPGPHHFEVTFQQSSTAKFATWTYSPLLKKLYCQIAKTCPIQIKVTPPPPGTAIRAMPVYKKAEHVTDVVKRCPNHELGRDFNEGQSAPASHLIRVEGNNLSQYVDDPVTGRQSVVVPYEPPQVGTEFTTILYNFMCNSSCVGGMNRRPILIIITLEMRDGQVLGRRSFEGRICACPGRDRKADEDHYRE 4gv1 A 1.49 BS01 0XZ A 1 K158 G162 V164 A177 K179 M227 Y229 A230 E234 E278 M281 D292 F438 K16 G20 V22 A35 K37 M85 Y87 A88 E92 E136 M139 D150 F296 D274 K276 N279 D292 T312 D132 K134 N137 D150 T170 2.7.11.1 0004672,0004674,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=4.2nM P31749 23394218 501 SRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITITPSMECVDSERRPHFPQFDYSAS 4gv8 A 2.1 BS01 DUP A 1 G78 I80 D81 Y84 G89 G76 I78 D79 Y82 G87 A25 R64 G66 L73 D81 A23 R62 G64 L71 D79 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 Kd=0.32uM remove_due_to_license_issue Q8SDV3 24311572 201 NTLQVRLLSENARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNDAIASNGYITPGVFDIKGEIDLSDAIRQYGTYQINEGDKLAQLVIVPIWTPELKQVEEFES 4gv8 A 2.1 BS02 DUP B 1 R64 S65 G66 R62 S63 G64 A25 R64 G66 L73 D81 A23 R62 G64 L71 D79 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 Kd=0.32uM remove_due_to_license_issue Q8SDV3 24311572 201 NTLQVRLLSENARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNDAIASNGYITPGVFDIKGEIDLSDAIRQYGTYQINEGDKLAQLVIVPIWTPELKQVEEFES 4gv8 B 2.1 BS01 DUP B 1 G78 I80 D81 Y84 G89 G76 I78 D79 Y82 G87 A25 R64 G66 L73 D81 A23 R62 G64 L71 D79 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 Kd=0.32uM remove_due_to_license_issue Q8SDV3 24311572 201 NTLQVRLLSENARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNDAIASNGYITPGVFDIKGEIDLSDAIRQYGTYQINEGDKLAQLVIVPIWTPELKQVEEFESF 4gv8 B 2.1 BS02 DUP C 1 N20 R64 S65 G66 N18 R62 S63 G64 A25 R64 G66 L73 D81 A23 R62 G64 L71 D79 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 Kd=0.32uM remove_due_to_license_issue Q8SDV3 24311572 201 NTLQVRLLSENARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNDAIASNGYITPGVFDIKGEIDLSDAIRQYGTYQINEGDKLAQLVIVPIWTPELKQVEEFESF 4gv8 C 2.1 BS01 DUP A 1 R64 S65 G66 R63 S64 G65 A25 R64 G66 L73 D81 A24 R63 G65 L72 D80 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 Kd=0.32uM remove_due_to_license_issue Q8SDV3 24311572 201 TNTLQVRLLSENARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNDAIASNGYITPGVFDIKGEIDLSDAIRQYGTYQINEGDKLAQLVIVPIWTPELKQVEEFEF 4gv8 C 2.1 BS02 DUP C 1 G78 I80 D81 Y84 G89 G77 I79 D80 Y83 G88 A25 R64 G66 L73 D81 A24 R63 G65 L72 D80 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 Kd=0.32uM remove_due_to_license_issue Q8SDV3 24311572 201 TNTLQVRLLSENARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNDAIASNGYITPGVFDIKGEIDLSDAIRQYGTYQINEGDKLAQLVIVPIWTPELKQVEEFEF 4gvm A 2.16 BS01 LF2 A 1 Q95 T124 T125 T128 W132 Q41 T70 T71 T74 W78 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=1.49uM remove_due_to_license_issue IC50=1.7e+2nM P12497 23615903 303 DCSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKTACWWAGIKQEFGIPYNPESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGGGYSAGERIVDIIATDIQ 4gw6 A 2.65 BS01 LF2 A 1 Q95 A128 W132 Q41 A74 W78 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue IC50=1.7e+2nM P12497 23615903 303 DCSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGIPESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGGYSAGERIVDIIATDIQ 4gw8 A 2.0 BS02 3RA A 1 L44 F49 A65 L120 R122 P123 V126 L174 I185 D186 L12 F17 A33 L88 R90 P91 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.88uM remove_due_to_license_issue P11309 22998443 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4gxs B 1.9634 BS01 0YS B 1 Y61 G62 L90 T91 R96 G141 S142 E145 E193 Y58 G59 L87 T88 R93 G138 S139 E142 E190 ? 0015276,0016020 remove_due_to_license_issue P19491 23076153 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4gxs D 1.9634 BS01 0YS D 1 K60 Y61 G62 L90 T91 R96 S140 G141 S142 E145 E193 K57 Y58 G59 L87 T88 R93 S137 G138 S139 E142 E190 ? 0015276,0016020 remove_due_to_license_issue P19491 23076153 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4gz3 A 1.9 BS02 UDP A 1 Q839 K842 L866 V895 A896 K898 H901 H920 T921 T922 D925 Q506 K509 L533 V562 A563 K565 H568 H587 T588 T589 D592 2.4.1.255 0006493,0016757 remove_due_to_license_issue IC50=1800nM O15294 23103939 1101 PTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKHIYDNRIVLNGIDLKAFLDSLPDVKIVKNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 4gzn C 0.99 BS01 dna A 0 S156 R157 R159 R160 D179 Q180 S181 S21 R22 R24 R25 D44 Q45 S46 ? remove_due_to_license_issue Q8C6P8 23059534 1 ~ 11 SERPFFCNFCGKTYRDASGLSRHRRAHLGYRPRSCPECGKCFRDQSEVNRHLKVHQNKP 4gzn C 0.99 BS02 dna B 0 R138 Y149 R150 S153 R166 K175 R178 E182 R185 H186 V189 R3 Y14 R15 S18 R31 K40 R43 E47 R50 H51 V54 ? remove_due_to_license_issue Q8C6P8 23059534 1 ~ 11 SERPFFCNFCGKTYRDASGLSRHRRAHLGYRPRSCPECGKCFRDQSEVNRHLKVHQNKP 4gzp A 2.3 BS02 G39 A 1 R118 E119 D151 R152 E276 R292 R371 Y406 R37 E38 D70 R71 E195 R211 R290 Y325 D151 E277 R292 R371 Y406 D70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 Ki=14.3nM remove_due_to_license_issue K7N5N3 23015718 512 AEYRNWSKPQCDITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPDKCYQFALGQGTTLNNVHSNNTVRDRTPYRTLLMNELGVPFHLGTKQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYNGRLVDSVVSWSKEILRTQESECVCINGTCTVVMTDGSASGKADTKILFIEEGKIVHTSTLSGSAQHVEECSCYPRYPGVRCVCRDNWKGSNRPIVDINIKDHSIVSSYVCSGLVGDTPRKNDSSSSSHCLDPNNEEGGHGVKGWAFDDGNDVWMGRTINETSRLGYETFKVIEGWSNPKSKLQINRQVIVDRGNRSGYSGIFSVEGKSCINRCFYVELIRGRKEETEVLWTSNSIVVFCGTSGTYGTGSWPDGADLNLMPI 4gzt A 2.19 BS02 G39 A 1 R118 E119 R152 R224 E276 R292 R371 Y406 R37 E38 R71 R143 E195 R211 R290 Y325 G151 E277 R292 R371 Y406 G70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 Ki=17nM remove_due_to_license_issue K7N5N3 23015718 501 AEYRNWSKPQCDITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPDKCYQFALGQGTTLNNVHSNNTVRGRTPYRTLLMNELGVPFHLGTKQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYNGRLVDSVVSWSKEILRTQESECVCINGTCTVVMTDGSASGKADTKILFIEEGKIVHTSTLSGSAQHVEECSCYPRYPGVRCVCRDNWKGSNRPIVDINIKDHSIVSSYVCSGLVGDTPRKNDSSSSSHCLDPNNEEGGHGVKGWAFDDGNDVWMGRTINETSRLGYETFKVIEGWSNPKSKLQINRQVIVDRGNRSGYSGIFSVEGKSCINRCFYVELIRGRKEETEVLWTSNSIVVFCGTSGTYGTGSWPDGADLNLMPI 4gzw A 2.45 BS01 SIA E 1 R118 E119 R224 E276 R292 R371 Y406 R37 E38 R143 E195 R211 R290 Y325 G151 E277 R292 R371 Y406 G70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 remove_due_to_license_issue K7N5N3 23015718 3 AEYRNWSKPQCDITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPDKCYQFALGQGTTLNNVHSNNTVRGRTPYRTLLMNELGVPFHLGTKQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYNGRLVDSVVSWSKEILRTQESECVCINGTCTVVMTDGSASGKADTKILFIEEGKIVHTSTLSGSAQHVEECSCYPRYPGVRCVCRDNWKGSNRPIVDINIKDHSIVSSYVCSGLVGDTPRKNDSSSSSHCLDPNNEEGGHGVKGWAFDDGNDVWMGRTINETSRLGYETFKVIEGWSNPKSKLQINRQVIVDRGNRSGYSGIFSVEGKSCINRCFYVELIRGRKEETEVLWTSNSIVVFCGTSGTYGTGSWPDGADLNLMPI 4gzx A 2.45 BS01 SIA E 1 R118 E119 R152 R224 E276 R292 R371 Y406 R37 E38 R71 R143 E195 R211 R290 Y325 G151 E277 R292 R371 Y406 G70 E196 R211 R290 Y325 3.2.1.18 0004308,0005975,0016020,0016798,0020002,0033644,0044423,0046761,0046872,0055036 remove_due_to_license_issue K7N5N3 23015718 2 AEYRNWSKPQCDITGFAPFSKDNSIRLSAGGDIWVTREPYVSCDPDKCYQFALGQGTTLNNVHSNNTVRGRTPYRTLLMNELGVPFHLGTKQVCIAWSSSSCHDGKAWLHVCITGDDKNATASFIYNGRLVDSVVSWSKEILRTQESECVCINGTCTVVMTDGSASGKADTKILFIEEGKIVHTSTLSGSAQHVEECSCYPRYPGVRCVCRDNWKGSNRPIVDINIKDHSIVSSYVCSGLVGDTPRKNDSSSSSHCLDPNNEEGGHGVKGWAFDDGNDVWMGRTINETSRLGYETFKVIEGWSNPKSKLQINRQVIVDRGNRSGYSGIFSVEGKSCINRCFYVELIRGRKEETEVLWTSNSIVVFCGTSGTYGTGSWPDGADLNLMPI 4h10 A 2.402 BS01 dna C 0 H77 S78 E81 R85 D110 K111 H9 S10 E13 R17 D42 K43 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue O00327 23229515 103 ~ 117 RIKNAREAHSQIEKRRRDKMNSFIDELASLVPTCNAMSRKLDKLTVLRMAVQHMKTLRGA 4h10 A 2.402 BS02 dna D 0 I80 E81 R84 I12 E13 R16 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue O00327 23229515 303 ~ 317 RIKNAREAHSQIEKRRRDKMNSFIDELASLVPTCNAMSRKLDKLTVLRMAVQHMKTLRGA 4h10 B 2.402 BS01 dna C 0 E43 R46 E13 R16 2.3.1.48 0000981,0032922,0046983 remove_due_to_license_issue O15516 23229515 103 ~ 117 KDKAKRVSRNKSEKKRRDQFNVLIKELGSMLPGNARKMDKSTVLQKSIDFLRKHKEITAWLEH 4h10 B 2.402 BS02 dna D 0 R39 N40 E43 R47 N51 D69 K70 R9 N10 E13 R17 N21 D39 K40 2.3.1.48 0000981,0032922,0046983 remove_due_to_license_issue O15516 23229515 303 ~ 317 KDKAKRVSRNKSEKKRRDQFNVLIKELGSMLPGNARKMDKSTVLQKSIDFLRKHKEITAWLEH 4h1e A 1.9 BS01 10J A 1 Q73 L91 D93 S96 V130 Y132 F169 W176 R189 D289 G291 Q16 L34 D36 S39 V73 Y75 F112 W119 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=3nM remove_due_to_license_issue P56817 22989333 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4h1j A 2.0 BS01 0YH A 1 K457 E474 M478 L504 Y505 L556 G566 D567 F568 R572 K39 E56 M60 L86 Y87 L138 G148 D149 F150 R154 D549 A551 R553 N554 D567 L587 D131 A133 R135 N136 D149 L160 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1200nM remove_due_to_license_issue IC50=1200nM Q14289 23153798 701 GIAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSRDEVTRLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA 4h1m A 1.99 BS01 0YJ A 1 G432 V439 K457 E474 M478 V487 M502 G566 D567 F568 G13 V20 K38 E55 M59 V68 M83 G147 D148 F149 D549 A551 R553 N554 D567 L587 D130 A132 R134 N135 D148 L153 2.7.10.2 0004672,0004713,0005524,0006468 ic50=78nM remove_due_to_license_issue IC50=78nM Q14289 23153798 701 IAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTLDNKEKFMSEAVIMKNLDHPHIVKLIGIIEEEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGLSLPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA 4h2j A 1.81 BS01 0YU A 1 K44 A47 V50 R51 V54 S55 F89 A92 L93 E96 S99 L100 H103 K32 A35 V38 R39 V42 S43 F66 A69 L70 E73 S76 L77 H80 D26 H43 L137 D14 H31 L114 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 301 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSELMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 4h2m A 1.78 BS01 0YV A 1 A47 V50 R51 V54 S55 A92 L93 E96 S99 L100 H103 A33 V36 R37 V40 S41 A66 L67 E70 S73 L74 H77 D26 H43 L137 D12 H29 L111 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 301 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSLMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 4h2o B 2.14 BS01 0YW B 1 S55 L93 E96 L100 H103 S42 L64 E67 L71 H74 D26 H43 L137 D13 H30 L108 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 301 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 4h2o B 2.14 BS02 0YW B 2 R51 F89 E96 N144 R38 F60 E67 N115 D26 H43 L137 D13 H30 L108 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 302 PAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 4h38 A 1.95 BS01 0YX A 1 A47 V50 R51 A92 L93 E96 S99 L100 A33 V36 R37 A66 L67 E70 S73 L74 D26 H43 L137 D12 H29 L111 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 301 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSLMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 4h3a A 1.98 BS01 0YY A 1 A47 V50 R51 E96 S99 L100 H103 A33 V36 R37 E65 S68 L69 H72 D26 H43 L137 D12 H29 L106 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 301 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFLFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 4h3c A 1.93 BS01 0YZ A 1 S55 A58 E96 H103 I141 S41 A44 E67 H74 I112 D26 H43 L137 D12 H29 L108 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 301 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 4h3c A 1.93 BS02 0YZ A 2 A47 Y68 V90 N144 A33 Y54 V61 N115 D26 H43 L137 D12 H29 L108 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 remove_due_to_license_issue P60472 23248302 302 AHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANR 4h3f A 1.7 BS01 10O A 1 S71 Q73 G74 D93 S96 N98 Y132 W137 I179 D289 G291 T292 T293 S14 Q16 G17 D36 S39 N41 Y75 W80 I122 D232 G234 T235 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=1nM remove_due_to_license_issue P56817 22989333 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4h3g A 1.85 BS01 10Q A 1 S71 Q73 G74 D93 S96 V130 Y132 W137 F169 I171 I179 R189 D289 G291 T292 T293 S14 Q16 G17 D36 S39 V73 Y75 W80 F112 I114 I122 R132 D232 G234 T235 T236 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=6nM remove_due_to_license_issue P56817 22989333 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4h3i A 1.96 BS01 10V A 1 Q73 L91 D93 S96 V130 F169 W176 D289 G291 Q16 L34 D36 S39 V73 F109 W116 D229 G231 D93 S96 N98 A100 D289 T292 D36 S39 N41 A43 D229 T232 3.4.23.46 0004190,0006508,0016020 Ki=3nM remove_due_to_license_issue P56817 22989333 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4h3j A 1.6 BS01 10W A 1 G72 Q73 G74 D93 S96 N98 V130 T133 Q134 I179 R189 D289 G291 G15 Q16 G17 D36 S39 N41 V73 T76 Q77 I122 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=90nM remove_due_to_license_issue P56817 22989333 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4h42 U 2.01 BS01 11E U 1 S190 Q192 G193 S195 W215 G219 C220 E244 S193 Q195 G196 S198 W218 G221 C222 E247 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE 4h4b A 2.9 BS01 11H A 1 N154 P293 F354 N152 P291 F352 2.7.1.77,3.1.3.5,3.1.3.99 0000255,0005515,0005524,0005737,0005829,0006204,0008253,0009117,0016740,0016787,0042802,0046037,0046040,0046054,0046085,0046872,0050146,0050483,0050484,0050689,0061630,0070936,0106411 remove_due_to_license_issue P49902 23220537 601 TSWSDRLQNAADMPANMDKHALKKYRREAYHRVFVNRSLAMEKIKCFGFDMDYTLAVYKSPEYESLGFELTVERLVSIGYPQELLSFAYDSTFPTRGLVFDTLYGNLLKVDAYGNLLVCAHGFNFIRGPETREQYPNKFIQRDDTERFYILNTLFNLPETYLLACLVDFFTNCPRYTSCETGFKDGDLFMSYRSMFQDVRDAVDWVHYKGSLKEKTVENLEKYVVKDGKLPLLLSRMKEVGKVFLATNSDYKYTDKIMTYLFDFPHGPKPGSSHRPWQSYFDLILVDARKPLFFGEGTVLRQVDTKTGKLKIGTYTGPLQHGIVYSGGSSDTICDLLGAKGKDILYIGDHIFGDILKSKKRQGWRTFLVIPELAQELHVWTDKSSLFEELQSLDIFLAIQRRIKKVTHDMDMCYGMMGSLFRSGSRQTLFASQVMRYADLYAASFINLLYYPFSYLFRAAHVLMPHES 4h4d A 1.35 BS02 10E A 1 V40 H41 A73 H74 H124 E126 S225 S226 N227 S269 V40 H41 A73 H74 H124 E126 S225 S226 N227 S269 1.17.7.4 0005829,0008299,0016114,0016491,0019288,0042380,0046872,0050992,0051538,0051539,0051745 ic50=0.15uM remove_due_to_license_issue P62623 23307751 402 MQILLANPRGFCAGVDRAISIVENALAIYGAPIYVRHEVVHNRYVVDSLRERGAIFIEQISEVPDGAILIFSAHGVSQAVRNEAKSRDLTVFDATCPLVTKVHMEVARASRRGEESILIGHAGHPEVEGTMGQYSNPEGGMYLVESPDDVWKLTVKNEEKLSFMTQTTLSVDDTSDVIDALRKRFPKIVGPRKDDICYATTNRQEAVRALAEQAEVVLVVGSKNSSNSNRLAELAQRMGKRAFLIDDAKDIQEEWVKEVKCVGVTAGASAPDILVQNVVARLQQLGGGEAIPLEGREENIVFEVPKELR 4h4e A 1.7 BS02 10G A 1 V40 H41 A73 H74 H124 S225 S226 N227 S269 V40 H41 A73 H74 H124 S225 S226 N227 S269 1.17.7.4 0005829,0008299,0016114,0016491,0019288,0042380,0046872,0050992,0051538,0051539,0051745 ic50=0.21uM remove_due_to_license_issue P62623 23307751 402 MQILLANPRGFCAGVDRAISIVENALAIYGAPIYVRHEVVHNRYVVDSLRERGAIFIEQISEVPDGAILIFSAHGVSQAVRNEAKSRDLTVFDATCPLVTKVHMEVARASRRGEESILIGHAGHPEVEGTMGQYSNPEGGMYLVESPDDVWKLTVKNEEKLSFMTQTTLSVDDTSDVIDALRKRFPKIVGPRKDDICYATTNRQEAVRALAEQAEVVLVVGSKNSSNSNRLAELAQRMGKRAFLIDDAKDIQEEWVKEVKCVGVTAGASAPDILVQNVVARLQQLGGGEAIPLEGREENIVFEVPKELR 4h4m A 2.85 BS01 494 A 1 P95 L100 K102 K103 V106 V108 Y181 Y188 W229 L234 P236 Y318 P95 L100 K102 K103 V106 V108 Y181 Y188 W229 L234 P236 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 23163887 601 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQV 4h58 A 3.1 BS01 10Z A 1 I462 V470 W530 C531 H538 F582 D593 I16 V24 W84 C85 H92 F136 D147 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 23398453 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP 4h5c F 2.02 BS01 YS4 F 1 F99 D103 R112 T167 E168 Q171 K200 D243 K257 F92 D96 R105 T160 E161 Q164 K193 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=28nM P14324 23234314 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4h5d F 2.02 BS01 YS4 F 1 F99 D103 R112 T167 E168 Q171 K200 D243 K257 F92 D96 R105 T160 E161 Q164 K193 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 Kd=0.58uM remove_due_to_license_issue IC50=28nM P14324 23234314 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4h5e F 2.04 BS02 IPR F 1 G56 K57 R60 Q96 R113 T201 F239 D243 G49 K50 R53 Q89 R106 T194 F232 D236 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 23234314 402 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4h71 A 1.93 BS01 PXE A 1 S412 L491 K492 A493 H538 K540 R557 S42 L121 K122 A123 H167 K169 R186 2.7.11.21 remove_due_to_license_issue P53350 23135290 702 DCHLSDMLQQLHSVNASKPSERGLVRQEEAEDPACIPIFWVSKWVDYSDKYGLGYQLCDNSVGVLFNDSTRLILYNDGDSLQYIERDGTESYLTVSSHPNSLMKKITLLKYFRNYMSEHLLKAGANITPREDELARLPYLRTWFRTRSAIILHLSNGSVQINFFQDHTKLILCPLMAAVTYIDEKRDFRTYRLSLLEEYGCCKELASRLRYARTMVDKLLSS 4h7q A 2.1 BS02 COI A 1 Y99 H132 R167 I170 R171 Y56 H89 R124 I127 R128 Y241 E245 K248 N249 Y198 E202 K205 N206 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 402 MMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYHFTTAGFGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHIDG 4h81 A 2.05 BS02 WJ2 A 1 I72 Y99 L128 H132 R167 I170 R171 I30 Y57 L86 H90 R125 I128 R129 Y241 E245 K248 N249 Y199 E203 K206 N207 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 404 TMMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYHFTTAGFGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHI 4h85 A 2.1 BS02 HRI A 1 I72 Y99 H132 R167 I170 R171 I29 Y56 H89 R124 I127 R128 Y241 E245 K248 N249 Y198 E202 K205 N206 2.7.11.1,2.7.11.4 0004672,0004674,0004722,0004740,0005524,0005739,0005759,0006550,0006552,0006574,0007283,0008610,0009083,0010510,0010906,0016301,0016310,0016772,0045252,0047323,0106310 remove_due_to_license_issue Q00972 23716694 404 MMLYSGRSQDGSHLLKSGRYLQQELPVRIAHRIKGFRSLPFIIGCNPTILHVHELYIRAFQKLTDFPPIKDQADEAQYCQLVRQLLDDHKDVVTLLAEGLRESRKHIEDEKLVRYFLDKTLTSRLGIRMLATHHLALHEDKPDFVGIICTRLSPKKIIEKWVDFARRLCEHKYGNAPRVRINGHVAARFPFIPMPLDYILPELLKNAMRATMESHLDTPYNVPDVVITIANNDVDLIIRISDRGGGIAHKDLDRVMDYHFTTAGFGFGLPTSRAYAEYLGGSLQLQSLQGIGTDVYLRLRHIDG 4ha5 A 1.83 BS01 13W A 1 Q73 D93 S96 Y132 W176 D289 G291 T292 Q16 D36 S39 Y75 W119 D232 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=56nM remove_due_to_license_issue P56817 22989333 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4hai A 2.55 BS02 I23 A 1 D335 W336 Y383 Q384 Y466 H524 D335 W336 Y383 Q384 Y466 H524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=7.9nM P34913 23237835 603 MTLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 4hbm A 1.9 BS01 0Y7 A 1 V14 T16 L54 G58 I61 V93 K94 H96 I99 Y100 V9 T11 L49 G53 I56 V88 K89 H91 I94 Y95 2.3.2.27 0005634,0043066,0051726 Kd=12nM remove_due_to_license_issue Q00987 22991965 201 MSVPTDGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 4hbn A 2.6 BS01 CMP A 1 V642 F658 G659 E660 I661 C662 R669 T670 R710 V123 F138 G139 E140 I141 C142 R149 T150 R190 ? remove_due_to_license_issue Q9Y3Q4 23103389 801 SDSSRRQYQEKYKQVEQYMSFHKLPPDTRQRIHDYYEHRYQGKMFDEESILGELSEPLREEIINFNCRKLVASMPLFANADPNFVTSMLTKLRFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTGNKETKLADGSYFGEICLLTRGRRTARVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVALDRLDRIGKKNS 4hbp A 2.91 BS01 17J A 1 S193 F194 I238 G239 S241 F381 M436 T488 S151 F152 I196 G197 S199 F339 M394 T446 K142 S217 S218 T236 I238 G239 G240 S241 F244 K100 S175 S176 T194 I196 G197 G198 S199 F202 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue IC50=8.7nM P97612 23218778 600 ARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMLSFDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSAGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNSMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAISYTVLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMT 4hbv A 1.63 BS01 15E A 1 W81 P82 F83 L92 I146 W40 P41 F42 L51 I105 ? ic50=23uM remove_due_to_license_issue IC50=23000nM O60885 23095041 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4hbw A 1.69 BS01 14Z A 1 W81 N140 I146 W40 N99 I105 ? ic50=4.8uM remove_due_to_license_issue IC50=1900nM O60885 23095041 202 SMNPPPPETSNPNKPKRETNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4hbx A 1.62 BS01 14X A 1 W81 L92 N140 I146 W40 L51 N99 I105 ? ic50=1.9uM remove_due_to_license_issue IC50=4800nM O60885 23095041 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4hby A 1.59 BS01 13F A 1 W81 L92 N140 W40 L51 N99 ? ic50=4.4uM remove_due_to_license_issue IC50=4400nM O60885 23095041 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4hco A 2.75 BS01 IMW A 1 A493 K540 R557 A121 K167 R184 2.7.11.21 remove_due_to_license_issue IC50=2180nM P53350 23135290 702 HLSDMLQQLHSVNASKPSERGLVRQEEAEDPACIPIFWVSKWVDYSDKYGLGYQLCDNSVGVLFNDSTRLILYNDGDSLQYIERDGTESYLTVSSHPNSLMKKITLLKYFRNYMSEHLLKAGANITPREGDLARLPYLRTWFRTRSAIILHLSNGSVQINFFQDHTKLILCPLMAAVTYIDEKRDFRTYRLSLLEEYGCCKELASRLRYARTMVDKLLSS 4hct A 1.48 BS01 18R A 1 I369 V377 A389 K391 M398 L433 F435 M438 G441 C442 D445 L489 D500 M503 V507 I16 V24 A36 K38 M45 L80 F82 M85 G88 C89 D92 L136 D147 M150 V154 D482 A484 R486 N487 D500 P521 D129 A131 R133 N134 D147 P168 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue IC50=10nM Q08881 23098091 701 GKWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4hcu A 1.43 BS01 13L A 1 I369 A389 K391 M398 F435 M438 G441 C442 D445 L489 D500 M503 I14 A34 K36 M43 F80 M83 G86 C87 D90 L134 D145 M148 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Q08881 23098091 701 WVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4hcv A 1.48 BS01 13J A 1 I369 F374 A389 K391 M398 F435 M438 C442 L489 D500 M503 I14 F19 A34 K36 M43 F80 M83 C87 L134 D145 M148 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Q08881 23098091 701 WVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4hdb A 1.49 BS01 G52 A 1 D25 G27 A28 N30 G48 P81 V82 I84 D25 G27 A28 N30 G48 P81 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8.9nM remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADNTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4hdb B 1.49 BS01 G52 A 1 D125 G127 D129 N130 G148 G149 I150 D25 G27 D29 N30 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADNTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4hdc A 2.05 BS01 13Y A 1 E37 R48 L52 F66 S69 R70 R92 S97 Y100 Q101 E36 R47 L51 F65 S68 R69 R91 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=1.2nM remove_due_to_license_issue P65249 23043329 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEKI 4hdf A 1.29 BS01 G52 A 1 R8 D25 G27 A28 D30 I84 R8 D25 G27 A28 D30 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.2nM remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 4hdf B 1.29 BS01 G52 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 4hdp A 1.22 BS01 G52 B 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4hdp B 1.22 BS01 G52 B 1 D25 G27 A28 D29 D30 G48 G49 V50 D25 G27 A28 D29 D30 G48 G49 V50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=30.9nM remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4hdu A 2.848 BS01 dna B 0 Y25 G26 R39 M45 K46 W56 N61 S62 S67 K68 R69 D70 Y25 G26 R39 M45 K46 W56 N61 S62 S67 K68 R69 D70 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 23112169 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4hdu A 2.848 BS02 dna C 0 M3 S36 Y37 Q40 M3 S36 Y37 Q40 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 23112169 14 ~ 26 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4hdv A 2.702 BS01 dna B 0 Y25 G26 A38 R39 M45 K46 W56 N61 S62 S67 R69 Y25 G26 A38 R39 M45 K46 W56 N61 S62 S67 R69 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 23112169 1 ~ 13 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4hdv A 2.702 BS02 dna C 0 M3 S36 Y37 R39 Q40 L94 M3 S36 Y37 R39 Q40 L94 ? 0003677,0003684,0003824,0003908,0005634,0005829,0006259,0006281,0006283,0032132,0070911 remove_due_to_license_issue Q9UTN9 23112169 14 ~ 26 MRMDEFYTKVYDAVCEIPYGKVSTYGEIARYVGMPSYARQVGQAMKHLHPETHVPWHRVINSRGTISKRDISAGEQRQKDRLEEEGVEIYQTSLGEYKLNLPEYMWKP 4he9 A 1.06 BS01 G52 A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.5nM remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4he9 B 1.06 BS01 G52 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23298236 401 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFMKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4heg A 1.46 BS01 G52 A 1 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.2nM remove_due_to_license_issue P03367 23298236 401 PQITLWKQPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4heg B 1.46 BS01 G52 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23298236 401 PQITLWKQPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4hej A 2.0 BS01 14D A 1 E37 R48 V51 L52 F66 S69 R70 R92 S96 S97 Y100 Q101 E36 R47 V50 L51 F65 S68 R69 R91 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=24000nM remove_due_to_license_issue P65249 23043329 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKNNRLDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLE 4heu A 2.0 BS02 15J A 1 Y514 L665 S667 T675 T678 A679 Y683 F686 P702 M703 E711 G715 Q716 F719 Y73 L224 S226 T234 T237 A238 Y242 F245 P261 M262 E270 G274 Q275 F278 3.1.4.17 0004114,0007165,0008081 ic50=0.097nM remove_due_to_license_issue IC50=0.097nM Q9Y233 23149228 1009 TSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4hev A 2.5 BS02 AXM A 1 F163 F194 E224 H227 E262 Y366 F163 F194 E218 H221 E242 Y346 H223 E224 H227 E262 R363 H217 E218 H221 E242 R343 3.4.24.69 0004222,0006508,0008270 Ki=460nM remove_due_to_license_issue P0DPI1 23340139 502 SSGLVPRGSHMQFVNKQFNYKDPVNGVDIAYIKIPQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEESLELGAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGTTASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLK 4hf1 A 2.222 BS01 dna C 0 R2 S5 K6 Y9 S38 S40 Y41 Q44 R59 G60 P61 R2 S5 K6 Y9 S38 S40 Y41 Q44 R59 G60 P61 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDESVDALTHALWRDLSDRLTGFLNNITLGELVNNQEVLDVSGRQHT 4hf1 A 2.222 BS02 dna D 0 P27 L28 E43 R50 S57 R59 G60 P61 Y65 P27 L28 E43 R50 S57 R59 G60 P61 Y65 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDESVDALTHALWRDLSDRLTGFLNNITLGELVNNQEVLDVSGRQHT 4hf1 B 2.222 BS01 dna C 0 P27 L28 E43 R50 S57 R59 P61 Y65 P27 L28 E43 R50 S57 R59 P61 Y65 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDAQGKGGAQGGDKALTHALWRDLSDRLTGFLNNITLGELVNNQEVL 4hf1 B 2.222 BS02 dna D 0 R2 S38 S40 Y41 Q44 R59 G60 P61 R2 S38 S40 Y41 Q44 R59 G60 P61 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLEQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDAQGKGGAQGGDKALTHALWRDLSDRLTGFLNNITLGELVNNQEVL 4hf2 A 2.99 BS01 dna C 0 R2 S5 K6 Y9 S38 S40 Y41 Q44 R59 P61 R2 S5 K6 Y9 S38 S40 Y41 Q44 R59 P61 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLAQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDESALTHALWRDLSDRLTGFLNNITLGELVNN 4hf2 A 2.99 BS02 dna D 0 P27 L28 R50 S57 P61 G62 G64 Y65 P27 L28 R50 S57 P61 G62 G64 Y65 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLAQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDESALTHALWRDLSDRLTGFLNNITLGELVNN 4hf2 B 2.99 BS01 dna C 0 P27 L28 R50 S57 P61 G63 G64 Y65 P27 L28 R50 S57 P61 G63 G64 Y65 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLAQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDGGDKALTHALWRDLSDRLTGFLNNITLGELVNNQEVL 4hf2 B 2.99 BS02 dna D 0 R2 S38 S40 Y41 Q44 R59 G60 P61 R2 S38 S40 Y41 Q44 R59 G60 P61 ? 0003677,0003690,0003700,0005506,0005829,0006355,0042802,0046872,0051537 remove_due_to_license_issue P0AGK8 23644595 1 ~ 29 MRLTSKGRYAVTAMLDVALNSEAGPVPLADISERQGISLSYLAQLFSRLRKNGLVSSVRGPGGGYLLGKDASSIAVGEVISAVDGGDKALTHALWRDLSDRLTGFLNNITLGELVNNQEVL 4hf4 A 2.0 BS02 15H A 1 Y514 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 Y73 I241 Y242 F245 P261 M262 E270 V271 G274 Q275 F278 3.1.4.17 0004114,0007165,0008081 ic50=2.4nM remove_due_to_license_issue IC50=2.4nM Q9Y233 23149228 1012 TSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4hfp B 2.4 BS02 15U B 1 H57 W60D D189 A190 E192 W215 G216 H43 W50 D199 A200 E202 W227 G228 H57 D102 E192 G193 D194 A195 G196 H43 D99 E202 G203 D204 A205 G206 3.4.21.5 0004252,0005509,0006508,0007596 Kd=42nM remove_due_to_license_issue P00734 23467412 402 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDAGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4hg7 A 1.6 BS01 NUT A 1 L54 G58 I61 M62 Q72 H73 V93 H96 Y100 L37 G41 I44 M45 Q55 H56 V76 H79 Y83 2.3.2.27 0005634,0043066,0051726 ic50=90nM remove_due_to_license_issue IC50=90nM, Ki=36nM, Kd=700nM Q00987 23897459 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDAAQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLV 4hge A 2.3 BS01 15V A 1 L855 G858 V863 A880 M929 Y931 L932 L983 D994 L13 G16 V21 A38 M83 Y85 L86 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 Ki=11.9nM remove_due_to_license_issue Ki=11.9nM O60674 23061660 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4hgl A 2.4 BS01 0YO A 1 G50 L57 K72 P100 E117 L118 L119 L169 I184 D185 P333 G18 L25 K40 P68 E85 L86 L87 L137 I152 D153 P301 D162 K164 T212 D130 K132 T180 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9Y6M4 24900428 401 GSGVLMVGPNFRVGKKIGCGNFGELRLGKNLYTNEYVAIKLEPMKSRAPQLHLEYRFYKQLGSGDGIPQVYYFGPCGKYNAMVLELLGPSLEDLFDLCDRTFSLKTVLMIAIQLISRMEYVHSKNLIYRDVKPENFLIGRPGNKTQQVIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGHMFMYFLRGSLPWQGLKADTLKERYQKIGDTKRATPIEVLCENFPEMATYLRYVRRLDFFEKPDYDYLRKLFTDLFDRKGYMFDYEYDWIGKQLPTPV 4hgs A 2.4 BS01 15G A 1 L57 A70 K72 P100 L116 L119 G120 P121 L169 I184 D185 P331 T332 P333 L25 A38 K40 P68 L84 L87 G88 P89 L137 I152 D153 P299 T300 P301 D162 K164 T212 D130 K132 T180 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9Y6M4 401 GSGVLMVGPNFRVGKKIGCGNFGELRLGKNLYTNEYVAIKLEPMKSRAPQLHLEYRFYKQLGSGDGIPQVYYFGPCGKYNAMVLELLGPSLEDLFDLCDRTFSLKTVLMIAIQLISRMEYVHSKNLIYRDVKPENFLIGRPGNKTQQVIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGHMFMYFLRGSLPWQGLKADTLKERYQKIGDTKRATPIEVLCENFPEMATYLRYVRRLDFFEKPDYDYLRKLFTDLFDRKGYMFDYEYDWIGKQLPTPV 4hgt A 1.8 BS01 15G A 1 I15 G18 I23 A36 K38 M82 L85 L135 I148 D149 I7 G10 I15 A28 K30 M71 L74 L124 I137 D138 D128 K130 D117 K119 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=40nM P48730 24900428 301 YRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 4hhy C 2.3637 BS01 15R C 1 L108 D109 V112 H201 G202 R217 A219 Y235 F236 S243 Y246 L103 D104 V107 H196 G197 R212 A214 Y230 F231 S238 Y241 S243 Y246 E327 S238 Y241 E322 2.4.2.-,2.4.2.30 0003950 ic50=1.92nM remove_due_to_license_issue IC50=1.9nM P09874 23473053 401 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 4hhz C 2.7199 BS01 15S C 1 Y49 L108 H201 G202 R217 I218 A219 P220 Y228 Y235 F236 S243 Y246 E327 Y49 L108 H201 G202 R217 I218 A219 P220 Y228 Y235 F236 S243 Y246 E327 S243 Y246 E327 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue P09874 23473053 401 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 4hid A 1.822 BS01 dna B 0 K25 T26 W27 Y28 F47 M49 S54 S55 R57 R68 W72 D73 E85 K97 H100 Y103 H109 K22 T23 W24 Y25 F44 M46 S51 S52 R54 R65 W69 D70 E82 K94 H97 Y100 H106 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 SFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4hik A 1.636 BS01 dna B 0 K25 W27 Y28 Y36 F47 M49 T53 S55 S56 R57 R68 I70 W72 D73 K97 D99 H100 L101 Y103 E105 H109 K22 W24 Y25 Y33 F44 M46 T50 S52 S53 R54 R65 I67 W69 D70 K94 D96 H97 L98 Y100 E102 H106 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 SFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4him A 1.75 BS01 dna B 0 K25 W27 Y28 Y36 F47 M49 S55 S56 R57 R68 I70 W72 D73 K97 D99 H100 Y103 E105 H109 K22 W24 Y25 Y33 F44 M46 S52 S53 R54 R65 I67 W69 D70 K94 D96 H97 Y100 E102 H106 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 SFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4hio A 1.753 BS01 dna B 0 K25 T26 W27 Y28 F47 M49 S54 S55 R57 R68 I70 W72 D73 E85 K97 D99 H100 E105 H109 K23 T24 W25 Y26 F45 M47 S52 S53 R55 R66 I68 W70 D71 E83 K95 D97 H98 E103 H107 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 DSFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4hiq A 1.18 BS01 16V A 1 K15 A108 A109 L110 S117 V121 K6 A99 A100 L101 S108 V112 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=6.2nM remove_due_to_license_issue Kd=4.8nM P02766 23716704 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVITNP 4hiq B 1.18 BS01 16V B 1 K15 L17 A108 L110 S117 V121 K6 L8 A99 L101 S108 V112 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=6.2nM remove_due_to_license_issue Kd=4.8nM P02766 23716704 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVITN 4his A 1.2 BS01 3MI A 1 K15 L17 L110 S117 T118 K5 L7 L100 S107 T108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=8.1nM remove_due_to_license_issue IC50=3100nM, Kd=274nM P02766 23716704 201 PLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVITNP 4hj2 A 2.1 BS01 LZ6 A 1 Y9 R45 Q54 V55 Q67 T68 L107 P110 M208 F220 Y6 R42 Q51 V52 Q64 T65 L104 P107 M205 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 remove_due_to_license_issue P08263 23460799 301 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIF 4hj2 A 2.1 BS02 LZ6 B 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 remove_due_to_license_issue P08263 23460799 301 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIF 4hj2 B 2.1 BS01 LZ6 A 1 D101 R131 D98 R124 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 remove_due_to_license_issue P08263 23460799 301 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIF 4hj2 B 2.1 BS02 LZ6 B 1 Y9 R45 Q54 V55 Q67 T68 L107 P110 M208 F220 Y6 R42 Q51 V52 Q64 T65 L104 P107 M201 F213 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 remove_due_to_license_issue P08263 23460799 301 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIF 4hj5 A 2.04 BS01 dna B 0 K25 W27 Y28 Y36 F47 M49 T53 S55 R57 R68 I70 W72 D73 H100 L101 E105 H109 K22 W24 Y25 Y33 F44 M46 T50 S52 R54 R65 I67 W69 D70 H97 L98 E102 H106 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 SFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4hj7 A 1.783 BS01 dna B 0 K25 W27 Y28 Y36 F47 M49 T53 S55 S56 R57 R68 I70 W72 D73 D99 H100 L101 Y103 E105 H109 K22 W24 Y25 Y33 F44 M46 T50 S52 S53 R54 R65 I67 W69 D70 D96 H97 L98 Y100 E102 H106 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 SFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4hj8 A 2.043 BS01 dna B 0 K25 W27 Y28 Y36 F47 M49 S54 S55 R57 R68 I70 W72 D73 K97 D99 H100 L101 E105 H109 K22 W24 Y25 Y33 F44 M46 S51 S52 R54 R65 I67 W69 D70 K94 D96 H97 L98 E102 H106 ? 0000723,0043047 remove_due_to_license_issue O13988 23201273 1 ~ 9 SFSLLSQITPHQRCSFYAQVIKTWYSDKNFTLYVTDYTENELFFPMSPYTSSSRWRGPFGRFSIRCILWDEHDFYCRNYIKEGDYVVMKNVRTKIDHLGYLECILHGDSAKRYNMSIEKVDSEEPELNEIKSRKRLYV 4hki A 2.15 BS02 FLN A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=140nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hkk A 1.95 BS02 AGI A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=2900nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4hkn A 2.05 BS02 LU2 A 1 H1031 G1032 Y1050 Y1060 Y1071 H80 G81 Y99 Y109 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=1100nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4hl5 A 2.2 BS02 15W A 1 H1031 G1032 F1035 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 F84 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=450nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hla A 1.95 BS01 017 A 1 D25 G27 D29 G48 G49 I50 I84 D25 G27 D29 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23877703 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4hla B 1.95 BS01 017 A 1 D25 A28 D30 G49 P81 V82 I84 D25 A28 D30 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 23877703 200 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4hlc A 1.55 BS01 T05 A 1 E37 R48 L52 F66 S69 R70 S96 S97 Y100 Q101 E36 R47 L51 F65 S68 R69 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=174nM remove_due_to_license_issue Q6GJI9 23206863 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKLDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLE 4hld A 2.0 BS01 16T A 1 E37 R48 L52 F66 S69 R70 R92 S96 S97 Y100 Q101 E36 R47 L51 F65 S68 R69 R91 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=0.5nM remove_due_to_license_issue Q6GJI9 23206863 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKNDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEK 4hlf A 2.15 BS02 15Z A 1 H1031 G1032 S1033 Y1050 Y1060 S1068 Y1071 H80 G81 S82 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=870nM Q9H2K2 23574272 1205 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hlg A 2.0 BS01 20B A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=310nM Q9H2K2 23574272 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hlh A 1.75 BS02 20D A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=1100nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hlk A 2.0 BS01 431 A 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 H80 G81 Y99 Y109 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=1100nM Q9H2K2 23574272 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hlm A 1.95 BS02 16S A 1 H1031 G1032 Y1050 Y1060 S1068 Y1071 H80 G81 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=170nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hlw A 2.5 BS02 17W A 1 F673 P723 N727 L830 E837 R840 F4 P54 N58 L161 E168 R171 ? remove_due_to_license_issue IC50=4200nM P10275 23301637 1002 QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIATSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 4hmh A 2.3 BS02 F94 A 1 H1031 G1032 S1033 Y1050 Y1060 S1068 Y1071 H80 G81 S82 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=620nM Q9H2K2 23574272 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4hmk A 3.0 BS01 LEU A 1 A22 G24 G26 Y108 F253 S256 F259 S355 I359 A19 G21 G23 Y105 F247 S250 F253 S349 I353 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 601 KREHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHES 4hmq A 2.1 BS01 FCE A 1 W63 N83 Y84 W158 M213 W223 Y225 R231 F255 W25 N45 Y46 W120 M175 W185 Y187 R193 F217 ? 0030288,0030313,1901678 remove_due_to_license_issue A0A0H2UPT5 23951167 401 KIVLDHAFGQTILDKKPERVATIAWGNHDVALALGIVPVGFSKANYGVSADKGVLPWTEEKIKELNGKANLFDDLDGLNFEAISNSKPDVILAGYSGITKEDYDTLSKIAPVAAYKSKPWQTLWRDMIKIDSKALGMEKEGDELIKNTEARISKELEKHPEIKGKIKGKKVLFTMINAADTSKFWIYTSKDPRANYLTDLGLVFPESLKEFESEDSFAKEISAEEANKINDADVIITYGDDKTLEALQKDPLLGKINAIKNGAVAVIPDNTPLAASCTPTPLSINYTIEEYLNLLGNACKNAK 4hn2 A 1.9 BS02 0EJ A 1 K53 K54 R213 K214 K248 R281 S326 K329 K12 K13 R172 K173 K207 R240 S285 K288 2.7.4.24 0000829 remove_due_to_license_issue O43314 23032903 402 RQIVVGICSMAKKSKSKPMKEILERISLFKYITVVVFEEEVILNEPVENWPLCDCLISFHSKGFPLDKAVAYAKLRNPFVINDLNMQYLIQDRREVYSILQAEGILLPRYAILNRDPNNPKECNLIEGEDHVEVNGEVFQKPFVEKPVSAEDHNVYIYYPTSAGGGSQRLFRKIGSRSSVYSPESNVRKTGSYIYEEFMPTDGTDVKVYTVGPDYAHAEARKSPALDGKVERDSEGKEVRYPVILNAREKLIAWKVCLAFKQTVCGFDLLRANGQSYVCDVNGFSFVKNSMKYYDDCAKILGNIVMRELAPQFHIPWSIPLEAED 4hn5 A 1.902 BS01 dna C 0 C431 H432 Y433 K442 K446 C13 H14 Y15 K24 K28 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 857 ~ 872 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn5 A 1.902 BS02 dna D 0 S440 V443 F444 R447 R470 K471 R477 S22 V25 F26 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 842 ~ 857 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn5 B 1.902 BS01 dna C 0 S440 R447 R470 K471 R477 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 857 ~ 872 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn5 B 1.902 BS02 dna D 0 C431 H432 Y433 K442 K446 C14 H15 Y16 K25 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 842 ~ 857 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn6 A 2.549 BS01 dna C 0 C431 H432 Y433 K442 K446 C13 H14 Y15 K24 K28 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 857 ~ 872 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGDNRCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn6 A 2.549 BS02 dna D 0 S440 V443 R447 R470 K471 R477 S22 V25 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 842 ~ 857 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGDNRCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn6 B 2.549 BS01 dna C 0 S440 R447 R470 K471 R477 S22 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 857 ~ 872 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGDNRCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hn6 B 2.549 BS02 dna D 0 C431 H432 Y433 K442 K446 C13 H14 Y15 K24 K28 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 23222642 842 ~ 857 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGDNRCIIDKIRRKNCPACRYRKCLQAGMNLEA 4hnc A 1.889 BS02 0UT A 1 K164 C166 D195 N197 E247 H297 E317 K162 C164 D193 N195 E245 H295 E315 V22 S139 K164 C166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 C164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=0.67mM remove_due_to_license_issue Ki=700000nM P11444 24472022 402 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFSLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTCIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGASRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 4hnc B 1.889 BS02 0UT B 1 K164 C166 D195 N197 E247 H297 E317 K156 C158 D187 N189 E239 H289 E309 V22 S139 K164 C166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S131 K156 C158 D187 N189 E213 G238 E239 D262 M286 H289 L290 F291 A305 E309 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 Ki=0.67mM remove_due_to_license_issue Ki=700000nM P11444 24472022 402 EVLITGLRTRAVNVPLAYPVHGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFSLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTCIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGASRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 4hnf A 2.07 BS01 16W A 1 G16 S17 A36 K38 E52 M80 M82 L85 G14 S15 A34 K36 E47 M75 M77 L80 D128 K130 D123 K125 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=711nM remove_due_to_license_issue IC50=711nM P48730 23106386 301 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 4hni A 2.74 BS01 16W A 1 I15 A36 K38 M80 M82 L84 L85 L135 F150 I13 A34 K36 M71 M73 L75 L76 L126 F141 D128 K130 D119 K121 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=32nM P49674 23106386 301 LRVGNKYRLGRKIGSGSFGDIYLGANIASGEEVAIKLECVHIESKFYKMMQGGVGIPSIKWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFSTYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4hnn A 2.4 BS01 LYS A 1 G73 M76 W78 H81 Y131 G53 M56 W58 H61 Y111 T69 Y132 Y156 R161 K184 I223 T49 Y112 Y136 R141 K164 I203 4.3.3.7 0008840,0009089,0016829 Kd=0.002mM remove_due_to_license_issue D7U7T8 23354837 401 SVDDIKSLRLITAIKTPYLPDGRFDLEAYDALVNMQIVDGAEGVIVGGTTGEGQLMSWDEHIMLIGHTVNCFGGSIKVIGNTGSNSTREAIHATEQGFAVGMHAALHINPYYGKTSLEGLVSHFESVLPMGPTVIYNVPSRTGQDIPPGVIHTVAQSANLAGVKECVGNDRIKQYTDNRIVVWSGNDDQCHDAKWDYGATGVISVTSNLIPGLMRQLLFKGKNPSLNAKIMPLVNWLFEEPNPIGLNTALAQLGVVRPVFRLPYVPLPLAKRVEFVNIVKEIGRENFVGEKDVKVLDDDDFILVGRY 4hnn A 2.4 BS02 LYS B 1 N105 E109 N85 E89 T69 Y132 Y156 R161 K184 I223 T49 Y112 Y136 R141 K164 I203 4.3.3.7 0008840,0009089,0016829 Kd=0.002mM remove_due_to_license_issue D7U7T8 23354837 401 SVDDIKSLRLITAIKTPYLPDGRFDLEAYDALVNMQIVDGAEGVIVGGTTGEGQLMSWDEHIMLIGHTVNCFGGSIKVIGNTGSNSTREAIHATEQGFAVGMHAALHINPYYGKTSLEGLVSHFESVLPMGPTVIYNVPSRTGQDIPPGVIHTVAQSANLAGVKECVGNDRIKQYTDNRIVVWSGNDDQCHDAKWDYGATGVISVTSNLIPGLMRQLLFKGKNPSLNAKIMPLVNWLFEEPNPIGLNTALAQLGVVRPVFRLPYVPLPLAKRVEFVNIVKEIGRENFVGEKDVKVLDDDDFILVGRY 4hnn B 2.4 BS01 LYS A 1 N105 E109 N85 E89 T69 Y132 Y156 R161 K184 I223 T49 Y112 Y136 R141 K164 I203 4.3.3.7 0008840,0009089,0016829 Kd=0.002mM remove_due_to_license_issue D7U7T8 23354837 401 SVDDIKSLRLITAIKTPYLPDGRFDLEAYDALVNMQIVDGAEGVIVGGTTGEGQLMSWDEHIMLIGHTVNCFGGSIKVIGNTGSNSTREAIHATEQGFAVGMHAALHINPYYGKTSLEGLVSHFESVLPMGPTVIYNVPSRTGQDIPPGVIHTVAQSANLAGVKECVGNDRIKQYTDNRIVVWSGNDDQCHDAKWDYGATGVISVTSNLIPGLMRQLLFKGKNPSLNAKIMPLVNWLFEEPNPIGLNTALAQLGVVRPVFRLPYVPLPLAKRVEFVNIVKEIGRENFVGEKDVKVLDDDDFILVGRY 4hnn B 2.4 BS02 LYS B 1 G73 M76 W78 H81 Y131 G53 M56 W58 H61 Y111 T69 Y132 Y156 R161 K184 I223 T49 Y112 Y136 R141 K164 I203 4.3.3.7 0008840,0009089,0016829 Kd=0.002mM remove_due_to_license_issue D7U7T8 23354837 401 SVDDIKSLRLITAIKTPYLPDGRFDLEAYDALVNMQIVDGAEGVIVGGTTGEGQLMSWDEHIMLIGHTVNCFGGSIKVIGNTGSNSTREAIHATEQGFAVGMHAALHINPYYGKTSLEGLVSHFESVLPMGPTVIYNVPSRTGQDIPPGVIHTVAQSANLAGVKECVGNDRIKQYTDNRIVVWSGNDDQCHDAKWDYGATGVISVTSNLIPGLMRQLLFKGKNPSLNAKIMPLVNWLFEEPNPIGLNTALAQLGVVRPVFRLPYVPLPLAKRVEFVNIVKEIGRENFVGEKDVKVLDDDDFILVGRY 4hnp H 2.8 BS01 ONK H 1 T1 S20 T21 G47 T48 A49 T1 S20 T21 G47 T48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 24930969 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4hod A 3.3 BS01 LEU A 1 A22 G24 G26 Y108 F253 T254 S256 F259 S355 I359 A18 G20 G22 Y104 F247 T248 S250 F253 S349 I353 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 601 REHWATRLGLILAMAGNAVGLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFTLSLGFGAIITYASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAIMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHESAGT 4hp0 A 1.19 BS01 NOJ A 1 E35 N46 D52 W108 E35 N46 D52 W108 E35 N46 D48 S50 D52 N59 E35 N46 D48 S50 D52 N59 3.2.1.17 0003796,0005515,0005576,0005615,0005737,0005783,0016231,0016798,0016998,0031640,0042742,0042802,0050829,0050830,0051672 remove_due_to_license_issue P00698 23303182 201 KVFGRCELAAAMKRHGLDNYRGYSLGNWVCAAKFESNFNTQATNRNTDGSTDYGILQINSRWWCNDGRTPGSRNLCNIPCSALLSSDITASVNCAKKIVSDGNGMNAWVAWRNRCKGTDVQAWIRGCR 4hp1 C 2.25 BS01 dna A 0 K61 R62 H90 Q91 R96 K97 R105 P108 M109 K3 R4 H32 Q33 R38 K39 R47 P50 M51 1.14.11.80 0003677,0008270 remove_due_to_license_issue A0JP82 23217707 1 ~ 12 NKKRKRCGVCVPCLRKEPCGACYNCVNRSTSHQICKMRKCEQLKKKRVVPM 4hp1 C 2.25 BS02 dna B 0 H90 Q91 H32 Q33 1.14.11.80 0003677,0008270 remove_due_to_license_issue A0JP82 23217707 1 ~ 12 NKKRKRCGVCVPCLRKEPCGACYNCVNRSTSHQICKMRKCEQLKKKRVVPM 4hp3 C 2.05 BS01 dna A 0 R62 H90 Q91 R96 K97 R105 M109 R4 H32 Q33 R38 K39 R47 M51 1.14.11.80 0003677,0008270 remove_due_to_license_issue A0JP82 23217707 1 ~ 12 NKKRKRCGVCVPCLRKEPCGACYNCVNRSTSHQICKMRKCEQLKKKRVVPM 4hp3 C 2.05 BS02 dna B 0 K61 K63 Y81 H90 Q91 K94 K3 K5 Y23 H32 Q33 K36 1.14.11.80 0003677,0008270 remove_due_to_license_issue A0JP82 23217707 1 ~ 12 NKKRKRCGVCVPCLRKEPCGACYNCVNRSTSHQICKMRKCEQLKKKRVVPM 4hpi A 1.19 BS01 NOJ A 1 E35 D52 E35 D52 E35 N46 D48 S50 D52 N59 E35 N46 D48 S50 D52 N59 3.2.1.17 0003796,0005515,0005576,0005615,0005737,0005783,0016231,0016798,0016998,0031640,0042742,0042802,0050829,0050830,0051672 remove_due_to_license_issue P00698 23303182 201 KVFGRCELAAAMKRHGLDNYRGYSLGNWVCAAKFESNFNTQATNRNTDGSTDYGILQINSRWWCNDGRTPGSRNLCNIPCSALLSSDITASVNCAKKIVSDGNGMNAWVAWRNRCKGTDVQAWIRGCR 4hqb A 2.301 BS01 dna M 0 R64 W66 L74 G79 A81 R83 R64 W66 L74 G79 A81 R83 ? remove_due_to_license_issue Q9RY80 23975200 1 ~ 4 MLQIEFITDLGARVTVNVEHESRLLDVQRHYGRLGWTSGEIPSGGYQFPIENEADFDWSLIGARKWKSPEGEELVIHRGHAYRRRELEAVDSRKLKLPAAIKYSRGAKVSDPQHVREKADGDIEYVSLAIFRGGKRQERYAVP 4hqb A 2.301 BS02 dna N 0 L95 L97 R132 G134 K135 L95 L97 R132 G134 K135 ? remove_due_to_license_issue Q9RY80 23975200 5 ~ 9 MLQIEFITDLGARVTVNVEHESRLLDVQRHYGRLGWTSGEIPSGGYQFPIENEADFDWSLIGARKWKSPEGEELVIHRGHAYRRRELEAVDSRKLKLPAAIKYSRGAKVSDPQHVREKADGDIEYVSLAIFRGGKRQERYAVP 4hqb B 2.301 BS01 dna N 0 R64 W66 G79 H80 A81 G106 R64 W66 G79 H80 A81 G98 ? remove_due_to_license_issue Q9RY80 23975200 5 ~ 9 MLQIEFITDLGARVTVNVEHESRLLDVQRHYGRLGWTSGEIPSGGYQFPIENEADFDWSLIGARKWKSPEGEELVIHRGHAYRRRELEAPAAIKYSRGAKVSDPQHVREKIEYVSLAIFRGGKRQERYAVP 4hqb E 2.301 BS01 dna M 0 G134 Q137 G118 Q121 ? remove_due_to_license_issue Q9RY80 23975200 1 ~ 4 TMLQIEFITDLGARVTVNVEHESRLLDVQRHYGRLGWTSGEIPSGGYQFPIENEADFDWSLIGARKWKSPEGEELVIHRGHAYRRRELEAVDSRKLKLPAAIKYSRGEYVSLAIFRGGKRQERYAVPG 4hqu A 2.2 BS01 dna C 0 E24 R27 N36 L38 V39 W40 P42 R73 K74 I75 I77 P82 I83 F84 K85 K86 E18 R21 N30 L32 V33 W34 P36 R67 K68 I69 I71 P76 I77 F78 K79 K80 ? 0008083,0016020 remove_due_to_license_issue P01127 23139410 1 IAEPAMIAECKTRTEVFEISRRLIDRTNANFLVWPPCVEVQRCSGCCNNRNVQCRPTQVQLRPVQVRKIEIVRKKPIFKKATVTLEDHLACKCET 4hqx A 2.3 BS01 dna C 0 R27 N36 L38 V39 W40 P42 R73 K74 I75 I77 P82 I83 F84 K85 K86 R21 N30 L32 V33 W34 P36 R67 K68 I69 I71 P76 I77 F78 K79 K80 ? 0008083,0016020 remove_due_to_license_issue P01127 23139410 1 IAEPAMIAECKTRTEVFEISRRLIDRTNANFLVWPPCVEVQRCSGCCNNRNVQCRPTQVQLRPVQVRKIEIVRKKPIFKKATVTLEDHLACKCET 4hra A 3.15 BS01 EP6 A 1 D161 G163 S164 V169 V185 E186 K187 G221 D222 F223 F239 N241 D150 G152 S153 V158 V174 E175 K176 G210 D211 F212 F228 N230 2.1.1.360 0031151,0051726 remove_due_to_license_issue Ki=0.080000nM, IC50=<0.100000nM Q8TEK3 23801631 501 KLELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPTSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVGKPVSYYLHTIDRTILENYFSSLKNPKL 4hrc H 2.8 BS01 OV2 H 1 T1 T21 G47 A49 G168 T1 T21 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 24930969 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4hrd H 2.8 BS01 OV1 H 1 T1 T21 G47 A49 G168 T1 T21 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 24930969 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4hrd I 2.8 BS01 OV1 H 1 D124 I126 D124 I126 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 24930969 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4hso A 2.1 BS01 TYR A 1 Q153 L177 L181 S182 Q148 L172 L176 S177 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Kd=22uM remove_due_to_license_issue Q9K169 23754471 401 PTDDIKIKEVKELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLGVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMARA 4hso B 2.1 BS01 TYR A 1 D8 D9 D1 D2 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Kd=22uM remove_due_to_license_issue Q9K169 23754471 401 DDIKIKEVKELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLGVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMARA 4hso B 2.1 BS02 TYR B 1 Q153 A156 L177 L181 S182 Q146 A149 L170 L174 S175 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Kd=22uM remove_due_to_license_issue Q9K169 23754471 401 DDIKIKEVKELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLGVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMARA 4ht0 A 1.6 BS02 V50 A 1 H94 H119 V121 F131 L198 T199 T200 P202 H91 H116 V118 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=10nM remove_due_to_license_issue Kd=10.0nM P00918 23394791 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ht2 B 1.45 BS02 V50 B 1 H91 S133 L197 T198 T199 P200 H89 S131 L195 T196 T197 P198 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=290nM remove_due_to_license_issue Kd=150nM O43570 23394791 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4ht4 A 2.907 BS01 dna B 0 A2 M3 H5 N8 F10 S12 R78 K79 N80 S81 Q82 R85 L91 N93 E128 N129 P130 R139 K150 R151 G153 N154 Y156 T162 K163 H166 N167 R170 A1 M2 H4 N7 F9 S11 R77 K78 N79 S80 Q81 R84 L90 N92 E127 N128 P129 R138 K149 R150 G152 N153 Y155 T161 K162 H165 N166 R169 ? remove_due_to_license_issue Q53632 23359708 2 ~ 29 AMYHFQNKFVSKANGQSATAKSAFNSASRIKDFKENEFKDYSNKQCDYSEILLPNNADDKFKDREYLWNKVHDVENRKNSQVAREIIIGLPNEFDPNSNIELAKEFAESLSNEGMIVDLNIHKINEENPHAHLLCTLRGLDKNNEFEPKRKGNDYIRDWNTKEKHNEWRKRWENVQNKHLEKNGFSVRVSADSY 4ht8 A 1.9 BS01 rna I 0 Y25 L26 G29 I30 K31 L32 Q33 Q52 S60 T61 Y21 L22 G25 I26 K27 L28 Q29 Q48 S56 T57 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 B 1.9 BS01 rna I 0 L26 N28 I30 L21 N23 I25 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 B 1.9 BS02 rna K 0 Y25 G29 T61 Y20 G24 T56 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 C 1.9 BS01 rna K 0 Y25 G29 I30 K31 L32 Q33 Q52 T61 Y20 G24 I25 K26 L27 Q28 Q47 T56 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 D 1.9 BS01 rna K 0 Y25 G29 I30 K31 L32 Q33 Q52 S60 T61 Y21 G25 I26 K27 L28 Q29 Q48 S56 T57 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 QSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 E 1.9 BS01 rna I 0 Y25 G29 T61 Y20 G24 T56 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 E 1.9 BS02 rna K 0 L26 I30 L21 I25 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht8 F 1.9 BS01 rna I 0 Y25 G29 I30 K31 L32 Q33 N48 Q52 T61 Y20 G24 I25 K26 L27 Q28 N43 Q47 T56 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht9 A 1.8 BS01 rna D 0 Y25 G29 I30 K31 L32 Q33 N48 Q52 T61 Y20 G24 I25 K26 L27 Q28 N43 Q47 T56 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht9 A 1.8 BS02 rna E 0 Q8 Q41 F42 H57 Q3 Q36 F37 H52 0003723,0006355 remove_due_to_license_issue 23605038 4 ~ 5 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht9 B 1.8 BS01 rna D 0 Y25 G29 I30 K31 L32 Q33 Q52 S60 T61 Y22 G26 I27 K28 L29 Q30 Q49 S57 T58 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 GQSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht9 B 1.8 BS02 rna E 0 F42 H57 F39 H54 0003723,0006355 remove_due_to_license_issue 23605038 4 ~ 5 GQSLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht9 C 1.8 BS01 rna D 0 Y25 G29 T61 Y20 G24 T56 0003723,0006355 remove_due_to_license_issue 23605038 1 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4ht9 C 1.8 BS02 rna E 0 Q8 Q41 F42 H57 Q3 Q36 F37 H52 0003723,0006355 remove_due_to_license_issue 23605038 4 ~ 5 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4htx A 1.9 BS02 19F A 1 Y655 L770 H773 L809 I826 F830 M847 L858 Q859 F862 I866 Y77 L192 H195 L231 I248 F252 M269 L280 Q281 F284 I288 3.1.4.17 0004114,0007165,0008081 ic50=4.7nM remove_due_to_license_issue IC50=4.7nM O00408 23899287 1003 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 4hu1 B 1.95 BS02 V13 B 1 Q94 H96 H121 V123 F133 L200 T201 V202 Q91 H93 H118 V120 F130 L197 T198 V199 H66 H96 H98 E108 H121 T201 H63 H93 H95 E105 H118 T198 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=29nM remove_due_to_license_issue Kd=29nM Q8N1Q1 23394791 302 RLSWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 4huo X 1.52 BS01 RS8 X 1 Y80 V81 G121 N122 Y123 I172 R180 N209 W211 Y76 V77 G117 N118 Y119 I168 R176 N205 W207 V81 V77 3.2.2.22 0017148,0030598 ic50=20uM remove_due_to_license_issue P02879 23214944 301 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 4hup X 1.699 BS01 19M X 1 Y80 V81 G121 N122 Y123 I172 S176 R180 N209 W211 Y76 V77 G117 N118 Y119 I168 S172 R176 N205 W207 V81 V77 3.2.2.22 0017148,0030598 ic50=15uM remove_due_to_license_issue P02879 23214944 301 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 4hv3 A 1.54 BS01 19L A 1 Y80 V81 G121 N122 Y123 I172 S176 R180 W211 R258 Y81 V82 G122 N123 Y124 I173 S177 R181 W212 R259 V81 E177 R180 V82 E178 R181 3.2.2.22 0017148,0030598 ic50=115uM remove_due_to_license_issue P02879 23214944 301 MIFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 4hv7 X 1.869 BS01 19J X 1 Y80 V81 G121 Y123 I172 S176 R180 Y76 V77 G117 Y119 I168 S172 R176 V81 V77 3.2.2.22 0017148,0030598 ic50=300uM remove_due_to_license_issue P02879 23214944 301 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 4hva A 2.074 BS02 4HV A 1 L61 P62 H121 H168 C264 L31 P32 H91 H138 C211 P62 E63 H121 G122 C163 R164 P32 E33 H91 G92 C133 R134 3.4.22.59 0004197,0006508,0008234 Kd=1.3uM remove_due_to_license_issue P55212 23227217 401 FDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQACRGNQHDVPVIPYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4hvb A 2.35 BS01 19P A 1 W812 I831 K833 Y867 I879 M953 I963 D964 W562 I581 K583 Y617 I629 M703 I713 D714 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=0.111000nM P48736 24900568 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNYVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 4hvd A 1.85 BS02 933 A 1 L828 V836 A853 Y904 L905 G908 L956 L14 V22 A39 Y84 L85 G88 L136 D949 A951 R953 N954 D967 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.4nM remove_due_to_license_issue IC50=1.4nM P52333 23214979 1202 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSG 4hvg A 2.75 BS01 19Q A 1 L828 V836 A853 Y904 L905 G908 L956 D967 L15 V23 A40 Y87 L88 G91 L139 D150 D949 A951 R953 N954 D967 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=17nM P52333 23214979 1201 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 4hvh A 2.3 BS01 19R A 1 L828 V836 A853 Y904 L905 G908 L956 L15 V23 A40 Y85 L86 G89 L137 D949 A951 R953 N954 D967 D130 A132 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 ic50=19nM remove_due_to_license_issue IC50=19nM P52333 23214979 1201 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGS 4hvi A 2.4 BS01 19S A 1 L828 G829 V836 A853 K855 M902 E903 Y904 L905 L956 L14 G15 V22 A39 K41 M80 E81 Y82 L83 L134 D949 A951 R953 N954 D967 D127 A129 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 ic50=68.9nM remove_due_to_license_issue IC50=69nM P52333 23214979 1201 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSG 4hvs A 1.9 BS01 647 A 1 W557 L595 V603 A621 K623 E640 I653 E671 Y672 C673 L799 I808 C809 D810 F811 W10 L48 V56 A74 K76 E93 I106 E124 Y125 C126 L194 I203 C204 D205 F206 D792 A794 R796 N797 D810 D187 A189 R191 N192 D205 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=0.016uM remove_due_to_license_issue IC50=16nM P10721 23493555 1001 HHMPMYEVQWKVVEESNGNNYSYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAQGLIKSDAAMTVAVKMLKPSAHSTEREALMSELKVLSYLGNHENIVNLLGACTHGGPTLVITEYCCYGDLLNFLRRKRDSFHSSDTSPASMEDDENALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVDKGNARLPVKWMAPESIFNSVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMSSPEHAPAEMYDIMKTCWDADPDKRPTFKQIVQDIEKQISES 4hw2 A 2.8 BS01 19H A 1 A227 F228 M231 M250 V253 F254 R263 L267 F270 I294 A55 F56 M59 M78 V81 F82 R91 L95 F98 I122 ? 0042981 remove_due_to_license_issue Ki=55nM Q07820 23244564 401 GDELYRQSLEIISRYLREQATGAKDTKPMSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4hw3 A 2.4 BS01 19G A 1 F228 M250 V253 R263 T266 L267 F270 F58 M80 V83 R93 T96 L97 F100 ? 0042981 Ki=0.32uM remove_due_to_license_issue IC50=400nM, Ki=320nM Q07820 23244564 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 4hw7 A 2.9001 BS01 64M A 1 L588 A614 E664 Y665 C666 L785 G795 D796 F797 L23 A49 E99 Y100 C101 L160 G170 D171 F172 D778 R782 N783 D796 D153 R157 N158 D171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue IC50=62nM P07333 23493555 1001 PTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCTYGDLLNFLRRKAEAMLGPSGRPLELRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGNARLPVKWMAPESIFDSVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQITSFLQEQA 4hwo A 1.907 BS02 409 A 1 R363 E365 M374 R375 V376 F379 Q381 D383 H385 Y462 K465 Q479 T482 Q484 H511 G516 S517 R520 R122 E124 M133 R134 V135 F138 Q140 D142 H144 Y221 K224 Q238 T241 Q243 H270 G275 S276 R279 C334 R363 Q381 D383 H385 K465 H511 C93 R122 Q140 D142 H144 K224 H270 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 Ki=2.9nM remove_due_to_license_issue P0A8M3 23362938 702 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEELEHHHHHH 4hwp A 1.807 BS02 X16 A 1 R363 E365 R375 V376 F379 Q381 D383 H385 Y462 K465 Q479 Q484 H511 G516 S517 R520 R122 E124 R134 V135 F138 Q140 D142 H144 Y221 K224 Q238 Q243 H270 G275 S276 R279 C334 R363 Q381 D383 H385 K465 H511 C93 R122 Q140 D142 H144 K224 H270 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 Ki=17.2nM remove_due_to_license_issue P0A8M3 23362938 702 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEELEHHHHHH 4hwr A 1.9 BS02 1B2 A 1 M332 R363 V376 F379 Q381 D383 H385 Y462 Q484 H511 M92 R123 V136 F139 Q141 D143 H145 Y222 Q244 H271 C334 R363 Q381 D383 H385 K465 H511 C94 R123 Q141 D143 H145 K225 H271 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 Ki=182nM remove_due_to_license_issue P0A8M3 23362938 702 ARDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEEL 4hws A 1.7 BS02 1B3 A 1 R363 E365 L373 M374 R375 V376 F379 Q381 D383 H385 Y462 K465 Q479 T482 Q484 H511 G516 S517 R520 R122 E124 L132 M133 R134 V135 F138 Q140 D142 H144 Y221 K224 Q238 T241 Q243 H270 G275 S276 R279 C334 R363 Q381 D383 H385 K465 H511 C93 R122 Q140 D142 H144 K224 H270 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 Ki=0.8nM remove_due_to_license_issue P0A8M3 23362938 702 RDHRKIGKQLDLYHMQEEAPGMVFWHNDGWTIFRELEVFVRSKLKEYQYQEVKGPFMMDRVLWEKTGHWDNYKDAMFTTSSENREYCIKPMNCPGHVQIFNQGLKSYRDLPLRMAEFGSCHRNEPSGSLHGLMRVRGFTQDDAHIFCTEEQIRDEVNGCIRLVYDMYSTFGFEKIVVKLSTRPEKRIGSDEMWDRAEADLAVALEENNIPFEYQLGEGAFYGPKIEFTLYDCLDRAWQCGTVQLDFSLPSRLSASYVGEDNERKVPVMIHRAILGSMERFIGILTEEFAGFFPTWLAPVQVVIMNITDSQSEYVNELTQKLSNAGIRVKADLRNEKIGFKIREHTLRRVPYMLVCGDKEVESGKVAVRTRRGKDLGSMDVNEVIEKLQQEIRSRSLKQLEELEHHHHHH 4hwt A 2.3 BS02 1B2 A 1 M444 C446 R475 Q493 D495 H497 Y573 D578 I579 Q590 C591 A592 Q595 H623 M91 C93 R122 Q140 D142 H144 Y220 D225 I226 Q237 C238 A239 Q242 H266 C446 R475 Q493 D495 H497 K576 H623 C93 R122 Q140 D142 H144 K223 H266 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 Ki>50000nM remove_due_to_license_issue P26639 23362938 802 RDHRKIGRDQELYFFHELSPGSCFFLPKGAYIYNALIEFIRSEYRKRGFQEVVTPNIFNSRLWMTSGHWQHYSENMFSFEVEKELFALKPMNCPGHCLMFDHRPRSWRELPLRLADFGVLHRNELSGALTGLTRVRRFQQDDAHIFCAMEQIEDEIKGCLDFLRTVYSVFGFSFKLNLSTRPEKFLGDIEVWDQAEKQLENSLNEFGEKWELNSGDGAFYGPKIDIQIKDAIGRYHQCATIQLDFQLPIRFNLTYVSDKKRPVIVHRAILGSVERMIAILTENYGGKWPFWLSPRQVMVVPVGPTCDEYAQKVRQQFHDAKFMADIDLDPGCTLNKKIRNAQLAQYNFILVVGEKEKISGTVNIRTRDNKVHGERTISETIERLQQLKEFRSKQA 4hww A 1.298 BS01 X7A A 1 H101 D124 H126 D128 S137 H141 G142 D183 D232 H97 D120 H122 D124 S133 H137 G138 D179 D228 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 ic50=223nM remove_due_to_license_issue P05089 23472952 901 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 4hww B 1.298 BS01 X7A B 1 D124 H126 D128 S137 H141 G142 D183 D232 D120 H122 D124 S133 H137 G138 D179 D228 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 ic50=223nM remove_due_to_license_issue P05089 23472952 401 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 4hxl A 1.52 BS01 1A9 A 1 W81 P82 Q85 L92 I146 W39 P40 Q43 L50 I104 ? ic50=2.2uM remove_due_to_license_issue IC50=2200nM O60885 23530754 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 4hxm A 1.5 BS01 1A8 A 1 W81 P82 Q85 L92 I146 W39 P40 Q43 L50 I104 ? ic50=0.79uM remove_due_to_license_issue IC50=790nM O60885 23530754 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4hxq A 1.45 BS01 X8A A 1 D124 H126 D128 S137 H141 G142 D183 D232 D120 H122 D124 S133 H137 G138 D179 D228 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 ic50=60nM remove_due_to_license_issue P05089 23472952 901 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 4hxq B 1.45 BS01 X8A B 1 D124 H126 D128 S137 H141 D183 D232 D120 H122 D124 S133 H137 D179 D228 H101 D124 H126 D128 H141 D232 D234 E277 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 ic50=60nM remove_due_to_license_issue P05089 23472952 401 SRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYL 4hxr A 1.53 BS01 1A4 A 1 P82 V87 L92 I146 P40 V45 L50 I104 ? ic50=4.1uM remove_due_to_license_issue IC50=4100nM O60885 23530754 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 4hxs A 1.43 BS01 1A3 A 1 W81 P82 Q85 L92 I146 W39 P40 Q43 L50 I104 ? ic50=4.1uM remove_due_to_license_issue IC50=4100nM O60885 23530754 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4hxw A 1.69 BS01 1A0 A 1 N55 S56 E59 D82 R85 G86 I87 P88 T174 N31 S32 E35 D58 R61 G62 I63 P64 T131 5.6.2.2 0003677,0003918,0005524,0006265 Ki=2nM remove_due_to_license_issue Q839Z1 23352267 301 GLEAVRKRPGMYIGSTSGEGLHHLVWEIVDNSIDEALAGFAKSIQVIIEPDDSITVIDDGRGIPVGIQAKTGRPAVETVFTVLVGSSVVNALSTSLDVRVYKDGKVYYQEYRRGAVVDDLKVIEETDRHGTTVHFIPDPEIFTETTVYDFDKLATRVRELAFLNRGLHISIEDRREGQEDKKEYHYEGLEH 4hxz A 2.7 BS01 19Y A 1 I38 N41 S42 E45 D68 G72 M73 V115 T162 I164 I31 N34 S35 E38 D61 G65 M66 V98 T145 I147 5.6.2.2 0003677,0003918,0005524,0005694,0006265 remove_due_to_license_issue A0A0J9WZF0 23352267 1401 SIEVLTGLDPVKKRPGMYTNIENPNHLIQEIIDNSVDEVLAGFASKINITLYEDNSIEVADDGRGMPVDIHPEHKMSGIELIMTKLHSGGKFSHGVGVSVVNALSTRLEAEIKRDGNVYHIVFEDGFKTKDLEIIDNVGKKNTGTKIRFWPNKKYFDDIKVNFKALKNLLEAKAILCKALTIKYSNEIKKEKLTWHFETGLKGYLDHKLEAETLPAEPFIIDNFSNGDSYLDAVFCWCEDPSESIKNSYVNLIPTPQDGTHVTGLKNGIYDAIKAYIEKNSLSVKNIKITANDSFAQLNYVISVKITNPQFAGQTKEKLSNKDVTNFVATAVKDLLTIWLNQNPDEARQIVENISKVAQKRINADL 4hy0 A 2.84 BS03 1AQ A 1 K297 G306 L307 T308 D309 K311 E314 Q319 W323 K44 G53 L54 T55 D56 K58 E61 Q66 W70 2.3.2.27 remove_due_to_license_issue IC50=200nM P98170 23298277 403 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLE 4hy0 A 2.84 BS04 1AQ F 1 T345 L348 T92 L95 2.3.2.27 remove_due_to_license_issue IC50=200nM P98170 23298277 403 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLE 4hy0 B 2.84 BS02 1AQ B 1 K297 K299 G306 L307 T308 D309 W310 E314 Q319 W323 K44 K46 G53 L54 T55 D56 W57 E61 Q66 W70 2.3.2.27 remove_due_to_license_issue IC50=200nM P98170 23298277 403 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLE 4hy0 B 2.84 BS03 1AQ E 1 T345 L348 T92 L95 2.3.2.27 remove_due_to_license_issue IC50=200nM P98170 23298277 403 TNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLE 4hy1 A 1.9 BS01 19X A 1 I38 N41 S42 E45 D68 R71 G72 M73 I89 R131 T162 I164 I32 N35 S36 E39 D62 R65 G66 M67 I83 R119 T150 I152 5.6.2.2 0003677,0003918,0005524,0005694,0006265 Ki=2nM remove_due_to_license_issue A0A0J9WZF0 23352267 1401 KSIEVLTGLDPVKKRPGMYTNIENPNHLIQEIIDNSVDEVLAGFASKINITLYEDNSIEVADDGRGMPVDIHPEHKMSGIELIMTKLHSGGKFSNGGLHGVGVSVVNALSTRLEAEIKRDGNVYHIVFEDGFKTKDLEIIDNVGKKNTGTKIRFWPNKKYFDDIKVNFKALKNLLEAKAILCKALTIKYSNEIKKEKLTWHFETGLKGYLDHKLEAETLPAEPFIIDNFSNGDSYLDAVFCWCEDPSESIKNSYVNLIPTPQDGTHVTGLKNGIYDAIKAYIEKNSIKITANDSFAQLNYVISVKITNPQFAGQTKEKLSNKDVTNFVATAVKDLLTIWLNQNPDEARQIVENISKVAQK 4hy4 A 1.249 BS02 1BG A 1 D297 G306 L307 R308 C309 W310 E311 D314 E319 W323 D43 G52 L53 R54 C55 W56 E57 D60 E65 W69 2.3.2.27 ic50=2.7nM remove_due_to_license_issue Q13490 23298277 402 ISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRY 4hy5 A 1.752 BS02 1AQ A 1 D297 G306 L307 R308 C309 E311 D314 W323 D46 G55 L56 R57 C58 E60 D63 W72 2.3.2.27 ic50=1.3nM remove_due_to_license_issue Q13490 23298277 402 GSSISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRY 4hyf A 2.8 BS03 1AK A 1 F1035 A1038 D1045 H1048 A1049 I1059 Y1060 Y1071 I1075 F100 A103 D110 H113 A114 I124 Y125 Y136 I140 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=86nM Q9H2K2 23473363 1203 GTENLYFQSMLNTSGSGTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPEG 4hyh A 1.7 BS01 1AM A 1 L15 Y20 A36 K38 E85 Y86 C87 S88 G90 E91 E134 L137 D148 L12 Y17 A33 K35 E76 Y77 C78 S79 G81 E82 E125 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1.000000nM, EC50=30nM O14757 23535330 301 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKG 4hyi A 1.399 BS01 1AO A 1 Y20 A36 K38 E85 Y86 C87 E91 E134 L137 D148 Y18 A34 K36 E80 Y81 C82 E86 E129 L132 D143 D130 K132 E134 N135 D148 T170 D125 K127 E129 N130 D143 T165 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=3nM remove_due_to_license_issue EC50=750nM, IC50=2.0nM O14757 23535330 304 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAK 4hym A 1.9 BS01 CJC A 1 I38 N41 S42 E45 D68 G72 M73 I89 T162 I164 I32 N35 S36 E39 D62 G66 M67 I83 T150 I152 5.6.2.2 0003677,0003918,0005524,0005694,0006265 Ki=6nM remove_due_to_license_issue A0A0J9WZF0 23352267 401 KSIEVLTGLDPVKKRPGMYTNIENPNHLIQEIIDNSVDEVLAGFASKINITLYEDNSIEVADDGRGMPVDIHPEHKMSGIELIMTKLHSGGKFSNGGLHGVGVSVVNALSTRLEAEIKRDGNVYHIVFEDGFKTKDLEIIDNVGKKNTGTKIRFWPNKKYFDDIKVNFKALKNLLEAKAILCKALTIKYSNEIKKEKLTWHFETGLKGYLDHKLEAETLPAEPFIIDNFSNGDSYLDAVFCWCEDPSESIKNSYVNLIPTPQDGTHVTGLKNGIYDAIKAYIEKNSNIKITANDSFAQLNYVISVKITNPQFAGQTKEKLSNKDVTNFVATAVKDLLTIWLNQNPDEARQIVENISKVAQK 4hys A 2.415 BS02 1BJ A 1 V40 A53 E109 L110 M111 L168 V33 A46 E102 L103 M104 L161 D151 K153 N156 D169 T188 D144 K146 N149 D162 T166 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.055uM remove_due_to_license_issue P45983 23352510 401 NNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLTRYYRAPEVILGMGYKENVDIWSVGCIMGEMIKGGVLFPGTDHIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPREHTIEEWKELIYKEVM 4hyu A 2.152 BS02 1BK A 1 I32 S34 G35 Q37 G38 V40 A53 K55 E109 M111 L168 I25 S27 G28 Q30 G31 V33 A46 K48 E102 M104 L161 D151 K153 N156 D169 T188 D144 K146 N149 D162 T166 2.7.11.24 0004672,0004707,0005524,0006468 ic50=6.2nM remove_due_to_license_issue IC50=6.2nM P45983 23352510 401 NNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLTRYYRAPEVILGMGYKENVDIWSVGCIMGEMIKGGVLFPGTDHIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPREHTIEEWKELIYKEVM 4hz5 A 2.7 BS01 19Y A 1 I46 N49 E53 D76 R79 G80 M81 P82 H118 T169 I28 N31 E35 D58 R61 G62 M63 P64 H84 T135 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue H7C794 23352267 301 GLEAVRKRPGMYIGSTDSRGLHHLVYEIVDNAVDEALSGYGNEINVTIQKDNSICVADSGRGMPTGMHASGIPTVEVIFTVLHHGVGASVVNALSKWLEVHIVRDGVEYMERFEDGGKPVGTLKKIGKTKKRNGTSVTFLPDDTIFSTTNFSYEILAERLRESAFLLKGVKITLTDERGEEPKEEVFHYEE 4hze A 1.602 BS03 X7A A 1 H120 D143 H145 D147 S156 H160 D202 D251 H97 D120 H122 D124 S133 H137 D179 D228 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=509nM remove_due_to_license_issue P78540 23472952 406 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 4hzm A 1.45 BS01 1BW A 1 I30 D62 A129 R133 K163 H164 H168 M210 D249 I30 D62 A129 R133 K163 H164 H168 M207 D246 3.2.1.52 0004553,0004563,0005737,0005975,0008360,0009252,0009254,0016231,0016798,0046677,0051301,0071555 Ki=23.2uM remove_due_to_license_issue Q8ZQ06 24009110 400 MGPVMLNVEGCELDAEEREILAHPLVGGLILFTRNYHDPEQLRELVRQIRAASRNHLVVAVDQEGGRVQRFREGFTRLPAAQSFFALHGLEEGGRLAQEAGWLMASEMIAMDIDISFAPVLDVGHISAAIGERSYHADPAKALAMATRFIDGMHDAGMKTTGKHFPGHGAVTHKETPCDPRPETDIRGKDMSVFRTLISENKLDAIMPAHVIYRAIDPRPASGSPYWLKTVLRQELGFDGVIFSDDLSMGSYAERAQASLDAGCDMILVCNNRKGAVSVLDNLSPIKAERVTRLYHKGSFSRRELMDSARWKTASAQLNQLHERWQEEKAG 4hzt A 1.8 BS04 0ZA A 1 Q73 G74 L91 D93 Y132 Q134 G135 F169 W176 G291 T292 T293 N294 Q16 G17 L34 D36 Y75 Q77 G78 F112 W119 G224 T225 T226 N227 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.75uM remove_due_to_license_issue P56817 23465612 504 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHHH 4hzw A 1.701 BS02 LNV A 1 R118 E119 D151 R152 W178 E227 A246 E276 R292 R371 Y406 R37 E38 D70 R71 W98 E147 A166 E197 R212 R289 Y324 D151 E277 R292 R371 Y406 D70 E198 R212 R289 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=1.31nM remove_due_to_license_issue A9YN63 23824808 509 FRPFKSPLPLCPFRGFFPFHKDNAIRLGENKDVIVTREPYVSCDNDNCWSFALAQGALLGTKHSNGTIKDRTPYRSLIRFPIGTAPVLGNYKEICIAWSSSSCFDGKEWMHVCMTGNDNDASAQIIYGGRMTDSIKSWRKDILRTQESECQCIDGTCVVAVTDGPAANSADYRVYWIREGKIIKYENVPKTKIQHLEECSCYVDIDVYCICRDNWKGSNRPWMRINNETILETGYVCSKFHSDTPRPADPSTMSCDSPSNVNGGPGVKGFGFKAGDDVWLGRTVSTSGRSGFEIIKVTEGWINSPNHVKSITQTLVSNNDWSGYSGSFIVKAKDCFQPCFYVELIRGRPNKNDDVSWTSNSIVTFCGLDNEPGSGNWPDGSNIGFMPK 4hzx A 2.2 BS02 G39 A 1 R118 E119 D151 R152 W178 R224 E276 R292 N294 R371 Y406 R37 E38 D70 R71 W98 R144 E197 R212 N214 R289 Y324 D151 E277 R292 R371 Y406 D70 E198 R212 R289 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=0.5nM remove_due_to_license_issue A9YN63 23824808 508 FRPFKSPLPLCPFRGFFPFHKDNAIRLGENKDVIVTREPYVSCDNDNCWSFALAQGALLGTKHSNGTIKDRTPYRSLIRFPIGTAPVLGNYKEICIAWSSSSCFDGKEWMHVCMTGNDNDASAQIIYGGRMTDSIKSWRKDILRTQESECQCIDGTCVVAVTDGPAANSADYRVYWIREGKIIKYENVPKTKIQHLEECSCYVDIDVYCICRDNWKGSNRPWMRINNETILETGYVCSKFHSDTPRPADPSTMSCDSPSNVNGGPGVKGFGFKAGDDVWLGRTVSTSGRSGFEIIKVTEGWINSPNHVKSITQTLVSNNDWSGYSGSFIVKAKDCFQPCFYVELIRGRPNKNDDVSWTSNSIVTFCGLDNEPGSGNWPDGSNIGFMPK 4hzz A 1.601 BS02 G39 A 1 R118 E119 D151 R152 R224 R292 R371 Y406 R36 E37 D69 R70 R143 R211 R288 Y323 D151 E277 R292 R371 Y406 D69 E197 R211 R288 Y323 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=8.31nM remove_due_to_license_issue A9YN63 23824808 509 RPFKSPLPLCPFRGFFPFHKDNAIRLGENKDVIVTREPYVSCDNDNCWSFALAQGALLGTKHSNGTIKDRTPYRSLIRFPIGTAPVLGNYKEICIAWSSSSCFDGKEWMHVCMTGNDNDASAQIIYGGRMTDSIKSWRKDILRTQESECQCIDGTCVVAVTDGPAANSADYRVYWIREGKIIKYENVPKTKIQYLEECSCYVDIDVYCICRDNWKGSNRPWMRINNETILETGYVCSKFHSDTPRPADPSTMSCDSPSNVNGGPGVKGFGFKAGDDVWLGRTVSTSGRSGFEIIKVTEGWINSPNHVKSITQTLVSNNDWSGYSGSFIVKAKDCFQPCFYVELIRGRPNKNDDVSWTSNSIVTFCGLDNEPGSGNWPDGSNIGFMPK 4i06 A 1.8 BS03 X8A A 1 H120 D143 H145 D147 S156 H160 G161 D202 D251 H97 D120 H122 D124 S133 H137 G138 D179 D228 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=67nM remove_due_to_license_issue P78540 23472952 406 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 4i0d A 1.91 BS04 1B7 A 1 Q73 G74 L91 D93 Y132 Q134 G135 K168 F169 I171 G291 T292 T293 Q14 G15 L32 D34 Y73 Q75 G76 K109 F110 I112 G218 T219 T220 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D216 T219 3.4.23.46 0004190,0006508,0016020 ic50=0.61uM remove_due_to_license_issue P56817 23570791 504 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHHH 4i0f A 1.8 BS04 1BF A 1 Q73 G74 L91 D93 Y132 Q134 G135 K168 F169 G291 T292 T293 Q16 G17 L34 D36 Y75 Q77 G78 K111 F112 G224 T225 T226 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.45uM remove_due_to_license_issue P56817 23570791 504 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHHH 4i0r A 2.1 BS01 1B4 A 1 A400 M448 M450 A451 E452 G454 P455 L501 A34 M77 M79 A80 E81 G83 P84 L130 D494 A496 R498 N499 D512 K533 D123 A125 R127 N128 D141 K158 2.7.10.2 0004672,0004713,0005524,0006468 ic50=14nM remove_due_to_license_issue IC50=190nM P43405 23350847 701 VYLDRKLLTLEDELGSGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 4i0s A 1.98 BS01 1B5 A 1 L377 A400 M448 E449 M450 A451 P455 K458 L501 L15 A38 M80 E81 M82 A83 P87 K90 L133 D494 A496 R498 N499 D512 K533 D126 A128 R130 N131 D144 K161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=36nM remove_due_to_license_issue IC50=16600nM P43405 23350847 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 4i0t A 1.7 BS01 1B6 A 1 L377 A400 M448 M450 A451 P455 L501 S511 L15 A38 M80 M82 A83 P87 L133 S143 D494 A496 R498 N499 D512 D126 A128 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 ic50=26nM remove_due_to_license_issue IC50=26nM P43405 23350847 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 4i0z A 1.8 BS01 1BB A 1 Q73 G74 L91 D93 Y132 G135 K168 F169 G291 T292 T293 N294 R296 Q14 G15 L32 D34 Y73 G76 K109 F110 G222 T223 T224 N225 R227 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.47uM remove_due_to_license_issue P56817 23465612 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4i10 A 2.07 BS03 1BS A 1 Q73 G74 L91 Y132 Q134 G135 W176 G291 T292 T293 N294 R296 Q14 G15 L32 Y73 Q75 G76 W117 G222 T223 T224 N225 R227 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.17uM remove_due_to_license_issue P56817 23465612 504 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4i11 A 1.89 BS04 1CH A 1 Q73 G74 L91 Y132 W176 G291 T292 T293 Q16 G17 L34 Y75 W119 G228 T229 T230 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D226 T229 3.4.23.46 0004190,0006508,0016020 ic50=27.2uM remove_due_to_license_issue P56817 23465612 504 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHHH 4i12 A 1.78 BS01 1BC A 1 Q73 G74 Y132 G135 K136 K168 F169 I171 W176 G291 T292 T293 N294 Q11 G12 Y70 G73 K74 K106 F107 I109 W114 G214 T215 T216 N217 D93 S96 N98 A100 Y132 D289 T292 D31 S34 N36 A38 Y70 D212 T215 3.4.23.46 0004190,0006508,0016020 ic50=40uM remove_due_to_license_issue P56817 23570791 501 MVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVTSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4i1c A 2.0 BS03 1BE A 1 Q73 G74 D93 Y132 G135 K168 F169 I171 G291 T292 T293 Q14 G15 D34 Y73 G76 K109 F110 I112 G217 T218 T219 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D215 T218 3.4.23.46 0004190,0006508,0016020 ic50=0.4uM remove_due_to_license_issue P56817 23570791 504 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHH 4i1r A 2.7 BS01 LZU A 1 V344 K379 V381 A394 E397 F398 L401 R576 W580 L715 V7 K42 V44 A57 E60 F61 L64 R209 W213 L348 3.4.22.- 0004197,0006508 remove_due_to_license_issue Q9UDY8 23946259 801 MLAKDKVALLIGNMNYREHPKLKAPLVDVYELTNLLRQLDFKVVSLLDLTEYEMRNAVDEFLLLLDKGVYGLLYYAGHGYENFGNSFMVPVDAPNPYRSENCLCVQNILKLMQEKETGLNVFLLDMCRKTANIVFGYATCQGASGLANGIFMKFLKDRLLEDKKITVLLDEVAEDMGKCHLTKGKQALEIRSSLSEKRALTDPIQSLVRNLQWAKAHELPESMCLKFDCGVQIQLGFAAEFSNVMIIYTSIVYKPPEIIMCDAYVTDFPLDLDIDPKDANKGTPEETGSYLVSKDLPKHCLYTRLSSLQKLKEHLVFTVCLSYQYSGLEDTVEDKQEVNVGKPLIAKLDMHRH 4i3z A 2.05 BS01 ADP A 1 I10 A31 K33 F82 L83 D86 Q131 L134 D145 I10 A31 K33 F82 L83 D86 Q131 L134 D145 D127 K129 Q131 N132 D145 T158 T165 D127 K129 Q131 N132 D145 T158 T165 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=51.3uM remove_due_to_license_issue P24941 22891849 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 4i47 A 2.65 BS01 MY6 A 1 Y70 I71 E85 G109 Y70 I71 E85 G109 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 23280611 303 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 4i4e A 1.55 BS01 1BQ A 1 R426 I428 A452 M499 E500 C502 L504 G505 L553 R13 I15 A38 M85 E86 C88 L90 G91 L139 D546 A548 R550 N551 D564 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5uM remove_due_to_license_issue Q05397 23414845 1000 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPNPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4i4f A 1.75 BS01 1BR A 1 M475 L534 H544 R550 N551 L562 G563 D564 D604 M607 F608 M58 L117 H127 R133 N134 L145 G146 D147 D173 M176 F177 D546 A548 R550 N551 D564 K583 D129 A131 R133 N134 D147 K152 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.64uM remove_due_to_license_issue IC50=2200nM Q05397 23414845 702 YEIQRERIELGRCIGEGQFGDVHQGIYMSPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4i54 A 2.5 BS01 1C1 A 1 S256 E370 S375 F376 F382 I424 N425 M426 W427 G429 T430 G473 S140 E231 S236 F237 F243 I271 N272 M273 W274 G276 T277 G320 ? 0019031 Kd=110nM remove_due_to_license_issue Q0ED31 23667716 501 VWKDADTTLFCASDAKAHETEVHNVWATHACVPTDPNPQEIHLENVTENFNMWKNNMVEQMQEDVISLWDQSLQPCVKLTGGSVIKQACPKISFDPIPIHYCTPAGYVILKCNDKNFNGTGPCKNVSSVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNKSVEINCTRPSNGDIRKAYCEINGTKWNKVLKQVTEKLKEHFNNKTIIFQPPSGGDLEITMHSFNCRGEFFYCNTTQLFNNTCINGTITLPCKIKQIINMWQGTGQAMYAPPIDGKINCVSNITGILLTRDGGANNTSNETFRPGGGNIKDNWRSELYKYKVVQIE 4i5c A 2.1 BS01 C5I A 1 L881 G882 E883 G884 G887 V889 A906 M956 E957 F958 L959 L1010 D1021 L17 G18 E19 G20 G23 V25 A42 M84 E85 F86 L87 L138 D149 D1003 A1005 R1007 N1008 D1021 D1040 D131 A133 R135 N136 D149 D167 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.5nM remove_due_to_license_issue Ki=1.5nM, EC50=114nM P23458 23642482 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4i5h A 1.9 BS01 G17 A 1 A50 K52 E69 I82 I101 M106 L154 L164 D165 A42 K44 E61 I74 I93 M98 L146 L156 D157 D147 K149 S151 N152 D165 T188 D139 K141 S143 N144 D157 T173 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 Ki<2nM remove_due_to_license_issue P63086 23790491 401 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVADLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKILDFGLARVADPLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKDLPKEKLKELIFEETARFQPGY 4i5m A 1.801 BS01 R78 A 1 K57 L59 K61 C67 A80 K82 L130 E131 Y132 C133 S134 R136 F183 K16 L18 K20 C26 A39 K41 L89 E90 Y91 C92 S93 R95 F142 D176 K178 G180 N181 D194 T214 D135 K137 G139 N140 D153 T162 2.7.11.21 0004672,0005524,0006468 ic50=0.0088uM remove_due_to_license_issue IC50=14nM, Ki=<1nM, Kd=0.810000nM Q9NYY3 23794260 401 RIIVDPTTGKRYSRGKTLGKGGFAKCYEMTDLTNNKVYAAKIIPHSRVSKPHQREKIDKEIELHRILHHKHVVQFYHYFEDKENIYILLEYCSRRSMAHILKARKVLTEPEVRYYLRQIVSGLKYLHEQEILHRDLKLGNFFINESMELKVGDFGLAARLETPNYLSPEVLNKQGHGAESDIWALGCVMYTMLLGRPPFETTNLKETYRSIREARYTMPSSLLAPAKHLIASMLSKNPEDRPSLDDIIRHDFFTQGFTPDRLSSSCCHTVPDF 4i5p A 1.738 BS01 1D1 A 1 L88 C96 A109 L159 E160 Y161 C162 F212 L18 C26 A39 L89 E90 Y91 C92 F142 D205 K207 G209 N210 D223 T243 D135 K137 G139 N140 D153 T173 2.7.11.21 0004672,0005524,0006468 ic50=0.377uM remove_due_to_license_issue Q9NYY3 23794260 401 RIIVDPTTGKRYSRGKTLGKGGFAKCYEMTDLTNNKVYAAKIIPHSRVSKPHQREKIDKEIELHRILHHKHVVQFYHYFEDKENIYILLEYCSRRSMAHILKARKVLTEPEVRYYLRQIVSGLKYLHEQEILHRDLKLGNFFINESMELKVGDFGLAARLEPLEHRRRTICGTPNYLSPEVLNKQGHGAESDIWALGCVMYTMLLGRPPFETTNLKETYRSIREARYTMPSSLLAPAKHLIASMLSKNPEDRPSLDDIIRHDFFTQGFTPDRLSSSCCHTVPDF 4i60 A 2.5 BS01 B1R A 1 L14 S16 Y33 T35 V37 T38 A39 T40 W70 S73 S75 T77 W97 S101 R114 N118 L14 S16 Y33 T35 V37 T38 A39 T40 W70 S73 S75 T77 W97 S101 R114 N118 ? 0005576,0009374,0019731 Kd=1.87uM remove_due_to_license_issue P02701 23603015 203 ARKCSLTGKWTNDLGSNMTIGAVNSKGEFTGTYTTAVTATSNEIKESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRLRTQKE 4i6b A 1.8 BS01 11G A 1 L88 C96 A109 V143 L159 E160 C162 F212 L18 C26 A39 V73 L89 E90 C92 F142 D205 K207 G209 N210 D223 T243 D135 K137 G139 N140 D153 T173 2.7.11.21 0004672,0005524,0006468 ic50=1.17uM remove_due_to_license_issue Q9NYY3 23794260 401 RIIVDPTTGKRYSRGKTLGKGGFAKCYEMTDLTNNKVYAAKIIPHSRVSKPHQREKIDKEIELHRILHHKHVVQFYHYFEDKENIYILLEYCSRRSMAHILKARKVLTEPEVRYYLRQIVSGLKYLHEQEILHRDLKLGNFFINESMELKVGDFGLAARLEPLEHRRRTICGTPNYLSPEVLNKQGHGAESDIWALGCVMYTMLLGRPPFETTNLKETYRSIREARYTMPSSLLAPAKHLIASMLSKNPEDRPSLDDIIRHDFFTQGFTPDRLSSSCCHTVPDFH 4i6f A 2.9 BS01 1C7 A 1 C96 A109 L159 E160 Y161 C162 F212 C26 A39 L89 E90 Y91 C92 F142 D205 K207 G209 N210 D223 T243 D135 K137 G139 N140 D153 T173 2.7.11.21 0004672,0005524,0006468 remove_due_to_license_issue IC50=5.0nM Q9NYY3 23794260 401 RIIVDPTTGKRYSRGKTLGKGGFAKCYEMTDLTNNKVYAAKIIPHSRVSKPHQREKIDKEIELHRILHHKHVVQFYHYFEDKENIYILLEYCSRRSMAHILKARKVLTEPEVRYYLRQIVSGLKYLHEQEILHRDLKLGNFFINESMELKVGDFGLAARLEPLEHRRRTICGTPNYLSPEVLNKQGHGAESDIWALGCVMYTMLLGRPPFETTNLKETYRSIREARYTMPSSLLAPAKHLIASMLSKNPEDRPSLDDIIRHDFFTQGFTPDRLSSSCCHTVPDFH 4i6h A 1.91 BS01 1C8 A 1 L88 K90 C96 A109 V143 L159 E160 Y161 C162 R165 F212 L18 K20 C26 A39 V73 L89 E90 Y91 C92 R95 F142 D205 K207 G209 N210 D223 T243 D135 K137 G139 N140 D153 T173 2.7.11.21 0004672,0005524,0006468 ic50=0.005uM remove_due_to_license_issue Q9NYY3 23794260 401 RIIVDPTTGKRYSRGKTLGKGGFAKCYEMTDLTNNKVYAAKIIPHSRVSKPHQREKIDKEIELHRILHHKHVVQFYHYFEDKENIYILLEYCSRRSMAHILKARKVLTEPEVRYYLRQIVSGLKYLHEQEILHRDLKLGNFFINESMELKVGDFGLAARLEPLEHRRRTICGTPNYLSPEVLNKQGHGAESDIWALGCVMYTMLLGRPPFETTNLKETYRSIREARYTMPSSLLAPAKHLIASMLSKNPEDRPSLDDIIRHDFFTQGFTPDRLSSSCCHTVPDFH 4i6q A 1.85 BS02 1DT A 1 L828 V836 A853 M902 Y904 L905 L956 L14 V22 A39 M82 Y84 L85 L136 D949 A951 R953 N954 D967 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.03uM remove_due_to_license_issue IC50=30nM P52333 23541670 1202 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGS 4i71 A 1.28 BS01 AGV A 1 N12 D14 D40 F79 W83 M164 N173 E184 N186 R252 Y257 W260 D261 N15 D17 D43 F82 W86 M167 N176 E187 N189 R255 Y260 W263 D264 3.2.2.1 0005829,0006139,0006152,0006166,0008477,0016798,0016799,0016810,0020015,0046872 Ki=18nM remove_due_to_license_issue Q57ZL6 23897478 401 GSHMAKTVILDHDGNKDDFVAMILLLSNPKKVNLIGCICTDADCFVENGFDVTGKIMCAMHRLIKTPLFPIGKSTATAVNAFPTEWRFSAKNLDDMPFLNIVEDVALWEKLKPENEAHNGQQLLADLVMKSKEKVTVCVTGPLSNMAWCIEKYGEAFTSKVEECVIMGGAVDVGGNVFLPTTDGSAEWNIYWDPPAAKKVLCCPNIRCVLFSLDATNTVPVRSVDVKGFGAQNQYLLSQMVGTMWAMSTHEEILRDGDAYYAWDALTAAYILEPTIATLEPVALDVDVSKGKSEGRTPRAPCVHVARNPSKQMFHDLVFASTRVC 4i72 A 2.05 BS02 UA2 A 1 N12 D14 D40 F79 W83 M164 E184 N186 R252 Y257 W260 D261 N15 D17 D43 F82 W86 M167 E187 N189 R255 Y260 W263 D264 3.2.2.1 0005829,0006139,0006152,0006166,0008477,0016798,0016799,0016810,0020015,0046872 Ki=0.9nM remove_due_to_license_issue Q57ZL6 23897478 402 GSHMAKTVILDHDGNKDDFVAMILLLSNPKKVNLIGCICTDADCFVENGFDVTGKIMCAMHRLIKTPLFPIGKSTATAVNAFPTEWRFSAKNLDDMPFLNIVEDVALWEKLKPENEAHNGQQLLADLVMKSKEKVTVCVTGPLSNMAWCIEKYGEAFTSKVEECVIMGGAVDVGGNVFLPTTDGSAEWNIYWDPPAAKKVLCCPNIRCVLFSLDATNTVPVRSVDVKGFGAQNQYLLSQMVGTMWAMSTHEEILRDGDAYYAWDALTAAYILEPTIATLEPVALDVDVSKGKSEGRTPRASGKPCVHVARNPSKQMFHDLVFASTRVC 4i73 A 2.18 BS02 MBY A 1 D14 D40 F79 W83 M164 N173 E184 W185 N186 R252 Y257 W260 D261 D17 D43 F82 W86 M167 N176 E187 W188 N189 R255 Y260 W263 D264 3.2.2.1 0005829,0006139,0006152,0006166,0008477,0016798,0016799,0016810,0020015,0046872 Ki=190nM remove_due_to_license_issue Q57ZL6 23897478 402 GSHMAKTVILDHDGNKDDFVAMILLLSNPKKVNLIGCICTDADCFVENGFDVTGKIMCAMHRLIKTPLFPIGKSTATAVNAFPTEWRFSAKNLDDMPFLNIVEDVALWEKLKPENEAHNGQQLLADLVMKSKEKVTVCVTGPLSNMAWCIEKYGEAFTSKVEECVIMGGAVDVGGNVFLPTTDGSAEWNIYWDPPAAKKVLCCPNIRCVLFSLDATNTVPVRSVDVKGFGAQNQYLLSQMVGTMWAMSTHEEILRDGDAYYAWDALTAAYILEPTIATLEPVALDVDVSKGKSEGRTPRAGKPCVHVARNPSKQMFHDLVFASTRVC 4i74 A 1.68 BS02 MBY A 1 N12 D14 D40 F79 W83 M164 N173 E184 W185 N186 E248 E249 W260 D261 N15 D17 D43 F82 W86 M167 N176 E187 W188 N189 E251 E252 W263 D264 3.2.2.1 0005829,0006139,0006152,0006166,0008477,0016798,0016799,0016810,0020015,0046872 remove_due_to_license_issue Q57ZL6 23897478 408 GSHMAKTVILDHDGNKDDFVAMILLLSNPKKVNLIGCICTDADCFVENGFDVTGKIMCAMHRLIKTPLFPIGKSTATAVNAFPTEWRFSAKNLDDMPFLNIVEDVALWEKLKPENEAHNGQQLLADLVMKSKEKVTVCVTGPLSNMAWCIEKYGEAFTSKVEECVIMGGAVDVGGNVFLPTTDGSAEWNIYWDPPAAKKVLCCPNIRCVLFSLDATNTVPVRSVDVKGFGAQNQYLLSQMVGTMWAMSTHEEILRDGDAYYAWDALTAAYILEPTIATLEPVALDVDVSKGKSEGRTPRASGPCVHVARNPSKQMFHDLVFASTRVC 4i7f A 2.5 BS01 NVE A 1 P95 L100 K103 K104 S105 V106 Y181 Y188 G190 R199 P225 F227 W229 L234 H235 P236 Y318 P95 L100 K103 K104 S105 V106 Y181 Y188 G190 R199 P225 F227 W229 L234 H235 P236 Y318 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=100nM remove_due_to_license_issue P04585 23375792 601 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 4i7m A 1.48 BS01 2LP A 1 A99 H102 V103 V111 L118 A110 H113 V114 V122 L129 E11 D20 E22 D31 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Ka=13900M^-1 remove_due_to_license_issue P00720 23473072 202 PTTENLYFQGSMNIFEMLRIDEGLRLKIYKDCEGYYTIGIGHLLTKSPDLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINHVFQMGVTGVAGFTNVLRMLQQKRWDEAAVNLAKSRWYNQCPDRAKRVITTFRTGTWDAYKNL 4i7p A 1.6 BS01 ES3 A 1 V87 Y88 A99 H102 V111 L118 L121 F153 V99 Y100 A111 H114 V123 L130 L133 F165 E11 D20 E23 D32 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Ka=3155M^-1 remove_due_to_license_issue Kd=317000nM P00720 23473072 202 IPTTENLYFQGSMNIFEMLRIDEGLRLKIYKDCEGYYTIGIGHLLTKSPDLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINHVFQMGVTGVAGFTNVLRMLQQKRWDEAAVNLAKSRWYNQCPDRAKRVITTFRTGTWDAYKNL 4i7y H 2.4 BS02 dna D 0 H91 P92 R93 Y94 N95 W96 R97 R126 L130 H230 R233 W237 Q244 F245 H87 P88 R89 Y90 N91 W92 R93 R123 L130 H234 R237 W241 Q248 F249 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 24311581 1 ~ 27 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4i8n A 2.5 BS01 1CG A 1 D48 D181 F182 C215 S216 A217 I219 G220 R221 M258 Q262 D47 D180 F181 C214 S215 A216 I218 G219 R220 M257 Q261 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P18031 23964742 401 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL 4i8w A 1.96 BS01 G07 B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 23877703 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4i8w B 1.96 BS01 G07 B 1 D25 G27 A28 D30 G48 P81 V82 I84 D25 G27 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=12.7pM remove_due_to_license_issue P0C6F2 23877703 300 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4i8x A 2.23 BS01 6P3 A 1 V30 T94 V135 N137 R168 A237 T247 V30 T94 V125 N127 R158 A227 T237 D165 R168 H192 D155 R158 H182 1.1.1.27 0003824,0004459,0005737,0006089,0006090,0016491,0016616,0019752 Kd=2300uM remove_due_to_license_issue P13491 23302067 401 AALKDQLIHNLLKEEHVPQNKITVVGVGAVGMACAISILMKDLADELALVDVMEDKLKGEMMDLQHGSLFLRTPKIVSGKDYSVTANSKLVIITAGALVQRNVNIFKFIIPNVVKYSPHCKLLVVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHALSCHGWILGEHGDSSVPVWSGMNVAGVSLKTLHPELGTDADKEQWKQVHKQVVDSAYEVIKLKGYTTWAIGLSVADLAESIMKNLRRVHPISTMLKGLYGIKEDVFLSVPCVLGQNGISDVVKVTLTSEEEAHLKKSADTLWGIQKELQF 4i8x C 2.23 BS01 6P3 C 1 V30 T94 R98 V135 N137 R168 T247 V30 T94 R98 V135 N137 R168 T247 R105 D165 R168 H192 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005737,0006089,0006090,0016491,0016616,0019752 Kd=2300uM remove_due_to_license_issue P13491 23302067 401 AALKDQLIHNLLKEEHVPQNKITVVGVGAVGMACAISILMKDLADELALVDVMEDKLKGEMMDLQHGSLFLRTPKIVSGKDYSVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPHCKLLVVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHALSCHGWILGEHGDSSVPVWSGMNVAGVSLKTLHPELGTDADKEQWKQVHKQVVDSAYEVIKLKGYTTWAIGLSVADLAESIMKNLRRVHPISTMLKGLYGIKEDVFLSVPCVLGQNGISDVVKVTLTSEEEAHLKKSADTLWGIQKELQF 4i8z A 1.75 BS01 G08 A 1 D25 G27 A28 D30 I47 G48 P81 V82 I84 D25 G27 A28 D30 I47 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8.9pM remove_due_to_license_issue P0C6F2 23877703 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4i8z B 1.75 BS01 G08 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 23877703 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4i9h A 2.17 BS01 1E4 A 1 G26 G28 V30 D51 V52 T94 A95 G96 R111 N114 I115 F118 V135 S136 N137 R168 A237 T247 G26 G28 V30 D51 V52 T94 A95 G96 R105 N108 I109 F112 V129 S130 N131 R162 A231 T241 D165 R168 H192 D159 R162 H186 1.1.1.27 0003824,0004459,0005737,0006089,0006090,0016491,0016616,0019752 Kd=0.068uM remove_due_to_license_issue P13491 23302067 401 AALKDQLIHNLLKEEHVPQNKITVVGVGAVGMACAISILMKDLADELALVDVMEDKLKGEMMDLQHGSLFLRTPKIVSGKDYSVTANSKLVIITAGARQLNLVQRNVNIFKFIIPNVVKYSPHCKLLVVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHALSCHGWILGEHGDSSVPVWSGMNVAGVSLKTLHPELGTDADKEQWKQVHKQVVDSAYEVIKLKGYTTWAIGLSVADLAESIMKNLRRVHPISTMLKGLYGIKEDVFLSVPCVLGQNGISDVVKVTLTSEEEAHLKKSADTLWGIQKELQF 4i9h C 2.17 BS01 1E4 C 1 G26 G28 V30 D51 V52 T94 A95 G96 R111 I115 F118 V135 S136 N137 R168 A237 T247 G26 G28 V30 D51 V52 T94 A95 G96 R108 I112 F115 V132 S133 N134 R165 A234 T244 R105 D165 R168 H192 R102 D162 R165 H189 1.1.1.27 0003824,0004459,0005737,0006089,0006090,0016491,0016616,0019752 Kd=0.068uM remove_due_to_license_issue P13491 23302067 401 AALKDQLIHNLLKEEHVPQNKITVVGVGAVGMACAISILMKDLADELALVDVMEDKLKGEMMDLQHGSLFLRTPKIVSGKDYSVTANSKLVIITAGARGESRLNLVQRNVNIFKFIIPNVVKYSPHCKLLVVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHALSCHGWILGEHGDSSVPVWSGMNVAGVSLKTLHPELGTDADKEQWKQVHKQVVDSAYEVIKLKGYTTWAIGLSVADLAESIMKNLRRVHPISTMLKGLYGIKEDVFLSVPCVLGQNGISDVVKVTLTSEEEAHLKKSADTLWGIQKELQF 4i9i A 2.4 BS02 1DY A 1 H1184 G1185 F1188 A1191 G1196 D1198 H1201 Y1203 I1212 Y1213 F1214 A1215 S1221 Y1224 E1291 H81 G82 F85 A88 G93 D95 H98 Y100 I109 Y110 F111 A112 S118 Y121 E188 2.4.2.-,2.4.2.30 0003950 ic50=0.008uM remove_due_to_license_issue IC50=8.0nM O95271 23316926 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEH 4i9o A 2.0 BS01 KI1 A 1 I611 L628 Y631 A632 V635 I660 E663 C664 I24 L41 Y44 A45 V48 I73 E76 C77 2.3.1.-,2.3.1.48 0003712,0004402,0006355 remove_due_to_license_issue P45481 23384013 701 RKGWHEHVTQDLRSHLVHKLVQAIFPTPDPAALKDRRMENLVAYAKKVEGDMYESANSRDEYYHLLAEKIYKIQKECE 4i9r A 2.6 BS01 RET A 1 F15 P39 V54 W109 K111 L121 M123 F15 P39 V54 W109 K111 L121 M123 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 remove_due_to_license_issue P29373 24059243 201 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIWVAAASKPAVEIKQEGDTFYIKVSTTVWTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTKELTNDGELILTMTADDVVCTLVFVRE 4i9s A 2.58 BS01 RET A 1 F15 A36 W59 K111 L121 F15 A36 W59 K111 L121 ? 0001972,0005501,0005504,0005515,0005634,0005654,0005737,0005783,0005829,0006355,0007165,0008289,0008544,0015908,0016918,0019841,0030332,0035115,0042573,0048672,0070062 remove_due_to_license_issue P29373 24059243 201 PNFSGNWKIIRSENFEELLKVLGVNVMLRKIAVAAASKPAVEIKQEGDTFYIKVSTTVWTTEINFKVGEEFEEQTVDGRPCKSLVKWESENKMVCEQKLLKGEGPKTSWTKELTNDGELILTMTADDVVCTLVFVRE 4i9u A 2.5 BS01 1E7 A 1 V25 G26 D51 V52 A95 R111 I115 F118 I119 V25 G26 D51 V52 A95 R103 I107 F110 I111 D165 R168 H192 D157 R160 H184 1.1.1.27 0003824,0004459,0005737,0006089,0006090,0016491,0016616,0019752 Kd=137uM remove_due_to_license_issue P13491 23302067 401 AALKDQLIHNLLKEEHVPQNKITVVGVGAVGMACAISILMKDLADELALVDVMEDKLKGEMMDLQHGSLFLRTPKIVSGKDYSVTANSKLVIITAGARNLVQRNVNIFKFIIPNVVKYSPHCKLLVVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHALSCHGWILGEHGDSSVPVWSGMNVAGVSLKTLHPELGTDADKEQWKQVHKQVVDSAYEVIKLKGYTTWAIGLSVADLAESIMKNLRRVHPISTMLKGLYGIKEDVFLSVPCVLGQNGISDVVKVTLTSEEEAHLKKSADTLWGIQKELQF 4i9z A 2.08 BS01 5BA A 1 Y612 A779 V782 F786 M816 Q817 F820 Y78 A238 V241 F245 M254 Q255 F258 3.1.4.35 0004114,0007165,0008081 ic50=18.2nM remove_due_to_license_issue IC50=18nM O76074 23867165 901 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 4ia0 A 2.17 BS01 5BB A 1 L725 D764 F786 M816 Q817 F820 L181 D220 F242 M250 Q251 F254 3.1.4.35 0004114,0007165,0008081 ic50=77nM remove_due_to_license_issue IC50=77nM O76074 23867165 901 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAE 4iaw A 2.4 BS01 LIZ A 1 Q33 R36 T52 Q54 V66 A68 R70 L79 Y106 F123 S136 Q33 R36 T52 Q54 V66 A68 R70 L79 Y106 F123 S136 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 Kd=0.234nM remove_due_to_license_issue P80188 23542582 201 QDSTSDLIPAPPLSKVPLQQNFQDNQFHGKWYQVGRAGNAAPREDKDLLKMTAQTYELKEDKSYNVTAVRFRKKMCEYLTMTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVQQNREYFSISLLGRTKELASELKENFIRFSKSLGLPENHIVFPVPIDQCIDGSA 4iax A 1.9 BS01 LIZ A 1 Q33 T52 Q54 V66 A68 R70 E77 Y78 L79 Y106 F123 S136 Q28 T47 Q49 V61 A63 R65 E72 Y73 L74 Y101 F118 S131 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 Kd=0.273nM remove_due_to_license_issue P80188 23542582 201 DLIPAPPLSKVPLQQNFQDNQFHGKWYQVGRAGNAAPPMDPELLLLTAQTYELKEDKSYDVTAVRFRKKMCEYLTMTFVPSPQPGEFTLGNIKNYPGLTSYFVRVVSTNYNQHAMVFFKKVQQNREYFSISLLGRTKELASELKENFIRFSKSLGLPENHIVFPVPIDQCID 4ibb A 1.752 BS01 1DK A 1 A221 Q241 Q244 K248 K251 I295 A4 Q24 Q27 K31 K34 I78 ? Kd=270.7uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibc A 1.745 BS01 12G A 1 A221 Q241 Q244 V245 K248 K251 I295 D302 A4 Q24 Q27 V28 K31 K34 I78 D85 ? Kd=1049uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibd A 1.84 BS01 1DL A 1 Q241 Q244 K248 P293 I295 Q24 Q27 K31 P76 I78 ? Kd=214.6uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibe A 1.95 BS01 11Y A 1 Q241 Q244 K248 K251 P293 I295 I297 Q24 Q27 K31 K34 P76 I78 I80 ? Kd=70.6uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibf A 2.291 BS01 1D5 A 1 Q241 Q244 K248 K251 P293 I295 D302 F328 Q24 Q27 K31 K34 P76 I78 D85 F111 ? Kd=36.8uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibg A 1.413 BS01 1D6 A 1 A221 Q241 Q244 K248 K251 P293 I295 I297 A4 Q24 Q27 K31 K34 P76 I78 I80 ? Kd=108uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibg B 1.413 BS01 1D6 B 1 Q241 V245 K248 K251 P293 I295 Q24 V28 K31 K34 P76 I78 ? Kd=108uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibi A 1.473 BS01 1D8 A 1 Q241 Q244 V245 K248 K251 P293 I295 D302 F328 Q24 Q27 V28 K31 K34 P76 I78 D85 F111 ? Kd=73uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibj A 1.54 BS01 1D9 A 1 K222 Q241 Q244 K248 K251 I295 F328 K6 Q25 Q28 K32 K35 I79 F112 ? Kd=47uM remove_due_to_license_issue Q05127 24495995 401 PDISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibk A 1.85 BS01 1DE A 1 Q241 Q244 V245 K248 K251 P293 I295 D302 F328 Q24 Q27 V28 K31 K34 P76 I78 D85 F111 ? Kd=50.4uM remove_due_to_license_issue Q05127 24495995 401 DISAKDLRNIMYDHLPGFGTAFHQLVQVICKLGKDSNSLDIIHAEFQASLAEGDSPQCALIQITKRVPIFQDAAPPVIHIRSRGDIPRACQKSLRPVPPSPKIDRGWVCVFQLQDGKTLGLKI 4ibm A 1.8 BS01 IR1 A 1 L1002 G1003 A1028 M1076 E1077 M1079 A1080 G1082 M1139 D1150 L21 G22 A47 M95 E96 M98 A99 G101 M158 D169 D1132 A1134 R1136 N1137 D1150 E1159 L1171 D151 A153 R155 N156 D169 E178 L190 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=1.8uM remove_due_to_license_issue P06213 23935097 1301 SVYVPDEWEVSREKITLLRELGQGSFGMVYEGNARDIIKGEAETRVAVKTVNESASLRERIEFLNEASVMKGFTCHHVVRLLGVVSKGQPTLVVMELMAHGDLKSYLRSLRPEAENNPGRPPPTLQEMIQMAAEIADGMAYLNAKKFVHRDLAARNCMVAHDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMAPESLKDGVFTTSSDMWSFGVVLWEITSLAEQPYQGLSNEQVLKFVMDGGYLDQPDNCPERVTDLMRMCWQFNPNMRPTFLEIVNLLKDDLHPSFPEVSFFHSEEN 4idn A 2.252 BS01 GNP A 1 F76 R77 G79 K80 S81 F82 W112 R113 R118 E119 T120 R217 D218 P272 V276 F47 R48 G50 K51 S52 F53 W83 R84 R89 E90 T91 R188 D189 P243 V247 3.6.5.- 0003924,0005525 Kd=5.77uM remove_due_to_license_issue Q8WXF7 23334294 501 KKAGPVQVLIVKDDHSFELDETALNRILLSEAVRDKEVVAVSVAGAFRKGKSFLMDFMLRYMYNQESVDWVGDYNEPLTGFSWRGGSERETTGIQIWSEIFLINKPDGKKVAVLLMDTQGTFDSQSTLRDSATVFALSTMISSIQVYNLSQNVQEDDLQHLQLFTEYGRLAMEETFLKPFQSLIFLVRDWSFPYEFSYGADGGAKFLEKRLKVSGNQHEELQNVRKHIHSCFTNISCFLLPHPGLKVATNPNFDGKLKEIDDEFIKNLKILIPWLLSPESLDIKEINGNKITCRGLVEYFKAYIKIYQGEELPHPKSMLQATAEANNLAAVATAKDTYNKKMEEICGGDKPFLAPNDLQTKHLQLKEESVKLFRGVKKMGGEEFSRRYLQQLESEIDELYIQYIKHNDSKNIFHAAR 4idn B 2.252 BS01 GNP B 1 F76 R77 G79 K80 S81 F82 W112 R113 R118 T120 R217 D218 P272 V276 F46 R47 G49 K50 S51 F52 W82 R83 R88 T90 R187 D188 P242 V246 3.6.5.- 0003924,0005525 Kd=5.77uM remove_due_to_license_issue Q8WXF7 23334294 501 KAGPVQVLIVKDDHSFELDETALNRILLSEAVRDKEVVAVSVAGAFRKGKSFLMDFMLRYMYNQESVDWVGDYNEPLTGFSWRGGSERETTGIQIWSEIFLINKPDGKKVAVLLMDTQGTFDSQSTLRDSATVFALSTMISSIQVYNLSQNVQEDDLQHLQLFTEYGRLAMEETFLKPFQSLIFLVRDWSFPYEFSYGADGGAKFLEKRLKVSGNQHEELQNVRKHIHSCFTNISCFLLPHPGLKVATNPNFDGKLKEIDDEFIKNLKILIPWLLSPESLDIKEINGNKITCRGLVEYFKAYIKIYQGEELPHPKSMLQATAEANNLAAVATAKDTYNKKMEEICGGDKPFLAPNDLQTKHLQLKEESVKLFRGVKKMGGEEFSRRYLQQLESEIDELYIQYIKHNDSKNIFHAARAAALEHH 4ido A 2.091 BS01 GDP A 1 R77 K78 G79 K80 S81 F82 W112 R113 G114 R217 D218 P272 V276 R47 K48 G49 K50 S51 F52 W82 R83 G84 R187 D188 P242 V246 3.6.5.- 0003924,0005525 remove_due_to_license_issue Q8WXF7 23334294 501 KAGPVQVLIVKDDHSFELDETALNRILLSEAVRDKEVVAVSVAGAFRKGKSFLMDFMLRYMYNQESVDWVGDYNEPLTGFSWRGGSERETTGIQIWSEIFLINKPDGKKVAVLLMDTQGTFDSQSTLRDSATVFALSTMISSIQVYNLSQNVQEDDLQHLQLFTEYGRLAMEETFLKPFQSLIFLVRDWSFPYEFSYGADGGAKFLEKRLKVSGNQHEELQNVRKHIHSCFTNISCFLLPHPGLKVATNPNFDGKLKEIDDEFIKNLKILIPWLLSPESLDIKEINGNKITCRGLVEYFKAYIKIYQGEELPHPKSMLQATAEANNLAAVATAKDTYNKKMEEICGGDKPFLAPNDLQTKHLQLKEESVKLFRGVKKMGGEEFSRRYLQQLESEIDELYIQYIKHNDSKNIF 4ido B 2.091 BS01 GDP B 1 R77 K78 G79 K80 S81 F82 W112 R113 G114 R217 D218 P272 V276 R47 K48 G49 K50 S51 F52 W82 R83 G84 R187 D188 P242 V246 3.6.5.- 0003924,0005525 remove_due_to_license_issue Q8WXF7 23334294 501 KAGPVQVLIVKDDHSFELDETALNRILLSEAVRDKEVVAVSVAGAFRKGKSFLMDFMLRYMYNQESVDWVGDYNEPLTGFSWRGGSERETTGIQIWSEIFLINKPDGKKVAVLLMDTQGTFDSQSTLRDSATVFALSTMISSIQVYNLSQNVQEDDLQHLQLFTEYGRLAMEETFLKPFQSLIFLVRDWSFPYEFSYGADGGAKFLEKRLKVSGNQHEELQNVRKHIHSCFTNISCFLLPHPGLKVATNPNFDGKLKEIDDEFIKNLKILIPWLLSPESLDIKEINGNKITCRGLVEYFKAYIKIYQGEELPHPKSMLQATAEANNLAAVATAKDTYNKKMEEICGGDKPFLAPNDLQTKHLQLKEESVKLFRGVKKMGGEEFSRRYLQQLESEIDELYIQYIKHNDSKNIFHAARAAALEH 4idt A 2.4 BS01 T28 A 1 G409 V414 K429 M469 L472 S476 L522 C533 D534 G77 V82 K97 M137 L140 S144 L190 C201 D202 D515 K517 N520 D534 T559 D183 K185 N188 D202 T218 2.7.11.25 0004672,0004674,0005524,0006468 ic50=0.1uM remove_due_to_license_issue IC50=4600nM Q99558 23374866 701 VEEYLVHALQGSVSSGQAHSLTSLAKTWAARGSRSREPSPKTEDNEGVLLTEKLKPVDYEYREEVHWATHQLRLGRGSFGEVHRMEDKQTGFQCAVKKVRLEVFRAEELMACAGLTSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLVKEQGCLPEDRALYYLGQALEGLEYLHSRRILHGDVKADNVLLSSDGSHAALCDFGHAVCLQTGDYIPGTETHMAPEVVLGRSCDAKVDVWSSCCMMLHMLNGCHPWTQFFRGPLCLKIASEPPPVREIPPSCAPLTAQAIQEGLRKEPIHRVSAAELGGKVNRALQQVGGLKSPWRGEYKEPRHP 4idv A 2.9 BS01 13V A 1 R408 V414 E440 I467 M469 E470 L472 G475 S476 Q479 L522 C533 D534 F535 R68 V74 E100 I127 M129 E130 L132 G135 S136 Q139 L182 C193 D194 F195 D515 K517 N520 D534 L551 T559 D175 K177 N180 D194 L211 T219 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=20nM Q99558 23374866 701 FSVEEYLVHALQGSVSSGQAHSLTSLAKTWAARTEDNEGVLLTEKLKPVDYEYREEVHWATHQLRLGRGSFGEVHRMEDKQTGFQCAVKKVRLEVFRAEELMACAGLTSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLVKEQGCLPEDRALYYLGQALEGLEYLHSRRILHGDVKADNVLLSSDGSHAALCDFGHAVCLQPDGLGKSLLTGDYIPGTETHMAPEVVLGRSCDAKVDVWSSCCMMLHMLNGCHPWTQFFRGPLCLKIASEPPPVREIPPSCAPLTAQAIQEGLRKEPIHRVSAAELGGKVNRALQQVGGLKSPWRGEYKEPRHP 4ie0 A 2.53 BS02 PD2 A 1 R96 H231 D233 Y295 H307 V309 R316 S318 T320 R70 H180 D182 Y233 H245 V247 R254 S256 T258 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue IC50=8300nM Q9C0B1 23547775 603 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAAKEKADEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4ie2 A 2.2082 BS03 1EC A 1 H120 D143 H145 D147 S156 H160 G161 D202 D251 H97 D120 H122 D124 S133 H137 G138 D179 D228 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=4500nM remove_due_to_license_issue P78540 23453840 405 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 4ie3 A 2.3522 BS03 1EE A 1 D143 H145 D147 N149 S156 H160 D202 D251 D120 H122 D124 N126 S133 H137 D179 D228 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=980nM remove_due_to_license_issue P78540 23453840 405 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 4ie4 A 2.5048 BS02 8XQ A 1 N205 H231 D233 V244 Y295 H307 V309 R316 S318 N151 H177 D179 V190 Y230 H242 V244 R251 S253 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 ic50=3.3uM remove_due_to_license_issue IC50=3300nM Q9C0B1 23547775 603 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNTEAEIAAACETFLKLNDYLQIETIQALEELAAKEKADEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4ie5 A 1.95 BS02 MD6 A 1 R96 N205 H231 D233 Y295 H307 V309 R316 S318 R322 R70 N153 H179 D181 Y232 H244 V246 R253 S255 R259 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 ic50=15uM remove_due_to_license_issue IC50=15000nM Q9C0B1 23547775 602 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNITEAEIAAACETFLKLNDYLQIETIQALEELAAKEKANDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4ie6 A 2.5036 BS02 UN9 A 1 R96 Y108 V228 H231 D233 Y295 H307 V309 R316 S318 T320 R322 R74 Y86 V183 H186 D188 Y239 H251 V253 R260 S262 T264 R266 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 ic50=2.8uM remove_due_to_license_issue IC50=2800nM Q9C0B1 23547775 602 GLVPRGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAAKEKANEDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4ie7 A 2.6004 BS02 RHN A 1 Y108 L109 V228 S229 H231 D233 E234 R322 Y82 L83 V175 S176 H178 D180 E181 R258 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 23547775 602 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNITEAEIAAACETFLKLNDYLQIETIQALEELAAKEKADEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCELEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4ieh A 2.1 BS01 1E9 A 1 A59 D62 F63 R66 Y67 M74 L96 G104 V107 Y161 A34 D37 F38 R41 Y42 M49 L71 G79 V82 Y136 ? 0042981 Kd=14nM remove_due_to_license_issue P10415,Q07817 24900652 201 YDNREIVMKYIHYKLSQRGYEWDSEVVHLTLRQAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGP 4ifh B 3.286 BS02 1EF B 1 H108 E111 H112 F115 S128 N139 E189 F820 Y831 V833 H66 E69 H70 F73 S86 N97 E147 F778 Y789 V791 E111 E69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 26394692 1102 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLEHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDLSQAPALPQPEVIQNMTEFKRGLPLFPLVKP 4igr A 2.65 BS01 3ZA A 1 Y491 P518 T520 R525 G690 A691 T692 E739 Y765 Y59 P86 T88 R93 G138 A139 T140 E187 Y213 ? 0015276,0016020 remove_due_to_license_issue Ki=123nM P42264 23414088 901 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGC 4igt A 1.24 BS01 3ZA A 1 Y471 P499 T501 R506 G674 S675 T676 E726 Y753 Y61 P89 T91 R96 G141 S142 T143 E193 Y220 ? 0015276,0016020 Kd=12.8nM remove_due_to_license_issue Ki=126000nM P19491 23414088 801 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECGS 4ih3 A 2.493 BS02 PDC A 1 H8 R47 P77 H174 W191 D291 L296 H8 R47 P77 H174 W191 D291 L296 4.1.1.45 0001760,0005515,0005737,0005829,0006569,0008270,0016787,0016831,0019748,0046872,1904985,1905004,1905012 remove_due_to_license_issue Q8TDX5 25392945 402 MKIDIHSHILPKEWPDLKKRFGYGGWVQLQHHSKGEAKLLKDGKVFRVVRENCWDPEVRIREMDQKGVTVQALSTVPVMFSYWAKPEDTLNLCQLLNNDLASTVVSYPRRFVGLGTLPMQAPELAVKEMERCVKELGFPGVQIGTHVNEWDLNAQELFPVYAAAERLKCSLFVHPWDMQMDGRMAKYWLPWLVGMPAETTIAICSMIMGGVFEKFPKLKVCFAHGGGAFPFTVGRISHGFSMRPDLCAQDNPMNPKKYLGSFYTDALVHDPLSLKLLTDVIGKDKVILGTDYPFPLGELEPGKLIESMEEFDEETKNKLKAGNALAFLGLER 4ih3 F 2.493 BS02 PDC F 1 R47 P77 H174 W191 D291 L296 R47 P77 H174 W191 D291 L296 4.1.1.45 0001760,0005515,0005737,0005829,0006569,0008270,0016787,0016831,0019748,0046872,1904985,1905004,1905012 remove_due_to_license_issue Q8TDX5 25392945 402 MKIDIHSHILPKEWPDLKKRFGYGGWVQLQHHSKGEAKLLKDGKVFRVVRENCWDPEVRIREMDQKGVTVQALSTVPVMFSYWAKPEDTLNLCQLLNNDLASTVVSYPRRFVGLGTLPMQAPELAVKEMERCVKELGFPGVQIGTHVNEWDLNAQELFPVYAAAERLKCSLFVHPWDMQMDGRMAKYWLPWLVGMPAETTIAICSMIMGGVFEKFPKLKVCFAHGGGAFPFTVGRISHGFSMRPDLCAQDNPMNPKKYLGSFYTDALVHDPLSLKLLTDVIGKDKVILGTDYPFPLGELEPGKLIESMEEFDEETKNKLKAGNALAFLGLER 4ih5 A 1.9 BS01 12R A 1 L384 N411 M414 Y415 Q446 I447 Y448 L379 N406 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=78uM remove_due_to_license_issue P26663 23509929 601 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4ih6 A 2.2 BS01 1EP A 1 R200 S368 G410 N411 M414 Y415 Q446 I447 Y448 R195 S363 G405 N406 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=18uM remove_due_to_license_issue P26663 23509929 601 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4ih7 A 2.3 BS01 1ER A 1 R200 C366 S368 G410 M414 Y415 Q446 I447 Y448 R195 C361 S363 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 Kd=5.8uM remove_due_to_license_issue P26663 23509929 602 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4ihv A 2.716 BS01 dna C 0 N84 T87 N77 T80 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihv A 2.716 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihv B 2.716 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihv B 2.716 BS02 dna D 0 I83 N84 T87 K90 I83 N84 T87 K90 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihw A 2.7 BS01 dna C 0 N84 T87 N77 T80 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihw A 2.7 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihw B 2.7 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihw B 2.7 BS02 dna D 0 N84 T87 K90 N84 T87 K90 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihx A 2.8 BS01 dna C 0 N84 T87 K90 N77 T80 K83 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihx A 2.8 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihx B 2.8 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihx B 2.8 BS02 dna D 0 I83 N84 T87 K90 I83 N84 T87 K90 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihy A 2.9 BS01 dna C 0 N84 T87 K90 N77 T80 K83 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihy A 2.9 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihy B 2.9 BS01 dna C 0 Q74 T75 R85 R89 Q74 T75 R85 R89 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ihy B 2.9 BS02 dna D 0 N84 T87 K90 N84 T87 K90 0003677,0006355,0043565 remove_due_to_license_issue 23661683 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 4ii9 A 1.66 BS03 UDP B 1 K36 W39 F70 Y103 I142 R211 K36 W39 F70 Y103 I142 R211 K36 D108 R211 F304 K305 E319 K36 D108 R211 F304 K305 E319 2.3.2.10 0008360,0009252,0016746,0016755,0044038,0047206,0071555 remove_due_to_license_issue Q9EY50 23744707 101 PVLNLNDPQAVERYEEFMRQSPYGQVTQDLGWAKVKNNWEPVDVYLEDDQGAIIAAMSMLLGDTPTDKKFAYASKGPVMDVTDVDLLDRLVDEAVKALDGRAYVLRFDPEVAYSDEFNTTLQDHGYVTRNRNVADAGMHATIQPRLNMVLDLTKFPDAKTTLDLYPSKTKSKIKRPFRDGVEVHSGNSATELDEFFKTYTTMAERHGITHRPIEYFQRMQAAFDADTMRIFVAEREGKLLSTGIALKYGRKIWYMYAGSMDGNTYYAPYAVQSEMIQWALDTNTDLYDLGGIESESTDDSLYVFKHVFVKDAPREYIGEIDKVLDPEVYAELVKDGH 4iic A 1.9 BS08 IFM A 1 V74 D92 R156 K189 H190 M245 Y248 D280 W281 S451 E509 V53 D71 R135 K168 H169 M224 Y227 D259 W260 S430 E488 D280 A507 D259 A486 3.2.1.21 0004553,0005975,0008422,0009251,0016798,0030245 Ki=14uM remove_due_to_license_issue P48825 23537284 944 LAFSPPFYPSPWANGQGEWAEAYQRAVAIVSQMTLDEKVNLTTGTGWELEKCVGQTGGVPRLNIGGMCLQDSPLGIRDSDYNSAFPAGVNVAATWDKNLAYLRGQAMGQEFSDKGIDVQLGPAAGPLGRSPDGGRNWEGFSPDPALTGVLFAETIKGIQDAGVVATAKHYILNEQEHFRQVAEAAGYGFNISDTISSNVDDKTIHEMYLWPFADAVRAGVGAIMCSYNQINNSYGCQNSYTLNKLLKAELGFQGFVMSDWGAHHSGVGSALAGLDMSMPGDITFDSATSFWGTNLTIAVLNGTVPQWRVDDMAVRIMAAYYKVGRDRLYQPPNFSSWTRDEYGFKYFYPQEGPYEKVNHFVNVQRNHSEVIRKLGADSTVLLKNNNALPLTGKERKVAILGEDAGSNSYGANGCSDRGCDNGTLAMAWGSGTAEFPYLVTPEQAIQAEVLKHKGSVYAITDNWALSQVETLAKQASVSLVFVNSDAGEGYISVDGNEGDRNNLTLWKNGDNLIKAAANNCNNTIVVIHSVGPVLVDEWYDHPNVTAILWAGLPGQESGNSLADVLYGRVNPGAKSPFTWGKTREAYGDYLVRELNNGNGAPQDDFSEGVFIDYRGFDKRNETPIYEFGHGLSYTTFNYSGLHIQVLNVATETGAAPTFGQVGNASDYVYPEGLTRISKFIYPWLNSTDLKASSGDPYYGVDTAEHVPEGATDGSPQPVLPAGGGSGGNPRLYDELIRVSVTVKNTGRVAGDAVPQLYVSLGGPNEPKVVLRKFDRLTLKPSEETVWTTTLTRRDLSNWDVAAQDWVITSYPKKVHVGSSSRQLPLHAALPKVQ 4iid A 2.3 BS06 NOJ A 1 D92 R156 K189 H190 Y248 D280 W281 E509 D71 R135 K168 H169 Y227 D259 W260 E488 D280 A507 D259 A486 3.2.1.21 0004553,0005975,0008422,0009251,0016798,0030245 Ki=2.4uM remove_due_to_license_issue P48825 23537284 940 LAFSPPFYPSPWANGQGEWAEAYQRAVAIVSQMTLDEKVNLTTGTGWELEKCVGQTGGVPRLNIGGMCLQDSPLGIRDSDYNSAFPAGVNVAATWDKNLAYLRGQAMGQEFSDKGIDVQLGPAAGPLGRSPDGGRNWEGFSPDPALTGVLFAETIKGIQDAGVVATAKHYILNEQEHFRQVAEAAGYGFNISDTISSNVDDKTIHEMYLWPFADAVRAGVGAIMCSYNQINNSYGCQNSYTLNKLLKAELGFQGFVMSDWGAHHSGVGSALAGLDMSMPGDITFDSATSFWGTNLTIAVLNGTVPQWRVDDMAVRIMAAYYKVGRDRLYQPPNFSSWTRDEYGFKYFYPQEGPYEKVNHFVNVQRNHSEVIRKLGADSTVLLKNNNALPLTGKERKVAILGEDAGSNSYGANGCSDRGCDNGTLAMAWGSGTAEFPYLVTPEQAIQAEVLKHKGSVYAITDNWALSQVETLAKQASVSLVFVNSDAGEGYISVDGNEGDRNNLTLWKNGDNLIKAAANNCNNTIVVIHSVGPVLVDEWYDHPNVTAILWAGLPGQESGNSLADVLYGRVNPGAKSPFTWGKTREAYGDYLVRELNNGNGAPQDDFSEGVFIDYRGFDKRNETPIYEFGHGLSYTTFNYSGLHIQVLNAVATETGAAPTFGQVGNASDYVYPEGLTRISKFIYPWLNSTDLKASSGDPYYGVDTAEHVPEGATDGSPQPVLPAGGGSGGNPRLYDELIRVSVTVKNTGRVAGDAVPQLYVSLGGPNEPKVVLRKFDRLTLKPSEETVWTTTLTRRDLSNWDVAAQDWVITSYPKKVHVGSSSRQLPLHAALPKVQ 4iie A 2.0 BS07 CGB A 1 D92 R156 K189 H190 M245 Y248 D280 S451 E509 D71 R135 K168 H169 M224 Y227 D259 S430 E488 D280 A507 D259 A486 3.2.1.21 0004553,0005975,0008422,0009251,0016798,0030245 Ki=4600uM remove_due_to_license_issue P48825 23537284 943 LAFSPPFYPSPWANGQGEWAEAYQRAVAIVSQMTLDEKVNLTTGTGWELEKCVGQTGGVPRLNIGGMCLQDSPLGIRDSDYNSAFPAGVNVAATWDKNLAYLRGQAMGQEFSDKGIDVQLGPAAGPLGRSPDGGRNWEGFSPDPALTGVLFAETIKGIQDAGVVATAKHYILNEQEHFRQVAEAAGYGFNISDTISSNVDDKTIHEMYLWPFADAVRAGVGAIMCSYNQINNSYGCQNSYTLNKLLKAELGFQGFVMSDWGAHHSGVGSALAGLDMSMPGDITFDSATSFWGTNLTIAVLNGTVPQWRVDDMAVRIMAAYYKVGRDRLYQPPNFSSWTRDEYGFKYFYPQEGPYEKVNHFVNVQRNHSEVIRKLGADSTVLLKNNNALPLTGKERKVAILGEDAGSNSYGANGCSDRGCDNGTLAMAWGSGTAEFPYLVTPEQAIQAEVLKHKGSVYAITDNWALSQVETLAKQASVSLVFVNSDAGEGYISVDGNEGDRNNLTLWKNGDNLIKAAANNCNNTIVVIHSVGPVLVDEWYDHPNVTAILWAGLPGQESGNSLADVLYGRVNPGAKSPFTWGKTREAYGDYLVRELNNGNGAPQDDFSEGVFIDYRGFDKRNETPIYEFGHGLSYTTFNYSGLHIQVLNAVATETGAAPTFGQVGNASDYVYPEGLTRISKFIYPWLNSTDLKASSGDPYYGVDTAEHVPEGATDGSPQPVLPAGGGSGGNPRLYDELIRVSVTVKNTGRVAGDAVPQLYVSLGGPNEPKVVLRKFDRLTLKPSEETVWTTTLTRRDLSNWDVAAQDWVITSYPKKVHVGSSSRQLPLHAALPKVQ 4iif A 2.45 BS05 CTS A 1 D92 R156 K189 H190 Y248 D280 W281 S451 E509 D71 R135 K168 H169 Y227 D259 W260 S430 E488 D280 A507 D259 A486 3.2.1.21 0004553,0005975,0008422,0009251,0016798,0030245 Ki=6.6uM remove_due_to_license_issue P48825 23537284 941 LAFSPPFYPSPWANGQGEWAEAYQRAVAIVSQMTLDEKVNLTTGTGWELEKCVGQTGGVPRLNIGGMCLQDSPLGIRDSDYNSAFPAGVNVAATWDKNLAYLRGQAMGQEFSDKGIDVQLGPAAGPLGRSPDGGRNWEGFSPDPALTGVLFAETIKGIQDAGVVATAKHYILNEQEHFRQVAEAAGYGFNISDTISSNVDDKTIHEMYLWPFADAVRAGVGAIMCSYNQINNSYGCQNSYTLNKLLKAELGFQGFVMSDWGAHHSGVGSALAGLDMSMPGDITFDSATSFWGTNLTIAVLNGTVPQWRVDDMAVRIMAAYYKVGRDRLYQPPNFSSWTRDEYGFKYFYPQEGPYEKVNHFVNVQRNHSEVIRKLGADSTVLLKNNNALPLTGKERKVAILGEDAGSNSYGANGCSDRGCDNGTLAMAWGSGTAEFPYLVTPEQAIQAEVLKHKGSVYAITDNWALSQVETLAKQASVSLVFVNSDAGEGYISVDGNEGDRNNLTLWKNGDNLIKAAANNCNNTIVVIHSVGPVLVDEWYDHPNVTAILWAGLPGQESGNSLADVLYGRVNPGAKSPFTWGKTREAYGDYLVRELNNGNGAPQDDFSEGVFIDYRGFDKRNETPIYEFGHGLSYTTFNYSGLHIQVLNAVATETGAAPTFGQVGNASDYVYPEGLTRISKFIYPWLNSTDLKASSGDPYYGVDTAEHVPEGATDGSPQPVLPAGGGSGGNPRLYDELIRVSVTVKNTGRVAGDAVPQLYVSLGGPNEPKVVLRKFDRLTLKPSEETVWTTTLTRRDLSNWDVAAQDWVITSYPKKVHVGSSSRQLPLHAALPKV 4ij1 A 1.79 BS01 17C A 1 N138 P180 H183 Y186 R187 A190 R193 N110 P145 H148 Y151 R152 A155 R158 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 Ki=4uM remove_due_to_license_issue P9WFX5 24623674 401 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGTVNLSTMAAIVVAAAGVPVVKHGNRAADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4ijh A 1.498 BS01 1EJ A 1 R31 I33 T34 R43 S55 M57 L87 D89 R91 V93 R34 I36 T37 R46 S58 M60 L90 D92 R94 V96 ? 0003677,0005634,0006260 Kd=47uM remove_due_to_license_issue P27694 23914285 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4ijh A 1.498 BS02 1EJ A 2 R41 L87 K88 V93 R44 L90 K91 V96 ? 0003677,0005634,0006260 Kd=47uM remove_due_to_license_issue P27694 23914285 204 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4ijh A 1.498 BS03 1EJ A 3 R43 R91 R46 R94 ? 0003677,0005634,0006260 Kd=47uM remove_due_to_license_issue P27694 23914285 205 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4ijl A 1.7 BS01 1EK A 1 R41 A59 T60 N85 R43 A61 T62 N87 ? 0003677,0005634,0006260 Kd=135uM remove_due_to_license_issue Kd=135000nM P27694 23914285 201 SHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4ijl A 1.7 BS02 1EK A 2 R31 R43 S55 V93 R33 R45 S57 V95 ? 0003677,0005634,0006260 Kd=135uM remove_due_to_license_issue Kd=135000nM P27694 23914285 202 SHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4ijp A 2.25 BS01 1EH A 1 T693 V701 A715 K717 L751 F767 L770 S771 M772 E776 L822 T24 V32 A46 K48 L82 F98 L101 S102 M103 E107 L153 D815 K817 N820 D834 S852 D146 K148 N151 D165 S183 2.7.11.1 0004672,0004674,0005524,0006468,0045292 ic50=0.016uM remove_due_to_license_issue IC50=16nM Q13523 24003220 1101 DAEGYYRVNIGEVLDKRYNVYGYTGQGVFSNVVRARDNARANQEVAVKIIRNNELMQKTGLKELEFLKKLNDADPDDKFHCLRLFRHFYHKQHLCLVFEPLSMNLREVLKKYGKDVGLHIKAVRSYSQQLFLALKLLKRCNILHADIKPDNILVNESKTILKLCDFGSASHVADNDITPYLVSRFYRAPEIIIGKSYDYGIDMWSVGCTLYELYTGKILFPGKTNNHMLKLAMDLKGKMPNKMIRKGVFKDQHFDQNLNFMYIEVDEREKVTVMSTINPTKDLLADLIQRLPEDQRKKVHQLKDLLDQILMLDPAKRISINQALQHAFIQE 4ijq A 2.004 BS01 SV2 A 1 K102 I135 D137 T138 G139 T141 K165 F186 V187 K99 I116 D118 T119 G120 T122 K146 F167 V168 E133 D134 D137 F186 R199 E114 D115 D118 F167 R180 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.03uM remove_due_to_license_issue P00492 23448281 301 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4ikr A 1.78 BS03 PVP A 1 Y195 Y196 F198 C203 H212 H310 W353 Y106 Y107 F109 C114 H123 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=0.59uM remove_due_to_license_issue IC50=1100nM P53582 23767698 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4iks A 1.7 BS01 TFD A 1 Y195 Y196 F198 C203 H212 Y300 H310 W353 Y106 Y107 F109 C114 H123 Y211 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=7.23uM remove_due_to_license_issue IC50=1000nM P53582 23767698 401 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4ikt A 1.6 BS01 TFV A 1 Y195 H212 H310 T311 N314 W353 Y106 H123 H221 T222 N225 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=0.67uM remove_due_to_license_issue IC50=2000nM, EC50=280nM P53582 23767698 401 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4iku A 1.3 BS01 SHX A 1 Y195 H212 Y300 H310 W353 Y106 H123 Y211 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=1.79uM remove_due_to_license_issue P53582 23767698 401 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4im0 A 2.4001 BS01 1FV A 1 L15 V23 A36 K38 V68 M86 E87 F88 C89 G92 M142 T156 D157 L17 V25 A38 K40 V66 M84 E85 F86 C87 G90 M140 T154 D155 N135 K137 N140 D157 T176 N133 K135 N138 D155 T158 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue Kd=79nM Q9UHD2 23453972 701 GSMQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFNNRPVDVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRNIKPGNIMRVIGEDGQSVYKLTDFGTEEYLHPDMYERVLRKDHATVDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVKVMEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 4inb A 1.8 BS01 1F6 A 1 W23 V27 E28 A31 F32 S33 V36 F40 V59 G61 H62 A65 L138 I141 V142 W23 V27 E28 A31 F32 S33 V36 F40 V59 G61 H62 A65 L138 I141 V142 ? 0016032 ic50=0.89uM remove_due_to_license_issue A9PKC6 23401268 201 PIVQNLQGQMVHQAISPRTLNAWVKVVEEKAFSPEVIPMFSALSEGATPQDLNTMLNTVGGHQAAMQMLKETINEEAAEWDRLHPVHAGPIAPGQMREPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYS 4inr H 2.7 BS01 1G1 H 1 T1 T21 K33 G47 A49 T1 T21 K33 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 23320547 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4inr I 2.7 BS01 1G1 H 1 D124 I126 D124 I126 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 23320547 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4inr Z 2.7 BS01 1G1 Y 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 23320547 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4int H 2.9 BS01 1G5 H 1 T1 T21 Q22 C31 K33 G47 A49 S129 T1 T21 Q22 C31 K33 G47 A49 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 23320547 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4int I 2.9 BS01 1G5 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 23320547 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4int Z 2.9 BS01 1G5 Y 1 D126 V128 D126 V128 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 23320547 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4inu H 3.1 BS01 1G6 H 1 T1 S20 T21 Q22 A27 K33 G47 A49 T52 S129 T1 S20 T21 Q22 A27 K33 G47 A49 T52 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 23320547 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4inu I 3.1 BS01 1G6 H 1 F123 D124 L125 I126 C128 D130 F123 D124 L125 I126 C128 D130 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 23320547 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4inu Z 3.1 BS01 1G6 Y 1 D126 P127 S130 R137 D126 P127 S130 R137 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 23320547 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4io2 A 1.37 BS02 GLU A 1 Y67 I86 T87 R92 R136 T139 D180 Y61 I80 T81 R86 R130 T133 D174 ? 0015276,0016020 Kd=203nM remove_due_to_license_issue E9P5T5 23434404 303 GSARLKGITLRIGVIESVPFTIVANVNTTKLTGYVLDLIEYLRDKMGFVADVQLAPPNTSYTGLVLALANGDYDIAIGDITVTSARREIVAFSNSISDNSMRILMRKGTLIDGMDDLKNGKIPYNRIGIRIGTAGEDYYLREISGGSRNFYPLKSRQEMYDSLLAGIIDVSFMDIGTAEYVTNNIYCNLTLVGEDFDKSTFGIVTPKEWLYAKDLDVNILSLRETGILDNLKKKWFQTKACP 4io3 A 1.66 BS01 ASP A 1 Y67 I86 T87 R92 R136 T139 R162 D180 Y61 I80 T81 R86 R130 T133 R156 D174 ? 0015276,0016020 Kd=875nM remove_due_to_license_issue E9P5T5 23434404 301 GSARLKGITLRIGVIESVPFTIVANVNTTKLTGYVLDLIEYLRDKMGFVADVQLAPPNTSYTGLVLALANGDYDIAIGDITVTSARREIVAFSNSISDNSMRILMRKGTLIDGMDDLKNGKIPYNRIGIRIGTAGEDYYLREISGGSRNFYPLKSRQEMYDSLLAGIIDVSFMDIGTAEYVTNNIYCNLTLVGEDFDKSTFGIVTPKEWLYAKDLDVNILSLRETGILDNLKKKWFQTKACP 4io4 A 1.941 BS01 SER A 1 Y67 T87 R92 T139 D180 Y63 T83 R88 T135 D176 ? 0015276,0016020 Kd=24uM remove_due_to_license_issue E9P5T5 23434404 301 SARLKGITLRIGVIESVPFTIVANVIDRNTTKLTGYVLDLIEYLRDKMGFVADVQLAPPNTSYTGLVLALANGDYDIAIGDITVTSARREIVAFSNSISDNSMRILMRKGTLIDGMDDLKNGKIPYNRIGIRIGTAGEDYYLREISGGSRNFYPLKSRQEMYDSLLAGIIDVSFMDIGTAEYVTNNIYCNLTLVGEDFDKSTFGIVTPKEWLYAKDLDVNILSLRETGILDNLKKKWFQTKACP 4io5 A 1.721 BS01 ALA A 1 Y67 I86 T87 R92 T139 D180 Y61 I80 T81 R86 T133 D174 ? 0015276,0016020 Kd=9uM remove_due_to_license_issue E9P5T5 23434404 301 GSARLKGITLRIGVIESVPFTIVANVNTTKLTGYVLDLIEYLRDKMGFVADVQLAPPNTSYTGLVLALANGDYDIAIGDITVTSARREIVAFSNSISDNSMRILMRKGTLIDGMDDLKNGKIPYNRIGIRIGTAGEDYYLREISGGSRNFYPLKSRQEMYDSLLAGIIDVSFMDIGTAEYVTNNIYCNLTLVGEDFDKSTFGIVTPKEWLYAKDLDVNILSLRETGILDNLKKKWFQTKACP 4io6 A 1.6 BS01 MET A 1 Y67 T87 R92 T139 M179 D180 Y62 T82 R87 T134 M174 D175 ? 0015276,0016020 Kd=15uM remove_due_to_license_issue E9P5T5 23434404 301 GSARLKGITLRIGVIESVPFTIVANVINTTKLTGYVLDLIEYLRDKMGFVADVQLAPPNTSYTGLVLALANGDYDIAIGDITVTSARREIVAFSNSISDNSMRILMRKGTLIDGMDDLKNGKIPYNRIGIRIGTAGEDYYLREISGGSRNFYPLKSRQEMYDSLLAGIIDVSFMDIGTAEYVTNNIYCNLTLVGEDFDKSTFGIVTPKEWLYAKDLDVNILSLRETGILDNLKKKWFQTKACP 4io7 A 1.92 BS01 PHE A 1 Y67 D85 T87 R92 T139 D180 Y63 D81 T83 R88 T135 D176 ? 0015276,0016020 remove_due_to_license_issue E9P5T5 23434404 301 GSARLKGITLRIGVIESVPFTIVANVIRNTTKLTGYVLDLIEYLRDKMGFVADVQLAPPNTSYTGLVLALANGDYDIAIGDITVTSARREIVAFSNSISDNSMRILMRKGTLIDGMDDLKNGKIPYNRIGIRIGTAGEDYYLREISGGSRNFYPLKSRQEMYDSLLAGIIDVSFMDIGTAEYVTNNIYCNLTLVGEDFDKSTFGIVTPKEWLYAKDLDVNILSLRETGILDNLKKKWFQTKACP 4io8 A 2.58 BS01 3FD A 1 Y15 T37 G202 E268 K271 R272 S275 G339 R342 D366 Y13 T35 G200 E266 K269 R270 S273 G337 R340 D364 D10 K71 E175 D199 D8 K69 E173 D197 ? 0005524,0140662 remove_due_to_license_issue Kd=3e+2nM, Ki=1.2e+2nM, IC50=500nM P0DMV8 24265689 401 KAAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGDTKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAI 4ipf A 1.7 BS01 1F0 A 1 L50 L53 I57 M58 Q68 H69 F87 V89 H92 Y96 L30 L33 I37 M38 Q48 H49 F67 V69 H72 Y76 2.3.2.27 0005634,0043066,0051726 ic50=18nM remove_due_to_license_issue P56273 23400593 201 EKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4iq6 A 3.12 BS01 IQ6 A 1 G63 F67 A83 K85 D133 Y134 V135 L188 C199 D200 G27 F31 A47 K49 D89 Y90 V91 L144 C155 D156 D181 K183 N186 D200 S219 D137 K139 N142 D156 S175 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue Ki=58nM P49841 24900653 501 VTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 4iqr A 2.9 BS01 dna C 0 K61 H62 Y63 K72 R76 R80 Q122 K13 H14 Y15 K24 R28 R32 Q74 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 3001 ~ 3020 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNEINALLQAEVLSRQITSPVSGINGDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr A 2.9 BS02 dna D 0 D69 G70 F74 R77 H83 R100 N101 R104 D21 G22 F26 R29 H35 R52 N53 R56 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 4000 ~ 4019 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNEINALLQAEVLSRQITSPVSGINGDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr B 2.9 BS01 dna C 0 H62 Y63 K72 R76 R80 Q122 E124 R125 R127 S129 H14 Y15 K24 R28 R32 Q74 E76 R77 R79 S81 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 3001 ~ 3020 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNERDRISTRRSSYEDSSLPSINALLQAEVLSDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr B 2.9 BS02 dna D 0 D69 G70 R77 R100 N101 R104 R107 R125 I128 D21 G22 R29 R52 N53 R56 R59 R77 I80 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 4000 ~ 4019 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNERDRISTRRSSYEDSSLPSINALLQAEVLSDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr E 2.9 BS01 dna G 0 K61 H62 Y63 R76 R80 Q122 K13 H14 Y15 R28 R32 Q74 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 3001 ~ 3020 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNPSINALLQAEVLSRQITSPVSGINGDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr E 2.9 BS02 dna H 0 D69 G70 R77 H83 R100 N101 R104 R107 D21 G22 R29 H35 R52 N53 R56 R59 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 4000 ~ 4019 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNPSINALLQAEVLSRQITSPVSGINGDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr F 2.9 BS01 dna G 0 Y63 R76 R80 Q122 E124 R125 R127 I128 S129 Y15 R28 R32 Q74 E76 R77 R79 I80 S81 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 3001 ~ 3020 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNERDRISTRRSSYEDSSLPSINALLQAEVLSRSGINGDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqr F 2.9 BS02 dna H 0 D69 G70 R77 R100 N101 R104 R125 I128 D21 G22 R29 R52 N53 R56 R77 I80 ? 0000978,0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P41235 23485969 4000 ~ 4019 ALCAICGDRATGKHYGASSCDGCKGFFRRSVRKNHMYSCRFSRQCVVDKDKRNQCRYCRLKKCFRAGMKKEAVQNERDRISTRRSSYEDSSLPSINALLQAEVLSRSGINGDIRAKKIASIADVCESMKEQLLVLVEWAKYIPAFCELPLDDQVALLRAHAGEHLLLGATKRSMVFKDVLLLGNDYIVPRHCPELAEMSRVSIRILDELVLPFQELQIDDNEYAYLKAIIFFDPDAKGLSDPGKIKRLRSQVQVSLEDYINDRQYDSRGRFGELLLLLPTLQSITWQMIEQIQFIKLFGMAKIDNLLQEMLLGG 4iqt A 2.6 BS01 1FO A 1 M192 T331 G332 G333 F334 R336 D343 D345 S453 R454 Q455 R458 M44 T183 G184 G185 F186 R188 D195 D197 S299 R300 Q301 R304 D343 D345 D434 D195 D197 D280 2.7.7.31,3.1.11.- 0003677,0003887,0006281,0016779,0034061 remove_due_to_license_issue P09838 23968551 601 KISQYACQRRTTLNNYNQLFTDALDILAENDELRENEGSCLAFMRASSVLKSLPFPITSMKDTEGIPCLGDKVKSIIEGIIEDGESSEAKAVLNDERYKSFKLFTSVFGVGLKTAEKWFRMGFRTLSKIQSDKSLRFTQMQKAGFLYYEDLVSCVNRPEAEAVSMLVKEAVVTFLPDALVTMTGGFRRGKMTGHDVDFLITSPEATEDEEQQLLHKVTDFWKQQGLLLYCDILESTFEKFKQPSRDALDHFQKCFLILKLDHGRVHSEKEGKGWKAIRVDLVMCPYDRRAFALLGWTGSRQFERDLRRYATHERKMMLDNHALYDRTKRVFLEAESEEEIFAHLGLDYIEPWERNA 4iqu A 2.4 BS01 1FQ A 1 R336 W450 S453 R454 Q455 A510 R188 W298 S301 R302 Q303 A358 D343 D345 D434 D195 D197 D282 2.7.7.31,3.1.11.- 0003677,0003887,0006281,0016779,0034061 remove_due_to_license_issue P09838 23968551 602 KISQYACQRRTTLNNYNQLFTDALDILAENDELRENEGSCLAFMRASSVLKSLPFPITSMKDTEGIPCLGDKVKSIIEGIIEDGESSEAKAVLNDERYKSFKLFTSVFGVGLKTAEKWFRMGFRTLSKIQSDKSLRFTQMQKAGFLYYEDLVSCVNRPEAEAVSMLVKEAVVTFLPDALVTMTGGFRRGKMTGHDVDFLITSPEATEDEEQQLLHKVTDFWKQQGLLLYCDILESTFEKFKQPSRKVDALDHFQKCFLILKLDHGRVHSEKEGKGWKAIRVDLVMCPYDRRAFALLGWTGSRQFERDLRRYATHERKMMLDNHALYDRTKRVFLEAESEEEIFAHLGLDYIEPWERNA 4ir5 A 1.7 BS01 IR5 A 1 P1888 V1893 N1894 L1897 V1898 N1944 I1950 P33 V38 N39 L42 V43 N89 I95 ? remove_due_to_license_issue IC50=610nM Q9UIF8 25799074 2013 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 4ir6 A 1.8 BS01 IR6 A 1 W1887 P1888 P1892 V1893 V1898 I1950 W32 P33 P37 V38 V43 I95 ? remove_due_to_license_issue IC50=840nM Q9UIF8 25799074 2007 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 4iri A 2.77 BS01 dna B 0 Y345 R350 R353 Y356 K363 R368 Y369 Y54 R59 R62 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P11308 23898196 1 ~ 12 GQIQLWQFLLELLSDSSNSSCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQPH 4iri A 2.77 BS02 dna C 0 Q295 W334 K338 M343 K347 R350 Y354 Y355 K358 Q4 W43 K47 M52 K56 R59 Y63 Y64 K67 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P11308 23898196 13 ~ 24 GQIQLWQFLLELLSDSSNSSCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQPH 4irx A 1.451 BS01 INS A 1 Q49 F51 D125 R126 N168 D169 S174 R178 S203 N231 D258 Q278 Q20 F22 D96 R97 N139 D140 S145 R149 S174 N202 D229 Q249 ? Kd=0.76uM remove_due_to_license_issue A0A0H3C834 23504019 401 GLVPRGSHMEVVVSFNDLSQPFFVAMRRELEDEAAKLGVKVQVLDAQNNSSKQISDLQAAAVQGAKVVIVAPTDSKALAGAADDLVEQGVAVISVDRNIAGGKTAVPHVGADNVAGGRAMADWVVKTYPAGARVVVITNDPGSSSSIERVKGVHDGLAAGGPAFKIVTEQTANSKRDQALTVTQNILTSMRDTPPDVILCLNDDMAMGALEAVRAAGLDSAKVKVIGFDAIPEALARIKAGEMVATVEQNPGLQIRTALRQAVDKIKSGAALKSVSLKPVLITSGNLTEASRIGEM 4is1 C 2.1 BS01 dna A 0 F480 R481 Y485 H489 T492 Y506 Q510 T512 S513 Y516 F10 R11 Y15 H19 T22 Y36 Q40 T42 S43 Y46 ? remove_due_to_license_issue O75362 23436653 1 ~ 20 RECSYCGKFFRSNYYLNIHLRTHTGEKPYKCEFCEYAAAQKTSLRYHLERHH 4is1 C 2.1 BS02 dna B 0 Y484 K511 T512 R515 Y14 K41 T42 R45 ? remove_due_to_license_issue O75362 23436653 1 ~ 20 RECSYCGKFFRSNYYLNIHLRTHTGEKPYKCEFCEYAAAQKTSLRYHLERHH 4is1 D 2.1 BS01 dna A 0 Y484 T512 R515 Y15 T43 R46 ? remove_due_to_license_issue O75362 23436653 1 ~ 20 SRECSYCGKFFRSNYYLNIHLRTHTGEKPYKCEFCEYAAAQKTSLRYHLERHHK 4is1 D 2.1 BS02 dna B 0 R481 Y485 H489 T492 Y506 Q510 T512 S513 Y516 R12 Y16 H20 T23 Y37 Q41 T43 S44 Y47 ? remove_due_to_license_issue O75362 23436653 1 ~ 20 SRECSYCGKFFRSNYYLNIHLRTHTGEKPYKCEFCEYAAAQKTSLRYHLERHHK 4ish H 1.82 BS01 1GE H 1 H57 D189 S190 C191 K192 S195 S214 W215 G216 G219 H41 D186 S187 C188 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=1.9nM remove_due_to_license_issue Ki=1.9nM P08709 23478148 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4isi H 1.94 BS01 1GG H 1 H57 T98 T99 D189 S190 C191 S195 V213 W215 G216 Q217 G219 H41 T86 T87 D186 S187 C188 S192 V210 W212 G213 Q214 G215 3.4.21.21 0004252,0006508 Ki=7.3nM remove_due_to_license_issue P08709 23416003 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4isu A 2.3 BS01 IKM A 1 Y61 T91 R96 L138 G141 S142 T174 E193 Y220 Y58 T88 R93 L135 G138 S139 T171 E190 Y217 ? 0015276,0016020 Ki=0.21mM remove_due_to_license_issue P19491 23432124 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4ith A 2.25 BS01 RCM A 1 M67 L70 V75 V76 M92 H136 I154 A155 D156 S161 F162 M39 L42 V47 V48 M64 H108 I126 A127 D128 S133 F134 D138 K140 E142 N143 D156 T189 D110 K112 E114 N115 D128 T142 2.7.11.1 0004672,0005524,0006468 ic50=0.3169uM remove_due_to_license_issue IC50=200nM, EC50=18nM Q13546 23473668 307 NVIKMKSSDFLVSLAFHRTQGLMIMKTVNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 4iti A 2.86 BS01 1HW A 1 A64 M67 V76 L78 L90 M92 H136 I154 A155 D156 L157 S161 F162 A57 M60 V69 L71 L83 M85 H129 I147 A148 D149 L150 S154 F155 D138 K140 E142 N143 D156 T189 D131 K133 E135 N136 D149 T172 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13546 23473668 301 NVIKMKSSDFLESAELDSGGFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELGGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 4itj A 1.8 BS01 1HX A 1 M67 L70 V76 L78 M92 I154 A155 D156 S161 F162 M52 L55 V61 L63 M77 I139 A140 D141 S146 F147 D138 K140 E142 N143 D156 T189 D123 K125 E127 N128 D141 T156 2.7.11.1 0004672,0005524,0006468 ic50=0.3772uM remove_due_to_license_issue Q13546 23473668 301 NVIKMKSSDFLEFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 4itp A 1.697 BS02 1GD A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=54nM remove_due_to_license_issue Ki=54nM P00918 24012377 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4iu0 A 1.77 BS03 ABH A 1 D137 H139 D141 S150 H154 D243 E288 D125 H127 D129 S138 H142 D231 E276 H114 D137 H139 D141 H154 D243 D245 E288 H102 D125 H127 D129 H142 D231 D233 E276 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Ki=1.3uM remove_due_to_license_issue Q6TUJ5 23583962 403 KKMSIVLAPFSGGQPHSGVELGPDYLLKQGLQQDMEKLGWDTRLERVFDGKVVEARKASDNGDRIGRVKRPRLTAECTEKIYKCVRRVAEQGRFPLTIGGDHSIALGTVAGVLSVHPDAGVIWVDAHADINTMSGTVSGNLHGCPLSILLGLDRENIPECFSWVPQVLKPNKIAYIGLRAVDDEEKKILHDLNIAAFSMHHVDRYGIDKVVSMAIEAVSPKGTEPVMVSYDVDTIDPLYVPATGTPVRGGLSFREALFLCERIAECGRLVALDVVECNPLLAATESHVNDTISVGCAIARCMMGETLLYT 4iu1 A 1.95 BS03 NNH A 1 H139 D141 N143 S150 H154 D194 T257 H127 D129 N131 S138 H142 D182 T245 H114 D137 H139 D141 H154 D243 D245 E288 H102 D125 H127 D129 H142 D231 D233 E276 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Ki~50uM remove_due_to_license_issue Q6TUJ5 23583962 403 KKMSIVLAPFSGGQPHSGVELGPDYLLKQGLQQDMEKLGWDTRLERVFDGKVVEARKASDNGDRIGRVKRPRLTAECTEKIYKCVRRVAEQGRFPLTIGGDHSIALGTVAGVLSVHPDAGVIWVDAHADINTMSGTVSGNLHGCPLSILLGLDRENIPECFSWVPQVLKPNKIAYIGLRAVDDEEKKILHDLNIAAFSMHHVDRYGIDKVVSMAIEAVSPKGTEPVMVSYDVDTIDPLYVPATGTPVRGGLSFREALFLCERIAECGRLVALDVVECNPLLAATESHVNDTISVGCAIARCMMGETLLYT 4iu4 A 1.8 BS03 S2C A 1 D137 H139 D141 S150 H154 D194 D243 D245 E288 D125 H127 D129 S138 H142 D182 D231 D233 E276 H114 D137 H139 D141 H154 D243 D245 E288 H102 D125 H127 D129 H142 D231 D233 E276 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Ki~10uM remove_due_to_license_issue Q6TUJ5 23583962 405 KKMSIVLAPFSGGQPHSGVELGPDYLLKQGLQQDMEKLGWDTRLERVFDGKVVEARKASDNGDRIGRVKRPRLTAECTEKIYKCVRRVAEQGRFPLTIGGDHSIALGTVAGVLSVHPDAGVIWVDAHADINTMSGTVSGNLHGCPLSILLGLDRENIPECFSWVPQVLKPNKIAYIGLRAVDDEEKKILHDLNIAAFSMHHVDRYGIDKVVSMAIEAVSPKGTEPVMVSYDVDTIDPLYVPATGTPVRGGLSFREALFLCERIAECGRLVALDVVECNPLLAATESHVNDTISVGCAIARCMMGETLLYT 4iue A 2.38 BS02 AJ4 A 1 H1031 G1032 P1034 A1049 Y1050 Y1060 S1068 Y1071 I1075 H80 G81 P83 A98 Y99 Y109 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 Kd=0.28uM remove_due_to_license_issue Q9H2K2 23672613 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4iuo A 1.8 BS01 QIC A 1 E46 R48 R82 H143 R213 F225 S232 A233 Q236 E54 R56 R90 H151 R221 F233 S240 A241 Q244 E86 H143 M170 E94 H151 M178 4.2.1.10 0003855,0008652,0009073,0009423,0016829,0046279 remove_due_to_license_issue P58687 24437575 301 NLYFQSNAMKTVTVRDLVVGEGAPKIIVSLMGKTITDVKSEALAYREADFDILEWRVDHFANVTTAESVLEAAGAIREIITDKPLLFTFRSAKEGGEQALTTGQYIDLNRAAVDSGLVDMIDLELFTGDDEVKATVGYAHQHNVAVIMSNHDFHKTPAAEEIVQRLRKMQELGADIPMIAVMPQTKADVLTLLTATVEMQERYADRPIITMSMSKTGVISRLAGEVFGSAATFGAVKKASAPGQISVADLRTVLTILHQ 4iva A 1.5 BS01 1J5 A 1 V863 A880 M929 Y931 L932 S936 L983 D994 V23 A40 M89 Y91 L92 S96 L143 D154 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue O60674 23659214 1201 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4ivb A 1.9 BS01 1J5 A 1 L881 V889 A906 M956 F958 L959 S963 E966 L1010 D1021 L29 V37 A54 M95 F97 L98 S102 E105 L149 D160 D1003 A1005 R1007 N1008 D1021 D1040 D142 A144 R146 N147 D160 D179 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.9nM remove_due_to_license_issue EC50=130nM, Ki=1.9nM P23458 23659214 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4ivc A 2.35 BS01 1J6 A 1 L881 G882 E883 V889 A906 M956 F958 L959 S963 E966 N1008 L1010 G1020 D1021 L29 G30 E31 V37 A54 M95 F97 L98 S102 E105 N147 L149 G159 D160 D1003 A1005 R1007 N1008 D1021 D1040 D142 A144 R146 N147 D160 D179 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.1nM remove_due_to_license_issue EC50=28nM, IC50=<0.200nM, Ki=0.100000nM P23458 23659214 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4ivd A 1.93 BS01 15T A 1 L881 E883 V889 A906 M956 F958 L959 S963 E966 L1010 D1021 L29 E31 V37 A54 M94 F96 L97 S101 E104 L148 D159 D1003 A1005 R1007 N1008 D1021 D1040 D141 A143 R145 N146 D159 D178 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.3nM remove_due_to_license_issue EC50=43nM, Ki=0.300000nM P23458 23659214 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4ivk A 1.8 BS01 CEP A 1 Y99 S100 F174 V175 Y218 I277 Q296 G383 A384 R409 Y75 S76 F150 V151 Y194 I253 Q272 G359 A360 R385 S100 K103 Y172 F174 L189 Y218 D223 M271 W381 A384 S76 K79 Y148 F150 L165 Y194 D199 M247 W357 A360 3.1.1.1 remove_due_to_license_issue K4HQE7 23737193 501 AEGPVTATKPKEAGFTSEGLARIDAYLKNEIQAKTMPGAVMMIKRNGETAYFSSFGLRDPDTKEPMTAETIFRIYSMSKPITTVAAMMLVEEGKLQLDEPVSKYIPSFANVKVGVETKGENGMALETGPVKRAITIQDLMRHTSGITYGFVGDGLVKKAYIASNLFDGDFDNAEFAERIAKLPLVYQPGTTWDYGHSTDILGRVVEVVSGKSLYQFEKERLLDPLGMKDTGFYVTDPAKKSLVAEAMPNDRKIGGSEMFDPRVQKKWEPGGQGMVSTIGDYARFTQMVLNGGTLDGKRYLSPKTIAYMGSNHIPQASGIVPGAYYLPGPGVGFGLGFAVRTEAGVTPVEGSVGDLSWGGAGGTVFWIDPKENLTVVFMAPMVSPRARVWRTLRNIVYGAFDRLE 4ivs A 2.636 BS01 VSI A 1 D32 Y71 T72 F108 W115 D228 T231 R235 D36 Y75 T76 F112 W119 D220 T223 R227 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 23681056 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4ivt A 1.6 BS01 VTI A 1 D32 Y71 T72 Q73 F108 I110 W115 D228 G230 R235 D37 Y76 T77 Q78 F113 I115 W120 D221 G223 R228 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=1.01uM remove_due_to_license_issue P56817 23681056 401 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4ivz A 3.1 BS01 dna C 0 R17 T23 Q24 R35 T36 S39 R43 R16 T22 Q23 R34 T35 S38 R42 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 4ivz A 3.1 BS02 dna D 0 L33 D34 T36 F37 R46 N47 L48 T49 S52 L32 D33 T35 F36 R45 N46 L47 T48 S51 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 4ivz B 3.1 BS01 dna C 0 L33 D34 T36 F37 N47 L48 T49 S52 L32 D33 T35 F36 N46 L47 T48 S51 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 4ivz B 3.1 BS02 dna D 0 R17 T23 Q24 R35 T36 R43 N44 R16 T22 Q23 R34 T35 R42 N43 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 4ivz E 3.1 BS01 dna G 0 R17 T23 Q24 R35 T36 S39 R43 R16 T22 Q23 R34 T35 S38 R42 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILKH 4ivz E 3.1 BS02 dna H 0 L33 D34 T36 F37 N47 L48 T49 S52 L32 D33 T35 F36 N46 L47 T48 S51 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILKH 4ivz F 3.1 BS01 dna G 0 L33 D34 T36 F37 R46 N47 L48 T49 L32 D33 T35 F36 R45 N46 L47 T48 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 4ivz F 3.1 BS02 dna H 0 R17 T23 Q24 R35 S39 R43 N44 R16 T22 Q23 R34 S38 R42 N43 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue Q8GGH0 24887147 1 ~ 19 ESFLLSKVSFVIKKIRLEKGMTQEDLAYKSNLDRTFISGIERNSRNLTIKSLELIMKGLEVSDVVFFEMLIKEILK 4iwd A 1.99 BS01 1JC A 1 I1084 R1086 G1087 H1088 V1092 A1108 L1140 Y1159 M1160 G1163 R1208 N1209 M1211 D1222 I38 R40 G41 H42 V46 A62 L94 Y113 M114 G117 R162 N163 M165 D176 D1204 A1206 R1208 N1209 D1222 D158 A160 R162 N163 D176 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1.000000nM P08581 23379595 1401 MQNTVHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHHHHH 4iwz A 1.598 BS01 1GO A 1 I91 Q92 H94 H96 H119 F131 L198 T199 T200 I88 Q89 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=51nM remove_due_to_license_issue Ki=51nM P00918 23993330 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ixh A 2.105 BS02 Q21 A 1 S22 V24 L25 P26 S354 Y358 S22 V24 L25 P26 S298 Y302 1.1.1.205 0003824,0003938,0006164,0016491 ic50=6.1nM remove_due_to_license_issue IC50=8.0nM, Ki=13nM Q8T6T2 23668331 504 MGTKNIGKGLTFEDILLVPNYSEVLPREVSLETKLTKNVSLKIPLISSAMDTVTEHLMAVGMARLGGIGIIHKNMDMESQVNEVLKVKNSGGLRVGAAIGVNEIERAKLLVEAGVDVIVLDSAHGHSLNIIRTLKEIKSKMNIDVIVGNVVTEEATKELIENGADGIKVGIGPGSICTTRIVAGVGVPQITAIEKCSSVASKFGIPIIADGGIRYSGDIGKALAVGASSVMIGSILAGTEESPGEKELIGDTVYKYYRGMGSVGAMKSGMVPEGIEGRVKYKGEMEGVVYQLVGGLRSCMGYLGSASIEELWKKSSYVEITTSGLRESHVHDVEIV 4ixh A 2.105 BS03 Q21 B 1 A165 S169 M302 G303 M326 E329 A123 S127 M260 G261 M270 E273 1.1.1.205 0003824,0003938,0006164,0016491 ic50=6.1nM remove_due_to_license_issue IC50=8.0nM, Ki=13nM Q8T6T2 23668331 501 MGTKNIGKGLTFEDILLVPNYSEVLPREVSLETKLTKNVSLKIPLISSAMDTVTEHLMAVGMARLGGIGIIHKNMDMESQVNEVLKVKNSGGLRVGAAIGVNEIERAKLLVEAGVDVIVLDSAHGHSLNIIRTLKEIKSKMNIDVIVGNVVTEEATKELIENGADGIKVGIGPGSICTTRIVAGVGVPQITAIEKCSSVASKFGIPIIADGGIRYSGDIGKALAVGASSVMIGSILAGTEESPGEKELIGDTVYKYYRGMGSVGAMKSGMVPEGIEGRVKYKGEMEGVVYQLVGGLRSCMGYLGSASIEELWKKSSYVEITTSGLRESHVHDVEIV 4ixh D 2.105 BS01 Q21 A 1 A165 S169 M302 G303 E329 A122 S126 M259 G260 E271 1.1.1.205 0003824,0003938,0006164,0016491 remove_due_to_license_issue IC50=8.0nM, Ki=13nM Q8T6T2 23668331 504 GTKNIGKGLTFEDILLVPNYSEVLPREVSLETKLTKNVSLKIPLISSAMDTVTEHLMAVGMARLGGIGIIHKNMDMESQVNEVLKVKNSGGLRVGAAIGVNEIERAKLLVEAGVDVIVLDSAHGHSLNIIRTLKEIKSKMNIDVIVGNVVTEEATKELIENGADGIKVGIGPGSICTTRIVAGVGVPQITAIEKCSSVASKFGIPIIADGGIRYSGDIGKALAVGASSVMIGSILAGTEESPGEKELIGDTVYKYYRGMGSVGAMKSMVPEGIEGRVKYKGEMEGVVYQLVGGLRSCMGYLGSASIEELWKKSSYVEITTSGLRESHVHDVEIV 4ixh D 2.105 BS02 Q21 C 1 S22 V24 L25 P26 S354 Y358 S21 V23 L24 P25 S296 Y300 1.1.1.205 0003824,0003938,0006164,0016491 remove_due_to_license_issue IC50=8.0nM, Ki=13nM Q8T6T2 23668331 502 GTKNIGKGLTFEDILLVPNYSEVLPREVSLETKLTKNVSLKIPLISSAMDTVTEHLMAVGMARLGGIGIIHKNMDMESQVNEVLKVKNSGGLRVGAAIGVNEIERAKLLVEAGVDVIVLDSAHGHSLNIIRTLKEIKSKMNIDVIVGNVVTEEATKELIENGADGIKVGIGPGSICTTRIVAGVGVPQITAIEKCSSVASKFGIPIIADGGIRYSGDIGKALAVGASSVMIGSILAGTEESPGEKELIGDTVYKYYRGMGSVGAMKSMVPEGIEGRVKYKGEMEGVVYQLVGGLRSCMGYLGSASIEELWKKSSYVEITTSGLRESHVHDVEIV 4ixu A 1.9 BS03 38I A 1 D143 H145 D147 N149 S156 H160 G161 D202 D251 D120 H122 D124 N126 S133 H137 G138 D179 D228 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=23nM remove_due_to_license_issue P78540 23886684 406 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 4ixv A 2.3 BS03 XA1 A 1 D143 H145 D147 S155 S156 H160 G161 D202 D251 E296 D120 H122 D124 S132 S133 H137 G138 D179 D228 E273 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=240nM remove_due_to_license_issue P78540 23886684 405 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 4iz0 A 2.22 BS01 2BI A 1 L419 R422 M423 I482 R501 W528 L415 R418 M419 I478 R497 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50~100uM remove_due_to_license_issue O92972 23545108 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4iz0 A 2.22 BS02 2BI A 2 F193 R200 N316 C366 G410 M414 Y415 Q446 I447 Y448 F189 R196 N312 C362 G406 M410 Y411 Q442 I443 Y444 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50~100uM remove_due_to_license_issue O92972 23545108 602 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4izm A 4.5 BS03 ASP A 1 R276 S277 S278 G354 A358 G359 D394 R397 T398 R264 S265 S266 G342 A346 G347 D382 R385 T386 ? 0005283,0005886,0006865,0015108,0015183,0015293,0015501,0016020,0035725,0042802,0046872,0046942,0070207,0070778,0140009,1902476 remove_due_to_license_issue O59010 23563139 503 LQKILIGLILGAIVGLILGHYGYAHAVHTYVKPFGDLFVRLLKMLVMPIVFASCVVGAASISPARLGRVGVKIVVYYLLTSAFAVTLGIIMARLFNPGAGIHLAVGGQQFQPHQAPPLVHILLDIVPTNPFGALANGQVLPTIFFAIILGIAITYLMNSENEKVRKSAETLLDAINGLAEAMYKIVNGVMQYAPIGVFALIAYVMAEQGVHVVGELAKVTAAVYVGLTLQILLVYFVLLKIYGIDPISFIKHAKDAMLTAFVTRSSSGTLPVTMRVAKEMGISEGIYCFTLPLGATINMDGTALYQGVATFFIANALGSHLTVGQQLTIVLTAVLASIGTAGVPGAGAIMLAMVLHSVGLPLTDPNVAAAYAMILGIDAILDMGRTMVNVTGDLTGTAIVAKTE 4izy A 2.3 BS02 1J2 A 1 I32 S34 G35 Q37 G38 V40 A53 K55 M111 L168 I25 S27 G28 Q30 G31 V33 A46 K48 M104 L161 D151 K153 N156 D169 T188 D144 K146 N149 D162 T166 2.7.11.24 0004672,0004707,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=3.1nM, Kd=0.140000nM P45983 23664880 401 NNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLTRYYRAPEVILGMGYKENVDIWSVGCIMGEMIKGGVLFPGTDHIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPREHTIEEWKELIYKEVM 4j03 A 2.92 BS02 FVS A 1 D335 W336 I363 F381 Y383 Y466 L499 W525 D335 W336 I363 F381 Y383 Y466 L499 W525 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue P34913 23684894 603 MTLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 4j04 A 2.0 BS01 1JF A 1 M423 L474 L497 W528 M419 L470 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=11uM remove_due_to_license_issue O92972 23545108 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4j04 A 2.0 BS02 1JF A 2 V205 W208 K209 D359 L360 E361 V370 V372 R380 Y382 V201 W204 K205 D355 L356 E357 V366 V368 R376 Y378 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=11uM remove_due_to_license_issue O92972 23545108 602 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4j06 A 2.0 BS01 1JG A 1 L419 R422 M423 L474 H475 S476 Y477 L497 W528 L415 R418 M419 L470 H471 S472 Y473 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=4.6uM remove_due_to_license_issue O92972 23545108 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4j08 A 2.1 BS01 1JH A 1 L419 R422 H475 S476 Y477 I482 L497 W528 L415 R418 H471 S472 Y473 I478 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.22uM remove_due_to_license_issue O92972 23545108 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4j0a A 2.4 BS01 1JL A 1 L419 R422 M423 H475 S476 L497 W528 L415 R418 M419 H471 S472 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.16uM remove_due_to_license_issue O92972 23545108 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4j0p A 1.97 BS01 1H8 A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 D222 G224 T226 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.051uM remove_due_to_license_issue IC50=54nM P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j0r A 1.72 BS01 1H2 A 1 W81 P82 F83 L92 I146 M149 W40 P41 F42 L51 I105 M108 ? ic50=0.386uM remove_due_to_license_issue IC50=386nM, Kd=360nM O60885 23517011 205 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4j0s A 1.84 BS01 1H3 A 1 W81 P82 F83 L92 Y139 I146 M149 W40 P41 F42 L51 Y98 I105 M108 ? ic50=0.382uM remove_due_to_license_issue IC50=382nM, Kd=390nM O60885 23517011 205 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4j0t A 2.05 BS01 6T9 A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 D224 G226 T228 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=184uM remove_due_to_license_issue P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j0v A 1.94 BS01 1H7 A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 A396 G16 Q17 G18 L35 D37 Y76 F113 D222 G224 T226 A329 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.028uM remove_due_to_license_issue IC50=1nM P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j0y A 1.77 BS01 1H6 A 1 G72 Q73 G74 L91 D93 Y132 F169 I179 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 I123 D222 G224 T226 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.435uM remove_due_to_license_issue IC50=1170nM P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j0z A 2.13 BS01 1H5 A 1 G72 Q73 G74 L91 D93 Y132 F169 I179 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 I123 D224 G226 T228 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.077uM remove_due_to_license_issue P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j17 A 1.81 BS01 1HQ A 1 G72 Q73 G74 L91 D93 Y132 F169 I179 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 I123 D222 G224 T226 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.054uM remove_due_to_license_issue IC50=46nM P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1c A 2.01 BS01 1HO A 1 G72 Q73 G74 L91 D93 S96 Y132 F169 D289 G291 T293 G16 Q17 G18 L35 D37 S40 Y76 F113 D222 G224 T226 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.049uM remove_due_to_license_issue P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1e A 1.78 BS01 1HM A 1 G72 Q73 G74 L91 D93 S96 Y132 F169 I179 D289 G291 T293 G16 Q17 G18 L35 D37 S40 Y76 F113 I123 D222 G224 T226 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.019uM remove_due_to_license_issue IC50=17.9nM P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1f A 2.25 BS01 1HL A 1 Q73 G74 L91 D93 Y132 F169 I179 D289 G291 T293 Q17 G18 L35 D37 Y76 F113 I123 D222 G224 T226 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=0.012uM remove_due_to_license_issue IC50=11.5nM P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVETSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1g A 2.789 BS01 rna E 0 V16 S17 S18 F20 N21 P22 K53 N78 H79 R84 V88 T94 R97 V125 P127 L128 E130 A131 R168 M174 F178 K181 K184 Q185 R186 A218 V11 S12 S13 F15 N16 P17 K48 N73 H74 R79 V83 T89 R92 V120 P122 L123 E125 A126 R163 M169 F173 K176 K179 Q180 R181 A213 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 45 DFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNI 4j1g B 2.789 BS01 rna E 0 A15 S17 S18 F20 N21 P22 K50 K53 N78 H79 R84 R97 P127 L128 E130 R168 M174 F178 R180 K181 R186 A10 S12 S13 F15 N16 P17 K45 K48 N73 H74 R79 R92 P122 L123 E125 R163 M169 F173 R175 K176 R181 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 45 DFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFN 4j1g C 2.789 BS01 rna E 0 A15 S17 S18 F20 L47 H49 K53 N78 H79 R97 V125 P127 L128 E130 R168 M174 F178 R180 K181 Q185 R186 A218 G219 A10 S12 S13 F15 L42 H44 K48 N73 H74 R92 V120 P122 L123 E125 R163 M169 F173 R175 K176 Q180 R181 A213 G214 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 45 DFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNI 4j1g D 2.789 BS01 rna E 0 S18 F20 N21 P22 L47 H49 K53 N78 H79 V88 R97 P127 L128 E130 R168 F178 R180 K181 K184 Q185 R186 S13 F15 N16 P17 L42 H44 K48 N73 H74 V83 R92 P122 L123 E125 R163 F173 R175 K176 K179 Q180 R181 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 45 DFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFN 4j1h A 2.2 BS01 1HJ A 1 G72 Q73 G74 L91 D93 Y132 F169 I179 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 I123 D221 G223 T225 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.776uM remove_due_to_license_issue P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1i A 2.05 BS01 1HH A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 G16 Q17 G18 L35 D37 Y76 F113 D221 G223 T225 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.04uM remove_due_to_license_issue P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1j A 2.65 BS01 dna H 0 L47 H49 K50 K53 N78 H79 T94 L95 H96 R97 V125 P127 L128 E130 M174 F178 K181 K184 L45 H47 K48 K51 N76 H77 T92 L93 H94 R95 V123 P125 L126 E128 M172 F176 K179 K182 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 17 TGPDFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNISV 4j1j A 2.65 BS02 dna I 0 P13 R84 P11 R82 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 17 TGPDFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNISV 4j1j B 2.65 BS01 dna H 0 A14 A15 S17 S18 L47 K50 K53 N78 H79 D85 T94 H96 L128 E130 R168 M174 F178 K181 Q185 A10 A11 S13 S14 L43 K46 K49 N74 H75 D81 T90 H92 L124 E126 R164 M170 F174 K177 Q181 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 17 PDFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNISV 4j1j C 2.65 BS01 dna H 0 R12 R84 R180 R11 R83 R179 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 17 STGPDFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNISV 4j1j C 2.65 BS02 dna I 0 L47 K50 K53 N78 H79 R84 V125 P127 L128 R168 M174 F178 L46 K49 K52 N77 H78 R83 V124 P126 L127 R167 M173 F177 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 17 STGPDFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNISV 4j1j D 2.65 BS01 dna I 0 A14 S18 L47 K53 N78 H79 V88 T94 H96 R97 P127 L128 E130 R168 F178 K181 A9 S13 L42 K48 N73 H74 V83 T89 H91 R92 P122 L123 E125 R163 F173 K176 ? 0003723,0019013,1990904 remove_due_to_license_issue F2WAD7 23569220 1 ~ 17 DFIYDDRPAAVSSTFNPEKGYMDFITAYGKNINADNVRIFFLNHKKAKDSLKGSPKVEVDLQFGTLRVKVVNNHNPRNRDNPVADNAITLHRLSGYLAKWCFDEIDHGQIEEAEVKSKVVIPLAEAKGCKWGDGVALYLAFAPGAEMFLKDFEFYPLAIDIQRVVKDGMDITFMRKVLKQRYGTKTADDWMISEVTAIQSAVKVVAKLPWAKAGFTAAAKNFLAKFNISV 4j1k A 2.18 BS01 1HG A 1 G72 Q73 G74 L91 D93 Y132 F169 D289 G291 T293 A396 G16 Q17 G18 L35 D37 Y76 F113 D221 G223 T225 A318 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.013uM remove_due_to_license_issue P56817 23590342 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4j1p A 1.08 BS01 1K0 A 1 P371 F372 V376 L381 L383 N429 V435 P30 F31 V35 L40 L42 N88 V94 ? Kd=0.206uM remove_due_to_license_issue Kd=5800nM, IC50=251nM P25440 24391744 501 SMGKLSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 4j21 A 1.93 BS02 AJ6 A 1 H1031 G1032 Y1050 Y1060 S1068 Y1071 G1074 I1075 E1138 H80 G81 Y99 Y109 S117 Y120 G123 I124 E186 2.4.2.-,2.4.2.30 0003950 Kd=0.039uM remove_due_to_license_issue Q9H2K2 23672613 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4j22 A 2.12 BS02 AJ7 A 1 H1031 G1032 F1035 A1049 Y1050 Y1060 S1068 Y1071 G1074 I1075 H80 G81 F84 A98 Y99 Y109 S117 Y120 G123 I124 2.4.2.-,2.4.2.30 0003950 Kd=0.018uM remove_due_to_license_issue Q9H2K2 23672613 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4j28 A 1.73 BS01 EAT A 1 H66 E87 W88 H135 D229 W232 W316 H32 E53 W54 H101 D195 W198 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=2uM remove_due_to_license_issue Q8A3I4 23830696 501 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAA 4j2t A 3.2 BS01 1HT A 1 F256 Q259 L260 V263 I267 I765 V769 V772 F776 I829 F834 F256 Q259 L260 V263 I267 I765 V769 V772 F776 I829 F834 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 23574308 1001 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 4j2x A 2.85 BS03 dna G 0 K84 Y86 S191 K192 R220 Q222 K32 Y34 S139 K140 R168 Q170 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 24290140 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMETDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKQSLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDESEGEEFTVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTP 4j2x A 2.85 BS04 dna H 0 K90 R91 F92 K192 R218 S221 T223 K295 K311 K38 R39 F40 K140 R166 S169 T171 K243 K259 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 24290140 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMETDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKQSLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDESEGEEFTVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTP 4j2x C 2.85 BS03 dna E 0 K84 Y86 S191 K196 R220 Q222 K32 Y34 S139 K144 R168 Q170 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 24290140 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMETDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKQSLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDESEGEEFTVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTPE 4j2x C 2.85 BS04 dna F 0 K90 R91 F92 K192 K195 R218 S221 T223 K311 K38 R39 F40 K140 K143 R166 S169 T171 K259 ? 0000978,0001228,0003677,0003700,0005634,0006355,0006357 remove_due_to_license_issue P31266 24290140 1 ~ 15 PPKRLTREAMRNYLKERGDQTVLILHAKVAQKSYGNEKRFFCPPPCVYLMGSGWKKKKEQMETDGCSEQESQPCAFIGIGNSDQEMQQLNLEGKNYCTAKTLYISDSDKRKHFMLSVKMFYGNSDDIGVFLSKRIKVISKPSKKKQSLKNADLCIASGTKVALFNRLRSQTVSTRYLHVEGGNFHASSQQWGAFYIHLLDDDESEGEEFTVRDGYIHYGQTVKLVCSVTGMALPRLIIRKVDKQTALLDADDPVSQLHKCAFYLKDTERMYLCLSQERIIQFQATPCPKEQNKEMINDGASWTIISTDKAEYTFYEGMGPVLAPVTPVPVVESLQLNGGGDVAMLELTGQNFTPNLRVWFGDVEAETMYRCGESMLCVVPDISAFREGWRWVRQPVQVPVTLVRNDGVIYSTSLTFTYTPE 4j3d A 2.0 BS03 1JS A 1 M62 E77 H78 T190 F191 G192 D196 I197 R201 G209 S210 V216 K238 D241 H264 M62 E77 H78 T180 F181 G182 D186 I187 R191 G199 S200 V206 K228 D231 H254 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=5.3nM remove_due_to_license_issue P47205 23499237 303 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYM 4j3e A 1.91 BS01 NUT A 1 L50 L53 G54 I57 M58 F87 V89 H92 Y96 L31 L34 G35 I38 M39 F68 V70 H73 Y77 2.3.2.27 0005634,0043066,0051726 ic50=0.088uM remove_due_to_license_issue P56273 24900694 201 MEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4j3i A 1.24 BS01 1K0 A 1 P82 F83 V87 N140 D144 I146 P41 F42 V46 N99 D103 I105 ? Kd=8.93uM remove_due_to_license_issue IC50=510nM, Kd=1100nM O60885 24391744 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4j3j A 3.2 BS01 D3C A 1 E205 E206 F357 Y585 S630 Y631 Y662 Y666 N710 V711 E166 E167 F318 Y546 S591 Y592 Y623 Y627 N671 V672 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 23671024 801 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFS 4j3l A 2.09 BS02 AJ5 A 1 H1031 G1032 F1035 Y1050 Y1060 S1068 Y1071 G1074 I1075 E1138 H80 G81 F84 Y99 Y109 S117 Y120 G123 I124 E186 2.4.2.-,2.4.2.30 0003950 Kd=0.016uM remove_due_to_license_issue Q9H2K2 23672613 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4j3m A 1.9 BS02 AJ8 A 1 H1031 G1032 F1035 Y1050 Y1060 S1068 Y1071 G1074 H80 G81 F84 Y99 Y109 S117 Y120 G123 2.4.2.-,2.4.2.30 0003950 ic50=0.021uM remove_due_to_license_issue Q9H2K2 23672613 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4j3u A 1.7 BS01 SGD C 1 F514 D541 R544 F499 D526 R529 N219 H311 F312 K366 D473 E510 D642 N204 H296 F297 K351 D458 E495 D627 3.2.1.41 0000272,0004553,0005975,0016798,0046872,0051060 remove_due_to_license_issue Q9FYY0 25562209 1 MPDARAYWVTSDLIAWNVGELEQSVCLYASRAAAMSLSGIQGYDSKVELQPESAGLPETVTQKFPFISSYRAFRVPSSVDVASLVKCQLVVASFDVTGLQLPGVLDDMFAYTGPLGAVFSEDSVSLHLWAPTAQGVSVCFFDGPAGPALETVQLKESNGVWSVTGPREWENRYYLYEVDVYHPTKAQVLKCLAGDPYARSLSANGARTWLVDINNETLKPASWDELADEKPKLDSFSDITIYELHIRDFSAHDGTVDSDSRGGFRAFAYQASAGMEHLRKLSDAGLTHVHLLPSFHFAGVDDIKSNWKFVDECELATFPPGSDMQQAAVVAIQEEDPYNWGYNPVLWGVPKGSYASDPDGPSRIIEYRQMVQALNRIGLRVVMDVVYNHLDSSGPCGISSVLDKIVPGYYVRRDTNGQIENSAAMNNTASEHFMVDRLIVDDLLNWAVNYKVDGFRFDLMGHIMKRTMMRAKSALQSLTTDAHGVDGSKIYLYGEGWDFAEVARNQRGINGSQLNMSGTGIGSFNDRIRDAINGGNPFGNPLQQGFNTGLFLEPNGFYQGNEADTRRSLATYADQIQIGLAGNLRDYVLISHTGEAKKGSEIHTFDGLPVGYTASPIETINYVSAHDNETLFDVISVKTPMILSVDERCRINHLASSMMALSQGIPFFHAGDEILRSKSIDRDSYNSGDWFNKLDFTYETNNWGVGLPPSEKNEDNWPLMKPRLENPSFKPAKGHILAALDSFVDILKIRYSSPLFRLSTANDIKQRVRFHNTGPSLVPGVIVMGIEDARGESPEMAQLDTNFSYVVTVFNVCPHEVSMDIPALASMGFELHPVQVNSSDTLVRKSAYEAATGRFTVPGRTVSVFVEPRC 4j3u A 1.7 BS02 GLC C 1 W512 N643 W497 N628 N219 H311 F312 K366 D473 E510 D642 N204 H296 F297 K351 D458 E495 D627 3.2.1.41 0000272,0004553,0005975,0016798,0046872,0051060 remove_due_to_license_issue Q9FYY0 25562209 2 MPDARAYWVTSDLIAWNVGELEQSVCLYASRAAAMSLSGIQGYDSKVELQPESAGLPETVTQKFPFISSYRAFRVPSSVDVASLVKCQLVVASFDVTGLQLPGVLDDMFAYTGPLGAVFSEDSVSLHLWAPTAQGVSVCFFDGPAGPALETVQLKESNGVWSVTGPREWENRYYLYEVDVYHPTKAQVLKCLAGDPYARSLSANGARTWLVDINNETLKPASWDELADEKPKLDSFSDITIYELHIRDFSAHDGTVDSDSRGGFRAFAYQASAGMEHLRKLSDAGLTHVHLLPSFHFAGVDDIKSNWKFVDECELATFPPGSDMQQAAVVAIQEEDPYNWGYNPVLWGVPKGSYASDPDGPSRIIEYRQMVQALNRIGLRVVMDVVYNHLDSSGPCGISSVLDKIVPGYYVRRDTNGQIENSAAMNNTASEHFMVDRLIVDDLLNWAVNYKVDGFRFDLMGHIMKRTMMRAKSALQSLTTDAHGVDGSKIYLYGEGWDFAEVARNQRGINGSQLNMSGTGIGSFNDRIRDAINGGNPFGNPLQQGFNTGLFLEPNGFYQGNEADTRRSLATYADQIQIGLAGNLRDYVLISHTGEAKKGSEIHTFDGLPVGYTASPIETINYVSAHDNETLFDVISVKTPMILSVDERCRINHLASSMMALSQGIPFFHAGDEILRSKSIDRDSYNSGDWFNKLDFTYETNNWGVGLPPSEKNEDNWPLMKPRLENPSFKPAKGHILAALDSFVDILKIRYSSPLFRLSTANDIKQRVRFHNTGPSLVPGVIVMGIEDARGESPEMAQLDTNFSYVVTVFNVCPHEVSMDIPALASMGFELHPVQVNSSDTLVRKSAYEAATGRFTVPGRTVSVFVEPRC 4j3u A 1.7 BS03 GLC C 2 N551 F553 N536 F538 N219 H311 F312 K366 D473 E510 D642 N204 H296 F297 K351 D458 E495 D627 3.2.1.41 0000272,0004553,0005975,0016798,0046872,0051060 remove_due_to_license_issue Q9FYY0 25562209 6 MPDARAYWVTSDLIAWNVGELEQSVCLYASRAAAMSLSGIQGYDSKVELQPESAGLPETVTQKFPFISSYRAFRVPSSVDVASLVKCQLVVASFDVTGLQLPGVLDDMFAYTGPLGAVFSEDSVSLHLWAPTAQGVSVCFFDGPAGPALETVQLKESNGVWSVTGPREWENRYYLYEVDVYHPTKAQVLKCLAGDPYARSLSANGARTWLVDINNETLKPASWDELADEKPKLDSFSDITIYELHIRDFSAHDGTVDSDSRGGFRAFAYQASAGMEHLRKLSDAGLTHVHLLPSFHFAGVDDIKSNWKFVDECELATFPPGSDMQQAAVVAIQEEDPYNWGYNPVLWGVPKGSYASDPDGPSRIIEYRQMVQALNRIGLRVVMDVVYNHLDSSGPCGISSVLDKIVPGYYVRRDTNGQIENSAAMNNTASEHFMVDRLIVDDLLNWAVNYKVDGFRFDLMGHIMKRTMMRAKSALQSLTTDAHGVDGSKIYLYGEGWDFAEVARNQRGINGSQLNMSGTGIGSFNDRIRDAINGGNPFGNPLQQGFNTGLFLEPNGFYQGNEADTRRSLATYADQIQIGLAGNLRDYVLISHTGEAKKGSEIHTFDGLPVGYTASPIETINYVSAHDNETLFDVISVKTPMILSVDERCRINHLASSMMALSQGIPFFHAGDEILRSKSIDRDSYNSGDWFNKLDFTYETNNWGVGLPPSEKNEDNWPLMKPRLENPSFKPAKGHILAALDSFVDILKIRYSSPLFRLSTANDIKQRVRFHNTGPSLVPGVIVMGIEDARGESPEMAQLDTNFSYVVTVFNVCPHEVSMDIPALASMGFELHPVQVNSSDTLVRKSAYEAATGRFTVPGRTVSVFVEPRC 4j3u A 1.7 BS04 GLC C 3 F514 F553 F499 F538 N219 H311 F312 K366 D473 E510 D642 N204 H296 F297 K351 D458 E495 D627 3.2.1.41 0000272,0004553,0005975,0016798,0046872,0051060 remove_due_to_license_issue Q9FYY0 25562209 8 MPDARAYWVTSDLIAWNVGELEQSVCLYASRAAAMSLSGIQGYDSKVELQPESAGLPETVTQKFPFISSYRAFRVPSSVDVASLVKCQLVVASFDVTGLQLPGVLDDMFAYTGPLGAVFSEDSVSLHLWAPTAQGVSVCFFDGPAGPALETVQLKESNGVWSVTGPREWENRYYLYEVDVYHPTKAQVLKCLAGDPYARSLSANGARTWLVDINNETLKPASWDELADEKPKLDSFSDITIYELHIRDFSAHDGTVDSDSRGGFRAFAYQASAGMEHLRKLSDAGLTHVHLLPSFHFAGVDDIKSNWKFVDECELATFPPGSDMQQAAVVAIQEEDPYNWGYNPVLWGVPKGSYASDPDGPSRIIEYRQMVQALNRIGLRVVMDVVYNHLDSSGPCGISSVLDKIVPGYYVRRDTNGQIENSAAMNNTASEHFMVDRLIVDDLLNWAVNYKVDGFRFDLMGHIMKRTMMRAKSALQSLTTDAHGVDGSKIYLYGEGWDFAEVARNQRGINGSQLNMSGTGIGSFNDRIRDAINGGNPFGNPLQQGFNTGLFLEPNGFYQGNEADTRRSLATYADQIQIGLAGNLRDYVLISHTGEAKKGSEIHTFDGLPVGYTASPIETINYVSAHDNETLFDVISVKTPMILSVDERCRINHLASSMMALSQGIPFFHAGDEILRSKSIDRDSYNSGDWFNKLDFTYETNNWGVGLPPSEKNEDNWPLMKPRLENPSFKPAKGHILAALDSFVDILKIRYSSPLFRLSTANDIKQRVRFHNTGPSLVPGVIVMGIEDARGESPEMAQLDTNFSYVVTVFNVCPHEVSMDIPALASMGFELHPVQVNSSDTLVRKSAYEAATGRFTVPGRTVSVFVEPRC 4j4n A 2.75 BS01 D44 A 1 D56 V74 W78 Y101 C106 I110 D50 V68 W72 Y95 C100 I104 Y44 F55 D56 I75 Y101 F118 Y38 F49 D50 I69 Y95 F112 5.2.1.8 0003755 remove_due_to_license_issue Q8I4V8 23974147 201 FEKVELTADGGVIKTILKKGDEGEENIPKKGNEVTVHYVGKLESTGKVFDSSFDRNVPFKFHLEQGEVIKGWDICVSSMRKNEKCLVRIESMYGYGDEGCGESIPGNSVLLFEIELLSFRELE 4j4o A 1.73 BS01 D44 A 1 D55 F64 E72 V73 I74 W77 Y100 C105 I109 D51 F60 E68 V69 I70 W73 Y96 C101 I105 Y43 F54 D55 I74 Y100 F117 Y39 F50 D51 I70 Y96 F113 5.2.1.8 0003755 remove_due_to_license_issue A5K8X6 23974147 201 TLEQVHLTEDGGVVKTILRKGEGGEENAPKKGNEVTVHYVGKLESSGKVFDSSRERNVPFKFHLGQGEVIKGWDICVASMTKNEKCSVRLDSKYGYGEEGCGESIPGNSVLIFEIELISFRE 4j4v A 2.303 BS01 SVR A 1 T63 R64 G65 N66 K67 R95 P127 M147 F177 I181 T62 R63 G64 N65 K66 R94 P126 M146 F176 I180 ? 0003723,0019013,0019028,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue I6WJ72 23576501 301 SEWSRIAVEFGEQQLNLTELEDFARELAYEGLDPALIIKKLKETGGDDWVKDTKFIIVFALTRGNKIVKASGKMSNSGSKRLMALQEKYGLVERAETRLSITPVRVAQSLPTWTCAAAAALKEYLPVGPAVMNLKVENYPPEMMCMAFGSLIPTAGVSEATTKTLMEAYSLWQDAFTKTINVKMRGASKTEVYNSFRDPLHAAVNSVFFPNDVRVKWLKAKGILGPDGVPSRAAEVAAAAYRNL 4j4v B 2.303 BS01 SVR B 1 T63 R64 G65 N66 P127 M147 F177 T62 R63 G64 N65 P126 M146 F176 ? 0003723,0019013,0019028,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue I6WJ72 23576501 301 SEWSRIAVEFGEQQLNLTELEDFARELAYEGLDPALIIKKLKETGGDDWVKDTKFIIVFALTRGNKIVKASGKMSNSGSKRLMALQEKYGLVERAETRLSITPVRVAQSLPTWTCAAAAALKEYLPVGPAVMNLKVENYPPEMMCMAFGSLIPTAGVSEATTKTLMEAYSLWQDAFTKTINVASKTEVYNSFRDPLHAAVNSVFFPNDVRVKWLKAKGILGPDGVPSRAAEVAAAAYRNL 4j4v E 2.303 BS01 SVR E 1 T63 R64 G65 N66 R95 A96 M147 F177 T62 R63 G64 N65 R94 A95 M146 F176 ? 0003723,0019013,0019028,0030430,0042025,0044172,0044177,1990904 remove_due_to_license_issue I6WJ72 23576501 301 SEWSRIAVEFGEQQLNLTELEDFARELAYEGLDPALIIKKLKETGGDDWVKDTKFIIVFALTRGNKIVKASGKMSNSGSKRLMALQEKYGLVERAETRLSITPVRVAQSLPTWTCAAAAALKEYLPVGPAVMNLKVENYPPEMMCMAFGSLIPTAGVSEATTKTLMEAYSLWQDAFTKTINGASKTEVYNSFRDPLHAAVNSVFFPNDVRVKWLKAKGILGPDGVPSRAAEVAAAAYRNL 4j51 A 2.3 BS01 N75 A 1 Y60 K61 D62 C227 S228 A229 C231 G232 R233 Q274 Q278 Y60 K61 D62 C226 S227 A228 C230 G231 R232 Q273 Q277 D195 C227 R233 T234 Q274 D194 C226 R232 T233 Q273 3.1.3.48 0004725,0004726,0006470,0016311 ic50=0.259uM remove_due_to_license_issue IC50=259nM, Ki=110nM Q9Y2R2 23713581 401 MDQREILQKFLDEAQSKKITKEEFANEFLKLKRQSTKYKADKTYPTTVAEKPKNIKKNRYKDILPYDYSRVELSLITDEDSSYINANFIKGVYGPKAYIATQGPLSTTLLDFWRMIWEYSVLIIVMACMEYEMGKKKCERYWAEPGEMQLEFGPFSVSCEAEKRKSDYIIRTLKVKFNSETRTIYQFHYKNWPDHDVPSSIDPILELIWDVRCYQEDDSVPICIHCSAGCGRTGVICAIDYTWMLLKDGIIPENFSVFSLIREMRTQRPSLVQTQEQYELVYNAVLELFKRQMDVIRDKHSG 4j52 A 2.3 BS01 1J3 A 1 L59 C67 A80 G81 K82 V114 L132 C133 R134 R136 F183 L22 C30 A43 G44 K45 V77 L95 C96 R97 R99 F146 D176 K178 G180 N181 D194 T214 D139 K141 G143 N144 D157 T177 2.7.11.21 0004672,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=3.0nM P53350 23664874 400 KEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAPS 4j53 A 2.5 BS02 1J4 A 1 L59 C67 V114 C133 R136 F183 L22 C30 V77 C96 R99 F146 D176 K178 G180 N181 D194 T214 D139 K141 G143 N144 D157 T177 2.7.11.21 0004672,0005524,0006468 ic50=2nM remove_due_to_license_issue IC50=2.0nM P53350 23664874 403 KEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAPS 4j58 A 1.28 BS01 53Z A 1 F102 M103 Q105 R124 A143 N144 Q153 F155 H168 F59 M60 Q62 R81 A100 N101 Q110 F112 H125 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 27652979 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 4j59 A 1.92 BS01 671 A 1 F102 M103 Q105 R124 A143 N144 Q153 F155 H168 F59 M60 Q62 R81 A100 N101 Q110 F112 H125 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 27652979 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 4j5b A 2.01 BS01 6B4 A 1 R97 M103 Q105 G114 R124 A143 N144 Q153 F155 H168 R54 M60 Q62 G71 R81 A100 N101 Q110 F112 H125 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 27652979 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 4j5c X 1.03 BS01 7I6 X 1 R97 F102 M103 Q105 R124 A143 N144 Q153 F155 H168 R54 F59 M60 Q62 R81 A100 N101 Q110 F112 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 27652979 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 4j5d X 1.32 BS01 728 X 1 R97 M103 Q105 R124 A143 N144 Q153 F155 H168 R54 M60 Q62 R81 A100 N101 Q110 F112 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 27652979 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 4j5e X 0.99 BS01 7B7 X 1 R97 M103 Q105 R124 A143 N144 T149 Q153 F155 H168 R54 M60 Q62 R81 A100 N101 T106 Q110 F112 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 27652979 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 4j5p A 2.3 BS01 BR1 A 1 S190 M191 F192 S193 S217 T236 D237 I238 G239 G240 S241 C269 F432 T488 S158 M159 F160 S161 S185 T204 D205 I206 G207 G208 S209 C237 F400 T456 K142 S217 S218 T236 I238 G239 G240 S241 F244 K110 S185 S186 T204 I206 G207 G208 S209 F212 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 23581831 601 GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTPQK 4j6i A 2.9 BS01 1JV A 1 W812 I831 K833 Y867 I879 E880 I881 V882 K883 D884 I963 D964 W570 I589 K591 Y625 I637 E638 I639 V640 K641 D642 I721 D722 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=1.4nM P48736 23540645 1201 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 4j70 K 2.8 BS01 1KR K 1 T1 K33 M45 A46 G47 S131 T1 K33 M45 A46 G47 S131 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 23547757 301 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4j74 A 1.2 BS01 I18 A 1 L50 I57 V89 H92 I95 Y96 L31 I38 V70 H73 I76 Y77 2.3.2.27 0005634,0043066,0051726 Kd=26uM remove_due_to_license_issue P56273 24900726 201 MEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4j74 A 1.2 BS02 I18 A 2 M58 Y63 Q68 M39 Y44 Q49 2.3.2.27 0005634,0043066,0051726 Kd=26uM remove_due_to_license_issue P56273 24900726 202 MEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4j7d A 1.25 BS01 I31 A 1 L50 I57 M58 F87 V89 H92 I95 Y96 L31 I38 M39 F68 V70 H73 I76 Y77 2.3.2.27 0005634,0043066,0051726 Kd=20uM remove_due_to_license_issue P56273 24900726 201 MEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4j7e A 1.63 BS01 I29 A 1 L50 L53 Y63 F87 V89 H92 I95 Y96 L31 L34 Y44 F68 V70 H73 I76 Y77 2.3.2.27 0005634,0043066,0051726 Kd=14uM remove_due_to_license_issue P56273 24900726 201 MEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4j8m A 1.853 BS01 CJ5 A 1 G145 N146 V147 K162 L164 L194 E211 Y212 A213 G216 L263 D274 V279 A281 P282 G21 N22 V23 K38 L40 L70 E87 Y88 A89 G92 L139 D150 V155 A157 P158 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=48nM remove_due_to_license_issue O14965 25175806 501 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 4j8t A 2.05 BS01 DOG A 1 L14 Y34 H54 F58 Y101 Y115 L117 V124 L14 Y34 H54 F58 Y101 Y115 L117 V124 ? Kd=168nM remove_due_to_license_issue Kd=474nM Q9HYR3 24005320 201 MNAKEIVVHALRLLENGDARGWCDLFHPEGVLEYPYPPPGYKTRFEGRETIWAHMRLFPEYMTIRFTDVQFYETADPDLAIGEFHGDGVHTVSGGKLAADYISVLRTRDGQILLYRLFFNPLRVLEPL 4j93 A 1.74 BS02 1JR A 1 N53 L56 N57 M66 K70 T107 N53 L56 N57 M66 K70 T107 ? 0016032 remove_due_to_license_issue Q79791 23817385 202 PIVQNLQGQMVHQAISPRTLNAWVKVVEEKAFSPEVIPMFSALSEGATPQDLNTMLNTVGGHQAAMQMLKETINEEAAEWDRLHPVHAGPIAPGQMREPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYS 4j9a A 3.2 BS01 DOG A 1 L14 Y34 Y41 M55 Y61 Y99 Y101 Y115 L117 L13 Y33 Y40 M54 Y60 Y98 Y100 Y114 L116 ? remove_due_to_license_issue Kd=474nM Q9HYR3 24005320 201 NAKEIVVHALRLLENGDARGWSDLFHPEGVLEYPYPPPGYKTRFEGRETIWAHMRLFPEYMTIRFTDVQFYETADPDLAIGEFHGDGVLTASGGKLAYDYIAVWRTRDGQILLYRLFFNPLR 4jai A 3.2 BS01 XU2 A 1 L139 V147 A160 K162 Q185 L208 L210 Y212 A213 G216 L263 F275 L14 V22 A35 K37 Q60 L83 L85 Y87 A88 G91 L138 F150 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T151 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=4.0nM O14965 23570792 401 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 4jaj A 2.7 BS01 XU1 A 1 L139 A213 G216 L263 L15 A89 G92 L139 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=5540nM O14965 23570792 900 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 4jal A 2.0 BS01 SAH A 1 L78 T79 T80 G100 E102 R121 I122 M124 M131 N132 L133 L79 T80 T81 G101 E103 R122 I123 M125 M132 N133 L134 2.1.1.207 0001510,0002131,0002132,0003723,0005737,0006396,0008033,0008168,0008173,0008175,0008757,0030488,0032259,0042803,0141098,0141102 remove_due_to_license_issue P0AGJ7 23804755 201 MALNIVLYEPEIPPNTGNIIRLCANTGFRLHIIEPMGFAWDDKRLRRAGLDYHEFTAVTRHHDYRAFLEAENPQRLFALTTKGTPAHSAVSYQDGDYLMFGPETRGLPASILDALPAEQKIRIPMVPDSRSMNLSNAVSVVVYEAWRQLGYPGAVL 4jal B 2.0 BS01 SAH B 1 L78 T79 T80 F99 G100 E102 I122 M124 S130 M131 L79 T80 T81 F100 G101 E103 I123 M125 S131 M132 2.1.1.207 0001510,0002131,0002132,0003723,0005737,0006396,0008033,0008168,0008173,0008175,0008757,0030488,0032259,0042803,0141098,0141102 remove_due_to_license_issue P0AGJ7 23804755 203 MALNIVLYEPEIPPNTGNIIRLCANTGFRLHIIEPMGFAWDDKRLRRAGLDYHEFTAVTRHHDYRAFLEAENPQRLFALTTKGTPAHSAVSYQDGDYLMFGPETRGLPASILDALPAEQKIRIPMVPDSRSMNLSNAVSVVVYEAWRQLGYPGAV 4jaz A 2.85 BS01 STL A 1 F264 H266 R280 I281 R288 I341 S342 F58 H60 R74 I75 R82 I135 S136 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 24796862 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 4jbl B 2.0 BS01 MET B 1 X58 T85 S86 N88 T89 M136 Q159 F160 G192 G236 I237 A239 X57 T84 S85 N87 T88 M135 Q158 F159 G191 G235 I236 A238 K58 S280 K57 S279 2.5.1.47 0004124,0006535 Kd=0.54mM remove_due_to_license_issue O15570 23747298 401 EQISISSPRKRIYHNILETIGGTPLVELHGVTEHPRIKKGTRILVKLEYFNPMSSVKDRVGFNIVYQAIKDGRLKPGMEIIESTSGNTGIALCQAGAVFGYRVNIAMPSTMSVERQMIMKAFGAELILTEGKKGMPGAIEEVNKMIKENPGKYFVANQFGNPDNTAAHHYTANEIWEDTDGEVDIVVSAVGTSGTVIGVAEKLKEKKKGIKIIAVEPEESAVLEGKAKGPHGIQGIGAGFIPDIYKKEFVDEIIPIKTQDAWKMARAVVKYDGIMCGMSSGAAILAGLKEAEKPENEGKTIVIIVPSCGERYLSTDLYKIKDEGTKIQILDSLLN 4jbo A 2.493 BS01 WPH A 1 R137 F144 A160 K162 V174 L178 E181 E211 Y212 A213 P214 G216 L263 D274 R12 F19 A35 K37 V49 L53 E56 E86 Y87 A88 P89 G91 L138 D149 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=24nM remove_due_to_license_issue IC50=24nM O14965 23610398 501 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTDLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 4jbp A 2.45 BS01 YPH A 1 R137 L139 F144 V147 A160 K162 L164 L169 L178 E181 E211 A213 P214 L215 G216 K224 L263 D274 R12 L14 F19 V22 A35 K37 L39 L44 L53 E56 E86 A88 P89 L90 G91 K99 L138 D149 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=41nM remove_due_to_license_issue IC50=41nM O14965 23610398 501 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 4jbs A 2.789 BS02 P52 A 1 E200 G334 A335 E337 H370 E371 H374 E393 F450 Y455 Y892 E144 G278 A279 E281 H314 E315 H318 E337 F394 Y399 Y800 E337 H370 E371 H374 E393 Q447 Y455 E281 H314 E315 H318 E337 Q391 Y399 3.4.11.- 0002250,0002474,0004175,0004177,0005515,0005615,0005737,0005783,0005788,0005789,0006508,0008217,0008237,0008270,0016020,0019885,0042277,0043171,0046872,0070006 remove_due_to_license_issue IC50=11nM Q6P179 24248368 1009 PVATNGERFPWQELRLPSVVIPLHYDLFVHPNLTSLDFVASEKIEVLVSNATQFIILHSKDLEITNATLQSEEYMKPGKELKVLSYPAHEQIALLVPEKLTPHLKYYVAMDFQAKLGDGFEGFYKSTYRTLGGETRILAVTDFEPTQARMAFPCFDEPLFKANFSIKIRRESRHIALSNMPKVKTIELEGGLLEDHFETTVKMSTYLVAYIVCDFHSLSGFTSSGVKVSIYASPDKRNQTHYALQASLKLLDFYEKYFDIYYPLSKLDLIAIPDFAPGAMENWGLITYRETSLLFDPKTSSASDKLWVTRVIAHELAHQWFGNLVTMEWWNDIWLKEGFAKYMELIAVNATYPELQFDDYFLNVCFEVITKDSLNSSRPISKPAETPTQIQEMFDEVSYNKGACILNMLKDFLGEEKFQKGIIQYLKKFSYRNAKNDDLWSSLSNSLGENAEVKEMMTTWTLQKGIPLLVVKQDGCSLRLQQERFLQGQERYLWHIPLTYSTSSSNVIHRHILKSKTDTLDLPEKTSWVKFNVDSNGYYIVHYEGHGWDQLITQLNQNHTLLRPKDRVGLIHDVFQLVGAGRLTLDKALDMTYYLQHETSSPALLEGLSYLESFYHMMDRRNISDISENLKRYLLQYFKPVIDRQSWSDKGSVWDRMLRSALLKLACDLNHAPCIQKAAELFSQWMESSGKLNIPTDVLKIVYSVGAQTTAGWNYLLEQYELSMSSAEQNKILYALSTSKHQEKLLKLIELGMEGKVIKTQNLAALLHAIARRPKGQQLAWDFVRENWTHLLKKFDLGSYDIRMIISGTTAHFSSKDKLQEVKLFFESLEAQGSHLDIFQTVLETITKNIKWLEKNLPTLRTWLMVNTR 4jda A 2.65 BS01 A9S A 1 K79 V107 A113 S116 F132 H139 L141 Y144 K57 V81 A87 S90 F106 H113 L115 Y118 ? 0004864,0005515,0005634,0005737,0005886,0009738,0010427,0038023,0042802,0042803,0062049 remove_due_to_license_issue Q9SSM7 23844015 301 YGLTKDEFSTLDSIIRTHHTFPRSPNTCTSLIAHRVDAPAHAIWRFVRDFANPNKYKHFIKSCTIRVNKEIKVGTIREVSVVSGLPASTSVEILEVLDEEKRILSFRVLGGEHRLNNYRSVTSVNEFVVLKKRVYSVVLESYIVDIPQGNTEEDTRMFVDTVVKSNLQNLAVISTAS 4jda B 2.65 BS01 A9S B 1 K79 V107 S116 L141 Y144 V192 N196 K57 V80 S89 L114 Y117 V157 N161 ? 0004864,0005515,0005634,0005737,0005886,0009738,0010427,0038023,0042802,0042803,0062049 remove_due_to_license_issue Q9SSM7 23844015 301 YGLTKDEFSTLDSIIRTHHTFPRSPNTCTSLIAHRVDAPAHAIWRFVRDFANPNKYKHFIKSCTIRVNEIKVGTIREVSVVSGLPASTSVEILEVLDEEKRILSFRVLGGEHRLNNYRSVTSVNEFVVVYSVVLESYIVDIPQGNTEEDTRMFVDTVVKSNLQNLAVISTA 4je7 A 2.1 BS01 BB2 A 1 P46 C47 V48 G49 Q54 R84 G110 C111 R118 W146 I150 H153 E154 H157 P45 C46 V47 G48 Q53 R83 G109 C110 R117 W145 I149 H152 E153 H156 G49 Q54 C111 E112 H153 E154 H157 G48 Q53 C110 E111 H152 E153 H156 3.5.1.88 0042586 Kd=395nM remove_due_to_license_issue IC50=27nM Q9FV53 24531459 201 DLPEIVASGDPVLHEKAREVDPGEIGSERIQKIIDDMIKVMRLAPCVGLAAPQIGVPLRIIVLEDTKEYISYAPKEEILAQERRHFDLMVMVNPVLKERSNKKALFFEGCESVDGFRAAVERYLEVVVTGYDRQGKRIEVNASGWQARILQHECDHLDGNLYVDKMVPRTFRTVDNLDLPLAEGCPKLGSHHH 4jfi A 1.05 BS01 1KT A 1 Y57 F67 D68 F77 V86 I87 W90 Y113 S118 K121 Y45 F55 D56 F65 V74 I75 W78 Y101 S106 K109 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=18.1uM remove_due_to_license_issue Q13451 23647266 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKG 4jfj A 1.08 BS01 1KU A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 I122 F130 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 I110 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=2.1uM remove_due_to_license_issue Ki=2100nM Q13451 23647266 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4jfk A 1.15 BS01 JFK A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 S118 L119 P120 K121 I122 F130 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 S106 L107 P108 K109 I110 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Kd=0.36uM remove_due_to_license_issue Ki=300nM, Kd=360nM Q13451 23647266 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4jfl A 1.2 BS01 1KY A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 I122 F130 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 I110 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Kd=10.5uM remove_due_to_license_issue Kd=10500nM, Ki=13900nM Q13451 23647266 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4jfm A 1.02 BS01 1KZ A 1 Y57 F67 D68 R73 F77 V86 W90 Y113 F130 Y45 F55 D56 R61 F65 V74 W78 Y101 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Kd=3.3uM remove_due_to_license_issue Ki=7600nM, Kd=3300nM Q13451 23647266 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4jfs A 2.0 BS01 16Z A 1 H66 E87 W88 H135 D229 W232 E288 W316 H32 E53 W54 H101 D195 W198 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=5.4uM remove_due_to_license_issue Q8A3I4 23740878 501 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAA 4jft A 2.1 BS01 1KN A 1 H66 E87 W88 H135 Y178 D229 W232 W316 H32 E53 W54 H101 Y144 D195 W198 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=3.5uM remove_due_to_license_issue Q8A3I4 23740878 501 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAA 4jfv A 1.88 BS01 H57 A 1 H66 E87 W88 H135 Y178 D229 E288 W316 H32 E53 W54 H101 Y144 D195 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=0.52uM remove_due_to_license_issue Q8A3I4 23740878 508 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAK 4jfw A 2.1 BS01 H58 A 1 H66 E87 W88 H135 D229 W232 E288 W316 H32 E53 W54 H101 D195 W198 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=0.46uM remove_due_to_license_issue Q8A3I4 23740878 501 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAK 4jg6 A 2.6 BS01 1LB A 1 C436 A449 M496 D561 C26 A39 M86 D151 D539 K541 N544 D561 T581 D129 K131 N134 D151 T171 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P51812 23540679 801 SIVQQLHRNSIQFTDGYEVKEDISVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNR 4jg7 A 3.0002 BS01 1LC A 1 I428 C436 A449 M496 L546 D561 I24 C30 A43 M90 L140 D155 D539 K541 N544 D561 T581 D133 K135 N138 D155 T175 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P51812 23540679 801 HSIVQQLHRNSIQFTDGYEVKEDIGVYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRN 4jg8 A 3.1002 BS01 1LE A 1 I428 C436 A449 K451 M493 L495 M496 D561 I14 C22 A35 K37 M79 L81 M82 D147 D539 K541 N544 D561 T581 D125 K127 N130 D147 T167 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P51812 23540679 801 SIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVMELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQ 4jgv A 3.01 BS01 T94 A 1 L509 V510 T513 Q528 L555 K558 L148 V149 T152 Q167 L190 K193 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P22736 24316735 601 ANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKWAEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFGDWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVAAVAEPPALSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF 4jh0 A 2.35 BS01 1MD A 1 R125 E205 E206 Y547 S630 Y662 Y666 N710 R87 E167 E168 Y509 S592 Y624 Y628 N672 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=0.94nM remove_due_to_license_issue P27487 23964740 801 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 4jhq A 1.99 BS01 B6F A 1 S16 Y33 V37 T38 A39 T40 W70 F72 S75 T77 W97 S101 K111 R114 N118 S15 Y32 V36 T37 A38 T39 W69 F71 S74 T76 W96 S100 K110 R113 N117 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 201 RKCSLTGKWTNDLGSNMTIGAVNSKGEFTGTYTTAVTATSNEIKESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRLRT 4jht A 1.18 BS01 8XQ A 1 Y122 H131 D133 S145 F154 H187 I189 R204 T208 Y109 H118 D120 S132 F141 H174 I176 R191 T195 1.14.11.33 0005515,0005737,0005829,0006281,0006307,0008198,0035513,0035515,0035516,0042245,0046872,0051213,0070989,0072702 remove_due_to_license_issue P05050 26682036 301 PLAAGAVILRRFAFNAAEQLIRDINDVASQSPFRQMVTPGGYTMSVAMTNCGHLGWTTHRQGYLYSPIDPQTNKPWPAMPQSFHNLCQRAATAAGYPDFQPDACLINRYAPGAKLSLHQDKDEPDLRAPIVSVSLGLPAIFQFGGLKRNDPLKRLLLEHGDVVVWGGESRLFYHGIQPLKAGFHPLTIDCRYNLTFRQAGK 4jhz A 2.831 BS01 1KV A 1 D163 L361 E413 M447 Y468 Y472 R562 D165 L363 E408 M442 Y463 Y467 R557 D163 H296 H330 V355 F357 E413 Y468 E504 K568 D165 H298 H332 V357 F359 E408 Y463 E499 K563 3.2.1.31 0004553,0004566,0005829,0005975,0016798,0030246,0032991,0042802 remove_due_to_license_issue Ki=9.6e+2nM P05804 23690068 701 SHMLRPVETPTREIKKLDGLWAFSLDRENCGIDQRWWESALQESRAIAVPGSFNDQFADADIRNYAGNVWYQREVFIPKGWAGQRIVLRFDAVTHYGKVWVNNQEVMEHQGGYTPFEADVTPYVIAGKSVRITVCVNNELNWQTIPPGMVITDENGKKKQSYFHDFFNYAGIHRSVMLYTTPNTWVDDITVVTHVAQDCNHASVDWQVVANGDVSVELRDADQQVVATGQGTSGTLQVVNPHLWQPGEGYLYELCVTAKSQTECDIYPLRVGIRSVAVKGEQFLINHKPFYFTGFGRHEDADLRGKGFDNVLMVHDHALMDWIGANSYRTSHYPYAEEMLDWADEHGIVVIDETAAVGFNLSLNKPKELYSEEAVNGETQQAHLQAIKELIARDKNHPSVVMWSIANEPDTRPQGAREYFAPLAEATRKLDPTRPITCVNVMFCDAHTDTISDLFDVLCLNRYYGWYVQSGDLETAEKVLEKELLAWQEKLHQPIIITEYGVDTLAGLHSMYTDMWSEEYQCAWLDMYHRVFDRVSAVVGEQVWNFADFATSQGILRVGGNKKGIFTRDRKPKSAAFLLQKRWTGMNFGEKPQQGG 4jia A 1.85 BS01 1K3 A 1 V863 A880 M929 Y931 L932 G935 L983 V31 A48 M97 Y99 L100 G103 L151 D976 A978 R980 N981 D994 S1016 D144 A146 R148 N149 D162 S184 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.0006uM remove_due_to_license_issue Ki=0.600000nM, IC50=22nM O60674 23870430 1201 SGAFEDRDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 4jib A 1.72 BS02 1L6 A 1 Q812 M847 Q859 S861 F862 Q236 M271 Q283 S285 F286 3.1.4.17 0004114,0007165,0008081 ic50=45nM remove_due_to_license_issue IC50=45nM O00408 23582272 1003 AMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 4jik A 1.9 BS01 1KO A 1 E17 V23 A36 C87 S88 G90 E91 E134 N135 L137 D148 E14 V19 A32 C71 S72 G74 E75 E118 N119 L121 D132 D130 K132 E134 N135 D148 T170 D114 K116 E118 N119 D132 T154 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.018uM remove_due_to_license_issue IC50=18nM O14757 23587425 301 PFVEDWDLVQTLGEGAGEVQLAVNRVTEEAVAVKIVNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKG 4jin A 2.095 BS01 1L7 A 1 S56 A78 K80 E148 F149 I150 I211 D212 S52 A74 K76 E144 F145 I146 I207 D208 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004711,0005524,0006338,0006468,0016787,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0046872,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue O28471 23523885 301 KKIESYLDKLRIKEKDGEERKIYAEVLDGRTLKTLYKLSAKGYITAMGGVISTGKEANVFYADGVFDGKPVAMAVKIYRIETSEFDKMDEYLYGDERFDMRRISPKEKVFIWTEKEFRNLERAKEAGVSVPQPYTYMKNVLLMEFIGEDELPAPTLVELGRELKELDVEGIFNDVVENVKRLYQEAELVHADLSEYNIMYIDKVYFIDMGQAVTLRHPMAESYLERDVRNIIRFFSKYGVKADFEEMLKEVKGE 4jit B 2.8 BS01 3ZF B 1 L90 D92 T93 G95 T96 W134 I135 L88 D90 T91 G93 T94 W132 I133 2.4.2.-,2.4.2.22 0000287,0000310,0004422,0005829,0005886,0006166,0016757,0032263,0032264,0032265,0032991,0042802,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M5 23927482 201 EKYIVTWDMLQIHARKLASRLMPSEQWKGIIAVSRGGLVPGALLARELGIRHVDTVCISSYDHDNQRELKVLKRAEGDGEGFIVIDDLVDTGGTAVAIREMYPKAHFVTIFAKPAGRPLVDDYVVDIPQDTWIEQPWDMGVVFVPPISGR 4jit C 2.8 BS01 3ZF C 1 R69 D92 T93 G95 T96 W134 I135 R67 D90 T91 G93 T94 W132 I133 2.4.2.-,2.4.2.22 0000287,0000310,0004422,0005829,0005886,0006166,0016757,0032263,0032264,0032265,0032991,0042802,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M5 23927482 201 EKYIVTWDMLQIHARKLASRLMPSEQWKGIIAVSRGGLVPGALLARELGIRHVDTVCISSYDHDNQRELKVLKRAEGDGEGFIVIDDLVDTGGTAVAIREMYPKAHFVTIFAKPAGRPLVDDYVVDIPQDTWIEQPWDMGVVFVPPISGR 4jjf A 2.2 BS01 FE9 A 1 G7 G9 A62 D63 P64 P110 P111 D131 W144 F145 P146 I154 C172 A206 V207 G7 G9 A62 D63 P64 P110 P111 D131 W144 F145 P146 I154 C172 A206 V207 1.12.98.2 0006730,0015948,0016491,0019386,0047068 remove_due_to_license_issue P32440 23873755 401 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjf A 2.2 BS02 N2I A 1 C172 G205 A206 C252 C172 G205 A206 C252 1.12.98.2 0006730,0015948,0016491,0019386,0047068 Ki=10nM remove_due_to_license_issue P32440 23873755 402 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjf B 2.2 BS01 FE9 B 1 L6 G7 G9 A62 D63 P64 P110 P111 D131 W144 F145 P146 I154 A171 C172 P204 A206 L6 G7 G9 A62 D63 P64 P110 P111 D131 W144 F145 P146 I154 A171 C172 P204 A206 1.12.98.2 0006730,0015948,0016491,0019386,0047068 remove_due_to_license_issue P32440 23873755 401 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjf B 2.2 BS02 N2I B 1 C172 C252 C172 C252 1.12.98.2 0006730,0015948,0016491,0019386,0047068 Ki=10nM remove_due_to_license_issue P32440 23873755 402 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjg A 2.5 BS01 FE9 A 1 G9 A62 D63 P64 P110 D131 W144 F145 P146 I154 A171 C172 T173 A206 G9 A62 D63 P64 P110 D131 W144 F145 P146 I154 A171 C172 T173 A206 1.12.98.2 0006730,0015948,0016491,0019386,0047068 remove_due_to_license_issue P32440 23873755 401 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjg B 2.5 BS01 FE9 B 1 L6 G7 G9 A62 D63 P64 P110 D131 W144 F145 P146 I154 A171 C172 T173 P204 L6 G7 G9 A62 D63 P64 P110 D131 W144 F145 P146 I154 A171 C172 T173 P204 1.12.98.2 0006730,0015948,0016491,0019386,0047068 remove_due_to_license_issue P32440 23873755 401 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjg B 2.5 BS02 IC9 B 1 T13 K147 T13 K147 1.12.98.2 0006730,0015948,0016491,0019386,0047068 remove_due_to_license_issue P32440 23873755 402 MKLAILGAGCYRTHAASGITNFSRACEVAEMVGKPEIAMTHSTITMGAELKELAGVDEVVVADPVFDNQFTVIDDFAYEDVIEAHKEDPEKIMPQIREKVNEVAKELPKPPEGAIHFTHPEDLGFEITTDDREAVADADFIMTWFPKGDMQPDIINKFIDDIKPGAIVTHACTIPTTKFYKIFEQKHGDLVTKPETLNVTSYHPGAVPEMKGQVYIAEGYASEDAIETLFELGQKARGNAYRLPAELLGPVCDMCSALTAITYAGILSYRDSVTQVLGAPASFAQMMAKESLEQITALMEKVGIDKMEENLDPGALLGTADSMNFGASAEILPTVFEILEKRKK 4jjs A 2.2 BS01 1M9 A 1 L419 R422 M423 H475 S476 Y477 I482 V485 A486 L497 W528 L415 R418 M419 H471 S472 Y473 I478 V481 A482 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 23768906 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4jju A 1.91 BS01 1MB A 1 L419 R422 M423 H475 S476 Y477 I482 V485 A486 L497 W528 L415 R418 M419 H471 S472 Y473 I478 V481 A482 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 23768906 3002 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4jkt A 2.77 BS01 04A D 1 K325 L326 F327 L328 N329 E330 Y399 K171 L172 F173 L174 N175 E176 Y245 S291 K294 Y419 Y471 V489 S137 K140 Y265 Y317 V335 3.5.1.2 0004359,0006541 remove_due_to_license_issue D3Z7P3 23935106 701 LEDLLFYTIKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSIGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRR 4jkt B 2.77 BS01 04A B 1 K325 L326 F327 L328 N329 E330 Y399 K159 L160 F161 L162 N163 E164 Y233 S291 K294 Y419 Y471 V489 S125 K128 Y253 Y305 V323 3.5.1.2 0004359,0006541 remove_due_to_license_issue D3Z7P3 23935106 701 LEDLLFYTIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVAPDLWGVSVCTVDGQRHSIGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRR 4jkt C 2.77 BS01 04A B 1 K325 L326 F327 L328 N329 Y399 K173 L174 F175 L176 N177 Y247 S291 K294 Y419 Y471 V489 S139 K142 Y267 Y319 V337 3.5.1.2 0004359,0006541 remove_due_to_license_issue D3Z7P3 23935106 701 LEDLLFYTIEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSIGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRR 4jkt D 2.77 BS01 04A D 1 R322 K325 L326 F327 L328 N329 E330 Y399 R161 K164 L165 F166 L167 N168 E169 Y238 S291 K294 Y419 Y471 V489 S130 K133 Y258 Y310 V328 3.5.1.2 0004359,0006541 remove_due_to_license_issue D3Z7P3 23935106 701 LEDLLFYTIQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADLWGVSVCTVDGQRHSIGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRR 4jkw A 2.01 BS01 IPE A 1 K39 Y100 Q102 K37 Y98 Q100 ? Kd=69.9uM remove_due_to_license_issue EC50=71000nM, IC50=513000nM O00481 23872678 201 QFSVLGPSGPILAMVGEDADLPCHLFPTMSAETMELKWVSSSLRQVVNVYADGKEVEDRQSAPYRGRTSILRDGITAGKAALRIHNVTASDSGKYLCYFQDGDFYEKALVELKVLEHHH 4jlg A 1.896 BS02 1L8 A 1 H252 V255 D256 T266 L267 S268 Y305 Y335 G336 Y337 H339 S340 H136 V139 D140 T150 L151 S152 Y189 Y219 G220 Y221 H223 S224 Y245 H293 H297 Y305 Y335 Y129 H177 H181 Y189 Y219 2.1.1.364 0005694,0006355,0016279,0140945 remove_due_to_license_issue IC50=2.0nM, Ki=0.330000nM Q8WTS6 25136132 402 GVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDERTALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCISTNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITHQEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPNCIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHSPPGKSGPEAPEWYQVELKAFQAT 4jlh A 2.09 BS01 0L9 A 1 Q95 T125 T128 A129 W132 Q40 T70 T73 A74 W77 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=15.6uM remove_due_to_license_issue IC50=4e+2nM P12497 23615903 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKTACWWAGIKQEFESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGGYSAGERIVDIIATDIQ 4jlj A 2.0 BS01 1NM A 1 V55 Y86 F96 Q97 D133 F137 Y204 V36 Y58 F68 Q69 D105 F109 Y176 E53 R128 E34 R100 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=726.4nM remove_due_to_license_issue IC50=230nM P27707 24419380 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNELTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jlj A 2.0 BS02 1NM A 2 S59 L82 Y86 E197 G199 I200 P201 Y204 S40 L54 Y58 E169 G171 I172 P173 Y176 E53 R128 E34 R100 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=726.4nM remove_due_to_license_issue IC50=230nM P27707 24419380 302 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNELTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jlm A 2.18 BS01 1NN A 1 E53 V55 M85 Y86 P89 Q97 D133 F137 S144 Y204 E35 V37 M58 Y59 P62 Q70 D106 F110 S117 Y177 E53 R128 E35 R101 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=6.1nM remove_due_to_license_issue IC50=7.0nM P27707 24419380 301 TRIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNELTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jlm A 2.18 BS02 1NN A 2 I30 Y86 R194 E196 E197 G199 I200 P201 Y204 I12 Y59 R167 E169 E170 G172 I173 P174 Y177 E53 R128 E35 R101 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=6.1nM remove_due_to_license_issue IC50=7.0nM P27707 24419380 302 TRIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNELTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jln A 2.15 BS01 18V A 1 E53 V55 L82 Y86 P89 F96 Q97 D133 F137 Y204 E34 V36 L54 Y58 P61 F68 Q69 D105 F109 Y176 E53 R128 E34 R100 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=1.5nM remove_due_to_license_issue Ki=1.5nM, IC50=3.0nM P27707 24419380 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNELTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4jls A 2.2 BS01 3ZE A 1 L90 V91 D92 T93 G94 G95 T96 K115 W134 I135 L71 V72 D73 T74 G75 G76 T77 K96 W115 I116 2.4.2.-,2.4.2.22 0000287,0000310,0004422,0005829,0005886,0006166,0016757,0032263,0032264,0032265,0032991,0042802,0046872,0051289,0052657,0097216 Ki=2.2uM remove_due_to_license_issue P0A9M5 23927482 201 EKYIVTWDMLQIHARKLASRLMPSEQWKGIIAVSRGGLVPGALLARELGIRHVDTVCISGDGEGFIVIDDLVDTGGTAVAIREMYPKAHFVTIFAKPAGRPLVDDYVVDIPQDTWIEQPWDMGVVFVPPISGR 4jmu A 2.0 BS01 1ML A 1 L21 R22 P23 Y29 H33 W36 S77 N80 L16 R17 P18 Y24 H28 W31 S72 N75 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0005198 ic50=3.4uM remove_due_to_license_issue P12497 24024973 202 SVLSGGELDKWEKIRLRPGGKKQYKLKHIVWASRELERFAVNPGLLETSEGCRQILGQLQPSLQTGSEELRSLYNTIAVLYCVHQRIDVKDTKEALDKIEEEQNK 4jmx A 2.55 BS01 IM2 A 1 M175 Y190 H208 S223 H224 G225 C226 N228 M141 Y156 H174 S189 H190 G191 C192 N194 2.3.2.- 0005576,0008360,0009252,0016740,0016746,0018104,0042597,0071555,0071972 remove_due_to_license_issue O53638 23999293 301 PIPGVASVSPANGAVVGVAHPVVVTFTTPVTDRRAVERSIRISTPHNTTGHFEWVASNVVRWVPHRYWPPHTRVSVGVQELTEGFETGDALIGVASISAHTFTVSRNGEVLRTMPASLGKPSRPTPIGSFHAMSKERTVVMDSRTIGIPLNSSDGYLLTAHYAVRVTWSGVYVHSAPWSVNSQGYANVSHGCINLSPDNAAWYFDAVTVGDPIEVV 4jn2 A 1.71 BS01 4CC A 1 Y32 Y38 S97 T98 F100 H102 Y31 Y37 S96 T97 F99 H101 remove_due_to_license_issue 23476049 301 DVVMTQSPLSLPVTLGQPASISCKSSQSLLYTDGKTYLYWFLQRPGQSPRRLIYLVSKLDSGVPDRFSGSGSGTDFTLKISRVEAEDVGVYYCLQSTHFPHTFGGGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 4jn2 B 1.71 BS01 4CC A 1 D36 W53 S57 T58 Y107 D30 W47 S51 T52 Y101 remove_due_to_license_issue 23476049 301 VQLQESGPGLVKPSETLSLTCTVSTSYIVDWIRQPPGKGLEWIGVIWAGGSTGYNSALRSRVSITKDTSKNQFSLKLSSVTAADTAVYYCASAAYYSYYNYDGFAYWGQGTLVTVSSASTKGPSVFPLAPGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 4jn4 A 2.3 BS01 ATP A 1 G10 T11 T12 N13 K70 G196 G197 G198 E267 K270 I271 S274 G341 G342 Q343 R345 G10 T11 T12 N13 K70 G196 G197 G198 E267 K270 I271 S274 G341 G342 Q343 R345 D8 K70 E171 D194 D8 K70 E171 D194 ? 0005515,0005524,0005737,0005829,0005886,0006260,0006457,0008270,0009408,0016020,0016234,0016887,0016989,0031072,0032991,0034620,0042026,0043335,0043531,0044183,0045892,0051082,0051085,0051087,0065003,0140662,1990169 remove_due_to_license_issue P0A6Y8 23708608 1002 SGKIIGIDLGTTNSCVAIMDGTTPRVLENAEGDRTTPSIIAYTQDGETLVGQPAKRQAVTNPQNTLFAIKRLIGRRFQDEEVQRDVSIMPFKIIAADNGDAWVEVKGQKMAPPQISAEVLKKMKKTAEDYLGEPVTEAVITVPAYFNDAQRQATKDAGRIAGLEVKRIINEPTAAALAYGLDKGTGNRTIAVYDLGGGAFDISIIEIDEVDGEKTFEVLATNGDTHLGGEDFDSRLINYLVEEFKKDQGIDLRNDPLAMQRLKEAAEKAKIELSSAQQTDVNLPYITADATGPKHMNIKVTRAKLESLVEDLVNRSIEPLKVALQDAGLSVSDIDDVILVGGQTRMPMVQKKVAEFFGKEPRKDVNPDEAVAIGAAVQGGVLTGDVKDVLLLDVTPLSLGIETMGGVMTTLIAKNTTIPTKHSQVFSMGGAVTIHVLQGERKRAADNKSLGQFNLDGINPAPRGMPQIEVTFDIDADGILHVSAKDKNSGKEQKITIKASSGLNEDEIQKMVRDAEANAEADRKFEELVQTRNQGDHLLHSTRKQVEEAGDKLPADDKTAIESALTALETALKGEDKAAIEAKMQELAQVSQKLMEIAQQ 4jn4 B 2.3 BS01 ATP B 1 G10 T11 T12 N13 K70 G196 G197 G198 A199 E267 K270 I271 S274 G341 G342 Q343 R345 G10 T11 T12 N13 K70 G196 G197 G198 A199 E267 K270 I271 S274 G341 G342 Q343 R345 D8 K70 E171 D194 D8 K70 E171 D194 ? 0005515,0005524,0005737,0005829,0005886,0006260,0006457,0008270,0009408,0016020,0016234,0016887,0016989,0031072,0032991,0034620,0042026,0043335,0043531,0044183,0045892,0051082,0051085,0051087,0065003,0140662,1990169 remove_due_to_license_issue P0A6Y8 23708608 1002 SGKIIGIDLGTTNSCVAIMDGTTPRVLENAEGDRTTPSIIAYTQDGETLVGQPAKRQAVTNPQNTLFAIKRLIGRRFQDEEVQRDVSIMPFKIIAADNGDAWVEVKGQKMAPPQISAEVLKKMKKTAEDYLGEPVTEAVITVPAYFNDAQRQATKDAGRIAGLEVKRIINEPTAAALAYGLDKGTGNRTIAVYDLGGGAFDISIIEIDEVDGEKTFEVLATNGDTHLGGEDFDSRLINYLVEEFKKDQGIDLRNDPLAMQRLKEAAEKAKIELSSAQQTDVNLPYITADATGPKHMNIKVTRAKLESLVEDLVNRSIEPLKVALQDAGLSVSDIDDVILVGGQTRMPMVQKKVAEFFGKEPRKDVNPDEAVAIGAAVQGGVLTGDVKDVLLLDVTPLSLGIETMGGVMTTLIAKNTTIPTKHSQVFSMGGAVTIHVLQGERKRAADNKSLGQFNLDGINPAPRGMPQIEVTFDIDADGILHVSAKDKNSGKEQKITIKASSGLNEDEIQKMVRDAEANAEADRKFEELVQTRNQGDHLLHSTRKQVEEAGDKLPADDKTAIESALTALETALKGEDKAAIEAKMQELAQVSQKLMEIAQQ 4jnc A 1.96 BS01 1LF A 1 F267 D335 W336 M339 P361 F381 Y383 M419 Y466 V498 L499 H524 F31 D99 W100 M103 P125 F145 Y147 M183 Y230 V262 L263 H288 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F31 H98 D99 W100 N123 N142 Y147 Y230 D260 H288 3.1.3.76,3.3.2.10 0003824 ic50=3nM remove_due_to_license_issue IC50=100nM P34913 23664879 601 GSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 4jne A 1.96 BS01 ATP A 1 G10 T11 T12 N13 K70 G196 G197 G198 A199 G229 E267 K270 I271 S274 G341 G342 Q343 R345 G10 T11 T12 N13 K70 G196 G197 G198 A199 G229 E267 K270 I271 S274 G341 G342 Q343 R345 D8 K70 E171 D194 D8 K70 E171 D194 ? 0005515,0005524,0005737,0005829,0005886,0006260,0006457,0008270,0009408,0016020,0016234,0016887,0016989,0031072,0032991,0034620,0042026,0043335,0043531,0044183,0045892,0051082,0051085,0051087,0065003,0140662,1990169 remove_due_to_license_issue P0A6Y8 23708608 1002 SGKIIGIDLGTTNSCVAIMDGTTPRVLENAEGDRTTPSIIAYTQDGETLVGQPAKRQAVTNPQNTLFAIKRLIGRRFQDEEVQRDVSIMPFKIIAADNGDAWVEVKGQKMAPPQISAEVLKKMKKTAEDYLGEPVTEAVITVPAYFNDAQRQATKDAGRIAGLEVKRIINEPTAAALAYGLDKGTGNRTIAVYDLGGGAFDISIIEIDEVDGEKTFEVLATNGDTHLGGEDFDSRLINYLVEEFKKDQGIDLRNDPLAMQRLKEAAEKAKIELSSAQQTDVNLPYITADATGPKHMNIKVTRAKLESLVEDLVNRSIEPLKVALQDAGLSVSDIDDVILVGGQTRMPMVQKKVAEFFGKEPRKDVNPDEAVAIGAAVQGGVLTGDVKDVLLLDVTPLSLGIETMGGVMTTLIAKNTTIPTKHSQVFSMGGAVTIHVLQGERKRAADNKSLGQFNLDGINPAPRGMPQIEVTFDIDADGILHVSAKDKNSGKEQKITIKASSGLNEDEIQKMVRDAEANAEADRKFEELVQTRNQGDHLLHSTRKQVEEAGDKLPADDKTAIESALTALETALKGEDKAAIEAKMQELAQVSQKLMEIAQQ 4jne B 1.96 BS01 ATP B 1 G10 T11 T12 N13 K70 G196 G197 G198 A199 G229 E267 K270 I271 S274 G341 G342 Q343 R345 G10 T11 T12 N13 K70 G196 G197 G198 A199 G229 E267 K270 I271 S274 G341 G342 Q343 R345 D8 K70 E171 D194 D8 K70 E171 D194 ? 0005515,0005524,0005737,0005829,0005886,0006260,0006457,0008270,0009408,0016020,0016234,0016887,0016989,0031072,0032991,0034620,0042026,0043335,0043531,0044183,0045892,0051082,0051085,0051087,0065003,0140662,1990169 remove_due_to_license_issue P0A6Y8 23708608 1002 SGKIIGIDLGTTNSCVAIMDGTTPRVLENAEGDRTTPSIIAYTQDGETLVGQPAKRQAVTNPQNTLFAIKRLIGRRFQDEEVQRDVSIMPFKIIAADNGDAWVEVKGQKMAPPQISAEVLKKMKKTAEDYLGEPVTEAVITVPAYFNDAQRQATKDAGRIAGLEVKRIINEPTAAALAYGLDKGTGNRTIAVYDLGGGAFDISIIEIDEVDGEKTFEVLATNGDTHLGGEDFDSRLINYLVEEFKKDQGIDLRNDPLAMQRLKEAAEKAKIELSSAQQTDVNLPYITADATGPKHMNIKVTRAKLESLVEDLVNRSIEPLKVALQDAGLSVSDIDDVILVGGQTRMPMVQKKVAEFFGKEPRKDVNPDEAVAIGAAVQGGVLTGDVKDVLLLDVTPLSLGIETMGGVMTTLIAKNTTIPTKHSQVFSMGGAVTIHVLQGERKRAADNKSLGQFNLDGINPAPRGMPQIEVTFDIDADGILHVSAKDKNSGKEQKITIKASSGLNEDEIQKMVRDAEANAEADRKFEELVQTRNQGDHLLHSTRKQVEEAGDKLPADDKTAIESALTALETALKGEDKAAIEAKMQELAQVSQKLMEIAQQ 4jnj A 1.902 BS01 BTN A 1 S27 Y43 N45 A47 G49 W79 S88 T90 W108 D128 S16 Y32 N34 A36 G40 W63 S72 T74 W92 D109 0009374 remove_due_to_license_issue 23670729 201 GAEAGITGTWYNQSGSTFTVTAGADGNLTGQYENRAQGTGCQNSPYTLTGRYNGTKLEWRVEWNNSTENCHSRTEWRGQYQGGAEARINTQWNLTYEGGSGPATEQGQDTFTKVK 4jnm A 2.2 BS01 1LJ A 1 H191 F193 D219 V242 A244 P273 S275 I309 R311 I351 H175 F177 D203 V226 A228 P257 S259 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=3nM remove_due_to_license_issue IC50=3.0nM P43490 23668988 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4jnm B 2.2 BS01 1LJ B 1 H191 F193 D219 V242 A244 P273 S275 I309 R311 I351 H175 F177 D203 V226 A228 P257 S259 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=3nM remove_due_to_license_issue IC50=3.0nM P43490 23668988 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEAA 4joa A 2.7 BS01 3DK A 1 A1148 E1167 I1171 I1194 L1196 E1197 M1199 L1256 G1269 A28 E38 I42 I65 L67 E68 M70 L121 G134 D1249 A1251 R1253 N1254 D1270 D114 A116 R118 N119 D135 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=29nM Q9UM73 23880539 1501 DLKEVPRKNITLIRGLGVYEGQVSLQVAVKTLPDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYAMLPVKWMPPEAGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALP 4joo A 1.8 BS01 1M4 A 1 L78 D80 Y119 F156 W163 I166 D276 G278 L34 D36 Y75 F112 W119 I122 D232 G234 D80 S83 N85 A87 Y119 D276 T279 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=36830nM remove_due_to_license_issue P56817 23537249 503 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4jp9 A 1.8 BS01 1M5 A 1 Q60 G61 D80 F156 I158 W163 I166 D276 G278 T279 Q16 G17 D36 F112 I114 W119 I122 D232 G234 T235 D80 S83 N85 A87 Y119 D276 T279 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=24nM remove_due_to_license_issue P56817 23537249 503 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4jpa A 2.0 BS05 AZ6 A 1 L185 A186 L218 H222 E223 H232 A238 L239 F241 P242 I243 T245 Y246 L82 A83 L115 H119 E120 H129 A135 L136 F138 P139 I140 T142 Y143 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=3.3nM remove_due_to_license_issue P45452 23810497 306 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYHFMLPDDDVQGIQSLYGPGDED 4jpc A 1.8 BS01 1M6 A 1 Q60 G61 D80 S83 Y119 F156 I158 I166 D276 G278 T279 Q16 G17 D36 S39 Y75 F112 I114 I122 D232 G234 T235 D80 S83 N85 A87 Y119 D276 T279 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=94nM remove_due_to_license_issue P56817 23537249 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4jpe A 1.8 BS01 1M7 A 1 Q60 G61 D80 Y119 I158 I166 D276 G278 Q16 G17 D36 Y75 I114 I122 D232 G234 D80 S83 N85 A87 Y119 D276 T279 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=48nM remove_due_to_license_issue P56817 23537249 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4jps A 2.2 BS01 1LT A 1 W780 K802 Y836 I848 V851 S854 H855 Q859 M922 I932 W726 K748 Y782 I794 V797 S800 H801 Q805 M860 I870 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue IC50=5.0nM P42336 23726034 1102 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRISTTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTTKMDWIFHT 4jpx A 1.55 BS01 PHE A 1 A158 Y159 K165 L175 T254 P256 F258 A150 Y151 K157 L167 T246 P248 F250 H138 H143 E184 P203 H130 H135 E176 P195 1.14.16.1 0004497,0004505,0005506,0006559,0009072,0016714,0019293,0046872 remove_due_to_license_issue P30967 23860686 301 FVVPDITTRKNVGLSHDANDFTLPQPLDRYSAEDHATWATLYQRQCKLLPGRACDEFLEGLERLEVDADRVPDFNKLNEKLMAATGWKIVAVPGLIPDDVFFEHLANRRFPVTWWLREPHQLLQEPDVFHDLFGHVPLLINPVFADYLEAYGKGGVKAKALGALPMLARLYWYTVEFGLINTPAGMRIYGAGILPSKSESIYCLDSASPNRVGFDLMRIMNTRYRIDTFQKTYFVIDSFKQLFDATAPDFAPLYLQLADAQPWGAGDIAPDDLVL 4jpy A 2.13 BS02 PHE A 1 A158 Y159 K165 L175 T254 A255 P256 D257 F258 A143 Y144 K150 L160 T239 A240 P241 D242 F243 H138 H143 E184 S203 H123 H128 E169 S188 1.14.16.1 0004497,0004505,0005506,0006559,0009072,0016714,0019293,0046872 remove_due_to_license_issue P30967 23860686 302 PDITTRKNVGLSHDANDFTLPQPLDRYSAEDHATWATLYQRQCKLLPGRACDEFLEGLERLEVDADRVPDFNKLNEKLMAATGWKIVAVPGLIPDDVFFEHLANRRFPVTWWLREPHEPDVFHDLFGHVPLLINPVFADYLEAYGKGGVKAKALGALPMLARLYWYTVEFGLINTPAGMRIYGAGILSSKSESIYCLDSASPNRVGFDLMRIMNTRYRIDTFQKTYFVIDSFKQLFDATAPDFAPLYLQLADAQPWGAGDIAPDDLVL 4jq7 A 2.73 BS01 KJQ A 1 L694 V702 A719 K721 T766 M769 G772 L820 L23 V31 A48 K50 T95 M98 G101 L149 D813 A815 R817 N818 D831 G850 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=223nM P00533 23611691 1001 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDMDDVVDADEYLIP 4jq8 A 2.83 BS01 KJ8 A 1 L694 F699 V702 A719 K721 T766 M769 G772 N818 L820 D831 L23 F28 V31 A48 K50 T95 M98 G101 N147 L149 D160 D813 A815 R817 N818 D831 G850 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=8.0nM P00533 23611691 1001 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDMDDVVDADEYLIP 4jql A 1.72 BS01 VJ6 A 1 N51 D54 A55 K58 D102 N106 L107 G135 V136 G137 F138 N42 D45 A46 K49 D93 N97 L98 G126 V127 G128 F129 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=1uM remove_due_to_license_issue P07900 23554224 301 QPMEEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4jr3 A 2.7 BS01 KJR A 1 L694 V702 A719 K721 T766 M769 G772 R817 L820 D831 L23 V31 A48 K50 T95 M98 G101 R146 L149 D160 D813 A815 R817 N818 D831 G850 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=218nM P00533 23611691 1001 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDMDDVVDADEYLIP 4jr5 A 1.906 BS01 1LS A 1 H191 F193 D219 V242 A244 S275 R311 I351 A379 H175 F177 D203 V226 A228 S259 R295 I335 A363 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.007uM remove_due_to_license_issue IC50=9.9nM P43490 23617784 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4jr5 B 1.906 BS01 1LS B 1 H191 F193 D219 V242 A244 S275 R311 I351 A379 H175 F177 D203 V226 A228 S259 R295 I335 A363 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.007uM remove_due_to_license_issue IC50=9.9nM P43490 23617784 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4jrg A 1.9 BS01 I09 A 1 L50 I57 M58 F82 V89 K90 H92 I95 Y96 L30 I37 M38 F62 V69 K70 H72 I75 Y76 2.3.2.27 0005634,0043066,0051726 ic50=196nM remove_due_to_license_issue P56273 23808545 201 EKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLV 4jrv A 2.8 BS01 KJV A 1 L694 V702 A719 K721 T766 Q767 M769 G772 N818 L820 D831 L23 V31 A48 K50 T92 Q93 M95 G98 N144 L146 D157 D813 A815 R817 N818 D831 G850 D139 A141 R143 N144 D157 G176 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=29nM P00533 23611691 1001 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDMDDVVDADEYLIP 4jsa A 1.5 BS02 FB2 A 1 H96 H119 V121 L198 T199 T200 H93 H116 V118 L194 T195 T196 H64 D94 H96 E106 H119 T199 H61 D91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11uM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 23706138 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFDFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4jsa A 1.5 BS03 FB2 A 2 W5 H15 W16 D19 W2 H12 W13 D16 H64 D94 H96 E106 H119 T199 H61 D91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11uM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 23706138 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFDFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4jsc A 2.5 BS01 1OY A 1 L50 G54 M58 V89 K90 H92 I95 Y96 L29 G33 M37 V68 K69 H71 I74 Y75 2.3.2.27 0005634,0043066,0051726 ic50=74nM remove_due_to_license_issue P56273 23808545 201 KLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLV 4jsr A 1.7 BS02 1NQ A 1 A146 D156 F157 F180 N229 I230 D231 H248 V292 F293 F294 E296 L298 A26 D36 F37 F60 N109 I110 D111 H128 V172 F173 F174 E176 L178 P155 D156 F157 R158 N229 D231 H248 P35 D36 F37 R38 N109 D111 H128 2.3.1.286 0017136,0051287,0070403 ic50=0.004uM remove_due_to_license_issue IC50=4.0nM Q9NTG7 23570514 402 GKLSLQDVAELIRARACQRVVVMVGAGISTPSGIPDFRSPGSGLYSNLQQYDLPYPEAIFELPFFFHNPKPFFTLAKELYPGNYKPNVTHYFLRLLHDKGLLLRLYTQNIDGLERVSGIPASKLVEAHGTFASATCTVCQRPFPGEDIRADVMADRVPRCPVCTGVVKPDIVFFGEPLPQRFLLHVVDFPMADLLLILGTSLEVEPFASLTEAVRSSVPRLLINRDLVGPLAWHPRSRDVAQLGDVVHGVESLVELLGWTEEMRDLVQRETGKL 4jss A 1.5 BS02 BEW A 1 Q92 D94 H96 H119 V121 T200 Q89 D91 H93 H116 V118 T196 H64 D94 H96 E106 H119 T199 H61 D91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=500uM remove_due_to_license_issue P00918 23706138 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFDFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4jsz A 1.9 BS02 FB2 A 1 W5 N11 H15 D19 W2 N8 H12 D16 H64 C94 H96 E106 H119 T199 H61 C91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5000uM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 23706138 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFCFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4jsz A 1.9 BS03 FB2 A 2 C94 H96 H119 V121 L198 T199 T200 C91 H93 H116 V118 L194 T195 T196 H64 C94 H96 E106 H119 T199 H61 C91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5000uM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 23706138 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFCFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4jt8 A 2.26 BS02 1NR A 1 A146 D156 F157 F180 N229 I230 D231 H248 V292 F294 A27 D37 F38 F61 N110 I111 D112 H129 V173 F175 P155 D156 F157 R158 N229 D231 H248 P36 D37 F38 R39 N110 D112 H129 2.3.1.286 0017136,0051287,0070403 ic50=0.033uM remove_due_to_license_issue IC50=33nM Q9NTG7 23570514 402 KGKLSLQDVAELIRARACQRVVVMVGAGISTPSGIPDFRSPGSGLYSNLQQYDLPYPEAIFELPFFFHNPKPFFTLAKELYPGNYKPNVTHYFLRLLHDKGLLLRLYTQNIDGLERVSGIPASKLVEAHGTFASATCTVCQRPFPGEDIRADVMADRVPRCPVCTGVVKPDIVFFGEPLPQRFLLHVVDFPMADLLLILGTSLEVEPFASLTEAVRSSVPRLLINRDLVGPLAWHPRSRDVAQLGDVVHGVESLVELLGWTEEMRDLVQRETGK 4jt9 A 2.24 BS02 1NS A 1 A146 D156 F157 F180 N229 I230 D231 H248 V292 A27 D37 F38 F61 N110 I111 D112 H129 V173 P155 D156 F157 R158 N229 D231 H248 P36 D37 F38 R39 N110 D112 H129 2.3.1.286 0017136,0051287,0070403 ic50=0.0072uM remove_due_to_license_issue IC50=7.2nM Q9NTG7 23570514 402 KGKLSLQDVAELIRARACQRVVVMVGAGISTPSGIPDFRSPGSGLYSNLQQYDLPYPEAIFELPFFFHNPKPFFTLAKELYPGNYKPNVTHYFLRLLHDKGLLLRLYTQNIDGLERVSGIPASKLVEAHGTFASATCTVCQRPFPGEDIRADVMADRVPRCPVCTGVVKPDIVFFGEPLPQRFLLHVVDFPMADLLLILGTSLEVEPFASLTEAVRSSVPRLLINRDLVGPLAWHPRSRDVAQLGDVVHGVESLVELLGWTEEMRDLVQRETGK 4ju3 A 2.0 BS01 1O1 A 1 L419 R422 H475 S476 Y477 I482 R490 L497 W528 L415 R418 H471 S472 Y473 I478 R486 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.085uM remove_due_to_license_issue O92972 24176401 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4ju4 A 2.4 BS01 1O3 A 1 L419 R422 M423 H475 S476 Y477 I482 L497 W528 L415 R418 M419 H471 S472 Y473 I478 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.34uM remove_due_to_license_issue O92972 24176401 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4ju6 A 2.2 BS01 1O6 A 1 L419 H475 S476 Y477 I482 L497 W528 L415 H471 S472 Y473 I478 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.67uM remove_due_to_license_issue O92972 24176401 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4ju7 A 2.2 BS01 1O6 A 1 L419 H475 S476 Y477 I482 L497 W528 L415 H471 S472 Y473 I478 L493 W524 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.67uM remove_due_to_license_issue O92972 24176401 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4jv6 B 1.87 BS01 18F B 1 M20 W32 A47 R61 Q78 I129 M19 W30 A45 R59 Q76 I125 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=217nM remove_due_to_license_issue Kd=2400nM O43924 23698361 201 SAKDERAREILRGFKLNWMNLRDATGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAASQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 4jv6 B 1.87 BS02 18F B 2 I53 L54 C56 W90 I109 A111 M117 L147 Y149 I51 L52 C54 W88 I107 A109 M113 L143 Y145 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=217nM remove_due_to_license_issue Kd=2400nM O43924 23698361 202 SAKDERAREILRGFKLNWMNLRDATGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAASQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 4jv7 A 2.2 BS01 1MN A 1 L54 F55 L57 G58 Q59 I61 M62 V93 I99 L29 F30 L32 G33 Q34 I36 M37 V68 I74 2.3.2.27 0005634,0043066,0051726 ic50=1uM remove_due_to_license_issue IC50=2000nM Q00987 23597064 201 TLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4jv8 B 1.45 BS01 1M1 B 1 L17 M20 W32 L38 R61 Q78 W90 L147 L16 M19 W31 L37 R60 Q77 W89 L144 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 remove_due_to_license_issue O43924 23698361 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAASQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 4jv8 B 1.45 BS02 1M1 B 2 I53 C56 V80 E88 I109 A111 M117 Y149 I52 C55 V79 E87 I108 A110 M114 Y146 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 remove_due_to_license_issue O43924 23698361 202 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAASQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 4jv9 A 2.5 BS01 1MO A 1 L54 F55 G58 Q59 I61 M62 V93 I99 L29 F30 G33 Q34 I36 M37 V68 I74 2.3.2.27 0005634,0043066,0051726 ic50=1.8uM remove_due_to_license_issue IC50=1800nM Q00987 23597064 201 TLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4jvb B 1.75 BS01 1M0 B 1 M20 L22 W32 V49 I53 R61 Q78 V80 I109 A111 M117 I129 L147 Y149 M19 L21 W31 V48 I52 R60 Q77 V79 I108 A110 M113 I125 L143 Y145 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=39nM remove_due_to_license_issue Kd=39nM O43924 23698361 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAAQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 4jve A 2.3 BS01 1MQ A 1 L54 F55 L57 G58 Q59 I61 M62 I99 L37 F38 L40 G41 Q42 I44 M45 I81 2.3.2.27 0005634,0043066,0051726 ic50=0.086uM remove_due_to_license_issue Q00987 23597064 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLGVPSFSVKEHRKIYTMIYRNLVVV 4jvh A 3.501 BS01 rna D 0 G100 R101 L103 G104 P105 R106 G107 K111 K120 M122 V123 R124 R130 K190 L194 L197 A198 Y204 G72 R73 L75 G76 P77 R78 G79 K83 K92 M94 V95 R96 R102 K162 L166 L169 A170 Y176 ? 0003676,0003723 remove_due_to_license_issue Q96PU8 23630077 4 ~ 11 KPTPDYLMQLMNDKKLMSNHLERLLDEEISRVRKDMYNDTSAELPDAVGPIVQLQEKLYVPVKEYPDFNFVGRILGPRGLTAKQLEAETGCKIMVRGKGSMRDKKKEEQNRGKPNWEHLNEDLHVLITVEDAQNRAEIKLKRAVEEVKKLLVPAAEGEDSLKKMQLMELAILNGTY 4jvi A 2.9 BS01 QZN A 1 I149 A168 L207 L208 I236 Y258 I56 A75 L114 L115 I143 Y165 ? remove_due_to_license_issue A0A0H2Z7A6 23935486 401 NLRVLLDTAIPPSFCDTVSSVLLDDFNMVSLIRTSPADSLATIKQDNAEIDIAITIDEELKISRFNQCVLGYTKAFVVAHPQHPLCNASLHSIASLANYRQISLGSRSGQHSNLLRPVSDKVLFVENFDDMLRLVEAGVGWGIAPHYFVEERLRNGTLAVLSELYEPGGIDTKVYCYYNTALESERSFLRFLESARQRLRELG 4jvj F 2.8 BS01 1MV F 1 F99 D103 M106 R112 T167 Q171 K200 T201 Y204 Q240 D243 F92 D96 M99 R105 T160 Q164 K193 T194 Y197 Q233 D236 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=390nM, Kd=3200nM P14324 23998921 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 4jvq A 2.4 BS01 1ML A 1 H475 S476 Y477 I482 R490 P496 L497 W528 H472 S473 Y474 I479 R487 P493 L494 W525 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.63uM remove_due_to_license_issue O92972 24024973 3002 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHS 4jwk A 1.87 BS01 CTN A 1 H22 Y68 M69 N70 N116 L150 H22 Y68 M69 N70 N116 L150 H22 N70 D95 N116 H22 N70 D95 N116 3.1.1.29 0004045,0005737,0006412,0016787 Kd=5.3nM remove_due_to_license_issue D0C9L6 23844024 201 MSNISLIVGLGNPGSEYAQTRHNAGFWFVEQLADKYGITLKNDPKFHGISGRGNIEGHDVRLLLPMTYMNRSGQSVVPFSKFYQIAPEAILIAHDELDMNPGVIRLKTGGGHGGHNGLRDIVPHIGPNFHRLRIGIGHPGSKERVSGHVLGKAPSNEQSLMDGAIDHALSKVKLLVQGQVPQAMNQINAYKPA 4jwr A 2.35 BS01 1MY A 1 L54 I61 H96 I99 L36 I43 H74 I77 2.3.2.27 0005634,0043066,0051726 ic50=0.61uM remove_due_to_license_issue IC50=610nM Q00987 23597064 201 IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4jx7 A 2.4 BS02 1N6 A 1 L44 G45 A65 E121 R122 V126 D128 L174 L12 G13 A33 E89 R90 V94 D96 L142 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=123nM remove_due_to_license_issue P11309 23936194 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4jx9 A 1.4 BS01 URI A 1 N12 Y17 H22 M69 N70 N116 N12 Y17 H22 M69 N70 N116 H22 N70 D95 N116 H22 N70 D95 N116 3.1.1.29 0004045,0005737,0006412,0016787 Kd=1.4nM remove_due_to_license_issue D0C9L6 23844024 201 MSNISLIVGLGNPGSEYAQTRHNAGFWFVEQLADKYGITLKNDPKFHGISGRGNIEGHDVRLLLPMTYMNRSGQSVVPFSKFYQIAPEAILIAHDELDMNPGVIRLKTGGGHGGHNGLRDIVPHIGPNFHRLRIGIGHPGSKERVSGHVLGKAPSNEQSLMDGAIDHALSKVKLLVQGQVPQAMNQINAYKPA 4jxs B 1.9 BS01 18U B 1 S64 Q120 N152 V211 S212 G317 A318 T319 G320 S61 Q117 N149 V208 S209 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=18uM remove_due_to_license_issue P00811 24835785 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4jxv A 1.76 BS01 1MU A 1 S64 L119 N152 V211 S212 Y221 G317 A318 S61 L116 N149 V208 S209 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=31uM remove_due_to_license_issue P00811 24835785 402 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4jxw A 2.3 BS01 1MW A 1 S64 L119 Q120 N152 H210 V211 S212 G317 A318 T319 G320 S61 L116 Q117 N149 H207 V208 S209 G314 A315 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=19uM remove_due_to_license_issue P00811 24835785 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4jxx A 2.3 BS01 rna B 0 Q13 E34 T68 N69 R130 R133 T135 L136 G168 P181 F182 I183 V189 R192 K194 M210 Y211 F233 Q234 D235 R238 R312 I313 T316 K317 Q318 D319 N320 T321 E323 A325 S326 S329 N336 R341 P369 N370 Q399 R402 R410 R412 N413 V455 Q517 E519 R520 L544 R545 T547 W548 Q7 E28 T62 N63 R124 R127 T129 L130 G162 P175 F176 I177 V183 R186 K188 M204 Y205 F227 Q228 D229 R232 R306 I307 T310 K311 Q312 D313 N314 T315 E317 A319 S320 S323 N330 R335 P363 N364 Q393 R396 R404 R406 N407 V443 Q505 E507 R508 L532 R533 T535 W536 E34 R260 K270 E28 R254 K264 6.1.1.18 0000166,0004812,0004819,0005524,0005737,0005829,0006412,0006418,0006424,0006425,0043039 remove_due_to_license_issue P00962 23727144 902 ~ 976 PTNFIRQIIDEDLASGKHTTVHTRFPPEPNGYLHIGHAKSICLNFGIAQDYKGQCNLRFDDTNPVKEDIEYVESIKNDVEWLGFHWSGNVRYSSDYFDQLHAYAIELINKGLAYVDELTPEQIREYRGTLTQPGKNSPYRDRSVEENLALFEKMRAGGFEEGKACLRAKIDMASPFIVMRDPVLYRIKFAEHHQTGNKWCIYPMYDFTHCISDALEGITHSLCTLEFQDNRRLYDWVLDNITIPVHPRQYEFSRLNLEYTVMSKRKLNLLVTDKHVEGWDDPRMPTISGLRRRGYTAASIREFCKRIGVTKQDNTIEMASLESCIREDLNENAPRAMAVIDPVKLVIENYQGEGEMVTMPNHPNKPEMGSRQVPFSGEIWIDRADFREEANKQYKRLVLGKEVRLRNAYVIKAERVEKDAEGNITTIFCTYDADTLSRKVKGVIHWVSAAHALPVEIRLYDRLFSVPNPGAADDFLSVINPESLVIKQGFAEPSLKDAVAGKAFQFEREGYFCLDSRHSTAEKPVFNRTVGLRDTW 4jxz A 2.4 BS01 rna B 0 Q13 E34 T68 N69 P126 R130 R133 T135 L136 G168 P181 F182 I183 R192 K194 M210 Y211 F233 Q234 D235 R238 I313 T316 K317 Q318 D319 N320 T321 E323 S326 S329 N336 R341 N370 Q399 R402 R410 R412 L442 S443 V455 Q517 E519 R520 R545 T547 W548 Q7 E28 T62 N63 P120 R124 R127 T129 L130 G162 P175 F176 I177 R186 K188 M204 Y205 F227 Q228 D229 R232 I307 T310 K311 Q312 D313 N314 T315 E317 S320 S323 N330 R335 N364 Q393 R396 R404 R406 L436 S437 V445 Q507 E509 R510 R535 T537 W538 E34 R260 K270 E28 R254 K264 6.1.1.18 0000166,0004812,0004819,0005524,0005737,0005829,0006412,0006418,0006424,0006425,0043039 remove_due_to_license_issue P00962 23727144 902 ~ 976 PTNFIRQIIDEDLASGKHTTVHTRFPPEPNGYLHIGHAKSICLNFGIAQDYKGQCNLRFDDTNPVKEDIEYVESIKNDVEWLGFHWSGNVRYSSDYFDQLHAYAIELINKGLAYVDELTPEQIREYRGTLTQPGKNSPYRDRSVEENLALFEKMRAGGFEEGKACLRAKIDMASPFIVMRDPVLYRIKFAEHHQTGNKWCIYPMYDFTHCISDALEGITHSLCTLEFQDNRRLYDWVLDNITIPVHPRQYEFSRLNLEYTVMSKRKLNLLVTDKHVEGWDDPRMPTISGLRRRGYTAASIREFCKRIGVTKQDNTIEMASLESCIREDLNENAPRAMAVIDPVKLVIENYQGEGEMVTMPNHPNKPEMGSRQVPFSGEIWIDRADFREEANKQYKRLVLGKEVRLRNAYVIKAERVEKDAEGNITTIFCTYDADTLSKGRKVKGVIHWVSAAHALPVEIRLYDRLFSVPNPGAADDFLSVINPESLVIKQGFAEPSLKDAVAGKAFQFEREGYFCLDSRHSTAEKPVFNRTVGLRDTW 4jyb A 2.1 BS01 GNP A 1 P64 G65 G67 K68 S69 T70 N201 K202 D204 S241 L243 P58 G59 G61 K62 S63 T64 N195 K196 D198 S235 L237 ? 0003924,0005525,0005737,0046872 remove_due_to_license_issue C5AP93 23873214 401 DMDTLRERLLAGDRAALARAITLAESRRADHRAAVRDLIDAVLPQTGRAIRVGITGVPGVGKSTTIDALGSLLTAAGHKVAVLAVDPSSTRTGGSILGDKTRMARLAIDRNAFIRPSPSSGTLGGVAAKTRETMLLCEAAGFDVILVETVGVGQSETAVADLTDFFLVLMLPGAGDELQGIKKGIFELADMIAVNKADDGDGERRASAAASEYRAALHILTPPSATWTPPVVTISGLHGKGLDSLWSRIEDHRSKLTATGEIAGKRREQDVKWMWALVHERLHQRLVGSAEVRQATAEAERAVAGGEHSPAAGADAIATLIGL 4jyc D 2.2 BS01 GDP D 1 G65 V66 G67 K68 S69 T70 N201 K202 D204 S241 L243 G60 V61 G62 K63 S64 T65 N188 K189 D191 S228 L230 ? 0003924,0005525,0005737,0046872 remove_due_to_license_issue C5AP93 23873214 501 PDMDTLRERLLAGDRAALARAITLAESRRADHRAAVRDLIDAVLPQTGRAIRVGITGVPGVGKSTTIDALGSLLTAAGHKVAVLAVDPSSTRTTRMARLAIDRNAFIRPSPSSGTLGGVAAKTRETMLLCEAAGFDVILVETVGVGQSETAVADLTDFFLVLMLPGAGDELQGIKKGIFELADMIAVNKADDGDGERRASAAASEYRAALHILTPPSATWTPPVVTISGLHGKGLDSLWSRIEDHRSKLTATGEIAGKRREQDVKWMWALVHERLHQRLVGSAEVRQATAEAERAVAGGEHSPAAGADAIATLI 4jym A 1.35 BS01 KKN A 1 Y124 F134 F157 F194 A219 Y123 F133 F156 F193 A218 F26 S95 V96 K216 F25 S94 V95 K215 ? 0005515,0005634,0005737,0005829,0009640,0009704,0016787,0080167 remove_due_to_license_issue Q9SZU7 23613584 301 GVVEEAHNVKVIGSGEATIVLGHGFGTDQSVWKHLVPHLVDDYRVVLYDNMGAGTTNPDYFDFDRYSNLEGYSFDLIAILEDLKIESCIFVGHSVSAMIGVLASLNRPDLFSKIVMISASPRYVNDVDYQGGFEQEDLNQLFEAIRSNYKAWCLGFAPLAVGGDMDSIAVQEFSRTLFNMRPDIALSVGQTIFQSDMRQILPFVTVPCHILQSVKDLAVPVVVSEYLHANLGCESVVEVIPSDGHLPQLSSPDSVIPVILRHIRNDI 4jyt A 2.0 BS01 N4A A 1 I41 C42 H57 C58 Y60G D189 S190 S195 W215 G216 G219 C220 I26 C27 H42 C43 Y52 D185 S186 S191 W212 G213 G215 C216 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 remove_due_to_license_issue Ki=40nM Q9Y5Y6 24900621 900 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 4jyu H 1.8 BS01 1OK H 1 H57 T99 P170I D189 S190 K192 S195 S214 W215 G216 G219 H41 T87 P169 D186 S187 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=10nM remove_due_to_license_issue Ki=9.7nM P08709 23845220 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4jyv H 2.19 BS01 1OJ H 1 H57 G97 T98 T99 P170I D189 S190 K192 S214 W215 G216 G219 G226 H41 G85 T86 T87 P169 D186 S187 K189 S211 W212 G213 G215 G223 3.4.21.21 0004252,0006508 Ki=17nM remove_due_to_license_issue Ki=17nM P08709 23845220 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4jyz A 2.5 BS01 rna B 0 Q13 E34 T68 N69 P126 R130 R133 T135 L136 G168 C171 P181 F182 I183 V189 R192 K194 M210 Y211 F233 Q234 D235 R238 I313 T316 K317 Q318 D319 N320 T321 E323 A325 S326 S329 N336 R341 N370 Q399 K401 R402 R410 R412 S443 K444 V455 Q517 E519 R520 L544 R545 T547 W548 Q7 E28 T62 N63 P120 R124 R127 T129 L130 G162 C165 P175 F176 I177 V183 R186 K188 M204 Y205 F227 Q228 D229 R232 I307 T310 K311 Q312 D313 N314 T315 E317 A319 S320 S323 N330 R335 N364 Q393 K395 R396 R404 R406 S437 K438 V449 Q511 E513 R514 L538 R539 T541 W542 E34 R260 K270 E28 R254 K264 6.1.1.18 0000166,0004812,0004819,0005524,0005737,0005829,0006412,0006418,0006424,0006425,0043039 remove_due_to_license_issue P00962 23727144 902 ~ 976 PTNFIRQIIDEDLASGKHTTVHTRFPPEPNGYLHIGHAKSICLNFGIAQDYKGQCNLRFDDTNPVKEDIEYVESIKNDVEWLGFHWSGNVRYSSDYFDQLHAYAIELINKGLAYVDELTPEQIREYRGTLTQPGKNSPYRDRSVEENLALFEKMRAGGFEEGKACLRAKIDMASPFIVMRDPVLYRIKFAEHHQTGNKWCIYPMYDFTHCISDALEGITHSLCTLEFQDNRRLYDWVLDNITIPVHPRQYEFSRLNLEYTVMSKRKLNLLVTDKHVEGWDDPRMPTISGLRRRGYTAASIREFCKRIGVTKQDNTIEMASLESCIREDLNENAPRAMAVIDPVKLVIENYQGEGEMVTMPNHPNKPEMGSRQVPFSGEIWIDRADFREEANKQYKRLVLGKEVRLRNAYVIKAERVEKDAEGNITTIFCTYDADTLSKDPADGRKVKGVIHWVSAAHALPVEIRLYDRLFSVPNPGAADDFLSVINPESLVIKQGFAEPSLKDAVAGKAFQFEREGYFCLDSRHSTAEKPVFNRTVGLRDTW 4jz1 A 1.9 BS01 F4D A 1 H57 T98 F99 D189 S190 Q192 G193 S195 W215 G216 G219 C220 H42 T93 F94 D185 S186 Q188 G189 S191 W212 G213 G215 C216 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 remove_due_to_license_issue Ki=200nM Q9Y5Y6 24900621 900 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 4jzb A 1.9 BS04 P2H A 1 F94 D98 R107 T163 Q167 K207 D250 K264 F94 D98 R107 T163 Q167 K207 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.1,2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Kd=342.5nM remove_due_to_license_issue Q4QBL1 24598749 405 MAHMERFQKVYEEVQEFLLGDAEKRFEMDVHRKGYLKSMMDTTCLGGKYNRGLCVVDVAEAMAKDTQMDAAAMERVLHDACVCGWMIEMLQAHFLVEDDIMDHSKTRRGKPCWYLHPGVTAQVAINDGLILLAWATQMALHYFADRPFLAEVLRVFHDVDLTTTIGQLYDVTSMVDSAKLDAKVAHANTTDYVEYTPFNHRRIVVYKTAYYTYWLPLVMGLLVSGTLEKVDKKATHKVAMVMGEYFQVQDDVMDCFTPPEKLGKIGTDIEDAKCSWLAVTFLTTAPAEKVAEFKANYGSTDPAAVAVIKQLYTEQNLLARFEEYEKAVVAEVEQLIAALEAQNAAFAASVKVLWSKTYKRQK 4jzb B 1.9 BS02 P2H B 1 F94 D98 R107 T163 Q167 K207 D250 K264 F94 D98 R107 T163 Q167 K207 D250 K264 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.1,2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Kd=342.5nM remove_due_to_license_issue Q4QBL1 24598749 402 MAHMERFQKVYEEVQEFLLGDAEKRFEMDVHRKGYLKSMMDTTCLGGKYNRGLCVVDVAEAMAKDTQMDAAAMERVLHDACVCGWMIEMLQAHFLVEDDIMDHSKTRRGKPCWYLHPGVTAQVAINDGLILLAWATQMALHYFADRPFLAEVLRVFHDVDLTTTIGQLYDVTSMVDSAKLDAKVAHANTTDYVEYTPFNHRRIVVYKTAYYTYWLPLVMGLLVSGTLEKVDKKATHKVAMVMGEYFQVQDDVMDCFTPPEKLGKIGTDIEDAKCSWLAVTFLTTAPAEKVAEFKANYGSTDPAAVAVIKQLYTEQNLLARFEEYEKAVVAEVEQLIAALEAQNAAFAASVKVLWSKTYKRQK 4jzd H 2.2 BS01 1NJ H 1 H57 T151 D189 S190 K192 G193 S195 S214 W215 G216 G219 H41 T141 D186 S187 K189 G190 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 ic50=0.005uM remove_due_to_license_issue Ki=10nM, IC50=5.0nM P08709 23927973 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4jze H 1.52 BS01 1NK H 1 H57 T151 D189 S190 K192 G193 S195 S214 W215 G216 G219 C220 H41 T141 D186 S187 K189 G190 S192 S211 W212 G213 G215 C216 3.4.21.21 0004252,0006508 ic50=0.007uM remove_due_to_license_issue IC50=7.0nM P08709 23927973 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4jzf H 1.84 BS01 1NL H 1 Q40 H57 T151 S190 C191 K192 G193 S195 S214 W215 G216 G219 C220 Q24 H41 T141 S187 C188 K189 G190 S192 S211 W212 G213 G215 C216 3.4.21.21 0004252,0006508 ic50=0.175uM remove_due_to_license_issue IC50=175nM P08709 23927973 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4jzi A 2.0 BS01 N4C A 1 H57 C58 F99 D189 S190 S195 W215 G216 H42 C43 F94 D185 S186 S191 W212 G213 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 remove_due_to_license_issue Ki=40nM Q9Y5Y6 24900621 900 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 4jzr A 2.1 BS01 4JR A 1 Y310 H313 D315 R322 H374 W389 F391 R396 Y115 H118 D120 R127 H179 W194 F196 R201 1.14.11.29 0005506,0016705,0031418 ic50=15.8nM remove_due_to_license_issue IC50=16nM Q9GZT9 24055079 402 PALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARA 4k0o A 2.15 BS01 MBG B 1 W109 S116 W109 S116 ? 0009289,0044406 remove_due_to_license_issue Q47200 24833052 1 VVSFIGSTENDVGPSQGSYSSTHAMDNLPFVYNTGYNIGYQNANVWRIGGGFCVGLDGKVDLPVVGSLDGQSIYGLTEEVGLLIWMGDTNYSRGTAMSGNSWENVFSGWCVGNYLSTQGLSVHVRPVILKRNSSAQYSVQKTSIGSIRMRPYNGSSAGSVQTTVNFSLNPFTLND 4k0y A 1.954 BS01 1OA A 1 F49 A65 K67 L120 N172 I185 D186 F17 A33 K35 L88 N140 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Ki=15nM remove_due_to_license_issue P11309 23623490 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4k10 A 2.3 BS02 NI9 A 1 D98 Q167 K207 D98 Q167 K207 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.1,2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Kd=119.5nM remove_due_to_license_issue Q4QBL1 24598749 406 MAHMERFQKVYEEVQEFLLGDAEKRFEMDVHRKGYLKSMMDTTCLGGKYNRGLCVVDVAEAMAKDTQMDAAAMERVLHDACVCGWMIEMLQAHFLVEDDIMDHSKTRRGKPCWYLHPGVTAQVAINDGLILLAWATQMALHYFADRPFLAEVLRVFHDVDLTTTIGQLYDVTSMVDSAKLDAKVAHANTTDYVEYTPFNHRRIVVYKTAYYTYWLPLVMGLLVSGTLEKVDKKATHKVAMVMGEYFQVQDDVMDCFTPPEKIGTDIEDAKCSWLAVTFLTTAPAEKVAEFKANYGSTDPAAVAVIKQLYTEQNLLARFEEYEKAVVAEVEQLIAALEAQNAAFAASVKVLWSKTYKRQ 4k10 B 2.3 BS02 NI9 B 1 D98 Q167 K207 D98 Q167 K207 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 K48 H93 D98 D102 R107 D170 K207 F246 D250 D251 2.5.1.1,2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 Kd=119.5nM remove_due_to_license_issue Q4QBL1 24598749 405 MAHMERFQKVYEEVQEFLLGDAEKRFEMDVHRKGYLKSMMDTTCLGGKYNRGLCVVDVAEAMAKDTQMDAAAMERVLHDACVCGWMIEMLQAHFLVEDDIMDHSKTRRGKPCWYLHPGVTAQVAINDGLILLAWATQMALHYFADRPFLAEVLRVFHDVDLTTTIGQLYDVTSMVDSAKLDAKVAHANTTDYVEYTPFNHRRIVVYKTAYYTYWLPLVMGLLVSGTLEKVDKKATHKVAMVMGEYFQVQDDVMDCFTPPEKLGKIGTDIEDAKCSWLAVTFLTTAPAEKVAEFKANYGSTDPAAVAVIKQLYTEQNLLARFEEYEKAVVAEVEQLIAALEAQNAAFAASVKVLWSKTY 4k18 A 2.051 BS01 1OB A 1 G45 F49 V52 A65 K67 R122 L174 I185 D186 G14 F18 V21 A34 K36 R91 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Ki=1.1nM remove_due_to_license_issue P11309 23623490 402 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLS 4k19 A 2.74 BS01 1OD A 1 S68 W79 L94 Y100 L103 Y106 K125 K134 S64 W75 L90 Y96 L99 Y102 K121 K130 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 remove_due_to_license_issue Kd=34nM P80188 23755875 206 SDLIPAPPLSKVPLQQNFQDNQFQGKWYVVGLAGNAILREDKDPQKMYATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKKVSQNREYFKITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDG 4k1b A 2.082 BS01 1OC A 1 L44 V52 A65 K67 E121 V126 D128 E171 L174 D186 L12 V20 A33 K35 E89 V94 D96 E139 L142 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Ki=0.003nM remove_due_to_license_issue Ki=0.003000nM P11309 23623490 402 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4k2f B 1.99 BS01 A08 B 1 F240 L266 L269 H284 V374 W378 P401 W402 V403 F24 L50 L53 H68 V158 W162 P185 W186 V187 S217 H239 V286 N485 T695 S1 H23 V70 N269 T479 3.5.1.97 0016787,0017000 ic50=0.04uM remove_due_to_license_issue Q9I194 24824984 805 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIRE 4k2g B 2.3 BS01 1OQ B 1 F240 M246 L266 H284 V374 W378 P401 W402 V403 F24 M30 L50 H68 V158 W162 P185 W186 V187 S217 H239 V286 N485 T695 S1 H23 V70 N269 T479 3.5.1.97 0016787,0017000 ic50=0.02uM remove_due_to_license_issue Q9I194 24824984 810 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIRE 4k2y A 2.3 BS02 ES2 A 1 A190 F191 K192 G216 R217 A168 F169 K170 G190 R191 H57 D102 K192 G193 D194 S195 G196 H45 D89 K170 G171 D172 S173 G174 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 ic50=470uM remove_due_to_license_issue IC50=470000nM P23946 23659209 303 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 4k3h A 2.45 BS01 1OM A 1 Y32 N34 F36 Y55 S89 L90 S91 Y96 F98 Y34 N36 F38 Y57 S91 L92 S93 Y98 F100 Kd=90pM remove_due_to_license_issue 23978698 201 QAVVTQEPSVTVSPGGTVILTCGSSTGAVTSGHYANWFQQKPGQAPRALIFETDKKYSWTPGRFSGSLLGAKAALTISDAQPEDEAEYYCSLSDVDGYLFGGGTQLTVL 4k3h B 2.45 BS01 1OM A 1 N34 F36 Y55 S89 S91 N36 F38 Y57 S91 S93 remove_due_to_license_issue 23978698 201 QAVVTQEPSVTVSPGGTVILTCGSSTGAVTSGHYANWFQQKPGQAPRALIFETDKKYSWTPGRFSGSLLGAKAALTISDAQPEDEAEYYCSLSDVDGYLFGGGTQLTVL 4k3k A 1.85 BS04 SFK A 1 T172 G174 H175 R176 P242 T164 G166 H167 R168 P234 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 ic50=4.44mM remove_due_to_license_issue P0A988 24090409 407 MKFTVEREHLLKPLQQVSLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4k3l A 1.5 BS01 LEU A 1 G174 R176 M362 G165 R167 M350 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 remove_due_to_license_issue P0A988 24090409 401 MKFTVEREHLLKPLQQVSPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMR 4k3l A 1.5 BS02 PHE A 1 T172 G174 P242 T163 G165 P230 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 remove_due_to_license_issue P0A988 24090409 402 MKFTVEREHLLKPLQQVSPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMR 4k3n A 2.0 BS04 1OT A 1 K374 D379 K386 M392 M396 F398 D399 D459 E461 T486 L487 L492 K290 D295 K302 M308 M312 F314 D315 D375 E377 T402 L403 L408 K386 R463 K302 R379 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.011uM remove_due_to_license_issue Q8IL11 23713488 1004 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4k3n F 2.0 BS04 1OT F 1 K374 D379 K386 M392 F398 D399 D459 E461 T486 L487 L492 K282 D287 K294 M300 F306 D307 D367 E369 T394 L395 L400 K386 R463 K294 R371 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.011uM remove_due_to_license_issue Q8IL11 23713488 1004 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4k42 A 2.9 BS02 NWM A 1 Y143 G168 Y169 I345 M355 Y129 G154 Y155 I331 M341 3.6.4.- 0000287,0001725,0003785,0005509,0005515,0005523,0005524,0005737,0005856,0005865,0005884,0010628,0016787,0019904,0030027,0030041,0030175,0030240,0031013,0031432,0031941,0032036,0032432,0042802,0044297,0048306,0048741,0051017,0090131,0098723,0140660 remove_due_to_license_issue P68135 25047814 403 TTALVCDNGSGLVKAGFAGDDAPRAVFPSIVGRPQKDSYVGDEAQSKRGILTLKYPIEHGIITNWDDMEKIWHHTFYNELRVAPEEHPTLLTEAPLNPKANREKMTQIMFETFNVPAMYVAIQAVLSLYASGRTTGIVLDSGDGVTHNVPIYEGYALPHAIMRLDLAGRDLTDYLMKILTERGYSFVTTAEREIVRDIKEKLCYVALDFENEMATAASSSSLEKSYELPDGQVITIGNERFRCPETLFQPSFIGMESAGIHETTYNSIMKCDIDIRKDLYANNVMSGGTTMYPGIADRMQKEITALAPSTMKIKIIAPPERKYSVWIGGSILASLSTFQQMWITKQEYDEAGPSIVHRKC 4k43 A 2.9 BS02 1PO A 1 Y143 A144 Y169 I345 L349 T351 Y129 A130 Y155 I331 L335 T337 3.6.4.- 0000287,0001725,0003785,0005509,0005515,0005523,0005524,0005737,0005856,0005865,0005884,0010628,0016787,0019904,0030027,0030041,0030175,0030240,0031013,0031432,0031941,0032036,0032432,0042802,0044297,0048306,0048741,0051017,0090131,0098723,0140660 remove_due_to_license_issue P68135 25047814 403 TTALVCDNGSGLVKAGFAGDDAPRAVFPSIVGRPQKDSYVGDEAQSKRGILTLKYPIEHGIITNWDDMEKIWHHTFYNELRVAPEEHPTLLTEAPLNPKANREKMTQIMFETFNVPAMYVAIQAVLSLYASGRTTGIVLDSGDGVTHNVPIYEGYALPHAIMRLDLAGRDLTDYLMKILTERGYSFVTTAEREIVRDIKEKLCYVALDFENEMATAASSSSLEKSYELPDGQVITIGNERFRCPETLFQPSFIGMESAGIHETTYNSIMKCDIDIRKDLYANNVMSGGTTMYPGIADRMQKEITALAPSTMKIKIIAPPERKYSVWIGGSILASLSTFQQMWITKQEYDEAGPSIVHRKC 4k4e A 2.3 BS02 K4E A 1 H1184 S1186 F1188 I1192 F1197 D1198 H1201 Y1203 I1212 Y1213 Y1224 G1227 H81 S83 F85 I89 F94 D95 H98 Y100 I109 Y110 Y121 G124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 23701517 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSAYAEYVIYRGEQAYPEYLITYQIMKPEH 4k4f A 2.9 BS02 K4F A 1 H1184 F1188 A1191 I1192 G1196 D1198 H1201 F1208 G1211 I1212 Y1213 H81 F85 A88 I89 G93 D95 H98 F105 G108 I109 Y110 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 23701517 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVLAYAEYVIYRGEQAYPEYLITYQIMKPEH 4k4j A 2.0 BS02 1O8 A 1 I268 A271 A272 Q275 F313 R316 L326 A327 I345 C432 L436 I24 A27 A28 Q31 F69 R72 L82 A83 I101 C188 L192 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue EC50=820nM, Kd=33nM P19793 24187139 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4k55 A 1.91 BS01 H6P A 1 K39 Y100 Q102 Y107 K37 Y98 Q100 Y105 ? Kd=3.06uM remove_due_to_license_issue EC50=0.510000nM, IC50=16100nM, Kd=1540nM O00481 23872678 201 QFSVLGPSGPILAMVGEDADLPCHLFPTMSAETMELKWVSSSLRQVVNVYADGKEVEDRQSAPYRGRTSILRDGITAGKAALRIHNVTASDSGKYLCYFQDGDFYEKALVELKVLEHH 4k5l A 1.91 BS02 19N A 1 E319 A461 M462 E463 H496 E497 H500 E519 E572 Y575 Y580 E124 A266 M267 E268 H301 E302 H305 E324 E377 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=11uM remove_due_to_license_issue O96935 23713488 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4k5m A 1.75 BS02 1OV A 1 E319 A461 M462 E463 H496 E497 H500 E519 Y575 Y580 E124 A266 M267 E268 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=193uM remove_due_to_license_issue O96935 23713488 1106 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4k5n A 1.91 BS02 1OU A 1 E319 V459 A461 M462 E463 H496 E497 E519 Y575 Y580 E124 V264 A266 M267 E268 H301 E302 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=127uM remove_due_to_license_issue O96935 23713488 1106 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4k5o A 1.9 BS02 1OT A 1 E319 V459 A461 M462 E463 H496 E497 H500 E519 Y575 Y580 M1034 E124 V264 A266 M267 E268 H301 E302 H305 E324 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=104uM remove_due_to_license_issue O96935 23713488 1106 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4k5p A 1.85 BS02 1OS A 1 E319 V459 A461 M462 E463 H496 E497 H500 E519 Y575 Y580 E124 V264 A266 M267 E268 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=345uM remove_due_to_license_issue O96935 23713488 1106 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4k5y A 2.977 BS01 1Q5 A 1 F203 M206 L280 N283 T316 L323 Y327 F89 M92 L323 N326 T359 L366 Y370 E1011 D1020 E116 D125 ?,3.2.1.17 0003796,0004888,0004930,0007166,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P34998 23863939 401 HYHVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLSVAKSELDKAIGRNSNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRSALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVIATFRTGTWDAYDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRPGVYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAFVNEVSRVVFIYFNAFLESFQGFFVSVFACFLNS 4k5z A 1.8 BS02 1P7 A 1 A190 F191 S195 G216 A226 A171 F172 S176 G193 A201 H57 D102 K192 G193 D194 S195 G196 H45 D89 K173 G174 D175 S176 G177 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 remove_due_to_license_issue IC50=>1000000nM P23946 23659209 703 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 4k60 A 1.5 BS02 1P8 A 1 A190 F191 K192 G216 A226 A170 F171 K172 G192 A200 H57 D102 K192 G193 D194 S195 G196 H44 D88 K172 G173 D174 S175 G176 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 ic50=570uM remove_due_to_license_issue IC50=570000nM P23946 23659209 703 IIGGTECKPHSRPYMAYLEIVTNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 4k63 A 3.1 BS01 SIA I 1 Y95 S136 S137 E190 Q226 Y92 S133 S134 E187 Q223 ? 0019031,0019064,0046789 remove_due_to_license_issue A8HWY8 23641058 3 QDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKTHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPTNDLCYPGSFNDYEELKHLLSRINHFEKIQIIPKSSWSDHEASSGVSSACPYLGSPSFFRNVVWLIKKNSTYPTIKKSYNNTNQEDLLVLWGIHHPNDAAEQTRLYQNPTTYISIGTSTLNQRLVPKIATRSKVNGQSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSAIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNS 4k64 A 2.604 BS01 SIA I 1 Y95 V135 S136 S137 W153 H183 E190 Q226 Y92 V132 S133 S134 W150 H180 E187 Q223 ? 0019031,0019064,0046789 remove_due_to_license_issue A8HWY8 23641058 2 QDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKTHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPTNDLCYPGSFNDYEELKHLLSRINHFEKIQIIPKSSWSDHEASSGVSSACPYLGSPSFFRNVVWLIKKNSTYPTIKKSYNNTNQEDLLVLWGIHHPNDAAEQTRLYQNPTTYISIGTSTLNQRLVPKIATRSKVNGQSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSAIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNS 4k66 A 3.005 BS01 SIA I 1 Y95 V135 S136 S137 W153 H183 E190 R193 Y92 V132 S133 S134 W150 H180 E187 R190 ? 0019031,0019064,0046789 remove_due_to_license_issue A8HWY8 23641058 2 QDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKTHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPTNDLCYPGSFNDYEELKYLLSRINHFEKIQIIPKSSWSDHEASSGVSSACPYLGSPSFFRNVVWLIKKNSAYPTIKKSYNNTNQEDLLVLWGIHHPNDAAEQTRLYQNPTTYISIGTSTLNQRLVPKIATRSKVNGLSSRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSAIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNS 4k67 A 2.7 BS01 SIA I 1 Y95 V135 S136 S137 W153 H183 E190 L226 S228 Y92 V132 S133 S134 W150 H180 E187 L223 S225 ? 0019031,0019064,0046789 remove_due_to_license_issue A8HWY8 23641058 2 QDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKTHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPTNDLCYPGSFNDYEELKYLLSRINHFEKIQIIPKSSWSDHEASSGVSSACPYLGSPSFFRNVVWLIKKNSAYPTIKKSYNNTNQEDLLVLWGIHHPNDAAEQTRLYQNPTTYISIGTSTLNQRLVPKIATRSKVNGLSSRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSAIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNS 4k69 A 1.5 BS03 1P9 A 1 C42 H57 A190 F191 K192 S195 S214 Y215 G216 C30 H45 A166 F167 K168 S171 S186 Y187 G188 H57 D102 K192 G193 D194 S195 G196 H45 D89 K168 G169 D170 S171 G172 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 ic50=0.04uM remove_due_to_license_issue IC50=40nM P23946 23659209 304 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGAAQGIVSYGRSDAKPPAVFTRISHYQPWINQILQAN 4k6i A 2.1 BS02 9RA A 1 I268 A272 L309 F313 R316 L326 C432 I24 A28 L65 F69 R72 L82 C188 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue EC50=33nM, Kd=36nM, Ki=379nM P19793 24187139 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4k6t A 2.0 BS01 SIA A 1 Y312 P317 D318 K345 Y133 P138 D139 K166 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 KYDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6t A 2.0 BS02 SIA C 1 Y308 V322 Y129 V143 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 KYDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6t B 2.0 BS01 SIA B 1 Y312 P317 D318 K345 Y133 P138 D139 K166 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 KYDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6t C 2.0 BS01 SIA C 1 Y312 P317 D318 K345 Y129 P134 D135 K162 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 RTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6u A 1.9 BS02 SIA A 1 Y312 P317 D318 K345 Y131 P136 D137 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6u B 1.9 BS01 SIA A 1 Y308 V322 Y130 V144 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 PKYDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6u B 1.9 BS03 SIA B 1 Y312 P317 D318 K345 Y134 P139 D140 K167 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 PKYDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6u C 1.9 BS01 SIA C 1 Y312 P317 D318 K345 Y130 P135 D136 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6v A 1.5 BS02 18D A 1 Y312 P317 D318 K345 Y131 P136 D137 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6v B 1.5 BS02 18D B 1 Y312 P317 D318 P320 K345 Y132 P137 D138 P140 K165 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 YDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6v C 1.5 BS01 18D C 1 Y312 P317 D318 K345 Y130 P135 D136 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 402 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6w A 1.5 BS01 18D A 1 Y312 P317 D318 K345 Y130 P135 D136 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6w B 1.5 BS01 18D B 1 Y312 P317 D318 P320 K345 Y132 P137 D138 P140 K165 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 YDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6w C 1.5 BS01 18D C 1 Y312 P317 D318 K345 Y131 P136 D137 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4k6z A 2.73 BS01 1Q3 A 1 L881 E883 V889 A906 M956 G962 E966 R1007 N1008 L1010 G1020 D1021 L17 E19 V25 A42 M83 G89 E93 R134 N135 L137 G147 D148 D1003 A1005 R1007 N1008 D1021 D1040 D130 A132 R134 N135 D148 D167 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P23458 24042009 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4k77 B 2.4 BS01 1Q4 B 1 L881 A906 F958 L959 R1007 N1008 L1010 L17 A42 F86 L87 R135 N136 L138 D1003 A1005 R1007 N1008 D1021 D1040 D131 A133 R135 N136 D149 D168 2.7.10.2 0004672,0004713,0005524,0006468 Ki=235nM remove_due_to_license_issue Ki=235nM P23458 24042009 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 4k7i A 2.25 BS01 CAQ A 1 P40 G46 C47 R127 P41 G47 C48 R128 1.11.1.24 0008379,0016491,0034599 Kd=1500uM remove_due_to_license_issue P30044 25025339 201 SAPIKVGDAIPAVEVFEGEPGNKVNLAELFKGKKGVLFGVPGAFTPGCSKTHLPGFVEQAEALKAKGVQVVACLSVNDAFVTGEWGRAHKAEGKVRLLADPTGAFGKETDLLLDDSLVSIFGNRRLKRFSMVVQDGIVKALNVEPDGTGLTCSLAPNIISQL 4k7n A 2.3 BS01 MCT A 1 P40 T44 P45 G46 C47 R127 P40 T44 P45 G46 C47 R127 1.11.1.24 0008379,0016491,0034599 Kd=330uM remove_due_to_license_issue P30044 25025339 201 APIKVGDAIPAVEVFEGEPGNKVNLAELFKGKKGVLFGVPGAFTPGCSKTHLPGFVEQAEALKAKGVQVVACLSVNDAFVTGEWGRAHKAEGKVRLLADPTGAFGKETDLLLDDSLVSIFGNRRLKRFSMVVQDGIVKALNVEPDGTGLTCSLAPNIISQL 4k7n B 2.3 BS01 MCT B 1 T44 P45 G46 C47 R127 T44 P45 G46 C47 R127 1.11.1.24 0008379,0016491,0034599 Kd=330uM remove_due_to_license_issue P30044 25025339 201 APIKVGDAIPAVEVFEGEPGNKVNLAELFKGKKGVLFGVPGAFTPGCSKTHLPGFVEQAEALKAKGVQVVACLSVNDAFVTGEWGRAHKAEGKVRLLADPTGAFGKETDLLLDDSLVSIFGNRRLKRFSMVVQDGIVKALNVEPDGTGLTCSLAPNIISQL 4k7o A 1.98 BS01 EKZ A 1 P40 T44 P45 G46 C47 F120 R127 T147 P41 T45 P46 G47 C48 F121 R128 T148 1.11.1.24 0008379,0016491,0034599 Kd=50uM remove_due_to_license_issue P30044 25025339 201 SAPIKVGDAIPAVEVFEGEPGNKVNLAELFKGKKGVLFGVPGAFTPGCSKTHLPGFVEQAEALKAKGVQVVACLSVNDAFVTGEWGRAHKAEGKVRLLADPTGAFGKETDLLLDDSLVSIFGNRRLKRFSMVVQDGIVKALNVEPDGTGLTCSLAPNIISQL 4k8a A 2.91 BS01 K8A A 1 I428 A452 M499 C502 L553 I15 A37 M84 C87 L138 D546 A548 R550 N551 D564 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q05397 23973211 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEE 4k8o A 2.65 BS01 ATP A 1 Y489 V497 N517 G518 S519 G520 K521 S522 T523 Q678 Y21 V29 N49 G50 S51 G52 K53 S54 T55 Q210 7.4.2.14 0005524,0016887 remove_due_to_license_issue P36370 25377891 801 GSLAPLNMKGLVKFQDVSFAYPNHPNVQVLQGLTFTLYPGKVTALVGPNGSGKSTVAALLQNLYQPTGGKVLLDGEPLVQYDHHYLHTQVAAVGQEPLLFGRSFRENIAYGLTRTPTMEEITAVAMESGAHDFISGFPQGYDTEVGETGNQLSGGQRQAVALARALIRKPRLLILDNATSALAAGNQLRVQRLLYESPEWASRTVLLITQQLSLAERAHHILFLKEGSVCEQGTHLQLMERGGCYRSMVEALAA 4k8s A 2.39 BS01 1QT A 1 L30 D32 G34 P70 Y71 T72 F108 Y198 K224 D228 G230 T329 L33 D35 G37 P73 Y74 T75 F111 Y190 K216 D220 G222 T315 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.036uM remove_due_to_license_issue P56817 23769639 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4k9h A 2.29 BS01 1QU A 1 D32 G34 Y71 T72 Q73 F108 I118 D228 G230 T232 N233 D35 G37 Y74 T75 Q76 F111 I121 D220 G222 T224 N225 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.076uM remove_due_to_license_issue P56817 23769639 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4k9y A 2.0 BS01 K9Y A 1 I428 A452 E471 M475 V484 M499 C502 F542 L553 G563 D564 F565 R569 Y570 I14 A38 E57 M61 V70 M85 C88 F128 L139 G149 D150 F151 R155 Y156 D546 A548 R550 N551 D564 K583 D132 A134 R136 N137 D150 K169 2.7.10.2 0004672,0004713,0005524,0006468 Kd=0.111uM remove_due_to_license_issue Kd=111nM, IC50=750nM Q05397 23973211 701 YEIQRERIELGRCIGEGQFGDVHQGIYMSPENPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSRYMEDSTYYKASKGKLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKA 4kab A 2.71 BS01 4KA A 1 A452 M499 L501 C502 L553 A39 M86 L88 C89 L140 D546 A548 R550 N551 D564 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q05397 23973211 701 TRDYEIQRERIELGRCIGEGQFGDVHQGIYMSPPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4kai A 2.3 BS01 1PV A 1 R200 L204 L314 N316 I363 S365 C366 S368 L384 M414 Y415 Y448 R196 L200 L310 N312 I359 S361 C362 S364 L380 M410 Y411 Y444 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 23672667 601 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPGWFVAGYSGGDIYHSL 4kai A 2.3 BS02 1PV A 2 S476 Y477 L497 R501 S472 Y473 L493 R497 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 23672667 602 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQPRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPGWFVAGYSGGDIYHSL 4kao A 2.39 BS01 KAO A 1 E471 T474 M475 V484 M499 L553 G563 D564 F565 E54 T57 M58 V67 M82 L136 G146 D147 F148 D546 A548 R550 N551 D564 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Kd=0.77uM remove_due_to_license_issue IC50=>10000nM, Kd=770nM Q05397 23973211 701 YEIQRERIELGRCIGEGQFGDVHQGIYMSPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4kax A 1.85 BS01 GTP A 1 D22 A23 G25 K26 T27 T28 T41 T44 G65 G66 N122 K123 D125 L126 C155 A156 T157 D11 A12 G14 K15 T16 T17 T30 T33 G54 G55 N111 K112 D114 L115 C144 A145 T146 L67 L56 3.6.5.2 0001726,0001889,0003924,0003925,0005515,0005525,0005737,0005768,0005769,0005794,0005829,0005886,0005925,0005938,0006886,0007155,0007399,0010975,0010976,0015031,0016020,0016192,0016787,0019003,0030139,0030154,0030496,0030838,0030866,0031527,0031901,0031996,0032154,0032456,0034394,0035020,0035591,0036010,0042995,0048261,0048488,0050714,0051301,0051489,0051549,0055037,0055038,0060998,0070062,0072659,0090162,0090543,0097178,0097284,0098793,0098794,0098978,0099562,0120183,1902217,1903078,1903438,1905345,1905606,1990090,2000009,2000171 remove_due_to_license_issue P62330 23940353 201 GSMRILMLGLDAAGKTTILYKLKLGQSVTTIPTVGFNVETVTYKNVKFNVWDVGGLDKIRPLWRHYYTGTQGLIFVVDCADRDRIDEARQELHRIINDREMRDAIILIFANKQDLPDAMKPHEIQEKLGLTRIRDRNWYVQPSCATSGDGLYEGLTWLTSNYN 4kb7 A 1.85 BS01 690 A 1 F193 R200 L204 L314 Y316 I363 S365 C366 S368 N411 M414 Y415 Y448 F188 R195 L199 L309 Y311 I358 S360 C361 S363 N406 M409 Y410 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 23672667 601 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVYGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPVAGYSGGDIYHS 4kb8 A 1.95 BS01 1QN A 1 I23 A36 K38 M80 M82 L85 G86 L135 I148 I21 A34 K36 M78 M80 L83 G84 L133 I146 D128 K130 D126 K128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=12.9nM remove_due_to_license_issue IC50=64nM P48730 23919824 401 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kb9 A 1.29 BS01 G79 A 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 Ki=0.01nM remove_due_to_license_issue Q7SSI0 23947685 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4kb9 B 1.29 BS01 G79 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 remove_due_to_license_issue Q7SSI0 23947685 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4kba A 1.98 BS01 1QM A 1 I23 A36 K38 M80 M82 L85 G86 L135 I148 I21 A34 K36 M78 M80 L83 G84 L133 I146 D128 K130 D126 K128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=6nM remove_due_to_license_issue IC50=6.0nM P48730 23919824 401 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLRISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kbc A 1.98 BS01 1QJ A 1 I23 A36 K38 M80 M82 L85 I148 I18 A31 K33 M75 M77 L80 I143 D128 K130 D123 K125 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue P48730 23919824 401 ELRVGNRYRLGRKIGSDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kbi A 2.06 BS01 1C0 A 1 R200 L204 L314 Y316 V321 I363 S365 C366 S368 L384 M414 Y415 Y448 R195 L199 L309 Y311 V316 I358 S360 C361 S363 L379 M409 Y410 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 23672667 601 SMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGQRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKYGYGAKDVRNLSSRAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVYGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPYSGGDIYHS 4kbk A 2.1 BS01 1QG A 1 I15 I23 A36 K38 M80 M82 L85 G86 L135 I148 I13 I19 A32 K34 M70 M72 L75 G76 L125 I138 D128 K130 D118 K120 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=6.6nM P48730 23919824 401 LRVGNRYRLGRKIGSGGDIYLGTDIAAGEEVAIKLECQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 4kby A 2.36 BS01 C2E A 1 Y162 Y166 R237 V238 T262 P263 Y10 Y14 R76 V77 T101 P102 ? 0002218,0032481 Ka=5390000M^-1 remove_due_to_license_issue Q3TBT3 23519410 401 NVAHGLAWSYYIGYLRLILPGLQARIRMFNQLHNNMLSGAGSRRLYILFPLDCGVPDNLSVVDPNIRFRDMLPQNRVYSNSVYEILENGQPAGVCILEYATPLQTLFAMSQDAKAGFSREDRLEQAKLFCRTLEEILEDVPESRNNCRLIVYQEPTDGNSFSLSQEVLRHIRQEE 4kby B 2.36 BS01 C2E A 1 Y162 Y166 V238 S240 T262 P263 Y10 Y14 V78 S80 T102 P103 ? 0002218,0032481 remove_due_to_license_issue Q3TBT3 23519410 401 NVAHGLAWSYYIGYLRLILPGLQARIRMFNQLHNNMLSGAGSRRLYILFPLDCGVPDNLSVVDPNIRFRDMLPQQNRVYSNSVYEILENGQPAGVCILEYATPLQTLFAMSQDAKAGFSREDRLEQAKLFCRTLEEILEDVPESRNNCRLIVYQEPTDGNSFSLSQEVLRHIRQEE 4kc1 A 1.5 BS02 WS1 A 1 F121 A122 I123 Y126 V184 R188 D211 V212 D213 F64 A65 I66 Y69 V127 R131 D154 V155 D156 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 remove_due_to_license_issue P16442 24108680 403 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPK 4kc2 A 1.7 BS02 WS2 A 1 F121 A122 I123 Y126 W181 V184 R188 D211 V212 D213 F64 A65 I66 Y69 W124 V127 R131 D154 V155 D156 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 remove_due_to_license_issue P16442 24108680 403 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPK 4kc4 A 1.6 BS02 WS3 A 1 F121 A122 I123 Y126 V184 R188 D211 V212 D213 K346 F64 A65 I66 Y69 V127 R131 D154 V155 D156 K289 H233 G266 W300 E303 A343 H176 G209 W243 E246 A286 2.4.1.37,2.4.1.40 0005975,0016020,0016758 remove_due_to_license_issue P16442 24108680 403 AIGEFMVSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVPK 4kcg A 2.09 BS01 1QC A 1 E53 V55 L82 M85 Y86 P89 Q97 D133 F137 S144 Y204 E34 V36 L52 M55 Y56 P59 Q67 D103 F107 S114 Y174 E53 R128 E34 R98 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 remove_due_to_license_issue IC50=4.9nM, Ki=0.500000nM P27707 24567448 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4kcx A 2.0 BS01 1QK A 1 W50 P51 F52 L61 D114 I115 M118 W22 P23 F24 L33 D86 I87 M90 ? Kd=37uM remove_due_to_license_issue Q58F21 24007471 201 TNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMP 4ke0 A 2.3 BS01 1R8 A 1 D32 G34 P70 Y71 T72 F108 I110 W115 Y198 K224 D228 G230 T329 D37 G39 P75 Y76 T77 F113 I115 W120 Y193 K219 D223 G225 T318 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=0.017uM remove_due_to_license_issue P56817 23769639 501 KGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4ke1 A 1.91 BS01 1R6 A 1 Q12 L30 D32 G34 S35 Y71 T72 F108 Y198 D228 G230 T329 Q14 L32 D34 G36 S37 Y73 T74 F110 Y190 D220 G222 T299 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.0025uM remove_due_to_license_issue P56817 23769639 404 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4keq A 2.279 BS03 5PN A 1 E65 H98 F99 L132 G133 F223 E63 H96 F97 L130 G131 F221 3.1.1.27 0016787,0042820,0046872,0047585 remove_due_to_license_issue Q988B9 24699732 303 DTKVYLLDGGSLVLDGYHVFWNRGPGGEVRFPVYSILIEHAEGRFLIDTGYDYDHVMKVLPFEKPIQEKHQTIPGALGLLGLEPRDIDVVVNSHFHFDHCGGNKYFPHAKKICHRSEVPQACNPQPFEHLGYSDLSFSAEAAEARGATAQLLEGTTRANSTFEGIDGDVDLARGVKLISTPGHSIGHYSLLVEFPRRKPILFTIDAAYTQKSLETLCQAAFHIDPVAGVNSMRKVKKLAEDHGAELMYSHDMDNFKTYRTGTQFYGHHHH 4keq A 2.279 BS04 5PN A 2 S13 I68 E70 Q73 K258 S11 I66 E68 Q71 K256 3.1.1.27 0016787,0042820,0046872,0047585 remove_due_to_license_issue Q988B9 24699732 304 DTKVYLLDGGSLVLDGYHVFWNRGPGGEVRFPVYSILIEHAEGRFLIDTGYDYDHVMKVLPFEKPIQEKHQTIPGALGLLGLEPRDIDVVVNSHFHFDHCGGNKYFPHAKKICHRSEVPQACNPQPFEHLGYSDLSFSAEAAEARGATAQLLEGTTRANSTFEGIDGDVDLARGVKLISTPGHSIGHYSLLVEFPRRKPILFTIDAAYTQKSLETLCQAAFHIDPVAGVNSMRKVKKLAEDHGAELMYSHDMDNFKTYRTGTQFYGHHHH 4kfp A 1.84 BS01 1R7 A 1 H191 F193 R196 D219 S241 V242 A244 P273 S275 R311 I351 H174 F176 R179 D202 S224 V225 A227 P256 S258 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.01uM remove_due_to_license_issue P43490 23899614 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4kfp B 1.84 BS01 1R7 B 1 H191 F193 R196 D219 S241 V242 A244 R311 I351 A379 H174 F176 R179 D202 S224 V225 A227 R294 I334 A362 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.01uM remove_due_to_license_issue P43490 23899614 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4kfq A 2.2 BS01 KFQ A 1 F92 P124 L125 T126 R131 S180 D224 F89 P121 L122 T123 R128 S177 D221 ? 0015276,0016020 remove_due_to_license_issue P35439 24072709 301 TRLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPNDTSPGSPRHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNSNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQECDS 4kif A 2.5 BS01 PPY A 1 R127 M240 H243 F287 F291 H295 R125 M238 H241 F285 F289 H293 2.1.1.281 0008168,0009058,0017000,0032259 remove_due_to_license_issue Q643C8 24914966 501 TEVSEAQARRAVADIFNSTLASSAIGAAWELGALDELRENGKLDVSDFAVRHDLHEPAVVGMFTALASVGIVRREGATVVVGPYFDEANHHRSLFHWLNQGSGELFRRMPQVLPNENRTGKFYQRDAGAISYACREISERYFDPAFWAAVDGLGYTPTTVADLGSGSGERLIQIARRFPGVRGLGVDIADGAIAMAEKEVAAKGFGDQISFVRGDARTIDQVSARGEFAEVDLLTCFMMGHDFWPRENCVQTLRKLRAAFPNVRRFLLGDATRTVGIPDRELPVFTLGFEFGHDMMGVYLPTLDEWDGVFEEGGWRCVKKHAIDSLSVSVVFELE 4kif A 2.5 BS04 PPY A 2 G206 F207 D209 G204 F205 D207 2.1.1.281 0008168,0009058,0017000,0032259 remove_due_to_license_issue Q643C8 24914966 504 TEVSEAQARRAVADIFNSTLASSAIGAAWELGALDELRENGKLDVSDFAVRHDLHEPAVVGMFTALASVGIVRREGATVVVGPYFDEANHHRSLFHWLNQGSGELFRRMPQVLPNENRTGKFYQRDAGAISYACREISERYFDPAFWAAVDGLGYTPTTVADLGSGSGERLIQIARRFPGVRGLGVDIADGAIAMAEKEVAAKGFGDQISFVRGDARTIDQVSARGEFAEVDLLTCFMMGHDFWPRENCVQTLRKLRAAFPNVRRFLLGDATRTVGIPDRELPVFTLGFEFGHDMMGVYLPTLDEWDGVFEEGGWRCVKKHAIDSLSVSVVFELE 4kii A 1.85 BS01 RHL A 1 K60 I71 I84 L103 F105 K59 I70 I83 L102 F104 ? 0005515,0005576,0019841,0036041,0036094,0042802 remove_due_to_license_issue P02754 201 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENDECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENQSLVCQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 4kij A 2.8 BS01 KIJ A 1 E20 Y24 N75 G77 H101 I102 S103 R112 E19 Y23 N74 G76 H100 I101 S102 R111 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P10 N11 R18 Y23 N74 G77 E98 H100 R107 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 25234229 202 ELIVNVINGPNLGRLARREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4kil A 1.75 BS03 1R5 A 1 I38 H41 E80 D108 E119 K134 I43 H46 E85 D113 E124 K139 0003723,0039694 ic50=0.5uM remove_due_to_license_issue 24936242 305 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4kin A 1.97 BS01 1M8 A 1 V30 A51 K53 E71 L75 L104 T106 A111 A157 D168 F169 V26 A47 K49 E67 L71 L100 T102 A107 A151 D162 F163 D150 K152 N155 D168 T185 D144 K146 N149 D162 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=4.8nM remove_due_to_license_issue IC50=4.8nM Q16539 23746475 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4kio A 2.18 BS01 G5K A 1 I369 A389 F435 F437 M438 G441 C442 L489 I15 A32 F72 F74 M75 G78 C79 L126 D482 A484 R486 N487 D500 P521 D119 A121 R123 N124 D137 P142 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=0.5uM remove_due_to_license_issue Q08881 23935099 701 GSVIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4kip A 2.27 BS01 1R9 A 1 A51 K53 E71 T106 M109 L167 D168 F169 A47 K49 E67 T102 M105 L163 D164 F165 D150 K152 N155 D168 T185 D146 K148 N151 D164 T170 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=7nM remove_due_to_license_issue IC50=7.0nM Q16539 23746475 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4kiq A 2.5 BS01 1RA A 1 S32 G33 A51 K53 E71 L104 T106 L108 L167 D168 F169 S29 G30 A48 K50 E68 L101 T103 L105 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=23nM remove_due_to_license_issue IC50=23nM Q16539 23746475 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLAATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4kis A 3.2 BS01 dna E 0 R135 M136 G139 K140 R143 A153 K154 R156 S189 T191 Y207 M254 N261 K262 K286 S290 R291 Y295 Y297 Y299 H309 R2 M3 G6 K7 R10 A20 K21 R23 S56 T58 Y74 M121 N128 K129 K153 S157 R158 Y162 Y164 Y166 H176 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 25 ~ 50 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFASRNIDKEDESLNEKLKIEHAKKKRLFDLYINGSYEVSELDSMMNDIDAQINYYEAQIEANEELKKNKTVDFNSLEFREKQLYLKSLINKIYIDGEQVTIEWLLEHHHHHH 4kis A 3.2 BS02 dna F 0 M136 R209 N212 Y225 K226 N259 S264 S266 N269 H283 R285 T288 K303 K306 M3 R76 N79 Y92 K93 N126 S131 S133 N136 H150 R152 T155 K170 K173 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 -1 ~ 24 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFASRNIDKEDESLNEKLKIEHAKKKRLFDLYINGSYEVSELDSMMNDIDAQINYYEAQIEANEELKKNKTVDFNSLEFREKQLYLKSLINKIYIDGEQVTIEWLLEHHHHHH 4kis B 3.2 BS01 dna G 0 R135 M136 G139 K140 R143 A153 K154 R156 S189 T191 Y207 N261 K262 K286 T288 S290 K293 Y295 Y297 Y299 R2 M3 G6 K7 R10 A20 K21 R23 S56 T58 Y74 N128 K129 K153 T155 S157 K160 Y162 Y164 Y166 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 25 ~ 50 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFELDSLNEKLKIEHAKKKRLFDLYSELDSMMNDIDAQINYYEAQIEANEELKKNKKIQENLADLATVDFNSLEFREKQLYLKSLINKIYIDGEQVTIEWLLE 4kis B 3.2 BS02 dna H 0 M136 L150 R209 Y225 K226 N259 S264 S266 N269 V282 H283 R285 T288 K303 K306 M3 L17 R76 Y92 K93 N126 S131 S133 N136 V149 H150 R152 T155 K170 K173 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 -1 ~ 24 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFELDSLNEKLKIEHAKKKRLFDLYSELDSMMNDIDAQINYYEAQIEANEELKKNKKIQENLADLATVDFNSLEFREKQLYLKSLINKIYIDGEQVTIEWLLE 4kis C 3.2 BS01 dna I 0 R135 M136 G139 K140 R143 A153 K154 S189 T191 Y207 M254 K262 K286 T288 K293 Y295 Y297 Y299 K313 R2 M3 G6 K7 R10 A20 K21 S56 T58 Y74 M121 K129 K153 T155 K160 Y162 Y164 Y166 K180 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 25 ~ 50 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFASRNIDKEDELDSLNEKLKIEHAKKKRLFDLYDSMMNDIDAQINYYEAQIEANEELKKNKKIQENLADLATVDFNSLEFREKQLYLKSLINKIYIDGEQVTIEWL 4kis C 3.2 BS02 dna J 0 M136 R156 R209 Y225 K226 N259 S264 S266 V282 H283 R285 T288 K306 M3 R23 R76 Y92 K93 N126 S131 S133 V149 H150 R152 T155 K173 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 -1 ~ 24 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFASRNIDKEDELDSLNEKLKIEHAKKKRLFDLYDSMMNDIDAQINYYEAQIEANEELKKNKKIQENLADLATVDFNSLEFREKQLYLKSLINKIYIDGEQVTIEWL 4kis D 3.2 BS01 dna K 0 R135 M136 K140 R143 T152 A153 K154 T165 S189 T191 Y207 M254 K262 K286 T288 S290 R291 K293 Y295 Y297 Y299 K313 R320 R3 M4 K8 R11 T20 A21 K22 T33 S57 T59 Y75 M122 K130 K154 T156 S158 R159 K161 Y163 Y165 Y167 K181 R188 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 25 ~ 50 RDRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFASRNIDKELNEKLKIEIDAQINYYEAQIEANEELKKNKKIQEFNSLEFREKQLYLKSLINKIYIDGEQVTIEWLLEHHHHHH 4kis D 3.2 BS02 dna L 0 R133 M136 L150 R156 R209 N212 Y225 K226 N259 S264 S266 N269 V282 H283 R285 T288 K303 K306 R1 M4 L18 R24 R77 N80 Y93 K94 N127 S132 S134 N137 V150 H151 R153 T156 K171 K174 ? 0000150,0003677 remove_due_to_license_issue Q928V6 23821671 -1 ~ 24 RDRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYSFASRNIDKELNEKLKIEIDAQINYYEAQIEANEELKKNKKIQEFNSLEFREKQLYLKSLINKIYIDGEQVTIEWLLEHHHHHH 4kiu A 2.4 BS01 KIU A 1 N12 R15 L16 E20 Y24 G77 H81 H101 I102 S103 R112 N10 R13 L14 E18 Y22 G75 H79 H99 I100 S101 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 25234229 201 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4kiu L 2.4 BS01 KIU L 1 N12 L16 R19 Y24 N75 G77 H81 H101 I102 S103 V105 R112 N10 L14 R17 Y22 N73 G75 H79 H99 I100 S101 V103 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 25234229 201 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4kiw A 2.57 BS01 KIW A 1 N12 L13 R15 L16 Y24 N75 G77 G78 H81 H101 I102 S103 V105 R112 N10 L11 R13 L14 Y22 N73 G75 G76 H79 H99 I100 S101 V103 R110 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y22 N73 G76 E97 H99 R106 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 25234229 500 LIVNVINGPNLGRLGRREPAVYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4kiw L 2.57 BS01 KIW L 1 N12 R15 L16 R19 Y24 N75 G77 H81 H101 I102 S103 R112 N10 R13 L14 R17 Y19 N70 G72 H76 H96 I97 S98 R107 P11 N12 R19 Y24 N75 G78 E99 H101 R108 P9 N10 R17 Y19 N70 G73 E94 H96 R103 4.2.1.10 0003855,0005829,0008652,0009073,0009423,0016829,0019631 remove_due_to_license_issue P9WPX7 25234229 201 LIVNVINGPNLGRLGRREYGGTTHDELVALIEREAAELGLKAVVRQSDSEAQLLDWIHQAADAAEPVILNAGGLTHTSVALRDACAELSAPLIEVHISNVHAREEFRRHSYLSPIATGVIVGLGIQGYLLALRYLAEH 4kji A 3.2 BS01 rna C 0 F3 L4 I5 L6 S7 R9 T41 G45 R49 A54 R56 V58 L59 I60 V61 R62 L65 F1 L2 I3 L4 S5 R7 T39 G43 R47 A52 R54 V56 L57 I58 V59 R60 L63 ? 0003723,0006109,0006402,0042802 remove_due_to_license_issue A0A0H2ZIZ8 23954502 1 ~ 16 FLILSRREGEGITLSLKADYPAEELIRQLREGGIRILVTDIIGNQARVGIEAPRGVLIVRDELK 4kji B 3.2 BS01 rna D 0 G2 F3 L4 I5 L6 S7 L39 T41 G45 N46 R49 A54 V58 L59 I60 V61 R62 L65 G1 F2 L3 I4 L5 S6 L38 T40 G44 N45 R48 A53 V57 L58 I59 V60 R61 L64 ? 0003723,0006109,0006402,0042802 remove_due_to_license_issue A0A0H2ZIZ8 23954502 1 ~ 16 GFLILSRREGEGITLSLKADYPAEELIRQLREGGIRILVTDIIGNQARVGIEAPRGVLIVRDELK 4kju A 1.6 BS02 1RH A 1 K206 L207 K208 N209 W210 E211 D214 E219 H223 K56 L57 K58 N59 W60 E61 D64 E69 H73 2.3.2.27 ic50=0.006uM remove_due_to_license_issue IC50=6.0nM P98170 24093940 502 GTIYPRNPAMYSEEARLKSFQNWPDYAHLTPRELASAGLYYTGIGDQVQCFACGGKLKNWEPGDRAWSEHRRHFPNCFFVLG 4kjv A 1.7 BS02 1RK A 1 K206 L207 K208 E211 D214 E219 H223 F224 K56 L57 K58 E61 D64 E69 H73 F74 2.3.2.27 ic50=0.018uM remove_due_to_license_issue IC50=18nM P98170 24093940 502 GTIYPRNPAMYSEEARLKSFQNWPDYAHLTPRELASAGLYYTGIGDQVQCFACGGKLKNWEPGDRAWSEHRRHFPNCFFVLGR 4klb A 2.62 BS01 1RV A 1 C25 G65 G66 C25 G65 G66 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.51 0006508,0008234 remove_due_to_license_issue P25779 23991231 301 APAAVDWRARGAVTAVKDQGQCGSCWAFSAIGNVECQWFLAGHPLTNLSEQMLVSCDKTDSGCSGGLMNNAFEWIVQENNGAVYTEDSYPYASGEGISPPCTTSGHTVGATITGHVELPQDEAQIAAWLAVNGPVAVAVDASSWMTYTGGVMTSCVSEQLDHGVLLVGYNDSAAVPYWIIKNSWTTQWGEEGYIRIAKGSNQCLVKEEASSAVVG 4kln A 2.62 BS01 AGS A 1 G207 G248 T249 G250 K251 T252 L253 N348 I380 G408 A409 G196 G237 T238 G239 K240 T241 L242 N337 I369 G397 A398 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKEIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 4kln A 2.62 BS02 AGS F 1 R359 F360 R348 F349 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKEIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 4kln B 2.62 BS01 AGS A 1 R359 F360 R348 F349 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKEIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 4kln B 2.62 BS02 AGS B 1 G207 G248 T249 G250 K251 T252 L253 N348 G408 A409 G196 G237 T238 G239 K240 T241 L242 N337 G397 A398 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 LSTAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVRGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKEIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPS 4klv A 1.3 BS01 KLV A 1 C29 P31 R49 Y68 G79 N80 R141 C29 P31 R49 Y68 G79 N80 R141 ? 0016747,0046872 Kd=165.3uM remove_due_to_license_issue Q9HV14 24003232 216 MQLSHRPAETGDLETVAGFPQDRDELFYCYPKAIWPFSVAQLAAAIAERRGSTVAVHDGQVLGFANFYQWQHGDFCALGNMMVAPAARGLGVARYLIGVMENLAREQYKARLMKISCFNANAAGLLLYTQLGYQPRAIAERHDPDGRRVALIQMDKPLE 4km0 A 1.3 BS01 CP6 A 1 I5 W6 D27 F31 L50 I94 I7 W8 D29 F33 L52 I96 I5 I20 W22 D27 Q28 F31 L57 T91 T113 I7 I22 W24 D29 Q30 F33 L59 T93 T115 1.5.1.3 0004146,0005829,0006730,0016491,0046452,0046654,0046655,0050661,0070401 Kd=0.91uM remove_due_to_license_issue P9WNX1 24210757 201 SHMVGLIWAQATSGVIGRGGDIPWRLPEDQAHFREITMGHTIVMGRRTWDSLPAKVRPLPGRRNVVLSRQADFMASGAEVVGSLEEALTSPETWVIGGGQVYALALPYATRCEVTEVDIGLPREAGDALAPVLDETWRGETGEWRFSRSGLRYRLYSYHRS 4km2 A 1.4 BS02 TOP A 1 I5 W6 D27 F31 I94 I5 W6 D27 F31 I94 I5 I20 W22 D27 Q28 F31 L57 T91 T113 I5 I20 W22 D27 Q28 F31 L57 T91 T113 1.5.1.3 0004146,0005829,0006730,0016491,0046452,0046654,0046655,0050661,0070401 Kd=1.43uM remove_due_to_license_issue IC50=88000nM P9WNX1 24210757 202 MVGLIWAQATSGVIGRGGDIPWRLPEDQAHFREITMGHTIVMGRRTWDSLPAKVRPLPGRRNVVLSRQADFMASGAEVVGSLEEALTSPETWVIGGGQVYALALPYATRCEVTEVDIGLPREAGDALAPVLDETWRGETGEWRFSRSGLRYRLYSYHRS 4kmu C 3.85 BS01 RFP C 1 Q513 F514 D516 R529 S531 L533 R540 N568 I572 Q506 F507 D509 R522 S524 L526 R533 N561 I565 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 23679862 1401 KKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4kmz A 2.3 BS01 FOL A 1 D97 Y101 W118 R119 W150 H151 R152 G153 W154 W156 W187 S190 Y191 D73 Y77 W94 R95 W126 H127 R128 G129 W130 W132 W163 S166 Y167 ? Kd=2.7nM remove_due_to_license_issue P14207 23934049 301 TDLLNVCMDAKHHKTKPGPEDKLHDQCSPWKKNACCTASTSQELHKDTSRLYNFNWDHCGKMEPACKRHFIQDTCLYECSPNLGPWIQQVNQSWRKERFLDVPLCKEDCQRWWEDCHTSHTCKSNWHRGWDWTSGVNKCPAGALCRTFESYFPTPAALCEGLWSHSYKVSNYSRGSGRCIQMWFDSAQGNPNEEVARFYAAAM 4kn0 A 2.1 BS01 MTX A 1 Y76 F78 Y101 Q116 W118 H151 R152 G153 W154 W156 W187 S190 Y53 F55 Y78 Q93 W95 H128 R129 G130 W131 W133 W164 S167 ? Kd=40nM remove_due_to_license_issue IC50=106nM P14207 23934049 301 RTDLLNVCMDAKHHKTKPGPEDKLHDQCSPWKKNACCTASTSQELHKDTSRLYNFNWDHCGKMEPACKRHFIQDTCLYECSPNLGPWIQQVNQSWRKERFLDVPLCKEDCQRWWEDCHTSHTCKSNWHRGWDWTSGVNKCPAGALCRTFESYFPTPAALCEGLWSHSYKVSNYSRGSGRCIQMWFDSAQGNPNEEVARFYAAAMH 4kn1 A 2.301 BS01 04J A 1 Y76 Y101 W118 H151 R152 G153 W154 W156 W187 S190 Y53 Y78 W95 H128 R129 G130 W131 W133 W164 S167 ? Kd=144nM remove_due_to_license_issue P14207 23934049 301 RTDLLNVCMDAKHHKTKPGPEDKLHDQCSPWKKNACCTASTSQELHKDTSRLYNFNWDHCGKMEPACKRHFIQDTCLYECSPNLGPWIQQVNQSWRKERFLDVPLCKEDCQRWWEDCHTSHTCKSNWHRGWDWTSGVNKCPAGALCRTFESYFPTPAALCEGLWSHSYKVSNYSRGSGRCIQMWFDSAQGNPNEEVARFYAAAMH 4kn2 A 2.6 BS01 LYA A 1 Y76 F78 D97 T98 Y101 W118 W150 H151 R152 G153 W154 W156 W187 Y52 F54 D73 T74 Y77 W94 W126 H127 R128 G129 W130 W132 W163 ? remove_due_to_license_issue IC50=60nM P14207 23934049 304 TDLLNVCMDAKHHKTKPGPEDKLHDQCSPWKKNACCTASTSQELHKDTSRLYNFNWDHCGKMEPACKRHFIQDTCLYECSPNLGPWIQQVNQSWRKERFLDVPLCKEDCQRWWEDCHTSHTCKSNWHRGWDWTSGVNKCPAGALCRTFESYFPTPAALCEGLWSHSYKVSNYSRGSGRCIQMWFDSAQGNPNEEVARFYAAA 4kn4 C 3.965 BS01 1RL C 1 Q513 F514 R529 S531 L533 R540 I572 Q506 F507 R522 S524 L526 R533 I565 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 23679862 1401 KKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4kn7 C 3.686 BS01 1RM C 1 Q513 F514 R529 S531 L533 R540 I572 Q506 F507 R522 S524 L526 R533 I565 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 23679862 1401 KKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4kn7 X 3.686 BS01 1RM C 1 D513 D514 E515 D421 D422 E423 ? 0000345,0003677,0003700,0005515,0005737,0005829,0006351,0006352,0006355,0009408,0010468,0016987,0045892,1903865,2000142 remove_due_to_license_issue P00579 23679862 1401 QSQLKLLVTRGKEQGYLTYAEVNDHLPEDIVDSDQIEDIIQMINDMGIQVMEEAPDADDTDPVRMYMREMGTVELLTREGEIDIAKRIEDGINQVQCSVAEYPEAITYLLEQYDRVEAEIDPELAREKFAELRAQYVVTRDTIKAKGRSHATAQEEILKLSEVFKQFRLVPKQFDYLVNSMRVMMDRVRTQERLIMKLCVEQCKMPKKNFITLFTGNETSDTWFNAAIAMNKPWSEKLHDVSEEVHRALQKLQQIEEETGLTIEQVKDINRRMSIGEAKARRAKKEMVEANLRLVISIAKKYTNRGLQFLDLIQEGNIGLMKAVDKFEYRRGYKFSTYATWWIRQAITRSIADQARTIRIPVHMIETINKLNRISRQMLQEMGREPTPEELAERMLMPEDKIRKVLKIAKEPISMETPIGDDEDSHLGDFIEDTTLELPLDSATTESLRAATHDVLAGLTAREAKVLRMRFGIDMNTDYTLEEVGKQFDVTRERIRQIEAKALRKLRHPSRSEVLRS 4knb A 2.4 BS01 1RU A 1 A1108 L1140 Y1159 M1160 K1161 M1211 Y1230 A40 L69 Y88 M89 K90 M140 Y159 D1204 A1206 R1208 N1209 D1222 A1243 D133 A135 R137 N138 D151 A172 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.047uM remove_due_to_license_issue IC50=47nM P08581 23773865 1401 QAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLTDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF 4kne A 2.0 BS01 1CY A 1 I5 W6 D27 Q28 F31 L50 I94 I5 W6 D27 Q28 F31 L50 I94 I5 I20 W22 D27 Q28 F31 L57 T91 T113 I5 I20 W22 D27 Q28 F31 L57 T91 T113 1.5.1.3 0004146,0005829,0006730,0016491,0046452,0046654,0046655,0050661,0070401 Kd=1.26uM remove_due_to_license_issue P9WNX1 24210757 201 MVGLIWAQATSGVIGRGGDIPWRLPEDQAHFREITMGHTIVMGRRTWDSLPAKVRPLPGRRNVVLSRQADFMASGAEVVGSLEEALTSPETWVIGGGQVYALALPYATRCEVTEVDIGLPREAGDALAPVLDETWRGETGEWRFSRSGLRYRLYSYHRS 4kni A 1.8 BS02 E1E A 1 Q92 H94 H96 H119 V121 F131 L198 T199 T200 Q89 H91 H93 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=16.7nM remove_due_to_license_issue Kd=17nM, Ki=11nM P00918 24103428 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4knj A 2.0 BS02 E1F A 1 H94 H119 V121 V143 L198 T199 T200 P202 H91 H116 V118 V139 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=11.1nM remove_due_to_license_issue Kd=11nM, kon=390000M-1-s-1, koff=0.0042s-1 P00918 24103428 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4knm A 1.9 BS02 E1E A 1 H96 H98 H121 V123 F133 V145 L200 T201 V202 W211 H92 H94 H117 V119 F129 V141 L196 T197 V198 W207 H66 H96 H98 E108 H121 T201 H62 H92 H94 E104 H117 T197 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=10nM remove_due_to_license_issue Kd=8.1nM Q8N1Q1 24103428 302 LSWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 4knn B 1.404 BS02 E1F B 1 R93 Q94 H96 H121 F133 L200 T201 V202 R88 Q89 H91 H116 F128 L195 T196 V197 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=16.7nM remove_due_to_license_issue Kd=5.6nM, koff=0.0046s-1, kon=720000M-1-s-1 Q8N1Q1 24103428 302 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 4knr A 2.1 BS01 1S8 A 1 L11 A12 A13 G14 T82 Y103 D105 Y139 V223 L8 A9 A10 G11 T79 Y100 D102 Y136 V220 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=1.8uM remove_due_to_license_issue P43889 25262942 501 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 4knx A 1.9 BS01 1S9 A 1 L11 A13 G14 Q76 Q79 T82 Y103 D105 Y139 T170 V223 G225 L8 A10 G11 Q73 Q76 T79 Y100 D102 Y136 T167 V220 G222 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=3.2uM remove_due_to_license_issue P43889 25262942 501 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 4ko8 A 1.98 BS01 AGS A 1 G207 P247 G248 T249 G250 K251 T252 L253 N348 I380 H384 G408 A409 G194 P234 G235 T236 G237 K238 T239 L240 N335 I367 H371 G395 A396 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 TAILKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNPSALRETVV 4ko8 B 1.98 BS01 AGS A 1 R359 F360 R343 F344 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 LKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSN 4ko8 B 1.98 BS02 AGS B 1 G207 P247 G248 T249 G250 K251 T252 L253 N348 I380 H384 G408 A409 G191 P231 G232 T233 G234 K235 T236 L237 N332 I364 H368 G392 A393 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 LKQKNRPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSN 4kod A 2.96 BS01 ADP A 1 I206 G207 G248 T249 G250 K251 T252 L253 I380 H384 G408 A409 I185 G186 G227 T228 G229 K230 T231 L232 I359 H363 G387 A388 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 RPNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQS 4kod E 2.96 BS01 ADP E 1 I206 G207 G248 T249 G250 K251 T252 L253 I380 H384 G408 A409 I184 G185 G226 T227 G228 K229 T230 L231 I358 H362 G386 A387 3.6.4.6 0005524,0016887 remove_due_to_license_issue P55072 24196964 800 PNRLIVDEAINEDNSVVSLSQPKMDELQLFRGDTVLLKGKKRREAVCIVLSDDTCSDEKIRMNRVVRNNLRVRLGDVISIQPCPDVKYGKRIHVLPIDDTVEGITGNLFEVYLKPYFLEAYRPIRKGDIFLVHGGMRAVEFKVVETDPSPYCIVAPDTVIHCEGEPIKREDEEESLNEVGYDDIGGCRKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRKKMDLIDLEDETIDAEVMNSLAVTMDDFRWALSQSNP 4kom A 2.604 BS01 SIA C 1 Y88 A125 T126 W142 H174 E181 L217 Y86 A123 T124 W140 H172 E179 L215 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRU4 24009358 4 ICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARPQVNGLSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4kon A 2.6 BS01 SIA C 1 Y88 A125 T126 S127 W142 H174 E181 Y86 A123 T124 S125 W140 H172 E179 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRU4 24009358 2 ICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARPQVNGLSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4kot A 1.55 BS01 CE3 A 1 C29 P31 R49 Y68 G79 N80 M81 F118 R141 L151 C29 P31 R49 Y68 G79 N80 M81 F118 R141 L151 ? 0016747,0046872 Kd=3.5uM remove_due_to_license_issue Q9HV14 24003232 205 MQLSHRPAETGDLETVAGFPQDRDELFYCYPKAIWPFSVAQLAAAIAERRGSTVAVHDGQVLGFANFYQWQHGDFCALGNMMVAPAARGLGVARYLIGVMENLAREQYKARLMKISCFNANAAGLLLYTQLGYQPRAIAERHDPDGRRVALIQMDKPLE 4kov A 1.6 BS01 KOV A 1 C29 P31 R49 Y68 G79 N80 M81 S116 F118 R141 L151 C29 P31 R49 Y68 G79 N80 M81 S116 F118 R141 L151 ? 0016747,0046872 Kd=176.7uM remove_due_to_license_issue Q9HV14 24003232 204 MQLSHRPAETGDLETVAGFPQDRDELFYCYPKAIWPFSVAQLAAAIAERRGSTVAVHDGQVLGFANFYQWQHGDFCALGNMMVAPAARGLGVARYLIGVMENLAREQYKARLMKISCFNANAAGLLLYTQLGYQPRAIAERHDPDGRRVALIQMDKPLE 4kow A 1.45 BS01 CFX A 1 C29 P31 R49 Y68 G79 N80 S116 F118 R141 L151 C29 P31 R49 Y68 G79 N80 S116 F118 R141 L151 ? 0016747,0046872 Kd=49.3uM remove_due_to_license_issue Kd=4.93e+4nM Q9HV14 24003232 204 MQLSHRPAETGDLETVAGFPQDRDELFYCYPKAIWPFSVAQLAAAIAERRGSTVAVHDGQVLGFANFYQWQHGDFCALGNMMVAPAARGLGVARYLIGVMENLAREQYKARLMKISCFNANAAGLLLYTQLGYQPRAIAERHDPDGRRVALIQMDKPLE 4kox A 1.8 BS01 CLS A 1 C29 P31 R49 Y68 G79 N80 M81 S116 R141 C29 P31 R49 Y68 G79 N80 M81 S116 R141 ? 0016747,0046872 Kd=16.9uM remove_due_to_license_issue Kd=1.69e+4nM Q9HV14 24003232 205 MQLSHRPAETGDLETVAGFPQDRDELFYCYPKAIWPFSVAQLAAAIAERRGSTVAVHDGQVLGFANFYQWQHGDFCALGNMMVAPAARGLGVARYLIGVMENLAREQYKARLMKISCFNANAAGLLLYTQLGYQPRAIAERHDPDGRRVALIQMDKPLE 4kp0 A 2.8 BS01 KPK A 1 H57 A190 F191 K192 G193 S195 Y215 G216 H45 A171 F172 K173 G174 S176 Y192 G193 H57 D102 K192 G193 D194 S195 G196 H45 D89 K173 G174 D175 S176 G177 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 remove_due_to_license_issue IC50=22nM P23946 24121339 301 IIGGTECKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGVAQGIVSYGRSDAKPPAVFTRISHYRPWINQILQAN 4kp4 A 3.0 BS01 ANP A 1 H243 N1347 R1350 Y1351 D1373 I1378 R1392 G1393 A1396 G1401 T1402 G1403 L1404 G1405 L1406 L1430 H13 N125 R128 Y129 D151 I156 R170 G171 A174 G179 T180 G181 L182 G183 L184 L208 2.7.13.3 0000155,0007165,0016310,0016772 remove_due_to_license_issue P0AEJ4,Q9WZV7 24500224 1501 ADDRTLLMAGVSHDLRTPLTRIRAYAETIYNSLGELDLSTLKELAESINKDIEECNAIIEQFIDYLRTGQEMPMEMADLNAVLGEVIAAESGYEREIETALYPGSIEVKMHPLSIKRAVANMVVNAARYGNGWIKVSSGTEPNRAWFQVEDDGPGIAPEQRKHLFQPFVRGDSARTISGTGLGLAIVQRIVDNHNGMLELGTSERGGLSIRAWLPVPVT 4kp5 A 1.45 BS02 E1F A 1 H91 H117 V119 S133 L197 T198 W208 H89 H115 V117 S131 L195 T196 W206 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=833nM remove_due_to_license_issue koff=0.31s-1, Kd=833nM, kon=1600000M-1-s-1 O43570 24103428 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4kp6 A 1.5 BS01 1S1 A 1 H234 N395 T407 I410 M431 Q443 F446 H73 N234 T246 I249 M270 Q282 F285 3.1.4.53 0004114,0007165,0008081 ic50=0.87nM remove_due_to_license_issue Q07343 23806553 501 NEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIP 4kp8 A 1.8 BS02 E1G A 1 Q89 H91 H93 H117 V119 S133 L197 T198 T199 P201 Q87 H89 H91 H115 V117 S131 L195 T196 T197 P199 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=3330nM remove_due_to_license_issue Kd=1300nM O43570 24103428 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4kpx A 2.21 BS01 1SE A 1 L11 A12 A13 G14 Y103 D105 Y139 T170 V223 G225 L8 A9 A10 G11 Y100 D102 Y136 T167 V220 G222 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=0.05uM remove_due_to_license_issue P43889 25262942 511 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 4kpz A 2.09 BS01 1SF A 1 L11 A12 A13 G14 V26 Q76 Q79 G81 D105 L8 A9 A10 G11 V23 Q73 Q76 G78 D102 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 remove_due_to_license_issue P43889 25262942 501 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 4kql A 2.31 BS01 1SG A 1 A12 A13 Q76 Q79 G81 T82 Y103 D105 Y139 T170 V223 G225 A9 A10 Q73 Q76 G78 T79 Y100 D102 Y136 T167 V220 G222 R18 R15 2.3.1.157,2.7.7.23 0000287,0000902,0003977,0005737,0006048,0008360,0009245,0009252,0016020,0016740,0016746,0016779,0019134,0046872,0071555 ic50=0.0017uM remove_due_to_license_issue P43889 25262942 511 KALSAVILAAGKGTRMYSDLPKVLHTIAGKPMVKHVIDTAHQLGSENIHLIYGHGGDLMRTHLANEQVNWVLQTEQLGTAHAVQQAAPFFKDNENIVVLYGDAPLITKETLEKLIEAKPENGIALLTVNLDNPTGYGRIIRENGNVVAIVEQKDANAEQLNIKEVNTGVMVSDGASFKKWLARVGNNNAQGEYYLTDLIALANQDNCQVVAVQATDVMEVEGANNRLQLAALERYFQNKQASKLLLEGVMIYDPARFDLRGTLEHGKDVEIDVNVIIEGNVKLGDRVKIGTGCVLKNVVIGNDVEIKPYSVLEDSIVGEKAAIGPFSRLRPGAELAAETHVGNFVEIKKSTVGKGSKVNHLTYVGDSEIGSNCNIGAGVITCNYDGANKFKTIIGDDVFVGSDTQLVAPVKVANGATIGAGTTITRDVGENELVITRVAQRHIQGWQRPI 4kqo A 2.31 BS01 JPP A 1 S294 Y328 S349 Y409 S485 G486 T487 A488 R489 Y498 S245 Y279 S300 Y360 S436 G437 T438 A439 R440 Y449 3.4.16.4 0000917,0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0043093,0051301,0071555 remove_due_to_license_issue G3XD46 23899657 601 ARSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKVSVGTKGYRENAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPT 4kqp A 0.95 BS01 GLN A 1 F270 F308 G326 M327 S328 R333 K373 T376 A377 D417 F16 F54 G72 M73 S74 R79 K119 T122 A123 D163 ? 0015276,0016020 Kd=0.9uM remove_due_to_license_issue Q9CES5 23994008 501 ATPKKDVYTIASDNSFAPFEFQNDDKQFTGIDVDLLNAIAKNQGFKLKWNFIGFQAAVDSVQSGHADGMMSGMSITDARKQVFDYGSPYYSSNLTIATSSTDDSIKSWKDLKGKTLGAKNGTASFDYLNAHAKEYGYTVKTFTDATTMYSSLNNGSINALMDDEPVIKYAIKQGQKFATPIKPIPDGQYGFAVKKGSNPELIEMFNNGLANLRANGEYDKIIDKYLESDA 4kqq A 2.1 BS01 VPP A 1 S294 V333 S349 Y407 Y409 S485 G486 T487 R489 Y498 Y503 F533 G534 G535 S244 V283 S299 Y357 Y359 S435 G436 T437 R439 Y448 Y453 F483 G484 G485 3.4.16.4 0000917,0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0043093,0051301,0071555 ic50=126uM remove_due_to_license_issue G3XD46 23899657 601 RSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKVSVGTKGYRENAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPTATEQQQVN 4kqr A 2.01 BS01 VPP A 1 S294 V333 S349 Y407 Y409 S485 G486 T487 R489 Y498 Y503 F533 G534 G535 S244 V283 S299 Y357 Y359 S435 G436 T437 R439 Y448 Y453 F483 G484 G485 3.4.16.4 0000917,0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0043093,0051301,0071555 ic50=126uM remove_due_to_license_issue G3XD46 23899657 601 RSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKVSVGTKGYRENAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPTATEQQQVN 4krs A 2.29 BS02 1SX A 1 H1184 G1185 S1186 F1188 Y1203 Y1213 S1221 Y1224 H80 G81 S82 F84 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=0.299uM remove_due_to_license_issue O95271 23879431 1406 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRAYAEYVIYRGEQAYPEYLITYQIMKPE 4ks1 A 2.2 BS02 2H8 A 1 R118 E119 D151 R152 R224 E276 E277 R292 R371 Y406 R36 E37 D69 R70 R143 E195 E196 R211 R288 Y322 D151 E277 R292 R371 Y406 D69 E196 R211 R288 Y322 3.2.1.18 0004308,0005975,0016020,0033644,0055036 Ki=1.5nM remove_due_to_license_issue Q07599 24129600 502 TYMNNTEAICDVKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVKVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVINSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQADISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDAQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQVRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEIADWSWHDGAILPFDIDK 4ks2 A 2.595 BS02 1SJ A 1 E119 D151 R152 W178 R224 E276 E277 R292 N294 R371 Y406 E37 D69 R70 W97 R143 E195 E196 R211 N213 R288 Y322 D151 E277 R292 R371 Y406 D69 E196 R211 R288 Y322 3.2.1.18 0004308,0005975,0016020,0033644,0055036 remove_due_to_license_issue Q0A480 24129600 502 TYMNNTEAICDVKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVKVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVINSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQADISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDAQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQVRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEIADWSWHDGAILPFDIDK 4ks3 A 2.6 BS01 1SL A 1 R118 E119 T148 K150 D151 R152 R156 W178 R224 E276 R371 Y406 R36 E37 T66 K68 D69 R70 R74 W97 R143 E195 R288 Y322 D151 E277 R292 R371 Y406 D69 E196 R211 R288 Y322 3.2.1.18 0004308,0005975,0016020,0033644,0055036 remove_due_to_license_issue Q0A480 24129600 501 TYMNNTEAICDVKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVKVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVINSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQADISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDAQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQVRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEIADWSWHDGAILPFDID 4ks4 A 2.495 BS01 1SN A 1 R118 E119 D151 R152 R156 W178 R224 E276 E277 R292 R371 Y406 R36 E37 D69 R70 R74 W97 R143 E195 E196 R211 R288 Y322 D151 E277 R292 R371 Y406 D69 E196 R211 R288 Y322 3.2.1.18 0004308,0005975,0016020,0033644,0055036 Ki=72nM remove_due_to_license_issue Q0A480 24129600 501 TYMNNTEAICDVKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVKVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVINSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQADISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDAQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQVRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEIADWSWHDGAILPFDIDK 4ks5 A 2.699 BS02 1SO A 1 E119 D151 R152 R156 W178 R224 E276 R292 Y406 E37 D69 R70 R74 W97 R143 E195 R211 Y322 D151 E277 R292 R371 Y406 D69 E196 R211 R288 Y322 3.2.1.18 0004308,0005975,0016020,0033644,0055036 remove_due_to_license_issue Q0A480 24129600 502 TYMNNTEAICDVKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVKVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVINSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQADISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDAQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQVRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEIADWSWHDGAILPFDID 4ksp A 2.93 BS01 1SU A 1 V470 A480 K482 E500 L504 I526 T528 W530 C531 G533 H573 F582 D593 F594 V24 A34 K36 E54 L58 I80 T82 W84 C85 G87 H127 F136 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S151 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=77nM P15056 23906342 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP 4ksq A 3.3 BS01 1SW A 1 A480 K482 E500 L504 I526 T528 W530 C531 G533 F582 I591 G592 D593 F594 A34 K36 E54 L58 I80 T82 W84 C85 G87 F136 I145 G146 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 23906342 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLP 4ksy A 1.881 BS01 1SY A 1 S162 Y163 Y167 R238 T263 S11 Y12 Y16 R87 T112 ? 0002218,0032481 Kd=3.79nM remove_due_to_license_issue Q86WV6 23747010 500 NFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPSFSLSQEVLRHLRQE 4ktc A 2.3 BS03 1X3 A 1 Q41 F43 H57 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 D168 Q41 F43 H57 D81 V132 L135 K136 G137 S139 F154 R155 A156 A157 D168 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 ic50=1nM remove_due_to_license_issue P26662 23672640 202 APITAYSQQTRGLLGCIITSLTGRDKNQVDGEVQVLSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWPAPPGARSMTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHVVGIFRAAVCTRGVAKAVDFIPVESM 4kud A 3.203 BS01 dna I 0 Y41 K42 R72 R83 F84 Q85 V117 T118 Y4 K5 R35 R46 F47 Q48 V80 T81 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006355,0006878,0008823,0009060,0009303,0030527,0031298,0042790,0043505,0043935,0045943,0046982,0070911 remove_due_to_license_issue P61830 23934152 1 ~ 146 PHRYKPGTVALREIRRFQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAIGALQESVEAYLVSLFEDTNLAAIHAKRVTIQKKDIKLARRLRGE 4kud A 3.203 BS02 dna J 0 R40 Y41 G44 V46 A47 R49 R63 L65 R69 R83 R3 Y4 G7 V9 A10 R12 R26 L28 R32 R46 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006355,0006878,0008823,0009060,0009303,0030527,0031298,0042790,0043505,0043935,0045943,0046982,0070911 remove_due_to_license_issue P61830 23934152 147 ~ 292 PHRYKPGTVALREIRRFQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAIGALQESVEAYLVSLFEDTNLAAIHAKRVTIQKKDIKLARRLRGE 4kud B 3.203 BS01 dna I 0 R17 R19 P32 R36 R45 R3 R5 P18 R22 R31 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006334,0006355,0030527,0031298,0042790,0042802,0045943,0046982 remove_due_to_license_issue P02309 23934152 1 ~ 146 AKRHRKILRDNIQGITKPAIRRLARRGGVKRISGLIYEEVRAVLKSFLESVIRDSVTYTEHAKRKTVTSLDVVYALKRQGRTLYGFGG 4kud B 3.203 BS02 dna J 0 R35 R45 I46 S47 R78 K79 T80 R21 R31 I32 S33 R64 K65 T66 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006334,0006355,0030527,0031298,0042790,0042802,0045943,0046982 remove_due_to_license_issue P02309 23934152 147 ~ 292 AKRHRKILRDNIQGITKPAIRRLARRGGVKRISGLIYEEVRAVLKSFLESVIRDSVTYTEHAKRKTVTSLDVVYALKRQGRTLYGFGG 4kud C 3.203 BS01 dna I 0 Q16 R18 R33 Q42 R43 R78 Q1 R3 R18 Q27 R28 R63 ? 0000786,0003677,0005634,0005694,0006281,0006325,0030527,0031298,0031507,0046982 remove_due_to_license_issue P04912 23934152 1 ~ 146 QSRSAKAGLTFPVGRVHRLLRRGNYAQRIGSGAPVYLTAVLEYLAAEILELAGNAARDNKKTRIIPRHLQLAIRNDDELNKLLGNVTIAQGGVLPNIHQNLLP 4kud C 3.203 BS02 dna J 0 R30 R43 I44 S46 T77 R78 R15 R28 I29 S31 T62 R63 ? 0000786,0003677,0005634,0005694,0006281,0006325,0030527,0031298,0031507,0046982 remove_due_to_license_issue P04912 23934152 147 ~ 292 QSRSAKAGLTFPVGRVHRLLRRGNYAQRIGSGAPVYLTAVLEYLAAEILELAGNAARDNKKTRIIPRHLQLAIRNDDELNKLLGNVTIAQGGVLPNIHQNLLP 4kud D 3.203 BS01 dna I 0 Y45 I57 S58 Q59 S90 T91 Y9 I21 S22 Q23 S54 T55 ? 0000122,0000786,0003677,0005515,0005634,0005694,0006301,0006325,0006355,0030527,0031298,0046982 remove_due_to_license_issue P02293 23934152 1 ~ 146 KETYSSYIYKVLKQTHPDTGISQKSMSILNSFVNDIFERIATEASKLAAYNKKSTISAREIQTAVRLILPGELAKHAVSEGTRAVTKYSSSTQ 4kud D 3.203 BS02 dna J 0 K37 T39 Y43 K1 T3 Y7 ? 0000122,0000786,0003677,0005515,0005634,0005694,0006301,0006325,0006355,0030527,0031298,0046982 remove_due_to_license_issue P02293 23934152 147 ~ 292 KETYSSYIYKVLKQTHPDTGISQKSMSILNSFVNDIFERIATEASKLAAYNKKSTISAREIQTAVRLILPGELAKHAVSEGTRAVTKYSSSTQ 4kud E 3.203 BS01 dna I 0 R40 Y41 G44 V46 A47 R63 K64 L65 R69 R83 R5 Y6 G9 V11 A12 R28 K29 L30 R34 R48 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006355,0006878,0008823,0009060,0009303,0030527,0031298,0042790,0043505,0043935,0045943,0046982,0070911 remove_due_to_license_issue P61830 23934152 1 ~ 146 KKPHRYKPGTVALREIRRFQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAIGALQESVEAYLVSLFEDTNLAAIHAKRVTIQKKDIKLARRLRGE 4kud E 3.203 BS02 dna J 0 Y41 K42 T45 R63 R72 R83 F84 Q85 S86 R116 V117 T118 Y6 K7 T10 R28 R37 R48 F49 Q50 S51 R81 V82 T83 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006355,0006878,0008823,0009060,0009303,0030527,0031298,0042790,0043505,0043935,0045943,0046982,0070911 remove_due_to_license_issue P61830 23934152 147 ~ 292 KKPHRYKPGTVALREIRRFQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAIGALQESVEAYLVSLFEDTNLAAIHAKRVTIQKKDIKLARRLRGE 4kud F 3.203 BS01 dna I 0 R45 I46 S47 G48 K79 T80 R33 I34 S35 G36 K67 T68 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006334,0006355,0030527,0031298,0042790,0042802,0045943,0046982 remove_due_to_license_issue P02309 23934152 1 ~ 146 GGAKRHRKILRDNIQGITKPAIRRLARRGGVKRISGLIYEEVRAVLKSFLESVIRDSVTYTEHAKRKTVTSLDVVYALKRQGRTLYGFGG 4kud F 3.203 BS02 dna J 0 R17 R19 T30 P32 R36 R45 R5 R7 T18 P20 R24 R33 ? 0000500,0000786,0003677,0005515,0005634,0005694,0006325,0006334,0006355,0030527,0031298,0042790,0042802,0045943,0046982 remove_due_to_license_issue P02309 23934152 147 ~ 292 GGAKRHRKILRDNIQGITKPAIRRLARRGGVKRISGLIYEEVRAVLKSFLESVIRDSVTYTEHAKRKTVTSLDVVYALKRQGRTLYGFGG 4kud G 3.203 BS01 dna I 0 S15 R30 R43 S46 K76 T77 R78 S1 R16 R29 S32 K62 T63 R64 ? 0000786,0003677,0005634,0005694,0006281,0006325,0030527,0031298,0031507,0046982 remove_due_to_license_issue P04912 23934152 1 ~ 146 SQSRSAKAGLTFPVGRVHRLLRRGNYAQRIGSGAPVYLTAVLEYLAAEILELAGNAARDNKKTRIIPRHLQLAIRNDDELNKLLGNVTIAQGGVLPNIHQNLLPK 4kud G 3.203 BS02 dna J 0 S15 R18 R33 Q42 R43 R78 S1 R4 R19 Q28 R29 R64 ? 0000786,0003677,0005634,0005694,0006281,0006325,0030527,0031298,0031507,0046982 remove_due_to_license_issue P04912 23934152 147 ~ 292 SQSRSAKAGLTFPVGRVHRLLRRGNYAQRIGSGAPVYLTAVLEYLAAEILELAGNAARDNKKTRIIPRHLQLAIRNDDELNKLLGNVTIAQGGVLPNIHQNLLPK 4kud H 3.203 BS01 dna I 0 R36 E38 T39 Y43 R1 E3 T4 Y8 ? 0000122,0000786,0003677,0005515,0005634,0005694,0006301,0006325,0006355,0030527,0031298,0046982 remove_due_to_license_issue P02293 23934152 1 ~ 146 RKETYSSYIYKVLKQTHPDTGISQKSMSILNSFVNDIFERIATEASKLAAYNKKSTISAREIQTAVRLILPGELAKHAVSEGTRAVTKYSSSTQ 4kud H 3.203 BS02 dna J 0 R36 Y45 Q59 K89 S90 T91 R1 Y10 Q24 K54 S55 T56 ? 0000122,0000786,0003677,0005515,0005634,0005694,0006301,0006325,0006355,0030527,0031298,0046982 remove_due_to_license_issue P02293 23934152 147 ~ 292 RKETYSSYIYKVLKQTHPDTGISQKSMSILNSFVNDIFERIATEASKLAAYNKKSTISAREIQTAVRLILPGELAKHAVSEGTRAVTKYSSSTQ 4kup A 1.311 BS01 1TZ A 1 D33 D35 Y79 G80 D81 F116 D219 G221 T222 Y226 I300 D33 D35 Y79 G80 D81 F116 D219 G221 T222 Y226 I300 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=6uM remove_due_to_license_issue P11838 24532096 401 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4kup A 1.311 BS02 1TZ A 2 D15 D119 T223 D15 D119 T223 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=6uM remove_due_to_license_issue P11838 24532096 402 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4kv9 A 1.93 BS01 GDP A 1 G51 G53 K54 S55 T56 K184 D186 V237 R253 G12 G14 K15 S16 T17 K127 D129 V180 R193 ? 0000287,0003924,0005525,0005737,0005856,0019003,0031105,0031982,0042802,0042803,0046872,0046982,0051260 Kd=0.000146M remove_due_to_license_issue A0A3Q0KDV9 24464615 500 FVFNILCVGETGIGKSTLLETLFNQKFDFKLKAVTYDLKEANVKLKLTVVETCENNIKPVVDYIDNQFENYLQEELKMKRSMQAFHDTRVHVCLYFIAPTGHSLKSIDLVAMKKLENKVNVIPVIAKSDTITKSELQKFKARILSEIQSNEIGIYQFPTDDEAVSETNSVMNQHIPFAVVGSSEEVKITVRVRQYPWGSVQVENENHCDFVRLREMLLRVNMEDLRERTHGVHYETYRRQRLIEMG 4kv9 B 1.93 BS01 GDP B 1 G51 G53 K54 S55 T56 K184 D186 V237 R253 G12 G14 K15 S16 T17 K131 D133 V184 R200 ? 0000287,0003924,0005525,0005737,0005856,0019003,0031105,0031982,0042802,0042803,0046872,0046982,0051260 Kd=0.000146M remove_due_to_license_issue A0A3Q0KDV9 24464615 500 FVFNILCVGETGIGKSTLLETLFNQKFDFSPKLKAVTYDLKEANVKLKLTVVETCNKENNIKPVVDYIDNQFENYLQEELKMKRSMQAFHDTRVHVCLYFIAPTGHSLKSIDLVAMKKLENKVNVIPVIAKSDTITKSELQKFKARILSEIQSNEIGIYQFPTDDEAVSETNSVMNQHIPFAVVGSSEEVKINGKTVRVRQYPWGSVQVENENHCDFVRLREMLLRVNMEDLRERTHGVHYETYRRQRLIEMG 4kva A 2.14 BS01 GTP A 1 T50 G51 G53 K54 S55 T56 E100 K184 D186 V237 R253 T11 G12 G14 K15 S16 T17 E48 K128 D130 V181 R193 ? 0000287,0003924,0005525,0005737,0005856,0019003,0031105,0031982,0042802,0042803,0046872,0046982,0051260 Kd=0.000115M remove_due_to_license_issue A0A3Q0KDV9 24464615 500 FVFNILCVGETGIGKSTLLETLFNQKFDFPKLKAVTYDLKKLKLTVVETCGYGDENNIKPVVDYIDNQFENYLQEELKMKRSMQAFHDTRVHVCLYFIAPTGHSLKSIDLVAMKKLENKVNVIPVIAKSDTITKSELQKFKARILSEIQSNEIGIYQFPTDDEAVSETNSVMNQHIPFAVVGSSEEVKTVRVRQYPWGSVQVENENHCDFVRLREMLLRVNMEDLRERTHGVHYETYRRQRLIEMG 4kva A 2.14 BS03 GTP B 1 T187 E192 T131 E136 ? 0000287,0003924,0005525,0005737,0005856,0019003,0031105,0031982,0042802,0042803,0046872,0046982,0051260 Kd=0.000115M remove_due_to_license_issue A0A3Q0KDV9 24464615 500 FVFNILCVGETGIGKSTLLETLFNQKFDFPKLKAVTYDLKKLKLTVVETCGYGDENNIKPVVDYIDNQFENYLQEELKMKRSMQAFHDTRVHVCLYFIAPTGHSLKSIDLVAMKKLENKVNVIPVIAKSDTITKSELQKFKARILSEIQSNEIGIYQFPTDDEAVSETNSVMNQHIPFAVVGSSEEVKTVRVRQYPWGSVQVENENHCDFVRLREMLLRVNMEDLRERTHGVHYETYRRQRLIEMG 4kva B 2.14 BS01 GTP B 1 T50 G51 G53 K54 S55 T56 K184 D186 V237 G238 R253 T11 G12 G14 K15 S16 T17 K136 D138 V189 G190 R205 ? 0000287,0003924,0005525,0005737,0005856,0019003,0031105,0031982,0042802,0042803,0046872,0046982,0051260 Kd=0.000115M remove_due_to_license_issue A0A3Q0KDV9 24464615 500 FVFNILCVGETGIGKSTLLETLFNQKFDFSPKLKAVTYDLKEANVKLKLTVVETCGYGDQNKENNIKPVVDYIDNQFENYLQEELKMKRSMQAFHDTRVHVCLYFIAPTGHSLKSIDLVAMKKLENKVNVIPVIAKSDTITKSELQKFKARILSEIQSNEIGIYQFPTDDEAVSETNSVMNQHIPFAVVGSSEEVKINGKTVRVRQYPWGSVQVENENHCDFVRLREMLLRVNMEDLRERTHGVHYETYRRQRLIEMG 4kvm E 2.597 BS02 1XE I 1 N21 L22 V76 S77 V78 R83 H84 G86 L87 A88 H111 V112 N116 A118 L122 Y123 N21 L22 V76 S77 V78 R83 H84 G86 L87 A88 H111 V112 N116 A118 L122 Y123 2.3.1.255 0004596,0006474,0016747,0031415 remove_due_to_license_issue Q9UTI3 23912279 5201 MDIRPARISDLTGMQNCNLHNLPENYQLKYYLYHAISWPMLSYVATDPKGRVVGYVLAKMEEEPKDGIPHGHITSVSVMRSYRHLGLAKRLMVQSQRAMVEVYGAKYMSLHVRKSNRAAIHLYRDTLQFDVQGIESKYYADGEDAYAMHKDFS 4kwf A 2.31 BS01 3AK A 1 F170 M174 W177 E268 C301 C302 C303 D457 F459 F465 F164 M168 W171 E262 C295 C296 C297 D451 F453 F459 N169 K192 E268 C302 E399 E476 N163 K186 E262 C296 E393 E470 1.2.1.3 0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627 Ki=15uM remove_due_to_license_issue Ki=34000nM, IC50=82000nM P05091 24444054 601 AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS 4kwg A 2.1 BS01 2AK A 1 F170 M174 C301 C302 C303 D457 F459 F164 M168 C295 C296 C297 D451 F453 N169 K192 E268 C302 E399 E476 N163 K186 E262 C296 E393 E470 1.2.1.3 0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627 Ki=1uM remove_due_to_license_issue Ki=1000nM, IC50=2400nM P05091 24444054 601 AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS 4kwo A 1.32 BS01 1UD A 1 D102 Y106 Q107 D156 C158 G229 L231 A232 M260 G261 D80 Y84 Q85 D125 C127 G198 L200 A201 M229 G230 D102 D280 C318 C320 C323 H349 D80 D249 C287 C289 C292 H318 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=353nM remove_due_to_license_issue P28720 25483606 401 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAAGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSTKQSEEGVTFKHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4kwp A 1.25 BS01 EXX A 1 V66 K68 F113 V116 N118 M163 I174 V65 K67 F112 V115 N117 M162 I173 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.04uM remove_due_to_license_issue P68400 24442476 408 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 4kww A 2.55 BS01 PHT A 1 T137 R138 H160 R161 M169 K171 T136 R137 H159 R160 M168 K170 R102 K139 K171 E201 D222 R101 K138 K170 E200 D221 2.4.2.19 0004514,0005515,0005737,0005829,0009435,0016757,0016763,0019363,0019674,0034213,0042802,0070062,1902494 remove_due_to_license_issue Q15274 24038671 300 DAEGLALLLPPVTLAALVDSWLREDCPGLNYAALVSGAGPSQAALWAKSPGVLAGQPFFDAIFTQLNCQVSWFLPEGSKLVPVARVAEVRGPAHCLLLGERVALNTLARCSGIASAAAAAVEAARGAGWTGHVAGTRKTTPGFRLVEKYGLLVGGAASHRYDLGGLVMVKDNHVVAAGGVEKAVRAARQAADFTLKVEVECSSLQEAVQAAEAGADLVLLDNFKPEELHPTATVLKAQFPSVAVEASGGITLDNLPQFCGPHIDVISMGMLTQAAPALDFSLKLF 4kww B 2.55 BS01 PHT B 1 T137 R138 H160 R161 M169 K171 T136 R137 H159 R160 M168 K170 R102 K139 K171 E201 D222 R101 K138 K170 E200 D221 2.4.2.19 0004514,0005515,0005737,0005829,0009435,0016757,0016763,0019363,0019674,0034213,0042802,0070062,1902494 remove_due_to_license_issue Q15274 24038671 300 DAEGLALLLPPVTLAALVDSWLREDCPGLNYAALVSGAGPSQAALWAKSPGVLAGQPFFDAIFTQLNCQVSWFLPEGSKLVPVARVAEVRGPAHCLLLGERVALNTLARCSGIASAAAAAVEAARGAGWTGHVAGTRKTTPGFRLVEKYGLLVGGAASHRYDLGGLVMVKDNHVVAAGGVEKAVRAARQAADFTLKVEVECSSLQEAVQAAEAGADLVLLDNFKPEELHPTATVLKAQFPSVAVEASGGITLDNLPQFCGPHIDVISMGMLTQAAPALDFSLKLF 4kww C 2.55 BS01 PHT C 1 T137 R138 H160 R161 M169 K171 T136 R137 H159 R160 M168 K170 R102 K139 K171 E201 D222 R101 K138 K170 E200 D221 2.4.2.19 0004514,0005515,0005737,0005829,0009435,0016757,0016763,0019363,0019674,0034213,0042802,0070062,1902494 remove_due_to_license_issue Q15274 24038671 300 DAEGLALLLPPVTLAALVDSWLREDCPGLNYAALVSGAGPSQAALWAKSPGVLAGQPFFDAIFTQLNCQVSWFLPEGSKLVPVARVAEVRGPAHCLLLGERVALNTLARCSGIASAAAAAVEAARGAGWTGHVAGTRKTTPGFRLVEKYGLLVGGAASHRYDLGGLVMVKDNHVVAAGGVEKAVRAARQAADFTLKVEVECSSLQEAVQAAEAGADLVLLDNFKPEELHPTATVLKAQFPSVAVEASGGITLDNLPQFCGPHIDVISMGMLTQAAPALDFSLKLF 4kxb A 2.4 BS02 BES A 1 E223 T356 G357 A358 M359 E360 H393 E394 H397 E416 F474 Y479 R887 E148 T281 G282 A283 M284 E285 H318 E319 H322 E341 F399 Y404 R808 E360 H393 E394 H397 E416 T471 Y479 E285 H318 E319 H322 E341 T396 Y404 3.4.11.7 0001525,0002003,0003081,0004177,0005615,0005737,0005765,0005886,0005903,0006508,0007267,0008217,0008233,0008237,0008270,0008283,0009897,0016324,0016477,0031410,0032835,0042277,0043171,0045177,0046872,0070006,0070062 remove_due_to_license_issue Q07075 23888046 1017 DICPASEDESGQWKNFRLPDFVNPVHYDLHVKPLLEEDTYTGTVSISINLSAPTRYLWLHLRETRITRLPELKRPSGDQVQVRRCFEYKKQEYVVVEAEEELTPSSGDGLYLLTMEFAGWLNGSLVGFYRTTYTENGRVKSIAATDHEPTDARKSFPCFDEPNKKATYTISITHPKEYGALSNMPVAKEESVDDKWTRTTFEKSVPMSTYLVCFAVHQFDSVKRISNSGKPLTIYVQPEQKHTAEYAANITKSVFDYFEEYFAMNYSLPKLDKIAIPDFGTGAMENWGLITYRETNLLYDPKESASSNQQRVATVVAHELVHQWFGNIVTMDWWEDLWLNEGFASFFEFLGVNHAETDWQMRDQMLLEDVLPVQEDDSLMSSHPIIVTVTTPDEITSVFDGISYSKGSSILRMLEDWIKPENFQKGCQMYLEKYQFKNAKTSDFWAALEEASRLPVKEVMDTWTRQMGYPVLNVNGVKNITQKRFLLDPRANPSQPPSDLGYTWNIPVKWTEDNITSSVLFNRSEKEGITLNSGNAFLKINPDHIGFYRVNYEVATWDSIATALSLNHKTFSSADRASLIDDAFALARAQLLDYKVALNLTKYLKREENFLPWQRVISAVTYIISMFEDDKELYPMIEEYFQGQVKPIADSLGWNDAGDHVTKLLRSSVLGFACKMGDREALNNASSLFEQWLNGTVSLPVNLRLLVYRYGMQNSGNEISWNYTLEQYQKTSLAQEKEKLLYGLASVKNVTLLSRYLDLLKDTNLIKTQDVFTVIRYISYNSYGKNMAWNWIQLNWDYLVNRYTLNNRNLGRIVTIAEPFNTELQLWQMESFFAKYPQAGAGEKPREQVLETVKNNIEWLKQHRNTIREWFFNLL 4kxl A 1.69 BS01 6C6 A 1 C15 G16 S17 I18 R19 H45 V46 I65 N69 S87 G89 E93 C7 G8 S9 I10 R11 H37 V38 I48 N52 S70 G72 E76 3.2.2.- 0009159,0070694 Kd=0.6uM remove_due_to_license_issue O35820 24260472 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVAEAAGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYLV 4kxl A 1.69 BS02 6C6 B 1 S117 M119 S100 M102 3.2.2.- 0009159,0070694 Kd=0.6uM remove_due_to_license_issue O35820 24260472 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVAEAAGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYLV 4kxl B 1.69 BS01 6C6 A 1 S117 M119 S92 M94 3.2.2.- 0009159,0070694 Kd=0.6uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYL 4kxl B 1.69 BS02 6C6 B 1 C15 G16 S17 I18 R19 G20 I65 N69 S87 G89 E93 C6 G7 S8 I9 R10 G11 I40 N44 S62 G64 E68 3.2.2.- 0009159,0070694 Kd=0.6uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYL 4kxm A 2.24 BS01 6IA A 1 G16 I18 R19 H45 V46 I65 N69 S87 G89 E93 G7 I9 R10 H36 V37 I44 N48 S66 G68 E72 3.2.2.- 0009159,0070694 Kd=2.6uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYL 4kxm A 2.24 BS02 6IA B 1 S117 M119 S96 M98 3.2.2.- 0009159,0070694 Kd=2.6uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYL 4kxm B 2.24 BS01 6IA A 1 S117 M119 S97 M99 3.2.2.- 0009159,0070694 Kd=2.6uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYLV 4kxm B 2.24 BS02 6IA B 1 G16 S17 I18 R19 H45 V46 I65 N69 S87 G89 E93 G7 S8 I9 R10 H36 V37 I45 N49 S67 G69 E73 3.2.2.- 0009159,0070694 Kd=2.6uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYLV 4kxn A 1.9 BS01 6K6 A 1 G16 I18 R19 G20 H45 V46 F64 I65 Q68 N69 S87 G89 E93 G7 I9 R10 G11 H36 V37 F45 I46 Q49 N50 S68 G70 E74 3.2.2.- 0009159,0070694 Kd=0.8uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADAGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAY 4kxn A 1.9 BS02 6K6 B 1 S117 M119 S98 M100 3.2.2.- 0009159,0070694 Kd=0.8uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADAGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAY 4kxn B 1.9 BS01 6K6 B 1 C15 G16 I18 R19 I65 N69 S87 G89 E93 C6 G7 I9 R10 I39 N43 S61 G63 E67 3.2.2.- 0009159,0070694 Kd=0.8uM remove_due_to_license_issue O35820 24260472 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYLV 4kyh A 2.5 BS03 ZST A 1 M36 R38 F68 E100 T102 N104 M31 R33 F63 E95 T97 N99 Q34 E100 H127 E173 Q29 E95 H122 E168 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 remove_due_to_license_issue Q9CPU0 23857942 203 PASSGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIAT 4kyk B 2.0 BS03 IMN B 1 K151 K157 M158 L161 F163 K144 K150 M151 L154 F156 Q34 E100 H127 E173 Q27 E93 H120 E166 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 Ki=18uM remove_due_to_license_issue Q9CPU0 23857942 300 SSGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIATII 4kz0 A 2.87 BS01 1UJ A 1 W812 I831 Y867 E880 V882 A885 M953 I963 D964 W565 I584 Y620 E633 V635 A638 M706 I716 D717 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=4200nM P48736 23820386 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEVSLWDCDRKFRVKIRGIDIPVLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVRLLYYVNLLLIDHRFLLRRGEYVLHMWQIFNADKLTSATNPDKENSMSISILLDNEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNRVPFVLTPDFLFVMGTSKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 4kz3 A 1.67 BS01 1U1 A 1 V211 S212 Y221 T319 V208 S209 Y218 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1.7mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kz4 B 1.42 BS01 4A1 B 1 G63 S64 L119 N152 Y221 G317 A318 G60 S61 L116 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.07mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kz5 A 1.35 BS01 1U3 A 1 S64 N152 Y221 T319 G320 S61 N149 Y218 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki<10mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kz6 B 1.68 BS01 ZB6 B 1 S64 Q120 A318 S61 Q117 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.8mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kz7 A 1.43 BS01 1U5 A 1 S64 G317 A318 S61 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=3.2mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kz8 A 2.282 BS01 1U6 A 1 Y221 A318 T319 Y218 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1.6mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kz8 A 2.282 BS02 1U6 A 2 Q253 L254 Q250 L251 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1.6mM remove_due_to_license_issue P00811 24807704 402 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kza A 1.6 BS01 NZ9 A 1 L254 S257 P306 L251 S254 P303 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.2mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kza A 1.6 BS02 NZ9 A 2 K24 P26 G206 K342 K21 P23 G203 K339 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.2mM remove_due_to_license_issue P00811 24807704 402 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kza A 1.6 BS03 NZ9 A 3 S64 L119 N152 L293 G317 A318 T319 S61 L116 N149 L290 G314 A315 T316 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.2mM remove_due_to_license_issue P00811 24807704 404 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kza A 1.6 BS04 NZ9 A 4 Q120 V211 S212 Y221 T319 G320 Q117 V208 S209 Y218 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=0.2mM remove_due_to_license_issue P00811 24807704 405 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kzb A 1.37 BS01 NZ2 A 1 S64 N152 Y221 G317 A318 T319 N343 S61 N149 Y218 G314 A315 T316 N340 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1.3mM remove_due_to_license_issue P00811 24807704 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kzb A 1.37 BS02 NZ2 A 2 K239 P240 L241 A307 P330 K236 P237 L238 A304 P327 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1.3mM remove_due_to_license_issue P00811 24807704 402 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kzb A 1.37 BS04 NZ2 A 3 Q120 V211 S212 Y221 T319 G320 Q117 V208 S209 Y218 T316 G317 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1.3mM remove_due_to_license_issue P00811 24807704 404 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4kzc A 3.25 BS01 1UK A 1 W812 I831 K833 Y867 I879 I881 V882 A885 M953 I963 D964 W554 I571 K573 Y607 I619 I621 V622 A625 M693 I703 D704 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=8.2nM P48736 23820386 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKNCIFIVIHRSTTSQTIKVSPDDTPGAISFFTQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTANETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGNERVPFVLTPDFLFVMGTSKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 4kze H 2.404 BS01 rna R 0 Y34 P56 Y57 S58 S60 Y62 Q102 Y104 R105 R110 Y31 P53 Y54 S55 S57 Y59 Q99 Y101 R102 R107 remove_due_to_license_issue 24952597 1 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPYSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARQGYRRRSGRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 4kze L 2.404 BS01 rna R 0 S92 F95 S92 F95 remove_due_to_license_issue 24952597 1 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSYSFPSTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 4kzl A 2.0 BS01 20D A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=1100nM Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4kzq A 2.25 BS01 DFL A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4kzu A 2.1 BS01 A73 A 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 I1075 H80 G81 Y99 Y109 A111 K116 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l02 A 2.75 BS01 1V2 A 1 D81 F173 I174 V177 D178 F192 T196 L268 F288 F303 H311 G342 D77 F169 I170 V173 D174 F188 T192 L264 F284 F299 H307 G338 2.3.1.-,2.7.1.91 0000287,0001568,0001727,0003376,0003677,0005515,0005516,0005524,0005634,0005654,0005737,0005768,0005829,0005886,0005905,0006473,0006629,0006670,0006954,0007420,0008283,0008284,0008289,0008481,0010008,0010800,0010803,0016020,0016301,0016407,0017050,0019722,0030100,0030139,0030148,0030307,0030335,0031398,0031901,0032651,0032740,0034612,0035556,0035924,0038036,0043066,0043231,0045202,0045766,0045840,0045931,0045987,0046512,0046521,0048146,0050764,0051092,0051721,0070301,0071363,0071897,0090520,0098793,0150077,1900060,1900745,1901224,1903978,1905364 remove_due_to_license_issue IC50=20nM Q9NYA1 23845219 401 AMGSGVLPRPCRVLVLLNPRGGKGKALQLFRSHVQPLLAEAEISFTLMLTERRNHARELVRSEELGRWDALVVMSGDGLMHEVVNGLMERPDWETAIQKPLCSLPAGSGNALAASLNHYAGYEQVTNEDLLTNCTLLLCRRLLSPMNLLSLHTASGLRLFSVLSLAWGFIADVDLESEKYRRLGEMRFTLGTFLRLAALRTYRGRLAYLPVGRVGSKTPASPVVVQQGPVDAHLVPLEEPVPSHWTVVPDEDFVLVLALLHSHLGSEMFAAPMGRCAAGVMHLFYVRAGVSRAMLLRLFLAMEKGRHMEYECPYLVYVPVVAFRLEPKDGKGVFAVDGELMVSEAVQGQVHPNYFWMVSG 4l09 A 2.05 BS01 1UR A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l0b A 1.8 BS02 1UT A 1 H1031 G1032 F1035 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 F84 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l0i A 2.3 BS01 1UW A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l0l A 2.1 BS01 PFV A 1 E291 S294 V333 S349 N351 Y409 S485 G486 T487 A488 R489 Y503 F533 E239 S242 V281 S297 N299 Y357 S433 G434 T435 A436 R437 Y441 F471 3.4.16.4 0000917,0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0016757,0043093,0051301,0071555 remove_due_to_license_issue Q51504 23755848 601 VRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKNAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPTA 4l0s A 1.9 BS01 1UZ A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l0t A 2.1 BS01 1V0 A 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 H80 G81 Y99 Y109 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=140nM remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l0v A 1.7 BS01 1V1 A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l0y A 2.5 BS01 dna C 0 R142 K167 T169 V170 D171 R93 K118 T120 V121 D122 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q03347 24646888 1 ~ 16 SMVEVLADHPGELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPR 4l0y A 2.5 BS02 dna D 0 R80 K83 R135 R142 R174 R177 R31 K34 R86 R93 R125 R128 ? 0003677,0003700,0005524,0005634,0006355 remove_due_to_license_issue Q03347 24646888 101 ~ 116 SMVEVLADHPGELVRTDSPNFLCSVLPTHWRCNKTLPIAFKVVALGDVPDGTLVTVMAGNDENYSAELRNATAAMKNQVARFNDLRFVGRSGRGKSFTLTITVFTNPPQVATYHRAIKITVDGPREPR 4l0y B 2.5 BS01 dna C 0 Q336 L337 W375 K379 K383 M384 K388 R391 Y395 Y396 Q3 L4 W42 K46 K50 M51 K55 R58 Y62 Y63 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P14921 24646888 1 ~ 16 PIQLWQFLLELLTDKSCQSFISWTGDGWEFKLSDPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTAGKRYVYRFVCDLQSLLGYTPEELHAMLDVKP 4l0y B 2.5 BS02 dna D 0 Y386 R391 R394 Y397 K404 R409 Y410 Y53 R58 R61 Y64 K71 R76 Y77 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P14921 24646888 101 ~ 116 PIQLWQFLLELLTDKSCQSFISWTGDGWEFKLSDPDEVARRWGKRKNKPKMNYEKLSRGLRYYYDKNIIHKTAGKRYVYRFVCDLQSLLGYTPEELHAMLDVKP 4l10 A 1.7 BS02 A63 A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l19 A 1.66 BS06 1UA A 1 H222 L239 F241 P242 I243 T245 T247 F252 P255 H119 L136 F138 P139 I140 T142 T144 F149 P152 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.8uM remove_due_to_license_issue IC50=2400nM, Ki=824nM P45452 25330343 307 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 4l19 A 1.66 BS07 1UA A 2 Y176 A188 F189 H226 Y73 A85 F86 H123 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.8uM remove_due_to_license_issue IC50=2400nM, Ki=824nM P45452 25330343 308 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 4l1a A 1.9 BS01 AB1 A 1 N25 G27 A28 D29 D30 I50 P81 T82 V84 N25 G27 A28 D29 D30 I50 P81 T82 V84 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 ic50=5.39nM remove_due_to_license_issue Q000H7 23792096 101 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKVIGTVLVGPTPTNVIGRNLMTQIGCTLNF 4l1a B 1.9 BS01 AB1 A 1 R8 N25 A28 D29 P81 R8 N25 A28 D29 P81 N25 T26 G27 N25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q000H7 23792096 101 PQITLWQRPIVTIKIGGQLKEALLNTGADDTVLEEVNLPGRWKPKLIGGIGGFVKVRQYDQVPIEICGHKTIGTVLVGPTPTNVIGRNLMTQIGCTLNF 4l23 A 2.501 BS01 X6K A 1 M772 D810 Y836 I848 E849 V850 V851 I932 D933 M736 D774 Y800 I812 E813 V814 V815 I887 D888 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue Kd=1.5nM, IC50=3.6nM P42336 24900786 1101 GELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSGETSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREANRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTTKMDWIF 4l2f A 2.05 BS01 1V3 A 1 H1031 G1032 S1033 Y1050 Y1060 F1061 S1068 Y1071 I1075 H80 G81 S82 Y99 Y109 F110 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l2g A 2.05 BS02 1V4 A 1 H1031 G1032 Y1050 Y1060 F1061 A1062 K1067 S1068 Y1071 H80 G81 Y99 Y109 F110 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1205 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l2k A 2.1 BS01 1V8 A 1 H1031 G1032 Y1050 Y1060 F1061 A1062 S1068 Y1071 H80 G81 Y99 Y109 F110 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l2l A 1.648 BS02 1V6 A 1 Q136 A137 Y267 W311 F314 F362 K364 L365 V367 P374 A377 Y378 P382 Q133 A134 Y264 W308 F311 F359 K361 L362 V364 P371 A374 Y375 P379 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 Ki=2.3uM remove_due_to_license_issue IC50=12400nM, Kd=130nM, Ki=360nM P09960 24591641 702 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 4l2x F 2.55 BS01 YL2 F 1 F99 D103 R112 T167 Q171 K200 T201 D243 K257 F92 D96 R105 T160 Q164 K193 T194 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=115nM P14324 23998921 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4l31 A 2.0 BS01 F08 A 1 H1031 G1032 A1049 Y1050 Y1060 F1061 A1062 S1068 Y1071 I1075 H80 G81 A98 Y99 Y109 F110 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l32 A 1.85 BS02 1VF A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l33 A 2.1 BS02 F70 A 1 H1031 G1032 A1049 Y1050 I1051 Y1060 A1062 S1068 Y1071 I1075 H80 G81 A98 Y99 I100 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l34 A 1.8 BS02 1VG A 1 H1031 G1032 Y1050 Y1060 S1068 Y1071 H80 G81 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 24116873 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4l3p A 2.68 BS01 1UH A 1 V42 G45 V50 A61 M104 Y106 A107 E108 G110 L163 C174 V17 G20 V25 A36 M79 Y81 A82 E83 G85 L138 C149 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 23850198 601 GSLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHGE 4l4l A 2.122 BS01 1XC A 1 H191 F193 R196 D219 V242 A244 S275 I309 R311 D313 I351 G353 G383 G384 H175 F177 R180 D203 V226 A228 S259 I293 R295 D297 I335 G337 G367 G368 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4l4l B 2.122 BS01 1XC A 1 Y18 R392 Y11 R376 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEAA 4l4l B 2.122 BS02 1XC B 1 Y188 H191 F193 R196 D219 S241 V242 A244 S275 R311 D313 G353 G383 G384 Y172 H175 F177 R180 D203 S225 V226 A228 S259 R295 D297 G337 G367 G368 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEAA 4l4m A 2.445 BS01 1XD A 1 H191 F193 R196 D219 V242 S275 I309 R311 I351 H175 F177 R180 D203 V226 S259 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.01uM remove_due_to_license_issue IC50=10nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4l4m B 2.445 BS01 1XD B 1 H191 F193 R196 D219 V242 S275 I309 R311 I351 H175 F177 R180 D203 V226 S259 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.01uM remove_due_to_license_issue IC50=10nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4l4v A 1.9 BS01 1VY A 1 Y7 R9 S24 K43 Y62 W69 R94 I96 Q153 W156 Y7 R9 S23 K42 Y61 W68 R93 I95 Q152 W155 ? Kd=1.65uM remove_due_to_license_issue Q95460 23846752 301 RTHSLRYFRLGVSDPIGVPEFISVGYVDSHPITTYDSVTRQKEPRAPWMAENLAPDHWERYTQLLRGWQQMFKVELKRLQRHYNHSGSHTYQRMIGCELLEDGSTTGFLQYAYDGQDFLIFNKDTLSWLAVDNVAHTIKQAWEANQHELLYQKNWLEEECIAWLKRFLEYGKDTLQRTEPPLVRVNRKETFPGVTALFCKAHGFYPPEIYMTWMKNGEEIVQEIDYGDILPSGDGTYQAWASIELLYSCHVEHSGVHMVLQV 4l4z A 2.3 BS01 D5X A 1 E126 A127 I210 G211 T220 D243 L245 E58 A59 I142 G143 T152 D175 L177 ? 0030246 Kd=2.1uM remove_due_to_license_issue P76141 24047255 501 EGCLEYETQLRRQFSLQHVRVIPGLADADVGGRLGIGAAHMLMSLLQPQQMLAIGFGEATMNTLQRLSGFISSQQIRLVTLSGGVGSYMTGIGQLNAACSVNIIPAPLRASSADIARTLKNENCVKDVLLAAQAADVAIVGIGAVSQQDDATIIRSGYISQGEQLMIGRKGAVGDILGYFFDAKGDVVTNIKIHNELIGLPLSALKTIPVRVGVAGGENKAEAIAAAMKGGYINALVTDQDTAAAILRS 4l50 A 2.1 BS01 D8X A 1 F124 G125 E126 A127 G211 T220 D243 L245 K288 F55 G56 E57 A58 G142 T151 D174 L176 K219 ? 0030246 Kd=0.88uM remove_due_to_license_issue P76141 24047255 501 FEGCLEYETQLRRQFSLQHVRVIPGLADVGGRLGIGAAHMLMSLLQPQQMLAIGFGEATMNTLQRLSGFISSQQIRLVTLSGGVGSYMTGIGQLNAACSVNIIPAPLRASSADIARTLKNENCVKDVLLAAQAADVAIVGIGAVSQQDDATIIRSGYISQGEQLMIGRKGAVGDILGYFFDAKGDVVTNIKIHNELIGLPLSALKTIPVRVGVAGGENKAEAIAAAMKGGYINALVTDQDTAAAILRS 4l51 A 1.9 BS01 HSX A 1 G125 E126 A127 G209 I210 G211 T220 D243 L245 K288 G54 E55 A56 G138 I139 G140 T149 D172 L174 K217 ? 0030246 Kd=995uM remove_due_to_license_issue P76141 24047255 501 EGCLEYETQLRRQFSLQHVRVIPGLDVGGRLGIGAAHMLMSLLQPQQMLAIGFGEATMNTLQRLSGFISSQQIRLVTLSGGVGSYMTGIGQLNAACSVNIIPAPLRASSADIARTLKNENCVKDVLLAAQAADVAIVGIGAVSQQDDATIIRSGYISQGEQLMIGRKGAVGDILGYFFDAKGDVVTNIKIHNELIGLPLSALKTIPVRVGVAGGENKAEAIAAAMKGGYINALVTDQDTAAAILRS 4l52 A 2.54 BS01 1UL A 1 V42 V50 A61 M104 E105 Y106 A107 E108 G110 L163 C174 V17 V25 A36 M79 E80 Y81 A82 E83 G85 L138 C149 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 23850198 501 GSLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 4l53 A 2.55 BS01 1UO A 1 V42 V50 A61 M104 Y106 A107 G110 L163 C174 D175 V17 V25 A36 M79 Y81 A82 G85 L138 C149 D150 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 23856049 501 GSLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTKGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 4l5j A 2.6 BS01 HSX A 1 F124 G125 E126 A127 G209 T220 D243 L245 K288 F115 G116 E117 A118 G200 T211 D234 L236 K279 ? 0000987,0003677,0005737,0005829,0006351,0009408,0030246,0042802,2000142 remove_due_to_license_issue P76141 24047255 501 EQGMCEEEQVARIAWFYYHDGLTQSEISDRLGLTRLKVSRLLEKGHQSGIIRVQINSRFEGCLEYETQLRRQFSLQHVRVIPGLADADVGGRLGIGAAHMLMSLLQPQQMLAIGFGEATMNTLQRLSGFISSQQIRLVTLSGGVGSYMTGIGQLNAACSVNIIPAPLRASSADIARTLKNENCVKDVLLAAQAADVAIVGIGAVSQQDDATIIRSGYISQGEQLMIGRKGAVGDILGYFFDAKGDVVTNIKIHNELIGLPLSALKTIPVRVGVAGGENKAEAIAAAMKGGYINALVTDQDTAAAILRS 4l5r C 1.873 BS01 dna A 0 S166 G167 H222 R224 G226 N227 G235 N236 S121 G122 H177 R179 G181 N182 G190 N191 ? 0002218,0035458 remove_due_to_license_issue Q9R002 23850291 1 ~ 20 TPKKNISKGAVLHEKPMTVMVLTATEPFNYKEGKENMFHATVATESKYYRVKVFNMDLKEKFTENQFITISKYFNSSGILEINETATVSEAAPNQMFEVPKNIIRSAKETLKISKIKELDSGTLIYGVFAVEKKKVNDKSITFKIKDNEDNIKVVWDKEQHNINYEKGDKLQLFSFHLRKGNGKPILHSGNHSFIKGE 4l5r C 1.873 BS02 dna B 0 K48 K53 K180 N182 D183 K184 S185 T187 K198 K3 K8 K135 N137 D138 K139 S140 T142 K153 ? 0002218,0035458 remove_due_to_license_issue Q9R002 23850291 1 ~ 20 TPKKNISKGAVLHEKPMTVMVLTATEPFNYKEGKENMFHATVATESKYYRVKVFNMDLKEKFTENQFITISKYFNSSGILEINETATVSEAAPNQMFEVPKNIIRSAKETLKISKIKELDSGTLIYGVFAVEKKKVNDKSITFKIKDNEDNIKVVWDKEQHNINYEKGDKLQLFSFHLRKGNGKPILHSGNHSFIKGE 4l6q A 2.79 BS01 1WU A 1 I98 A119 K121 M169 E170 Y171 M172 N219 L221 D232 I72 A93 K95 M143 E144 Y145 M146 N193 L195 D206 D214 K216 N219 D232 T253 D188 K190 N193 D206 T227 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O75116 24049062 501 QRKLEALIRDPRSPINVESLLDGLNSLVLDLDFPALRKNKNIDNFLNRYEKIVKKIRGLQMKAEDYDVVKVIGRGAFGEVQLVRHKASQKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWAKFYTAEVVLALDAIHSMGLIHRDVKPDNMLLDKHGHLKLADFGTCMKMDETGMVHCDTAVGTPDYISPEVLKSQGGDGFYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMDHKNSLCFPEDAEISKHAKNLICAFLTDREVRLGRNGVEEIRQHPFFKNDQWHWDNIRETAAPVVPELSSDIDSSNFDDIEDDVETFPIPKAFVGNQLPFIGFTYYR 4l6s A 2.2 BS01 1WQ A 1 D766 L769 D770 H862 G863 R878 A880 Y896 S904 Y907 D106 L109 D110 H202 G203 R218 A220 Y236 S244 Y247 S904 Y907 E988 S244 Y247 E328 2.4.2.-,2.4.2.30 0003950 Kd=0.003uM remove_due_to_license_issue Kd=3.0nM P09874 23850199 1100 HMKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 4l6t B 1.859 BS01 GAL G 1 E73 Q83 W110 N112 K113 E52 Q62 W89 N91 K92 ? 0005576 remove_due_to_license_issue Q8GAV3 24095060 4 MTPQNITDLCNEYQNTMIYSLNKEIATYTESLAGKREMVIISFSNGATFQVEVPGSQHLESQKRPLERMKDTLRAAYFTGIKISKLCAWTNKSPNSIAAIELSNL 4l6t B 1.859 BS02 SIA G 1 E33 Y34 Q35 L80 E12 Y13 Q14 L59 ? 0005576 remove_due_to_license_issue Q8GAV3 24095060 5 MTPQNITDLCNEYQNTMIYSLNKEIATYTESLAGKREMVIISFSNGATFQVEVPGSQHLESQKRPLERMKDTLRAAYFTGIKISKLCAWTNKSPNSIAAIELSNL 4l6t C 1.859 BS01 GAL H 1 E73 Q78 Q83 W110 N112 K113 E52 Q57 Q62 W89 N91 K92 ? 0005576 remove_due_to_license_issue Q8GAV3 24095060 4 MTPQNITDLCNEYQNTMIYSLNKEIATYTESLAGKREMVIISFSNGATFQVEVPGSQHLESQKRPLERMKDTLRAAYFTGIKISKLCAWTNKSPNSIAAIELSNL 4l6t C 1.859 BS02 SIA H 1 E33 Y34 Q35 L80 E12 Y13 Q14 L59 ? 0005576 remove_due_to_license_issue Q8GAV3 24095060 5 MTPQNITDLCNEYQNTMIYSLNKEIATYTESLAGKREMVIISFSNGATFQVEVPGSQHLESQKRPLERMKDTLRAAYFTGIKISKLCAWTNKSPNSIAAIELSNL 4l70 A 2.0 BS01 1V9 A 1 H384 G385 T386 Y414 S422 Y425 E514 H206 G207 T208 Y236 S244 Y247 E336 S422 Y425 E514 S244 Y247 E336 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 24188023 601 SMKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 4l7b B 2.41 BS01 1VV B 1 Y334 N414 R415 A556 Y572 F577 Y14 N94 R95 A236 Y252 F257 ? ic50=2.3uM remove_due_to_license_issue Kd=1900nM, IC50=792nM, Ki=560nM, EC50=26000nM Q14145 24504667 701 APKVGRLIYTAGGYFRQSLSYLEAYNPSDGTWLDLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVTLEH 4l7c A 2.4 BS01 1VW A 1 Y334 N382 R415 A556 Y572 S602 Y9 N57 R90 A231 Y247 S277 ? ic50=7.4uM remove_due_to_license_issue Q14145 24504667 701 RLIYTAGGYFRQSLSYLEAYNPSDGTWLDLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVTLE 4l7d A 2.25 BS01 1VX A 1 Y334 N414 R415 G509 A556 Y572 F577 S602 Y9 N89 R90 G184 A231 Y247 F252 S277 ? ic50=0.75uM remove_due_to_license_issue IC50=750nM Q14145 24504667 701 RLIYTAGGYFRQSLSYLEAYNPSDGTWLDLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVTLE 4l7f A 1.95 BS01 1V5 A 1 I32 Q37 G38 V40 A53 K55 L57 M111 A113 N114 Q117 V158 L168 I28 Q33 G34 V36 A49 K51 L53 M107 A109 N110 Q113 V154 L164 D151 K153 N156 D169 T188 D147 K149 N152 D165 T171 2.7.11.24 0004672,0004707,0005524,0006468 ic50=160nM remove_due_to_license_issue P45983 23916259 401 SLDNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDWRKGIITIT 4l7g A 1.38 BS01 1W0 A 1 G11 Q12 G13 D32 Y71 F108 W115 D228 G230 G13 Q14 G15 D34 Y73 F110 W117 D223 G225 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTDCGYNI 4l7h A 1.85 BS01 1W1 A 1 D32 G34 S35 Y71 W115 I118 D228 G230 D34 G36 S37 Y73 W117 I120 D223 G225 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4l7j A 1.651 BS01 1W2 A 1 D32 S35 Y71 F108 W115 D228 D34 S37 Y73 F110 W117 D223 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4l7l A 2.1 BS01 1VA A 1 D284 H384 G385 Y414 F415 S422 Y425 E514 D105 H205 G206 Y235 F236 S243 Y246 E335 S422 Y425 E514 S243 Y246 E335 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 24188023 601 MKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 4l7n A 1.8 BS01 1VB A 1 D284 L287 D291 H384 G385 R400 M402 Y414 S422 Y425 E514 D105 L108 D112 H205 G206 R221 M223 Y235 S243 Y246 E335 S422 Y425 E514 S243 Y246 E335 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 24188023 601 MKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 4l7o A 2.0 BS01 1VD A 1 D284 L287 D291 H384 G385 R400 M402 Y414 S422 Y425 E514 D106 L109 D113 H206 G207 R222 M224 Y236 S244 Y247 E336 S422 Y425 E514 S244 Y247 E336 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 24188023 601 SMKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 4l7r A 2.2 BS01 M00 A 1 D284 H384 G385 Y414 F415 S422 Y425 E514 D105 H205 G206 Y235 F236 S243 Y246 E335 S422 Y425 E514 S243 Y246 E335 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 24188023 601 MKRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 4l7u A 2.8 BS01 1VC A 1 V288 H384 G385 T386 N387 V390 Y414 K421 S422 Y425 E514 V108 H204 G205 T206 N207 V210 Y234 K241 S242 Y245 E334 S422 Y425 E514 S242 Y245 E334 2.4.2.- 0003950 remove_due_to_license_issue Q9Y6F1 24188023 601 KRVQPCSLDPATQKLITNIFSKEMFKNTMALMDLDVKKMPLGKLSKQQIARGFEALEALEEALKDGGQSLEELSSHFYTVIPHNFGHSQPPPINSPELLQAKKDMLLVLADIELAQALQAVSEQEKTVEEVPHPLDRDYQLLKCQLQLLDSGAPEYKVIQTYLEQTGSNHRCPTLQHIWKVNQEGEEDRFQAHSKLGNRKLLWHGTNMAVVAAILTSGLRIMPHSGGRVGKGIYFASENSKSAGYVIGMKCGAHHVGYMFLGEVALGREHHINTDNPSLKSPPPGFDSVIARGHTEPDPTQDTELELDGQQVVVPQGQPVPCPEFSSSTFSQSEYLIYQESQCRLRYLLEVH 4l8m A 2.1 BS01 F46 A 1 A51 K53 E71 L74 L75 L104 T106 L108 M109 G110 A111 D112 L167 D168 F169 L171 A47 K49 E67 L70 L71 L100 T102 L104 M105 G106 A107 D108 L161 D162 F163 L165 D150 K152 N155 D168 T185 D144 K146 N149 D162 T172 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.001uM remove_due_to_license_issue IC50=1.000000nM, Kd=17nM Q16539 24131218 403 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4l9i A 2.32 BS01 8PR A 1 R195 V201 A214 T265 M267 D271 E318 L321 R166 V172 A185 T236 M238 D242 E289 L292 D314 K316 E318 N319 D332 A341 T352 D285 K287 E289 N290 D303 A312 T323 2.7.11.14 0001750,0004672,0004674,0004703,0005515,0005524,0005737,0006468,0007165,0007601,0009966,0016020,0022400,0042995,0046777,0050254,0097381 Kd=13uM remove_due_to_license_issue IC50=398100nM P28327 24220010 601 SRDRKYLARLKLPPLSKCEALRESLDLGFEGMCLEQPIGKRLFQQFLRTHEQHGPALQLWKDIEDYDTADDALRPQKAQALRAAYLEPQAQLFCSFLDAETVARARAGAGDGLFQPLLRAVLAHLGQAPFQEFLDSLYFLRFLQWKWLEAQPMGEDWFLDFRVLGRGGFGEVFACQMKATGKLYACKKLNKKRLKKRKGYQGAMVEKKILAKVHSRFIVSLAYAFETKTDLCLVMTIMNGGDIRYHIYNVDEDNPGFQEPRAIFYTAQIVSGLEHLHQRNIIYRDLKPENVLLDDDGNVRISDLGLAVELKAGQTKTKGYAGTPGFMAPELLLGEEYDFSVDYFALGVTLYEMIAARGPFRARGEKVENKELKQRVLEQAVTYPDKFSPASKDFCEALLQKDPEKRLGFRDGSCDGLRTHPLFRDISWRQLEAGMLTPPFVPDSRTVYAKNIQDVGAFSTVKGVAFEKADTEFFQEFASGTCPIPWQEEMIETGVFGDLNVWRP 4la7 A 1.98 BS01 A1O A 1 P60 K64 V85 S96 E98 F112 L121 Y124 F165 P50 K54 V75 S86 E88 F102 L111 Y114 F155 ? 0004864,0005515,0005634,0005737,0005886,0009738,0010427,0038023,0042802,0042803,0062049 ic50=267nM remove_due_to_license_issue O80992 23818638 201 TDEEQKTLEPVIKTYHQFEPDPTTCTSLITQRIHAPASVVWPLIRRFDNPERYKHFVKRCRLISGDGDVGSVREVTVISGLPASTSTERLEFVDDDHRVLSFRVVGGEHRLKNYKSVTSVNEFLNQDSGKVYTVVLESYTVDIPEGNTEEDTKMFVDTVVKLNLQKLGVAATSAPM 4lar H 2.38 BS01 1WE H 1 Y33 F98 E106 H213 W215 F220 Y33 F98 E106 H213 W215 F220 remove_due_to_license_issue 24349338 300 EVQLQESGPSLVKPSQTLSLTCSVTGDSVTSGYWSWIRQFPGNKLDYMGYISYRGSTYYNPSLKSRISITRDTSKNQVYLQLKSVSSEDTATYYCSYFDSDDYAMEYWGQGTSVTVSSGGGGSQIVLTQSPAIMSASPGEKVTLTCSASSSVSSSHLYWYQQKPGSSPKLWIYSTSNLASGVPARFSGSGSGTSYSLTISSMEAEDAASYFCHQWSSFPFTFGSGTKLEIKR 4lbl A 1.58 BS01 BGC B 1 R162 E184 R50 E72 ? 0030246 remove_due_to_license_issue P17931 24326249 1 MLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTLLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 4lbl A 1.58 BS02 GAL B 1 H158 R162 N174 W181 E184 H46 R50 N62 W69 E72 ? 0030246 remove_due_to_license_issue P17931 24326249 2 MLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTLLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 4lbo A 1.65 BS01 BGC B 1 R162 E184 R186 R50 E72 R74 ? 0030246 remove_due_to_license_issue P17931 24326249 1 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 4lbo A 1.65 BS02 GAL B 1 H158 R162 N174 W181 E184 H46 R50 N62 W69 E72 ? 0030246 remove_due_to_license_issue P17931 24326249 2 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 4lbp A 1.87 BS01 1WG A 1 Y21 H24 P40 S56 Y21 H24 P40 S56 ? Kd=11.4uM remove_due_to_license_issue Q45075 23955343 201 MLFLIYRKDRPGSLQVRIDNYAAHLAYLEPLKAKIQVGGPTLGAGTGTDDKDMTGSFLIMEAESWDEVHSFVENDPFTKAGLFAATIVERWKHGKHND 4lbu A 1.17 BS01 1WJ A 1 T47 L68 G69 N70 D102 Y106 Q107 D156 C158 G229 A232 M260 G261 D280 T38 L59 G60 N61 D93 Y97 Q98 D142 C144 G215 A218 M246 G247 D266 D102 D280 C318 C320 C323 H349 D93 D266 C304 C306 C309 H335 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=276nM remove_due_to_license_issue P28720 25483606 401 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4lc7 A 1.7 BS01 1WP A 1 Q73 G74 D93 Y132 F169 I171 W176 D289 G291 T292 Q16 G17 D36 Y75 F112 I114 W119 D232 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4lch A 1.596 BS03 1WN A 1 L18 M62 E77 T190 F191 I197 G209 S210 H237 D241 H264 L18 M62 E77 T190 F191 I197 G209 S210 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue P47205 23914798 304 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISY 4lck A 3.2 BS01 rna C 0 I14 G15 T16 K17 Q18 M62 V73 A75 A76 I13 G14 T15 K16 Q17 M61 V72 A74 A75 ? 0003723,0005737,0005840,1990904 remove_due_to_license_issue P46350 23892783 1 ~ 102 SYDKVSQAKSIIIGTKQTVKALKRGSVKEVVVAKDADPILTSSVVSLAEDQGISVSMVESMKKLGKACGIEVGAAAVAIIL 4lck D 3.2 BS01 rna F 0 I14 G15 Q18 M62 V73 G74 A75 A76 I13 G14 Q17 M61 V72 G73 A74 A75 ? 0003723,0005737,0005840,1990904 remove_due_to_license_issue P46350 23892783 1 ~ 102 SYDKVSQAKSIIIGTKQTVKALKRGSVKEVVVAKDADPILTSSVVSLAEDQGISVSMVESMKKLGKACGIEVGAAAVAIIL 4led A 2.37 BS01 XXR A 1 Q148 D150 N152 Y156 Q147 D149 N151 Y155 ? remove_due_to_license_issue T2LG16 24516380 301 ASSLAPRQVIRDGQFITSPNGKYKLVMQADGNLVLYEDGTKPIWNTTPVGPGAKAVMEFNLNLYNKAGQVAWSSNVYTAYLFEEFKDEAYLNLQDDGDFGIFSDEAKWGSIVLSRPEVGVKNKIIPTGTVMVPGTEYINGNYRLAFQGDGNLVIYQINPQVVIWATYTMGADRAVVQEDGNFVIYKGTTALWHTHTATGMPAYLKFTNTGKLFLSQPTLLWTLKRGSLSKPPKVIPGQHGPLDTTPIWSWPHDY 4led A 2.37 BS02 XXR A 2 Q178 D180 N182 Y186 Q177 D179 N181 Y185 ? remove_due_to_license_issue T2LG16 24516380 302 ASSLAPRQVIRDGQFITSPNGKYKLVMQADGNLVLYEDGTKPIWNTTPVGPGAKAVMEFNLNLYNKAGQVAWSSNVYTAYLFEEFKDEAYLNLQDDGDFGIFSDEAKWGSIVLSRPEVGVKNKIIPTGTVMVPGTEYINGNYRLAFQGDGNLVIYQINPQVVIWATYTMGADRAVVQEDGNFVIYKGTTALWHTHTATGMPAYLKFTNTGKLFLSQPTLLWTLKRGSLSKPPKVIPGQHGPLDTTPIWSWPHDY 4led A 2.37 BS03 XXR A 3 G149 D150 G148 D149 ? remove_due_to_license_issue T2LG16 24516380 303 ASSLAPRQVIRDGQFITSPNGKYKLVMQADGNLVLYEDGTKPIWNTTPVGPGAKAVMEFNLNLYNKAGQVAWSSNVYTAYLFEEFKDEAYLNLQDDGDFGIFSDEAKWGSIVLSRPEVGVKNKIIPTGTVMVPGTEYINGNYRLAFQGDGNLVIYQINPQVVIWATYTMGADRAVVQEDGNFVIYKGTTALWHTHTATGMPAYLKFTNTGKLFLSQPTLLWTLKRGSLSKPPKVIPGQHGPLDTTPIWSWPHDY 4len A 1.5 BS01 2GK A 1 C69 S70 N104 Y105 S130 N132 E166 N170 T235 G236 S237 C44 S45 N79 Y80 S105 N107 E141 N145 T210 G211 S212 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9L5C8 24882105 300 QTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTAGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 4leq A 1.405 BS01 1WK A 1 T47 L68 N70 D102 Y106 Q107 D156 C158 G229 L231 A232 M260 G261 D280 T38 L59 N61 D93 Y97 Q98 D146 C148 G219 L221 A222 M250 G251 D270 D102 D280 C318 C320 C323 H349 D93 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=288nM remove_due_to_license_issue P28720 25483606 401 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4lg2 A 2.7 BS01 rna F 0 I267 Q268 K271 R311 I60 Q61 K64 R104 ? remove_due_to_license_issue Q8JPY0 23824825 4 ~ 12 ISAKDLKEIMYDHLPGFGTAFHQLVQVICKIGKDNNLLDTIHAEFQASLADGDSPQCALIQITKRVPIFQDVPPPIIHIRSRGDIPRACQKSLRPAPPSPKIDRGWVCLFKMQDGKTLGLKI 4lg2 D 2.7 BS01 rna J 0 C264 I267 Q268 K271 R311 C57 I60 Q61 K64 R104 ? remove_due_to_license_issue Q8JPY0 23824825 1 ~ 12 ISAKDLKEIMYDHLPGFGTAFHQLVQVICKIGKDNNLLDTIHAEFQASLADGDSPQCALIQITKRVPIFQDVPPPIIHIRSRGDIPRACQKSLRPAPPSPKIDRGWVCLFKMQDGKTLGLKI 4lg2 D 2.7 BS02 rna I 0 F228 Q263 F21 Q56 ? remove_due_to_license_issue Q8JPY0 23824825 1 ~ 12 ISAKDLKEIMYDHLPGFGTAFHQLVQVICKIGKDNNLLDTIHAEFQASLADGDSPQCALIQITKRVPIFQDVPPPIIHIRSRGDIPRACQKSLRPAPPSPKIDRGWVCLFKMQDGKTLGLKI 4lge A 1.55 BS02 1Y0 A 1 D297 G306 L307 R308 C309 W310 E311 D314 E319 W323 D43 G52 L53 R54 C55 W56 E57 D60 E65 W69 2.3.2.27 ic50=3.5nM remove_due_to_license_issue Q13490 23928071 402 ISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRY 4lgg A 2.41 BS01 VGG A 1 L273 V281 A293 K295 M341 L393 L10 V16 A28 K30 M68 L120 D386 R388 A390 N391 D404 D113 R115 A117 N118 D131 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3nM remove_due_to_license_issue P00523 23841803 601 RESLRLEVKLGQGGEVWMGTWNGTTRVAIKTLKPGLQEAQVMKKLRHEKLVQLYAVVSEEIYIVGEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4lgh A 2.84 BS01 0JN A 1 L273 A293 K295 M314 I336 G338 Y340 M341 L393 L17 A34 K36 M43 I65 G67 Y69 M70 L122 D386 R388 A390 N391 D404 D115 R117 A119 N120 D133 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=620nM P00523 23841803 601 KDAWEIPRESLRLEVKLGQGGEVWMGTWNGTRVAIKTLEAQVMKKLRHEKLVQLYAVVSEEPIYIVGEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4lgu A 2.0 BS02 1YH A 1 D297 G306 L307 R308 C309 E311 D314 E319 W323 D41 G50 L51 R52 C53 E55 D58 E63 W67 2.3.2.27 ic50=2.1nM remove_due_to_license_issue Q13490 23928071 402 NLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRY 4lh3 A 1.813 BS01 GUA A 1 F212 K347 C348 S349 G512 S513 F520 F182 K317 C318 S319 G482 S483 F490 N211 K233 E314 C348 E447 P532 N181 K203 E284 C318 E417 P502 1.2.1.88 0003842,0004029,0005739,0005759,0005829,0006560,0010133,0016491,0016620,0042802 Ki=30mM remove_due_to_license_issue Q8CHT0 23928095 602 KVANEPILAFSQGSPERDALQKALKDLKGQTEAIPCVVGDEEVWTSDIQYQLSPFNHAHKVAKFCYADKALLNRAIDAALAARKEWDLKPMADRAQVFLKAADMLSGPRRAEVLAKTMVGQGKTVIQAEIDAAAELIDFFRFNAKFAVELEGEQPISVPPSTNHTVYRGLEGFVAAISPFNFTAIGGNLAGAPALMGNVVLWKPSDTAMLASYAVYRILREAGLPPNIIQFVPADGPTFGDTVTSSEHLCGINFTGSVPTFKHLWRQVAQNLDRFRTFPRLAGECGGKNFHFVHSSADVDSVVSGTLRSAFEYGGQKCSACSRLYVPKSLWPQIKGRLLEEHSRIKVGDPAEDFGTFFSAVIDAKAFARIKKWLEHARSSPSLSILAGGQCNESVGYYVEPCIIESKDPQEPIMKEEIFGPVLTVYVYPDDKYRETLKLVDSTTSYGLTGAVFAQDKAIVQEATRMLRNAAGNFYINDKSTGSVVGQQPFGGARASGTNDKPGGPHYILRWTSPQVIKETHKPLGDWRYSYMQ 4lh5 A 2.19 BS01 LF0 A 1 A169 E170 H171 T174 M178 A97 E98 H99 T102 M106 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=0.23uM remove_due_to_license_issue P12497 24261564 301 SPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKYSAGERIVDIIATDI 4lh6 A 1.65 BS01 1X7 A 1 E118 L119 K120 I121 E175 Y227 V289 K291 E117 L118 K119 I120 E174 Y226 V288 K290 E118 K120 D122 Y227 K315 E117 K119 D121 Y226 K314 6.5.1.2 0003911 ic50=77uM remove_due_to_license_issue Q837V6 24287382 401 EQQPLTLTAATTRAQELRKQLNQYSHEYYVKDQPSVEDYVYDRLYKELVDIETEFPDLITPDSPTQRVGGKVLSGFEKAPHDIPMYSLNDGFSKEDIFAFDERVRKAIGKPVAYCCELKIDGLAISLRYENGVFVRGATRGDGTVGENITENLRTVRSVPMRLTEPISVEVRGECYMPKQSFVALNEEREENGQDIFANPRNAAAGSLRQLDTKIVAKRNLNTFLYTVADFGPMKAKTQFEALEELSAIGFRTNPERQLCQSIDEVWAYIEEYHEKRSTLPYEIDGIVIKVNEFALQDELGFTVKAPRWAIAYKFPPEEAET 4lh7 A 1.9 BS01 1X8 A 1 Y87 L89 E118 K120 I121 E175 Y227 K291 Y86 L88 E117 K119 I120 E174 Y226 K290 E118 K120 D122 Y227 K315 E117 K119 D121 Y226 K314 6.5.1.2 0003911 ic50=34uM remove_due_to_license_issue Q837V6 24287382 401 EQQPLTLTAATTRAQELRKQLNQYSHEYYVKDQPSVEDYVYDRLYKELVDIETEFPDLITPDSPTQRVGGKVLSGFEKAPHDIPMYSLNDGFSKEDIFAFDERVRKAIGKPVAYCCELKIDGLAISLRYENGVFVRGATRGDGTVGENITENLRTVRSVPMRLTEPISVEVRGECYMPKQSFVALNEEREENGQDIFANPRNAAAGSLRQLDTKIVAKRNLNTFLYTVADFGPMKAKTQFEALEELSAIGFRTNPERQLCQSIDEVWAYIEEYHEKRSTLPYEIDGIVIKVNEFALQDELGFTVKAPRWAIAYKFPPEEAE 4lhm A 1.52 BS06 AZZ A 1 T87 Y168 R171 V177 S186 K190 F210 T87 Y168 R171 V177 S186 K190 F210 D83 K84 H85 S86 T123 D164 R171 S186 K190 K191 D83 K84 H85 S86 T123 D164 R171 S186 K190 K191 2.4.2.4 0004645,0005829,0006206,0006213,0006974,0009032,0016020,0016154,0016757,0016763,0046104 Ki=0.68mM remove_due_to_license_issue P07650 24699659 510 LFLAQEIIRKKRDGHALSDEEIRFFINGIRDNTISEGQIAALAMTIFFHDMTMPERVSLTMAMRDSGTVLDWKSLHLNGPIVDKHSTGGVGDVTSLMLGPMVAACGGYIPMISGRGLGHTGGTLDKLESIPGFDIFPDDNRFREIIKDVGVAIIGQTSSLAPADKRFYATRDITATVDSIPLITASILAKKLAEGLDALVMDVKVGSGAFMPTYELSEALAEAIVGVANGAGVRTTALLTDMNQVLASSAGNAVEVREAVQFLTGEYRNPRLFDVTMALCVEMLISGKLAKDDAEARAKLQAVLDNGKAAEVFGRMVAAQKGPTDFVENYAKYLPTAMLTKAVYADTEGFVSEMDTRALGMAVVAMGGGRRQASDTIDYSVGFTDMARLGDQVDGQRPLAVIHAKDENNWQEAAKAVKAAIKLADKAPESTPTVYRRISE 4lhv A 1.95 BS01 GDP A 1 G18 V19 G20 K21 T22 C23 F33 N34 N121 K122 D124 S151 A152 K153 G16 V17 G18 K19 T20 C21 F31 N32 N110 K111 D113 S140 A141 K142 3.6.5.2 0003924,0005525 remove_due_to_license_issue P61006 24072714 201 GSHDYLFKLLLIGDSGVGKTCVLFRFSEDAFNSTFISTIGIDFKIRTIELDGKRIKLQIWDTTTAYYRGAMGIMLVYDITNEKSFDNIRNWIRNIEEHASADVEKMILGNKCDVNDKRQVSKERGEKLALDYGIKFMETSAKANINVENAFFTLARDIKAKMDKK 4li0 A 3.3 BS01 GDP A 1 G18 G20 K21 T22 C23 K122 D124 S151 A152 K153 G13 G15 K16 T17 C18 K117 D119 S146 A147 K148 Q67 Q62 3.6.5.2 0003924,0005525 remove_due_to_license_issue P61006 24072714 200 DYLFKLLLIGDSGVGKTCVLFRFSEDAFNSTFISTIGIDFKIRTIELDGKRIKLQIWDTAGQERFRTITTAYYRGAMGIMLVYDITNEKSFDNIRNWIRNIEEHASADVEKMILGNKCDVNDKRQVSKERGEKLALDYGIKFMETSAKANINVENAFFTLARDIKAKMDKK 4li5 A 2.64 BS01 1WY A 1 L718 G719 F723 V726 A743 M793 G796 C797 D800 L844 L26 G27 F31 V34 A51 M101 G104 C105 D108 L152 D837 A839 R841 N842 D855 G874 D145 A147 R149 N150 D163 G182 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 23930994 1101 GSMGEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDEDDVVDADEYLIPQ 4li6 A 2.05 BS02 1XO A 1 H1184 G1185 P1187 F1188 Y1203 Y1213 A1215 K1220 S1221 Y1224 I1228 H80 G81 P83 F84 Y99 Y109 A111 K116 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 23844574 1406 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPYAEYVIYRGEQAYPEYLITYQIMKPE 4li7 A 2.2 BS01 1XP A 1 H1184 G1185 F1188 A1191 K1195 G1196 F1197 D1198 H1201 Y1213 S1221 Y1224 I1228 H80 G81 F84 A87 K91 G92 F93 D94 H97 Y106 S114 Y117 I121 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 23844574 1405 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKPEA 4li8 A 2.521 BS02 1XQ A 1 H1184 G1185 F1188 A1191 F1197 D1198 H1201 A1202 G1211 Y1213 F1214 A1215 K1220 S1221 Y1224 I1228 E1291 H80 G81 F84 A87 F93 D94 H97 A98 G104 Y106 F107 A108 K113 S114 Y117 I121 E177 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=15.4nM O95271 23844574 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRYAEYVIYRGEQAYPEYLITYQIMKP 4lil A 2.6 BS03 UTP A 1 S160 R162 R163 H166 K318 S150 R152 R153 H156 K303 2.7.7.102 0000287,0000428,0003896,0005515,0005654,0005658,0006260,0006269,0006270,0008270,0016020,0016779,0032553,0046872 remove_due_to_license_issue P49642 24239947 504 PTELPELLKLYYRRLFPYSQYYRWLNYIKNYFQHREFSFTLKDDIYIRYQSFNNQSDLEKEMQKMNPYKIDIGAVYSHRPNQHNTVKLGAFQAQEKELVFDIDMTDYDDVRRCCSDICPKCWTLMTMAIRIIDRALKEDFGFKHRLWVYSGRRGVHCWVCDESVRKLSSAVRSGIVEYLSLVKKKKVHLSEKIHPFIRKSINIIKKYFEEYALVNQDILENKESWDKILALVPETIHDELQQSFQKSHNSLQRWEHLKKVASRYQNNIKNDKYGPWLEWEIMLQYCFPRLDINVSKGINHLLKSPFSVHPKTGRISVPIDLQKVDQFDPFTVPTISFICRELDATRDYKKTSLAPYVKVFEHFLENLDKS 4lj0 A 2.15 BS01 rna C 0 Y407 N410 C411 A412 Y6 N9 C10 A11 ? remove_due_to_license_issue G0SCL7 24071581 1 ~ 4 EQDCKYWPNCANPLCAFRHPTMPPCRNGGECKVPGCKFTHLKTPCKFRPCTNRSCPFLHEEGQRG 4lj0 A 2.15 BS02 rna D 0 N410 A412 C446 K447 F448 C451 T452 N453 F458 N9 A11 C45 K46 F47 C50 T51 N52 F57 ? remove_due_to_license_issue G0SCL7 24071581 1 ~ 4 EQDCKYWPNCANPLCAFRHPTMPPCRNGGECKVPGCKFTHLKTPCKFRPCTNRSCPFLHEEGQRG 4lj0 A 2.15 BS03 rna E 0 C426 R427 N428 F439 C25 R26 N27 F38 ? remove_due_to_license_issue G0SCL7 24071581 1 ~ 2 EQDCKYWPNCANPLCAFRHPTMPPCRNGGECKVPGCKFTHLKTPCKFRPCTNRSCPFLHEEGQRG 4lj3 A 1.7 BS01 C2E A 1 Q127 L143 V144 R145 P156 N200 D262 K286 G320 E322 G340 Y341 P346 Q24 L40 V41 R42 P53 N97 D159 K183 G217 E219 G237 Y238 P243 3.1.4.52 0071111 Kd<1nM remove_due_to_license_issue P21514 24451384 401 YHHIVTPEAISLALENHEFKPWIQPVFCAQTGVLTGCEVLVRWEHPQTGIIPPDQFIPLAESSGLIVIMTRQLMKQTADILMPVKHLLPDNFHIGINVSAGCFLAAGFEKECLNLVNKLGNDKIKLVLELTERNPIPVTPEARAIFDSLHQHNITFALDDFGTGYATYRYLQAFPVDFIKIDKSFVQMASVDEISGHIVDNIVELARKPGLSIVAEGVETQEQADLMIGKGVHFLQGYLYSPPVPGNKFISEWVMK 4lj5 A 2.4 BS01 ADP A 1 R559 V561 T597 G598 V599 G600 K601 T602 I765 Q769 A805 R37 V39 T75 G76 V77 G78 K79 T80 I236 Q240 A276 ? 0005524,0016887 remove_due_to_license_issue Q9RA63 24531492 901 MEVTEEDIAEIVSRWTGIPVSKLLEKLLRLEEELHKRVVGQDEAIRAVADAIRRARAGLKDPNRPIGSFLFLGPTGVGKTELAKTLAATLFDTEEAMIRIDMTEYMEKHAVSRLIGAPPGGQLTEAVRRRPYSVILFDEIEKAHPDVFNILLQILDDGRLTDSHGRTVDFRNTVIILTSNLGSPLILEGLQKGWPYERIRDEVFKVLQQHFRPEFLNRLDEIVVFRPLTKEQIRQIVEIQLSYLRARLAEKRISLELTEAAKDFLAERGYDPVFGARPLRRVIQRELETPLAQKILAGEVKEGDRVQVDVGPAGLVFAVP 4lj8 A 2.1 BS01 ADP A 1 V560 V561 G598 V599 G600 K601 T602 I765 Q769 R806 V40 V41 G78 V79 G80 K81 T82 I239 Q243 R280 ? 0005524,0016887 remove_due_to_license_issue Q9RA63 24531492 901 HMEVTEEDIAEIVSRWTGIPVSKLLEGELLRLEEELHKRVVGQDEAIRAVADAIRRARAGLKDPNRPIGSFLFLGPTGVGKTELAKTLAATLFDTEEAMIQIDMTEYMEKHAVSRLIGAPPGGGQLTEAVRRRPYSVILFDEIEKAHPDVFNILLQILDDGRLTDSHGRTVDFRNTVIILTSNLGSPLILEGLQKGWPYERIRDEVFKVLQQHFRPEFLNRLDEIVVFRPLTKEQIRQIVEIQLSYLRARLAEKRISLELTEAAKDFLAERGYDPVFGARPLRRVIQRELETPLAQKILAGEVKEGDRVQVDVGPAGLVFAVP 4ljh A 1.45 BS02 GAL A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 23869965 203 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4ljr A 1.8 BS01 dna D 0 R52 F140 R48 F136 ? 0009294 remove_due_to_license_issue O25100 24369431 5 MKSHFQYSTLENIPKAFDILKDPPKKLYCVGDTKLLDTPLKVAIIGTRRPTPYSKQHTITLARELAKNGAVIVSGGALGVDIIAQENALPKTIMLSPCSLDFIYPTNNHKVIQEIAQNGLILSEYEKDFMPIKGSFLARNRLVIALSDVVIIPQADLKSGSMSSARLAQKYQKPLFVLPQRLNESDGTNELLEKGQAQGIFNIQNFINTLLKD 4ljr B 1.8 BS01 dna C 0 R52 Y108 P135 K137 F140 K162 R48 Y104 P131 K133 F136 K158 ? 0009294 remove_due_to_license_issue O25100 24369431 1 ~ 6 MKSHFQYSTLENIPKAFDILKDPPKKLYCVGDTKLLDTPLKVAIIGTRRPTPYSKQHTITLARELAKNGAVIVSGGALGVDIIAQENALPKTIMLSPCSLDFIYPTNNHKVIQEIAQNGLILSEYEKDFMPIKGSFLARNRLVIALSDVVIIPQADLKSGSMSSARLAQKYQKPLFVLPQRLNESDGTNELLEKGQAQGIFNIQNFINTLLKD 4lk6 A 2.859 BS02 LRD A 1 H50 Q53 H50 Q53 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 23869965 902 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lk6 A 2.859 BS03 GAL A 1 H50 Q53 H50 Q53 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 23869965 903 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lk7 A 1.758 BS02 GAL A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 23869965 203 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lkd A 2.307 BS01 GAL A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 24307364 201 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lke A 1.653 BS01 GAL A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 24307364 201 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lkf A 1.64 BS01 GAL A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 24307364 201 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lkf B 1.64 BS01 GAL B 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 24307364 201 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4lkg A 2.994 BS01 GAL G 1 G216 Q217 G216 Q217 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRV0 24009358 2 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSSCRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKNPALIVWGIHHSGSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARTQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDADCEGDCYYSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4lkg A 2.994 BS02 SIA G 1 Y88 A125 T126 S127 W142 H174 E181 L185 Q217 Y88 A125 T126 S127 W142 H174 E181 L185 Q217 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRV0 24009358 3 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSSCRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKNPALIVWGIHHSGSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARTQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDADCEGDCYYSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4lkh A 3.099 BS01 SIA A 1 Y88 A125 T126 S127 H174 E181 Q217 Y88 A125 T126 S127 H174 E181 Q217 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRV0 24009358 603 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSSCRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKNPALIVWGIHHSGSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARTQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDADCEGDCYYSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4lkj A 2.798 BS01 SIA C 1 Y88 A125 T126 W142 H174 Q217 Y86 A123 T124 W140 H172 Q215 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRV5 24009358 3 ICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARPQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4lkk A 2.491 BS01 GAL C 1 G216 Q217 G214 Q215 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRV5 24009358 1 ICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARPQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4lkk A 2.491 BS02 SIA C 1 Y88 A125 T126 S127 W142 H174 E181 Q217 Y86 A123 T124 S125 W140 H172 E179 Q215 ? 0016020,0019031,0019062,0019064,0020002,0039654,0046718,0046789,0075512 remove_due_to_license_issue V5IRV5 24009358 2 ICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSACRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARPQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPE 4lkl A 1.58 BS02 ADM B 1 L491 R518 L120 R139 2.7.11.21 remove_due_to_license_issue P53350 24223211 101 CHLSDMLQQLHSVNASKPSERGLVRQEEAEDPACIPIFWVSKWVDYSDKYGLGYQLCDNSVGVLFNDSTRLILYNDGDSLQYIERDGTESYLTVSSHPNSLMKKITLLKYFRNYMSEHLLKAGANITPLPYLRTWFRTRSAIILHLSNGSVQINFFQDHTKLILCPLMAAVTYIDEKRDFRTYRLSLLEEYGCCKELASRLRYARTMVDKLLSS 4lko A 2.43 BS01 1WH A 1 E205 E206 Y547 S630 Y662 Y666 N710 H740 E167 E168 Y509 S592 Y624 Y628 N672 H702 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=8.3nM remove_due_to_license_issue P27487 23964740 801 SRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 4lkq A 1.62 BS01 1XM A 1 Q726 F729 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=450uM remove_due_to_license_issue Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4lkt A 2.57 BS01 EIC A 1 M23 L32 M35 L60 R129 Y131 M25 L34 M37 L62 R131 Y133 ? 0001972,0005324,0005504,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005886,0006006,0006629,0006656,0006869,0008289,0008544,0010829,0014069,0015908,0015909,0030667,0031392,0035360,0035578,0042593,0042802,0045202,0051930,0070062,0098921,0098978,0099092,0099178,0099524,0120162,1990379 remove_due_to_license_issue Ki=1.26e+3nM Q01469 24692551 601 NAMATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTLKTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVECVMNNVTCTRIYEKVE 4ll3 A 1.95 BS01 017 A 1 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=2.7pM remove_due_to_license_issue Q9WFL7 24785545 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4ll3 A 1.95 BS02 017 A 2 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Kd=2.7pM remove_due_to_license_issue Q9WFL7 24785545 202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4ll3 B 1.95 BS01 017 A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q9WFL7 24785545 201 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4ll3 B 1.95 BS02 017 A 2 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q9WFL7 24785545 202 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4llk A 1.55 BS01 MEW A 1 S677 I692 F729 S232 I247 F284 3.1.4.17 0004114,0007165,0008081 Ki=990uM remove_due_to_license_issue Ki=990000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4llp A 1.75 BS01 4ZE A 1 I692 F729 I247 F284 3.1.4.17 0004114,0007165,0008081 Ki=16uM remove_due_to_license_issue Ki=16000nM Q9Y233 24375910 801 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4llp A 1.75 BS02 4ZE A 2 Q726 F729 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=16uM remove_due_to_license_issue Ki=16000nM Q9Y233 24375910 802 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4llx A 1.75 BS01 5ZE A 1 Q726 F729 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=1300uM remove_due_to_license_issue Ki=1300000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4lm0 A 1.66 BS01 5NI A 1 F696 Q726 F729 F251 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=560uM remove_due_to_license_issue Ki=560000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4lm1 A 1.6 BS01 7ZE A 1 I692 F696 M713 Q726 F729 I247 F251 M268 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=590uM remove_due_to_license_issue Ki=590000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWISS 4lm2 A 1.55 BS01 8ZE A 1 S677 I692 Q726 F729 S232 I247 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=940uM remove_due_to_license_issue Ki=940000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4lm3 A 1.49 BS01 9ZE A 1 S677 I692 M713 Q726 F729 S232 I247 M268 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=1200uM remove_due_to_license_issue Ki=1200000nM Q9Y233 24375910 801 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWIS 4lm4 A 1.48 BS01 JPZ A 1 L675 S677 I692 Q726 F729 L230 S232 I247 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=910uM remove_due_to_license_issue Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4lm5 A 2.25 BS01 Q17 A 1 F49 V52 A65 K67 E121 L174 I185 D186 F15 V18 A31 K33 E81 L134 I145 D146 D167 K169 N172 D186 L193 T204 D127 K129 N132 D146 L153 T164 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 24531473 401 ESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGEVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4lmn A 2.8 BS03 EUI A 1 K97 L118 V127 I141 M143 D190 D208 F209 S212 L215 K37 L58 V67 I81 M83 D130 D148 F149 S152 L155 D190 K192 S194 N195 D208 D217 T226 D130 K132 S134 N135 D148 D157 T166 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=4.2nM Q02750 23934108 503 MELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMANSFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGLN 4lmu A 2.38 BS01 QUE A 1 L44 A65 K67 L120 E121 R122 V126 L174 I185 D186 L9 A30 K32 L81 E82 R83 V87 L135 I146 D147 D167 K169 N172 D186 L193 T204 D128 K130 N133 D147 L154 T165 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=1100nM, Kd=25nM P11309 24531473 401 SQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGETRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHL 4ln7 A 1.73 BS03 1ZQ A 1 A20 Y24 K34 I38 H41 E80 D108 E119 K134 A25 Y29 K39 I43 H46 E85 D113 E124 K139 0003723,0039694 ic50=0.041uM remove_due_to_license_issue 23978130 306 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERG 4lnb B 1.752 BS03 ED5 B 1 A168 L169 R274 D387 C389 D452 Y454 H455 A79 L80 R185 D298 C300 D360 Y362 H363 H333 R381 K384 D387 C389 Y390 D445 D452 H455 H244 R292 K295 D298 C300 Y301 D353 D360 H363 2.5.1.58 0003824,0004659,0004660,0005965,0008270,0008318,0018343,0046872,0097354 remove_due_to_license_issue Q4WPS9 24347326 603 VHPGIPALFREPPLIHDLLSTETTELQSETVNKCLPLLKGIHNSQKGPFNKYGIPALQRKDHLEYLYDSLEDYPASFVALDASRPWMVYWALAGLCLLGEDVTRFRERVISTFTAAQNSTGGIGGGHGQMSHVASSYAAVLSIAMVGGEEAFKLIDRKAMWKWLGKLKQPDGGFTVCEGGEEDVRGAYCAMVVHALLDLPLALPPEAEARQNGLETFTDGLPEYLSRCQTYEGGISGSPGSEAHGAYAFCALACLCLLGRPEVVVPRYMNIATLLPWLSARQYAPEGGFSGRTNKLVDGCYSHWVGNCWPLVQAALDGTQPLARSSVGNLYSREGLTRYILSCCQCKLGGLRDKPGKHPDSYHTCYALTGLSTVQYYHYCTDSSVSSKFSSAFSWKHDPNFASDGQGSDIGVFTENDRLVPFHPIFVIPHKSAEDIRVWFENQSFDL 4lnf A 2.949 BS03 GLN A 1 E134 Y156 E189 R298 E304 E133 Y155 E188 R297 E303 D53 E132 E134 E189 E196 H245 R316 E333 R335 D52 E131 E133 E188 E195 H244 R315 E332 R334 6.3.1.2 0000287,0003824,0004356,0005515,0005524,0005737,0006542,0016595,0016874,0043562,0045892,0046872,0070406,0090295,0140297,1904797 remove_due_to_license_issue P12425 24158439 503 AKYTREDIEKLVKEENVKYIRLQFTDILGTIKNVEIPVSQLGKALDNKVMFDGSSIEGFVRIEESDMYLYPDLNTFVIFPWTAEKGKVARFICDIYNPDGTPFEGDPRNNLKRILKEMEDLGFSDFNLGPEPEFFLFKLDEKGEPTLELNDKGGYFDLAPTDLGENCRRDIVLELEEMGFEIEASHHEVAPGQHEIDFKYAGAVRSCDDIQTFKLVVKTIARKHGLHATFMPKPLFGVNGSGMHCNLSLFKNGVNAFFDENADLQLSETAKHFIAGIVKHATSFTAVTNPTVNSYKRLVPGYEAPCYVAWSAQNRSPLIRIPASRGISTRVEVRSVDPAANPYLALSVLLAAGLDGIKNKLEAPAPIDRNIYVMSKEERMENGIVDLPATLAEALEEFKSNEVMVKALGEHLFEHFIEAKEIEWDMFRTQVHPWEREQYMSQY 4lnf B 2.949 BS03 GLN B 1 E134 E189 G241 R298 E304 E133 E188 G240 R297 E303 D53 E132 E134 E189 E196 H245 R316 E333 R335 D52 E131 E133 E188 E195 H244 R315 E332 R334 6.3.1.2 0000287,0003824,0004356,0005515,0005524,0005737,0006542,0016595,0016874,0043562,0045892,0046872,0070406,0090295,0140297,1904797 remove_due_to_license_issue P12425 24158439 503 AKYTREDIEKLVKEENVKYIRLQFTDILGTIKNVEIPVSQLGKALDNKVMFDGSSIEGFVRIEESDMYLYPDLNTFVIFPWTAEKGKVARFICDIYNPDGTPFEGDPRNNLKRILKEMEDLGFSDFNLGPEPEFFLFKLDEKGEPTLELNDKGGYFDLAPTDLGENCRRDIVLELEEMGFEIEASHHEVAPGQHEIDFKYAGAVRSCDDIQTFKLVVKTIARKHGLHATFMPKPLFGVNGSGMHCNLSLFKNGVNAFFDENADLQLSETAKHFIAGIVKHATSFTAVTNPTVNSYKRLVPGYEAPCYVAWSAQNRSPLIRIPASRGISTRVEVRSVDPAANPYLALSVLLAAGLDGIKNKLEAPAPIDRNIYVMSKEERMENGIVDLPATLAEALEEFKSNEVMVKALGEHLFEHFIEAKEIEWDMFRTQVHPWEREQYMSQY 4lng B 1.905 BS02 JAN B 1 W157 D365 C367 D430 Y432 H433 W89 D297 C299 D357 Y359 H360 H311 R359 K362 D365 C367 Y368 D423 D430 H433 H243 R291 K294 D297 C299 Y300 D350 D357 H360 2.5.1.58 0003824,0004659,0004660,0005965,0008270,0008318,0018343,0046872,0097354 remove_due_to_license_issue Q4WPS9 24347326 602 HPGIPALFREPPLIHDLLSTETTELQSETVNKCLPLLKGIHNSQKGPFNKYGIPALQRKDHLEYLYDSLEDYPASFVALDASRPWMVYWALAGLCLLGEDVTRFRERVISTFTAAQNSTGGIGGGHGQMSHVASSYAAVLSIAMVGGEEAFKLIDRKAMWKWLGKLKQPDGGFTVCEGGEEDVRGAYCAMVVHALLDLPLALPPEAEARQNGLETFTDGLPEYLSRCQTYEGGISGSPGSEAHGAYAFCALACLCLLGRPEVVVPRYMNIATLLPWLSARQYAPEGGFSGRTNKLVDGCYSHWVGNCWPLVQAALDGTQPLSSVGNLYSREGLTRYILSCCQCKLGGLRDKPGKHPDSYHTCYALTGLSTVQYYHYCTDSSVSSKDDFSSAFSWKHDPNFASDGQGSDIGVFTENDRLVPFHPIFVIPHKSAEDIRVWFENQSFDL 4lno A 2.9 BS03 GLN A 1 E134 Y156 E189 R298 E304 E133 Y155 E188 R297 E303 D53 E132 E134 E189 E196 H245 R316 E333 R335 D52 E131 E133 E188 E195 H244 R315 E332 R334 6.3.1.2 0000287,0003824,0004356,0005515,0005524,0005737,0006542,0016595,0016874,0043562,0045892,0046872,0070406,0090295,0140297,1904797 remove_due_to_license_issue P12425 24158439 503 AKYTREDIEKLVKEENVKYIRLQFTDILGTIKNVEIPVSQLGKALDNKVMFDGSSIEGFVRIEESDMYLYPDLNTFVIFPWTAEKGKVARFICDIYNPDGTPFEGDPRNNLKRILKEMEDLGFSDFNLGPEPEFFLFKLDEKGEPTLELNDKGGYFDLAPTDLGENCRRDIVLELEEMGFEIEASHHEVAPGQHEIDFKYAGAVRSCDDIQTFKLVVKTIARKHGLHATFMPKPLFGVNGSGMHCNLSLFKNGVNAFFDENADLQLSETAKHFIAGIVKHATSFTAVTNPTVNSYKRLVPGYEAPCYVAWSAQNRSPLIRIPASRGISTRVEVRSVDPAANPYLALSVLLAAGLDGIKNKLEAPAPIDRNIYVMSKEERMENGIVDLPATLAEALEEFKSNEVMVKALGEHLFEHFIEAKEIEWDMFRTQVHPWEREQYMSQY 4lno B 2.9 BS03 GLN B 1 E134 E189 H245 R298 E304 R335 E133 E188 H244 R297 E303 R334 D53 E132 E134 E189 E196 H245 R316 E333 R335 D52 E131 E133 E188 E195 H244 R315 E332 R334 6.3.1.2 0000287,0003824,0004356,0005515,0005524,0005737,0006542,0016595,0016874,0043562,0045892,0046872,0070406,0090295,0140297,1904797 remove_due_to_license_issue P12425 24158439 503 AKYTREDIEKLVKEENVKYIRLQFTDILGTIKNVEIPVSQLGKALDNKVMFDGSSIEGFVRIEESDMYLYPDLNTFVIFPWTAEKGKVARFICDIYNPDGTPFEGDPRNNLKRILKEMEDLGFSDFNLGPEPEFFLFKLDEKGEPTLELNDKGGYFDLAPTDLGENCRRDIVLELEEMGFEIEASHHEVAPGQHEIDFKYAGAVRSCDDIQTFKLVVKTIARKHGLHATFMPKPLFGVNGSGMHCNLSLFKNGVNAFFDENADLQLSETAKHFIAGIVKHATSFTAVTNPTVNSYKRLVPGYEAPCYVAWSAQNRSPLIRIPASRGISTRVEVRSVDPAANPYLALSVLLAAGLDGIKNKLEAPAPIDRNIYVMSKEERMENGIVDLPATLAEALEEFKSNEVMVKALGEHLFEHFIEAKEIEWDMFRTQVHPWEREQYMSQY 4lnq A 2.0 BS01 dna C 0 S166 H222 R224 G226 S118 H174 R176 G178 ? 0002218,0035458 remove_due_to_license_issue Q9R002 24419611 1 ~ 20 GPHMKGAVLHEKPMTVMVLTATEPFNYKEGKENMFHATVATESKYYRVKVFNMDLKEKFTENKFITISKYFNSSGILEINETATVSEAAPNQMFEVPKNIIRSAKETLKISKIKELDSGTLIYGVFAVEKKKVNDKSITFKIKDNEDNIKVVWDKEQHNINYEKGDKLQLFSFHLRKGNGKPILHSGNHSFIKGE 4lnq A 2.0 BS02 dna D 0 K180 N182 K184 S185 T187 K132 N134 K136 S137 T139 ? 0002218,0035458 remove_due_to_license_issue Q9R002 24419611 1 ~ 20 GPHMKGAVLHEKPMTVMVLTATEPFNYKEGKENMFHATVATESKYYRVKVFNMDLKEKFTENKFITISKYFNSSGILEINETATVSEAAPNQMFEVPKNIIRSAKETLKISKIKELDSGTLIYGVFAVEKKKVNDKSITFKIKDNEDNIKVVWDKEQHNINYEKGDKLQLFSFHLRKGNGKPILHSGNHSFIKGE 4lnq B 2.0 BS01 dna C 0 N182 D183 K184 S185 T187 K198 N129 D130 K131 S132 T134 K145 ? 0002218,0035458 remove_due_to_license_issue Q9R002 24419611 1 ~ 20 GAVLHEKPMTVMVLTATEPFNYKEGKENMFHATVATESKYYRVKVFNMDLKEKFTENKFITISKYFNSSGILEINETATVSEAAPNQMFEVPKNIIRSAKETLKISKIKELDSGTLIYGVFAVEKKKVNDKSITFKIKDNEDNIKVVWDKEQHNINYEKGDKLQLFSFHLRKGNGKPILHSGNHSFIKGEKL 4lnq B 2.0 BS02 dna D 0 S166 H222 R224 K225 G226 S113 H169 R171 K172 G173 ? 0002218,0035458 remove_due_to_license_issue Q9R002 24419611 1 ~ 20 GAVLHEKPMTVMVLTATEPFNYKEGKENMFHATVATESKYYRVKVFNMDLKEKFTENKFITISKYFNSSGILEINETATVSEAAPNQMFEVPKNIIRSAKETLKISKIKELDSGTLIYGVFAVEKKKVNDKSITFKIKDNEDNIKVVWDKEQHNINYEKGDKLQLFSFHLRKGNGKPILHSGNHSFIKGEKL 4lnw A 1.9 BS01 T3 A 1 F215 F218 I222 R228 M256 M259 R262 L276 S277 L292 H381 F401 F71 F74 I78 R84 M112 M115 R118 L132 S133 L148 H237 F257 ? 0003677,0004879,0006355 remove_due_to_license_issue P10827 24552590 501 SHMEEMIRSLQQRPEPTPEEWDLIHIATEAHRSTNAQGSHWKQRRKFLPDDIGQSPIVSMPDGDKVDLEAFSEFTKIITPAITRVVDFAKKLPMFSELPCEDQIILLKGCCMEIMSLRAAVRYDPESDTLTLSGEMAVKREQLKNGGLGVVSDAIFELGKSLSAFNLDDTEVALLQAVLLMSTDRSGLLCVDKIEKSQEAYLLAFEHYVNHRKHNIPHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 4lnw A 1.9 BS02 T3 A 2 Q342 L368 V371 R375 Q198 L224 V227 R231 ? 0003677,0004879,0006355 remove_due_to_license_issue P10827 24552590 502 SHMEEMIRSLQQRPEPTPEEWDLIHIATEAHRSTNAQGSHWKQRRKFLPDDIGQSPIVSMPDGDKVDLEAFSEFTKIITPAITRVVDFAKKLPMFSELPCEDQIILLKGCCMEIMSLRAAVRYDPESDTLTLSGEMAVKREQLKNGGLGVVSDAIFELGKSLSAFNLDDTEVALLQAVLLMSTDRSGLLCVDKIEKSQEAYLLAFEHYVNHRKHNIPHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED 4loh A 2.25 BS01 1SY A 1 S162 Y163 Y167 R238 Y240 T263 P264 S9 Y10 Y14 R85 Y87 T110 P111 ? 0002218,0032481 Kd=5.3uM remove_due_to_license_issue Q86WV6 23910378 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDHAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEE 4loh B 2.25 BS01 1SY A 1 S162 Y167 R238 T263 S9 Y14 R85 T110 ? 0002218,0032481 remove_due_to_license_issue Q86WV6 23910378 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDHAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEE 4loi A 1.89 BS01 1YC B 1 S162 Y167 R238 T263 S9 Y14 R80 T105 ? 0002218,0032481 remove_due_to_license_issue EC50=30nM, Kd=287000nM Q86WV6 23910378 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDHAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEK 4loi B 1.89 BS01 1YC B 1 S162 Y163 Y167 R238 T263 S9 Y10 Y14 R85 T110 ? 0002218,0032481 Kd=0.17uM remove_due_to_license_issue EC50=30nM, Kd=287000nM Q86WV6 23910378 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDHAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQE 4loj A 1.77 BS01 1SY B 1 S161 Y162 Y166 R237 Y239 T262 S7 Y8 Y12 R83 Y85 T108 ? 0002218,0032481 remove_due_to_license_issue Q3TBT3 23910378 401 AHGLAWSYYIGYLRLILPGLQARIRMFNQLHNNMLSGAGSRRLYILFPLDCGVPDNLSVVDPNIRFRDMLPQQNIDRAGIKNRVYSNSVYEILENGQPAGVCILEYATPLQTLFAMSQDAKAGFSREDRLEQAKLFCRTLEEILEDVPESRNNCRLIVYQEPTDGNSFSLSQEVLRHIRQ 4loj B 1.77 BS01 1SY B 1 S161 Y166 R237 Y239 T262 S6 Y11 R82 Y84 T107 ? 0002218,0032481 remove_due_to_license_issue Q3TBT3 23910378 401 HGLAWSYYIGYLRLILPGLQARIRMFNQLHNNMLSGAGSRRLYILFPLDCGVPDNLSVVDPNIRFRDMLPQQNIDRAGIKNRVYSNSVYEILENGQPAGVCILEYATPLQTLFAMSQDAKAGFSREDRLEQAKLFCRTLEEILEDVPESRNNCRLIVYQEPTDGNSFSLSQEVLRHIRQ 4loo A 1.95 BS02 SB4 A 1 V38 A51 K53 L104 V105 T106 M109 L167 V34 A47 K49 L100 V101 T102 M105 L163 D150 K152 N155 D168 T185 D146 K148 N151 D164 T181 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 remove_due_to_license_issue P47811 24037507 401 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 4lop A 2.049 BS03 SB4 A 1 V38 A51 L104 V105 T106 L108 M109 D112 L167 V36 A49 L102 V103 T104 L106 M107 D110 L165 D150 K152 N155 D168 T185 D148 K150 N153 D166 T183 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 remove_due_to_license_issue P47811 24037507 401 QERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 4loq A 2.319 BS03 SB4 A 1 V38 A51 L104 T106 M109 L167 V36 A49 L102 T104 M107 L165 D150 K152 N155 D168 T185 D148 K150 N153 D166 T183 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006974,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030278,0030316,0031098,0031663,0032495,0032496,0032735,0032868,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051403,0051525,0060045,0060348,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090400,0098586,0098978,0099179,0106310,1900015,1901741,2000379 remove_due_to_license_issue P47811 24037507 401 QERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLD 4lov A 1.5 BS01 KGM A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 ? 0007155,0009289 Kd=17.1nM remove_due_to_license_issue P08191 24476493 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4loy H 1.77 BS03 6XS H 1 H57 Y60A W60D D189 A190 V213 W215 G216 G219 G226 F227 Y228 H43 Y47 W50 D192 A193 V218 W220 G221 G223 G231 F232 Y233 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 24175584 304 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4lp0 A 1.95 BS01 1YM A 1 E55 D78 R81 M83 P84 I98 E39 D62 R65 M67 P68 I82 5.6.2.2 0003677,0003918,0005524,0006265 ic50<10nM remove_due_to_license_issue Q8DQB5 24098982 301 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4lp6 A 2.15 BS01 Q4I A 1 H94 H119 F130 L197 T198 T199 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 24288253 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4lp6 A 2.15 BS04 Q4I B 1 H4 W5 D19 F20 H64 H1 W2 D16 F17 H61 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 24288253 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4lpb A 1.75 BS01 1YP A 1 N51 E55 D78 R81 M83 P84 I98 R140 T172 N35 E39 D62 R65 M67 P68 I82 R107 T139 5.6.2.2 0003677,0003918,0005524,0006265 ic50<10nM remove_due_to_license_issue Q8DQB5 24098982 301 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHAVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4lpf A 2.3 BS01 3TR A 1 H73 H74 E77 H64 H65 E68 0000105,0004424 remove_due_to_license_issue 301 SRRARIERRTRESDIVIELDLDGTGQVAVDTGVPFYDHMLTALGSHASFDLTVRATGDVEIEAHHTIEDTAIALGTALGQALGDKRGIRRFGDAFIPMDETLAHAAVDLSGRPYCVHTGEPDHLQHTTIAGSSVPYHTVINRHVFESLAANARIALHVRVLYGRDPHHITEAQYKAVARALRQAVEPDPR 4lpg F 2.35 BS01 1MV F 1 K57 N59 F206 F239 L344 K49 N51 F198 F231 L336 2.5.1.1,2.5.1.10 0004659,0008299,0016765 Kd=55.6uM remove_due_to_license_issue IC50=390nM, Kd=3200nM P14324 24911527 402 DVYAQEKQDFVQHFSQIVRVLTEEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 4lph F 2.3 BS02 YL3 F 1 N59 F239 L344 N52 F232 L337 2.5.1.1,2.5.1.10 0004659,0008299,0016765 Kd=9.2uM remove_due_to_license_issue IC50=5000nM, Kd=9200nM P14324 24911527 402 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 4lps A 2.0 BS02 GDP A 1 G56 G58 K59 T60 T61 R89 K183 D185 S214 S215 G29 G31 K32 T33 T34 R62 K156 D158 S187 S188 ? 0003924,0005525,0008270,0016151,0016787,0046872,0051604 remove_due_to_license_issue O25560 24338018 302 SKNDIKAAEMKERYLKEGLYVLNFMSSPGSGKTTMLENLADFKDFKFCVVEGDLQTNRDADRLRKKGVSAHQITTGEACHLEASMIEGAFDLLKDEGALEKSDFLIIENVGNLVCPSSYNLGAAMNIVLLSVPEGDDKVLKYPTMFMCADAVIISKADMVEVFNFRVSQVKEDMQKLKPEAPIFLMSSKDPKSLEDFKNFLLEKKRENYQSTHSF 4lps A 2.0 BS04 GDP B 1 P160 K165 P133 K138 ? 0003924,0005525,0008270,0016151,0016787,0046872,0051604 remove_due_to_license_issue O25560 24338018 302 SKNDIKAAEMKERYLKEGLYVLNFMSSPGSGKTTMLENLADFKDFKFCVVEGDLQTNRDADRLRKKGVSAHQITTGEACHLEASMIEGAFDLLKDEGALEKSDFLIIENVGNLVCPSSYNLGAAMNIVLLSVPEGDDKVLKYPTMFMCADAVIISKADMVEVFNFRVSQVKEDMQKLKPEAPIFLMSSKDPKSLEDFKNFLLEKKRENYQSTHSF 4lq3 A 2.6 BS02 20V A 1 V324 N326 D354 V317 N319 D347 3.6.1.15 0000166,0001172,0003723,0003968,0004386,0005524,0006351,0008234,0039694,0046872 remove_due_to_license_issue Q2N379 24316032 601 GTYCGAPILGPGSAPKLSTKTKFWRSSTTPLPPGTYEPAYLGGKDPRVKGGPSLQQVMRDQLKPFTEPRGKPPKPSVLEAAKKTIINVLEQTIDPPEKWSFTQACASLDKTTSSGHPHHMRKNDCWNGESFTGKLADQASKANLMFEGGKNMTPVYTGALKDELVKTDKIYGKIKKRLLWGSDLATMIRCARAFGGLMDELKAHCVTLPIRVGMNMNEDGPIIFERHSRYKYHYDADYSRWDSTQQRAVLAAALEIMVKFSSEPHLAQVVAEDLLSPSVVDVGDFKISINEPSGVPCTSQWNSIAHWLLTLCALSEVTNLSPDIIQANSLFSFYGDDEIVSTDIKLDPEKLTAKLKEYGLKPTRPDGPLVISEDLNGLTFLRRTVTRDPAGWFGKLEQSSILRQMYWTRGPNHEDPSETMSQRPIQLMSLLGEAALHGPAFYSKISKLVIAELKEGMDYVPRQEPMFRWMRFSDLSTWEGDRNLAPSFVNEDGVE 4lq3 A 2.6 BS03 20V A 2 K166 E168 R392 L406 S410 I411 Q414 R419 D507 E510 K161 E163 R382 L396 S400 I401 Q404 R409 D492 E495 3.6.1.15 0000166,0001172,0003723,0003968,0004386,0005524,0006351,0008234,0039694,0046872 remove_due_to_license_issue Q2N379 24316032 603 GTYCGAPILGPGSAPKLSTKTKFWRSSTTPLPPGTYEPAYLGGKDPRVKGGPSLQQVMRDQLKPFTEPRGKPPKPSVLEAAKKTIINVLEQTIDPPEKWSFTQACASLDKTTSSGHPHHMRKNDCWNGESFTGKLADQASKANLMFEGGKNMTPVYTGALKDELVKTDKIYGKIKKRLLWGSDLATMIRCARAFGGLMDELKAHCVTLPIRVGMNMNEDGPIIFERHSRYKYHYDADYSRWDSTQQRAVLAAALEIMVKFSSEPHLAQVVAEDLLSPSVVDVGDFKISINEPSGVPCTSQWNSIAHWLLTLCALSEVTNLSPDIIQANSLFSFYGDDEIVSTDIKLDPEKLTAKLKEYGLKPTRPDGPLVISEDLNGLTFLRRTVTRDPAGWFGKLEQSSILRQMYWTRGPNHEDPSETMSQRPIQLMSLLGEAALHGPAFYSKISKLVIAELKEGMDYVPRQEPMFRWMRFSDLSTWEGDRNLAPSFVNEDGVE 4lq3 A 2.6 BS04 20V A 3 I463 A464 K467 I450 A451 K454 3.6.1.15 0000166,0001172,0003723,0003968,0004386,0005524,0006351,0008234,0039694,0046872 remove_due_to_license_issue Q2N379 24316032 604 GTYCGAPILGPGSAPKLSTKTKFWRSSTTPLPPGTYEPAYLGGKDPRVKGGPSLQQVMRDQLKPFTEPRGKPPKPSVLEAAKKTIINVLEQTIDPPEKWSFTQACASLDKTTSSGHPHHMRKNDCWNGESFTGKLADQASKANLMFEGGKNMTPVYTGALKDELVKTDKIYGKIKKRLLWGSDLATMIRCARAFGGLMDELKAHCVTLPIRVGMNMNEDGPIIFERHSRYKYHYDADYSRWDSTQQRAVLAAALEIMVKFSSEPHLAQVVAEDLLSPSVVDVGDFKISINEPSGVPCTSQWNSIAHWLLTLCALSEVTNLSPDIIQANSLFSFYGDDEIVSTDIKLDPEKLTAKLKEYGLKPTRPDGPLVISEDLNGLTFLRRTVTRDPAGWFGKLEQSSILRQMYWTRGPNHEDPSETMSQRPIQLMSLLGEAALHGPAFYSKISKLVIAELKEGMDYVPRQEPMFRWMRFSDLSTWEGDRNLAPSFVNEDGVE 4lq9 A 2.04 BS01 21D A 1 Q414 W417 T418 R419 R436 Q439 Q409 W412 T413 R414 R431 Q434 3.6.1.15 0000166,0001172,0003723,0003968,0004386,0005524,0006351,0008234,0039694,0046872 remove_due_to_license_issue Q2N379 24316032 601 GTYCGAPILGPGSAPKLSTKTKFWRSSTTPLPPGTYEPAYLGGKDPRVKGGPSLQQVMRDQLKPFTEPRGKPPKPSVLEAAKKTIINVLEQTIDPPEKWSFTQACASLDKTTSSGHPHHMRKNDCWNGESFTGKLADQASKANLMFEGGKNMTPVYTGALKDELVKTDKIYGKIKKRLLWGSDLATMIRCARAFGGLMDELKAHCVTLPIRVGMNMNEDGPIIFERHSRYKYHYDADYSRWDSTQQRAVLAAALEIMVKFSSEPHLAQVVAEDLLSPSVVDVGDFKISINEGLPSGVPCTSQWNSIAHWLLTLCALSEVTNLSPDIIQANSLFSFYGDDEIVSTDIKLDPEKLTAKLKEYGLKPTRPDKTEGPLVISEDLNGLTFLRRTVTRDPAGWFGKLEQSSILRQMYWTRGPNHEDPSETMIPHSQRPIQLMSLLGEAALHGPAFYSKISKLVIAELKEGGMDFYVPRQEPMFRWMRFSDLSTWEGDRNLAPSFVNE 4lq9 A 2.04 BS02 21D A 2 Q66 V170 K171 K174 K180 R182 Q61 V165 K166 K169 K175 R177 3.6.1.15 0000166,0001172,0003723,0003968,0004386,0005524,0006351,0008234,0039694,0046872 remove_due_to_license_issue Q2N379 24316032 602 GTYCGAPILGPGSAPKLSTKTKFWRSSTTPLPPGTYEPAYLGGKDPRVKGGPSLQQVMRDQLKPFTEPRGKPPKPSVLEAAKKTIINVLEQTIDPPEKWSFTQACASLDKTTSSGHPHHMRKNDCWNGESFTGKLADQASKANLMFEGGKNMTPVYTGALKDELVKTDKIYGKIKKRLLWGSDLATMIRCARAFGGLMDELKAHCVTLPIRVGMNMNEDGPIIFERHSRYKYHYDADYSRWDSTQQRAVLAAALEIMVKFSSEPHLAQVVAEDLLSPSVVDVGDFKISINEGLPSGVPCTSQWNSIAHWLLTLCALSEVTNLSPDIIQANSLFSFYGDDEIVSTDIKLDPEKLTAKLKEYGLKPTRPDKTEGPLVISEDLNGLTFLRRTVTRDPAGWFGKLEQSSILRQMYWTRGPNHEDPSETMIPHSQRPIQLMSLLGEAALHGPAFYSKISKLVIAELKEGGMDFYVPRQEPMFRWMRFSDLSTWEGDRNLAPSFVNE 4lqg A 1.77 BS05 CTW A 1 R210 N257 D387 E424 E425 L428 R463 G518 N519 R534 W541 Y552 H553 K699 Y700 R156 N203 D333 E370 E371 L374 R409 G464 N465 R480 W487 Y496 H497 K641 Y642 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue IC50=1300nM Q04609 27228467 823 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4lqy A 1.54 BS01 AMP A 1 D34 T70 F71 N91 D104 Y154 Y184 D189 H336 D11 T47 F48 N68 D81 Y131 Y161 D166 H313 3.6.1.29 ic50=129uM remove_due_to_license_issue Q9Y6X5 24338010 505 LPPKLLLVSFDGFRADYLKNYEFPHLQNFIKEGVLVEHVKNVFITKTFPNHYSIVTGLYEESHGIVANSMYDAVTKKHFSDSNDKDPFWWNEAVPIWVTNQLQENRSSAAAMWPGTDVPIHDTISSYFMNYNSSVSFEERLNNITMWLNNSNPPVTFATLYWEEPDASGHKYGPEDKENMSRVLKKIDDLIGDLVQRLKMLGLWENLNVIITSDHGMTQCSQDRLINLDSCIDHSYYTLIDLSPVAAILPKINRTEVYNKLKNCSPHMNVYLKEDIPNRFYYQHNDRIQPIILVADEGWTIVLNESSQKLGDHGYDNSLPSMHPFLAAHGPAFHKGYKHSTINIVDIYPMMCHILGLKPHPNNGTFGHTKCLLVDQWCI 4lrh A 2.8 BS01 FOL A 1 Y60 D81 Y85 W102 W134 H135 K136 G137 W140 W171 S174 Y175 Y53 D74 Y78 W95 W127 H128 K129 G130 W133 W164 S167 Y168 ? remove_due_to_license_issue P15328 23851396 301 RTELLNVCMNAKHHKEKPGPEDKLHEQCRPWRKNACCSTNTSQEAHKDVSYLYRFNWNHCGEMAPACKRHFIQDTCLYECSPNLGPWIQQVDQSWRKERVLNVPLCKEDCEQWWEDCRTSYTCKSNWHKGWNWTSGFNKCAVGAACQPFHFYFPTPTVLCNEIWTHSYKVSNYSRGSGRCIQMWFDPAQGNPNEEVARFYAAAMSGT 4lrr A 2.41 BS01 CF9 A 1 E58 F62 W80 W83 Y94 L143 C146 H147 Q165 S167 D169 G173 N177 E58 F62 W80 W83 Y94 L143 C146 H147 Q165 S167 D169 G173 N177 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Ki=6uM remove_due_to_license_issue P0A886 24147825 309 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4lsj A 2.35 BS02 LSJ A 1 L563 N564 L566 M601 M604 L608 F623 L732 Y735 C736 T739 L38 N39 L41 M76 M79 L83 F98 L199 Y202 C203 T206 ? Ki=0.268nM remove_due_to_license_issue Ki=0.268000nM P04150 24446728 801 PQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQK 4lts A 1.692 BS01 LTS A 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 S275 R311 I351 Y173 H176 F178 R181 D204 Y225 S226 V227 A229 S260 R296 I336 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=4.4nM remove_due_to_license_issue IC50=6.20nM P43490 24279990 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4lts B 1.692 BS01 LTS B 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 S275 R311 I351 Y172 H175 F177 R180 D203 Y224 S225 V226 A228 S259 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=4.4nM remove_due_to_license_issue IC50=6.20nM P43490 24279990 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEAA 4luo A 1.54 BS01 1DZ A 1 R31 I33 R43 S55 M57 L87 V93 R34 I36 R46 S58 M60 L90 V96 ? 0003677,0005634,0006260 Kd=580uM remove_due_to_license_issue Kd=580000nM P27694 24147804 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4luo A 1.54 BS02 1DZ A 2 R41 N85 L87 V93 I95 R44 N88 L90 V96 I98 ? 0003677,0005634,0006260 Kd=580uM remove_due_to_license_issue Kd=580000nM P27694 24147804 202 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4luv A 1.4 BS01 1XS A 1 R41 M57 A59 T60 N85 I95 R44 M60 A62 T63 N88 I98 ? 0003677,0005634,0006260 Kd=1400uM remove_due_to_license_issue Kd=710000nM P27694 24147804 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4luz A 1.9 BS01 1XT A 1 I33 R41 R43 S55 M57 A59 T60 V93 I95 I36 R44 R46 S58 M60 A62 T63 V96 I98 ? 0003677,0005634,0006260 Kd=20uM remove_due_to_license_issue Kd=26000nM P27694 24147804 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4lv1 A 1.74 BS01 NL9 A 1 S64 Q120 Y150 N152 Y221 A318 S61 Q117 Y147 N149 Y218 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 25344815 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4lv1 A 1.74 BS02 NL9 A 2 L254 Y259 P304 L251 Y256 P301 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 25344815 402 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4lv2 A 1.65 BS01 N95 A 1 S64 Q120 Y150 N152 Y221 G317 A318 S61 Q117 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 25344815 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4lv3 A 1.42 BS01 25N A 1 S64 Q120 Y150 N152 Y221 G317 A318 S61 Q117 Y147 N149 Y218 G308 A309 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K306 A309 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 25344815 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4lv4 A 2.08 BS03 8HC A 1 H96 E161 E178 H252 H95 E160 E166 H226 D95 H96 H252 N274 D94 H95 H226 N248 4.1.2.13 0004332,0005576,0005829,0005886,0005975,0006096,0008270,0009274,0016829,0016832,0035375,0046872 Kd=9.39uM remove_due_to_license_issue Kd=6940nM, IC50=14000nM P9WQA3 24325645 403 PIATPEVYAEMLGQAKQNSYAFPAINCTSSETVNAAIKGFADAGSDGIIQFSTGGAEFGSGLGVKDMVTGAVALAEFTHVIAAKYPVNVALHTDHCPKDKLDSYVRPLLAISAQRVSKGGNPLFQSHMWDGSAVPIDENLAIAQELLKAAAAAKIILEIEIGVVGEKLYTSPEDFEKTIEALGAGEHGKYLLAATFGPDILAQGQQVAAAKLGLPADAKPFDFVFHGGSGSLKSEIEEALRYGVVKMNVDTDTQYAFTRPIAGHMFTNYDGVLKVDGEVGVKKVYDPRSYLKKAEASMSQRVVQACNDLHCAGKSLTHHH 4lvt A 2.05 BS01 1XJ A 1 D100 F101 R104 Y105 D108 M112 L134 N140 W141 G142 R143 F195 L198 Y199 D38 F39 R42 Y43 D46 M50 L72 N78 W79 G80 R81 F133 L136 Y137 ? 0042981 remove_due_to_license_issue Ki=<1.000000nM, IC50=<15nM P10415 23291630 301 YDNREIVMKYIHYKLSQRGYEWDASEVVHLTLRQAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGP 4lw1 A 1.631 BS01 1XS A 1 R41 M57 A59 T60 I95 R44 M60 A62 T63 I98 ? 0003677,0005634,0006260 Kd=710uM remove_due_to_license_issue Kd=710000nM P27694 24147804 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4lw1 A 1.631 BS02 1XS A 2 R31 I33 R43 S55 L87 R91 V93 R34 I36 R46 S58 L90 R94 V96 ? 0003677,0005634,0006260 Kd=710uM remove_due_to_license_issue Kd=710000nM P27694 24147804 202 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4lwc A 1.61 BS01 1XU A 1 I33 R41 R43 S55 M57 A59 T60 N85 L87 V93 I95 M97 I36 R44 R46 S58 M60 A62 T63 N88 L90 V96 I98 M100 ? 0003677,0005634,0006260 remove_due_to_license_issue Kd=1.7nM P27694 24147804 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4lwe A 1.5 BS01 FJ2 A 1 N51 A55 K58 D93 I96 G97 M98 F138 T184 N35 A39 K42 D77 I80 G81 M82 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=70nM P07900 25313505 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4lwh A 1.7 BS01 FJ5 A 1 N51 A55 K58 D93 I96 G97 M98 L107 T109 F138 T184 N36 A40 K43 D78 I81 G82 M83 L92 T94 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=27nM P07900 25313505 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4lwi A 1.7 BS01 FJ6 A 1 N51 D54 A55 K58 D93 I96 G97 M98 L107 G108 T109 F138 T184 N35 D38 A39 K42 D77 I80 G81 M82 L91 G92 T93 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=23nM P07900 25313505 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4lwt A 1.6 BS01 20Q A 1 L50 I57 Y63 V89 H92 L31 I38 Y44 V70 H73 2.3.2.27 0005634,0043066,0051726 ic50=3.9uM remove_due_to_license_issue P56273 24997575 201 MEKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4lwu A 1.14 BS01 20U A 1 L50 L53 I57 M58 H69 F82 V89 K90 H92 I95 Y96 L30 L33 I37 M38 H49 F62 V69 K70 H72 I75 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.005uM remove_due_to_license_issue P56273 24997575 201 EKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4lwv A 2.32 BS01 20W A 1 L50 L53 G54 I57 H69 F82 V89 H92 I95 Y96 L30 L33 G34 I37 H49 F62 V69 H72 I75 Y76 2.3.2.27 0005634,0043066,0051726 ic50=7nM remove_due_to_license_issue P56273 24900784 201 EKLVQPTPLLLSLLKSAGAQKETFTMKEVLYHLGQYIMAKQLYDEKQQHIVHCSNDPLGELFGVQEFSVKEHRRIYAMISRNLVS 4lww A 1.641 BS01 LWW A 1 Y188 H191 F193 R196 D219 S241 V242 A244 S275 R311 Y172 H175 F177 R180 D203 S225 V226 A228 S259 R295 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=29nM remove_due_to_license_issue IC50=29nM P43490 24279990 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4lww B 1.641 BS01 LWW B 1 H191 F193 R196 D219 S241 V242 A244 S275 R311 H175 F177 R180 D203 S225 V226 A228 S259 R295 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=29nM remove_due_to_license_issue IC50=29nM P43490 24279990 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4lxa A 1.95 BS01 1YS A 1 Q12 G13 L30 D32 G34 S35 P70 Y71 T72 F108 I110 I126 Y198 D228 G230 T231 Q15 G16 L33 D35 G37 S38 P73 Y74 T75 F111 I113 I129 Y189 D219 G221 T222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.002uM remove_due_to_license_issue P56817 23981898 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4lxb H 1.61 BS03 7R9 H 1 H57 Y60A W60D E97A N98 I174 D189 A190 V213 W215 G216 E217 G219 G226 F227 Y228 H43 Y47 W50 E94 N95 I172 D192 A193 V218 W220 G221 E222 G223 G231 F232 Y233 3.4.21.5 0004252,0005509,0006508,0007596 ic50=7nM remove_due_to_license_issue P00734 24175584 304 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4lxd A 1.9 BS01 1XV A 1 D100 Y105 M112 E133 N140 W141 G142 R143 Y199 D42 Y47 M54 E75 N82 W83 G84 R85 Y141 ? 0042981 remove_due_to_license_issue Ki=59nM P10415 23291630 301 RTGYDNREIVMKYIHYKLSQRGYEWDAGSEVVHLTLRQAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGP 4lxk A 2.05 BS01 1YT A 1 Q12 G13 L30 D32 G34 S35 P70 Y71 T72 Q73 F108 I126 Y198 D228 G230 T231 Q15 G16 L33 D35 G37 S38 P73 Y74 T75 Q76 F111 I129 Y189 D219 G221 T222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.004uM remove_due_to_license_issue P56817 23981898 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4lxm A 2.3 BS01 1YU A 1 Q12 G13 L30 D32 G34 S35 P70 Y71 T72 F108 Y198 D228 G230 Q15 G16 L33 D35 G37 S38 P73 Y74 T75 F111 Y190 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.088uM remove_due_to_license_issue P56817 23981898 501 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4lxz A 1.85 BS03 SHH A 1 P34 D104 H145 H146 F155 D181 H183 Y308 P23 D93 H134 H135 F144 D170 H172 Y297 3.5.1.-,3.5.1.98 0004407 Kd=0.182uM remove_due_to_license_issue IC50=921nM, Kd=182nM, Ki=40nM Q92769 23897821 407 GKKKVCYYYDGDIGNYYYGQGHPMKPHRIRMTHNLLLNYGLYRKMEIYRPHKATAEEMTKYHSDEYIKFLRSIRPDNMSEYSKQMQRFNVGEDCPVFDGLFEFCQLSTGGSVAGAVKLNRQQTDMAVNWAGGLHHAKKSEASGFCYVNDIVLAILELLKYHQRVLYIDIDIHHGDGVEEAFYTTDRVMTVSFHKYGEYFPGTGDLRDIGAGKGKYYAVNFPMRDGIDDESYGQIFKPIISKVMEMYQPSAVVLQCGADSLSGDRLGCFNLTVKGHAKCVEVVKTFNLPLLMLGGGGYTIRNVARCWTYETAVALDCEIPNELPYNDYFEYFGPDFKLHISPSNMTNQNTPEYMEKIKQRLFENLRMLP 4ly1 A 1.57 BS03 20Y A 1 Y29 M35 L144 H145 H146 G154 F155 C156 D181 H183 F210 L276 G305 G306 Y308 Y18 M24 L133 H134 H135 G143 F144 C145 D170 H172 F199 L265 G294 G295 Y297 3.5.1.-,3.5.1.98 0004407 Kd=0.0552uM remove_due_to_license_issue IC50=100nM, Ki=1.5nM, Kd=55.2nM Q92769 23897821 407 GKKKVCYYYDGDIGNYYYGQGHPMKPHRIRMTHNLLLNYGLYRKMEIYRPHKATAEEMTKYHSDEYIKFLRSIRPDNMSEYSKQMQRFNVGEDCPVFDGLFEFCQLSTGGSVAGAVKLNRQQTDMAVNWAGGLHHAKKSEASGFCYVNDIVLAILELLKYHQRVLYIDIDIHHGDGVEEAFYTTDRVMTVSFHKYGEYFPGTGDLRDIGAGKGKYYAVNFPMRDGIDDESYGQIFKPIISKVMEMYQPSAVVLQCGADSLSGDRLGCFNLTVKGHAKCVEVVKTFNLPLLMLGGGGYTIRNVARCWTYETAVALDCEIPNELPYNDYFEYFGPDFKLHISPSNMTNQNTPEYMEKIKQRLFENLRMLP 4ly9 A 2.35 BS02 1YY A 1 V10 I11 Y24 V28 P29 E32 R215 H504 A521 R525 V10 I11 Y24 V28 P29 E32 R213 H483 A500 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 Kd=0.007uM remove_due_to_license_issue IC50=21nM Q14397 24226772 714 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4lyn A 2.0 BS01 1YG A 1 I10 V18 A31 K33 F80 F82 L83 Q85 D86 K89 L134 D145 I10 V18 A31 K33 F80 F82 L83 Q85 D86 K89 L134 D145 D127 K129 Q131 N132 D145 T165 D127 K129 Q131 N132 D145 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=60nM P24941 12190313 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4lys A 1.83 BS01 2SJ A 1 W81 P82 F83 L92 N140 I146 W39 P40 F41 L50 N98 I104 ? remove_due_to_license_issue O60885 24272870 203 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4lyw A 1.95 BS01 21Q A 1 W81 P82 F83 V87 L92 N140 W40 P41 F42 V46 L51 N99 ? Kd=237nM remove_due_to_license_issue Kd=240nM O60885 24272870 1001 AMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4lzr A 1.85 BS01 LOC A 1 W81 F83 V87 L92 L94 N140 I146 W40 F42 V46 L51 L53 N99 I105 ? Kd=20uM remove_due_to_license_issue O60885 24272870 201 AMNPPPPETSNPNKPKRQTNQLEYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLEDNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALESLFLQKINELPTEE 4lzs A 2.2 BS01 L46 A 1 P82 F83 V87 L92 N140 I146 P41 F42 V46 L51 N99 I105 ? Kd=16uM remove_due_to_license_issue Kd=6800nM O60885 24272870 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4m0e A 2.0 BS01 1YL A 1 Y72 Y124 W286 V294 F295 Y337 F338 Y341 Y69 Y121 W278 V286 F287 Y329 F330 Y333 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G118 G119 G151 S200 A201 G239 F289 F291 E326 H439 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 Ki=0.7uM remove_due_to_license_issue Ki=600nM, IC50=1000nM P22303 24900610 604 EDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSA 4m0f A 2.304 BS01 1YK A 1 W86 Y124 W286 Y337 F338 Y341 H447 W83 Y121 W277 Y328 F329 Y332 H438 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G118 G119 G151 S200 A201 G239 F288 F290 E325 H438 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 Ki=1.7nM remove_due_to_license_issue Ki=1.7nM, IC50=8nM P22303 24900610 604 EDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSA 4m0r A 1.96 BS01 644 A 1 N138 A179 H183 Y186 R187 A190 R193 R194 G206 N111 A152 H156 Y159 R160 A163 R166 R167 G179 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 Ki=6.2uM remove_due_to_license_issue P9WFX5 24623674 600 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQ 4m0y A 1.7 BS01 M0Y A 1 G370 S371 G372 V377 A389 F437 M438 E439 G441 C442 L489 G15 S16 G17 V22 A34 F82 M83 E84 G86 C87 L134 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=0.35uM remove_due_to_license_issue Q08881 24593284 701 WVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4m0y A 1.7 BS02 M0Y A 2 F403 A407 M410 M411 V419 L421 F435 S499 D500 F501 F506 F48 A52 M55 M56 V64 L66 F80 S144 D145 F146 F151 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=0.35uM remove_due_to_license_issue Q08881 24593284 702 WVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4m0z A 2.0 BS01 M0Z A 1 F403 E406 A407 M410 V419 L421 F435 S499 D500 F501 F506 F49 E52 A53 M56 V65 L67 F81 S145 D146 F147 F152 D482 A484 R486 N487 D500 P521 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=6.4uM remove_due_to_license_issue Q08881 24593284 701 KWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4m0z A 2.0 BS02 M0Z A 2 I369 G370 A389 K391 E436 F437 M438 G441 L489 I15 G16 A35 K37 E82 F83 M84 G87 L135 D482 A484 R486 N487 D500 P521 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=6.4uM remove_due_to_license_issue Q08881 24593284 702 KWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4m12 A 2.15 BS01 1YZ A 1 F403 E406 A407 M410 L413 V419 L421 F435 S499 D500 F501 F506 F49 E52 A53 M56 L59 V65 L67 F81 S145 D146 F147 F152 D482 A484 R486 N487 D500 P521 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=0.9uM remove_due_to_license_issue Q08881 24593284 701 KWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4m13 A 1.85 BS01 1E0 A 1 F403 A407 M410 V419 Q420 L421 G423 V424 F435 S499 D500 F501 F506 F49 A53 M56 V65 Q66 L67 G69 V70 F81 S145 D146 F147 F152 D482 A484 R486 N487 D500 P521 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Kd=0.2uM remove_due_to_license_issue Q08881 24593284 701 KWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAES 4m14 A 1.55 BS01 QWS A 1 I369 A389 K391 E436 F437 M438 G441 L489 I15 A35 K37 E82 F83 M84 G87 L135 D482 A484 R486 N487 D500 P521 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Q08881 24593284 701 KWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAE 4m14 A 1.55 BS02 QWS A 2 F403 E406 A407 M410 M411 V419 L421 F435 S499 D500 F501 F506 F49 E52 A53 M56 M57 V65 L67 F81 S145 D146 F147 F152 D482 A484 R486 N487 D500 P521 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Q08881 24593284 702 KWVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTRFVLDDQYTSSTGTKFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWRERPEDRPAFSRLLRQLAEIAE 4m1j C 1.8 BS01 B0S C 1 S217 H239 F240 V286 V374 W378 N485 S1 H23 F24 V70 V158 W162 N269 S217 S1 3.5.1.97 0016787,0017000 remove_due_to_license_issue Q9I194 23883096 801 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIREAA 4m2r A 1.993 BS02 BZ1 A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.2nM remove_due_to_license_issue Ki=3nM, IC50=3.2nM, Kd=0.13nM P00918 24090602 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4m2u A 1.999 BS02 ETS A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=9.1nM remove_due_to_license_issue Ki=9nM, IC50=26.61nM, Kd=0.043000nM P00918 24090602 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4m2v A 1.718 BS02 BZ1 A 1 H94 H119 V121 L198 T199 T200 H91 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=3nM, IC50=3.2nM, Kd=0.13nM P00918 24090602 302 HWGYGAHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4m2w A 1.658 BS02 ETS A 1 H94 H119 V121 L198 T199 T200 H91 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=9nM, IC50=26.61nM, Kd=0.043000nM P00918 24090602 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4m3b A 2.001 BS01 2B2 A 1 M102 W103 G106 I107 F110 W138 Y148 T149 N176 N179 E180 W207 M73 W74 G77 I78 F81 W109 Y119 T120 N147 N150 E151 W178 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.4uM remove_due_to_license_issue P9WMC1 24818704 301 RELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAEDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 4m3d A 1.9 BS01 2H2 A 1 M102 W103 G106 I107 F110 Y148 T149 V152 N176 N179 E180 W207 M80 W81 G84 I85 F88 Y126 T127 V130 N154 N157 E158 W185 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=3.9uM remove_due_to_license_issue P9WMC1 24818704 301 DDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 4m3e A 2.109 BS01 2B3 A 1 L90 P94 M102 W103 I107 F110 W138 M142 W145 Y148 N176 N179 E180 W207 L69 P73 M81 W82 I86 F89 W117 M121 W124 Y127 N155 N158 E159 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.56uM remove_due_to_license_issue P9WMC1 24818704 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 4m3f A 2.0 BS01 2D1 A 1 M102 W103 G106 I107 F110 W138 M142 Y148 T149 N176 N179 W207 M81 W82 G85 I86 F89 W117 M121 Y127 T128 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=4.9uM remove_due_to_license_issue P9WMC1 24818704 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 4m3g A 2.3 BS01 2G1 A 1 M102 W103 G106 F110 M142 W145 Y148 T149 N176 N179 E180 W207 M79 W80 G83 F87 M119 W122 Y125 T126 N153 N156 E157 W184 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.55uM remove_due_to_license_issue P9WMC1 24818704 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 4m3m A 2.1 BS01 22N A 1 D151 R224 A246 E276 E277 R292 Y347 R371 Y406 D70 R144 A166 E196 E197 R212 Y265 R289 Y323 D151 E277 R292 R371 Y406 D70 E197 R212 R289 Y323 3.2.1.18 0004308,0005975,0016020,0033644,0055036 remove_due_to_license_issue Q07599 24425043 501 GTYMNNTEAICDVKGFAPFSKDNGIRIGSRGHIFVIREPFVSCSPIECRTFFLTQGSLLNDKHSNGTVKDRSPFRTLMSVKVGQSPNVYQARFEAVAWSATACHDGKKWMTVGVTGPDSKAVAVIHYGGVPTDVINSWAGDILRTQESSCTCIQGDCYWVMTDGPANRQAQYRIYKANQGRIIGQADISFNGGHIEECSCYPNDGKVECVCRDNWTGTNRPVLVISPDLSYRVGYLCAGIPSDTPRGEDAQFTGSCTSPMGNQGYGVKGFGFRQGTDVWMGRTISRTSRSGFEILRIKNGWTQTSKEQVRKQVVVDNLNWSGYSGSFTLPVELSGKDCLVPCFWVEMIRGKPEEKTIWTSSSSIVMCGVDYEIADWSWHDGAILPFDIDK 4m3q A 2.718 BS02 24K A 1 L593 G594 A617 M674 M730 L16 G17 A40 M78 M134 D723 A725 R727 N728 D741 D127 A129 R131 N132 D145 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=55nM Q12866 24195762 906 EDVVIDRNLLILGKILGEGEFGSVMEGNLKQEDGTSLKVAVKTCMKDFSHPNVIRLLGVCIEMSSQGIPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFPVKWIAIESLRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESL 4m48 A 2.955 BS03 21B A 1 F43 D46 V120 Y124 F325 S421 G425 F19 D22 V96 Y100 F258 S354 G358 ? 0016020 remove_due_to_license_issue Q7K4Y6 24037379 704 DERETWSGKVDFLLSVIGFAVDLANVWRFPYLCYKNGGGAFLVPYGIMLAVGGIPLFYMELALGQHNRKGAITCWGRLVPLFKGIGYAVVLIAFYVDFYYNVIIAWSLRFFFASFTNSLPWTSCNNIWNTPNCRPFESQGFQSAASEYFNRYILELNRSEGIHDLGAIKWDMALCLLIVYLICYFSLWKGISTSGKVVWFTALFPYAALLILLIRGLTLPGSFLGIQYYLTPNFSAIYKAEVWADAATQVFFSLGPGFGVLLAYASYNKYHNNVYKDALLTSFINSATSFIAGFVIFSVLGYMAHTLGVRIEDVATEGPGLVFVVYPAAIATMPASTFWALIFFMMLATLGLDSSFGGSEAIITALSDEFPKIKRNRELFVAGLFSLYFVVGLASCTQGGFYFFHLLDRYAAGYSILVAVFFEAIAVSWIYGTNRFSEDIRDMIGFPPGRYWQVCWRFVAPIFLLFITVYLLIGYEPLTYADYVYPSWANALGWCIAGSSVVMIPAVAIFKLLSTPGSLRQRFTILTTPWRD 4m4q A 2.502 BS03 21A A 1 A20 K34 A37 I38 H41 E80 D108 E119 K134 A25 K39 A42 I43 H46 E85 D113 E124 K139 0003723,0039694 ic50=0.011uM remove_due_to_license_issue 23978130 304 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4m59 A 2.46 BS01 rna D 0 G431 K432 K537 V597 S604 K608 I632 N635 D639 V668 N671 T672 N675 C678 K679 V703 H706 T707 G710 G711 S714 L738 R742 G347 K348 K453 V513 S520 K524 I548 N551 D555 V584 N587 T588 N591 C594 K595 V619 H622 T623 G626 G627 S630 L654 R658 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 24162847 1 ~ 18 PDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPSVVTYNALLQVFGKAGNYTEALRVLGEMEQNGCQPDAVTYNELAGTEEAARCLDTMASPNAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYGSGAVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAFEEARGFLSEVKALEAYIEDA 4m59 A 2.46 BS02 rna C 0 R175 T178 H182 V210 N213 R221 G245 F246 S249 T250 V281 N284 A285 Q288 V316 N319 E320 R102 T105 H109 V137 N140 R148 G172 F173 S176 T177 V208 N211 A212 Q215 V243 N246 E247 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 24162847 1 ~ 18 PDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPSVVTYNALLQVFGKAGNYTEALRVLGEMEQNGCQPDAVTYNELAGTEEAARCLDTMASPNAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYGSGAVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAFEEARGFLSEVKALEAYIEDA 4m59 B 2.46 BS01 rna D 0 E151 R175 H182 V210 N213 V214 F246 S249 T250 V281 N284 A285 E80 R104 H111 V139 N142 V143 F175 S178 T179 V210 N213 A214 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 24162847 1 ~ 18 LSPDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPSVVTYNALLQVFGKAEALRVLGEMEQNGPDAVTYNELAGTYARAGFFEEAARCLDTMAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAKRFEEARGFLKALEAYIEDAQF 4m59 B 2.46 BS02 rna C 0 R565 N600 I632 N635 D639 N671 T672 N675 C678 K679 H706 G710 G711 S714 R742 R476 N511 I543 N546 D550 N582 T583 N586 C589 K590 H617 G621 G622 S625 R653 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 24162847 1 ~ 18 LSPDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPSVVTYNALLQVFGKAEALRVLGEMEQNGPDAVTYNELAGTYARAGFFEEAARCLDTMAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAKRFEEARGFLKALEAYIEDAQF 4m5g A 1.31 BS02 YH1 A 1 T42 P43 L45 Y53 N55 W89 R121 F123 T43 P44 L46 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=9.7uM remove_due_to_license_issue P26281 24613625 302 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5h A 1.11 BS02 YH2 A 1 T42 P43 L45 G46 Y53 N55 W89 R121 F123 T43 P44 L46 G47 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=29uM remove_due_to_license_issue P26281 24613625 302 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5i A 1.08 BS05 YH6 A 1 T42 P43 L45 Y53 N55 W89 R121 F123 T43 P44 L46 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=6.7uM remove_due_to_license_issue IC50=64000nM, Kd=6700nM P26281 24613625 205 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5j A 1.696 BS02 YH5 A 1 T42 P43 P44 L45 Y53 N55 W89 R92 R121 F123 T43 P44 P45 L46 Y54 N56 W88 R91 R120 F122 R82 R92 D95 D97 R83 R91 D94 D96 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=14.5uM remove_due_to_license_issue IC50=44000nM, Kd=14500nM P26281 24613625 302 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5k A 1.296 BS05 YH3 A 1 T42 P43 L45 Y53 N55 W89 D117 R121 F123 T43 P44 L46 Y54 N56 W90 D118 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=5.9uM remove_due_to_license_issue P26281 24613625 305 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5l A 1.094 BS05 YH4 A 1 T42 P43 L45 Y53 N55 W89 R121 F123 T43 P44 L46 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=18.9uM remove_due_to_license_issue Kd=18900nM, IC50=243000nM P26281 24613625 306 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5m A 1.118 BS01 DX4 A 1 L45 Y53 N55 F123 L46 Y54 N56 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=18uM remove_due_to_license_issue P26281 24613625 401 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5n A 2.0 BS04 YH7 A 1 T42 P44 L45 Y53 N55 D95 F123 T44 P46 L47 Y55 N57 D97 F125 R82 R92 D95 D97 R84 R94 D97 D99 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=7.5uM remove_due_to_license_issue P26281 24613625 504 HMTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 4m5o A 2.0 BS03 X48 A 1 K34 I38 H41 E80 D108 E119 K134 K39 I43 H46 E85 D113 E124 K139 0003723,0039694 ic50=0.38uM remove_due_to_license_issue 23978130 306 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4m5o A 2.0 BS04 X48 A 2 K19 E23 Y24 G81 R82 D83 K24 E28 Y29 G86 R87 D88 0003723,0039694 ic50=0.38uM remove_due_to_license_issue 23978130 307 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4m5o A 2.0 BS05 X48 A 3 Y24 E26 E80 Y29 E31 E85 0003723,0039694 ic50=0.38uM remove_due_to_license_issue 23978130 308 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4m5r A 1.4 BS02 MSR A 1 L16 K19 A20 E23 E80 G81 R82 D83 L21 K24 A25 E28 E85 G86 R87 D88 0003723,0039694 ic50=1000uM remove_due_to_license_issue 23978130 304 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 4m5r A 1.4 BS03 MSR A 2 Y24 E26 K34 Y29 E31 K39 0003723,0039694 ic50=1000uM remove_due_to_license_issue 23978130 306 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 4m5u A 2.2 BS03 20F A 1 A20 K34 A37 I38 H41 E80 D108 E119 K134 A25 K39 A42 I43 H46 E85 D113 E124 K139 0003723,0039694 ic50=0.023uM remove_due_to_license_issue 24055080 305 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4m6p A 1.75 BS01 20R A 1 H191 F193 R196 D219 V242 A244 S275 R311 I351 H175 F177 R180 D203 V226 A228 S259 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.054uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4m6p A 1.75 BS02 20R B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.054uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4m6p B 1.75 BS01 20R B 1 H191 F193 R196 D219 V242 A244 R311 I351 H174 F176 R179 D202 V225 A227 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.054uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4m6q A 2.406 BS01 20T A 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 I309 R311 D313 I351 G353 G383 G384 Y172 H175 F177 R180 D203 Y224 S225 V226 A228 I293 R295 D297 I335 G337 G367 G368 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.0061uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4m6q A 2.406 BS03 20T B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.0061uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4m6q B 2.406 BS01 20T A 1 Y18 R392 Y11 R376 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.0061uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4m6q B 2.406 BS02 20T B 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 S275 I309 R311 I351 G353 G383 G384 Y172 H175 F177 R180 D203 Y224 S225 V226 A228 S259 I293 R295 I335 G337 G367 G368 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.0061uM remove_due_to_license_issue P43490 24021463 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4m6u A 1.8 BS02 TTN A 1 K164 K166 D195 E247 H297 E317 K162 K164 D193 E245 H295 E315 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 remove_due_to_license_issue P11444 24472022 402 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 4m6u B 1.8 BS02 TTN B 1 K164 K166 D195 E247 H297 E317 K162 K164 D193 E245 H295 E315 V22 S139 K164 K166 D195 N197 E221 G246 E247 D270 M294 H297 L298 F299 A313 E317 V20 S137 K162 K164 D193 N195 E219 G244 E245 D268 M292 H295 L296 F297 A311 E315 5.1.2.2 0000287,0009063,0016052,0016836,0016853,0018838,0018924,0019596,0046872 remove_due_to_license_issue P11444 24472022 402 EVLITGLRTRAVNVPLAYPVHTAVGTVGTAPLVLIDLATSAGVVGHSYLFAYTPVALKSLKQLLDDMAAMIVNEPLAPVSLEAMLAKRFCLAGYTGLIRMAAAGIDMAAWDALGKVHETPLVKLLGANARPVQAYDSHSLDGVKLATERAVTAAELGFRAVKTKIGYPALDQDLAVVRSIRQAVGDDFGIMVDYNQSLDVPAAIKRSQALQQEGVTWIEEPTLQHDYEGHQRIQSKLNVPVQMGENWLGPEEMFKALSIGACRLAMPDAMKIGGVTGWIRASALAQQFGIPMSSHLFQEISAHLLAATPTAHWLERLDLAGSVIEPTLTFEGGNAVIPDLPGVGIIWREKEIGKYLV 4m7b A 1.95 BS02 28C A 1 G1032 F1035 Y1050 Y1060 S1068 Y1071 I1075 G81 F84 Y99 Y109 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=200nM remove_due_to_license_issue IC50=200nM Q9H2K2 24527792 1202 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4m7j H 1.95 BS01 KDA A 1 W52 S53 G54 S56 W52 S53 G54 S56 remove_due_to_license_issue 24682362 1 EVQLKESGPGLVQPSQSLSITCTVSGFSLTTYGVHWVRQSPGKGLEWLGVIWSGGSTDYNAAFISRLSISKDNSKSHVFFKMNSLQANDTAIYYCARMRITTDWFAYWGQGTLVTVSAAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRD 4m7x A 1.42 BS02 27Q A 1 E70 G100 R113 G116 I117 E70 G100 R113 G116 I117 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q8NVG0 27759386 315 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLEKHHHHHH 4m7y A 1.8 BS01 2GH A 1 F71 T99 G100 T101 R113 G116 I117 F71 T99 G100 T101 R113 G116 I117 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q8NVG0 27759386 301 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLE 4m7y A 1.8 BS03 2GH B 1 T172 A173 E202 Y240 T172 A173 E202 Y240 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q8NVG0 27759386 301 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLE 4m7y B 1.8 BS01 2GH A 1 T172 A173 E202 Y240 T172 A173 E202 Y240 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q8NVG0 27759386 301 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLE 4m7y B 1.8 BS02 2GH B 1 F71 T99 G100 R113 G116 F71 T99 G100 R113 G116 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q8NVG0 27759386 301 MKVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLE 4m84 A 1.998 BS01 21E A 1 L57 G58 V65 A78 K80 M112 L126 L181 L14 G15 V22 A35 K37 M69 L83 L138 D174 K176 E178 N179 D195 T214 D131 K133 E135 N136 D152 T171 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 ic50=0.049uM remove_due_to_license_issue IC50=49.0nM Q9BJF5 24494061 601 TAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 4m8b R 2.61 BS01 dna A 0 R62 W63 S72 L79 V181 G182 N183 R62 W63 S72 L79 V173 G174 N175 ? remove_due_to_license_issue P38867 24994900 1 ~ 20 SSPGPTCYGYIDDEQDLALVFQGVFNGNLRCIERRPYDAEKVELVNPGNIFVFNEEKSGIKRWTDGFSWSPSRISGKFLVYREYNRLGSHNVPEYNIFERAHRKYFYTGLLKKTFSLKFNMTDSTKLETFHLIAYYTEKDIHQGSLRRPSENPFFHKFRPSQKLLDALQKVAVGNGRSNPS 4m8b R 2.61 BS02 dna B 0 R35 K61 R62 R73 R185 N187 P188 R35 K61 R62 R73 R177 N179 P180 ? remove_due_to_license_issue P38867 24994900 2 ~ 21 SSPGPTCYGYIDDEQDLALVFQGVFNGNLRCIERRPYDAEKVELVNPGNIFVFNEEKSGIKRWTDGFSWSPSRISGKFLVYREYNRLGSHNVPEYNIFERAHRKYFYTGLLKKTFSLKFNMTDSTKLETFHLIAYYTEKDIHQGSLRRPSENPFFHKFRPSQKLLDALQKVAVGNGRSNPS 4m8e A 2.4 BS02 29V A 1 I268 A271 A272 Q275 W305 F313 R316 V342 C432 I24 A27 A28 Q31 W61 F69 R72 V98 C188 ? 0003677,0003707,0005634,0006355,0008270 Kd=13nM remove_due_to_license_issue P19793 24359708 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4m8h A 2.2 BS02 R4M A 1 I268 A271 A272 Q275 F313 R316 A327 C432 I24 A27 A28 Q31 F69 R72 A83 C188 ? 0003677,0003707,0005634,0006355,0008270 Kd=25nM remove_due_to_license_issue P19793 24359708 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4m8t A 3.0 BS01 RMM A 1 I428 V430 C436 A449 K451 I477 E494 L495 M496 D561 I19 V21 C27 A40 K42 I68 E85 L86 M87 D152 D539 K541 N544 D561 T581 D130 K132 N135 D152 T172 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P18654 25344815 801 QLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVMELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNR 4m8x A 2.05 BS01 KGQ B 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90JJ9 24371077 101 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8x A 2.05 BS02 KGQ B 2 D25 G27 A28 D30 I32 G48 P81 D25 G27 A28 D30 I32 G48 P81 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90JJ9 24371077 102 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8x B 2.05 BS01 KGQ B 1 D25 G27 A28 D30 I32 G48 P81 I84 D25 G27 A28 D30 I32 G48 P81 I84 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.063nM remove_due_to_license_issue Q90JJ9 24371077 101 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8x B 2.05 BS02 KGQ B 2 D25 A28 D29 G48 G49 D25 A28 D29 G48 G49 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.063nM remove_due_to_license_issue Q90JJ9 24371077 102 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8y A 2.22 BS01 KGQ A 1 D25 G27 D29 V48 G49 G50 I51 I85 D25 G27 D29 V48 G49 G50 I51 I85 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.11nM remove_due_to_license_issue Q90JJ9 24371077 201 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8y A 2.22 BS02 KGQ A 2 D25 G27 A28 D30 V48 G49 G50 P82 D25 G27 A28 D30 V48 G49 G50 P82 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 Ki=0.11nM remove_due_to_license_issue Q90JJ9 24371077 202 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8y B 2.22 BS01 KGQ A 1 D25 G27 A28 D30 V48 G49 P82 I85 D25 G27 A28 D30 V48 G49 P82 I85 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90JJ9 24371077 201 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m8y B 2.22 BS02 KGQ A 2 D25 G27 D29 V48 G49 G50 D25 G27 D29 V48 G49 G50 D25 T26 G27 D25 T26 G27 3.1.26.13 0004190,0006508 remove_due_to_license_issue Q90JJ9 24371077 202 PQITLWQRPFVTVKIAGQLMEALLDTGADDTILEEEMSLPGRWTPKVVGGIGGFMKVRQYDQILVEICGHKVIGTVLVGPTPANIIGRNLLTQIGCTLNF 4m9e A 1.851 BS01 dna B 0 Y411 K413 H416 R443 E446 R449 R471 H474 Y13 K15 H18 R45 E48 R51 R73 H76 ? remove_due_to_license_issue Q60793 24520114 1 ~ 10 THTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDELTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 4m9e A 1.851 BS02 dna C 0 K413 S415 Y430 S472 D473 K15 S17 Y32 S74 D75 ? remove_due_to_license_issue Q60793 24520114 1 ~ 10 THTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDELTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 4m9v C 0.969 BS01 dna A 0 S156 R157 R159 R160 D179 Q180 S181 Q182 S22 R23 R25 R26 D45 Q46 S47 Q48 ? remove_due_to_license_issue Q8C6P8 24236546 1 ~ 11 PSERPFFCNFCGKTYRDASGLSRHRRAHLGYRPRSCPECGKCFRDQSQVNRHLKVHQNKP 4m9v C 0.969 BS02 dna B 0 R138 K147 Y149 R150 D151 S153 R166 K175 R178 Q182 R185 V189 R4 K13 Y15 R16 D17 S19 R32 K41 R44 Q48 R51 V55 ? remove_due_to_license_issue Q8C6P8 24236546 1 ~ 11 PSERPFFCNFCGKTYRDASGLSRHRRAHLGYRPRSCPECGKCFRDQSQVNRHLKVHQNKP 4m9v F 0.969 BS01 dna D 0 S156 R157 R159 R160 S181 Q182 S22 R23 R25 R26 S47 Q48 ? remove_due_to_license_issue Q8C6P8 24236546 1 ~ 11 PSERPFFCNFCGKTYRDASGLSRHRRAHLGYRPRSCPECGKCFRDQSQVNRHLKVHQNKP 4m9v F 0.969 BS02 dna E 0 R138 Y149 R150 D151 S153 R166 K175 R178 Q182 R185 H186 V189 R4 Y15 R16 D17 S19 R32 K41 R44 Q48 R51 H52 V55 ? remove_due_to_license_issue Q8C6P8 24236546 1 ~ 11 PSERPFFCNFCGKTYRDASGLSRHRRAHLGYRPRSCPECGKCFRDQSQVNRHLKVHQNKP 4man A 2.07 BS01 1Y1 A 1 A97 D100 F101 Y105 F109 M112 L134 W141 G142 A146 Y199 A32 D35 F36 Y40 F44 M47 L69 W76 G77 A81 Y134 ? 0042981,0043066 remove_due_to_license_issue Ki=<0.100000nM P10415 23291630 301 GYDNREIVMKYIHYKLSQRGYEEVVHLTLRQAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGP 4mao A 2.6 BS01 28D A 1 I428 V430 C436 A449 K451 I477 M493 E494 M496 N544 L546 C560 D561 I14 V16 C22 A35 K37 I63 M79 E80 M82 N130 L132 C146 D147 D539 K541 N544 D561 T581 D125 K127 N130 D147 T167 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P18654 25153195 801 SIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVMELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNR 4mb9 A 1.85 BS01 28F A 1 I48 N51 E55 V76 D78 R81 M83 P84 R140 T172 I32 N35 E39 V60 D62 R65 M67 P68 R112 T144 0003677,0003918,0005524,0006265 remove_due_to_license_issue 24088190 302 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHAGGLHGVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4mbc A 1.75 BS01 28G A 1 I48 N51 A52 E55 V76 D78 R81 M83 P84 R140 T172 I32 N35 A36 E39 V60 D62 R65 M67 P68 R107 T139 0003677,0003918,0005524,0006265 remove_due_to_license_issue 24088190 301 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHAVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4mbf A 1.54 BS03 2AW A 1 S70 Y105 N132 N170 T235 G236 A237 R244 S45 Y80 N107 N145 T210 G211 A212 R218 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 24454944 303 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 4mbf A 1.54 BS04 2AW A 2 V224 P226 A227 V199 P201 A202 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 24454944 304 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 4mbi A 2.3 BS01 26K A 1 L44 F49 A65 L120 L174 I185 D186 L12 F17 A33 L88 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=7.0nM P11309 24091081 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4mbj A 3.6 BS01 DFS A 1 V471 A481 K483 L505 L514 I527 W531 C532 G593 D594 G596 L597 V24 A34 K36 L58 L67 I80 W84 C85 G146 D147 G149 L150 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 24042006 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 4mbl A 2.6 BS01 26L A 1 L44 F49 A65 K67 D128 L174 D186 L12 F17 A33 K35 D96 L142 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=2.9nM P11309 24091081 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4mc1 A 1.39 BS01 526 A 1 D25 G27 A28 D29 D30 I84 D25 G27 A28 D29 D30 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc1 A 1.39 BS02 526 B 1 D25 G27 A28 D30 I50 D25 G27 A28 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc1 B 1.39 BS01 526 A 1 D25 G27 A28 D30 G49 I50 D25 G27 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc1 B 1.39 BS02 526 B 1 D25 G27 A28 D29 D30 G48 G49 P81 V82 I84 D25 G27 A28 D29 D30 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc2 A 1.56 BS01 525 A 1 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc2 A 1.56 BS02 525 B 1 R8 D25 G27 A28 D30 I50 R8 D25 G27 A28 D30 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc2 B 1.56 BS01 525 A 1 D25 G27 A28 D30 G49 I50 D25 G27 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc2 B 1.56 BS02 525 B 1 D25 A28 D29 D30 G48 P81 V82 I84 D25 A28 D29 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc6 A 1.31 BS01 23K A 1 R8 L23 D25 G27 G49 I50 R8 L23 D25 G27 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc6 B 1.31 BS01 23K A 1 D25 G27 A28 D29 D30 I47 P81 V82 I84 D25 G27 A28 D29 D30 I47 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc9 A 1.19 BS01 23L A 1 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc9 A 1.19 BS02 23L B 1 R8 D25 G27 A28 D30 G49 I50 R8 D25 G27 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc9 B 1.19 BS01 23L A 1 R8 D25 G27 A28 D30 G49 I50 R8 D25 G27 A28 D30 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mc9 B 1.19 BS02 23L B 1 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 G27 A28 D29 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4mcb A 1.94 BS01 21W A 1 L87 S88 P89 E116 S132 I133 Y136 L138 G140 G141 P144 L87 S88 P89 E116 S132 I133 Y136 L138 G140 G141 P144 P89 E116 R154 P89 E116 R154 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 ic50=1.5uM remove_due_to_license_issue P43912 23981144 303 MWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLGLLDCPHYTRPEVLEGLTVPPVLMSHHEEIRKWRLKQSLQRTWLR 4mcb B 1.94 BS01 21W A 1 D169 A172 D173 D169 A172 D173 P89 E116 R154 D169 P89 E116 R154 D169 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 ic50=1.5uM remove_due_to_license_issue P43912 23981144 303 MWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLGKQASAEEDSFADGLLDCPHYTRPEVLEGLTVPPVLMSGHHEEIRKWRLKQSLQRTWLRRPELLEGLALTDEQRKLLKEAQAE 4mcb B 1.94 BS02 21W B 1 L87 S88 P89 E116 S132 Y136 L138 G140 G141 P144 L87 S88 P89 E116 S132 Y136 L138 G140 G141 P144 P89 E116 R154 D169 P89 E116 R154 D169 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 ic50=1.5uM remove_due_to_license_issue P43912 23981144 303 MWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLGKQASAEEDSFADGLLDCPHYTRPEVLEGLTVPPVLMSGHHEEIRKWRLKQSLQRTWLRRPELLEGLALTDEQRKLLKEAQAE 4mcc A 1.95 BS01 21X A 1 L87 S88 P89 E116 S132 I133 Y136 L138 G140 P144 L87 S88 P89 E116 S132 I133 Y136 L138 G140 P144 P89 E116 R154 P89 E116 R154 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 ic50=0.56uM remove_due_to_license_issue P43912 23981144 301 MWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLGLLDCPHYTRPEVLEGLTVPPVLMSGHHEEIRKWRLKQSLQRTWLR 4mcc B 1.95 BS01 21X B 1 L87 S88 P89 S132 Y136 V137 L138 G140 G141 P144 L87 S88 P89 S132 Y136 V137 L138 G140 G141 P144 P89 E116 R154 P89 E116 R154 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 ic50=0.56uM remove_due_to_license_issue P43912 23981144 301 MWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLDGLLDCPHYTRPEVLEGLTVPPVLMSGHHEEIRKWRLKQSLQRTWLRRPELLEGLALTDEQRKLLKEAQAEHN 4mcd A 1.55 BS01 22L A 1 L87 S88 P89 S132 I133 Y136 L138 G140 P144 L87 S88 P89 S132 I133 Y136 L138 G140 P144 P89 E116 R154 P89 E116 R154 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 ic50=4.7uM remove_due_to_license_issue P43912 23981144 301 MWIGVISLFPEMFKAITEFGVTGRAVKHNLLKVECWNPRDFTFDKHKTVDDRPYGGGPGMLMMVQPLRDAIHTAKAAAGEGAKVIYLSPQGRKLDQGGVTELAQNQKLILVCGRYEGIDERLIQTEIDEEWSIGDYVLTGGELPAMTLIDAVARFIPGVLSFADGLLDCPHYTRPEVLEGLTVPPVLMSGHHEEIRKWRLKQSLQRTWLRRPELLEGLALTDEQRKLLKEAQAEHNS 4mcv A 2.73 BS01 29K A 1 L273 V281 A293 K295 G338 E339 Y340 M341 G344 A390 N391 L393 L18 V26 A38 K40 G83 E84 Y85 M86 G89 A135 N136 L138 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F158 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 24171479 601 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVGEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4md6 A 2.0 BS01 24E A 1 L725 A767 I768 V782 A783 F787 I813 M816 Q817 F820 L181 A223 I224 V238 A239 F243 I252 M255 Q256 F259 3.1.4.35 0004114,0007165,0008081 ic50=17nM remove_due_to_license_issue IC50=17nM O76074 24565909 902 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGEKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 4mdn A 1.905 BS01 Y30 A 1 E23 M50 L54 G58 I61 V93 H96 Y100 E7 M34 L38 G42 I45 V77 H80 Y84 2.3.2.27 0005634,0043066,0051726 Ki=0.6uM remove_due_to_license_issue Ki=600nM Q00987 24207125 201 MQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4mdq A 2.119 BS01 28W A 1 L54 G58 F91 V93 H96 L30 G34 F67 V69 H72 2.3.2.27 0005634,0043066,0051726 Ki=1.2uM remove_due_to_license_issue Ki=1200nM Q00987 24207125 201 ETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4mdq A 2.119 BS02 28W A 2 M50 K51 R97 Y100 M26 K27 R73 Y76 2.3.2.27 0005634,0043066,0051726 Ki=1.2uM remove_due_to_license_issue Ki=1200nM Q00987 24207125 202 ETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4mds A 1.598 BS01 23H A 1 H41 M49 F140 L141 C145 H163 M165 E166 Q189 H41 M49 F140 L141 C145 H163 M165 E166 Q189 H41 G143 C145 H41 G143 C145 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0008233,0019082 ic50=6.2uM remove_due_to_license_issue P0C6U8 24080461 401 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDRQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGA 4mdt A 2.59 BS02 24G A 1 L62 K143 I159 D160 F161 F192 M195 I198 G210 S211 K239 K262 H265 L62 K143 I159 D160 F161 F192 M195 I198 G210 S211 K239 K262 H265 0009245,0103117 remove_due_to_license_issue 24108127 402 MIKQRTLKRIVQATGVGLHTGKKVTLTLRPAPANTGVIYRRTDLNPPVDFPADAKSVRDTMLCTCLVNEHDVRISTVEHLNAALAGLGIDNIVIEVNAPEIPIMDGSAAPFVYLLLDAGIDELNSAKKFVRIKETVRVEDGDKWAEFKPYNGFSLDFTIDFNHPAIDSSNQRYAMNFSADAFMRQISRARTFGFMRDIEYLQSRGLCLGGSFDCAIVVDDYRVLNEDGLRFEDEFVRHKMLDAIGDLFMCGHNIIGAFTAYKSGHALNNKLLQAVLAKQEAWEYVTFQDDAELPLAFKAP 4mdx A 1.5 BS01 rna C 0 N32 I34 G35 F38 S39 P40 N33 I35 G36 F39 S40 P41 3.1.27.- 0003677,0003723,0004519,0004521,0006402,0016075 remove_due_to_license_issue P96622 24120662 1 ~ 9 SMIVKRGDVYFADLSPVVGSEQGGVRPVLVIQNDIGNRFSPTAIVAAITAQIQKAKLPTHVEIDAKRYGFERDSVILLEQIRTIDKQRLTDKITHLDDEMMDKVDEALQISLALI 4mdx B 1.5 BS01 rna C 0 F10 S19 E20 Q21 G22 V24 R25 P26 T48 A49 Q50 K53 L56 P57 H59 F69 E70 S73 E78 Q79 D90 F11 S20 E21 Q22 G23 V25 R26 P27 T49 A50 Q51 K54 L57 P58 H60 F70 E71 S74 E79 Q80 D91 3.1.27.- 0003677,0003723,0004519,0004521,0006402,0016075 remove_due_to_license_issue P96622 24120662 1 ~ 9 SMIVKRGDVYFADLSPVVGSEQGGVRPVLVIQNDIGNRFSPTAIVAAITAQIQKAKLPTHVEIDAKRYGFERDSVILLEQIRTIDKQRLTDKITHLDDEMMDKVDEALQISLALI 4men A 1.81 BS01 25K A 1 W81 P82 F83 L92 L94 N140 W40 P41 F42 L51 L53 N99 ? remove_due_to_license_issue O60885 24090311 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4meo A 1.72 BS01 25V A 1 W81 P82 Q85 V87 D88 L92 L94 N140 I146 W40 P41 Q44 V46 D47 L51 L53 N99 I105 ? remove_due_to_license_issue IC50=42000nM O60885 24090311 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4mep A 1.85 BS01 24Y A 1 W81 P82 F83 Q85 L92 W40 P41 F42 Q44 L51 ? ic50=4.7uM remove_due_to_license_issue O60885 24090311 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4meq A 1.77 BS01 25O A 1 W81 P82 F83 V87 L92 N140 I146 W40 P41 F42 V46 L51 N99 I105 ? remove_due_to_license_issue O60885 24090311 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4mf0 A 2.67 BS01 29Z A 1 A389 K391 F435 F437 M438 G441 L489 S499 A30 K32 F72 F74 M75 G78 L126 S136 D482 A484 R486 N487 D500 P521 D119 A121 R123 N124 D137 P142 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Ki=8.4nM, IC50=10000nM Q08881 24138940 701 VIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4mf0 A 2.67 BS02 29Z B 1 I369 L379 I13 L20 D482 A484 R486 N487 D500 P521 D119 A121 R123 N124 D137 P142 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Ki=8.4nM, IC50=10000nM Q08881 24138940 701 VIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4mf0 B 2.67 BS01 29Z B 1 K387 A389 F435 F437 M438 G441 L489 S499 K28 A30 F72 F74 M75 G78 L126 S136 D482 A484 R486 N487 D500 P521 D119 A121 R123 N124 D137 P139 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Ki=8.4nM, IC50=10000nM Q08881 24138940 701 VIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4mf1 A 2.113 BS01 29Y A 1 I369 A389 K391 F435 F437 M438 E439 G441 L489 S499 I15 A33 K35 F76 F78 M79 E80 G82 L130 S140 D482 A484 R486 N487 D500 P521 D123 A125 R127 N128 D141 P145 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=0.7nM remove_due_to_license_issue Ki=0.600000nM, IC50=91nM Q08881 24138940 701 GSVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEASVIHRDLAARNCLVGENQVIKVSDFGMPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAAIAASG 4mfe A 2.61 BS02 3PY A 1 R548 Q552 G586 L619 R621 V881 T882 R78 Q82 G116 L149 R151 V411 T412 D549 D655 K718 H747 H749 T882 D79 D185 K248 H277 H279 T412 6.4.1.1 0003824 remove_due_to_license_issue Q2K340 24157795 1102 DRATKLLTYLADVTVNGHPEAKDRPKPLENAARPVVPYANGNGVKDGTKQLLDTLGPKKFGEWMRNEKRVLLTDTTMRDGHQSLLATRMRTYDIARIAGTYSHALPNLLSLECWGGATFDVSMRFLTEDPWERLALIREGAPNLLLQMLLRGANGVGYTNYPDNVVKYFVRQAAKGGIDLFRVFDCLNWVENMRVSMDAIAEENKLCEAAICYTGDILNSARPKYDLKYYTNLAVELEKAGAHIIAVKDMAGLLKPAAAKVLFKALREATGLPIHFHTHDTSGIAAATVLAAVEAGVDAVDAAMDALSGNTSQPCLGSIVEALSGSERDPGLDPAWIRRISFYWEAVRNQYAAFESDLKGPASEVYLHEMPGGQFTNLKEQARSLGLETRWHQVAQAYADANQMFGDIVKVTPSSKVVGDMALMMVSQDLTVADVVSPDREVSFPESVVSMLKGDLGQPPSGWPEALQKKALKGEKPYTVRPGSLLKEADLDAERKVIEKKLEREVSDFEFASYLMYPKVFTDFALASDTYGPVSVLPTPAYFYGLADGEELFADIEKGKTLVIVNQAVSATDSQGMVTVFFELNGQPRRIKVPDRA 4mg5 A 2.05 BS02 27E A 1 M343 L346 L384 M388 F404 M421 G521 M39 L42 L80 M84 F100 M117 G215 ? remove_due_to_license_issue P03372 25260197 602 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAH 4mg6 A 2.1 BS02 27G A 1 L346 L349 A350 E353 M388 F404 M421 I424 L428 L42 L45 A46 E49 M84 F100 M111 I114 L118 ? remove_due_to_license_issue P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 4mg7 A 2.15 BS02 27H A 1 L346 L349 A350 E353 M421 L42 L45 A46 E49 M113 ? remove_due_to_license_issue IC50=33nM P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL 4mg8 A 1.85 BS02 27J A 1 L346 A350 E353 L387 M388 L391 M421 G521 L525 L42 A46 E49 L83 M84 L87 M117 G215 L219 ? remove_due_to_license_issue P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 4mg9 A 2.0 BS02 27K A 1 A350 E353 L387 L391 A46 E49 L83 L87 ? remove_due_to_license_issue IC50=1420nM P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 4mga A 1.8 BS02 27L A 1 E353 L391 E49 L87 ? remove_due_to_license_issue P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL 4mgb A 1.85 BS02 XDH A 1 L346 L349 A350 L387 M388 F404 I424 F425 G521 H524 L42 L45 A46 L83 M84 F100 I118 F119 G213 H216 ? remove_due_to_license_issue P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHR 4mgc A 2.15 BS02 27M A 1 L349 A350 E353 M388 H524 L525 L43 A44 E47 M82 H213 L214 ? remove_due_to_license_issue P03372 25260197 601 LALSLTADQMVSALLDAEPPILYSEYDPTRFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL 4mgd A 1.9 BS02 27N A 1 T347 A350 E353 L387 F404 M421 T43 A46 E49 L83 F100 M115 ? remove_due_to_license_issue EC50=31nM, IC50=43nM P03372 25260197 601 SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL 4mgv A 1.72 BS01 D5I A 1 Y43 D55 F64 V73 I74 W77 Y100 Y39 D51 F60 V69 I70 W73 Y96 Y43 F54 D55 I74 Y100 F117 Y39 F50 D51 I70 Y96 F113 5.2.1.8 0003755 remove_due_to_license_issue A5K8X6 24900611 201 TLEQVHLTEDGGVVKTILRKGEGGEENAPKKGNEVTVHYVGKLESSGKVFDSSRERNVPFKFHLGQGEVIKGWDICVASMTKNEKCSVRLDSKYGYGEEGCGESIPGNSVLIFEIELISFRE 4mh7 A 2.51 BS02 MH7 A 1 G594 A617 F673 M674 K675 A740 G18 A41 F80 M81 K82 A147 D723 A725 R727 N728 D741 D130 A132 R134 N135 D148 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=5900nM Q12866 24219778 906 LEDVVIDRNLLILGKILGEGEFGSVMEGNLKQEDGTSLKVAVKTAACMKDFSHPNVIRLLGVCIEMSSQGIPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESL 4mha A 2.59 BS01 4MH A 1 L593 A617 F673 M674 G677 M730 D741 L14 A35 F85 M86 G89 M142 D153 D723 A725 R727 N728 D741 D135 A137 R139 N140 D153 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=5.2nM Q12866 24219778 904 VVIDRNLLILGKILGEGSVMEGNLKQEDGTSLKVAVKTMKLDNSSQREIEEFLSEAACMKDFSHPNVIRLLGVCIEPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFGPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESLPD 4mhg A 2.199 BS01 dna B 0 Y387 E388 R392 R395 Y398 K405 R410 L411 Y53 E54 R58 R61 Y64 K71 R76 L77 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P97360 24333486 1 ~ 14 RLLWDYVYQLLSDSRYENFIRWEDKESKIFRIVDPNGLARLWGNHKNRTNMTYEKMSRALRHYYKLNIIRKEPGQRLLFRFMKTPDEIMS 4mhg A 2.199 BS02 dna C 0 L336 W376 K380 R382 M385 K389 R392 H396 Y397 L2 W42 K46 R48 M51 K55 R58 H62 Y63 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue P97360 24333486 1 ~ 14 RLLWDYVYQLLSDSRYENFIRWEDKESKIFRIVDPNGLARLWGNHKNRTNMTYEKMSRALRHYYKLNIIRKEPGQRLLFRFMKTPDEIMS 4mho A 2.0 BS01 26M A 1 E88 G135 L136 D283 R292 H341 H377 N484 E672 S674 G675 E77 G124 L125 D263 R272 H312 H348 N455 E643 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=8.25uM remove_due_to_license_issue Ki=8250nM P00489 25092521 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mhs A 2.0 BS01 26Q A 1 E88 G135 L136 D283 R292 H341 H377 N484 E672 S674 G675 E77 G124 L125 D267 R276 H315 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=5.14uM remove_due_to_license_issue Ki=5140nM P00489 25092521 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mhy A 1.38 BS02 PBD A 1 D144 E183 E184 W189 D238 E296 F317 W321 H322 D115 E154 E155 W160 D209 E267 F288 W292 H293 2.3.2.5 0005576,0008270,0016603,0016746,0017186,0046872 remove_due_to_license_issue B7QK46 24598748 401 LKWPRDLRPLAHHDLLYMGQIEDRGDFNATLRNFLVPRVVGSQKHREVREFIVRSLKDLDWDVEEDCFDGQTPHGIKPFCNVIATLNPSACHRLVLACHYDSLLHKEGTFIGATDSAVPCAQLLYLARSLNGKLQNQKTRGDGLTLQLVFFDGEEAFERWSSHDSLYGSRHLAQKWHEDRTSAERLESCLERSEIANQIDRMEVMVLLDLLGAENPRFYSYFGETQPVYRRLVNIESRLNDAGLMELPRRRRRTNYFSNSSTVGFIEDDHIPFLKRSVPIVHIIPSPFPDVWHTLDDNEQNLHHPTISNLNKIFKAFVSEYLQL 4mhz A 1.95 BS01 PBD A 1 D144 E183 D238 L239 I295 E296 F317 W321 D116 E155 D210 L211 I267 E268 F289 W293 2.3.2.5 0005576,0008270,0016603,0016746,0017186,0046872 remove_due_to_license_issue B7QK46 24598748 401 LKWPRDLRPLAHHDLLYMGQISEDRGDFNATLRNFLVPRVVGSQKHREVREFIVRSLKDLDWDVEEDCFDGQTPHGIKPFCNVIATLNPSACHRLVLACHYDSLLHKEGTFIGATDSAVPCAQLLYLARSLNGKLQNQKTRGDGLTLQLVFFDGEEAFERWSSHDSLYGSRHLAQKWHEDRTSAERLESCLERSEIANQIDRMEVMVLLDLLGAENPRFYSYFGETQPVYRRLVNIESRLNDAGLMELPRRRRRTNYFSNSSTVGFIEDDHIPFLKRSVPIVHIIPSPFPDVWHTLDDNEQNLHHPTISNLNKIFKAFVSEYLQL 4mi3 A 2.15 BS01 26R A 1 G135 L136 D283 H377 N484 E672 S674 G675 G124 L125 D263 H348 N455 E643 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=75.29uM remove_due_to_license_issue P00489 25092521 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mi6 A 1.9 BS01 26V A 1 L136 D283 N284 H377 N484 E672 S674 G675 L125 D267 N268 H351 N458 E646 S648 G649 H377 K568 R569 K574 T676 K680 H351 K542 R543 K548 T650 K654 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=48.68uM remove_due_to_license_issue Ki=48680nM P00489 25092521 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mi9 A 1.85 BS01 26W A 1 G135 L136 N282 N284 H341 H377 N484 E672 S674 G675 G124 L125 N265 N267 H314 H350 N457 E645 S647 G648 H377 K568 R569 K574 T676 K680 H350 K541 R542 K547 T649 K653 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=376.87uM remove_due_to_license_issue Ki=376870nM P00489 25092521 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mib A 2.3 BS01 28M A 1 R200 N291 N316 G317 D318 C366 S368 L384 G410 M414 Y415 Q446 I447 Y448 R195 N286 N311 G312 D313 C361 S363 L379 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.2nM remove_due_to_license_issue P26663 24195700 602 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4mic A 2.45 BS01 26Y A 1 G135 L136 N282 D283 F285 H341 H377 N484 E672 S674 G675 G124 L125 N262 D263 F265 H312 H348 N455 E643 S645 G646 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Ki=4.98uM remove_due_to_license_issue Ki=4980nM P00489 25092521 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mjo A 2.4 BS01 2C1 A 1 V17 M18 G21 R22 R25 G26 G28 L30 T31 V9 M10 G13 R14 R17 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 Kd=0.6uM remove_due_to_license_issue IC50=80nM P09467 24128068 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYARDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 4mjo C 2.4 BS01 2C1 C 1 M18 G21 R22 R25 G26 G28 L30 T31 M177 M10 G13 R14 R17 G18 G20 L22 T23 M159 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 Kd=0.6uM remove_due_to_license_issue IC50=80nM P09467 24128068 401 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYARDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 4mjp B 1.855 BS01 27O B 1 T172 R240 P242 D243 R246 V247 T165 R233 P235 D236 R239 V240 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=131uM remove_due_to_license_issue P0A988 24631121 403 MKFTVEREHLLKPLQQVSGPPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4mjq A 1.73 BS01 27R A 1 R152 Y154 H175 R176 P242 V247 R148 Y150 H171 R172 P238 V243 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=193uM remove_due_to_license_issue P0A988 24631121 401 MKFTVEREHLLKPLQQVSGRPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4mjr A 1.62 BS01 0LA A 1 R152 Y154 G174 R176 L177 V247 V360 M362 R146 Y148 G168 R170 L171 V241 V354 M356 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=283uM remove_due_to_license_issue P0A988 24631121 404 MKFTVEREHLLKPLQQVSGPLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4mk0 A 2.4 BS01 29X A 1 I197 R199 G200 G203 V205 A218 K220 D272 L273 M274 A321 L324 S334 D335 A480 I168 R170 G171 G174 V176 A189 K191 D243 L244 M245 A292 L295 S305 D306 A451 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 ic50=6.3uM remove_due_to_license_issue P25098 24220010 702 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVNAADAFTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKPA 4mk1 A 1.85 BS03 27Y A 1 H41 E80 D108 E119 K134 H46 E85 D113 E124 K139 3.1.-.- 0003723,0039694 ic50=16uM remove_due_to_license_issue M9V5A4 23978130 307 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4mk1 A 1.85 BS04 27Y A 2 A20 Y24 E26 E80 A25 Y29 E31 E85 3.1.-.- 0003723,0039694 ic50=16uM remove_due_to_license_issue M9V5A4 23978130 308 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4mk1 A 1.85 BS05 27Y A 3 A20 E23 Y24 G81 R82 D83 A25 E28 Y29 G86 R87 D88 3.1.-.- 0003723,0039694 ic50=16uM remove_due_to_license_issue M9V5A4 23978130 309 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4mk2 A 1.85 BS04 28B A 1 Y24 K34 I38 H41 E80 D108 E119 K134 Y29 K39 I43 H46 E85 D113 E124 K139 3.1.-.- 0003723,0039694 ic50=0.73uM remove_due_to_license_issue M9V5A4 23978130 306 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4mk5 A 1.9 BS03 28A A 1 Y24 K34 I38 H41 E80 D108 E119 K134 Y29 K39 I43 H46 E85 D113 E124 K139 3.1.-.- 0003723,0039694 ic50=0.45uM remove_due_to_license_issue M9V5A4 23978130 306 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4mk7 A 2.8 BS02 28O A 1 R200 G410 M414 Y415 Y448 R195 G405 M409 Y410 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 24069953 603 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4mk8 A 2.09 BS01 28Q A 1 S288 N291 N316 G317 D318 D319 G410 M414 Y415 Q446 I447 Y448 S556 S283 N286 N311 G312 D313 D314 G405 M409 Y410 Q441 I442 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=1nM remove_due_to_license_issue P26663 24069953 602 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4mk9 A 2.05 BS01 28R A 1 F193 N316 G317 D318 D319 C366 S368 G410 M414 Y415 Q446 I447 Y448 S556 F188 N311 G312 D313 D314 C361 S363 G405 M409 Y410 Q441 I442 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=9nM remove_due_to_license_issue P26663 24069953 601 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4mka A 2.05 BS01 2AY A 1 F193 N291 N316 G317 D318 D319 C366 S368 G410 M414 Y415 Q446 I447 Y448 S556 F188 N286 N311 G312 D313 D314 C361 S363 G405 M409 Y410 Q441 I442 Y443 S551 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=1nM remove_due_to_license_issue P26663 24069953 602 HMSYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPAASRLDLSGWFVAGYSGGDIYH 4mlt A 2.0 BS02 TM4 A 1 H94 V121 L198 T199 T200 H91 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.4mM remove_due_to_license_issue P00918 24635441 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4mlx A 1.65 BS02 TM7 A 1 H94 H96 H119 L198 T200 H91 H93 H116 L194 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.65mM remove_due_to_license_issue P00918 24635441 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4mm4 A 2.886 BS03 8PR A 1 Y21 A22 D24 P101 A105 Y108 F253 F259 S356 G359 T408 Y17 A18 D20 P97 A101 Y104 F246 F252 S349 G352 T401 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYTHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mm5 A 3.2 BS03 SRE A 1 Y21 D24 P101 Y108 F253 G256 F259 S355 G359 Y17 D20 P97 Y104 F246 G249 F252 S348 G352 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYTHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mm6 A 3.1 BS03 29E A 1 Y21 A22 D24 P101 V104 A105 Y108 F253 S254 F259 S356 G359 T408 Y17 A18 D20 P97 V100 A101 Y104 F246 S247 F252 S349 G352 T401 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mm7 A 2.85 BS03 29J A 1 Y21 V104 Y108 F253 F259 S355 Y17 V100 Y104 F246 F252 S348 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPTHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mm8 A 3.31 BS03 RFX A 1 Y21 A22 D24 V104 A105 Y108 F253 G256 F259 G359 T408 Y17 A18 D20 V100 A101 Y104 F246 G249 F252 G352 T401 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYITHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mm9 A 2.9 BS03 FVX A 1 Y21 A22 D24 V104 A105 Y108 F253 S254 F259 G359 Y17 A18 D20 V100 A101 Y104 F246 S247 F252 G352 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mma A 3.3 BS03 CXX A 1 Y21 D24 P101 V104 A105 Y108 F259 S355 S356 G359 T408 Y17 D20 P97 V100 A101 Y104 F252 S348 S349 G352 T401 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVASYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGVLITFASYVRKDQDIVLSGLTAATLNEKASVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQGMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWATGIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mme A 2.5 BS03 29Q A 1 Y21 A22 D24 V104 A105 Y108 F253 G256 F259 S355 G359 Y17 A18 D20 V100 A101 Y104 F246 G249 F252 S348 G352 ? 0005886,0016020,0035725 Kd=318nM remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGAIITFASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mmf A 2.7 BS03 29Q A 1 Y21 A22 D24 V104 A105 Y108 F253 G256 F259 G359 Y17 A18 D20 V100 A101 Y104 F246 G249 F252 G352 ? 0005886,0016020,0035725 remove_due_to_license_issue O67854 24121440 603 REHWATRLGLILAMAGYAVDLGNFLRFPVQAAENGGGAFMIPYIIAFLLVGIPLMWIEWAMGRYGGAQGHGTTPAIFYLLWRNRFAKILGVFGLWIPLVVAIYYVYIESWTLGFAIKFLVGLVPEPPTDPDSILRPFKEFLYSYIGVPKGDEPILKPSLFAYIVFLITMFINVSILIRGISKGIERFAKIAMPTLFILAVFLVIRVFLLETPNGTAADGLNFLWTPDFEKLKDPGVWIAAVGQIFFSLGLGFGAIITYASYVRKDQDIVLSGLTAATLNEKAEVILGGSISIPAAVAFFGVANAVAIAKAGAFNLGFITLPAIFSQTAGGTFLGFLWFFLLFFAGLTSSIAGMQPMIAFLEDELKLSRKHAVLWTAAIVFFSAHLVMFLNKSLDEMDFWAGTIGVVFFGLTELIIFFWIFGADKAWEEINRGGIIKVPRIYYYVMRYITPAFLAVLLVVWAREYIPKIMEETHWTVWITRFYIIGLFLFLTFLVFLAERRRNHE 4mmm A 1.47 BS01 BP7 A 1 T44 G46 C47 I119 T45 G47 C48 I120 1.11.1.24 0008379,0016491,0034599 Kd=150uM remove_due_to_license_issue P30044 25025339 201 SAPIKVGDAIPAVEVFEGEPGNKVNLAELFKGKKGVLFGVPGAFTPGCSKTHLPGFVEQAEALKAKGVQVVACLSVNDAFVTGEWGRAHKAEGKVRLLADPTGAFGKETDLLLDDSLVSIFGNRRLKRFSMVVQDGIVKALNVEPDGTGLTCSLAPNIISQL 4mmp A 1.57 BS01 SLB A 1 V12 D51 L67 E69 R72 R129 R149 F172 N189 Q216 V11 D50 L66 E68 R71 R128 R148 F171 N188 Q215 0030288,0055085 Kd=19.7nM remove_due_to_license_issue 25004958 401 GADYDLKFGMVAGPSSNEYKAVEFFAKEVKEKSNGKIDVAIFPSSQLGDDRVMIKQLKDGALDFTLGESARFQIYFPEAEVFALPYMIPNFETSKKALLDTKFGQGLLKKIDKELNVQVLSVAYNGTRQTTSNRAINSIEDMKGLKLRVPNAATNLAYAKYVGAAPTPMAFSEVYLALQTNSVDGQENPLPTIQAQKFYEVQKYLALTNHILNDQLYLISNDTLADLPEDLQKVVKDAAAKAAEYHTKLFVDGENSLVEFFKSQGVTVTQPDLKPFKAALTPYYDEYLKKNGEVGKMAIEEISNLAKL 4mnp A 2.5 BS01 SLB A 1 D51 F67 E69 R72 R128 R148 F171 N188 D49 F65 E67 R70 R126 R146 F169 N186 ? 0030288,0042597,0055085 Kd=45.5nM remove_due_to_license_issue Q8RDN9 25004958 401 KYNLKMGMTAGTSQNEYKAAEVFAKELKKRSNGEIELKLYPNAQLGKDDLAMMQQLEGGALDFTFAETGRFSTFFPEAEVFTLPYMIKDFNHMKKAVNTKFGKDLFKKVHDKKGMTVLAQAYNGTRQTTSNKAIKSLADMKGMKLRVPGAAANLAYAKYTEAAPTPMAFSEVYLALQTNAVDGQENPLSTIKAQKFYEVQKYLAMTNHILNDQLYLVSNITMEELPENLQKVVKESAEVAAEYHTKLFMDEEKSLKDFFKSKGVTITEPNLVDFKKAMKPFYDEYIKKNGKVGENAIKAIEAVRL 4mo4 A 1.67 BS01 ACP A 1 G164 N187 D191 F202 D203 R204 D205 G291 G292 F295 G163 N186 D190 F201 D202 R203 D204 G273 G274 F277 2.7.1.170 0005524,0006040,0009254,0016301,0016773,0046677,0097175 Kd=0.06mM remove_due_to_license_issue Q9I5Q5 24362022 500 PRYLGLMSGTSLDGMDIVLIEQGDRTTLLASHYLPMPAGLREDILALCVPGPDEIARAAEVEQRWVALAAQGVRELLLQQQMSPDEVRAIGSHGQTIRHEPARHFTVQIGNPALLAELTGIDVVADFRRRDVAAGGQGAPLVPAFHQALFGDDDTSRAVLNIGGFSNVSLLSPGKPVRGFDCGPGNVLMDAWIHHQRGEHFDRDGAWAASGQVNHALLASLLANLPWLQEHLARHPALPAADIQATLLELSARSISESLLDAQPDCEEVLVCGGGAFNTALMKRLAMLMPEARVASTDEYGIPPAWMEGMAFAWLAHRFLERLPGNCPDVTGALGPRTLGALYPA 4mo8 A 1.85 BS02 2VQ A 1 H64 H94 H96 L198 T199 T200 H61 H91 H93 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10.1nM remove_due_to_license_issue Ki=10nM P00918 24128000 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4mot A 1.75 BS01 2B7 A 1 I48 N51 A52 E55 V76 D78 R81 G82 M83 P84 I98 R140 T172 I32 N35 A36 E39 V60 D62 R65 G66 M67 P68 I82 R107 T139 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue Q8DQB5 24405701 301 QVLEGLDAVRKRPGMYIGSTDGAGLHHLVWEIVDNAVDEALSGFGDRIDVTINKDGSLTVQDHGRGMPTGMHAMGIPTVEVIFTILHAVGSSVVNALSSWLEVEITRDGAVYKQRFENGGKPVTTLKKIGTALKSKTGTKVTFMPDATIFSTTDFKYNTISERLNESAFLLKNVTLSLTDKRTDEAIEFHYEN 4mp2 A 1.751 BS01 PV1 A 1 N255 R258 A259 E262 D290 G294 V295 T354 N240 R243 A244 E247 D275 G279 V280 T322 H247 E251 K254 N255 H232 E236 K239 N240 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=3570nM remove_due_to_license_issue IC50=6.78e+3nM, Kd=3570nM Q15119 24356970 501 SLAGAPKYIEHFSKFSPSPLSMKQFLDFGSSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPAHPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWC 4mp7 A 1.8 BS01 PFT A 1 N255 R258 A259 E262 D290 G294 V295 T354 N240 R243 A244 E247 D275 G279 V280 T323 H247 E251 K254 N255 H232 E236 K239 N240 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=1827nM remove_due_to_license_issue IC50=5.68e+3nM, Kd=1827nM Q15119 24356970 501 SLAGAPKYIEHFSKFSPSPLSMKQFLDFGSSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPAHPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWCVP 4mpc A 1.699 BS01 PV2 A 1 N255 R258 A259 E262 D290 G294 V295 T354 N240 R243 A244 E247 D275 G279 V280 T323 H247 E251 K254 N255 H232 E236 K239 N240 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=711nM remove_due_to_license_issue IC50=2.11e+3nM, Kd=711nM Q15119 24356970 502 SLAGAPKYIEHFSKFSPSPLSMKQFLDFGSSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPAHPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWCVP 4mpe A 1.953 BS01 PV8 A 1 N255 R258 A259 E262 D290 G294 V295 T354 N240 R243 A244 E247 D275 G279 V280 T323 H247 E251 K254 N255 H232 E236 K239 N240 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=426nM remove_due_to_license_issue Kd=426nM, IC50=570nM Q15119 24356970 501 SLAGAPKYIEHFSKFSPSPLSMKQFLDFGSSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPAHPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWCVP 4mpn A 1.752 BS01 PV0 A 1 N255 R258 A259 E262 D290 G294 V295 T354 N240 R243 A244 E247 D275 G279 V280 T323 H247 E251 K254 N255 H232 E236 K239 N240 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=239nM remove_due_to_license_issue EC50=456nM, Kd=156nM, IC50=456nM Q15119 24356970 501 SLAGAPKYIEHFSKFSPSPLSMKQFLDFGSSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPAHPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWCVP 4mq1 A 2.35 BS01 2C3 A 1 I165 G166 K167 G168 F170 G171 V173 K188 F238 M240 L241 S242 N292 L294 V306 D307 I31 G32 K33 G34 F36 G37 V39 K54 F104 M106 L107 S108 N158 L160 V172 D173 D287 K289 N292 D307 S324 D153 K155 N158 D173 S190 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=12nM Q13627 24239188 501 VYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDGKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 4mq2 A 2.8 BS01 2C4 A 1 F170 K188 F238 M240 L241 S242 Y243 L294 V306 D307 F35 K53 F103 M105 L106 S107 Y108 L159 V171 D172 D287 K289 N292 D307 S324 D152 K154 N157 D172 S189 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=97nM Q13627 24239188 501 YNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 4mq6 A 1.7 BS01 29W A 1 P38 T39 H44 G46 H47 K160 Q164 V187 M195 S196 S197 P36 T37 H42 G44 H45 K158 Q162 V185 M193 S194 S195 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 0004592,0015940 remove_due_to_license_issue 26486566 404 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4mq6 A 1.7 BS02 29W A 2 L114 P133 T134 G138 L112 P131 T132 G136 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 0004592,0015940 remove_due_to_license_issue 26486566 405 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4mqp A 1.83 BS01 2B1 A 1 W64 W65 G124 S125 Y157 H158 E220 A226 D254 I256 K283 Y407 W57 W58 G117 S118 Y150 H151 E213 A219 D247 I249 K276 Y400 Y25 Y157 E220 D254 A257 K283 Y407 Y18 Y150 E213 D247 A250 K276 Y400 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 24482078 501 LTPEQIIAVDGAHLWHPYSSIGREAVSPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHGGMHSLWTDVLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLVGS 4mqp B 1.83 BS01 2B1 A 1 P317 T318 P310 T311 Y25 Y157 E220 D254 A257 K283 Y407 Y18 Y150 E213 D247 A250 K276 Y400 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 24482078 501 LTPEQIIAVDGAHLWHPYSSIGREAVSPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHGGMHSLWTDVLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLVG 4mqp B 1.83 BS02 2B1 B 1 W65 G124 S125 Y157 H158 E220 A226 D254 I256 K283 F402 Y407 W58 G117 S118 Y150 H151 E213 A219 D247 I249 K276 F395 Y400 Y25 Y157 E220 D254 A257 K283 Y407 Y18 Y150 E213 D247 A250 K276 Y400 2.6.1.62 0004015,0005737,0008483,0009102,0030170 remove_due_to_license_issue P9WQ81 24482078 501 LTPEQIIAVDGAHLWHPYSSIGREAVSPVVAVAAHGAWLTLIRDGQPIEVLDAMSSWWTAIHGHGHPALDQALTTQLRVMNHVMFGGLTHEPAARLAKLLVDITPAGLDTVFFSDSGSVSVEVAAKMALQYWRGRGLPGKRRLMTWRGGYHGDTFLAMSICDPHGGMHSLWTDVLAAQVFAPQVPRDYDPAYSAAFEAQLAQHAGELAAVVVEPVVQGAGGMRFHDPRYLHDLRDICRRYEVLLIFDEIATGFGRTGALFAADHAGVSPDIMCVGKALTGGYLSLAATLCTADVAHTISAGAAGALMHGPTFMANPLACAVSVASVELLLGQDWRTRITELAAGLTAGLDTARALPAVTDVRVCGAIGVIECDRPVDLAVATPAALDRGVWLRPFRNLVYAMPPYICTPAEITQITSAMVEVARLVG 4mqu A 2.22 BS01 MG9 A 1 P29 E32 G181 M213 R215 H504 K514 W517 A521 M522 R525 P29 E32 G179 M211 R213 H483 K493 W496 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue IC50=4.0nM Q14397 24405213 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4mr3 A 1.68 BS01 1K0 A 1 W81 P82 Q85 V87 L92 N140 I146 W40 P41 Q44 V46 L51 N99 I105 ? remove_due_to_license_issue IC50=510nM, Kd=1100nM O60885 24248379 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4mr4 A 1.66 BS01 1K0 A 1 P82 F83 V87 L92 Y139 N140 I146 P41 F42 V46 L51 Y98 N99 I105 ? remove_due_to_license_issue IC50=510nM, Kd=1100nM O60885 24248379 204 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4mr5 A 1.63 BS01 1K0 A 1 P371 F372 V376 L383 N429 H433 V435 P26 F27 V31 L38 N84 H88 V90 ? remove_due_to_license_issue Kd=5800nM, IC50=251nM P25440 24248379 506 LSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 4mr6 A 1.67 BS01 1K0 A 1 P371 F372 V376 L383 N429 H433 V435 P26 F27 V31 L38 N84 H88 V90 ? remove_due_to_license_issue Kd=5800nM, IC50=251nM P25440 24248379 505 LSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 4mra A 2.34 BS01 QUE A 1 E121 E124 K544 Y548 R551 K655 E110 E113 K515 Y519 R522 K626 H377 K568 R569 K574 T676 K680 H348 K539 R540 K545 T647 K651 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 ic50=33.5uM remove_due_to_license_issue P00489 24556570 901 QISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVLPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPA 4mrd A 2.55 BS01 BDP B 1 Y83 I100 A102 Y59 I76 A78 ? 0005540,0007155,0016020 remove_due_to_license_issue P15379 24606063 2 QIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4mrd A 2.55 BS02 BDP B 2 C81 R82 I100 C57 R58 I76 ? 0005540,0007155,0016020 remove_due_to_license_issue P15379 24606063 4 QIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4mre A 1.58 BS01 2C9 A 1 N29 V30 R155 N6 V7 R132 ? 0005540,0007155,0016020 Kd=6.4mM remove_due_to_license_issue Kd=6400000nM P15379 24606063 202 NQIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4mrf A 1.55 BS01 2CK A 1 N29 V30 V153 N154 R155 N6 V7 V130 N131 R132 ? 0005540,0007155,0016020 Kd=11.2mM remove_due_to_license_issue Kd=11200000nM P15379 24606063 203 NQIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4mrg A 1.69 BS01 24W A 1 N29 V30 E41 N154 R155 N6 V7 E18 N131 R132 ? 0005540,0007155,0016020 Kd=1.1mM remove_due_to_license_issue Kd=1100000nM P15379 24606063 201 NQIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4mrh A 1.12 BS01 2CQ A 1 R33 F38 F60 V137 T138 R10 F15 F37 V114 T115 ? 0005540,0007155,0016020 Kd=12.6mM remove_due_to_license_issue Kd=12600000nM P15379 24606063 201 NQIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4mro A 2.2 BS01 MG0 A 1 V28 P29 E32 R215 H504 W517 A521 M522 R525 V28 P29 E32 R213 H483 W496 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 24405213 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4mrw A 1.96 BS01 MRW A 1 I692 F696 Q726 F729 I247 F251 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=500uM remove_due_to_license_issue Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4mrz A 1.58 BS01 2ZV A 1 F696 Q726 F729 F251 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=300uM remove_due_to_license_issue Ki=300000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4ms0 A 1.79 BS01 2ZX A 1 I692 M713 Q726 F729 I247 M268 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=410uM remove_due_to_license_issue Ki=410000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4msa A 1.62 BS01 2ZM A 1 L675 S677 I692 F696 Q726 F729 L230 S232 I247 F251 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=500uM remove_due_to_license_issue Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4msa A 1.62 BS02 2ZM A 2 C469 Y492 R496 C24 Y47 R51 3.1.4.17 0004114,0007165,0008081 Ki=500uM remove_due_to_license_issue Q9Y233 24375910 903 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4msc A 2.47 BS01 2ZT A 1 Y693 P712 M713 E721 G725 F729 Y246 P265 M266 E274 G278 F282 3.1.4.17 0004114,0007165,0008081 Ki=1.1uM remove_due_to_license_issue Ki=1100nM Q9Y233 24375910 900 TSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4mse A 2.81 BS01 2ZU A 1 Y693 M713 E721 G725 F729 Y248 M268 E276 G280 F284 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Ki=5500nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4msg A 1.8 BS02 2C6 A 1 H1184 G1185 S1186 F1188 A1191 I1192 K1195 G1196 F1197 D1198 H1201 A1202 Y1213 F1214 A1215 K1220 S1221 Y1224 E1291 H80 G81 S82 F84 A87 I88 K91 G92 F93 D94 H97 A98 Y109 F110 A111 K116 S117 Y120 E187 2.4.2.-,2.4.2.30 0003950 ic50=0.1nM remove_due_to_license_issue O95271 24294969 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEH 4msk A 2.3 BS02 2C8 A 1 H1184 G1185 S1186 F1188 A1191 K1195 F1197 D1198 H1201 Y1203 I1212 Y1213 F1214 A1215 K1220 S1221 Y1224 E1291 H81 G82 S83 F85 A88 K92 F94 D95 H98 Y100 I109 Y110 F111 A112 K117 S118 Y121 E188 2.4.2.-,2.4.2.30 0003950 ic50=0.063uM remove_due_to_license_issue O95271 24294969 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPE 4msl A 2.7 BS01 2ET A 1 Y271 S283 R292 F317 Y318 Y212 S224 R233 F258 Y259 ? 0016020 remove_due_to_license_issue IC50=4000nM Q99523 24531479 809 CGRVRDFVAKLANNTHQHVFDDLRGSVSLSWVGDSTGVILVLTTFHVGQSKLYRSEDYGKNFKDITDLINNTFIRTEFGMAIGPENSGKVVLTAEVSGGSRGGRIFRSSDFAKNFVQTDLPFHPLTQMMYSPQNSDYLLALSTENGLWVSKNFGGKWEEIHKAVCLAKWGSDNTIFFTTYANGSCKADLGALELWRTSDLGKSFKTIGVKIYSFGLGGRFLFASVMADKDTTRRIHVSTDQGDTWSMAQLPSVGQEQFYSILAANDDMVFMHVDEPGDTGFGTIFTSDDRGIVYSKSLDRHLYTTTGGETDFTNVTSLRGVYITSVLSEDNSIQTMITFDQGGRWTHLRKPENSECDATAKNKNECSLHIHASYSISQKLNVPMAPLSEPNAVGIVIAHGSVGDAISVMVPDVYISDDGGYSWTKMLEGPHYYTILDSGGIIVAIEHSSRPINVIKFSTDEGQCWQTYTFTRDPIYFTGLASEPGARSMNISIWGFTESTSQWVSYTIDFKDILERNCEEKDYTIWLAHSTDPEDYEDGCILGYKEQFLRLRKSSMCQNGRDYVVTKQPSICLCSLEDFLCDFGYYRPENDSKCVEQPELKGHDLEFCLYGREEHLTTNGYRKIPGDKCQGGVNPVREVKDLKKKCTSNFLSPE 4msn A 2.3 BS01 2ZQ A 1 M713 Q726 F729 M268 Q281 F284 3.1.4.17 0004114,0007165,0008081 Ki=94uM remove_due_to_license_issue Ki=94000nM Q9Y233 24375910 900 AGTSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATWI 4mss A 1.8 BS01 2CZ A 1 D65 R140 K170 H171 H183 D253 D254 D63 R138 K168 H169 H181 D251 D252 3.2.1.52 0004553,0004563,0005737,0005975,0008360,0009252,0009254,0016231,0016798,0051301,0071555 Ki=3.6uM remove_due_to_license_issue B4EA43 24136176 401 TTPGPVMLDVVGTTLSRDDARRLAHPNTGGVILFARHFQNRAQLTALTDSIRAVREDILIAVDHEGGRVQRFRTDGFTVLPAMRRLGELWDRDVLLATKVATAVGYILAAELRACGIDMSFTPVLDLDYGHSKVIGDRAFHRDPRVVTLLAKSLNHGLSLAGMANCGKHFPGHGFAEADSHVALPTDDRTLDAILEQDVAPYDWLGLSLAAVIPAHVIYTQVDKRPAGFSRVWLQDILRGKLGFTGAIFSDDLSMEAAREGGTLTQAADAALAAGCDMVLVCNQPDAAEVVLNGLKARASAESVRRIKRMRARGKALKWDKLIAQPEYLQAQALLSSAL 4msu A 2.5 BS01 2EU A 1 V28 P29 E32 R215 H504 W517 A521 M522 R525 V28 P29 E32 R213 H483 W496 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 ic50=1.42uM remove_due_to_license_issue IC50=1420nM, Kd=240nM Q14397 24405172 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4mt9 A 2.0 BS02 2D6 A 1 H1184 G1185 F1188 H1201 I1212 Y1213 F1214 A1215 K1220 S1221 Y1224 H80 G81 F84 H97 I108 Y109 F110 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=0.1nM remove_due_to_license_issue O95271 24294969 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPE 4mti A 2.15 BS02 2DX A 1 D297 G306 L307 R308 C309 W310 D314 E319 W323 D45 G54 L55 R56 C57 W58 D62 E67 W71 2.3.2.27 ic50=1.2nM remove_due_to_license_issue Q13490 24169315 402 SSISNLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRY 4mu7 A 1.79 BS02 2DY A 1 R294 G306 L307 R308 C309 W310 D314 E319 W323 R38 G50 L51 R52 C53 W54 D58 E63 W67 2.3.2.27 ic50=1.4nM remove_due_to_license_issue Q13490 24169315 402 NLSMQTHAARMRTFMYWPSSVPVQPEQLASAGFYYVGRNDDVKCFCCDGGLRCWESGDDPWVEHAKWFPRCEFLIRMKGQEFVDEIQGRY 4mue A 2.06 BS01 2DH A 1 P38 T39 M40 H44 G46 H47 K160 Q164 T186 V187 M195 S196 P35 T36 M37 H41 G43 H44 K146 Q150 T172 V173 M181 S182 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D74 D75 Q78 K146 S182 S183 R184 0004592,0015940 remove_due_to_license_issue 26486566 401 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 4mue A 2.06 BS02 2DH A 2 L114 P133 T134 G138 L100 P119 T120 G124 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D74 D75 Q78 K146 S182 S183 R184 0004592,0015940 remove_due_to_license_issue 26486566 402 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTF 4muf A 2.5 BS01 2DJ A 1 P38 T39 M40 H44 G46 H47 G158 K160 D161 Q164 M195 S196 S197 P35 T36 M37 H41 G43 H44 G147 K149 D150 Q153 M184 S185 S186 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M37 H41 H44 D77 D78 Q81 K149 S185 S186 R187 0004592,0015940 remove_due_to_license_issue 26486566 403 PAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGT 4muk A 1.9 BS01 2DV A 1 P38 T39 M40 H44 G46 H47 V142 D161 V187 M195 P36 T37 M38 H42 G44 H45 V125 D144 V170 M178 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D71 D72 Q75 K143 S179 S180 R181 0004592,0015940 remove_due_to_license_issue 26486566 401 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4mul A 1.75 BS01 2DW A 1 P38 T39 M40 H44 G46 H47 Q72 V139 K160 Q164 V187 M195 S196 S197 P36 T37 M38 H42 G44 H45 Q70 V137 K158 Q162 V185 M193 S194 S195 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 0004592,0015940 remove_due_to_license_issue 26486566 404 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4mul A 1.75 BS02 2DW A 2 M71 L114 P133 T134 M69 L112 P131 T132 M40 H44 H47 D88 D89 Q92 K160 S196 S197 R198 M38 H42 H45 D86 D87 Q90 K158 S194 S195 R196 0004592,0015940 remove_due_to_license_issue 26486566 407 IPAFHPGELNVYSAPGDVADVSRALRLTGRRVMLVPTMGALHEGHLALVRAAKRVPGSVVVVSIFVNPMQFGAGGDLDAYPRTPDDDLAQLRAEGVEIAFTPTTAAMYPDGLRTTVQPGPLAAELEGGPRPTHFAGVLTVVLKLLQIVRPDRVFFGEKDYQQLVLIRQLVADFNLDVAVVGVPTVREADGLAMSSRNRYLDPAQRAAAVALSAALTAAAHAATAGAQAALDAARAVLDAAPGVAVDYLELRDIGLGPMPLNGSGRLLVAARLGTTRLLDNIAIEIGTFA 4muv A 1.25 BS01 PCG A 1 V282 F296 G297 E298 M299 A300 R307 S308 R348 D352 V69 F83 G84 E85 M86 A87 R94 S95 R135 D139 ? 0005221 Kd=336nM remove_due_to_license_issue Q98GN8 24981229 401 GSQEVRRGDFVRNWQLVAAVPLFQKLGPAVLVEIVRALRARTVPAGAVICRIGEPGDRMFFVVEGSVSVASPNPSELGPGAFFGEMALISGEPRSATVSAATTVSLLSLHSADFQMLCSSSPEIAEIFRKTALERRGADASA 4muw A 2.639 BS02 2F4 A 1 L625 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 L184 I241 Y242 F245 P261 M262 E270 V271 G274 Q275 F278 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=9.7nM Q9Y233 24102193 1012 TSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4mvh A 2.496 BS02 2F5 A 1 Y514 I682 Y683 F686 P702 M703 E711 G715 Q716 F719 Y62 I230 Y231 F234 P250 M251 E259 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=4.5nM remove_due_to_license_issue IC50=4.5nM Q9Y233 24102193 1010 TLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4mvn A 1.7 BS01 I1S A 1 H39 A149 Q150 P151 S154 A171 G172 S173 G174 H39 A149 Q150 P151 S154 A171 G172 S173 G174 3.4.21.- 0004252,0005576,0006508,0008236 remove_due_to_license_issue Q2FXC2 24375505 301 EKNVKEITDATKEPYNSVVAFVGGTGVVVGKNTIVTNKHIAKSNDIFKNRVSAHHSSKGKGGGNYDVKDIVEYPGKEDLAIVHVHETSTEGLNFNKNVSYTKFADGAKVKDRISVIGYPKGAQTKYKMFESTGTINHISGTFMEFDAYAQPGNSGSPVLNSKHELIGILYAGSGKSEKNFGVYFTPQLKEFIQNNIEK 4mvn A 1.7 BS02 I1S C 1 K76 E77 K76 E77 3.4.21.- 0004252,0005576,0006508,0008236 remove_due_to_license_issue Q2FXC2 24375505 301 EKNVKEITDATKEPYNSVVAFVGGTGVVVGKNTIVTNKHIAKSNDIFKNRVSAHHSSKGKGGGNYDVKDIVEYPGKEDLAIVHVHETSTEGLNFNKNVSYTKFADGAKVKDRISVIGYPKGAQTKYKMFESTGTINHISGTFMEFDAYAQPGNSGSPVLNSKHELIGILYAGSGKSEKNFGVYFTPQLKEFIQNNIEK 4mwq A 2.0 BS02 G39 A 1 R119 E120 D152 R153 W180 I224 R226 R294 N296 R372 Y406 R37 E38 D70 R71 W98 I142 R144 R212 N214 R290 Y324 D152 E279 R294 R372 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.79nM remove_due_to_license_issue A0A024E3Q2 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCRDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mwr A 1.797 BS02 ZMR A 1 R119 E120 D152 R153 W180 E229 A248 E278 R294 R372 Y406 R37 E38 D70 R71 W98 E147 A166 E196 R212 R290 Y324 D152 E279 R294 R372 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.41nM remove_due_to_license_issue A0A024E3Q2 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCRDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mwu A 1.799 BS02 LNV A 1 R119 E120 D152 R153 W180 E229 A248 E278 R294 R372 Y406 R37 E38 D70 R71 W98 E147 A166 E196 R212 R290 Y324 D152 E279 R294 R372 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=3.24nM remove_due_to_license_issue A0A024E3Q2 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCRDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mwv A 2.0 BS02 BCZ A 1 R119 E120 D152 R153 W180 E229 E278 R294 R372 Y406 R37 E38 D70 R71 W98 E147 E196 R212 R290 Y324 D152 E279 R294 R372 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=0.4nM remove_due_to_license_issue A0A024E3Q2 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCRDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mww A 1.9 BS02 G39 A 1 R119 E120 D152 R153 W180 I224 R372 Y406 R37 E38 D70 R71 W98 I142 R290 Y324 D152 E279 K294 R372 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue A0A067Y7N7 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCKDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mwx A 1.801 BS02 ZMR A 1 R119 E120 D152 R153 W180 R226 E229 A248 E278 K294 R372 Y406 R37 E38 D70 R71 W98 R144 E147 A166 E196 K212 R290 Y324 D152 E279 K294 R372 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=75.7nM remove_due_to_license_issue A0A067Y7N7 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCKDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mwy A 1.8 BS02 LNV A 1 R119 E120 D152 R153 W180 R226 E229 A248 E278 K294 R372 Y406 R37 E38 D70 R71 W98 R144 E147 A166 E196 K212 R290 Y324 D152 E279 K294 R372 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=89.6nM remove_due_to_license_issue A0A067Y7N7 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCKDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mx0 A 2.101 BS02 BCZ A 1 R119 E120 D152 R153 W180 R226 E229 E279 R372 Y406 R37 E38 D70 R71 W98 R144 E147 E197 R290 Y324 D152 E279 K294 R372 Y406 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 ic50=184.7nM remove_due_to_license_issue A0A067Y7N7 24165891 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCKDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 4mx1 A 1.59 BS01 1MX A 1 Y80 V81 G121 N122 Y123 I172 R180 W211 G212 Y81 V82 G122 N123 Y124 I173 R181 W212 G213 V81 E177 R180 V82 E178 R181 3.2.2.22 0017148,0030598 ic50=209uM remove_due_to_license_issue IC50=209000nM P02879 24432385 301 MIFPKQYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 4mx5 X 1.52 BS01 5MX X 1 Y80 V81 G121 N122 Y123 I172 S176 R180 Y76 V77 G117 N118 Y119 I168 S172 R176 V81 V77 3.2.2.22 0017148,0030598 ic50=28uM remove_due_to_license_issue IC50=28000nM P02879 24432385 301 QYPIINFTTAGATVQSYTNFIRAVRGRLTTGADVRHEIPVLPNRVGLPINQRFILVELSNHAELSVTLALDVTNAYVVGYRAGNSAYFFHPDNQEDAEAITHLFTDVQNRYTFAFGGNYDRLEQLAGNLRENIELGNGPLEEAISALYYYSTGGTQLPTLARSFIICIQMISEAARFQYIEGEMRTRIRYNRRSAPDPSVITLENSWGRLSTAIQESNQGAFASPIQLQRRNGSKFSVYDVSILIPIIALMVYRCAPPPSSQF 4mx9 A 3.1 BS01 2E8 A 1 V64 A77 K79 M111 L125 Y130 E134 D194 V23 A36 K38 M70 L84 Y89 E93 D153 D173 K175 E177 N178 D194 T213 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue F0V9W9 24681759 601 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYYYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMKSMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSSELATIFGVSDVDSETWKNVLAEVDKNNDGEVDFDEFQQMLLKLCGN 4mxa A 3.0 BS01 BK7 A 1 V64 A77 K79 M111 L125 E134 I193 D194 V23 A36 K38 M70 L84 E93 I152 D153 D173 K175 E177 N178 D194 T213 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue F0V9W9 24681759 601 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYYYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMKSMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSSELATIFGVSDVDSETWKNVLAEVDKNNDGEVDFDEFQQMLLKLCGN 4mxc A 1.632 BS01 DWF A 1 I1084 V1092 A1108 K1110 E1127 M1131 F1134 Y1159 M1160 G1163 D1164 F1200 M1211 A1221 D1222 F1223 I33 V41 A57 K59 E76 M80 F83 Y108 M109 G112 D113 F149 M160 A170 D171 F172 D1204 A1206 R1208 N1209 D1222 A1243 D153 A155 R157 N158 D171 A187 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=6.7nM P08581 24944742 1401 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4my6 A 1.7 BS01 3VH A 1 Y16 W23 K69 N71 F77 Q79 W80 R81 V86 Y15 W22 K68 N70 F76 Q78 W79 R80 V85 ? remove_due_to_license_issue Q8N8S7 25848013 201 SEQSICQARAAVMVYDDANKKWVPAGGSTGFSRVHIYHHTGNNTFRVVGRKIQDHQVVINCAIPKGLKYNQATQTFHQWRDARQVYGLNFGSKEDANVFASAMMHALEVL 4my6 A 1.7 BS02 3VH B 1 Y16 D18 Y15 D17 ? remove_due_to_license_issue Q8N8S7 25848013 201 SEQSICQARAAVMVYDDANKKWVPAGGSTGFSRVHIYHHTGNNTFRVVGRKIQDHQVVINCAIPKGLKYNQATQTFHQWRDARQVYGLNFGSKEDANVFASAMMHALEVL 4myd A 1.374 BS01 164 A 1 G22 F23 Y85 S86 L87 R90 R124 W147 Y148 F153 G22 F23 Y85 S86 L87 R90 R124 W147 Y148 F153 4.2.99.20 0005829,0009234,0016829,0070205 Kd=28uM remove_due_to_license_issue P37355 24737327 301 MILHAQAKHGKPGLPWLVFLHGFSGDCHEWQEVGEAFADYSRLYVDLPGHGGSAAISVDGFDDVTDLLRKTLVSYNILDFWLVGYSLGGRVAMMAACQGLAGLCGVIVEGGHPGLQNAEQRAERQRSDRQWVQRFLTEPLTAVFADWYQQPVFASLNDDQRRELVALRSNNNGATLAAMLEATSLAVQPDLRANLSARTFAFYYLCGERDSKFRALAAELAADCHVIPRAGHNAHRENPAGVIASLAQILRF 4myh B 3.38 BS01 GSH B 1 R280 R284 S394 R183 R187 S297 7.-.-.- 0005524,0016020,0016887,0055085,0140359 remove_due_to_license_issue P40416 24604199 701 YIWPKGNNKVRIRVLIALGLLISAKILNVQVPFFFKQTIDSMNIAWDDPTVALPAAIGLTILCYGVARFGSVLFGELRNAVFAKVAQNAIRTVSLQTFQHLMKLDLGWHLSRQTGGLTRAMDRGTKGISQVLTAMVFHIIPISFEISVVCGILTYQFGASFAAITFSTMLLYSIFTIKTTAWRTHFRRDANKADNKAASVALDSLINFEAVKYFNNEKYLADKYNGSLMNYRDSQIKVSQSLAFLNSGQNLIFTTALTAMMYMGCTGVIGGNLTVGDLVLINQLVFQLSVPLNFLGSVYRDLKQSLIDMETLFKLRKNEVKIKNAERPLMLPENVPYDITFENVTFGYHPDRKILKNASFTIPAGWKTAIVGSSGSGKSTILKLVFRFYDPESGRILINGRDIKEYDIDALRKVIGVVPQDTPLFNDTIWENVKFGRIDATDEEVITVVEKAQLAPLIKKLPQGFDTIVGERGLMISGGEKQRLAIARVLLKNARIMFFDEATSALDTHTEQALLRTIRDNFTSGSRTSVYIAHRLRTIADADKIIVLDNGRVREEGKHLELLAMPGSLYRELWTIQEDLDHLENELKDQQELWSHPQ 4myq A 1.9 BS01 19T A 1 Y405 M519 N567 I582 F586 M603 Q615 F618 L674 K677 Y82 M196 N244 I259 F263 M280 Q292 F295 L339 K342 3.1.4.53 0004114,0007165,0008081 ic50=32nM remove_due_to_license_issue IC50=32nM Q07343 24361374 701 SISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPQCQGLMEKFQF 4mz4 A 1.63 BS01 2F3 A 1 F193 R200 N316 D319 C366 G410 M414 Y415 Q446 I447 Y448 F188 R195 N311 D314 C361 G405 M409 Y410 Q441 I442 Y443 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 24252545 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLGKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAAICGRYLFNWAVRTKLKLTPIPAASQLDLSGWFVAGYSGGDIYHSLSRAR 4mzo A 1.47 BS01 2EW A 1 G145 C147 G191 G192 Y193 V285 N286 Y334 G23 C25 G69 G70 Y71 V163 N164 Y212 Q141 C147 H287 N307 Q19 C25 H165 N185 3.4.22.27 0006508,0008234 remove_due_to_license_issue O70370 24224654 401 LPDTVDWREKGCVTEVKYQGSCGACWAFSAVGALEGQLKLKTGKLISLSAQNLVDCSNEEKYGNKGCGGGYMTEAFQYIIDNGGIEADASYPYKAMDEKCHYNSKNRAATCSRYIQLPFGDEDALKEAVATKGPVSVGIDASHSSFFFYKSGVYDDPSCTGNVNHGVLVVGYGTLDGKDYWLVKNSWGLNFGDQGYIRMARNNKNHCGIASYCSYPEI 4mzo A 1.47 BS02 2EW C 1 N312 Q316 N190 Q194 Q141 C147 H287 N307 Q19 C25 H165 N185 3.4.22.27 0006508,0008234 remove_due_to_license_issue O70370 24224654 401 LPDTVDWREKGCVTEVKYQGSCGACWAFSAVGALEGQLKLKTGKLISLSAQNLVDCSNEEKYGNKGCGGGYMTEAFQYIIDNGGIEADASYPYKAMDEKCHYNSKNRAATCSRYIQLPFGDEDALKEAVATKGPVSVGIDASHSSFFFYKSGVYDDPSCTGNVNHGVLVVGYGTLDGKDYWLVKNSWGLNFGDQGYIRMARNNKNHCGIASYCSYPEI 4mzr A 2.9 BS01 dna K 0 S241 R273 C275 A276 R280 S148 R180 C182 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 3 ~ 28 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzr A 2.9 BS02 dna L 0 R248 R283 R155 R190 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzr B 2.9 BS01 dna K 0 K120 F121 K27 F28 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 3 ~ 28 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzr B 2.9 BS02 dna L 0 F121 S241 R248 R273 A276 R280 F28 S148 R155 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzr C 2.9 BS01 dna K 0 R273 A276 R280 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 3 ~ 28 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzr C 2.9 BS02 dna L 0 K120 F121 R248 K27 F28 R155 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzr D 2.9 BS01 dna L 0 S241 R273 A276 R280 S148 R180 A183 R187 ? 0000976,0003677,0003700,0005634,0006355,0006915,0051262 remove_due_to_license_issue P04637 24374182 27 ~ 52 SSSVPSQKTYQGSYGFRLGFLHSGTAKFGTCTYSPALNKMFVQLAKTVPVQLYVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERSSDSDGLAPPQHLIRVEGNLRAEYLDDPNTFRHSVVVPYEPPEVGSDYTTIYFKFMCNSSCMGGMNRRPILVIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKKTMDGEYFTLQIRGRERFEQFRERNEALELKDAQAT 4mzs A 1.85 BS01 2EV A 1 G145 C147 K187 G191 G192 Y193 M194 V285 N286 Y334 G23 C25 K65 G69 G70 Y71 M72 V163 N164 Y212 Q141 C147 H287 N307 Q19 C25 H165 N185 3.4.22.27 0006508,0008234 remove_due_to_license_issue O70370 24224654 401 LPDTVDWREKGCVTEVKYQGSCGACWAFSAVGALEGQLKLKTGKLISLSAQNLVDCSNEEKYGNKGCGGGYMTEAFQYIIDNGGIEADASYPYKAMDEKCHYNSKNRAATCSRYIQLPFGDEDALKEAVATKGPVSVGIDASHSSFFFYKSGVYDDPSCTGNVNHGVLVVGYGTLDGKDYWLVKNSWGLNFGDQGYIRMARNNKNHCGIASYCSYPEI 4n00 A 1.8 BS01 2EX A 1 G72 Q73 G74 L91 D93 Y132 W137 F169 W176 D289 G291 G13 Q14 G15 L32 D34 Y73 W78 F110 W117 D223 G225 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=9.5nM remove_due_to_license_issue IC50=9.9nM P56817 24397738 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4n07 A 1.87 BS01 2J9 A 1 K104 P105 F106 M107 S108 K104 P105 F106 M107 S108 ? 0015276,0016020 Kd=0.35uM remove_due_to_license_issue EC50=900nM P19491 24131202 301 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECG 4n07 B 1.87 BS01 2J9 B 1 P105 S217 K218 G219 P104 S216 K217 G218 ? 0015276,0016020 Kd=0.35uM remove_due_to_license_issue EC50=900nM P19491 24131202 301 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGEC 4n07 B 1.87 BS04 2J9 C 1 P105 F106 M107 P104 F105 M106 ? 0015276,0016020 Kd=0.35uM remove_due_to_license_issue EC50=900nM P19491 24131202 301 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGEC 4n1b A 2.55 BS01 2FS A 1 Y334 N382 N414 R415 A556 Y572 S602 Y9 N57 N89 R90 A231 Y247 S277 ? remove_due_to_license_issue Q14145 24504667 701 RLIYTAGGYFRQSLSYLEAYNPSDGTWLDLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVTLE 4n1t A 1.6 BS01 2GD A 1 N33 G37 F72 M81 V83 W117 D119 D120 F139 N31 G35 F70 M79 V81 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=0.8nM remove_due_to_license_issue IC50=0.800000nM P36639 24695224 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 4n1u A 1.6 BS01 2GE A 1 F27 N33 F72 F74 W117 D119 D120 F139 F25 N31 F70 F72 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=5nM remove_due_to_license_issue IC50=5.0nM, EC50=126nM P36639 24695224 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDT 4n1z F 2.35 BS05 N1Z F 1 F99 D103 D107 R112 Q171 K200 D243 K257 F86 D90 D94 R99 Q158 K185 D228 K242 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 25411474 406 VYAQEKQDFVQHFSQIVRVLTHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKI 4n2q A 2.8 BS01 rna B 0 Y169 T172 R176 D203 Y205 Y126 T129 R133 D160 Y162 ? 0000373,0003723,0009658,0042802 remove_due_to_license_issue I1HB13 24186060 5 ~ 9 SLSTEAIHAVQALKRLTAADRSPPAATAAASAALGRLLRADLLAAMAELQRQGHWSLALAALHVARAEPWYRPDPELYATFVSSSPSNDPAAAAAVDALVEAFIEEKERGAAGGSSEGVWVGEDVYKLTRLVRALVAKGRARAAWRVYEAAVRKGGCEVDEYMYRVMAKGMKRLGLDEEAAEVEADLADWEARHLPDE 4n2s A 3.0 BS01 rna B 0 Y169 T172 R173 R176 D203 Y205 Y126 T129 R130 R133 D160 Y162 ? 0000373,0003723,0009658,0042802 remove_due_to_license_issue I1HB13 24186060 3 ~ 6 SLSTEAIHAVQALKRLTAADRSPPAATAAASAALGRLLRADLLAAMAELQRQGHWSLALAALHVARAEPWYRPDPELYATFVSSSPSNDPAAAAAVDALVEAFIEEKERGAAGGSSEGVWVGEDVYKLTRLVRALVAKGRARAAWRVYEAAVRKGGCEVDEYMYRVMAKGMKRLGLDEEAAEVEADLADWEARHLPD 4n3r A 1.9 BS02 2GU A 1 H1184 G1185 F1188 D1198 H1201 I1212 Y1213 S1221 Y1224 E1291 H81 G82 F85 D95 H98 I109 Y110 S118 Y121 E188 2.4.2.-,2.4.2.30 0003950 ic50=0.15uM remove_due_to_license_issue O95271 24900633 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEH 4n4s A 2.2 BS01 2H1 A 1 V37 A50 K52 I54 I82 I101 M106 L154 L164 V30 A43 K45 I47 I75 I94 M99 L147 L157 D147 K149 S151 N152 D165 T188 D140 K142 S144 N145 D158 T174 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 remove_due_to_license_issue P63086 24704509 401 GPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVADLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKILDFGLARVADPDTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 4n4t A 2.315 BS02 2GV A 1 H1184 F1188 A1191 I1192 F1197 D1198 H1201 F1208 Y1213 H81 F85 A88 I89 F94 D95 H98 F105 Y110 2.4.2.-,2.4.2.30 0003950 ic50=0.049uM remove_due_to_license_issue Q6PFX9 24900633 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEH 4n4v A 2.0 BS02 2GY A 1 H1184 S1186 P1187 F1188 A1191 F1197 D1198 H1201 F1208 Y1213 H81 S83 P84 F85 A88 F94 D95 H98 F105 Y110 2.4.2.-,2.4.2.30 0003950 ic50=0.002uM remove_due_to_license_issue O95271 24900633 1402 QGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPE 4n5d A 2.06 BS01 2FQ A 1 N125 Y198 L200 N101 Y163 L165 P62 E63 H121 G122 A163 R164 P38 E39 H97 G98 A139 R140 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 Kd=607uM remove_due_to_license_issue P55212 24259468 401 FYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPDTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4n5d B 2.06 BS01 2FQ A 1 Y198 L200 Y150 L152 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4n5g A 2.11 BS01 K09 A 1 L433 L436 F438 F439 I442 G443 L171 L174 F176 F177 I180 G181 ? 0003677,0003707,0005634,0006355,0008270 ic50=14.5uM remove_due_to_license_issue IC50=10000nM P19793 24704507 501 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4n6g A 2.142 BS01 2GQ B 1 Y198 L200 Y163 L165 P62 E63 H121 G122 A163 R164 P38 E39 H97 G98 A139 R140 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 FYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPDTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4n6g B 2.142 BS01 2GQ B 1 Y198 L200 Y150 L152 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4n6h A 1.8 BS01 EJ4 A 1 D128 Y129 M132 V217 W274 V281 G307 Y308 D198 Y199 M202 V287 W344 V351 G377 Y378 ? 0004930,0004985,0005506,0007186,0009055,0016020,0020037,0022900,0038046,0042597,0046872 remove_due_to_license_issue P0ABE7,P41143 24413399 1219 DLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCG 4n6y A 2.6 BS01 2HV A 1 L44 F49 V52 K67 R122 V126 L174 I185 D186 L13 F18 V21 K36 R91 V95 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue Ki=90nM P11309 24900629 401 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4n6z A 2.2 BS01 2HW A 1 F49 V52 A65 K67 I104 R122 D128 E171 L174 I185 D186 F17 V20 A33 K35 I72 R90 D96 E139 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=16nM remove_due_to_license_issue Ki=16nM P11309 24900629 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4n70 A 2.1 BS01 2HX A 1 L44 F49 A65 K67 I104 R122 V126 D128 E171 L174 I185 D186 L13 F18 A34 K36 I73 R91 V95 D97 E140 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=0.001nM remove_due_to_license_issue IC50=1nM, Ki=<1.000000nM P11309 24900629 401 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 4n7e A 2.7 BS01 2JQ A 1 Y271 F273 G274 F281 A282 S283 R292 I294 F317 Y318 Y362 Y211 F213 G214 F221 A222 S223 R232 I234 F257 Y258 Y302 ? 0016020 remove_due_to_license_issue Ki=429nM, IC50=450nM Q99523 24355129 807 GRVRDFVAKLANNTHQHVFDDLRGSVSLSWVGDSTGVILVLTTFHVPQSKLYRSEDYGKNFKDITDLINNTFIRTEFGMAIGPENSGKVVLTAEVSGGSRGGRIFRSSDFAKNFVQTDLPFHPLTQMMYSPQNSDYLLALSTENGLWVSKNFGGKWEEIHKAVCLAKWGSDNTIFFTTYANGSCKADLGALELWRTSDLGKSFKTIGVKIYSFGLGGRFLFASVMADKDTTRRIHVSTDQGDTWSMAQLPSVGQEQFYSILAANDDMVFMHVDEPGDTGFGTIFTSDDRGIVYSKSLDRHLYTTTGGETDFTNVTSLRGVYITSVLSEDNSIQTMITFDQGGRWTHLRKPENSECDATAKNKNECSLHIHASYSISQKLNVPMAPLSEPNAVGIVIAHGSVGDAISVMVPDVYISDDGGYSWTKMLEGPHYYTILDSGGIIVAIEHSSRPINVIKFSTDEGQCWQTYTFTRDPIYFTGLASEPGARSMNISIWGFTESTSQWVSYTIDFKDILERNCEEKDYTIWLAHSTDPEDYEDGCILGYKEQFLRLRKSSMCQNGRDYVVTKQPSICLCSLEDFLCDFGYYRPENDSKCVEQPELKGHDLEFCLYGREEHLTTNGYRKIPGDKCQGGVNPVREVKDLKKKCTSNFLSPE 4n7j A 1.673 BS01 2GQ B 1 Y198 T199 L200 Y162 T163 L164 P62 E63 H121 G122 A163 R164 P38 E39 H97 G98 A139 R140 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 FYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4n7j B 1.673 BS01 2GQ B 1 Y198 T199 Y150 T151 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4n7m A 2.125 BS01 2GQ A 1 Y198 T199 L200 Y162 T163 L164 P62 E63 H121 G122 A163 R164 P38 E39 H97 G98 A139 R140 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 Kd=3.4uM remove_due_to_license_issue P55212 24259468 401 FYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4n7m B 2.125 BS01 2GQ A 1 Y198 T199 Y150 T151 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4n7u A 1.4598 BS01 2JA A 1 R412 R418 R469 R116 R122 R173 ? Kd=0.51uM remove_due_to_license_issue IC50=7870nM, EC50=2.0nM O00481 24703779 501 GAYNEWKKALFKPADVILDPKTADPILLVSEDQRSVERAKEPQDLPDNPERFNWHYCVLGCESFISGRHYWEVEVGDRKEWHIGVCSKNVQRKGWVKMTPENGFWTMGLTDGNKYRTLTEPRTNLKLPKPPKKVGVFLDYETGDISFYNAVDGSHIHTFLDVSFSEALYPVFRILTLEPTALTICP 4n8d A 1.65 BS01 2KS A 1 E205 E206 R358 Y662 Y666 V711 E166 E167 R319 Y623 Y627 V672 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=11.9uM remove_due_to_license_issue P27487 24439847 815 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLIDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 4n8e A 2.3 BS01 2KV A 1 E205 E206 F357 S630 Y662 Y666 E166 E167 F318 S591 Y623 Y627 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.02uM remove_due_to_license_issue P27487 24439847 815 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLIDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 4n8q A 2.08 BS01 FA0 A 1 N138 A179 P180 H183 Y186 R187 A190 N115 A155 P156 H159 Y162 R163 A166 V106 V83 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 Ki=380uM remove_due_to_license_issue P9WFX5 24712732 601 VPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4n8r A 2.03 BS01 K08 A 1 A271 L436 F438 F439 I442 A9 L174 F176 F177 I180 ? 0003677,0003707,0005634,0006355,0008270 ic50=16.8uM remove_due_to_license_issue Kd=2050nM, IC50=10000nM P19793 24704507 501 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPH 4n98 A 1.7 BS01 4FC A 1 R152 Y154 T172 G174 R176 P242 V247 M362 R146 Y148 T166 G168 R170 P236 V241 M356 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=280uM remove_due_to_license_issue P0A988 24592885 401 MKFTVEREHLLKPLQQVSGTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4n99 A 2.3 BS01 2J1 A 1 H175 P242 V247 S346 H169 P232 V237 S336 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=216uM remove_due_to_license_issue P0A988 24592885 401 MKFTVEREHLLKPLQQVSGPLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4n9a A 1.9 BS02 2J2 A 1 G174 R176 L177 V247 M362 G166 R168 L169 V239 M354 2.7.7.7 0003677,0003887,0005515,0005737,0005829,0006260,0006261,0006271,0006974,0008408,0009360,0030174,0030894,0032297,0042276,0042802,0042803,0044787,1990078,1990085 Ki=64uM remove_due_to_license_issue P0A988 24592885 404 MKFTVEREHLLKPLQQVSLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4n9b A 2.859 BS01 2HH A 1 F193 R196 D219 V242 A244 S275 R311 I351 F176 R179 D202 V225 A227 S258 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue IC50=91000nM, Kd=5200nM P43490 24433859 602 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9b B 2.859 BS01 2HH B 1 F193 R196 D219 V242 A244 S275 R311 I351 F176 R179 D202 V225 A227 S258 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 remove_due_to_license_issue IC50=91000nM, Kd=5200nM P43490 24433859 602 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9c A 1.751 BS01 2ZM A 1 H191 F193 D219 S241 V242 A244 S275 I351 H174 F176 D202 S224 V225 A227 S258 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Kd=126uM remove_due_to_license_issue P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9c B 1.751 BS01 2ZM B 1 H191 F193 D219 S241 V242 A244 S275 I351 H174 F176 D202 S224 V225 A227 S258 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Kd=126uM remove_due_to_license_issue P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9d A 1.701 BS01 2HJ A 1 Y188 H191 F193 R196 D219 V242 A244 S275 Y171 H174 F176 R179 D202 V225 A227 S258 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.019uM remove_due_to_license_issue IC50=19nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9d A 1.701 BS02 2HJ B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.019uM remove_due_to_license_issue IC50=19nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9d B 1.701 BS01 2HJ A 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.019uM remove_due_to_license_issue IC50=19nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9d B 1.701 BS02 2HJ B 1 Y188 H191 F193 R196 D219 V242 S275 Y171 H174 F176 R179 D202 V225 S258 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.019uM remove_due_to_license_issue IC50=19nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9e A 1.72 BS01 2HL A 1 K189 H191 F193 R196 D219 V242 A244 S275 I309 R311 R349 I351 E376 N377 I378 A379 K173 H175 F177 R180 D203 V226 A228 S259 I293 R295 R333 I335 E360 N361 I362 A363 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM remove_due_to_license_issue IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9e A 1.72 BS02 2HL B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM remove_due_to_license_issue IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4n9e B 1.72 BS01 2HL A 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM remove_due_to_license_issue IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4n9e B 1.72 BS02 2HL B 1 K189 H191 F193 R196 D219 V242 A244 S275 I309 R311 R349 I351 E376 N377 I378 A379 K172 H174 F176 R179 D202 V225 A227 S258 I292 R294 R332 I334 E359 N360 I361 A362 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM remove_due_to_license_issue IC50=15nM P43490 24433859 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4na4 A 2.5 BS01 A1R A 1 T718 I719 E720 F731 N733 V746 Q747 E748 E749 Y788 N862 G864 G866 A867 F868 F895 T268 I269 E270 F281 N283 V296 Q297 E298 E299 Y338 N412 G414 G416 A417 F418 F445 3.2.1.143 0004649,0005975,0006282 remove_due_to_license_issue O88622 24465839 1001 KKWLGTPIEEMRKMPRCGIHLPSLRPSASHTVTVRVDLLRAGEVPKPFPTHYKDLWDNKHVKMPCSEQNLYPVTAGSRWELIQTALLNKFTRPQNLKDAILKYNVAYSKKWDFTALVDFWDKVLEEAEAQHLYQSILPDMVKIALCLPNICTQPIPLLKQKMNHSVTMSQEQIASLLANAFFCTFPRRNAKMKSEYSSYPDINFNRLFEGRSSRKPEKLKTLFCYFRRVTEKKPTGLVTFTRQSLEDFPEWERCEKPLTRLHVTYEGTIEGNGRGMLQVDFANRFVGGGVTGAGLVQEEIRFLINPELIVSRLFTEVLDHNECLIITGTEQYSEYTGYAETYRWARSHEDGSEKDDWQRRCTEIVAIDALHFRRYLDQFVPEKVRRELNKAYCGFLRPGVPSENLSAVATGNWGCGAFGGDARLKALIQILAAAAAERDVVYFTFGDSELMRDIYSMHTFLTERKLDVGKVYKLLLRYYNEECRNCSTPGPDIKLYPFIYHAVES 4na7 A 2.8 BS01 1T5 A 1 L41 H57 Y58B D189 A190 K192 G193 S195 S214 W215 G216 G218 C219 L28 H44 Y47 D182 A183 K185 G186 S188 S207 W208 G209 G211 C212 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue Ki=0.200000nM P03951 24405333 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYTDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4na8 A 2.3 BS01 1T6 A 1 R39 L41 H57 D189 A190 K192 G193 S195 S214 W215 G216 G218 C219 R26 L28 H44 D182 A183 K185 G186 S188 S207 W208 G209 G211 C212 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=1.5nM remove_due_to_license_issue Ki=1.5nM P03951 24405333 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYTDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4na9 H 2.24 BS01 1T7 H 1 H57 D189 S190 K192 G193 S195 S214 W215 G216 G219 C220 H41 D186 S187 K189 G190 S192 S211 W212 G213 G215 C216 3.4.21.21 0004252,0006508 Ki=41nM remove_due_to_license_issue P08709 24405333 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4nah A 2.38 BS02 2VJ A 1 E135 Y139 E134 Y138 H19 K43 R92 S130 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 remove_due_to_license_issue P63820 24041904 202 EHTIAVIPGSFDPITYGHLDIIERSTDRFDEIHVCVLKNSKKEGTFSLEERMDLIEQSVKHLPNVKVHQFSGLLVDYCEQVGAKTIIRGLRAVSDFEYELRLTSMNKKLNNEIETLYMMSSTNYSFISSSIVKEVAAYRADISEFVPPYVEKALKKKFK 4nah A 2.38 BS03 2VJ A 2 P9 S11 C36 V37 L75 R89 Y99 N107 P8 S10 C35 V36 L74 R88 Y98 N106 H19 K43 R92 S130 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 remove_due_to_license_issue P63820 24041904 203 EHTIAVIPGSFDPITYGHLDIIERSTDRFDEIHVCVLKNSKKEGTFSLEERMDLIEQSVKHLPNVKVHQFSGLLVDYCEQVGAKTIIRGLRAVSDFEYELRLTSMNKKLNNEIETLYMMSSTNYSFISSSIVKEVAAYRADISEFVPPYVEKALKKKFK 4nah C 2.38 BS01 2VJ A 1 P9 C36 L74 L75 R89 N107 P9 C36 L74 L75 R89 N107 H19 K43 R92 S130 H19 K43 R92 S130 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 remove_due_to_license_issue P63820 24041904 202 MEHTIAVIPGSFDPITYGHLDIIERSTDRFDEIHVCVLKNSKKEGTFSLEERMDLIEQSVKHLPNVKVHQFSGLLVDYCEQVGAKTIIRGLRAVSDFEYELRLTSMNKKLNNEIETLYMMSSTNYSFISSSIVKEVAAYRADISEFVPPYVEKALKKKFK 4nak A 1.8 BS01 PBQ A 1 V161 Q238 V239 S264 I265 V266 V77 Q149 V150 S175 I176 V177 2.7.7.60 0003824,0008299,0050518,0070567 ic50=1.4uM remove_due_to_license_issue P69834 24446431 401 EKSVSVILLAGGPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERIL 4nal A 1.8 BS01 H70 A 1 V161 Q238 V239 S264 I265 V266 V78 Q151 V152 S177 I178 V179 2.7.7.60 0003824,0008299,0050518,0070567 ic50=2.2uM remove_due_to_license_issue P69834 24446431 401 MEKSVSVILLAGGPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILSE 4nan A 1.8 BS01 2JM A 1 V161 V204 Q238 I265 V76 V119 Q148 I175 2.7.7.60 0003824,0008299,0050518,0070567 ic50=19uM remove_due_to_license_issue P69834 24446431 401 EKSVSVILLAGPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERIL 4nat A 1.72 BS01 2W5 A 1 C36 G73 L74 L75 L103 N107 C35 G66 L67 L68 L96 N100 H19 R92 S130 H18 R85 S123 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 remove_due_to_license_issue P63820 24041904 201 EHTIAVIPGSFDPITYGHLDIIERSTDRFDEIHVCVLGTFSLEERMDLIEQSVKHLPNVKVHQFSGLLVDYCEQVGAKTIIRGLRAVSDFEYELRLTSMNKKLNNEIETLYMMSSTNYSFISSSIVKEVAAYRADISEFVPPYVEKALKKKFK 4nat B 1.72 BS01 2W5 B 1 C36 L38 F71 G73 L74 L75 N107 C36 L38 F67 G69 L70 L71 N103 H19 R92 S130 H19 R88 S126 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 remove_due_to_license_issue P63820 24041904 201 MEHTIAVIPGSFDPITYGHLDIIERSTDRFDEIHVCVLKEGTFSLEERMDLIEQSVKHLPNVKVHQFSGLLVDYCEQVGAKTIIRGLRAVSDFEYELRLTSMNKKLNNEIETLYMMSSTNYSFISSSIVKEVAAYRADISEFVPPYVEKALKKKFK 4nau A 2.33 BS02 2W3 A 1 P9 C36 L38 K43 F71 G73 L74 L75 R89 Y99 L103 M106 N107 P8 C35 L37 K42 F70 G72 L73 L74 R88 Y98 L102 M105 N106 H19 K43 R92 S130 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 remove_due_to_license_issue P63820 24041904 202 EHTIAVIPGSFDPITYGHLDIIERSTDRFDEIHVCVLKNSKKEGTFSLEERMDLIEQSVKHLPNVKVHQFSGLLVDYCEQVGAKTIIRGLRAVSDFEYELRLTSMNKKLNNEIETLYMMSSTNYSFISSSIVKEVAAYRADISEFVPPYVEKALKKKFK 4nb6 A 2.85 BS01 444 A 1 W296 C299 L303 V340 M344 F367 H458 W52 C55 L59 V96 M100 F123 H214 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=60nM, EC50=54nM, Ki=51nM P51449 24239186 501 SLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIF 4nbk A 1.936 BS01 2J5 A 1 Y198 L200 P201 Y162 L164 P165 P62 E63 H121 G122 A163 R164 P38 E39 H97 G98 A139 R140 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 Kd=136uM remove_due_to_license_issue P55212 24259468 401 FYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4nbk B 1.936 BS01 2J5 A 1 V197 Y198 T199 E214 V149 Y150 T151 E166 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4nbl A 1.756 BS01 2J6 A 1 Y198 T199 L200 P201 Y164 T165 L166 P167 P62 E63 H121 G122 A163 R164 P39 E40 H98 G99 A140 R141 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 Kd=0.47uM remove_due_to_license_issue Kd=470nM P55212 24259468 401 AFYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPDTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4nbl B 1.756 BS01 2J6 A 1 A195 S196 V197 Y198 T199 E214 A146 S147 V148 Y149 T150 E165 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue Kd=470nM P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4nbn A 1.75 BS01 2J7 B 1 V197 Y198 T199 L200 P201 E214 V162 Y163 T164 L165 P166 E179 P62 E63 H121 G122 A163 R164 P38 E39 H97 G98 A139 R140 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 remove_due_to_license_issue P55212 24259468 401 FYKREMFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNQHDVPVIPDTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPKS 4nbn B 1.75 BS01 2J7 B 1 V197 Y198 T199 P201 E214 V148 Y149 T150 P152 E165 P62 E63 H121 G122 A163 R164 P33 E34 H92 G93 A134 R135 3.4.22.59 0002218,0004175,0004197,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0008234,0016540,0030855,0042802,0043065,0043067,0043525,0051604,0060545,0070269,0072332,0072734,0097153,0097284 Kd=44uM remove_due_to_license_issue P55212 24259468 401 MFDPAEKYKMDHRRRGIALIFNHERFFWHLTLPERRGTCADRDNLTRRFSDLGFEVKCFNDLKAEELLLKIHEVSTVSHADADCFVCVFLSHGEGNHIYAYDAKIEIQTLTGLFKGDKCHSLVGKPKIFIIQAARGNTNITEVDAASVYTLPAGADFLMCYSVAEGYYSHRETVNGSWYIQDLCEMLGKYGSSLEFTELLTLVNRKVSQRRVDFCKDPSAIGKKQVPCFASMLTKKLHFFPK 4ncg A 2.58 BS01 2KW A 1 L100 K103 V106 V179 Y181 Y188 V189 G190 W229 L234 H235 P236 Y318 L97 K100 V103 V176 Y178 Y185 V186 G187 W226 L231 H232 P233 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P04585 24412110 601 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGI 4ncm A 2.82 BS01 704 A 1 F323 F325 H357 E361 F404 M431 F3 F5 H37 E41 F84 M111 ? remove_due_to_license_issue P31345 25019388 501 SSFSFGGFTFKRTSGSSIKREEEVLTGNLQTLKIRVHEGYEEFTMVGKRATAILRKATRRLVQLIVSGKDEQSIAEAIIVAMVFSQEDCMIKAVRGDLNFVNRANQRLNPMHQLLRHFQKDAKVLFQNWGIEHIDNVMGMVGVLPDMTPSTEMSMRGIRVSKM 4ncn A 1.87 BS01 GTP A 1 V532 D533 T534 G535 K536 T537 K538 Q549 I556 T557 G597 N648 K649 D651 R652 S716 A717 H718 V16 D17 T18 G19 K20 T21 K22 Q33 I40 T41 G81 N132 K133 D135 R136 S200 A201 H202 3.6.5.3 0003924,0005525 remove_due_to_license_issue G0S8G9 24686316 1001 NKDNLRSPICCILGHVDTGKTKLLDKIRQTNVQEGEAGGITQQIGATYFPVEAIKQKTAVVNKDGKFEFKVPGLLIIDTPGHESFSNLRSRGSSLCNIAILVVDIMHGLEPQTIESLRLLRERKTPFVVALNKIDRLYGWKKIENNGFRESFALQNKAVQNEFRNRLDQVKLQFAEQGFNSELFYENKNFARYVSLVPTSAHTGEGIPDMLKLIVQLCQERMASSLMYLSELQATVLEVKAIEGFGVTIDVILSNGILREGDRIVLCGLEGPIKTNIRALLTPAPMRELRIKGQYIHHKEVKAAQGVKISAPGLEGAIAGSRLLVVGPDDDEEELEEEVESDLQ 4nct A 2.597 BS01 2K2 A 1 I165 G166 V173 A186 M240 E291 D307 I32 G33 V40 A53 M107 E158 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Kd=100nM Q13627 25945585 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 4ndu A 1.301 BS01 AMG A 1 N6 F13 H69 G70 S72 N73 N6 F13 H69 G70 S72 N73 ? 0005534,0030246 remove_due_to_license_issue A7UNK4 25504801 101 ACWKANSCPGSAFESKDRLRSFALLYCRYNYKPPYGQGAFGYASAVSTHGWETEAQCINTFEQIITSCHGQSNGGTLELNSGRLSLAFGNCEEL 4ng9 H 2.2 BS01 2KE H 1 H57 D60 G97 T98 T99 D102 D189 S190 K192 S195 S214 W215 G216 G219 H41 D44 G85 T86 T87 D90 D182 S183 K185 S188 S207 W208 G209 G211 3.4.21.21 0004252,0006508 remove_due_to_license_issue P08709 24900796 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4nga H 2.15 BS01 2KF H 1 L41 H57 K60A P170I D189 S190 K192 S195 V213 S214 W215 G216 Q217 G219 L25 H41 K45 P169 D186 S187 K189 S192 V210 S211 W212 G213 Q214 G215 3.4.21.21 0004252,0006508 remove_due_to_license_issue P08709 24900796 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4ngb A 2.25 BS01 rna B 0 Y926 R927 F950 P951 S952 F958 Y961 Y962 K965 Y966 S1006 W1014 L1017 Q1021 I1022 Y160 R161 F184 P185 S186 F192 Y195 Y196 K199 Y200 S229 W237 L240 Q244 I245 3.1.26.3 0003723 remove_due_to_license_issue Q9UPY3 24486018 1 ~ 12 QPCYLYVIGMVLTTPLPDELNFRRRKLYPPEDTTRCFGILTAKPIPQIPHFPVYTRSGEVTISIELAASGFMLSLQMLELITRLHQYIFSHILRLEKPALAYCVLPLNVVSSTLDIDFKFMEDIEKSEARIGIPSTKYTKETPFVFKLEDYQDAVIIPRYRNFDQPHRFYVADVYTDLTPLSKFPSPEYETFAEYYKTKYNLDLTNLNQPLLDVDHTSSRLNLLTPLSSAEKRKAKWESLQNKQILVPELCAIHPIPASLWRKAVCLPSILYRLHC 4ngm A 1.84 BS04 JB7 A 1 G206 K207 R210 E424 L428 G518 N519 R536 F546 S547 G548 Y552 H553 K699 Y700 A701 G152 K153 R156 E370 L374 G464 N465 R482 F492 S493 G494 Y498 H499 K645 Y646 A647 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Ki=0.044900nM Q04609 24954515 821 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4ngn A 1.64 BS04 J96 A 1 R210 N257 E424 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 L374 G464 N465 R480 R482 Y498 H499 K645 Y646 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Q04609 24954515 819 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4ngp A 1.63 BS01 J31 A 1 R210 E424 L428 E457 R463 G518 N519 R536 W541 N544 F546 Y552 H553 K699 Y700 A701 R156 E370 L374 E403 R409 G464 N465 R482 W487 N490 F492 Y498 H499 K644 Y645 A646 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Ki=11nM Q04609 24954515 817 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4ngq A 2.08 BS04 J37 A 1 R210 N257 E424 L428 R463 D465 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 L374 R409 D411 G464 N465 R480 R482 Y496 H497 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Q04609 24954515 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4ngr A 1.9 BS01 J21 A 1 K207 R210 N257 E424 L428 R463 G518 N519 R534 R536 G548 Y552 H553 N698 K699 Y700 K153 R156 N203 E370 L374 R409 G464 N465 R480 R482 G487 Y491 H492 N637 K638 Y639 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Ki=0.268000nM Q04609 24954515 814 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4ngs A 1.68 BS01 J34 A 1 R210 E424 L428 E457 R463 G518 N519 R536 W541 N544 F546 G548 Y552 H553 N698 K699 Y700 R156 E370 L374 E403 R409 G464 N465 R482 W487 N490 F492 G494 Y498 H499 N644 K645 Y646 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Ki=0.377000nM Q04609 24954515 815 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4ngt A 2.31 BS04 J42 A 1 R210 N257 E424 R463 G518 N519 R536 T538 W541 Y552 H553 K699 Y700 A701 R156 N203 E370 R409 G464 N465 R482 T484 W487 Y494 H495 K641 Y642 A643 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Ki=3.9nM Q04609 24954515 815 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4nh7 A 2.0 BS01 E0G A 1 A55 K58 M98 L107 F138 Y139 W162 A39 K42 M82 L91 F122 Y123 W146 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=4nM remove_due_to_license_issue Kd=4.0nM P07900 24332488 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSFIGYPITLFVEK 4nh8 A 1.65 BS01 2LC A 1 A55 K58 M98 F138 Y139 W162 A40 K43 M83 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=3nM remove_due_to_license_issue P07900 24332488 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4nh9 A 2.77 BS01 2LC A 1 N107 A111 M154 N162 F199 Y200 W223 T245 N35 A39 M82 N90 F116 Y117 W140 T162 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Ki=375nM P14625 24332488 401 SEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALSGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNFLNKMTEAQEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTEKTVWDWELMN 4nhj A 2.701 BS01 dna C 0 S162 R190 V203 R207 R226 S29 R57 V70 R74 R93 ? 0000160,0003677,0006355 remove_due_to_license_issue A6T8N1 24990372 2 ~ 23 PHKTISFGSLTIDPVNRQVMLGGENVALSTADFDMLWELATHAGQIMDRDALLKNLRGVTYDGMDRSVDVAISRLRKKLLDNATEPYRIKTVRNKGYLFAPH 4nhj A 2.701 BS02 dna D 0 R182 R199 V203 S206 A216 T224 R226 N227 Y230 R49 R66 V70 S73 A83 T91 R93 N94 Y97 ? 0000160,0003677,0006355 remove_due_to_license_issue A6T8N1 24990372 1 ~ 23 PHKTISFGSLTIDPVNRQVMLGGENVALSTADFDMLWELATHAGQIMDRDALLKNLRGVTYDGMDRSVDVAISRLRKKLLDNATEPYRIKTVRNKGYLFAPH 4nhj B 2.701 BS01 dna C 0 S162 A164 R190 R199 V203 R207 S28 A30 R56 R65 V69 R73 ? 0000160,0003677,0006355 remove_due_to_license_issue A6T8N1 24990372 2 ~ 23 HKTISFGSLTIDPVNRQVMLGGENVALSTADFDMLWELATHAGQIMDRDALLKNLRGVTYDGMDRSVDVAISRLRKKLLDNATEPYRIKTVRNKGYLFAPH 4nhj B 2.701 BS02 dna D 0 R182 R199 S206 A216 T224 R226 N227 Y230 R48 R65 S72 A82 T90 R92 N93 Y96 ? 0000160,0003677,0006355 remove_due_to_license_issue A6T8N1 24990372 1 ~ 23 HKTISFGSLTIDPVNRQVMLGGENVALSTADFDMLWELATHAGQIMDRDALLKNLRGVTYDGMDRSVDVAISRLRKKLLDNATEPYRIKTVRNKGYLFAPH 4nhx A 2.105 BS02 OGA A 1 L152 H155 I167 Y169 H218 V220 R230 L129 H132 I144 Y146 H195 V197 R207 1.14.11.- 0005506,0005515,0005634,0005654,0005737,0005829,0006449,0008283,0010494,0016705,0016706,0018126,0019511,0031418,0031543,0031544,0034063,0046872,0051213 remove_due_to_license_issue Q8N543 25728928 603 AEFSDAVTEETLKKQVAEAWSRRTPFSHEVIVMDMDPFLHCVIPNFIQSQDFLEGLQKELMNLDFHEKYNDLYKFQQSDDLKKRREPHISTLRKILFEDFRSWLSDISKIDLESTIDMSCAKYEFTDALLCHDDELEGRRIAFILYLVPPWDRSMGGTLDLYSIDEHFQPKQIVKSLIPSWNKLVFFEVSPVSFHQVSEVLSEEKSRLSISGWFHGPSLTRPPNYFEPPIPRSPHIPQDHEILYDWINPTYLDMDYQVQIQEEFEESSEILLKEFLKPEKFTKVCEALEHGHVEWSSRGPPNKRFYEKAEESKLPEILKECMKLFRSEALFLLLSNFTGLKLHFLAPSSSVPMCQGELRHWKTGHYTLIHAEFALDLILYCGCEGWEPEYGGFTSYIAKGEDEELLTVNPESNSLALVYRDRETLKFVKHINHRSLEQKKTFPNRTGFWDFSFIYYE 4nhy A 2.603 BS02 PD2 A 1 L152 I167 L182 H218 V220 R230 L129 I144 L159 H195 V197 R207 1.14.11.- 0005506,0005515,0005634,0005654,0005737,0005829,0006449,0008283,0010494,0016705,0016706,0018126,0019511,0031418,0031543,0031544,0034063,0046872,0051213 remove_due_to_license_issue Q8N543 25728928 603 AEFSDAVTEETLKKQVAEAWSRRTPFSHEVIVMDMDPFLHCVIPNFIQSQDFLEGLQKELMNLDFHEKYNDLYKFQQSDDLKKRREPHISTLRKILFEDFRSWLSDISKIDLESTIDMSCAKYEFTDALLCHDDELEGRRIAFILYLVPPWDRSMGGTLDLYSIDEHFQPKQIVKSLIPSWNKLVFFEVSPVSFHQVSEVLSEEKSRLSISGWFHGPSLTRPPNYFEPPIPRSPHIPQDHEILYDWINPTYLDMDYQVQIQEEFEESSEILLKEFLKPEKFTKVCEALEHGHVEWSSRGPPNKRFYEKAEESKLPEILKECMKLFRSEALFLLLSNFTGLKLHFLAPSSSVPMCQGELRHWKTGHYTLIHDHSKAEFALDLILYCGCEGWEPEYGGFTSYIAKGEDEELLTVNPESNSLALVYRDRETLKFVKHINHRSLEQKKTFPNRTGFWDFSFIYYE 4ni7 A 2.4 BS01 dna B 0 R16 R24 K27 Q28 R30 Y31 L33 M117 S118 V121 F125 K171 Q175 L178 R1 R9 K12 Q13 R15 Y16 L18 M89 S90 V93 F97 K138 Q142 L145 ? 0005125,0005138,0005576,0005615,0006955,0030154 remove_due_to_license_issue P05231 24415767 1 RQPLTSSERIDKQIRYILDGISALRKETCNKSNLNLPKMAEKDGCFQSGFNEETCLVKIITGLLEFEVYLEYLQNRFESSEEQARAVQMSTKVLIQFLQKKAITTPDPTTNASLLTKLQAQNQWLQDMTTHLILRSFKEFLQSSLRALRQM 4nie A 2.01 BS03 NBH A 1 Q286 L287 W317 C320 R364 M365 R367 A368 F377 F378 F388 Q23 L24 W54 C57 R101 M102 R104 A105 F114 F115 F125 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=20nM, IC50=>25000nM P51449 24900774 601 YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFST 4nj3 A 1.848 BS01 2KD A 1 V18 A31 K33 L55 V64 F80 E81 F82 L134 A144 D145 F146 G147 L148 V18 A31 K33 L47 V56 F72 E73 F74 L126 A136 D137 F138 G139 L140 D127 K129 Q131 N132 D145 T165 D119 K121 Q123 N124 D137 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=0.3uM remove_due_to_license_issue Kd=300nM, IC50=>10000nM, Ki=140nM P24941 24332088 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLAEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 4nj9 H 1.95 BS01 2M9 H 1 G97 Y98 G99 R100A G100B G101 Y102 G103 R105 G106 ? remove_due_to_license_issue Q9D8L4 25756188 501 EVQLQQSGPELVKPGTSVKMSCKASGYTFTDYYMHWVKQSHGKSLEWIGYIYPNNGGNGYNQKFKGKATLTVDKSSSTAYMELRSLTSEDSAVYYCARRGGYGSRGYFDVWGTGTTVTVSSAKTTAPSVYPLAPVGSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPALLQSGLYTLSSSVTVTSNTWPSQTITCNVAHPASSTKVDKKIEPRG 4nj9 L 1.95 BS04 2M9 H 1 Y28 I30 F32 R50 Y32 I34 F36 R54 ? remove_due_to_license_issue Q52L95 25756188 501 DIVLTQSPASLAVSLGQRATISCRASESVDSYGISFMHWYQQKPGQPPKLLIYRASNLESGIPARFSGSGSRTDFTLTIIPVEADDVATYYCQQSNEDPRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATSPIVKSFNRNE 4nja H 2.204 BS01 2M9 H 1 G97 Y98 G99 I100 R100A G100B G101 Y102 G103 I104 R105 G106 ? remove_due_to_license_issue A0A0F7R1P3 25756188 501 EVQLQQSGPELVKPGASVKMSCKASGYTFTDYYMHWVKQSHGKSLEWIGYIYPNNGGNGYNQKFKGKATLTVDKSSSTAYMELRSLTSDDSAVYYCARRGGYGIRGYFDVWGTGTTVTVSSAKTTPPSVYPLAPGCGDTTGSSVTSGCLVKGYFPEPVTVTWNSGSLSSSVHTFPALLQSGLYTMSSSVTVPSSTWPSQTVTCSVAHPASSTTVDKKLEPS 4nja L 2.204 BS02 2M9 H 1 Y28 N30 F32 R50 Y32 N34 F36 R54 ? 0002250,0006955,0019814 remove_due_to_license_issue P01660,Q52L95 25756188 501 DIVLTQSPASLAVSLGQRATISCRASESVDSYGNSFMHWYQQKPGQPPKLLIYRASNLESGIPARFSGSGSRTDFTLTINPVEADDVATYYCQQSNEDPRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 4njd A 2.5 BS01 NJD A 1 G328 E329 V335 A348 M395 E396 F397 L398 G401 L447 S457 D458 G30 E31 V37 A50 M97 E98 F99 L100 G103 L149 S159 D160 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 ic50=0.79uM remove_due_to_license_issue IC50=790nM O96013 24704155 600 MSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 4nk3 A 1.9 BS01 MK7 A 1 S90 Q146 Y177 N179 Y249 T343 G344 S345 N347 S62 Q118 Y149 N151 Y221 T315 G316 S317 N319 S90 K93 Y177 E299 K342 S345 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 24433862 401 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLEQ 4nk9 A 2.57 BS01 2K5 A 1 L484 G485 G487 V492 A512 K514 E531 I545 V561 A564 G567 L630 D641 F642 L21 G22 G24 V29 A48 K50 E67 I81 V97 A100 G103 L153 D164 F165 D623 A625 R627 N628 D641 D146 A148 R150 N151 D164 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 24900792 807 ELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4nka A 2.19 BS01 2K7 A 1 L484 A512 E531 E562 Y563 A564 G567 L630 D641 L21 A45 E64 E95 Y96 A97 G100 L151 D162 D623 A625 R627 N628 D641 D144 A146 R148 N149 D162 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=447nM remove_due_to_license_issue P11362 24900792 805 ELPEDPRWELPRDRLVLGKPLGEQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4nks A 2.5 BS01 2M2 A 1 A512 K514 E531 V561 A564 L630 A36 K38 E54 V84 A87 L139 D623 A625 R627 N628 D641 D132 A134 R136 N137 D150 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=69.1nM remove_due_to_license_issue P11362 24900792 801 LPEDPRWELPRDRLVLGKPLGQVVLAEAINRVTKVAVKMLKDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS 4nkt A 1.9 BS01 2KH A 1 F88 S90 N171 K197 S211 Y212 H336 F51 S53 N127 K153 S167 Y168 H278 2.7.7.19,2.7.7.52 remove_due_to_license_issue O13833 24322298 401 DMSHKEFTKFCYEVYNEIKISDKEFKEKRAALDTLRLCLKRISPDAELVAFGSLESGLALKNSDMDLCVLMTIALQFYEELIAEGFEGKFLQRARIPIIKLTSDTKNGFGASFQCAIGFNNRLAIHNTLLLSSYTKLDARLKPMVLLVKHWAKRKQINSPYFGTLSSYGYVLMVLYYLIHVIKPPVFPNLLLSPLKQEKIVDGFDVGFDDKLEDIPPSQNYSSLGSLLHGFFRFYAYKFEPREKVVTFRRPDGYLTKQEKGWTSRYILAIEDPFEISHNVGRTVSSSGLYRIRGEFMAASRLLNSRSYPIPYDSLFEEA 4nl1 A 2.3 BS01 Z13 A 1 E236 M264 E235 M263 V28 D54 K220 R254 V27 D53 K219 R253 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue Q81VW8 24650357 301 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGESTRPGFAKVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4nl1 B 2.3 BS01 Z13 B 1 L235 M264 L223 M252 V28 D54 K220 R254 V27 D51 K208 R242 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue Q81VW8 24650357 301 KWDYDLRCGEYTLNLNEKTLIMGILNVTPFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 4nl3 A 3.1 BS01 rna R 0 Q6 Q9 N42 F43 K58 H59 Q5 Q8 N41 F42 K57 H58 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 17 ~ 22 KQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALN 4nl3 B 3.1 BS01 rna R 0 Q6 Q9 N42 F43 K58 H59 Q5 Q8 N41 F42 K57 H58 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 17 ~ 22 KQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVAL 4nl3 C 3.1 BS01 rna Z 0 Q6 N42 F43 K58 H59 Q6 N42 F43 K58 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 27 ~ 32 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALNP 4nl3 D 3.1 BS01 rna R 0 Q6 Q9 N42 F43 H59 Q6 Q9 N42 F43 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 17 ~ 22 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALN 4nl3 E 3.1 BS01 rna Z 0 Q6 N42 F43 K58 H59 Q5 N41 F42 K57 H58 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 27 ~ 32 KQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALN 4nl3 F 3.1 BS01 rna Z 0 Q6 Q9 N42 F43 K58 H59 Q6 Q9 N42 F43 K58 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 27 ~ 32 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALNPD 4nl3 G 3.1 BS01 rna R 0 Q6 Q9 N42 F43 K58 H59 Q6 Q9 N42 F43 K58 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 17 ~ 22 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALN 4nl3 H 3.1 BS01 rna R 0 Q6 Q9 N42 F43 K58 H59 Q5 Q8 N41 F42 K57 H58 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 17 ~ 22 KQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVAL 4nl3 I 3.1 BS01 rna Z 0 Q6 Q9 N42 F43 K58 H59 Q6 Q9 N42 F43 K58 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 27 ~ 32 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALNP 4nl3 J 3.1 BS01 rna R 0 Q6 Q9 N42 F43 H59 Q6 Q9 N42 F43 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 17 ~ 22 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALN 4nl3 K 3.1 BS01 rna Z 0 Q6 Q9 N42 F43 K58 H59 Q6 Q9 N42 F43 K58 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 27 ~ 32 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALN 4nl3 L 3.1 BS01 rna Z 0 Q6 Q9 N42 F43 K58 H59 Q6 Q9 N42 F43 K58 H59 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue Q92C58 25150227 27 ~ 32 MKQGGQGLQDYYLNQLRKEKILATVFLTNGFQLRGRVVSFDNFTVLLDVEGKQQLVFKHAISTFSPQKNVALNP 4nld A 2.75 BS01 2N7 A 1 L392 A393 A395 A396 I424 H428 L492 G493 V494 P495 W500 R503 L334 A335 A337 A338 I366 H370 L434 G435 V436 P437 W442 R445 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 24397558 601 FDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGG 4nm6 A 2.026 BS01 dna B 0 R1261 R1262 S1286 S1290 Y1294 K1299 S1303 D1384 Y1902 H1904 R122 R123 S147 S151 Y155 K160 S164 D245 Y385 H387 1.14.11.80 0070579,0141167 remove_due_to_license_issue Q6N021 24315485 1 ~ 11 SCRCEGPFYTHLGAGPNVAAIREIMEERFGQKGKAIRIERVIYTGKEGKSSQGCPIAKWVVRRSSSEEKLLCLVRERAGHTCEAAVIVILILVWEGIPLSLADKLYSELTETLRKYGTLTNRRCALNEERTCACQGLDPETCGASFSFGCSWSMYYNGCKFARSKIPRKFKLLGDDPKEEEKLESHLQNLSTLMAPTYKKLAPDAYNNQIEYEHRAPECRLGLKEGRPFSGVTACLDFCAHAHRDLHNMQNGSTLVCTLTREDNREFGGKPEDEQLHVLPLYKVSDVDEFGSVEAQEEKKRSGAIQVLSSFRRKVRMLAEPVKTGSDEVWSDSEQSFLDPDIGGVAVAPTHGSILIECAKRELHATTPLKNPNRNHPTRISLVFYQHKSMNEPKHGLALWEAKMAEK 4nm6 A 2.026 BS02 dna C 0 W1291 M1293 Y1294 N1296 W152 M154 Y155 N157 1.14.11.80 0070579,0141167 remove_due_to_license_issue Q6N021 24315485 3 ~ 12 SCRCEGPFYTHLGAGPNVAAIREIMEERFGQKGKAIRIERVIYTGKEGKSSQGCPIAKWVVRRSSSEEKLLCLVRERAGHTCEAAVIVILILVWEGIPLSLADKLYSELTETLRKYGTLTNRRCALNEERTCACQGLDPETCGASFSFGCSWSMYYNGCKFARSKIPRKFKLLGDDPKEEEKLESHLQNLSTLMAPTYKKLAPDAYNNQIEYEHRAPECRLGLKEGRPFSGVTACLDFCAHAHRDLHNMQNGSTLVCTLTREDNREFGGKPEDEQLHVLPLYKVSDVDEFGSVEAQEEKKRSGAIQVLSSFRRKVRMLAEPVKTGSDEVWSDSEQSFLDPDIGGVAVAPTHGSILIECAKRELHATTPLKNPNRNHPTRISLVFYQHKSMNEPKHGLALWEAKMAEK 4nni A 2.64 BS01 VGL A 1 F307 R357 F30 R80 ? 0003676 remove_due_to_license_issue P9WH43 25430994 501 NLYFQHMRHFARTHAIGQIVPGKVTKLVPFGAFVRVEEGIEGLVHISELAERHVEVPDQVVAVGDDAMVKVIDIDLERRRISLSLKQANEDYTEEFDPAKYGMADSYDEQGNYIFPEGFDAETNEWLEGFEKQRAEWEARYAEAERRHKMHTAQMEKFAAA 4nni A 2.64 BS02 VGL A 2 F310 E318 R357 F33 E41 R80 ? 0003676 remove_due_to_license_issue P9WH43 25430994 502 NLYFQHMRHFARTHAIGQIVPGKVTKLVPFGAFVRVEEGIEGLVHISELAERHVEVPDQVVAVGDDAMVKVIDIDLERRRISLSLKQANEDYTEEFDPAKYGMADSYDEQGNYIFPEGFDAETNEWLEGFEKQRAEWEARYAEAERRHKMHTAQMEKFAAA 4nnn H 2.5 BS01 ALD H 1 T1 T21 G47 A49 T1 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 24403024 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4nnr A 1.98 BS01 FK5 A 1 Y56 D67 F76 V85 I86 W89 Y112 K120 F129 Y16 D27 F36 V45 I46 W49 Y72 K80 F89 Y56 F66 D67 I86 Y112 F129 Y16 F26 D27 I46 Y72 F89 5.2.1.8 0000413,0003755,0061077 remove_due_to_license_issue P26885 201 HCPIKSRKGDVLHMHYTGKLEDGTEFDSSLPQNQPFVFSLGTGQVIKGWDQGLLGMCEGEKRKLVIPSELGYGERGAPPKIPGGATLVFEVELLKIERRTEL 4nnu A 2.81 BS01 dna C 0 L58 L65 K69 K139 R140 R157 S160 Y162 Q179 L182 K186 K190 E208 Y211 R232 R233 T234 K236 L15 L22 K26 K96 R97 R114 S117 Y119 Q136 L139 K143 K147 E165 Y168 R189 R190 T191 K193 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 4nnu A 2.81 BS02 dna D 0 Y57 T78 I81 R82 A85 W88 R89 M143 K156 R157 R159 N163 F170 P178 Y14 T35 I38 R39 A42 W45 R46 M100 K113 R114 R116 N120 F127 P135 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 4nnu A 2.81 BS03 dna F 0 K52 Y103 K9 Y60 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 4nnu B 2.81 BS01 dna E 0 L58 L65 K69 R140 R157 Y162 L182 K183 K186 W189 K190 E208 Y211 R232 R233 T234 L15 L22 K26 R97 R114 Y119 L139 K140 K143 W146 K147 E165 Y168 R189 R190 T191 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTI 4nnu B 2.81 BS02 dna D 0 K52 Y103 W107 K9 Y60 W64 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTI 4nnu B 2.81 BS03 dna F 0 Y57 T78 I81 A85 W88 R89 Q100 K139 M143 K146 K147 K156 R157 R159 N163 P178 Y14 T35 I38 A42 W45 R46 Q57 K96 M100 K103 K104 K113 R114 R116 N120 P135 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTI 4nnw H 2.6 BS01 2MK H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 24403024 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4no1 K 2.5 BS01 CIX K 1 T1 A20 T21 G47 A49 T1 A20 T21 G47 A49 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 24403024 301 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4no6 K 3.0 BS01 2M1 K 1 T1 A20 T21 G47 A49 S131 T1 A20 T21 G47 A49 S131 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 24403024 301 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4no6 L 3.0 BS01 2M1 K 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 24403024 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4no8 K 2.7 BS01 2LV K 1 T1 T21 G47 A49 S131 T1 T21 G47 A49 S131 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 24403024 301 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4no9 H 2.9 BS01 2L0 H 1 T1 S20 T21 K33 G47 A49 G168 T1 S20 T21 K33 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 24403024 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4nod A 2.897 BS01 dna C 0 L58 L65 T77 R140 M143 K146 Y162 Q179 K186 W189 L15 L22 T34 R97 M100 K103 Y119 Q136 K143 W146 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod A 2.897 BS02 dna E 0 R232 R233 R189 R190 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod A 2.897 BS03 dna D 0 Y57 T78 I81 A85 W88 R89 Y103 W107 R140 R157 N163 A167 F170 P178 Y14 T35 I38 A42 W45 R46 Y60 W64 R97 R114 N120 A124 F127 P135 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod B 2.897 BS01 dna C 0 R232 R233 R189 R190 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod B 2.897 BS02 dna E 0 L58 L65 T77 R140 M143 K146 Y162 Q179 L182 K186 W189 E208 L15 L22 T34 R97 M100 K103 Y119 Q136 L139 K143 W146 E165 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod B 2.897 BS03 dna F 0 K52 S55 Y57 T78 I81 A85 R89 Y103 W107 R140 M143 K147 K156 R157 N163 A167 F170 P178 K9 S12 Y14 T35 I38 A42 R46 Y60 W64 R97 M100 K104 K113 R114 N120 A124 F127 P135 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod G 2.897 BS01 dna I 0 L58 L65 T77 R140 M143 K146 Y162 Q179 L182 K186 W189 E208 L15 L22 T34 R97 M100 K103 Y119 Q136 L139 K143 W146 E165 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod G 2.897 BS02 dna J 0 K52 S55 Y57 T78 A85 R89 Y103 W107 R140 M143 K156 R157 N163 V166 A167 F170 P178 K9 S12 Y14 T35 A42 R46 Y60 W64 R97 M100 K113 R114 N120 V123 A124 F127 P135 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod H 2.897 BS01 dna K 0 L58 L65 T77 R140 M143 K146 Y162 Q179 L182 K186 W189 E208 L15 L22 T34 R97 M100 K103 Y119 Q136 L139 K143 W146 E165 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4nod H 2.897 BS02 dna L 0 Y57 T78 I81 R82 A85 W88 R89 Y103 W107 R140 K156 R157 N163 A167 F170 P178 Y14 T35 I38 R39 A42 W45 R46 Y60 W64 R97 K113 R114 N120 A124 F127 P135 ? remove_due_to_license_issue Q00059 24435062 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRR 4non A 2.5 BS01 GDP A 1 N11 G13 K14 T15 S16 M114 D116 V117 S142 S143 L144 N11 G13 K14 T15 S16 M114 D116 V117 S142 S143 L144 ? 0005525 Kd=5.71uM remove_due_to_license_issue Q5M586 24649829 301 MTEIALIGNPNSGKTSLFNLITGHNQRVGNWPGVTVERKSGLVKKNKDLEIQDLPGIYSMSPYSPEEKVARDYLLSQRADSILNVVDATNLERNLYLTTQLIETGIPVTIALNMIDVLDGQGKKINVDKLSYHLGVPVVATSSLKQTGVDQVVKKAAHTTTSTVGDLAFPIYDDRLEAAISQILEVLGNSVPQRSARFYAIKLFEQDSLVEAELDLSQFQRKEIEDIIRITEEIFTEDAESIVINERYAFIERVCQMAES 4np2 A 1.75 BS01 2L1 A 1 N29 E41 R82 R155 N6 E18 R59 R132 ? 0005540,0007155,0016020 Kd=5.5mM remove_due_to_license_issue Kd=5500000nM P15379 24606063 201 NQIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4np3 A 1.61 BS01 2L2 A 1 N29 V30 E41 R82 V153 N154 R155 N6 V7 E18 R59 V130 N131 R132 ? 0005540,0007155,0016020 Kd=0.5mM remove_due_to_license_issue Kd=500000nM P15379 24606063 201 NQIDLNVTCRYAGVFHVEKNGRYSISRTEAADLCQAFNSTLPTMDQMKLALSKGFETCRYGFIEGNVVIPRIHPNAICAANHTGVYILVTSNTSHYDTYCFNASAPPEEDCTSVTDLPNSFDGPVTITIVNRDGTRYSKKGEYRTHQEDI 4np9 A 1.92 BS01 I3P A 1 Y421 K423 K435 R437 N481 V509 Y40 K42 K54 R56 N100 V128 ? 0016020 remove_due_to_license_issue P47709 24302762 601 TLGALEFSLLYDQDNSNLQCTIIRAKGLKPMDSNGLADPYVKLHLLPGASKSNKLRTKTLRNTRNPVWNETLQYHGITEEDMQRKTLRISVCDEDKFGHNEFIGETRFSLKKLKANQRKNFNICLERV 4npv A 2.4 BS01 0NK A 1 H223 I371 H373 L388 F392 L409 Q421 F424 H73 I221 H223 L238 F242 L259 Q271 F274 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=35nM Q01064 601 STAVLNCLKNLDLWCFDVFSLNQAADDHALRTIVFELLTRHNLISRFKIPTVFLMSFLDALETGYGKYKNPYHNQIHAADVTQTVHCFLLRTGMVHCLSEIELLAIIFAAAIHDYEHTGTTNSFHIQTKSECAIVYNDRSVLENHHISSVFRLMQDDEMNIFINLTKDEFVELRALVIEMVLATDMSCHFQQVKTMKTALQQLERIDKPKALSLLLHAADISHPTKQWLVHSRWTKALMEEFFRQGDKEAELGLPFSPLCDRTSTLVAQSQIGFIDFIVEPTFSVLTDVAEKSVQPPDVVSFRSTWVKRIQENKQKWKERAAS 4nq6 A 1.8 BS03 3R9 A 1 F34 W59 H88 D90 H149 C168 H210 F29 W54 H83 D85 H144 C163 H205 H86 H88 D90 H149 C168 K171 N180 H210 H81 H83 D85 H144 C163 K166 N175 H205 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P04190 27303030 304 KTVIKNETGTISISQLNKNVWVHTELGSFNGEAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 4nra A 1.85 BS01 2LW A 1 P1888 N1944 I1950 P33 N89 I95 ? Kd=65uM remove_due_to_license_issue IC50=37000nM, Kd=65000nM Q9UIF8 24304323 2006 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 4nrb A 2.08 BS01 2LX A 1 P1888 F1889 V1893 V1898 F1943 N1944 I1950 P33 F34 V38 V43 F88 N89 I95 ? ic50=38uM remove_due_to_license_issue IC50=38000nM Q9UIF8 24304323 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTF 4nrc A 1.86 BS01 2LY A 1 P1888 F1889 P33 F34 ? ic50=241uM remove_due_to_license_issue IC50=241000nM Q9UIF8 24304323 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFK 4nrk A 2.63 BS01 SIA K 1 Y95 T139 S140 G141 W158 D195 Q241 Y95 T139 S140 G141 W158 D195 Q241 ? 0019031,0019064,0046789 remove_due_to_license_issue P03460 24503069 3 DRICTGITSSNSPHVVKTATQGEVNVTGVIPLTTTPTRSHFANLKGTQTRGKLCPNCFNCTDLDVALGRPKCMGNIPSAKVSILHEVKPVTSGCYPIMHDRTKIRQLPNLLRGYENIRLSTSNVINTETAPGGPYKVGTSGSCPNVTNGNGFFNTMAWVIPKDNNKIAINPVTVEVPYICSEGEDQITVWGFHSDDKTQMERLYGDSNPQKFTSSANGVTTHYVSQIGGFPNQTEDEGLKQSGRIVVDYMVQKPGKTGTIVYQRGILLPQKVWCASGRSKVIKGSLPLIGEADCLHEKYGGLNKSKPYYTGEHAKAIGNCPIWVKTPLKLANGTKYRPPA 4nrl A 2.72 BS01 SIA G 1 Y95 T139 S140 G141 D195 Q241 Y95 T139 S140 G141 D195 Q241 ? 0019031,0019064,0046789 remove_due_to_license_issue P03460 24503069 5 DRICTGITSSNSPHVVKTATQGEVNVTGVIPLTTTPTRSHFANLKGTQTRGKLCPNCFNCTDLDVALGRPKCMGNIPSAKVSILHEVKPVTSGCYPIMHDRTKIRQLPNLLRGYENIRLSTSNVINTETAPGGPYKVGTSGSCPNVTNGNGFFNTMAWVIPKDNNKIAINPVTVEVPYICSEGEDQITVWGFHSDDKTQMERLYGDSNPQKFTSSANGVTTHYVSQIGGFPNQTEDEGLKQSGRIVVDYMVQKPGKTGTIVYQRGILLPQKVWCASGRSKVIKGSLPLIGEADCLHEKYGGLNKSKPYYTGEHAKAIGNCPIWVKTPLKLANGTKYRPPAK 4nro A 2.3 BS02 AKG A 1 N193 I201 H204 H266 I268 R277 I281 N114 I122 H125 H187 I189 R198 I202 1.14.11.53 0006397,0035515 remove_due_to_license_issue Q6P6C2 24616105 302 EQQLQKEEEARKVKSGIRQMRLFSQDECAKIEARIDEVVSRAEKGLYNEHTVDRAPLRNKYFFGEGYTYGPGQERLYPPGDVDEIPEWVHQLVIQKLVEHRVIPEGFVNSAVINDYQPGGCIVSHVDPIHIFERPIVSVSFFSDSALCFGCKFQFKPIRVSEPVLSLPVRRGSVTVLSGYAADEITHCIRPQDIKERRAVIILRKTRLDAPRL 4nrq A 2.5 BS01 PD2 A 1 N193 Y195 I201 H204 L226 H266 I268 R277 V279 I281 N111 Y113 I119 H122 L144 H184 I186 R195 V197 I199 1.14.11.53 0006397,0035515 remove_due_to_license_issue Q6P6C2 24616105 301 EQQLQKEEEARKVKSGIRQMRLFSQDECAKIEARIDEVVSRAEKGLYNEHTVDRAPLRNKYFFGEGYTGQERLYPPGDVDEIPEWVHQLVIQKLVEHRVIPEGFVNSAVINDYQPGGCIVSHVDPIHIFERPIVSVSFFSDSALCFGCKFQFKPIRVSEPVLSLPVRRGSVTVLSGYAADEITHCIRPQDIKERRAVIILRKTRLDAPRL 4nrt A 2.022 BS01 2NG A 1 W417 T418 R419 H433 R436 Q439 N505 W412 T413 R414 H428 R431 Q434 N500 3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 ic50=1000nM remove_due_to_license_issue A0ZNP5 24622391 601 GTYCGAPILGPGSAPKLSTKTKFWRSSTTPLPPGTYEPAYLGGKDPRVKGGPSLQQVMRDQLKPFTEPRGKPPKPSVLEAAKKTIINVLEQTIDPPEKWSFTQACASLDKTTSSGHPHHMRKNDCWNGESFTGKLADQASKANLMFEGGKNMTPVYTGALKDELVKTDKIYGKIKKRLLWGSDLATMIRCARAFGGLMDELKAHCVTLPIRVGMNMNEDGPIIFERHSRYKYHYDADYSRWDSTQQRAVLAAALEIMVKFSSEPHLAQVVAEDLLSPSVVDVGDFKISINEGLPSGVPCTSQWNSIAHWLLTLCALSEVTNLSPDIIQANSLFSFYGDDEIVSTDIKLDPEKLTAKLKEYGLKPTRPDKTEGPLVISEDLNGLTFLRRTVTRDPAGWFGKLEQSSILRQMYWTRGPNHEDPSETMIPHSQRPIQLMSLLGEAALHGPAFYSKISKLVIAELKEGGMDFYVPRQEPMFRWMRFSDLSTWEGDRNLAPSFVN 4nru A 2.3 BS01 2NG A 1 L391 R392 Q414 W417 T418 K419 R436 Q439 L389 R390 Q412 W415 T416 K417 R432 Q435 2.7.7.48,3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 ic50=115nM remove_due_to_license_issue Q80J95 24622391 1101 PRPSGTYAGLPIADYGDAPPLSTKTMFWRTSPEKLPPGAWEPAYLGSKDERVDGPSLQQVMRDQLKPYSEPRGLLPPQEILDAVCDAIENRLENTLEPQKPWTFKKACESLDKNTSSGYPYHKQKSKDWTGSAFIGDLGDQATHANNMYEMGKSMRPIYTAALKDELVKPDKIYGKIKKRLLWGSDLGTMIRAARAFGPFCDALKETCIFNPIRVGMSMNEDGPFIFARHANFRYHMDADYTRWDSTQQRAILKRAGDIMVRLSPEPDLARVVMDDLLAPSLLDVGDYKIVVEEGLPSGCPCTTQLNSLAHWILTLCAMVEVTRVDPDIVMQESEFSFYGDDEVVSTNLELDMVKYTMALRRYGLLPTRADKEEGPLERRQTLQGISFLRRAIVGDQFGWYGRLDRASIDRQLLWTKGPNHQNPFETLPGHRPSQLMALLGEAAMHGEKYYRTVASRVSKEAVVPRHRSVLRWVRFG 4ntj A 2.62 BS01 AZJ A 1 V102 Y105 F106 Y109 S156 N159 V190 N191 C194 R256 Y259 K280 V83 Y86 F87 Y90 S134 N137 V152 N153 C156 R313 Y316 K337 ? 0004930,0005506,0007186,0007194,0007596,0009055,0016020,0020037,0022900,0042597,0045028,0046872 remove_due_to_license_issue P0ABE7,Q9H244 24670650 1201 LCTRDYKITQVLFPLLYTVLFFVGLITNGLAMRIFFQIRSKSNFIIFLKNTVISDLLMILTFPFKILSDAKLLRTFVCQVTSVIFYFTMYISISFLGLITIDRYQKTTRPFKTKNLLGAKILSVVIWAFMFLLSLPNMILKSEFGLVWHEIVNYICQVIFWINFLIVIVCYTLITKELYRSYVRTADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLRGVGKVRKKVNVKVFIIIAVFFICFVPFHFARIPYTLSQTRDVFDCTAENTLFYVKESTLWLTSLNACLNPFIYFFLCKSFRNSLISM 4nuc A 1.4 BS01 435 A 1 W81 P82 V87 Y139 N140 I146 W40 P41 V46 Y98 N99 I105 ? Ki=0.91uM remove_due_to_license_issue Ki=4300nM O60885 24144283 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 4nud A 1.2 BS01 NUD A 1 W81 L92 N140 I146 W38 L49 N97 I103 ? Ki<0.0845uM remove_due_to_license_issue Ki=340nM O60885 24144283 201 NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4nue A 1.3 BS01 NUE A 1 W81 P82 V87 L92 N140 W40 P41 V46 L51 N99 ? Ki=0.15uM remove_due_to_license_issue Ki=440nM O60885 24144283 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 4nus A 2.39 BS01 2NK A 1 F79 V82 A98 K100 L150 L200 T210 D211 F212 F27 V30 A46 K48 L98 L148 T158 D159 F160 D193 K195 E197 N198 D211 T231 D141 K143 E145 N146 D159 T179 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.005uM remove_due_to_license_issue IC50=5.0nM P51812 24554780 1001 THHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRTKMERDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKESIDHEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKPATFYFDP 4nvp A 2.5 BS01 7CH A 1 F658 G659 E660 I661 C662 R669 T670 A671 R710 F141 G142 E143 I144 C145 R152 T153 A154 R193 ? Kd=27nM remove_due_to_license_issue Q9Y3Q4 24605759 800 SPMDSSRRQYQEKYKQVEQYMSFHKLPPDTRQRIHDYYEHRYQGKMFDEESILGELSEPLREEIINFNCRKLVASMPLFANADPNFVTSMLTKLRFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKETKLADGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVALDRLDRIGKKN 4nvq A 2.03 BS01 2OD A 1 Y1067 A1077 D1078 D1083 L1086 F1087 D1088 F1152 Y1154 R1157 F1158 I1161 Y152 A162 D163 D168 L171 F172 D173 F233 Y235 R238 F239 I242 Y1067 Y1154 Y152 Y235 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 ic50=3.3nM remove_due_to_license_issue IC50=3.3nM Q96KQ7 24900801 1201 IRTEKIICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLGEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKSYFTCQCGSEKCKHSAEAIALEQS 4nw5 A 1.94 BS01 2NR A 1 G75 Q76 V82 A98 F149 L150 G153 L200 T210 G25 Q26 V32 A48 F99 L100 G103 L150 T160 D193 K195 E197 N198 D211 T231 D143 K145 E147 N148 D161 T181 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.02uM remove_due_to_license_issue IC50=20nM P51812 24534486 1001 AITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRTKMERDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKESIDHEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKPTFYFDP 4nw6 A 1.74 BS01 2NS A 1 L74 Q76 V82 A98 F149 L150 G153 L200 T210 L24 Q26 V32 A48 F99 L100 G103 L150 T160 D193 K195 E197 N198 D211 T231 D143 K145 E147 N148 D161 T181 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.004uM remove_due_to_license_issue P51812 24534486 1001 AITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRTKMERDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKESIDHEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKPTFYFDP 4nw7 A 2.15 BS02 2O5 A 1 M519 N567 I582 F586 M603 Q615 F618 F678 M198 N246 I261 F265 M282 Q294 F297 F342 3.1.4.53 0004114,0007165,0008081 ic50=237nM remove_due_to_license_issue IC50=237nM Q07343 24998378 704 HMSISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPQLMEKFQF 4nwc A 2.012 BS01 2QE A 1 E443 Y491 P518 L519 T520 R525 G690 A691 T692 N722 E739 Y765 E12 Y60 P87 L88 T89 R94 G139 A140 T141 N171 E188 Y214 ? 0015276,0016020 Ki=1.74uM remove_due_to_license_issue Ki=1010nM P42264 25044437 905 TNRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 4nwd A 2.6 BS01 2QD A 1 E15 Y63 P90 L91 T92 R97 G142 A143 T144 N174 E191 Y217 E11 Y59 P86 L87 T88 R93 G138 A139 T140 N170 E187 Y213 ? 0015276,0016020 remove_due_to_license_issue Ki=57.3nM P42264 25044437 301 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 4nwk A 1.62 BS01 2R8 A 1 Q41 H57 D81 I132 L135 K136 G137 S139 F154 R155 A156 A157 Q52 H68 D92 I143 L146 K147 G148 S150 F165 R166 A167 A168 H57 D81 G137 S139 H68 D92 G148 S150 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue A8DG50 24555570 301 GSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLET 4nwm A 2.03 BS01 2P5 A 1 L408 T410 Q412 F413 V416 A428 K430 Y476 M477 A478 N479 G480 L528 D539 L542 Y551 L14 T16 Q18 F19 V22 A34 K36 Y82 M83 A84 N85 G86 L133 D144 L147 Y156 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.008uM remove_due_to_license_issue Q06187 24685542 701 MEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLRERHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDE 4nxo A 2.73 BS02 2H7 A 1 H108 Q111 H112 F115 S128 N139 E189 R824 Y831 V833 H66 Q69 H70 F73 S86 N97 E147 R782 Y789 V791 Q111 Q69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue IC50=56nM P14735 26394692 1102 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNPVLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4nxs A 2.5493 BS01 2OZ A 1 W47 D92 Y134 C142 K168 D170 E203 L206 Y207 R227 D231 W16 D61 Y103 C111 K137 D139 E172 L175 Y176 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue IC50=3.4e+2nM P06280 24783948 508 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTM 4nxs B 2.5493 BS01 2OZ B 1 W47 D92 C142 K168 D170 E203 L206 Y207 D231 W16 D61 C111 K137 D139 E172 L175 Y176 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue IC50=3.4e+2nM P06280 24783948 507 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTMQ 4nxu A 2.3 BS01 ADP A 1 S187 S189 H201 Q203 V324 K326 S340 R342 K368 S56 S58 H70 Q72 V189 K191 S205 R207 K233 ? 0005741,0007005 Kd=2.9uM remove_due_to_license_issue Q9NQG6 24515348 501 RMSLQEKLLTYYRNRAAIPAGEQARAKQAAVDICAELRSFLRAKLPDMPLRDMYLSGSLYDDLQVVTADHIQLIVPLVLEQNLWSCIPGEDTIMNVPGFFLVRRENPEYFPRGSSYWDRCVVGGYLSPKTVADTFEKVVAGSINWPAIGSLLDYVIRPAALTLEVQYERDKHLFIDFLPSVTLGDTVLVAKPHRLAQYDNLWRLSLRPAETARLRALDQADSGCRSLCLKILKAICKSTPALGHLTASQLTNVILHLAQEEADWSPDMLADRFLQALRGLISYLEAGVLPSALNPKVNLFAELTPEEIDELGYTLYCSLSEPEVLLQ 4nxv A 2.3 BS01 GDP A 1 S189 H201 Q203 K326 S340 R342 K368 A382 S58 H70 Q72 K194 S208 R210 K236 A250 ? 0005741,0007005 Kd=3.8uM remove_due_to_license_issue Q9NQG6 24515348 501 RMSLQEKLLTYYRNRAAIPAGEQARAKQAAVDICAELRSFLRAKLPDMPLRDMYLSGSLYDDLQVVTADHIQLIVPLVLEQNLWSCIPGEDTIMNVPGFFLVRRENPEYFPRGSSYWDRCVVGGYLSPKTVADTFEKVVAGSINWPAIGSLLDYVIRPAPPEALTLEVQYERDKHLFIDFLPSVTLGDTVLVAKPHRLAQYDNLWRLSLRPAETARLRALDQADSGCRSLCLKILKAICKSTPALGHLTASQLTNVILHLAQEEADWSPDMLADRFLQALRGLISYLEAGVLPSALNPKVNLFAELTPEEIDELGYTLYCSLSEPEVLLQ 4nyf A 1.9 BS01 4BI A 1 A169 E170 H171 T174 A108 E109 H110 T113 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 Kd=49nM remove_due_to_license_issue P0C6F2 24900852 301 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTIHTDNGSNFTSATVKAACDWAGIKQEPQSQGVVESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGIGGYSAGERIVDIIATDIQT 4nyf B 1.9 BS01 4BI A 1 Q95 L102 T125 A128 A129 W132 Q40 L47 T70 A73 A74 W77 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P0C6F2 24900852 301 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTIHTDNGSNFTSATVKAACDWAGIKQEDGIPYNPESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRYSAGERIVDIIATD 4nyi S 2.9612 BS01 2PX S 1 M878 Y884 F890 K898 L901 M304 Y310 F316 K324 L327 ? 0005085,0007264 remove_due_to_license_issue EC50=25100nM Q07889 24550516 1101 QMRLPSADVYRFAEPDSEENIIFEENMAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAHNITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 4nyj S 2.8522 BS01 2PZ S 1 M878 N879 Y884 F890 M300 N301 Y306 F312 ? 0005085,0007264 remove_due_to_license_issue EC50=>100000nM Q07889 24550516 1101 QMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 4nym S 3.5529 BS01 RND S 1 M878 Y884 F890 K898 E902 H905 M301 Y307 F313 K321 E325 H328 ? 0005085,0007264 remove_due_to_license_issue Q07889 24550516 1101 QMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAHNITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 4nyt A 2.25 BS01 PC A 1 R132 D133 T136 K221 R57 D58 T61 K146 ? Kd=3.7mM remove_due_to_license_issue Q15485 25344472 303 GPRTCKDLLDRGHFLSGWHTIYLPDCRPLTVLCDMDTDGGGWTVFQRRVDGSVDFYRDWATYKQGFGSRLGEFWLGNDNIHALTAQGTSELRTDLVDFEDNYQFAKYRSFKVADEAEKYNLVLGAFVEGSAGDSLTFHNNQSFSTKDQDNDLNTGNCAVMFQGAWWYKNCHTSNLNGRYLRGTHGSFANGINWKSGKGYNYSYKVSEMKVRP 4nzb I 2.68 BS01 NSE I 1 Y89 W143 Y185 Y192 Y89 W143 Y179 Y183 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 24982426 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTSEYFSQYSRFEILDVTQKKNSVTYPEAYEDVEVSLNFRKK 4nzb J 2.68 BS01 NSE I 1 W53 L112 W53 L112 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 24982426 301 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 4nzm A 2.0 BS02 0EJ A 1 K54 R213 K214 K248 R262 K329 K13 R172 K173 K207 R221 K288 2.7.4.24 0000829 remove_due_to_license_issue O43314 24768307 402 RQIVVGICSMAKKSKSKPMKEILERISLFKYITVVVFEEEVILNEPVENWPLCDCLISFHSKGFPLDKAVAYAKLRNPFVINDLNMQYLIQDRREVYSILQAEGILLPRYAILNRDPNNPKECNLIEGEDHVEVNGEVFQKPFVEKPVSAEDHNVYIYYPTSAGGGSQRLFRKIGSRSSVYSPESNVRKTGSYIYEEFMPTDGTDVKVYTVGPDYAHAEARKSPALDGKVERDSEGKEVRYPVILNAREKLIAWKVCLAFKQTVCGFDLLRANGQSYVCDVNGFSFVKNSMKYYDDCAKILGNIVMRELAPQFHIPWSIPLEAED 4nzn A 1.75 BS02 2OU A 1 K53 K54 K103 E192 H194 R213 K12 K13 K62 E151 H153 R172 2.7.4.24 0000829 remove_due_to_license_issue O43314 24768307 402 RQIVVGICSMAKKSKSKPMKEILERISLFKYITVVVFEEEVILNEPVENWPLCDCLISFHSKGFPLDKAVAYAKLRNPFVINDLNMQYLIQDRREVYSILQAEGILLPRYAILNRDPNNPKECNLIEGEDHVEVNGEVFQKPFVEKPVSAEDHNVYIYYPTSAGGGSQRLFRKIGSRSSVYSPESNVRKTGSYIYEEFMPTDGTDVKVYTVGPDYAHAEARKSPALDGKVERDSEGKEVRYPVILNAREKLIAWKVCLAFKQTVCGFDLLRANGQSYVCDVNGFSFVKNSMKYYDDCAKILGNIVMRELAPQFHIPWSIPLEAED 4nzo A 1.9 BS02 2OV A 1 K53 K54 H101 S102 K103 E192 R213 K12 K13 H60 S61 K62 E151 R172 2.7.4.24 0000829 remove_due_to_license_issue O43314 24768307 402 RQIVVGICSMAKKSKSKPMKEILERISLFKYITVVVFEEEVILNEPVENWPLCDCLISFHSKGFPLDKAVAYAKLRNPFVINDLNMQYLIQDRREVYSILQAEGILLPRYAILNRDPNNPKECNLIEGEDHVEVNGEVFQKPFVEKPVSAEDHNVYIYYPTSAGGGSQRLFRKIGSRSSVYSPESNVRKTGSYIYEEFMPTDGTDVKVYTVGPDYAHAEARKSPALDGKVERDSEGKEVRYPVILNAREKLIAWKVCLAFKQTVCGFDLLRANGQSYVCDVNGFSFVKNSMKYYDDCAKILGNIVMRELAPQFHIPWSIPLEAED 4o04 A 1.82 BS01 2Q8 A 1 N51 M98 G135 F138 Y139 W162 N36 M83 G120 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.69uM remove_due_to_license_issue Ki=690nM P07900 24673104 4000 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4o05 A 1.79 BS01 2Q9 A 1 N51 D93 M98 G135 F138 Y139 W162 T184 N36 D78 M83 G120 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.037uM remove_due_to_license_issue Ki=37nM P07900 24673104 4000 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4o07 A 1.86 BS01 FGH A 1 N51 A55 D93 M98 L107 G135 F138 Y139 W162 T184 N36 A40 D78 M83 L92 G120 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.042uM remove_due_to_license_issue Ki=42nM P07900 24673104 4000 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4o09 A 1.96 BS01 2R6 A 1 N51 A55 D93 M98 F138 Y139 W162 T184 N36 A40 D78 M83 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.02uM remove_due_to_license_issue Ki=20nM P07900 24673104 4000 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4o0a A 1.2 BS01 2P9 A 1 R31 I33 T34 R41 R43 S55 M57 A59 T60 N85 V93 I95 R34 I36 T37 R44 R46 S58 M60 A62 T63 N88 V96 I98 ? 0003677,0005634,0006260 remove_due_to_license_issue Kd=190nM P27694 24147804 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4o0b A 1.93 BS01 2QA A 1 N51 D93 M98 F138 Y139 W162 T184 N36 D78 M83 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=0.005uM remove_due_to_license_issue Ki=5.0nM P07900 24673104 4000 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4o0j A 2.05 BS01 LF8 A 1 L102 T124 T125 A128 A129 W132 L47 T69 T70 A73 A74 W77 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=13uM remove_due_to_license_issue P12497 24874515 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGGYSAGERIVDIIATDIQ 4o0t A 2.6 BS01 2OL A 1 V284 A297 K299 E315 M319 M344 Y346 L347 L396 T406 D407 F408 V34 A47 K49 E65 M69 M94 Y96 L97 L146 T156 D157 F158 N389 K391 D393 N394 D407 T427 N139 K141 D143 N144 D157 T177 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=5420nM, Ki=2900nM Q13153 24432870 601 EEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 4o0v A 2.8 BS01 2OL A 1 I327 V335 K350 E366 V379 M395 L398 G401 L447 S457 D458 F459 I29 V37 K52 E68 V81 M97 L100 G103 L149 S159 D160 F161 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=4.8nM, Ki=3.3nM O96013 24432870 601 GSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 4o0x A 2.483 BS01 2OQ A 1 V335 E366 V379 M395 L398 L447 S457 D458 F459 V37 E68 V81 M97 L100 L149 S159 D160 F161 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 Ki=0.068uM remove_due_to_license_issue Ki=68nM O96013 24432870 601 GSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 4o0y A 2.2 BS01 2OO A 1 I327 V335 A348 E366 M395 E396 F397 L398 L447 S457 D458 I29 V37 A50 E68 M97 E98 F99 L100 L149 S159 D160 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 Ki=0.06uM remove_due_to_license_issue IC50=66nM, Ki=60nM O96013 24432870 601 GSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 4o0z A 2.049 BS01 2RM A 1 H191 F193 R196 D219 V242 A244 I309 R311 I351 H175 F177 R180 D203 V226 A228 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.057uM remove_due_to_license_issue IC50=57nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o0z B 2.049 BS01 2RM B 1 Y188 H191 F193 R196 D219 V242 A244 S275 R311 I351 Y171 H174 F176 R179 D202 V225 A227 S258 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.057uM remove_due_to_license_issue IC50=57nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4o10 A 1.55 BS01 2QF A 1 Y188 H191 F193 R196 D219 V242 A244 R311 I351 Y172 H175 F177 R180 D203 V226 A228 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.078uM remove_due_to_license_issue IC50=78nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o10 A 1.55 BS02 2QF B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.078uM remove_due_to_license_issue IC50=78nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o10 B 1.55 BS01 2QF B 1 H191 F193 R196 D219 V242 A244 R311 I351 H174 F176 R179 D202 V225 A227 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.078uM remove_due_to_license_issue IC50=78nM P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4o12 A 2.498 BS01 2QG A 1 Y188 H191 F193 R196 D219 V242 S275 R311 Y172 H175 F177 R180 D203 V226 S259 R295 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.002uM remove_due_to_license_issue P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4o12 B 2.498 BS01 2QG A 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.002uM remove_due_to_license_issue P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4o12 B 2.498 BS02 2QG B 1 H191 F193 R196 D219 V242 A244 S275 I309 R311 R349 I351 I378 A379 H174 F176 R179 D202 V225 A227 S258 I292 R294 R332 I334 I361 A362 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.002uM remove_due_to_license_issue P43490 24797455 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELEA 4o13 A 1.75 BS01 2P1 A 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 S275 I309 R311 I351 Y172 H175 F177 R180 D203 Y224 S225 V226 A228 S259 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM remove_due_to_license_issue P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o13 B 1.75 BS01 2P1 B 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 I309 R311 I351 Y171 H174 F176 R179 D202 Y223 S224 V225 A227 I292 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.015uM remove_due_to_license_issue P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4o15 A 1.8 BS01 2P1 A 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 I309 R311 I351 Y172 H175 F177 R180 D203 Y224 S225 V226 A228 I293 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.095uM remove_due_to_license_issue P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o15 B 1.8 BS01 2P1 A 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.095uM remove_due_to_license_issue P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o15 B 1.8 BS02 2P1 B 1 Y188 H191 F193 R196 D219 Y240 S241 V242 A244 R311 I351 Y171 H174 F176 R179 D202 Y223 S224 V225 A227 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.095uM remove_due_to_license_issue P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o1b A 1.65 BS01 DGB A 1 G185 K189 H191 F193 R196 D219 V242 A244 S275 I309 R311 I378 A379 G169 K173 H175 F177 R180 D203 V226 A228 S259 I293 R295 I362 A363 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.385uM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKRTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o1b A 1.65 BS04 DGB B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.385uM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKRTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o1b B 1.65 BS01 DGB B 1 G185 K189 H191 F193 R196 D219 A244 S275 I309 R311 I378 A379 G168 K172 H174 F176 R179 D202 A227 S258 I292 R294 I361 A362 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.385uM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKRTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4o1d A 1.705 BS01 DGB A 1 F193 V242 A244 P273 S275 Q305 I309 R311 F177 V226 A228 P257 S259 Q289 I293 R295 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.024uM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLRDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o1d B 1.705 BS01 DGB B 1 F193 R196 V242 A244 P273 S275 Q305 P307 R311 F176 R179 V225 A227 P256 S258 Q288 P290 R294 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.024uM remove_due_to_license_issue IC50=3.0nM, Ki=0.30nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLRDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIEL 4o1l A 2.5 BS01 HO4 A 1 N14 L16 D18 G64 S65 N68 C123 A136 F170 N296 G297 D300 N11 L13 D15 G61 S62 N65 C120 A133 F167 N291 G292 D295 R132 G297 A298 G299 D300 R129 G292 A293 G294 D295 2.7.1.20 0003723,0004001,0004136,0005524,0005634,0005654,0005737,0005829,0005886,0006144,0006166,0006175,0006753,0009156,0016301,0032263,0034654,0044209,0046872,0106383 ic50=0.2uM remove_due_to_license_issue IC50=200nM P55263 25259627 403 LRENILFGMGNPLLDISAVVDKDFLDKYSLKPNDQILAEDKHKELFDELVKKFKVEYHAGGSTQNSIKVAQWMIQQPHKAATFFGCIGIDKFGEILKRKAAEAHVDAHYYEQNEQPTGTCAACITGDNRSLIANLAAANCYKKEKHLDLEKNWMLVEKARVCYIAGFFLTVSPESVLKVAHHASENNRIFTLNLSAPFISQFYKESLMKVMPYVDILFGNETEAATFAREQGFETKDIKEIAKKTQALPKMNSKRQRIVIFTQGRDDTIMATESEVTAFAVLDQDQKIDTNGAGDAFVGGFLSQLVSDKPLTECIRAGHYAASIII 4o1l A 2.5 BS02 HO4 A 2 G267 V284 D286 A298 G299 A327 I331 G264 V281 D283 A293 G294 A322 I326 R132 G297 A298 G299 D300 R129 G292 A293 G294 D295 2.7.1.20 0003723,0004001,0004136,0005524,0005634,0005654,0005737,0005829,0005886,0006144,0006166,0006175,0006753,0009156,0016301,0032263,0034654,0044209,0046872,0106383 ic50=0.2uM remove_due_to_license_issue IC50=200nM P55263 25259627 404 LRENILFGMGNPLLDISAVVDKDFLDKYSLKPNDQILAEDKHKELFDELVKKFKVEYHAGGSTQNSIKVAQWMIQQPHKAATFFGCIGIDKFGEILKRKAAEAHVDAHYYEQNEQPTGTCAACITGDNRSLIANLAAANCYKKEKHLDLEKNWMLVEKARVCYIAGFFLTVSPESVLKVAHHASENNRIFTLNLSAPFISQFYKESLMKVMPYVDILFGNETEAATFAREQGFETKDIKEIAKKTQALPKMNSKRQRIVIFTQGRDDTIMATESEVTAFAVLDQDQKIDTNGAGDAFVGGFLSQLVSDKPLTECIRAGHYAASIII 4o24 A 2.3 BS01 2Q0 A 1 N64 P66 W96 L99 F115 N71 P73 W103 L106 F122 3.1.-.- 0004519,0006259,0008408,0016787 remove_due_to_license_issue Q9X1X0 24316220 401 IHHHHHHVINLKELKILHTSDWHLGVTSWTSSRPVDRREELKKALDKVVEEAEKREVDLILLTGDLLHSRNNPSVVALHDLLDYLKRMMRTAPVVVLPGNHDWKGLKLFGNFVTSISSDITFVMSFEPVDVEAKRGQKVRILPFPYPDESEALRKNEGDFRFFLESRLNKLYEEALKKEDFAIFMGHFTVEGLAGYAGIEQGREIIINRALIPSVVDYAALGHIHSFREIQKQPLTIYPGSLIRIDFGEEADEKGAVFVELKRGEPPRYERIDASPLPLKTLYYKKIDTSALKSIRDFCRNFPGYVRVVYEEDSGILPDLMGEIDNLVKIE 4o24 B 2.3 BS01 2Q0 B 1 R63 N64 P66 L74 H94 L99 F115 R60 N61 P63 L71 H91 L96 F112 3.1.-.- 0004519,0006259,0008408,0016787 remove_due_to_license_issue Q9X1X0 24316220 401 LKELKILHTSDWHLGVTSWTSSRPVDRREELKKALDKVVEEAEKREVDLILLTGDLLHSRNNPSVVALHDLLDYLKRMMRTAPVVVLPGNHDWKGLKLFGNFVTSISSDITFVMSFEPVDVEAKRGQKVRILPFPYPDESEALRKNEGDFRFFLESRLNKLYEEALKKEDFAIFMGHFTVEGLAGYAGIEQGREIIINRALIPSVVDYAALGHIHSFREIQKQPLTIYPGSLIRIDFGEEADEKGAVFVELKRGEPPRYERIDASPLPLKTLYYKKIDTSALKSIRDFCRNFPGYVRVVYEEDSGILPDLMGEIDNLVKIE 4o26 A 3.001 BS01 rna E 0 K370 L371 P372 L373 R374 F376 I479 K480 V481 M482 L489 R490 R495 F496 P497 P498 S499 L501 Y503 R506 K47 L48 P49 L50 R51 F53 I151 K152 V153 M154 L161 R162 R167 F168 P169 P170 S171 L173 Y175 R178 2.7.7.49 0000723,0003677,0003720,0003964 remove_due_to_license_issue Q1PS67 24793650 170 ~ 220 GSGFLYGGRGMHGFCLNRKRRTAAGPRRLQGQDLVRLVFFEGLKPKKLPLRYFNMVPVFGRLLQRHRKCRYSSVLHRMCPVVELSRAAQGELSSLIPQHCAPHRVYLFVRECLTAVVPEELWGSDHNRLQFFSRVRGFLKSGSVAELMWKIKVMDCDWLKLRRTAGRFPPSELAYRTRILSQFLTWLLDGFVVGLVRACFYATESNAIRFYRQEVWSKLQDLAFRRHIAKGEMEELSPAQ 4o26 B 3.001 BS01 rna F 0 K370 L371 P372 L373 R374 F376 K478 I479 K480 V481 M482 L489 P497 P498 S499 Y503 R506 K42 L43 P44 L45 R46 F48 K149 I150 K151 V152 M153 L160 P161 P162 S163 Y167 R170 2.7.7.49 0000723,0003677,0003720,0003964 remove_due_to_license_issue Q1PS67 24793650 170 ~ 220 SGFLYGGRGMHGFCLNRKRRTAAGPRRLQGQDLVRLVFFEKKLPLRYFNMVPVFGRLLQRHRKCRYSSVLHRMCPVVELSRAAQGELSSLIPQHCAPHRVYLFVRECLTAVVPEELWGSDHNRLQFFSRVRGFLKSGKFERISVELMWKIKVMDCDWLKLPPSELAYRTRILSQFLTWLLDGFVVGLVRACFYATESVGQKNAIRFYRQEVWSKLQDLAFRRHIAKGE 4o28 A 2.0 BS01 1QS A 1 H191 F193 R196 D219 V242 A244 R311 I351 H173 F175 R178 D201 V224 A226 R293 I333 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.029uM remove_due_to_license_issue IC50=5.0nM, EC50=1.1nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o28 A 2.0 BS04 1QS B 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.029uM remove_due_to_license_issue IC50=5.0nM, EC50=1.1nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o28 B 2.0 BS01 1QS A 1 D16 Y18 D9 Y11 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.029uM remove_due_to_license_issue IC50=5.0nM, EC50=1.1nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o28 B 2.0 BS02 1QS B 1 H191 F193 R196 D219 V242 A244 P273 R311 I351 H174 F176 R179 D202 V225 A227 P256 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.029uM remove_due_to_license_issue IC50=5.0nM, EC50=1.1nM P43490 25285661 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNFREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 4o2a B 2.5 BS02 2RR B 1 L248 L255 N258 M259 V315 A316 I318 N350 K352 I378 L246 L253 N256 M257 V303 A304 I306 N338 K340 I358 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 Kd=1.8uM remove_due_to_license_issue Q6B856 24530796 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLLTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 4o2b A 2.3 BS03 LOC B 1 S178 A180 V181 S178 A180 V181 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 24530796 503 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVDS 4o2b B 2.3 BS02 LOC B 1 L248 A250 K254 L255 N258 M259 I318 K352 L246 A248 K252 L253 N256 M257 I310 K344 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 Ki=1.8uM remove_due_to_license_issue IC50=800nM, Ki=780nM Q6B856 24530796 503 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 4o2p A 2.1 BS01 11V A 1 L273 V281 A293 K295 I336 T338 Y340 M341 G344 L393 D404 L17 V25 A37 K39 I78 T80 Y82 M83 G86 L135 D146 D386 R388 A390 N391 D404 F424 D128 R130 A132 N133 D146 F156 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.2uM remove_due_to_license_issue P00523 25469771 601 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEDFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4o3a A 1.8 BS01 ASP A 1 Y61 T91 R96 G141 S142 T143 E193 Y61 T91 R96 G141 S142 T143 E193 ? 0015276,0016020 Ki=2.57mM remove_due_to_license_issue P19491 24673938 302 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4o3b B 1.906 BS01 GLU B 1 Y61 T91 R96 G141 S142 T143 E193 Y58 T88 R93 G138 S139 T140 E190 ? 0015276,0016020 Ki=0.82uM remove_due_to_license_issue P19491 24673938 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4o3c A 1.5 BS01 ASP A 1 Y61 T91 R96 G141 S142 T143 E193 Y61 T91 R96 G141 S142 T143 E193 ? 0015276,0016020 Ki=2.57mM remove_due_to_license_issue P19491 24673938 301 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 4o3f A 2.106 BS01 TZN A 1 G238 G239 T255 L257 F292 M312 G313 L314 P339 G341 V342 G238 G239 T255 L257 F292 M312 G313 L314 P339 G341 V342 R39 K216 G374 G397 R39 K216 G374 G389 2.7.2.3 0004618,0005515,0005524,0005615,0005737,0005759,0005829,0006094,0006096,0016301,0016525,0030855,0031639,0045121,0046166,0047134,0061621,0071456 Kd=2.78uM remove_due_to_license_issue P09411 25383758 501 MSLSNKLTLDKLDVKGKRVVMRVDFNVPMKNNQITNNQRIKAAVPSIKFCLDNGAKSVVLMSHLGRPDGVPMPDKYSLEPVAAELKSLLGKDVLFLKDCVGPEVENACANPAAGTVILLENLRFHVEEEGKGKDASGNKVKAEPAKIDAFRASLSKLGDVYVNDAFGTAHRAHSSMVGVNLPQKAGGFLMKKELNYFAKALESPERPFLAILGGAKVADKIQLINNMLDKVNEMIIGGGMAFTFLKVLNNMEIGTSLYDEEGAKIVKDLMSKAEKNGVKITLPVDFVTADKFDENAKTGQATVASGIPAGWMGLDCGTESSKKYAEAVGRAKQIVWNGPVGVFEWEAFARGTKSLMDEVVKATSRGCITIIGGGDTATDKVSHVSTGGGASLELLEGKVLPGVDALSNV 4o3m A 2.3 BS01 dna P 0 K870 P871 K872 T1110 N1112 M1113 A1163 N1164 K222 P223 K224 T444 N446 M447 A497 N498 5.6.2.4 0000166,0003676,0004386,0005524,0006260,0006281,0006310,0043138,0044237 remove_due_to_license_issue P54132 24816114 2 ~ 13 KHERFQSLSFPHTKEMMKIFHKKFGLHNFRTNQLEAINAALLGEDCFILMPTGGGKSLCYQLPACVSPGVTVVISPLRSLIVDQVQKLTSLDIPATYLTGDKTDSEATNIYLQLSKKDPIIKLLYVTPEKICASNRLISTLENLYERKLLARFVIDEAHRQDYKRMNMLRQKFPSVPVMALTATANPRVQKDILTQLKILRPQVFSMSFNRHNLKYYVLPKKPKKVAFDCLEWIRKHHPYDSGIIYCLSRRECDTMADTLQRDGLAALAYHAGLSDSARDEVQQKWINQDGCQVICATIAFGMGIDKPDVRFVIHASLPKSVEGYYQESGRAGRDGEISHCLLFYTYHDVTRLKRLIMMEKDHTRETHFNNLYSMVHYCENITECRRIQLLAYFGENGFNPDFCKKHPDVSCDNCCKYKTRDVTDDVKSIVRFVQEHSPSGRFTMNMLVDIFLGSKSAKIQSGIFGKGSAYSRHNAERLFKKLILDKILDEDLYINANDQAIAYVMLGNKAQTVLNGNLKVDFMETENKVSQREEMVKKCLGELTEVCKSLGKVFGVHYFNIFNTVTLKKLAESLSSDPEVLLQIDGVTEDKLEKYGAEVISVLQKYSEWTSP 4o3m A 2.3 BS02 dna T 0 L896 S897 R898 A920 T946 I947 A948 R1000 R1003 L1004 M1007 E1008 S1121 K1122 N1164 D1165 Q1166 L248 S249 R250 A272 T298 I299 A300 R352 R355 L356 M359 E360 S455 K456 N498 D499 Q500 5.6.2.4 0000166,0003676,0004386,0005524,0006260,0006281,0006310,0043138,0044237 remove_due_to_license_issue P54132 24816114 4 ~ 19 KHERFQSLSFPHTKEMMKIFHKKFGLHNFRTNQLEAINAALLGEDCFILMPTGGGKSLCYQLPACVSPGVTVVISPLRSLIVDQVQKLTSLDIPATYLTGDKTDSEATNIYLQLSKKDPIIKLLYVTPEKICASNRLISTLENLYERKLLARFVIDEAHRQDYKRMNMLRQKFPSVPVMALTATANPRVQKDILTQLKILRPQVFSMSFNRHNLKYYVLPKKPKKVAFDCLEWIRKHHPYDSGIIYCLSRRECDTMADTLQRDGLAALAYHAGLSDSARDEVQQKWINQDGCQVICATIAFGMGIDKPDVRFVIHASLPKSVEGYYQESGRAGRDGEISHCLLFYTYHDVTRLKRLIMMEKDHTRETHFNNLYSMVHYCENITECRRIQLLAYFGENGFNPDFCKKHPDVSCDNCCKYKTRDVTDDVKSIVRFVQEHSPSGRFTMNMLVDIFLGSKSAKIQSGIFGKGSAYSRHNAERLFKKLILDKILDEDLYINANDQAIAYVMLGNKAQTVLNGNLKVDFMETENKVSQREEMVKKCLGELTEVCKSLGKVFGVHYFNIFNTVTLKKLAESLSSDPEVLLQIDGVTEDKLEKYGAEVISVLQKYSEWTSP 4o43 A 2.4 BS03 2PW A 1 L60 P66 L74 W96 L99 F115 L67 P73 L81 W103 L106 F122 3.1.-.- 0004519,0006259,0008408,0016787 remove_due_to_license_issue Q9X1X0 24316220 403 IHHHHHHVINLKELKILHTSDWHLGVTSWTSSRPVDRREELKKALDKVVEEAEKREVDLILLTGDLLHSRNNPSVVALHDLLDYLKRMMRTAPVVVLPGNHDWKGLKLFGNFVTSISSDITFVMSFEPVDVEAKRGQKVRILPFPYPDESEALRKNEGDFRFFLESRLNKLYEEALKKEDFAIFMGHFTVEGLAGYAGIEQGREIIINRALIPSVVDYAALGHIHSFREIQKQPLTIYPGSLIRIDFGEEADEKGAVFVELKRGEPPRYERIDASPLPLKTLYYKKIDTSALKSIRDFCRNFPGYVRVVYEEDSGILPDLMGEIDNLVKIE 4o44 A 2.889 BS01 2RS A 1 L100 K101 K103 V106 V179 Y181 Y188 F227 W229 L234 H235 P236 L100 K101 K103 V106 V179 Y181 Y188 F227 W229 L234 H235 P236 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 24726448 601 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 4o4g A 2.712 BS01 2RT A 1 L100 K101 K103 V106 Y181 Y188 F227 L234 H235 P236 Y318 L102 K103 K105 V108 Y183 Y190 F229 L236 H237 P238 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 24726448 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 4o4k A 2.1 BS03 2PK A 1 D58 L59 R63 N93 L99 D65 L66 R70 N100 L106 3.1.-.- 0004519,0006259,0008408,0016787 remove_due_to_license_issue Q9X1X0 24316220 403 IHHHHHHVINLKELKILHTSDWHLGVTSWTSSRPVDRREELKKALDKVVEEAEKREVDLILLTGDLLHSRNNPSVVALHDLLDYLKRMMRTAPVVVLPGNHDWKGLKLFGNFVTSISSDITFVMSFEPVDVEAKRGQKVRILPFPYPDESEALRKNEGDFRFFLESRLNKLYEEALKKEDFAIFMGHFTVEGLAGYAGIEQGREIIINRALIPSVVDYAALGHIHSFREIQKQPLTIYPGSLIRIDFGEEADEKGAVFVELKRGEPPRYERIDASPLPLKTLYYKKIDTSALKSIRDFCRNFPGYVRVVYEEDSGILPDLMGEIDNLVKIE 4o4r A 2.4 BS01 20V A 1 M219 L391 R392 R393 Q414 K419 M216 L384 R385 R386 Q407 K412 2.7.7.48,3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 ic50=0.88uM remove_due_to_license_issue Q80J95 24657439 601 RPSGTYAGLPIADYGDAPPLSTKTMFWRTSPEKLPPGAWEPAYLGSKDERVDGPSLQQVMRDQLKPYSEPRGLLPPQEILDAVCDAIENRLENTLEPQKPWTFKKACESLDKNTSSGYPYHKQKSKDWTGSAFIGDLGDQATHANNMYEMGKSMRPIYTAALKDELVKPDKIYGKIKKRLLWGSDLGTMIRAARAFGPFCDALKETCIFNPIRVGMSMNEDGPFIFARHANFRYHMDADYTRWDSTQQRAILKRAGDIMVRLSPEPDLARVVMDDLLAPSLLDVGDYKIVVEEGLPSGCPCTTQLNSLAHWILTLCAMVEVTRVDPDIVMQESEFSFYGDDEVVSTNLELDMVKYTMALRRYGLLPTRADPLERRQTLQGISFLRRAIVGDQFGWYGRLDRASIDRQLLWTKGPNHQNPFETLPGHAQRPSQLMALLGEAAMHGEKYYRTVASRVSKEAAQVVPRHRSVLRWVRFG 4o4r A 2.4 BS02 20V A 2 F29 L169 Y341 R392 S410 R413 Q414 F26 L166 Y338 R385 S403 R406 Q407 2.7.7.48,3.4.22.66,3.6.1.15 0003723,0003968,0004386,0005524,0006351,0039694 ic50=0.88uM remove_due_to_license_issue Q80J95 24657439 602 RPSGTYAGLPIADYGDAPPLSTKTMFWRTSPEKLPPGAWEPAYLGSKDERVDGPSLQQVMRDQLKPYSEPRGLLPPQEILDAVCDAIENRLENTLEPQKPWTFKKACESLDKNTSSGYPYHKQKSKDWTGSAFIGDLGDQATHANNMYEMGKSMRPIYTAALKDELVKPDKIYGKIKKRLLWGSDLGTMIRAARAFGPFCDALKETCIFNPIRVGMSMNEDGPFIFARHANFRYHMDADYTRWDSTQQRAILKRAGDIMVRLSPEPDLARVVMDDLLAPSLLDVGDYKIVVEEGLPSGCPCTTQLNSLAHWILTLCAMVEVTRVDPDIVMQESEFSFYGDDEVVSTNLELDMVKYTMALRRYGLLPTRADPLERRQTLQGISFLRRAIVGDQFGWYGRLDRASIDRQLLWTKGPNHQNPFETLPGHAQRPSQLMALLGEAAMHGEKYYRTVASRVSKEAAQVVPRHRSVLRWVRFG 4o55 A 2.24 BS01 LF9 A 1 Q95 T124 T125 A128 A129 Q40 T69 T70 A73 A74 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 ic50=5.03uM remove_due_to_license_issue P12497 24874515 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGGYSAGERIVDIIATDIQ 4o5b A 2.37 BS01 LF9 A 1 Q95 T124 T125 T128 A129 Q40 T69 T70 T73 A74 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 24874515 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKTACWWAGIKQEFGIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGGYSAGERIVDIIATDIQ 4o5g A 2.301 BS03 2PV A 1 G57 D58 L60 H61 S62 R63 P91 G92 N93 G64 D65 L67 H68 S69 R70 P98 G99 N100 3.1.-.- 0004519,0006259,0008408,0016787 remove_due_to_license_issue Q9X1X0 24316220 403 IHHHHHHVINLKELKILHTSDWHLGVTSWTSSRPVDRREELKKALDKVVEEAEKREVDLILLTGDLLHSRNNPSVVALHDLLDYLKRMMRTAPVVVLPGNHDWKGLKLFGNFVTSISSDITFVMSFEPVDVEAKRGQKVRILPFPYPDESEALRKNEGDFRFFLESRLNKLYEEALKKEDFAIFMGHFTVEGLAGYAGIEQGREIIINRALIPSVVDYAALGHIHSFREIQKQPLTIYPGSLIRIDFGEEADEKGAVFVELKRGEPPRYERIDASPLPLKTLYYKKIDTSALKSIRDFCRNFPGYVRVVYEEDSGILPDLMGEIDNLVKIE 4o6e A 1.95 BS01 2SH A 1 E33 G34 G37 V39 A52 K54 Q105 M108 E109 T110 K114 N154 L156 D167 E21 G22 G25 V27 A40 K42 Q93 M96 E97 T98 K102 N142 L144 D155 D149 K151 S153 N154 D167 T190 D137 K139 S141 N142 D155 T167 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=1nM remove_due_to_license_issue IC50=1.000000nM, Ki=0.400000nM P28482 24813737 401 MVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPVATRWYRAPEIMLNYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKELDDLPKEKLKELIFEETARFQPG 4o70 A 1.55 BS01 1QK A 1 W81 F83 N140 D144 D145 I146 W40 F42 N99 D103 D104 I105 ? ic50=19uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o70 A 1.55 BS02 1QK A 2 K91 N93 K50 N52 ? ic50=19uM remove_due_to_license_issue O60885 24568369 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o71 A 1.36 BS01 CPB A 1 W81 P82 L92 N140 W40 P41 L51 N99 ? ic50=18uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o71 A 1.36 BS02 CPB B 1 F79 L148 M149 F38 L107 M108 ? ic50=18uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o72 A 1.4 BS01 2R4 A 1 W81 P82 F83 V87 L92 N140 I146 W40 P41 F42 V46 L51 N99 I105 ? ic50=1uM remove_due_to_license_issue IC50=1000nM O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o74 A 1.45 BS01 R78 A 1 W81 P82 V87 L92 Y97 Y139 N140 I146 W40 P41 V46 L51 Y56 Y98 N99 I105 ? ic50=0.025uM remove_due_to_license_issue IC50=25nM, Kd=37nM, Ki=56nM O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o75 A 1.55 BS01 2RC A 1 W81 P82 K91 L92 Y97 Y139 N140 W40 P41 K50 L51 Y56 Y98 N99 ? ic50=21uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o76 A 1.7 BS01 1M3 A 1 W81 P82 F83 L92 L94 N140 W40 P41 F42 L51 L53 N99 ? ic50=0.13uM remove_due_to_license_issue IC50=130nM, Kd=123nM O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o76 A 1.7 BS02 1M3 B 1 F79 W81 D145 M149 F38 W40 D104 M108 ? ic50=0.13uM remove_due_to_license_issue IC50=130nM, Kd=123nM O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o77 A 2.0 BS01 2RE A 1 W81 P82 V87 Y97 C136 N140 W40 P41 V46 Y56 C95 N99 ? ic50=2.5uM remove_due_to_license_issue IC50=2500nM, Kd=3400nM O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o78 A 1.34 BS01 SAV A 1 W81 P82 Q85 V87 L92 Y97 Y139 I146 W40 P41 Q44 V46 L51 Y56 Y98 I105 ? ic50=4.6uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7a A 1.34 BS01 2RF A 1 W81 P82 L92 N140 I146 W40 P41 L51 N99 I105 ? ic50=19uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7b A 1.5 BS01 2RJ A 1 W81 P82 F83 V87 L92 L94 Y97 N140 I146 W40 P41 F42 V46 L51 L53 Y56 N99 I105 ? ic50=20uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7c A 1.55 BS01 2RK A 1 W81 P82 V87 L92 N140 I146 W40 P41 V46 L51 N99 I105 ? ic50=10uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7d A 2.3 BS01 ONL A 1 Y249 Q285 S286 N335 E381 Y414 Y466 G483 V484 Y31 Q67 S68 N117 E163 Y196 Y248 G265 V266 S286 K289 Y414 Y466 V484 S68 K71 Y196 Y248 V266 3.5.1.2 0004359,0006541 remove_due_to_license_issue O94925 24451979 601 SMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 4o7e A 1.85 BS01 2RN A 1 W81 V87 L92 W40 V46 L51 ? ic50=5.7uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7e A 1.85 BS02 2RN A 2 F79 D145 M149 F38 D104 M108 ? ic50=5.7uM remove_due_to_license_issue O60885 24568369 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7e A 1.85 BS03 2RN B 1 W81 K91 L92 W40 K50 L51 ? ic50=5.7uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o7f A 1.8 BS01 2RQ A 1 W81 P82 F83 V87 L92 Y97 C136 N140 I146 W40 P41 F42 V46 L51 Y56 C95 N99 I105 ? ic50=13uM remove_due_to_license_issue O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4o91 A 2.393 BS01 NG2 A 1 A61 K63 E77 Q80 L81 I89 V90 M104 E105 A107 I153 H154 C174 D175 A35 K37 E51 Q54 L55 I63 V64 M78 E79 A81 I127 H128 C148 D149 D156 K158 P160 N161 I173 D175 D130 K132 P134 N135 I147 D149 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 25075558 601 SLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 4o97 A 2.2 BS02 NTX A 1 T98 F99 Q175 D189 S190 C191 Q192 S195 V213 W215 G216 T93 F94 Q169 D185 S186 C187 Q188 S191 V210 W212 G213 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 Ki=3nM remove_due_to_license_issue Ki=3.0nM Q9Y5Y6 24794746 900 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 4o9s A 2.3 BS01 2RY A 1 L35 F36 L37 A55 A57 M73 G75 M88 Y90 Y133 F135 L35 F36 L37 A55 A57 M73 G75 M88 Y90 Y133 F135 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 ic50=0.28uM remove_due_to_license_issue IC50=60nM P02753 24835984 201 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYCD 4o9v A 1.9 BS02 NT4 A 1 H57 I60 F99 D189 S190 S195 V213 W215 G216 G219 C220 H42 I45 F94 D185 S186 S191 V210 W212 G213 G215 C216 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 Ki=10nM remove_due_to_license_issue Ki=10.0nM Q9Y5Y6 24794746 900 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 4oag A 2.0 BS01 ADP A 1 S187 S189 H201 Q203 R326 S340 R342 K368 A382 S54 S56 H68 Q70 R191 S205 R207 K233 A247 ? 0005741,0007005 Kd=0.5uM remove_due_to_license_issue Q8BGV8 24508339 501 SLQEKLLSYYRNRAAIPAGEQARAKQAAVDICAELRSFLRAKLPDMPLRDMYLSGSLYDDLQVVTADHIQLIVPLVLEQNLWSCIPGEDTIMNVPGFFLVRRENPEYFPRGSSYWDRCVVGGYLSPKTVADTFEKVVAGSINWPAIGSLLDYVIRPAPEALTLEVQYEKDKHLVIDFLPSVTLGDTVLVARPHRLAQYDNLWRLSLRPAETARLRALDQADSGCRSLCLKILKAICKSTPALGHLTASQLTNVILHLAQEEADWSPDMLADRFLQALRGLISYLEAGVLPSALNPKVNLFAELTPQEIDELGYTLYCSLSEPEVLLQT 4oak A 2.0 BS02 DAL A 1 H95 D102 E153 W155 H156 H95 D102 E153 W155 H156 ? 0004180,0006508,0008233,0046872 remove_due_to_license_issue Q9JN36 24711382 202 MNTLQLINKNHPLKKNQEPPHLVLAPFSDHDVYLQPEVAKQWERLVRATGLEKDIRLVSGYRTEKEQRRLWEYSLKENGLAYTKQFVALPGCSEHQIGLAIDVGLKKQEDDDLICPHFRDSAAADLFMQQMMNYGFILRYPEDKQEITGISYEPWHFRYVGLPHSQVITAQKWTLEEYHDYLAQTVRQFA 4oak A 2.0 BS03 DAL A 2 F86 A88 S93 F86 A88 S93 ? 0004180,0006508,0008233,0046872 remove_due_to_license_issue Q9JN36 24711382 203 MNTLQLINKNHPLKKNQEPPHLVLAPFSDHDVYLQPEVAKQWERLVRATGLEKDIRLVSGYRTEKEQRRLWEYSLKENGLAYTKQFVALPGCSEHQIGLAIDVGLKKQEDDDLICPHFRDSAAADLFMQQMMNYGFILRYPEDKQEITGISYEPWHFRYVGLPHSQVITAQKWTLEEYHDYLAQTVRQFA 4oak B 2.0 BS02 DAL B 1 F86 H95 D102 I114 H156 F86 H95 D102 I114 H156 ? 0004180,0006508,0008233,0046872 remove_due_to_license_issue Q9JN36 24711382 202 MNTLQLINKNHPLKKNQEPPHLVLAPFSDHDVYLQPEVAKQWERLVRATGLEKDIRLVSGYRTEKEQRRLWEYSLKENGLAYTKQFVALPGCSEHQIGLAIDVGLKKQEDDDLICPHFRDSAAADLFMQQMMNYGFILRYPEDKQEITGISYEPWHFRYVGLPHSQVITAQKWTLEEYHDYLAQTVRQFA 4oak B 2.0 BS03 DAL B 2 R62 F86 A88 S93 H95 Y140 R62 F86 A88 S93 H95 Y140 ? 0004180,0006508,0008233,0046872 remove_due_to_license_issue Q9JN36 24711382 203 MNTLQLINKNHPLKKNQEPPHLVLAPFSDHDVYLQPEVAKQWERLVRATGLEKDIRLVSGYRTEKEQRRLWEYSLKENGLAYTKQFVALPGCSEHQIGLAIDVGLKKQEDDDLICPHFRDSAAADLFMQQMMNYGFILRYPEDKQEITGISYEPWHFRYVGLPHSQVITAQKWTLEEYHDYLAQTVRQFA 4oar A 2.41 BS02 2S0 A 1 N719 G722 Q725 M759 F794 L797 C891 T894 N38 G41 Q44 M78 F113 L116 C210 T213 ? ic50=0.038nM remove_due_to_license_issue EC50=>100nM, IC50=0.2nM P06401 25204619 1001 QLIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLGERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHDLVKQLHLYCLNTFIQSRMSEVIAAQLPKILAGMVKPLLFH 4oas A 1.7 BS01 2SW A 1 L54 G58 Q59 I61 V93 K94 H96 I99 Y100 L37 G41 Q42 I44 V76 K77 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 Kd=0.045nM remove_due_to_license_issue IC50=0.100000nM, Kd=0.036000nM Q00987 24456472 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4oaz A 2.25 BS01 C2E R 1 Q113 R114 R125 D128 Q31 R32 R43 D46 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 201 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADA 4oaz A 2.25 BS02 C2E R 2 R114 D116 R32 D34 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 202 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADA 4oaz A 2.25 BS03 C2E A 1 K84 R114 S123 I124 R125 Q126 K2 R32 S41 I42 R43 Q44 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 201 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADA 4oaz A 2.25 BS04 C2E A 2 D116 N118 L122 S123 D34 N36 L40 S41 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 202 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADA 4oaz R 2.25 BS01 C2E R 1 K84 R114 S123 I124 R125 Q126 K2 R32 S41 I42 R43 Q44 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 201 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLD 4oaz R 2.25 BS02 C2E R 2 R114 D116 N118 V121 L122 S123 R32 D34 N36 V39 L40 S41 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 202 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLD 4oaz R 2.25 BS03 C2E A 1 I110 Q113 R114 R125 D128 I28 Q31 R32 R43 D46 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 201 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLD 4oaz R 2.25 BS04 C2E A 2 R114 G115 D116 R32 G33 D34 ? 0045892 remove_due_to_license_issue Q7AKQ8 25171413 202 PKLVLDLERLATVPAEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLD 4ob0 A 1.2 BS02 PBC A 1 Q89 A111 S112 C113 Q88 A110 S111 C112 C108 C111 S112 C113 C107 C110 S111 C112 4.2.1.84 0003824,0005515,0016829,0018822,0046872,0046914,0050897,0050899 Ki=5uM remove_due_to_license_issue Q7SID2 24383915 302 TENILRKSDEEIQKEITARVKALESMLIEQGILTTSMIDRMAEIYENEVGPHLGAKVVVKAWTDPEFKKRLLADGTEACKELGIGGLQGEDMMWVENTDEVHHVVVCTLCSCYPWPVLGLPPNWFKEPQYRSRVVREPRQLLKEEFGFEVPPSKEIKVWDSSSEMRFVVLPQRPAGTDGWSEEELATLVTRESMIGVEPAKAV 4ob0 B 1.2 BS01 PBC A 1 F37 R52 F37 R52 R52 Y68 W72 R52 Y68 W72 4.2.1.84 0005515,0016829,0018822,0046914,0050899 remove_due_to_license_issue Q7SID3 24383915 302 MNGVYDVGGTDGLGPINRPADEPVFRAEWEKVAFAMFPATFRAGFMGLDEFRFGIEQMNPAEYLESPYYWHWIRTYIHHGVRTGKIDLEELERRTQYYRENPDAPLPEHEQKPELIEFVNQAVYGGLPASREVDRPPKFKEGDVVRFSTASPKGHARRARYVRGKTGTVVKHHGAYIYPDTAGNGLGECPEHLYTVRFTAQELWGPEGDPNSSVYYDCWEPYIELVDT 4ob1 A 1.631 BS02 BUB A 1 A111 S112 C113 W116 A110 S111 C112 W115 C108 C111 S112 C113 C107 C110 S111 C112 4.2.1.84 0003824,0005515,0016829,0018822,0046872,0046914,0050897,0050899 remove_due_to_license_issue Q7SID2 24383915 302 TENILRKSDEEIQKEITARVKALESMLIEQGILTTSMIDRMAEIYENEVGPHLGAKVVVKAWTDPEFKKRLLADGTEACKELGIGGLQGEDMMWVENTDEVHHVVVCTLCSCYPWPVLGLPPNWFKEPQYRSRVVREPRQLLKEEFGFEVPPSKEIKVWDSSSEMRFVVLPQRPAGTDGWSEEELATLVTRESMIGVEPAKAV 4ob2 A 1.52 BS01 BUB A 1 A111 S112 C113 A110 S111 C112 C108 C111 S112 C113 C107 C110 S111 C112 4.2.1.84 0003824,0005515,0016829,0018822,0046872,0046914,0050897,0050899 remove_due_to_license_issue Q7SID2 24383915 301 TENILRKSDEEIQKEITARVKALESMLIEQGILTTSMIDRMAEIYENEVGPHLGAKVVVKAWTDPEFKKRLLADGTEACKELGIGGLQGEDMMWVENTDEVHHVVVCTLCSCYPWPVLGLPPNWFKEPQYRSRVVREPRQLLKEEFGFEVPPSKEIKVWDSSSEMRFVVLPQRPAGTDGWSEEELATLVTRESMIGVEPAKAV 4oba A 1.602 BS01 2TW A 1 L54 G58 Q59 I61 M62 Y67 V93 H96 I99 Y100 L36 G40 Q41 I43 M44 Y49 V71 H74 I77 Y78 2.3.2.27 0005634,0043066,0051726 ic50=0.4nM remove_due_to_license_issue IC50=0.400000nM Q00987 24548297 501 IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4obo A 2.1 BS01 2QV A 1 Y36 V39 A52 K54 M105 F107 C108 L160 V170 D171 Y21 V24 A37 K39 M81 F83 C84 L136 V146 D147 D153 K155 Q157 N158 D171 T191 D129 K131 Q133 N134 D147 T156 2.7.11.1 0004672,0005524,0006468 ic50=0.077uM remove_due_to_license_issue IC50=92.7nM, Ki=108nM O95819 24673130 403 SSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEIKLEINMLKKYSHHRNIATYYGAFIKKSDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGRNTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTR 4obp A 2.27 BS02 2QU A 1 Y36 V39 A52 K54 M105 F107 C108 L160 D171 Y24 V27 A40 K42 M89 F91 C92 L144 D155 D153 K155 Q157 N158 D171 T191 D137 K139 Q141 N142 D155 T166 2.7.11.1 0004672,0005524,0006468 ic50=0.017uM remove_due_to_license_issue IC50=11.5nM O95819 24673130 403 IDLSSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEDEEEEIKLEINMLKKYSHHRNIATYYGAFIKKSDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVSANTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTR 4obq A 2.19 BS02 2QT A 1 Y36 V39 A52 K54 M105 F107 C108 L160 V170 D171 Y21 V24 A37 K39 M80 F82 C83 L135 V145 D146 D153 K155 Q157 N158 D171 T191 D128 K130 Q132 N133 D146 T155 2.7.11.1 0004672,0005524,0006468 ic50=0.065uM remove_due_to_license_issue IC50=58.6nM O95819 24673130 403 SSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVEINMLKKYSHHRNIATYYGAFIKKSPPGHDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVNTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTRK 4obv B 2.84 BS02 2SU B 1 P102 S105 F309 P462 E463 P87 S90 F294 P444 E445 4.1.1.105 0004058,0005737,0006520,0006568,0016830,0016831,0019752,0030170,0036469 remove_due_to_license_issue A7B1V0 25263219 501 TEYILNSTQLEEAIKSFVHDFCAEKHEIHDQPVVVEAKEHQEDKIKQIKIPEKGRPVNEVVSEMMNEVYRYRGDANHPRFFSFVPGPASSVSWLGDIMTSAYNIHAGGSKLAPMVNCIEQEVLKWLAKQVGFTENPGGVFVSGGSMANITALTAARDNKLTDINLHLGTAYISDQTHSSVAKGLRIIGITDSRIRRIPTNSHFQMDTTKLEEAIETDKKSGYIPFVVIGTAGTTNTGSIDPLTEISALCKKHDMWFHIDGAYGASVLLSPKYKSLLTGTGLADSISWDAHKWLFQTYGCAMVLVKDIRNLFHSFHVNPEYLKDLEDNVNTWDIGMELTRPARGLKLWLTLQVLGSDLIGSAIEHGFQLAVWAEEALNPKKDWEIVSPAQMAMINFRYAPKDLTKEEQDILNEKISHRILESGYAAIFTTVLNGKTVLRICAIHPEATQEDMQHTIDLLDQYGREIYTEMK 4obv D 2.84 BS01 2SU D 1 P102 A103 S104 S105 F309 P462 E463 P87 A88 S89 S90 F294 P444 E445 4.1.1.105 0004058,0005737,0006520,0006568,0016830,0016831,0019752,0030170,0036469 remove_due_to_license_issue A7B1V0 25263219 501 TEYILNSTQLEEAIKSFVHDFCAEKHEIHDQPVVVEAKEHQEDKIKQIKIPEKGRPVNEVVSEMMNEVYRYRGDANHPRFFSFVPGPASSVSWLGDIMTSAYNIHAGGSKLAPMVNCIEQEVLKWLAKQVGFTENPGGVFVSGGSMANITALTAARDNKLTDINLHLGTAYISDQTHSSVAKGLRIIGITDSRIRRIPTNSHFQMDTTKLEEAIETDKKSGYIPFVVIGTAGTTNTGSIDPLTEISALCKKHDMWFHIDGAYGASVLLSPKYKSLLTGTGLADSISWDAHKWLFQTYGCAMVLVKDIRNLFHSFHVNPEYLKDLEDNVNTWDIGMELTRPARGLKLWLTLQVLGSDLIGSAIEHGFQLAVWAEEALNPKKDWEIVSPAQMAMINFRYAPKDLTKEEQDILNEKISHRILESGYAAIFTTVLNGKTVLRICAIHPEATQEDMQHTIDLLDQYGREIYTEM 4obz A 2.9 BS01 2S4 B 1 D33 Y78 D32 Y77 D33 S36 N38 W40 Y78 D32 S35 N37 W39 Y77 3.4.23.5 0004190,0006508 remove_due_to_license_issue IC50=1900nM P07339 25086681 401 PIPEVLKNYMDAQYYGEIGIGTPPQCFTVVFDTGSSNLWVPSIHCKLLDIACWIHHKYNSDKSSTYVKNGTSFDIHYGSGSLSGYLSQDTVSVPCQS 4obz B 2.9 BS01 2S4 B 1 F131 I134 Y205 I229 D231 F25 I28 Y99 I123 D125 D231 T234 D125 T128 3.4.23.5 0004190,0006508 remove_due_to_license_issue IC50=1900nM P07339 25086681 401 GVKVERQVFGEATKQPGITFIAAKFDGILGMAYPRISVNNVLPVFDNLMQQKLVDQNIFSFYLSRDPDAQPGGELMLGGTDSKYYKGSLSYLNVTRKAYWQVHLDQVEVASGLTLCKEGCEAIVDTGTSLMVGPVDEVRELQKAIGAVPLIQGEYMIPCEKVSTLPAITLKLGGKGYKLSPEDYTLKVSQAGKTLCLSGFMGMDIPPPSGPLWILGDVFIGRYYTVFDRDNNRVGFAEAA 4oc0 A 1.85 BS04 2R7 A 1 R210 E424 E425 R463 D465 G518 N519 R534 R536 Y552 H553 Y700 R156 E370 E371 R409 D411 G464 N465 R480 R482 Y498 H499 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=318nM remove_due_to_license_issue Ki=318nM Q04609 24731280 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4oc1 A 1.75 BS04 2QS A 1 F209 R210 N257 E424 G427 L428 R463 D465 G518 N519 R534 A535 R536 F546 Y552 H553 K699 Y700 F155 R156 N203 E370 G373 L374 R409 D411 G464 N465 R480 A481 R482 F492 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=254nM remove_due_to_license_issue Q04609 24731280 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4oc2 A 1.65 BS05 2QQ A 1 R210 N257 E424 R463 D465 G518 N519 R534 R536 Y552 H553 Y700 R156 N203 E370 R409 D411 G464 N465 R480 R482 Y498 H499 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=5.3nM remove_due_to_license_issue Ki=5.3nM Q04609 24731280 821 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4oc3 A 1.79 BS04 2QP A 1 F209 R210 N257 E424 L428 R463 D465 G518 N519 R534 R536 Y552 H553 K699 Y700 F155 R156 N203 E370 L374 R409 D411 G464 N465 R480 R482 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=5.3nM remove_due_to_license_issue Ki=5.3nM Q04609 24731280 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4oc4 A 1.66 BS04 2QN A 1 F209 R210 E424 L428 R463 D465 G518 N519 R534 R536 F546 Y552 H553 K699 Y700 F154 R155 E369 L373 R408 D410 G463 N464 R479 R481 F488 Y494 H495 K639 Y640 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=105nM remove_due_to_license_issue Ki=105nM Q04609 24731280 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYNVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4oc5 A 1.7 BS04 2QM A 1 F209 R210 N257 E424 G427 L428 R463 D465 G518 N519 R534 R536 F546 Y552 H553 K699 Y700 F155 R156 N203 E370 G373 L374 R409 D411 G464 N465 R480 R482 F492 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=85nM remove_due_to_license_issue Ki=85.1nM Q04609 24731280 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4oc6 A 2.64 BS01 2S1 B 1 D33 G35 Y78 G79 S80 D33 G35 Y78 G79 S80 D33 S36 N38 W40 Y78 D33 S36 N38 W40 Y78 3.4.23.5 0004190,0006508 remove_due_to_license_issue IC50=85nM, Ki=0.700000nM P07339 25086681 402 GPIPEVLKNYMDAQYYGEIGIGTPPQCFTVVFDTGSSNLWVPSIHCKLLDIACWIHHKYNSDKSSTYVKNGTSFDIHYGSGSLSGYLSQDTVSVPCQS 4oc6 B 2.64 BS01 2S1 B 1 T125 F131 I134 I142 Y205 D231 G233 T234 S235 I311 S315 T20 F26 I29 I37 Y100 D126 G128 T129 S130 I206 S210 D231 T234 D126 T129 3.4.23.5 0004190,0006508 remove_due_to_license_issue IC50=85nM, Ki=0.700000nM P07339 25086681 402 GGVKVERQVFGEATKQPGITFIAAKFDGILGMAYPRISVNNVLPVFDNLMQQKLVDQNIFSFYLSRDPDAQPGGELMLGGTDSKYYKGSLSYLNVTRKAYWQVHLDQVEVASGLTLCKEGCEAIVDTGTSLMVGPVDEVRELQKAIGAVPLIQGEYMIPCEKVSTLPAITLKLGGKGYKLSPEDYTLKVSQAGKTLCLSGFMGMDIPPPSGPLWILGDVFIGRYYTVFDRDNNRVGFAEAARL 4occ A 1.8 BS01 2TZ A 1 L54 G58 Q59 I61 F86 K94 H96 I99 Y100 L37 G41 Q42 I44 F69 K77 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 ic50=2nM remove_due_to_license_issue IC50=2.0nM, Kd=0.392000nM Q00987 24601644 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4ock A 1.72 BS01 ANP A 1 Y27 G30 H31 I32 N33 I46 Q48 F104 I105 K210 I227 D228 Y25 G28 H29 I30 N31 I44 Q46 F102 I103 K208 I225 D226 2.7.1.162 0005524,0005975,0016301,0016773 remove_due_to_license_issue E8MF12 24816108 402 ESNEVLFGIASHFALEGAVTGIEPYGDGHINTTYLVTTDGPRYILQQMNTSIFPDTVNLMRNVELVTSTLKAQGKETLDIVPTTSGATWAEIDGGAWRVYKFIEHTVSYNLVPNPDVFREAGSAFGDFQNFLSEFDASQLTETIAHFHDTPHRFEDFKAALAADKLGRAAACQPEIDFYLSHADQYAVVMDGLRDGSIPLRVTHNDTKLNNILMDATTGKARAIIDLDTIMPGSMLFDFGDSIRFGASTALEDEKDLSKVHFSTELFRAYTEGFVGELRGSITAREAELLPFSGNLLTMECGMRFLADYLEGDIYFATKYPEHNLVRTRTQIKLVQEMEQKASETRAIVADIMEA 4ocp A 1.938 BS02 ADP A 1 G30 N33 I46 Q48 F104 I105 I227 D228 G28 N31 I44 Q46 F102 I103 I225 D226 2.7.1.162 0005524,0005975,0016301,0016773 remove_due_to_license_issue E8MF12 24816108 402 ESNEVLFGIASHFALEGAVTGIEPYGDGHINTTYLVTTDGPRYILQQMNTSIFPDTVNLMRNVELVTSTLKAQGKETLDIVPTTSGATWAEIDGGAWRVYKFIEHTVSYNLVPNPDVFREAGSAFGDFQNFLSEFDASQLTETIAHFHDTPHRFEDFKAALAADKLGRAAACQPEIDFYLSHADQYAVVMDGLRDGSIPLRVTHNDTKLNNILMDATTGKARAIIDLDTIMPGSMLFDFGDSIRFGASTALEDEKDLSKVHFSTELFRAYTEGFVGELRGSITAREAELLPFSGNLLTMECGMRFLADYLEGDIYFATKYPEHNLVRTRTQIKLVQEMEQKASETRAIVADIMEA 4oct A 2.28 BS02 AKG A 1 N193 Y195 H204 D206 H266 I268 R277 V279 I281 N110 Y112 H121 D123 H183 I185 R194 V196 I198 1.14.11.53 0006397,0035515 ic50=9uM remove_due_to_license_issue Q6P6C2 24778178 502 QKEEEARKVKSGIRQMRLFSQDECAKIEARIDEVVSRAEKGLYNEHTVDRAPLRNKYFFGEGYTRGPGQERLYPPGDVDEIPEWVHQLVIQKLVEHRVIPEGFVNSAVINDYQPGGCIVSHVDPIHIFERPIVSVSFFSDSALCFGCKFQFKPIRVSEPVLSLPVRRGSVTVLSGYAADEITHCIRPQDIKERRAVIILRKTRLDAPRL 4ocv A 1.472 BS01 ANP A 1 Y27 G30 H31 I32 N33 I46 Q48 F104 I105 K210 I227 Y24 G27 H28 I29 N30 I43 Q45 F101 I102 K207 I224 2.7.1.162 0016740 remove_due_to_license_issue B7GN78 24816108 402 TNEALFDVASHFALEGTVDSIEPYGDGHINTTYLVTTDGPRYILQRMNTGIFPDTVNLMRNVELVTSTLKAQGKETLDIVRTTSGDTWAEIDGGAWRVYKFIEHTMSYNLVPNPDVFREAGRAFGDFQNFLSGFDANQLTETIAHFHDTPHRFEDFKKALAADELGRAAGCGPEIEFYLSHADQYAVVMDGLRDGSIPLRVTHNDTKLNNILMDATTGKARAIIDLDTIMPGSMLFDFGDSIRFGASTALEDERDLDKVHFSTELFRAYTEGFVGELRDSITAREAELLPFSGNLLTMECGMRFLADYLEGDVYFATKYPEHNLVRSRTQIKLVREMEQRADETRAIVADVMETT 4ocx H 2.39 BS01 MT1 L 1 Y33 N36 Y51 Y99 Y33 N36 Y51 Y99 remove_due_to_license_issue 24832237 301 DVQLQESGPGLVKPSQSLSLTCTVTGFSITSPYAWNWIRQFPGNTLEWMGYISYRGSTTYHPSLKSRISITRDTSKNQFFLQLNSVTTEDTATYFCSSYGNYGAYSGQGTLVTVSAAKTTPPSVYPLAPGSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPR 4ocx L 2.39 BS01 MT1 L 1 H31 Y37 E39 F94 G96 L101 H31 Y37 E39 F94 G96 L101 ? 0046872 Kd~3.6pM remove_due_to_license_issue A2NHM3 24832237 301 DVLLTQIPLSLPVSLGDQASISCRSSQSIVHSNGNTYLEWYLQKPGQSPKLLIYKVSTRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFQGSHVPLTFGAGTQLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSPIVKSFNR 4ocz A 2.94 BS02 2RU A 1 F267 D335 M339 Y383 Y466 F267 D335 M339 Y383 Y466 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue Ki=0.660000nM P34913 25079952 603 MTLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 4od0 A 2.92 BS02 2RV A 1 F267 D335 W336 Y383 L408 M419 L428 Y466 F267 D335 W336 Y383 L408 M419 L428 Y466 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=3.7nM, Ki=0.910nM P34913 25079952 603 MTLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4od9 A 1.9 BS01 2RZ A 1 D33 G35 Y78 G79 S80 D32 G34 Y77 G78 S79 D33 S36 N38 W40 Y78 D32 S35 N37 W39 Y77 3.4.23.5 0004190,0006508 ic50=58nM remove_due_to_license_issue IC50=58nM P07339 25086681 103 PIPEVLKNYMDAQYYGEIGIGTPPQCFTVVFDTGSSNLWVPSIHCKLLDIACWIHHKYNSDKSSTYVKNGTSFDIHYGSGSLSGYLSQDTVSVPCQS 4od9 B 1.9 BS01 2RZ A 1 F126 F131 I134 Y205 I229 D231 G233 T234 M309 I311 F20 F25 I28 Y99 I123 D125 G127 T128 M203 I205 D231 T234 D125 T128 3.4.23.5 0004190,0006508 remove_due_to_license_issue IC50=58nM P07339 25086681 103 GVKVERQVFGEATKQPGITFIAAKFDGILGMAYPRISVNNVLPVFDNLMQQKLVDQNIFSFYLSRDPDAQPGGELMLGGTDSKYYKGSLSYLNVTRKAYWQVHLDQVEVASGLTLCKEGCEAIVDTGTSLMVGPVDEVRELQKAIGAVPLIQGEYMIPCEKVSTLPAITLKLGGKGYKLSPEDYTLKVSQAGKTLCLSGFMGMDIPPPSGPLWILGDVFIGRYYTVFDRDNNRVGFAEAA 4ode A 1.8 BS01 2U0 A 1 V14 L54 I61 V93 K94 H96 I99 Y100 V9 L49 I56 V88 K89 H91 I94 Y95 2.3.2.27 0005634,0043066,0051726 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM Q00987 24601644 201 MSVPTDGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4odf A 2.2006 BS01 2U1 A 1 V14 T16 S17 L54 G58 I61 Y67 V93 H96 I99 Y100 V3 T5 S6 L43 G47 I50 Y56 V82 H85 I88 Y89 2.3.2.27 0005634,0043066,0051726 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM Q00987 24601644 201 GAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4oe1 A 2.8 BS01 rna D 0 G431 K537 V597 S604 K608 I632 N635 D639 V668 N671 T672 N675 C678 K679 V703 T707 G710 G711 S714 L738 R742 G347 K453 V513 S520 K524 I548 N551 D555 V584 N587 T588 N591 C594 K595 V619 T623 G626 G627 S630 L654 R658 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 25231995 1 ~ 18 PDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPCVVTYNALLQVFGKAGNYTEALRVLGEMEQNGCQPDAVTYNELAGTEEAARCLDTMASPNAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYGSGAVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAFEEARGFLSEVKALEAYIEDA 4oe1 A 2.8 BS02 rna C 0 R175 T178 H182 V210 N213 R221 G245 F246 S249 T250 V281 N284 A285 Q288 V316 E320 R102 T105 H109 V137 N140 R148 G172 F173 S176 T177 V208 N211 A212 Q215 V243 E247 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 25231995 1 ~ 18 PDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPCVVTYNALLQVFGKAGNYTEALRVLGEMEQNGCQPDAVTYNELAGTEEAARCLDTMASPNAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYGSGAVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAFEEARGFLSEVKALEAYIEDA 4oe1 B 2.8 BS01 rna D 0 E151 G152 R175 H182 V210 N213 V214 F246 S249 T250 V281 N284 A285 E80 G81 R104 H111 V139 N142 V143 F175 S178 T179 V210 N213 A214 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 25231995 1 ~ 18 LSPDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPCVVTYNALLQVFGKAEALRVLGEMEQNGPDAVTYNELAGTYARAGFFEEAARCLDTMAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAKRFEEARGFLKALEAYIEDAQF 4oe1 B 2.8 BS02 rna C 0 R565 I632 N635 D639 N671 T672 N675 C678 K679 H706 G710 G711 S714 R742 R476 I543 N546 D550 N582 T583 N586 C589 K590 H617 G621 G622 S625 R653 ? 0003723,0003729,0006397,0009507,0009570,0042802,0048255 remove_due_to_license_issue B8Y6I0 25231995 1 ~ 18 LSPDAQVLVLAISSHPLPTLAAFLASRRDELLRADITSLLKALELSGHWEWALALLRWAGKEGAADASALEMVVRALGREGQHDAVCALLDETPLPPGSRLDVRAYTTVLHALSRAGRYERALELFAELRRQGVAPTLVTYNVVLDVYGRMGRSWPRIVALLDEMRAAGVEPDGFTASTVIAACSRDGLVDEAVAFFEDLKARGHAPCVVTYNALLQVFGKAEALRVLGEMEQNGPDAVTYNELAGTYARAGFFEEAARCLDTMAFTYNTVMTAYGNVGKVDEALALFDQMKKTGFVPNVNTYNLVLGMLGKKSRFTVMLEMLGEMSRSGCTPNRVTWNTMLAVSGKRGMEDYVTRVLEGMRSSGVELSRDTYNTLIAAYGRCGSRTNAFKMYNEMTSAGFTPCITTYNALLNVLSRQGDWSTAQSIVSKMRTKGFKPNEQSYSLLLQCYAKGGNVAGIAAIENEVYVFPSWVILRTLVIANFKCRRLDGMETAFQEVKARGYNPDLVIFNSMLSIYAKNGMYSKATEVFDSIKRSGLSPDLITYNSLMDMYAKCSESWEAEKILNQLKCSQTMKPDVVSYNTVINGFCKQGLVKEAQRVLSEMVADGMAPCAVTYHTLVGGYSSLEMFSEAREVIGYMVQHGLKPMELTYRRVVESYCRAKRFEEARGFLKALEAYIEDAQF 4oee A 1.5 BS01 IDY B 1 N27 R120 K125 Q134 K135 A136 N16 R109 K114 Q123 K124 A125 ? 0008083 remove_due_to_license_issue P09038 24959968 1 FPPGHFKDPKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVSANRYLAMKEDGRLLASKSVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMS 4oee A 1.5 BS02 GNX B 1 N27 K119 R120 K125 N16 K108 R109 K114 ? 0008083 remove_due_to_license_issue P09038 24959968 2 FPPGHFKDPKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVSANRYLAMKEDGRLLASKSVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMS 4oef A 1.8 BS01 IDY B 1 N27 R120 Q134 K135 A136 N9 R102 Q116 K117 A118 ? 0008083 remove_due_to_license_issue P09038 24959968 1 DPKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVSANRYLAMKEDGRLLASKSVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMS 4oef A 1.8 BS02 SGN B 1 N27 K119 R120 K125 N9 K101 R102 K107 ? 0008083 remove_due_to_license_issue P09038 24959968 2 DPKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVSANRYLAMKEDGRLLASKSVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMS 4oeg A 1.6 BS01 IDY B 1 N27 R120 Q134 K135 A136 N8 R101 Q115 K116 A117 ? 0008083 remove_due_to_license_issue P09038 24959968 1 PKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVSANRYLAMKEDGRLLASKSVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMS 4oeg A 1.6 BS02 SUS B 1 N27 K119 R120 K125 N8 K100 R101 K106 ? 0008083 remove_due_to_license_issue P09038 24959968 2 PKRLYCKNGGFFLRIHPDGRVDGVREKSDPHIKLQLQAEERGVVSIKGVSANRYLAMKEDGRLLASKSVTDECFFFERLESNNYNTYRSRKYTSWYVALKRTGQYKLGSKTGPGQKAILFLPMS 4oel A 1.4 BS01 SER A 1 D1 C234 G276 G277 F278 D1 C148 G190 G191 F192 Q228 C234 Q142 C148 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 22928782 501 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKVLHLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 4oel A 1.4 BS02 TYR A 1 G232 C234 E275 G146 C148 E189 Q228 C234 Q142 C148 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 22928782 502 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKVLHLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 4oem A 1.52 BS02 LYS A 1 G232 C234 G145 C147 Q228 C234 Q141 C147 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 22928782 502 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKVHLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 4oeu A 2.2 BS02 HIS A 1 H26 R344 Y374 I382 G383 W384 H480 H481 H25 R343 Y373 I381 G382 W383 H479 H480 ? 0015833,0042597,0043190,0046872,0055085,1904680 remove_due_to_license_issue Q0P844 25199691 502 IPKDTLIIAVENEIARINPAYSEDHDAVINLVFSGLTRFDENMSLKPDLAKSWDISKDGLVYDIFLRDDVLWHDGVKFSADDVKFSIEAFKNPKNNSSIYVNFEDIKSVEILNPSHVKITLFKPYPAFLDALSIGMLPKHLLENENLNTSSFNQNPIGTGPYKFVKWKKGEYVEFKANEHFYLDKVKTPRLIIKHIFDPSIASAELKNGKIDAALIDVSLLNIFKNDENFGILREKSADYRALMFNLDNEFLKDLKVRQALNYAVDKESIVKNLLHDYAFVANHPLERSWANSKNFKIYKYDPKKAEDLLVSAGFKKNKDGNFEKDGKILEFEIWAMSNDPLRVSLAGILQSEFRKIGVVSKVVAKPAGSFDYSKVDSFLIGWGSPLDPDFHTFRVFESSQDSALNDEGWNFGHYHDKKVDIALQKARNTSNLEERKKYYKDFIDALYENPPFIFLAYLDFALVYNKDLKGIKTRTLGHHGVGFTWNVYEWSK 4oew A 2.44 BS02 5IO A 1 A779 V782 A783 F786 Q817 F820 A227 V230 A231 F234 Q246 F249 3.1.4.35 0004114,0007165,0008081 Kd=0.000000064M remove_due_to_license_issue Kd=150nM O76074 24702184 903 TRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 4oex A 2.14 BS01 5EO A 1 V782 F786 M816 Q817 F820 V238 F242 M253 Q254 F257 3.1.4.35 0004114,0007165,0008081 Kd=0.000000064M remove_due_to_license_issue Kd=1500nM O76074 24702184 901 MEETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 4ofl A 2.7 BS01 HIS A 1 R344 W369 F383 G384 W385 Y406 H482 R342 W367 F381 G382 W383 Y404 H480 ? 0030288,0043190,0055085 remove_due_to_license_issue A0A5P8YI66 25199691 502 HTLQLAIGDEPTEGFDPMLGWSHGSYLLLHSPLLKQNEDFSWDSLLLSQYQPSDDGKTWLLTLKPDLKFSDGSPLTAKDVAFTYNNAAASGGKVDMGNFLSAEVIDPLNVRIHLKAPQSTFVNVLGSLGIVSADKYNAKTYAQKPIGAGPYRLVSFQPGQQMIVEANPYYAGNKNDFDKLIFVFLDEDSAFAAAQSGQLGVVRIPPSMAVGSVNNMKLWVRPSVENRGIVFPTTPAGKKDAHGYPIGNDVTADVAIRRAINYAINRQLLADQIMEGHAIPAYTGVQGLPWNNPDSAIKDGDIDKAKQILEQAGWQLNSQGTREKNGLPAKITLWYTSGDTTRRDLAQALRSMLKPIGIDVDLKSGSWETVERNMHANPTLFGWGSLDPMELYHHYSSNAAGVEYYNPGYYKNPMVDKHLQQALDAPTWQQAVPFWQQVDWDGTTGAGIRGDAAWAWLLNIQHTYLANNCVDLGKGTPEIHGSWSLLNSIDSWKWTC 4og3 A 2.01 BS01 2S6 A 1 S178 H181 F238 A242 M278 Y319 M322 Y323 W341 E363 S157 H160 F217 A221 M257 Y298 M301 Y302 W320 E342 ? 0005634 Kd=285nM remove_due_to_license_issue IC50=390nM, Kd=285nM O00255 24472025 602 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQ 4og4 A 1.45 BS01 2VK A 1 F238 A242 M278 Y319 M322 Y323 E363 F217 A221 M257 Y298 M301 Y302 E342 ? 0005634 Kd=952nM remove_due_to_license_issue IC50=529nM, Kd=952nM O00255 24472025 602 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPAPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 4og5 A 1.63 BS01 2S7 A 1 S155 S178 H181 F238 C241 A242 Y319 M322 Y323 E363 S134 S157 H160 F217 C220 A221 Y298 M301 Y302 E342 ? 0005634 ic50=302nM remove_due_to_license_issue IC50=195nM O00255 24472025 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPAPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 4og6 A 1.49 BS01 2S9 A 1 S178 D180 H181 F238 A242 M278 Y319 M322 Y323 E363 S157 D159 H160 F217 A221 M257 Y298 M301 Y302 E342 ? 0005634 ic50=197nM remove_due_to_license_issue IC50=197nM O00255 24472025 602 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 4og7 A 2.08 BS01 2SE A 1 E179 F238 C241 A242 Y319 M322 Y323 G326 E363 E158 F217 C220 A221 Y298 M301 Y302 G305 E342 ? 0005634 ic50=114nM remove_due_to_license_issue IC50=114nM O00255 24472025 602 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPGPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQM 4og8 A 1.53 BS02 2SF A 1 S178 H181 F238 A242 M278 Y319 M322 Y323 E363 S157 H160 F217 A221 M257 Y298 M301 Y302 E342 ? 0005634 ic50=56nM remove_due_to_license_issue Kd=110000nM, IC50=67nM, Ki=58nM O00255 24472025 602 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPGPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 4ogi A 1.73 BS01 R78 A 1 W81 P82 V87 L92 Y97 Y139 N140 I146 W40 P41 V46 L51 Y56 Y98 N99 I105 ? Kd=37nM remove_due_to_license_issue IC50=25nM, Kd=37nM, Ki=56nM O60885 24584101 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4ogj A 1.65 BS01 2TA A 1 W81 P82 F83 L92 L94 N140 W40 P41 F42 L51 L53 N99 ? Kd=164nM remove_due_to_license_issue Kd=164nM, IC50=290nM O60885 24584101 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4ogj A 1.65 BS02 2TA B 1 D145 M149 D104 M108 ? Kd=164nM remove_due_to_license_issue Kd=164nM, IC50=290nM O60885 24584101 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4ogn A 1.377 BS01 2U5 A 1 V14 T15 T16 L54 I61 Y67 V93 K94 H96 I99 V4 T5 T6 L44 I51 Y57 V83 K84 H86 I89 2.3.2.27 0005634,0043066,0051726 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM Q00987 24601644 201 DGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4ogt A 1.5361 BS01 2U6 A 1 T16 L54 I61 M62 V93 K94 H96 I99 Y100 T5 L43 I50 M51 V82 K83 H85 I88 Y89 2.3.2.27 0005634,0043066,0051726 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM Q00987 24601644 201 GAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4ogv A 2.197 BS01 2U7 A 1 L54 L57 I61 V93 H96 I99 Y100 L37 L40 I44 V72 H75 I78 Y79 2.3.2.27 0005634,0043066,0051726 ic50=9nM remove_due_to_license_issue IC50=9.0nM Q00987 24601644 501 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4ohk A 2.8 BS01 2TE A 1 P29 E32 G181 M213 R215 H504 W517 R518 A521 M522 R525 F526 P29 E32 G179 M211 R213 H483 W496 R497 A500 M501 R504 F505 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 24611879 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4ohm A 2.4 BS01 2TF A 1 P29 E32 G181 R215 K514 W517 A521 R525 P29 E32 G179 R213 K493 W496 A500 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue IC50=28nM Q14397 24611879 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4oho A 2.58 BS01 2TG A 1 V28 P29 E32 R215 H504 W517 R518 A521 R525 V28 P29 E32 R213 H483 W496 R497 A500 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue IC50=45nM Q14397 24611879 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4ohp A 2.4 BS01 2TJ A 1 V28 P29 E32 S34 G181 R215 K514 W517 A521 R525 V28 P29 E32 S34 G179 R213 K493 W496 A500 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue IC50=35nM Q14397 24611879 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4oiv A 1.7 BS01 XX9 A 1 A295 H298 M332 F333 S336 I366 M369 Y373 A452 L455 A32 H35 M69 F70 S73 I103 M106 Y110 A189 L192 ? 0003677,0004879,0006355,0032052,0038183 Kd=8.29uM remove_due_to_license_issue Q96RI1 26100621 501 ELTPDQQTLLHFIMDSYNKSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEERIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFAELLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLEEIW 4oiv B 1.7 BS01 XX9 B 1 L291 A295 H298 M332 F333 S336 M369 Y373 A452 L455 L44 A48 H51 M85 F86 S89 M115 Y119 A198 L201 ? 0003677,0004879,0006355,0032052,0038183 Kd=8.29uM remove_due_to_license_issue Q96RI1 26100621 501 ELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEEFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNSDLLEERIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFAELLGRLTELRTFNHHHAEMLMSWRVNDHKTPLLEEIW 4ojq A 2.25 BS01 2SX A 1 V232 T254 G255 T269 G271 Y502 V47 T69 G70 T84 G86 Y312 3.4.21.98,3.6.1.15,3.6.4.13 0004386,0005524 ic50=500uM remove_due_to_license_issue K4KA16 24467709 701 DNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGVDPNIRTGVRTITTGSPITYSTYGKFLADGGCSGGAYDIIICDECHSTDATSILGIGTVLDQAETAGARLVVLATATPPGSVTVSHPNIEEVALSTTGEIPFYGKAIPLEVIKGGRHLIFCHSKKKCDELAAKLVALGINAVAYYLDVSVIPDVVVVSTDALMTGFTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTLPQDAVSRTQRRGRTGRGKPGIYRFVAPGERPSGMFDSSVLCECYDAGCAWYELMPAETTVRLRAYMNTPGLPVCQDHLEFWEGVFTGLTHIDAHFLSQTKQSGENFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMTCMSADLEVV 4ojr A 1.82 BS01 2SQ A 1 A169 E170 H171 T174 M178 A101 E102 H103 T106 M110 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P03366 24904063 301 PGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTIHTDNGSNFTSATVKAACWWAGIKQGVVESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKSAGERIVDIIATD 4ok3 A 2.3 BS01 2SY A 1 V232 G255 T269 G271 K272 A275 A297 T298 A497 W501 Y502 V46 G69 T83 G85 K86 A89 A111 T112 A294 W298 Y299 3.4.21.98,3.6.1.15,3.6.4.13 0004386,0005524 ic50=71uM remove_due_to_license_issue K4KA16 24467709 701 NSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGVDPNIRTGVRTITTGSPITYSTYGKFLADGGCSGGAYDIIICDECHSTDATSILGIGTVLDQAETAGARLVVLATATPPGSVTVSHPNIEEVALSTTGEIPFYGKAIPLEVIKGGRHLIFCHSKKKCDELAAKLNAVASVIPDVVVVSTDALMTGGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTLPQDAVSRTQRRGRTGRGKPGIYRFVAPGERPSGMFDSSVLCECYDAGCAWYELMPAETTVRLRAYMNTPGLPVCQDHLEFWEGVFTGLTHIDAHFLSQTKQSGENFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMTCMSADLEV 4ok5 A 2.15 BS02 2T2 A 1 V232 G255 T269 G271 K272 A275 A297 T298 A497 W501 Y502 V49 G72 T86 G88 K89 A92 A114 T115 A309 W313 Y314 3.4.21.98,3.6.1.15,3.6.4.13 0004386,0005524 ic50=31uM remove_due_to_license_issue K4KA16 24467709 1003 FTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGVDPNIRTGVRTITTGSPITYSTYGKFLADGGCSGGAYDIIICDECHSTDATSILGIGTVLDQAETAGARLVVLATATPPGSVTVSHPNIEEVALSTTGEIPFYGKAIPLEVIKGGRHLIFCHSKKKCDELAAKLVALGINAVAYYRGLDVSVIPDVVVVSTDALMTTGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTLPQDAVSRTQRRGRTGRGKPGIYRFVAPGERPSGMFDSSVLCECYDAGCAWYELMPAETTVRLRAYMNTPGLPVCQDHLEFWEGVFTGLTHIDAHFLSQTKQSGENFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMTCMSADLEV 4ok6 A 2.4 BS02 2T7 A 1 V232 T254 G255 T269 G271 A275 T298 W501 Y502 V48 T70 G71 T85 G87 A91 T114 W302 Y303 3.4.21.98,3.6.1.15,3.6.4.13 0004386,0005524 ic50=14uM remove_due_to_license_issue K4KA16 24467709 1003 TDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGVDPNIRTGVRTITTGSPITYSTYGKFLADGGCSGGAYDIIICDECHSTDATSILGIGTVLDQAETAGARLVVLATATPPGSVTVSHPNIEEVALSTTGEIPFYGKAIPLEVIKGGRHLIFCHSKKKCDELAAKLINAVAYYRGLDVSVDVVVVSTDALMFDSVIDCNTCVTQTVDFSLDPTFTIETTTLPQDAVSRTQRRGRTGRGKPGIYRFVAPGERPSGMFDSSVLCECYDAGCAWYELMPAETTVRLRAYMNTPGLPVCQDHLEFWEGVFTGLTHIDAHFLSQTKQSGENFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMTCMSADLEV 4okg A 2.06 BS02 2SZ A 1 M62 E77 H78 T190 F191 M194 I197 R201 G209 S210 V216 D241 H264 M62 E77 H78 T190 F191 M194 I197 R201 G209 S210 V216 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue P47205 302 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 4okp B 1.37 BS01 2V0 B 1 W93 A160 K164 W90 A157 K161 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 24791931 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4oks A 2.25 BS01 2T9 A 1 V232 T254 G255 T269 G271 K272 A275 T298 A497 W501 Y502 V49 T71 G72 T86 G88 K89 A92 T115 A307 W311 Y312 3.4.21.98,3.6.1.15,3.6.4.13 0004386,0005524 Kd=33uM remove_due_to_license_issue K4KA16 24467709 701 FTDNSSPPAVPQSFQVAHLHAPTGSGKSTKVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGVDPNIRTGVRTITTGSPITYSTYGKFLADGGCSGGAYDIIICDECHSTDATSILGIGTVLDQAETAGARLVVLATATPPGSVTVSHPNIEEVALSTTGEIPFYGKAIPLEVIGRHLIFCHSKKKCDELAAKLVALGINAVAYYRGLDVSVIPTNGDVVVVSTDALGDFDSVIDCNTCVTQTVDFSLDPTFTIETTTLPQDAVSRTQRRGRTGRGKPGIYRFVAPGERPSGMFDSSVLCECYDAGCAWYELMPAETTVRLRAYMNTPGLPVCQDHLEFWEGVFTGLTHIDAHFLSQTKQSGENFPYLVAYQATVCARAQAPPPSWDQMWKCLIRLKPTLHGPTPLLYRLGAVQNEVTLTHPITKYIMTCMSADLEVV 4olc A 2.6 BS01 DCD A 1 D237 L239 S299 D236 L238 S291 G13 N14 K131 K216 K278 G12 N13 K130 K215 K270 2.7.2.2 0005829,0006525,0008804,0016301,0019546 remove_due_to_license_issue A8BB85 24558036 402 SAGKTVVIALGGNAMLQAKEKGDYDTQRKNVEIAASEIYKIHKAGYKVVLTSGNGPQVGAIKLQNQAAAGVSPEMPLHVCGAMSQGFIGYMMSQAMDNVFCANNEPANCVTCVTQTLVDPKDQAFTNPTKPVGRFYTEQEAKDLMAANPGKILREDAGRGWRVVVPSPRPLEIVEYGVIKTLIDNNVLVICTNGGGIPCKRENKVISGVDAVIDKDLATSLLAKTLNSDYLMILTDVLNACIRKLEEIKLSEILALEKDGHFAAGSMGPKVRAAIEFTQATGKMSIITSLSTAVDALNGKCGTRIIKD 4old A 1.48 BS01 2UZ A 1 V211 Y221 A318 T319 G320 V208 Y218 A308 T309 G310 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K305 A308 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 24791931 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 4olh A 2.4 BS01 2TO A 1 Y24 V28 P29 E32 R215 H504 K514 W517 R518 A521 M522 R525 Y24 V28 P29 E32 R213 H483 K493 W496 R497 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 25001129 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4oma A 1.6 BS01 LCS A 1 G88 I89 Y113 D185 S207 T209 K210 V338 S339 R374 G87 I88 Y112 D184 S206 T208 K209 V337 S338 R373 R60 Y113 D185 K210 R59 Y112 D184 K209 4.4.1.11 0005737,0016829,0016846,0018826,0019346,0030170 remove_due_to_license_issue Q84AR1 25398880 401 SDCRTYGFNTQIVHAGQQPDPSTGALSTPIFQTSTFVFDSAEQGAARFALEESGYIYTRLGNPTTDALEKKLAVLERGEAGLATASGISAITTTLLTLCQQGDHIVSASAIYGCTHAFLSHSMPKFGINVSFVDAAKPEEIRAAMRPETKVVYIETPANPTLSLVDIETVAGIAHQQGALLVVDNTFMSPYCQQPLQLGADIVVHSVTKYINGHGDVIGGIIVGKQEFIDQARFVGLKDITGGCMSPFNAWLTLRGVKTLGIRMERHCENALKIARFLEGHPSITRVYYPGLSSHPQYELGQRQMSLPGGIISFEIAGGLEAGRRMINSVELCLLAVSLGDTETLIQHPASMTHSPVAPEERLKAGITDGLIRLSVGLEDPEDIINDLEHAIRKAT 4omj A 1.6 BS01 2TX A 1 A108 Y153 H162 A167 A170 Y171 F174 L175 L189 A201 Y202 I205 A108 Y153 H162 A167 A170 Y171 F174 L175 L189 A201 Y202 I205 ? Kd=5.44uM remove_due_to_license_issue O76054 25987292 310 MSGRVGDLSPRQKEALAKFRENVQDVLPALPNPDDYFLLRWLRARSFDLQKSEAMLRKHVEFRKQKDIDNIISWQPPEVIQQYLSGGMCGYDLDGCPVWYDIIGPLDAKGLLFSASKQDLLRTKMRECELLLQECAHQTTKLGRKVETITIIYDCEGLGLKHLWKPAVEAYGEFLCMFEENYPETLKRLFVVKAPKLFPVAYNLIKPFLSEDTRKKIMVLGANWKEVLLKHISPDQVPVEYGGTMTDPDGNPKCKSKINYGGDIPRKYYVRDQV 4omk A 1.75 BS01 SQL A 1 A108 Y153 H162 A167 V168 L175 L189 F198 A201 Y202 I205 A108 Y153 H162 A167 V168 L175 L189 F198 A201 Y202 I205 ? Kd=40.1uM remove_due_to_license_issue O76054 25987292 305 MSGRVGDLSPRQKEALAKFRENVQDVLPALPNPDDYFLLRWLRARSFDLQKSEAMLRKHVEFRKQKDIDNIISWQPPEVIQQYLSGGMCGYDLDGCPVWYDIIGPLDAKGLLFSASKQDLLRTKMRECELLLQECAHQTTKLGRKVETITIIYDCEGLGLKHLWKPAVEAYGEFLCMFEENYPETLKRLFVVKAPKLFPVAYNLIKPFLSEDTRKKIMVLGANWKEVLLKHISPDQVPVEYGGTMTDPDGNPKCKSKINYGGDIPRKYYVRDQV 4omy A 3.062 BS01 dna E 0 V45 Q56 S57 S60 Q61 T80 I81 V40 Q51 S52 S55 Q56 T75 I76 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy A 3.062 BS02 dna F 0 N28 R31 S57 Q61 H62 N23 R26 S52 Q56 H57 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy B 3.062 BS01 dna E 0 N28 R31 S57 Q61 H62 R76 A78 Q79 N23 R26 S52 Q56 H57 R71 A73 Q74 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy B 3.062 BS02 dna F 0 A44 V45 G46 Q56 S57 S60 T80 I81 Y83 A39 V40 G41 Q51 S52 S55 T75 I76 Y78 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy C 3.062 BS01 dna G 0 N28 R31 S55 Q61 H62 R76 A78 Q79 N23 R26 S50 Q56 H57 R71 A73 Q74 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy C 3.062 BS02 dna H 0 V45 S57 S60 Q79 T80 I81 Y83 V40 S52 S55 Q74 T75 I76 Y78 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy D 3.062 BS01 dna G 0 V45 Q56 S57 S60 Q61 T80 I81 V40 Q51 S52 S55 Q56 T75 I76 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4omy D 3.062 BS02 dna H 0 N28 R31 L54 S55 S57 Q61 H62 N23 R26 L49 S50 S52 Q56 H57 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 A 3.0 BS01 dna E 0 V45 Q56 S57 S60 Q79 T80 I81 Y83 V40 Q51 S52 S55 Q74 T75 I76 Y78 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 A 3.0 BS02 dna F 0 N28 R31 S57 Q61 H62 K65 N23 R26 S52 Q56 H57 K60 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 B 3.0 BS01 dna E 0 N28 K30 R31 S57 Q61 H62 R76 A78 Q79 N23 K25 R26 S52 Q56 H57 R71 A73 Q74 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 B 3.0 BS02 dna F 0 A44 V45 Q56 S57 S60 R67 Q79 T80 I81 Y83 A39 V40 Q51 S52 S55 R62 Q74 T75 I76 Y78 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 C 3.0 BS01 dna G 0 V45 Q56 S57 S60 Q79 T80 I81 Y83 V40 Q51 S52 S55 Q74 T75 I76 Y78 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 C 3.0 BS02 dna H 0 N28 R31 S57 Q61 H62 N23 R26 S52 Q56 H57 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 D 3.0 BS01 dna G 0 N28 K30 R31 S57 Q61 H62 K65 R76 A78 Q79 N23 K25 R26 S52 Q56 H57 K60 R71 A73 Q74 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 1 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4on0 D 3.0 BS02 dna H 0 V45 Q56 S57 S60 R67 Q79 T80 I81 V40 Q51 S52 S55 R62 Q74 T75 I76 ? 0003700,0006355 remove_due_to_license_issue Q83TD2 24733893 2 ~ 22 QPLSPEKHEEAEIAAGFLSAMANPKRLLILDSLVKEEMAVGALANKVGLSQSALSQHLSKLRAQNLVSTRRDAQTIYYSSSSDSVMKILGALSEIYG 4ona A 2.4 BS01 UW1 A 1 L57 G58 V65 A78 K80 M112 L126 V130 Y131 L181 I194 D195 L198 L15 G16 V23 A36 K38 M70 L84 V88 Y89 L139 I152 D153 L156 D174 K176 E178 N179 D195 T214 D132 K134 E136 N137 D153 T172 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 ic50=0.002uM remove_due_to_license_issue IC50=2.00nM Q9BJF5 24494061 601 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 4ono A 2.705 BS01 PMK A 1 V127 Q129 S144 G145 H153 W155 I162 F185 Y188 L189 L192 V274 C282 V111 Q113 S128 G129 H137 W139 I146 F169 Y172 L173 L176 V253 C261 ? 0000139,0001913,0001916,0002237,0002474,0002481,0002502,0002503,0002726,0005198,0005515,0005576,0005615,0005765,0005783,0005788,0005794,0005829,0005886,0005925,0006826,0006879,0006955,0007608,0007611,0009897,0009986,0010977,0012507,0016020,0019885,0019886,0023026,0030670,0031901,0031902,0031905,0032092,0033077,0034756,0035580,0042026,0042605,0042612,0042613,0042802,0042803,0042824,0045646,0048260,0050680,0050768,0050778,0050870,0051289,0055038,0060586,0070062,0071281,0071283,0071316,1900121,1900122,1904434,1904437,1904724,1990000,1990712,2000774,2000978 remove_due_to_license_issue P29016,P29017,P61769 25298532 401 PIQRTPKIQVYSRHPAENGKSNFLNCYVSGFHPSDIEVDLLKNGERIEKVEHSDLSFSKDWSFYLLYYTEFTPTEKDEYACRVNHVTLSQPKIVKWDRDMGGGGEHVSFHVIQIFSFVNQSWARGQGSGWLDELQTHGWDSESGTIIFLHQWSKGQFSNEELSDLELLFRFYLFGLTREIQDHASYPFEVQVKAGCELHSGGSPEGFFQVAFNGLDLLSFQQTTWVPSPGCGSLAQSVCHLLNHQYEGVTETVYNLIRSTCPRFLLGLLDAGKMYVHRQVKPEAWLSSGPSPGPGRLQLVCHVSGFYPKPVWVMWMRGEQEQQGTQLGDILPNAQGTWYLRATLDVADGEAAGLSCRVKHSSLEGQDIILYWHH 4oo9 A 2.6 BS01 2U8 A 1 I625 S654 P655 S658 Y659 P743 L744 N747 W785 F788 S805 V806 S809 A810 I58 S87 P88 S91 Y92 P320 L321 N324 W362 F365 S382 V383 S386 A387 E1011 D1020 E121 D130 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P41594 25042998 4005 SPVQYLRWGDPAPIAAVVFACLGLLATLFVTVVFIIYRDTPVVKSSSRELCYIILAGICLGYLCTFCLIAKPKQIYCYLQRIGIGLSPAMSYSALVTKTYRAARILAMSKKNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKISACAQLVIAFILICIQLGIIVALFIMEPPDIMVYLICNTTNLGVVAPLGYNGLLILACTFYAFKTRNVPANFNEAKYIAFTMYTTCIIWLAFVPIYFGSNYKIITMCFSVSLSATVALGCMFVPKVYIILAKPERN 4ool A 2.3 BS01 2U2 A 1 E291 S294 R331 V333 S349 Y409 S485 G486 T487 A488 R489 F533 E239 S242 R279 V281 S297 Y357 S433 G434 T435 A436 R437 F471 0005886,0008658,0008955,0009252,0051301 remove_due_to_license_issue 24694215 601 VRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKNAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLP 4oon A 3.2 BS01 2U4 A 1 Q458 S461 N522 L559 T696 G697 T698 T699 N700 Y733 Q221 S224 N274 L311 T406 G407 T408 T409 N410 Y443 2.4.99.28,3.4.16.4 0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0016757,0030288,0046677,0071555 remove_due_to_license_issue Q07806 24694215 901 PLKVYSEDGKLISEFGEMTPELNAPYIAEMARAEMVGRYGSEAYTEGYKVITTVRSDLQNAASQSVRDGLIDYDQRHGYRGPETRLPGQTRDAWLKHLGQQRSIGGLEPAIVTQVEKSGIMVMTRDGKEEAVTWDSMKWARPFLSNNSMGPMPRQPADVAQAGDQIRVQRQEDGTLRFVQIPAAQSALISLDPKDGAIRSLVGGFSFEQSNYNRAIQAKRQPGSSFKPFIYSAALDNGFTAASLVNDAPIVFVDEYLTFLGPIPLREALYKSRNMVSIRVLQGLGIERAISYITKFGFQRDELPRNFSLALGTATVTPMEIAGAWSVFANGGYKVNPYVIERIESRDGQVLYQANPPRVPVEPTPAERIIDARTAYIMTSMLQDVIKRGTGRRALALKRTDLAGKTGTTNDSKDGWFSGYNSDYVTSVWVGFDQPETLGRREYGGTVALPIWIRYMGFALKDKPMHTMAEPPGIVSLRIDPVTGRSAAPGTPGAYFEMFKNE 4oow A 2.57 BS01 CAQ A 1 A97 R168 A97 R165 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue O92972 25053847 601 SMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPADLSGWFVAGYSGGDIYH 4op1 A 2.39 BS01 2UW A 1 V28 P29 E32 R215 H504 K514 W517 R518 A521 M522 R525 V28 P29 E32 R213 H483 K493 W496 R497 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 25914941 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4op2 A 2.24 BS01 2UX A 1 V28 P29 E32 G181 R215 H504 K514 W517 R518 A521 M522 R525 V28 P29 E32 G179 R213 H483 K493 W496 R497 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 25914941 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4op3 A 2.82 BS01 2UY A 1 A27 P29 E32 G181 M213 R215 H504 K514 W517 R518 A521 M522 R525 A27 P29 E32 G179 M211 R213 H483 K493 W496 R497 A500 M501 R504 ? 0001678,0005515,0005634,0005654,0005737,0005739,0005829,0006606,0009749,0009750,0019210,0033132,0034504,0046415,0070095,0070328,0097367,0141089,1901135 remove_due_to_license_issue Q14397 25914941 701 MPGTKRFQHVIETPEPGKWELSGYEAAVPITEKSNPLTQDLDKADAENIVRLLGQCDAEIFQEEGQSTYQRLYSESILTTMVQVAGKVQEVLKEPDGGLVVLSGGGTSGRMAFLMSVSFNQLMKGLGQKPLYTYLIAGGDRSVVASREGTEDSALHGIEELKKVAAGKKRVIVIGISVGLSAPFVAGQMDCCMNNTAVFLPVLVGFNPVSMARNDPIEDWSSTFRQVAERMQKMQEKQKAFVLNPAIGPEGLSGSSRMKGGSATKILLETLLLAAHKTVDQGIAASQRCLLEILRTFERAHQVTYSQSPKIATLMKSVSTSLEKKGHVYLVGWQTLGIIAIMDGVECIHTFGADFRDVRGFLIFTFSQEDFLTSILPSLTEIDTVVFIFTLDDNLTEVQTIVEQVKEKTNHIQALAHSTVGQTLPIPLKKLFPSIISITWPLLFFEYEGNFIQKFQRELSTKWVLNTVSTGAHVLLGKILQNHMLDLRISNSKLFWRALAMLQRFSGQSKARCIESLLRAIHFPQPLSDDIRAAPISCHVQVAHEKEQVIPIALLSLLFRCSITEAQAHLAAAPSVCEAVRSALA 4oq3 A 2.3 BS01 2V8 A 1 L54 G58 I61 F91 V93 H96 I99 L37 G41 I44 F74 V76 H79 I82 2.3.2.27 0005634,0043066,0051726 ic50=0.008uM remove_due_to_license_issue IC50=8.0nM Q00987 24704029 201 QIPASEQETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4oq3 A 2.3 BS02 2V8 C 1 Y76 P89 Y59 P72 2.3.2.27 0005634,0043066,0051726 ic50=0.008uM remove_due_to_license_issue IC50=8.0nM Q00987 24704029 201 QIPASEQETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4oq5 A 2.86 BS01 2UU A 1 M231 L235 M250 V253 R263 T266 L267 F270 M60 L64 M79 V82 R92 T94 L95 F98 ? 0042981 remove_due_to_license_issue IC50=500nM Q07820 24582986 401 MDLYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4oq5 A 2.86 BS02 2UU F 1 A227 G230 M231 A56 G59 M60 ? 0042981 remove_due_to_license_issue IC50=500nM Q07820 24582986 401 MDLYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4oq6 A 1.81 BS01 2UV A 1 M231 M250 F254 R263 T266 L267 M52 M71 F75 R84 T87 L88 ? 0042981 ic50=3.3uM remove_due_to_license_issue IC50=3300nM Q07820 24582986 401 DLYRQSLEIISRYLREQATGAKSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 4or0 A 2.58 BS01 NPS A 1 N390 R409 Y410 K413 V432 G433 L452 S488 N389 R408 Y409 K412 V431 G432 L451 S487 ? 0003677,0005504,0005515,0005576,0005615,0005737,0008289,0009267,0015643,0019825,0030170,0032991,0046872,0051902,0072732,1903981 remove_due_to_license_issue P02769 24753230 601 THKSEIAHRFKDLGEEHFKGLVLIAFSQYLQQCPFDEHVKLVNELTEFAKTCVADESHAGCEKSLHTLFGDELCKVASLRETYGDMADCCEKQEPERNECFLSHKDDSPDLPKLKPDPNTLCDEFKADEKKFWGKYLYEIARRHPYFYAPELLYYANKYNGVFQECCQAEDKGACLLPKIETMREKVLTSSARQRLRCASIQKFGERALKAWSVARLSQKFPKAEFVEVTKLVTDLTKVHKECCHGDLLECADDRADLAKYICDNQDTISSKLKECCDKPLLEKSHCIAEVEKDAIPENLPPLTADFAEDKDVCKNYQEAKDAFLGSFLYEYSRRHPEYAVSVLLRLAKEYEATLEECCAKDDPHACYSTVFDKLKHLVDEPQNLIKQNCDQFEKLGEYGFQNALIVRYTRKVPQVSTPTLVEVSRSLGKVGTRCCTKPESERMPCTEDYLSLILNRLCVLHEKTPVSEKVTKCCTESLVNRRPCFSALTPDETYVPKAFDEKLFTFHADICTLPDTEKQIKKQTALVELLKHKPKATEEQLKTVMENFVAFVDKCCAADDKEACFAVEGPKLVVSTQTALA 4or0 A 2.58 BS02 NPS A 2 F205 R208 A209 A212 K350 S479 L480 V481 F204 R207 A208 A211 K349 S478 L479 V480 ? 0003677,0005504,0005515,0005576,0005615,0005737,0008289,0009267,0015643,0019825,0030170,0032991,0046872,0051902,0072732,1903981 remove_due_to_license_issue P02769 24753230 602 THKSEIAHRFKDLGEEHFKGLVLIAFSQYLQQCPFDEHVKLVNELTEFAKTCVADESHAGCEKSLHTLFGDELCKVASLRETYGDMADCCEKQEPERNECFLSHKDDSPDLPKLKPDPNTLCDEFKADEKKFWGKYLYEIARRHPYFYAPELLYYANKYNGVFQECCQAEDKGACLLPKIETMREKVLTSSARQRLRCASIQKFGERALKAWSVARLSQKFPKAEFVEVTKLVTDLTKVHKECCHGDLLECADDRADLAKYICDNQDTISSKLKECCDKPLLEKSHCIAEVEKDAIPENLPPLTADFAEDKDVCKNYQEAKDAFLGSFLYEYSRRHPEYAVSVLLRLAKEYEATLEECCAKDDPHACYSTVFDKLKHLVDEPQNLIKQNCDQFEKLGEYGFQNALIVRYTRKVPQVSTPTLVEVSRSLGKVGTRCCTKPESERMPCTEDYLSLILNRLCVLHEKTPVSEKVTKCCTESLVNRRPCFSALTPDETYVPKAFDEKLFTFHADICTLPDTEKQIKKQTALVELLKHKPKATEEQLKTVMENFVAFVDKCCAADDKEACFAVEGPKLVVSTQTALA 4or0 A 2.58 BS03 NPS A 3 R194 L197 W213 R217 L480 R193 L196 W212 R216 L479 ? 0003677,0005504,0005515,0005576,0005615,0005737,0008289,0009267,0015643,0019825,0030170,0032991,0046872,0051902,0072732,1903981 remove_due_to_license_issue P02769 24753230 603 THKSEIAHRFKDLGEEHFKGLVLIAFSQYLQQCPFDEHVKLVNELTEFAKTCVADESHAGCEKSLHTLFGDELCKVASLRETYGDMADCCEKQEPERNECFLSHKDDSPDLPKLKPDPNTLCDEFKADEKKFWGKYLYEIARRHPYFYAPELLYYANKYNGVFQECCQAEDKGACLLPKIETMREKVLTSSARQRLRCASIQKFGERALKAWSVARLSQKFPKAEFVEVTKLVTDLTKVHKECCHGDLLECADDRADLAKYICDNQDTISSKLKECCDKPLLEKSHCIAEVEKDAIPENLPPLTADFAEDKDVCKNYQEAKDAFLGSFLYEYSRRHPEYAVSVLLRLAKEYEATLEECCAKDDPHACYSTVFDKLKHLVDEPQNLIKQNCDQFEKLGEYGFQNALIVRYTRKVPQVSTPTLVEVSRSLGKVGTRCCTKPESERMPCTEDYLSLILNRLCVLHEKTPVSEKVTKCCTESLVNRRPCFSALTPDETYVPKAFDEKLFTFHADICTLPDTEKQIKKQTALVELLKHKPKATEEQLKTVMENFVAFVDKCCAADDKEACFAVEGPKLVVSTQTALA 4or4 A 2.21 BS01 M7G A 1 F327 R334 K341 W359 E363 F406 S431 F6 R13 K20 W38 E42 F85 S110 ? 0033650 remove_due_to_license_issue A0A0J9X1Y8 25691568 501 RQRFRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSKMKLEKLLINSAKKEDMRDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSSDLFDQWGYEESPKASELHGINESMNASDYTLKGVVVTKN 4or6 A 2.293 BS01 GDP A 1 F327 R334 K341 W359 E363 F406 S431 F6 R13 K20 W38 E42 F85 S110 ? 0033650 remove_due_to_license_issue A0A0J9X1Y8 25691568 501 RQRFRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSKMKLEKLLINSAKKEDMRDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSSDLFDQWGYEESPKASELHGINESMNASDYTLKGVVVTKN 4osf A 1.62 BS01 4MT A 1 P2 M3 K33 Y37 H63 S64 I65 V107 P1 M2 K32 Y36 H62 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4osf A 1.62 BS02 4MT B 1 Y96 N98 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4osf C 1.62 BS01 4MT A 1 Y96 N98 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4osf C 1.62 BS02 4MT C 1 P2 M3 K33 H63 I65 V107 P1 M2 K32 H62 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 25743213 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4ot6 A 2.05 BS01 2V1 A 1 L408 T410 V416 A428 M477 A478 G480 N484 L528 L15 T17 V23 A35 M84 A85 G87 N91 L135 D521 A523 R525 N526 D539 F559 D128 A130 R132 N133 D146 F166 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 24712864 701 SWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4otf A 1.95 BS01 2VL A 1 L408 T410 G411 Q412 F413 V416 A428 K430 Y476 M477 G480 L528 D539 L13 T15 G16 Q17 F18 V21 A33 K35 Y81 M82 G85 L133 D144 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.006uM remove_due_to_license_issue IC50=6.0nM, EC50=380nM Q06187 25701252 704 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 4otg A 2.6 BS01 2V9 A 1 L627 G628 F632 V635 A648 Y703 S704 G707 L753 L17 G18 F22 V25 A38 Y93 S94 G97 L143 D746 K748 D750 N751 D764 T784 D136 K138 D140 N141 D154 T174 2.7.11.13 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q16512 25111382 1001 LRKSPLTLEDFKFLAVLGRGHFGKVLLSEFRPSGELFAIKALKKGDIVARDEVESLMCEKRILAAVTSAGHPFLVNLFGCFQTPEHVCFVMEYSAGGDLMLHIHSDVFSEPRAIFYSACVVLGLQFLHEHKIVYRDLKLDNLLLDTEGYVKIADFGLCKEGMGYGDRTSTFCGTPEFLAPEVLTDTSYTRAVDWWGLGVLLYEMLVGESPFPGDDEEEVFDSIVNDEVRYPRFLSAEAIGIMRRLLRRNPERRLGSSERDAEDVKKQPFFRTLGWEALLARRLPPPFVPTLFTGEAPTLSPPRDARPLTAAEQAAFLDFDFVAG 4oth A 1.8 BS01 DRN A 1 G628 F632 A648 K650 M701 S704 D708 D750 L753 A763 D764 F910 G17 F21 A37 K39 M90 S93 D97 D139 L142 A152 D153 F270 D746 K748 D750 N751 D764 D135 K137 D139 N140 D153 2.7.11.13 0004672,0004674,0005524,0006468 ic50=9nM remove_due_to_license_issue Q16512 25111382 1001 RKSPLTLEDFKFLAVLGRGHFGKVLLSEFRPSGELFAIKALKKGDIVARDEVESLMCEKRILAAVTSAGHPFLVNLFGCFQTPEHVCFVMEYSAGGDLMLHIHSDVFSEPRAIFYSACVVLGLQFLHEHKIVYRDLKLDNLLLDTEGYVKIADFGLCKTRAVDWWGLGVLLYEMLVGESPFPGDDEEEVFDSIVNDEVRYPRFLSAEAIGIMRRLLRRNPERRLGSSERDAEDVKKQPFFRTLGWEALLARRLPPPFVPTLSGRTDVSNFDEEFTGEAPTLSPPRDARPLTAAEQAAFLDFDFVAG 4oti A 1.93 BS01 MI1 A 1 G628 R629 G630 G633 V635 A648 S704 L753 F910 G17 R18 G19 G22 V24 A37 S93 L142 F268 D746 K748 D750 N751 D764 D135 K137 D139 N140 D153 2.7.11.13 0004672,0004674,0005524,0006468 ic50=43nM remove_due_to_license_issue Kd=200nM Q16512 25111382 1001 RKSPLTLEDFKFLAVLGRGHFGKVLLSEFRPSGELFAIKALKKGDIVARDEVESLMCEKRILAAVTSAGHPFLVNLFGCFQTPEHVCFVMEYSAGGDLMLHIHSDVFSEPRAIFYSACVVLGLQFLHEHKIVYRDLKLDNLLLDTEGYVKIADFGLTRAVDWWGLGVLLYEMLVGESPFPGDDEEEVFDSIVNDEVRYPRFLSAEAIGIMRRLLRRNPERRLGSSERDAEDVKKQPFFRTLGWEALLARRLPPPFVPTLSGRTDVSNFDEEFTGEAPTLSPPRDARPLTAAEQAAFLDFDFVAG 4oty A 2.354 BS01 LUR A 1 Y348 V349 L352 Y385 W387 M522 G526 A527 S530 Y317 V318 L321 Y354 W356 M491 G495 A496 S499 Q203 H207 L384 Y385 H388 G526 S530 Q172 H176 L353 Y354 H357 G495 S499 1.14.99.1 0001516,0001525,0004601,0004666,0005515,0005634,0005637,0005640,0005737,0005783,0005789,0005901,0006979,0007566,0007612,0007613,0008217,0008284,0008285,0009410,0009624,0009750,0010042,0010269,0010575,0016020,0016702,0019371,0019899,0020037,0030216,0030282,0031394,0031622,0031915,0032227,0032310,0032355,0032496,0032991,0033138,0033280,0034097,0034605,0034612,0035633,0042127,0042307,0042633,0042803,0043005,0043065,0043066,0045429,0045786,0045907,0045986,0045987,0046697,0046872,0048661,0050873,0051213,0051384,0051926,0051968,0070542,0071222,0071260,0071284,0071318,0071456,0071471,0071498,0071636,0090050,0090271,0090336,0090362,0098869,0150077,1902219,1905375,1990776,2000117 ic50=0.04uM remove_due_to_license_issue IC50=40nM Q05769 24060487 705 ANPCCSNPCQNRGECMSTGFDQYKCDCTRTGFYGENCTTPEFLTRIKLLLKPTPNTVHYILTHFKGVWNIVNNIPFLRSLIMKYVLTSRSYLIDSPPTYNVHYGYKSWEAFSNLSYYTRALPPVADDCPTPMGVKGNKELPDSKEVLEKVLLRREFIPDPQGSNMMFAFFAQHFTHQFFKTDHKRGPGFTRGLGHGVDLNHIYGETLDRQHKLRLFKDGKLKYQVIGGEVYPPTVKDTQVEMIYPPHIPENLQFAVGQEVFGLVPGLMMYATIWLREHNRVCDILKQEHPEWGDEQLFQTSRLILIGETIKIVIEDYVQHLSGYHFKLKFDPELLFNQQFQYQNRIASEFNTLYHWHPLLPDTFNIEDQEYSFKQFLYNNSILLEHGLTQFVESFTRQIAGRVAGGRNVPIAVQAVAKASIDQSREMKYQSLNEYRKRFSLKPYTSFEELTGEKEMAAELKALYSDIDVMELYPALLVEKPRPDAIFGETMVELGAPFSLKGLMGNPICSPQYWKPSTFGGEVGFKIINTASIQSLICNNVKGCPFTSFNVQ 4oue A 2.35 BS01 IPT A 1 D188 G189 A190 T219 W230 E234 E254 D277 D165 G166 A167 T196 W207 E211 E231 D254 3.2.1.111 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A5P6 24527659 502 SLAPCGLVPSARQLEWYNREMIAFFHFGINTFEEYVNEGDGKASTAIFNPTALDCRQWMQTLKAAGIPAAILTAKHADGFCLWPSKYTDYSVKNAAWKNGKGDVVREFVDACEEYGLKAGIYLGPHDRHEHLSPLYTTERYKEYYAHQLGELMSDYGKIWETWWDGAGADELTTPVYRHWYKIVREKQPDCVIFGTKNSYPFADVRWMGNEAGEAGDPCWATTDSVAIRDEAQYYKGLNEGMLDGDAYIPAETDVSIRPSWFYHAEEDSRVKSVRELWDIYCTSVGRNSVLLLNFPPDRRGLIHSTDSLHAALLKQGIDETFSTNLLRGAKVKATNVRGAKYSPEKMLDNEKNTYFAGKDGEVKADIIFTLPKTIEFDCLMIEEVIELGHRTTKWSVEYTVDGKNWITIPEATDKQAIGHKWIVRLAPVKAKQVRLRIQDGKACPAIHTFGVYKQSPVF 4ovf A 2.05 BS02 2VG A 1 R152 Y154 T172 G174 R176 L177 P242 V247 M362 R148 Y150 T168 G170 R172 L173 P238 V243 M358 0003677,0003887,0006260,0008408,0009360 remove_due_to_license_issue 25970224 407 MKFTVEREHLLKPLQQVSGPPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4ovg A 1.9 BS01 2VF A 1 R152 Y154 T172 G174 R176 L177 V247 V360 M362 R147 Y149 T167 G169 R171 L172 V242 V355 M357 0003677,0003887,0006260,0008408,0009360 remove_due_to_license_issue 25970224 401 MKFTVEREHLLKPLQQVSGPLGPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPMRL 4ovh A 2.25 BS01 2VE A 1 R152 Y154 G174 H175 R176 L177 V247 V360 M362 R150 Y152 G172 H173 R174 L175 V245 V358 M360 0003677,0003887,0006260,0008408,0009360 remove_due_to_license_issue 25970224 405 MKFTVEREHLLKPLQQVSGPLGGRLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4ovz A 2.5 BS01 P85 A 1 G164 D165 P249 Y269 Q270 Y274 T302 G156 D157 P241 Y261 Q262 Y266 T294 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0006508,0008234 ic50=0.49uM remove_due_to_license_issue IC50=490nM P0C6U8 24568342 902 FTTVDNTNLHTQLVDMSMTYGQQFGPTYLDGADVTKIKPHVNHEGKTFFVLPSDDTLRSEAFEYYHTLDESFLGRYMSALNHTKKWKFPQVGGLTSIKWADNNCYLSSVLLALQQLEVKFNAPALQEAYYRARAGDAANFCALILAYSNKTVGELGDVRETMTHLLQHANLESAKRVLNVVCKHCGQKTTTLTGVEAVMYMGTLSYDNLKTGVSIPCVCGRDATQYLVQQESSFVMMSAPPAEYKLQQGTFLCANEYTGNYQCGHYTHITAKETLYRIDGAHLTKMSEYKGPVTDVFYKETSYTT 4ovz A 2.5 BS02 P85 B 1 M209 Y269 M201 Y261 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0006508,0008234 ic50=0.49uM remove_due_to_license_issue IC50=490nM P0C6U8 24568342 902 FTTVDNTNLHTQLVDMSMTYGQQFGPTYLDGADVTKIKPHVNHEGKTFFVLPSDDTLRSEAFEYYHTLDESFLGRYMSALNHTKKWKFPQVGGLTSIKWADNNCYLSSVLLALQQLEVKFNAPALQEAYYRARAGDAANFCALILAYSNKTVGELGDVRETMTHLLQHANLESAKRVLNVVCKHCGQKTTTLTGVEAVMYMGTLSYDNLKTGVSIPCVCGRDATQYLVQQESSFVMMSAPPAEYKLQQGTFLCANEYTGNYQCGHYTHITAKETLYRIDGAHLTKMSEYKGPVTDVFYKETSYTT 4ow0 A 2.1 BS01 S88 A 1 L163 G164 D165 P249 Y265 Y269 Q270 Y274 L160 G161 D162 P246 Y262 Y266 Q267 Y271 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0006508,0008234 ic50=0.15uM remove_due_to_license_issue IC50=150nM P0C6U8 24568342 902 KTIKVFTTVDNTNLHTQLVDMSMTYGQQFGPTYLDGADVTKIKPHVNHEGKTFFVLPSDDTLRSEAFEYYHTLDESFLGRYMSALNHTKKWKFPQVGGLTSIKWADNNCYLSSVLLALQQLEVKFNAPALQEAYYRARAGDAANFCALILAYSNKTVGELGDVRETMTHLLQHANLESAKRVLNVVCKHCGQKTTTLTGVEAVMYMGTLSYDNLKTGVSIPCVCGRDATQYLVQQESSFVMMSAPPAEYKLQQGTFLCANEYTGNYQCGHYTHITAKETLYRIDGAHLTKMSEYKGPVTDVFYKETSYTTTI 4ow0 A 2.1 BS02 S88 B 1 P248 Y269 P245 Y266 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0006508,0008234 ic50=0.15uM remove_due_to_license_issue IC50=150nM P0C6U8 24568342 902 KTIKVFTTVDNTNLHTQLVDMSMTYGQQFGPTYLDGADVTKIKPHVNHEGKTFFVLPSDDTLRSEAFEYYHTLDESFLGRYMSALNHTKKWKFPQVGGLTSIKWADNNCYLSSVLLALQQLEVKFNAPALQEAYYRARAGDAANFCALILAYSNKTVGELGDVRETMTHLLQHANLESAKRVLNVVCKHCGQKTTTLTGVEAVMYMGTLSYDNLKTGVSIPCVCGRDATQYLVQQESSFVMMSAPPAEYKLQQGTFLCANEYTGNYQCGHYTHITAKETLYRIDGAHLTKMSEYKGPVTDVFYKETSYTTTI 4owm A 1.99 BS04 3F0 A 1 P180 H183 Y186 R187 A190 R194 P156 H159 Y162 R163 A166 R170 V106 V82 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 24712732 404 PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4own A 2.11 BS04 5RG A 1 V106 G107 H136 G137 N138 G206 V83 G84 H113 G114 N115 G180 V106 V83 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 24712732 404 VPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRALSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4own A 2.11 BS05 5RG A 2 N138 A179 P180 H183 Y186 R187 A190 N115 A153 P154 H157 Y160 R161 A164 V106 V83 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 24712732 405 VPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRALSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4owo A 1.99 BS04 6F0 A 1 N138 A179 P180 H183 Y186 A190 N116 A157 P158 H161 Y164 A168 V106 V84 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 24712732 404 SVPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4owo A 1.99 BS05 6F0 A 2 V106 G107 T108 H136 N138 R193 G206 V84 G85 T86 H114 N116 R171 G184 V106 V84 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 remove_due_to_license_issue P9WFX5 24712732 405 SVPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI 4owv A 1.9 BS01 BE2 A 1 N138 H183 Y186 R187 A190 N111 H154 Y157 R158 A161 V106 V84 2.4.2.18 0000162,0000287,0004048,0005576,0005829,0005886,0016757,0016763,0046872 Ki=45uM remove_due_to_license_issue P9WFX5 24712732 401 SVPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGTVNLSTMAAIVVAAAGVPVVKHGNRASLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQILE 4owx B 2.3 BS01 dna L 0 G13 K15 T32 K33 W55 D56 Y74 F78 Y85 T86 R88 G9 K11 T28 K29 W51 D52 Y70 F74 Y81 T82 R84 ? 0000724,0000781,0003677,0003697,0005515,0005634,0005654,0005829,0006281,0006974,0010212,0035861,0044818,0061730,0070182,0070200,0070876,0098505,1904355 remove_due_to_license_issue Q9BQ15 24630995 1 ~ 9 TFVKDIKPGLKNLNLIFIVLETGRVTKTKDGHEVRTCKVADKTGSINISVWDDVGNLIQPGDIIRLTKGYASVFKGCLTLYTGRGGDLQKIGEFCMVYSEVPNFSEP 4oya A 2.03 BS01 1VE A 1 F45 K95 A97 D99 L102 L166 V167 R176 F296 F336 M337 F338 S343 F45 K95 A97 D99 L102 L166 V167 R176 F296 F336 M337 F338 S343 4.6.1.1 0009190,0035556 ic50=0.36uM remove_due_to_license_issue Q96PN6 24616449 501 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oyb A 1.7 BS01 1VJ A 1 F45 K95 A97 L102 L166 V167 F336 M337 F338 F45 K95 A97 L102 L166 V167 F336 M337 F338 4.6.1.1 0009190,0035556 ic50=1.6uM remove_due_to_license_issue Q96PN6 24616449 502 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oyi A 1.7 BS01 1VK A 1 F45 K95 A97 L102 L166 V167 F336 M337 F338 F45 K95 A97 L102 L166 V167 F336 M337 F338 4.6.1.1 0009190,0035556 ic50=19uM remove_due_to_license_issue Q96PN6 24616449 501 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oym A 1.7 BS01 1ZC A 1 F45 K95 A97 L102 L166 V167 F336 M337 F338 F45 K95 A97 L102 L166 V167 F336 M337 F338 4.6.1.1 0009190,0035556 ic50=11uM remove_due_to_license_issue Q96PN6 24616449 501 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oyo A 1.75 BS01 1WC A 1 D47 D99 R176 F338 D47 D99 R176 F338 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24616449 501 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oyo A 1.75 BS02 1WC A 2 F45 K95 L102 L166 V167 F336 M337 F338 F45 K95 L102 L166 V167 F336 M337 F338 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24616449 502 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oyo A 1.75 BS03 1WC A 3 T52 G98 V411 A415 T52 G98 V411 A415 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24616449 503 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oyp A 2.28 BS01 BZ2 A 1 F45 K95 A97 L102 R176 F336 F45 K95 A97 L102 R176 F336 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24616449 502 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oys A 2.9 BS01 1TT A 1 F612 P618 I634 Y670 M682 Q683 F684 I685 L750 I760 F292 P298 I314 Y350 M362 Q363 F364 I365 L430 I440 2.7.1.137 0016301,0046854 remove_due_to_license_issue Q8NEB9 25326666 905 LKPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEPINSAEIDSSQIITSPLPNLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHALFAA 4oyt A 2.4 BS02 FON A 1 L124 G127 G128 H129 L130 T183 L124 G127 G128 H129 L130 T183 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25478836 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4oyt A 2.4 BS04 FON B 1 Y63 Y64 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25478836 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4oyt B 2.4 BS02 FON A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25478836 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4oyt B 2.4 BS04 FON B 1 L124 G127 G128 H129 L130 T183 L124 G127 G128 H129 L130 T183 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25478836 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4oz1 A 1.74 BS01 LYS A 1 H451 A480 H40 A69 ? 0003676,0003723,0005634,0006397 remove_due_to_license_issue Q14498 24795046 603 VQPLATQCFQLSNMFNPQTEEEVGWDTEIKDDVIEECNKHGGVIHIYVDKNSAQGNVYVKCPSIAAAIAAVNALHGRWFAGKMITAAYVPLPTYHNLFPDSMTATQLLVPS 4oz2 A 2.1 BS01 1Z6 A 1 A97 G98 F336 L345 V406 V411 A415 A97 G98 F336 L345 V406 V411 A415 4.6.1.1 0009190,0035556 remove_due_to_license_issue Q96PN6 24616449 501 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4oz3 A 1.7 BS01 1Z8 A 1 F45 K95 L102 L166 V167 V172 R176 F336 M337 F45 K95 L102 L166 V167 V172 R176 F336 M337 4.6.1.1 0009190,0035556 ic50=28uM remove_due_to_license_issue Q96PN6 24616449 501 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 4ozj A 1.45 BS01 ADP A 1 I18 G46 R47 G48 K97 G98 G100 K101 I13 G41 R42 G43 K78 G79 G81 K82 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue B8ZYW1 24946894 201 LPNDGGIKLVMAIIRPDKLADVKTALAEVGAPSLTVTNVSGRGSVDLHQKVKVECVVADTPAEDVADAIADAAHTGEKGDGKIFILPVENAIQVRTGKTGRDAV 4ozl A 1.4942 BS01 AMP A 1 I18 G46 R47 G98 G100 K101 I14 G42 R43 G79 G81 K82 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue B8ZYW1 24946894 201 DLPNDGGIKLVMAIIRPDKLADVKTALAEVGAPSLTVTNVSGRGSDLHQKVKVECVVADTPAEDVADAIADAAHTGEKGDGKIFILPVENAIQVRTGKTGRDAV 4ozn A 2.6 BS01 ATP A 1 I18 G46 R47 G48 G98 G100 K101 I14 G42 R43 G44 G91 G93 K94 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue B8ZYW1 24946894 201 DLPNDGGIKLVMAIIRPDKLADVKTALAEVGAPSLTVTNVSGRGSQKSQWRGEEYTVDLHQKVKVECVVADTPAEDVADAIADAAHTGEKGDGKIFILPVENAIQVRTGKTGRDAV 4ozn A 2.6 BS02 ATP C 1 S38 L39 T40 V75 R114 S34 L35 T36 V68 R107 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue B8ZYW1 24946894 201 DLPNDGGIKLVMAIIRPDKLADVKTALAEVGAPSLTVTNVSGRGSQKSQWRGEEYTVDLHQKVKVECVVADTPAEDVADAIADAAHTGEKGDGKIFILPVENAIQVRTGKTGRDAV 4ozn B 2.6 BS01 ATP A 1 S38 L39 T40 V75 R114 S34 L35 T36 V56 R95 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue B8ZYW1 24946894 201 DLPNDGGIKLVMAIIRPDKLADVKTALAEVGAPSLTVTNVSGRGSDLHQKVKVECVVADTPAEDVADAIADAAHTGEKGDGKIFILPVENAIQVRTGKTGRDAV 4ozn B 2.6 BS02 ATP B 1 I18 G46 R47 G48 K97 G98 G100 K101 I14 G42 R43 G44 K78 G79 G81 K82 ? 0005524,0005737,0005829,0006808,0030234 remove_due_to_license_issue B8ZYW1 24946894 201 DLPNDGGIKLVMAIIRPDKLADVKTALAEVGAPSLTVTNVSGRGSDLHQKVKVECVVADTPAEDVADAIADAAHTGEKGDGKIFILPVENAIQVRTGKTGRDAV 4ozo A 2.6 BS01 OTN A 1 D188 G189 A190 T219 W230 E234 E254 D277 D165 G166 A167 T196 W207 E211 E231 D254 3.2.1.111 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A5P6 24527659 503 SLAPCGLVPSARQLEWYNREMIAFFHFGINTFEEYVNEGDGKASTAIFNPTALDCRQWMQTLKAAGIPAAILTAKHADGFCLWPSKYTDYSVKNAAWKNGKGDVVREFVDACEEYGLKAGIYLGPHDRHEHLSPLYTTERYKEYYAHQLGELMSDYGKIWETWWDGAGADELTTPVYRHWYKIVREKQPDCVIFGTKNSYPFADVRWMGNEAGEAGDPCWATTDSVAIRDEAQYYKGLNEGMLDGDAYIPAETDVSIRPSWFYHAEEDSRVKSVRELWDIYCTSVGRNSVLLLNFPPDRRGLIHSTDSLHAALLKQGIDETFSTNLLRGAKVKATNVRGAKYSPEKMLDNEKNTYFAGKDGEVKADIIFTLPKTIEFDCLMIEEVIELGHRTTKWSVEYTVDGKNWITIPEATDKQAIGHKWIVRLAPVKAKQVRLRIQDGKACPAIHTFGVYKQSPVF 4p00 A 3.2 BS11 C2E A 1 R579 R580 R584 D609 S613 G614 V615 R616 R658 G670 I672 R567 R568 R572 D597 S601 G602 V603 R604 R646 G658 I660 2.4.1.12 0000166,0005515,0005886,0006011,0012505,0016020,0016757,0016758,0016759,0016760,0030244,0035438 remove_due_to_license_issue Q3J125 24704788 919 VVPVLLFLLWVALLVPFGLLAAAPVAPSAQGLIALSAVVLVALLKPFADKMVPRFLLLSAASMLVMRYWFWRLFETLPPPALDASFLFALLLFAVETFSISIFFLNGFLSADPTDRPFPRPLQPEELPTVDILVPSYNEPADMLSVTLAAAKNMIYPARLRTVVLCDDGGTDQRCMSPDPELAQKAQERRRELQQLCRELGVVYSTRERNEHAKAGNMSAALERLKGELVVVFDADHVPSRDFLARTVGYFVEDPDLFLVQTPHFFINPDPIQRNLALGDRCPPENEMFYGKIHRGLDRWGGAFFCGSAAVLRRRALDEAGGFAGETITEDAETALEIHSRGWKSLYIDRAMIAGLQPETFASFIQQRGRWATGMMQMLLLKNPLFRRGLGIAQRLCYLNSMSFWFFPLVRMMFLVAPLIYLFFGIEIFVATFEEVLAYMPGYLAVSFLVQNALFARQRWPLVSEVYEVAQAPYLARAIVTTLLRPRSARFAVTAKDETLSENYISPIYRPLLFTFLLCLSGVLATLVRWVAFPGDRSVLLVVGGWAVLNVLLVGFALRAVAEKQQRRAAPRVQMEVPAEAQIPAFGNRSLTATVLDASTSGVRLLVRLPGVGDPHPALEAGGLIQFQPKFPDAPQLERMVRGRIRSARREGGTVMVGVIFEAGQPIAVRETVAYLIFGESAHWRTMREATMRPIGLLHGMARILWMAAASLPKTARDFMDEPARRRR 4p00 A 3.2 BS12 C2E A 2 Q578 R579 R580 R584 R616 Q566 R567 R568 R572 R604 2.4.1.12 0000166,0005515,0005886,0006011,0012505,0016020,0016757,0016758,0016759,0016760,0030244,0035438 remove_due_to_license_issue Q3J125 24704788 920 VVPVLLFLLWVALLVPFGLLAAAPVAPSAQGLIALSAVVLVALLKPFADKMVPRFLLLSAASMLVMRYWFWRLFETLPPPALDASFLFALLLFAVETFSISIFFLNGFLSADPTDRPFPRPLQPEELPTVDILVPSYNEPADMLSVTLAAAKNMIYPARLRTVVLCDDGGTDQRCMSPDPELAQKAQERRRELQQLCRELGVVYSTRERNEHAKAGNMSAALERLKGELVVVFDADHVPSRDFLARTVGYFVEDPDLFLVQTPHFFINPDPIQRNLALGDRCPPENEMFYGKIHRGLDRWGGAFFCGSAAVLRRRALDEAGGFAGETITEDAETALEIHSRGWKSLYIDRAMIAGLQPETFASFIQQRGRWATGMMQMLLLKNPLFRRGLGIAQRLCYLNSMSFWFFPLVRMMFLVAPLIYLFFGIEIFVATFEEVLAYMPGYLAVSFLVQNALFARQRWPLVSEVYEVAQAPYLARAIVTTLLRPRSARFAVTAKDETLSENYISPIYRPLLFTFLLCLSGVLATLVRWVAFPGDRSVLLVVGGWAVLNVLLVGFALRAVAEKQQRRAAPRVQMEVPAEAQIPAFGNRSLTATVLDASTSGVRLLVRLPGVGDPHPALEAGGLIQFQPKFPDAPQLERMVRGRIRSARREGGTVMVGVIFEAGQPIAVRETVAYLIFGESAHWRTMREATMRPIGLLHGMARILWMAAASLPKTARDFMDEPARRRR 4p02 A 2.65 BS13 C2E A 1 R579 R580 A581 R584 D609 S613 G614 V615 R616 R658 G670 V671 I672 R567 R568 A569 R572 D597 S601 G602 V603 R604 R646 G658 V659 I660 2.4.1.12 0000166,0005515,0005886,0006011,0012505,0016020,0016757,0016758,0016759,0016760,0030244,0035438 remove_due_to_license_issue Q3J125 24704788 918 VVPVLLFLLWVALLVPFGLLAAAPVAPSAQGLIALSAVVLVALLKPFADKMVPRFLLLSAASMLVMRYWFWRLFETLPPPALDASFLFALLLFAVETFSISIFFLNGFLSADPTDRPFPRPLQPEELPTVDILVPSYNEPADMLSVTLAAAKNMIYPARLRTVVLCDDGGTDQRCMSPDPELAQKAQERRRELQQLCRELGVVYSTRERNEHAKAGNMSAALERLKGELVVVFDADHVPSRDFLARTVGYFVEDPDLFLVQTPHFFINPDPIQRNLALGDRCPPENEMFYGKIHRGLDRWGGAFFCGSAAVLRRRALDEAGGFAGETITEDAETALEIHSRGWKSLYIDRAMIAGLQPETFASFIQQRGRWATGMMQMLLLKNPLFRRGLGIAQRLCYLNSMSFWFFPLVRMMFLVAPLIYLFFGIEIFVATFEEVLAYMPGYLAVSFLVQNALFARQRWPLVSEVYEVAQAPYLARAIVTTLLRPRSARFAVTAKDETLSENYISPIYRPLLFTFLLCLSGVLATLVRWVAFPGDRSVLLVVGGWAVLNVLLVGFALRAVAEKQQRRAAPRVQMEVPAEAQIPAFGNRSLTATVLDASTSGVRLLVRLPGVGDPHPALEAGGLIQFQPKFPDAPQLERMVRGRIRSARREGGTVMVGVIFEAGQPIAVRETVAYLIFGESAHWRTMREATMRPIGLLHGMARILWMAAASLPKTARDFMDEPARRRR 4p02 A 2.65 BS14 C2E A 2 Q578 R579 R580 R584 R616 S659 Q566 R567 R568 R572 R604 S647 2.4.1.12 0000166,0005515,0005886,0006011,0012505,0016020,0016757,0016758,0016759,0016760,0030244,0035438 remove_due_to_license_issue Q3J125 24704788 919 VVPVLLFLLWVALLVPFGLLAAAPVAPSAQGLIALSAVVLVALLKPFADKMVPRFLLLSAASMLVMRYWFWRLFETLPPPALDASFLFALLLFAVETFSISIFFLNGFLSADPTDRPFPRPLQPEELPTVDILVPSYNEPADMLSVTLAAAKNMIYPARLRTVVLCDDGGTDQRCMSPDPELAQKAQERRRELQQLCRELGVVYSTRERNEHAKAGNMSAALERLKGELVVVFDADHVPSRDFLARTVGYFVEDPDLFLVQTPHFFINPDPIQRNLALGDRCPPENEMFYGKIHRGLDRWGGAFFCGSAAVLRRRALDEAGGFAGETITEDAETALEIHSRGWKSLYIDRAMIAGLQPETFASFIQQRGRWATGMMQMLLLKNPLFRRGLGIAQRLCYLNSMSFWFFPLVRMMFLVAPLIYLFFGIEIFVATFEEVLAYMPGYLAVSFLVQNALFARQRWPLVSEVYEVAQAPYLARAIVTTLLRPRSARFAVTAKDETLSENYISPIYRPLLFTFLLCLSGVLATLVRWVAFPGDRSVLLVVGGWAVLNVLLVGFALRAVAEKQQRRAAPRVQMEVPAEAQIPAFGNRSLTATVLDASTSGVRLLVRLPGVGDPHPALEAGGLIQFQPKFPDAPQLERMVRGRIRSARREGGTVMVGVIFEAGQPIAVRETVAYLIFGESAHWRTMREATMRPIGLLHGMARILWMAAASLPKTARDFMDEPARRRR 4p0n A 2.08 BS01 1IS A 1 I682 Y683 P702 M703 E711 V712 G715 Q716 F719 I230 Y231 P250 M251 E259 V260 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 ic50=0.8nM remove_due_to_license_issue IC50=0.800000nM Q9Y233 24944747 801 TLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4p0v A 2.4 BS02 1WO A 1 G56 K57 Y58 R60 E93 Q96 R113 F239 K257 G49 K50 Y51 R53 E86 Q89 R106 F232 K250 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K193 F232 D236 D237 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 24927548 402 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4p0w A 2.406 BS01 1XH A 1 G56 K57 Y58 N59 R60 G61 E93 Q96 R113 F239 G49 K50 Y51 N52 R53 G54 E86 Q89 R106 F232 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K193 F232 D236 D237 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 24927548 500 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4p0x A 2.5 BS01 1WO A 1 G56 K57 Y58 N59 R60 R113 F239 G43 K44 Y45 N46 R47 R98 F221 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F83 D88 D92 R97 D159 K182 F221 D225 D226 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 24927548 1001 AQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRAPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 4p0x A 2.5 BS02 1WO A 2 N59 K347 N46 K328 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F83 D88 D92 R97 D159 K182 F221 D225 D226 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 24927548 1002 AQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRAPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 4p10 A 2.0 BS01 2B8 A 1 H181 E184 N256 R257 H310 S311 Y312 S321 L362 D370 E385 H157 E160 N232 R233 H286 S287 Y288 S297 L338 D346 E361 H181 E184 R239 H310 E385 H157 E160 R215 H286 E361 3.4.17.20 0003331,0004180,0004181,0005576,0005615,0006508,0007596,0008237,0008270,0009410,0010757,0030163,0042730,0046872,0051918,0070062,0071333,0097421,2000346 remove_due_to_license_issue IC50=8.0nM Q96IY4 24588961 501 SGQVLAALPRTSRQVQVLQNLTTTYEIVLWQPVTADLIVKKKQVHFFVNASDVDNVKAHLNVSGIPCSVLLADVEDLIQQQISNDTVSPRASASYYEQYHSLNEIYSWIEFITERHPDMLTKIHIGSSFEKYPLYVLKVSGKEQAAKNAIWIDCGIHAREWISPAFCLWFIGHITQFYGIIGQYTNLLRLVDFYVMPVVNVDGYDYSWKKNRMWRKNRSFYANNHCIGTDLNRNFASKHWCEEGASSSSCSETYCGLYPESEPEVKAVASFLRRNINQIKAYISMHSYSQHIVFPYSYTRSKSKDHEELSLVASEAVRAIEKTSKNTRYTYGQGSETLYLAPGGGDDWIYDLGIKYSFTIELRDTGTYGFLLPERYIKPTCREAFAAVSKIAWHVIRNVLEP 4p1r A 2.243 BS02 2KR A 1 Y683 P702 M703 K708 E711 G715 Q716 F719 Y242 P261 M262 K267 E270 G274 Q275 F278 3.1.4.17 0004114,0007165,0008081 ic50=4.1nM remove_due_to_license_issue IC50=4.1nM Q9Y233 24944747 1020 TSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4p1u A 2.52 BS01 21G A 1 F23 H57 E61 F63 K76 F104 Q106 M131 F3 H37 E41 F43 K56 F84 Q86 M106 ? remove_due_to_license_issue P31345 25019388 4000 SSFSFGGFTFKRTSGSSIKREEEVLTGNLQTLKIRVHEGYEEFTMVGKRATAILRKATRRLVQLIVSGKDEQSIAEAIIVAMVFSQEDCMIKAVRGDLNFVNLNPMHQLLRHFQKDAKVLFQNWGIEHIDNVMGMVGVLPDMTPSTEMSMRGIRVSKM 4p2t A 2.15 BS01 24Q A 1 F76 L79 L110 F189 P192 L193 L196 F74 L77 L108 F185 P188 L189 L192 H46 S114 S116 H134 R142 R143 H44 S112 S114 H130 R138 R139 3.4.21.97 0004252,0006508 ic50=3.7uM remove_due_to_license_issue Q2HRB6 24977643 201 QGLYVGGFVDVVSCPKLEQELYLDPDQVTDYLPVTEPLPITIEHLPETEVGWTLGLFQVSHGIFCTGAITSPAFLELASRLADTSHVARAPVKNLPKEPLLEILHTWLPGLSLSSIHPRELTPSGPVFQHVSLCALGRRRGTVAVYGHDAEWVVSRFSSVSKSERAHILQHVSSCRLEDLSTPNFVSPLETL 4p3h A 1.45 BS01 25G A 1 I44 F76 L79 L110 F189 P192 I41 F73 L76 L107 F186 P189 H46 S114 S116 H134 R142 R143 H43 S111 S113 H131 R139 R140 3.4.21.97 0004252,0006508 ic50=1uM remove_due_to_license_issue Q2HRB6 24977643 201 GLYVGGFVDVVSCPKLEQELYLDPDQVTDYLPVTEPLPITIEHLPETEVGWTLGLFQVSHGIFCTGAITSPAFLELASRLADTSHVARAPVKNLPKEPLLEILHTWLPGLSLSSIHPRELSQTPSGPVFQHVSLCALGRRRGTVAVYGHDAEWVVSRFSSVSKSERAHILQHVSSCRLEDLSTPNFVSPL 4p44 A 1.75 BS04 2F7 A 1 K207 V208 R210 N257 D387 E424 E425 L428 G518 N519 R534 G548 Y549 Y552 H553 K699 Y700 K153 V154 R156 N203 D333 E370 E371 L374 G464 N465 R480 G491 Y492 Y495 H496 K640 Y641 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=16nM remove_due_to_license_issue Q04609 26460595 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p45 A 1.87 BS05 2F9 A 1 R210 D387 E424 E425 L428 G518 N519 R534 G548 Y552 H553 N698 K699 Y700 A701 R156 D333 E370 E371 L374 G464 N465 R480 G490 Y494 H495 N638 K639 Y640 A641 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=16nM remove_due_to_license_issue Q04609 26460595 822 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4b A 1.93 BS04 2G2 A 1 R210 Y234 N257 D387 E424 E425 L428 G518 N519 R534 R536 S547 Y552 H553 K699 Y700 R156 Y180 N203 D333 E370 E371 L374 G464 N465 R480 R482 S493 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=14nM remove_due_to_license_issue IC50=14nM Q04609 26460595 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4d A 1.65 BS04 2GR A 1 R210 N257 D387 E424 E425 L428 G518 R534 Y552 H553 K699 Y700 R156 N203 D333 E370 E371 L374 G464 R480 Y491 H492 K636 Y637 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=1800nM remove_due_to_license_issue Q04609 26460595 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4e A 1.67 BS05 2G4 A 1 R210 D387 E424 E425 L428 E457 G518 K545 G548 Y549 Y552 H553 K699 Y700 R156 D333 E370 E371 L374 E403 G464 K491 G494 Y495 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=180nM remove_due_to_license_issue Q04609 26460595 822 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4f A 1.86 BS04 2GB A 1 R210 D387 E424 E425 L428 E457 R463 G518 N544 K545 G548 Y549 Y552 H553 K699 Y700 R156 D333 E370 E371 L374 E403 R409 G464 N490 K491 G494 Y495 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=168nM remove_due_to_license_issue Q04609 26460595 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4i A 1.87 BS04 2G5 A 1 R210 D387 E424 E425 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 D333 E370 E371 L374 G464 N465 R480 R482 Y496 H497 K641 Y642 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=35nM remove_due_to_license_issue Q04609 26460595 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4j A 1.66 BS04 2H9 A 1 R210 N257 D387 E424 E425 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 D333 E370 E371 L374 G464 N465 R480 R482 Y490 H491 K635 Y636 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=700nM remove_due_to_license_issue Q04609 26460595 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4p4t A 2.3 BS01 GDP A 1 S80 S81 G82 K83 S84 S85 K248 D250 K279 C280 R281 G282 Q283 S37 S38 G39 K40 S41 S42 K197 D199 K228 C229 R230 G231 Q232 ? 0003924,0005525 remove_due_to_license_issue P20591 25295396 701 QYEEKVRPCIDLIDSLRALGVEQDLALPAIAVIGDQSSGKSSVLEALSGVALPRRCPLVLKLKKLVNEDKWRGKVSYQDYEIEISDASEVEKEINKAQNAIAGEGISHELITLEISSRDVPDLTLIDLPGITRVAVGNQPADIGYKIKTLIKKYIQRQETISLVVVPSNVDIATTEALSMAQEVDPEGDRTIGILTKPDLVDKGTEDKVVDVVRNLVFHLKKGYMIVKCRGQQEIQDQLSLSEALQREKIFFENHPYFRDLLEEGKATVPSLAEKLTSELITHISKSLPLLENQIKETHQRITEELQKYGVKRKFLKERLARLTQARRRLAQFPG 4p58 A 2.06 BS01 2F6 A 1 Y111 M132 E133 I134 A161 S162 H185 W186 Y58 M79 E80 I81 A108 S109 H132 W133 D184 K187 D212 N213 E242 D131 K134 D159 N160 E189 2.1.1.6 0000287,0006584,0008171,0016206 Kd=63uM remove_due_to_license_issue Ki=63000nM O88587 24847974 301 TKEQRILRYVQQNAKPGDPQSVLEAIDTYCSEGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDYAAITQQMLNFAGLQDKVTILIGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 4p5d A 2.11 BS01 N6P A 1 G16 S17 I18 R19 H45 E57 I65 N69 S87 G89 E93 G8 S9 I10 R11 H37 E49 I57 N61 S79 G81 E85 3.2.2.- 0009159,0070694 Ki=1.5uM remove_due_to_license_issue Ki=1500nM O35820 25108359 201 RRSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADAELEPLGEEAAGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYLV 4p5d C 2.11 BS01 N6P C 1 G16 S17 I18 R19 G20 H45 E57 A58 I65 N69 S87 G89 E93 G7 S8 I9 R10 G11 H36 E48 A49 I56 N60 S78 G80 E84 3.2.2.- 0009159,0070694 Ki=1.5uM remove_due_to_license_issue Ki=1500nM O35820 25108359 201 RSVYFCGSIRGGREDQALYARIVSRLRRYGKVLTEHVADAELEPLGEEAAGGDQFIHEQNLNWLQQADVVVAEVTQPSLGVGYELGRAVALGKPILCLFRPQSGRVLSAMIRGAADGSRFQVWDYAEGEVETMLDRYFEAYL 4p5e B 1.35 BS01 N6P B 1 C26 G27 S28 I29 R30 I76 D80 S98 G100 E104 C7 G8 S9 I10 R11 I48 D52 S70 G72 E76 3.2.2.- 0009159,0070694 Ki=2.8uM remove_due_to_license_issue Ki=2800nM O43598 25108359 201 RPALYFCGSIRGGREDRTLYERIVSRLRRFGTVLTEHVAAAELGDRLIHEQDLEWLQQADVVVAEVTQPSLGVGYELGRAVAFNKRILCLFRPQSGRVLSAMIRGAADGSRFQVWDYEEGEVEALLDRYFEADPLE 4p5z A 2.002 BS01 Q7M A 1 V635 A651 K653 E670 I673 M674 F677 I683 M702 Y742 L753 S763 D764 F765 V27 A43 K45 E62 I65 M66 F69 I75 M94 Y134 L145 S155 D156 F157 D746 A748 R750 N751 D764 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 Kd=39.3nM remove_due_to_license_issue Kd=3.9nM P29320 25076195 1001 VHEFAKELDATNISIDKVVGAGEFGEVCSGRLKLPSKKEISVAIKTLKVGYTEKQRRDFLGEASIMGQFDHPNIIRLEGVVTKSKPVMIVTEYMENGSLDSFLRKHDAQFTVIQLVGMLRGIASGMKYLSDMGYVHRDLAARNILINSNLVCKVSDFPIRWTSPEAIAYRKFTSASDVWSYGIVLWEVMSYGERPYWEMSNQDVIKAVDEGYRLPPPMDCPAALYQLMLDCWQKDRNNRPKFEQIVSILDKLIRNPGSLKIITNLLL 4p6c A 1.86 BS01 RES A 1 R38 E39 C68 T94 F96 R151 G153 H154 T155 E175 R38 E39 C68 T94 F96 R151 G153 H154 T155 E175 E39 D43 C68 N92 F96 E101 H137 H154 E175 E39 D43 C68 N92 F96 E101 H137 H154 E175 4.1.99.12 0000287,0003824,0005829,0008686,0009231,0016829,0030145,0046872 Ki=100uM remove_due_to_license_issue Q9KKP2 25792735 500 MNQSSLLAEFGDPITRVENALQALREGRGVLLLDDEDRENEGDIIYAVESLTTAQMALMIRECSGIVCLCLTEAQADRLALPPMVVNNNSANQTAFTVSIEAKHGVTTGVSAQDRVTTIKTAANPQAKPEDLARPGHVFPLRARAGGVLARRGHTEGTVDLMQMAGLQPAGVLCELTNPDGSMAKTPEIIEFGKLHNMPVLTIEDMVQYRIQFDLKL 4p6c B 1.86 BS01 RES B 1 R38 E39 C68 T94 F96 R151 G153 H154 T155 E175 R34 E35 C64 T90 F92 R147 G149 H150 T151 E171 E39 D43 C68 N92 F96 E101 H137 H154 E175 E35 D39 C64 N88 F92 E97 H133 H150 E171 4.1.99.12 0000287,0003824,0005829,0008686,0009231,0016829,0030145,0046872 Ki=100uM remove_due_to_license_issue Q9KKP2 25792735 500 SLLAEFGDPITRVENALQALREGRGVLLLDDEDRENEGDIIYAVESLTTAQMALMIRECSGIVCLCLTEAQADRLALPPMVVNNNSANQTAFTVSIEAKHGVTTGVSAQDRVTTIKTAANPQAKPEDLARPGHVFPLRARAGGVLARRGHTEGTVDLMQMAGLQPAGVLCELTNPDGSMAKTPEIIEFGKLHNMPVLTIEDMVQYRIQFDLKL 4p6e A 1.8 BS01 2FC A 1 G62 G68 G69 F70 M71 N163 G165 F211 G63 G69 G70 F71 M72 N164 G166 F212 Q19 C25 H164 N184 Q20 C26 H165 N185 3.4.22.27 0006508,0008234 ic50=1290nM remove_due_to_license_issue IC50=1290nM P25774 25313327 302 ILPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEIE 4p6e A 1.8 BS02 2FC B 1 F70 E115 F71 E116 Q19 C25 H164 N184 Q20 C26 H165 N185 3.4.22.27 0006508,0008234 ic50=1290nM remove_due_to_license_issue IC50=1290nM P25774 25313327 301 ILPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEIE 4p6g A 1.58 BS01 2FZ A 1 C25 K64 G68 G69 F70 M71 V162 N163 G165 F211 C26 K65 G69 G70 F71 M72 V163 N164 G166 F212 Q19 C25 H164 N184 Q20 C26 H165 N185 3.4.22.27 0006508,0008234 ic50=7.7nM remove_due_to_license_issue IC50=7.7nM P25774 25313327 301 ILPDSVDWREKGCVTEVKYQGSCGACWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEIE 4p6w A 1.951 BS02 MOF A 1 M560 L563 N564 G567 Q570 M601 M604 F623 M639 C643 C736 F749 M35 L38 N39 G42 Q45 M76 M79 F98 M114 C118 C211 F224 ? Ki=0.7nM remove_due_to_license_issue Ki=0.700000nM P04150 24763108 801 PQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMALMAFALGWRSYRQSSANLLYFAPDLIINEQRMTLPCMYDQCKHMLYVSSELHRLQVSYEEYLCMKVLLLLSTIPKDGLKSQELFDEIRMTYIKELGAAIVAREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQK 4p6x A 2.5 BS02 HCY A 1 L563 N564 Q570 M604 F623 Y735 C736 T739 L38 N39 Q45 M79 F98 Y210 C211 T214 ? Ki=91nM remove_due_to_license_issue Ki=30nM P04150 24763108 900 PQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMALMAFALGWRSYRQSSANLLYFAPDLIINEQRMTLPCMYDQCKHMLYVSSELHRLQVSYEEYLCMKVLLLLSTIPKDGLKSQALFDAIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQK 4p72 C 2.62 BS01 2NL C 1 L64 E131 F169 F171 T172 G203 C204 A226 G228 L54 E121 F159 F161 T162 G179 C180 A202 G204 H76 H90 R116 Q129 T172 A226 H66 H80 R106 Q119 T162 A202 6.1.1.20 0000049,0000166,0000287,0004812,0004826,0005524,0005737,0006412,0006432,0043039,0046872 remove_due_to_license_issue Q9I0A3 24936059 301 ERIDVTLPGRGQLSGGLHPVTRTLERIEQCFSRIGYEVAEGPEVEDDYHNFEALNIPGHHPARAMHDTFYFNANMLLRTHTSPVQVRTMESQQPPIRIVCPGRVYRCDSDLTHSPMFHQVEGLLVDEGVSFADLKGTIEEFLRAFFEKQLEVRFRPSFFPFTEPSAEVDIQCGWLEVMGCGMVHPNVLRMSNIDPEKFQGFAFGMGAERLAMLRYGVNDLRLFFDNDLRFLGQFR 4p73 C 3.03 BS01 GAX C 1 L64 S92 Q95 M99 E131 F169 F171 G203 C204 A226 F227 G228 L56 S84 Q87 M91 E123 F161 F163 G183 C184 A206 F207 G208 H76 H90 R116 Q129 T172 A226 H68 H82 R108 Q121 T164 A206 6.1.1.20 0000049,0000166,0000287,0004812,0004826,0005524,0005737,0006412,0006432,0043039,0046872 remove_due_to_license_issue Q9I0A3 24936059 301 AAERIDVTLPGRGQLSGGLHPVTRTLERIEQCFSRIGYEVAEGPEVEDDYHNFEALNIPGHHPARAMHDTFYFNANMLLRTHTSPVQVRTMESQQPPIRIVCPGRVYRCDSDLTHSPMFHQVEGLLVDEGVSFADLKGTIEEFLRAFFEKQLEVRFRPSFFPFTEPSAEVDIQCQTGWLEVMGCGMVHPNVLRMSNIDPEKFQGFAFGMGAERLAMLRYGVNDLRLFFDNDLRFLGQFR 4p74 C 2.7 BS01 2U9 C 1 L64 S92 Q95 Q129 E131 F169 F171 G203 C204 A226 F227 G228 G230 L54 S82 Q85 Q119 E121 F159 F161 G179 C180 A202 F203 G204 G206 H76 H90 R116 Q129 T172 A226 H66 H80 R106 Q119 T162 A202 6.1.1.20 0000049,0000166,0000287,0004812,0004826,0005524,0005737,0006412,0006432,0043039,0046872 remove_due_to_license_issue Q9I0A3 24936059 301 ERIDVTLPGRGQLSGGLHPVTRTLERIEQCFSRIGYEVAEGPEVEDDYHNFEALNIPGHHPARAMHDTFYFNANMLLRTHTSPVQVRTMESQQPPIRIVCPGRVYRCDSDLTHSPMFHQVEGLLVDEGVSFADLKGTIEEFLRAFFEKQLEVRFRPSFFPFTEPSAEVDIQCGWLEVMGCGMVHPNVLRMSNIDPEKFQGFAFGMGAERLAMLRYGVNDLRLFFDNDLRFLGQFR 4p75 C 2.96 BS01 2NM C 1 S92 Q95 E131 F171 G203 C204 A226 G228 S82 Q85 E121 F161 G179 C180 A202 G204 H76 H90 R116 Q129 T172 A226 H66 H80 R106 Q119 T162 A202 6.1.1.20 0000049,0000166,0000287,0004812,0004826,0005524,0005737,0006412,0006432,0043039,0046872 remove_due_to_license_issue Q9I0A3 24936059 301 ERIDVTLPGRGQLSGGLHPVTRTLERIEQCFSRIGYEVAEGPEVEDDYHNFEALNIPGHHPARAMHDTFYFNANMLLRTHTSPVQVRTMESQQPPIRIVCPGRVYRCDSDLTHSPMFHQVEGLLVDEGVSFADLKGTIEEFLRAFFEKQLEVRFRPSFFPFTEPSAEVDIQCGWLEVMGCGMVHPNVLRMSNIDPEKFQGFAFGMGAERLAMLRYGVNDLRLFFDNDLRFLGQFR 4p7e A 2.4 BS01 2HB A 1 L855 G856 G861 S862 V863 A880 M929 Y931 L932 G935 L983 D994 L13 G14 G19 S20 V21 A38 M83 Y85 L86 G89 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>10000nM O60674 25369270 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG 4p7m A 3.02 BS01 2OE A 1 P1 Y37 S64 N106 P1 Y37 S64 N96 5.3.2.1,5.3.3.12 0005125,0005576,0005615,0007165,0016853,0050178 remove_due_to_license_issue Q6Q3H7 25268646 201 PCCEVITNVNLPDDNVQSTLSQIENAISDVMGKPLGYIMSNYDYQKNLRFGGSNEAYCFVRITSSNNSALADQITKLLVSNLNVKSRRIYVEFRDNFAFSGSLF 4p7s A 2.87 BS01 2OK B 1 F50 E98 F99 R100 F50 E92 F93 R94 5.3.2.1,5.3.3.12 0005125,0005576,0005615,0007165,0016853,0050178 remove_due_to_license_issue Q6Q3H7 25268646 201 PCCEVITNVNLPDDNVQSTLSQIENAISDVMGKPLGYIMSNYDYQKNLRFGGSNEAYCFVRITSSNNSALADQITKLLVSNLNVKSRRIYVEFRDNFAFSGSLF 4p7s B 2.87 BS01 2OK B 1 P1 Y37 N106 F107 P1 Y35 N95 F96 5.3.2.1,5.3.3.12 0005125,0005576,0005615,0007165,0016853,0050178 remove_due_to_license_issue Q6Q3H7 25268646 201 PCCEVITNVNLPDDNVQSTLSQIENAISDVKPLGYIMSNYDYQKNLRFGGSNEAYCFVRITSINNSALADQITKLLVSNLNVKSRRIYVEFRDCNFAFGS 4p7s B 2.87 BS02 2OK C 1 F50 Y57 F48 Y55 5.3.2.1,5.3.3.12 0005125,0005576,0005615,0007165,0016853,0050178 remove_due_to_license_issue Q6Q3H7 25268646 201 PCCEVITNVNLPDDNVQSTLSQIENAISDVKPLGYIMSNYDYQKNLRFGGSNEAYCFVRITSINNSALADQITKLLVSNLNVKSRRIYVEFRDCNFAFGS 4p90 A 2.49 BS01 2K0 A 1 I276 V284 A297 K299 M344 Y346 L347 L396 D407 I27 V35 A42 K44 M79 Y81 L82 L131 D142 N389 K391 D393 N394 D407 T427 N124 K126 D128 N129 D142 T157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13153 601 DEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMEVAIKQMKELIINEILVMRENKNPNIVNYLDSYLELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQIKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLDMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 4pax A 2.8 BS01 NU1 A 1 H862 G863 Y896 F897 K903 S904 Y907 H201 G202 Y235 F236 K242 S243 Y246 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue P26446 9521710 1 KSKLAKPIQDLIKMIFDVESMKKAMVEFEIDLQKMPLGKLSKRQIQSAYSILNEVQQAVSDGGSESQILDLSNRFYTLIPHDFGMKKPPLLSNLEYIQAKVQMLDNLLDIEVAYSLLRGGNEDGDKDPIDINYEKLRTDIKVVDKDSEEAKIIKQYVKNTHAATHNAYDLKVVEIFRIEREGESQRYKPFKQLHNRQLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQADPIGLILLGEVALGNMYELKNASHITKLPKGKHSVKGLGKTAPDPTATTTLDGVEVPLGNGISTGINDTCLLYNEYIVYDVAQVNLKYLLKLKFNYKT 4pb1 A 2.803 BS01 RBV A 1 L259 N331 E332 F333 F366 L247 N319 E320 F321 F354 ? 0005337,0005886,0015293,0016020,0042802,1901642 remove_due_to_license_issue Q9KPL5 25082345 501 SLFMSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pb2 A 2.302 BS01 5UD A 1 Q154 E332 F366 S371 Q153 E320 F354 S359 ? 0005337,0005886,0015293,0016020,0042802,1901642 Kd=16uM remove_due_to_license_issue Q9KPL5 25082345 501 SLFMSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pce A 1.293 BS01 2N0 A 1 W81 V87 N140 I146 W40 V46 N99 I105 ? ic50=7uM remove_due_to_license_issue IC50=7000nM O60885 24767840 302 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4pci A 1.25 BS01 2NJ A 1 P82 L92 L94 N140 I146 P41 L51 L53 N99 I105 ? ic50=7.5uM remove_due_to_license_issue IC50=7500nM O60885 24767840 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 4pcs A 1.77 BS01 2M7 A 1 H66 E87 W88 H135 Y178 D229 W232 E288 W316 H32 E53 W54 H101 Y144 D195 W198 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A3I4 25427942 505 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAK 4pct A 2.1 BS01 H76 A 1 H66 E87 W88 H135 D229 E288 W316 H32 E53 W54 H101 D195 E254 W282 3.2.1.51 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A3I4 25427942 504 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAA 4pd5 A 2.906 BS01 GEO A 1 Q154 E332 F333 F366 I374 Q152 E319 F320 F353 I361 ? 0005337,0005886,0015293,0016020,0042802,1901642 remove_due_to_license_issue Q9KPL5 25082345 501 LFMSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pd6 A 2.08 BS01 URI A 1 Q154 E332 F366 S371 I374 Q150 E317 F351 S356 I359 ? 0005337,0005886,0015293,0016020,0042802,1901642 Kd=36uM remove_due_to_license_issue Q9KPL5 25082345 501 MSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pd7 A 2.909 BS01 ZE8 A 1 Q154 E332 F333 F366 I374 Q153 E320 F321 F354 I362 ? 0005337,0005886,0015293,0016020,0042802,1901642 remove_due_to_license_issue Q9KPL5 25082345 501 SLFMSLIGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pd8 A 2.75 BS01 P0C A 1 Q154 A185 L259 E332 F366 S371 I374 Q153 A184 L247 E320 F354 S359 I362 ? 0005337,0005886,0015293,0016020,0042802,1901642 remove_due_to_license_issue Q9KPL5 25082345 501 SLFMSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pd9 A 3.096 BS01 ADN A 1 Q154 N331 E332 F333 F366 S371 I374 Q153 N319 E320 F321 F354 S359 I362 ? 0005337,0005886,0015293,0016020,0042802,1901642 remove_due_to_license_issue Q9KPL5 25082345 501 SLFMSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pda A 2.608 BS01 CTN A 1 Q154 E332 F366 S371 I374 Q153 E320 F354 S359 I362 ? 0005337,0005886,0015293,0016020,0042802,1901642 remove_due_to_license_issue Q9KPL5 25082345 501 SLFMSCCGMAVLLGIAVLLSSNRKAINLRTVGGAFAIQFSLGAFILYVPWGQELLRGFSDAVSNVINYGNDGTSFLFGGLVSGKMFEVFGGGGFIFAFRVLPTLIFFSALISVLYYLGVMQWVIRILGGGLQKALGTSRAESMSAAANIFVGQTEAPLVVRPFVPKMTQSELFAVMCGGLASIAGGVLAGYASMGVKIEYLVAASFMAAPGGLLFAKLMMPETEKPQDKPANVIDAAAGGASAGLQLALNVGAMLIAFIGLIALINGMLGGIGGWFGMPELKLEMLLGWLFAPLAFLIGVPWNEATVAGEFIGLKTVANEFVAYSQFAPYLTEAAPVVLSEKTKAIISFALCGFANLSSIAILLGGLGSLAPKRRGDIARMGVKAVIAGTLSNLMAATIAGFFL 4pdb A 2.6 BS01 rna I 0 P29 S53 K54 Q80 R109 Y111 K113 A114 S130 T131 S132 K133 G134 G147 E149 P3 S27 K28 Q54 R83 Y85 K87 A88 S104 T105 S106 K107 G108 G121 E123 ? 0003735,0005737,0005840,0006412,0019843,1990904 remove_due_to_license_issue Q81VR6 25140011 1 ~ 38 TDPIADMLTRIRNANMVRHEKLEVPASKIKKEIAELLKREGFIRDVEYIEDNKQGILRIFLKYGANNERVITGLKRISKPGLRVYAKADEVPRVLNGLGIALVSTSKGVMTDKDARQLQTGGEVVAYVW 4pde A 2.8 BS01 GDP A 1 S240 F260 K262 R265 S207 F227 K229 R232 ? 0003824,0005515,0005737,0005829,0006777,0016783,0042803,0043546,0097163 remove_due_to_license_issue P32177 25649206 300 ITGVRQIELWRRDDLQHPRLDEVAEEVPVALVYNGISHVVMMASPKDLEYFALGFSLSEGIIESPRDIFGMDVVPSCNGLEVQIELSSRRFMGLKERRIGKPVQPLPFTQTFDLNKLDDALRHLNDFQPVGQLTGCTHAAAWMLPSGELVGGHEDVGRHVALDKLLGRRSQEGESWQQGAVLVSSRASYEMVQKSAMCGVEILFAVSAATTLAVEVAERCNLTLVGFCKPGRATVYTHPQRLSN 4pdk A 2.8 BS01 3VV A 1 L101 L102 A103 R105 T106 I108 L208 Y212 V215 G216 Y219 R253 G256 S259 G260 L94 L95 A96 R98 T99 I101 L201 Y205 V208 G209 Y212 R246 G249 S252 G253 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 301 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQM 4pdk A 2.8 BS02 3VV A 2 N130 Y153 K156 Y184 M187 R191 F194 H195 I200 L203 N123 Y146 K149 Y177 M180 R184 F187 H188 I193 L196 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 302 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQM 4pdk A 2.8 BS03 3VV B 1 I111 R114 Y115 I104 R107 Y108 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 301 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQM 4pdk A 2.8 BS04 3VV B 2 P27 M75 P20 M68 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 302 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQM 4pdk B 2.8 BS01 3VV A 2 W21 I82 W14 I75 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 302 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQMKMTLPS 4pdk B 2.8 BS02 3VV B 1 L101 L102 A104 R105 T106 L208 Y212 V215 G216 Y219 R253 G256 I257 S259 G260 L94 L95 A97 R98 T99 L201 Y205 V208 G209 Y212 R246 G249 I250 S252 G253 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 301 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQMKMTLPS 4pdk B 2.8 BS03 3VV B 2 R126 N130 Y153 Y184 M187 R191 F194 L203 I204 L208 R119 N123 Y146 Y177 M180 R184 F187 L196 I197 L201 ? 0000062,0003677,0003700,0005737,0006355,0006631,0019217,0071072 remove_due_to_license_issue Q9KQU8 25607896 302 PAGFAEKYIIESIWNGRFPPGSILPAERELSELIGVTRTTLREVLQRLARDGWLTIQHGKPTKVNQFMETSGLHILDTLMTLDAENATSIVEDLLAARTNISPIFMRYAFKLNKESAERIMINVIESCEALVNAPSWDAFIAASPYAEKIQQHVKEDSEKDELKRQEILIAKTFNFYDYMLFQRLAFHSGNQIYGLIFNGLKKLYDRVGSYYFSNPQARELAMEFYRQLLAVCQSGEREHLPQVIRQYGIASGHIWNQMKMTLPS 4pee A 1.95 BS01 2OX A 1 H66 E87 W88 H135 Y178 D229 W232 E288 W316 H32 E53 W54 H101 Y144 D195 W198 E254 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A3I4 25427942 504 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAKGTKSIY 4pf3 A 1.1 BS01 HFN A 1 N770 A773 Q776 M807 L810 F829 M845 M852 L938 F941 C942 T945 N36 A39 Q42 M73 L76 F95 M111 M118 L204 F207 C208 T211 ? ic50=51nM remove_due_to_license_issue P08235 25187277 1001 TPSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKCPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNVKPLYFHR 4pf5 A 2.04 BS03 M3N A 1 Y12 N14 G98 L99 Y100 A207 D208 R228 Y12 N14 G98 L99 Y100 A207 D208 R228 ? 0005537,0006952,0030246,0046872,0050688 remove_due_to_license_issue P02866 25483029 303 ADTIVAVELDTYPNTDIGDPSYPHIGIDIKSVRSKKTAKWNMQNGKVGTAHIIYNSVDKRLSAVVSYPNADSATVSYDVDLDNVLPEWVRVGLSASTGLYKETNTILSWSFTSKLKSNSTHETNALHFMFNQFSKDQKDLILQGDATTGTDGNLELTRVSSNGSPQGSSVGRALFYAPVHIWESSAVVASFEATFTFLIKSPDSHPADGIAFFISNIDSSIPSGSTGRLLGLFPDAN 4pg3 A 2.696 BS02 KRS A 1 E332 H338 N339 F342 E500 V501 N503 G554 G556 R559 E251 H257 N258 F261 E419 V420 N422 G457 G459 R462 R330 E332 T337 H338 E500 N503 R559 R249 E251 T256 H257 E419 N422 R462 6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 remove_due_to_license_issue IC50=120nM Q8IDJ8 24935905 602 PRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKYGLTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAGGANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFLDSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRP 4pgh A 2.8 BS01 SAM A 1 G206 D229 L230 D249 M250 K263 G198 D221 L222 D241 M242 K255 H267 D268 E296 E328 H259 D260 E288 E320 2.1.1.68 0008168,0008171,0008757,0009058,0009809,0017096,0030187,0032259,0046983,0047763,0051555,0102822 remove_due_to_license_issue C5YH12 24948836 401 AAVADEEACMYAMQLASSSILPMTLKNALELGLLEVLQKDAGKALAAEEVVARLPVAPTNPAAADMVDRMLRLLASYDVVKCQMEDKDGKYERRYSAAPVGKWLTPNEDGVSMAALALMNQDKVLMESWYYLKDAVLDGGIPFNKAYGMTAFEYHGTDPRFNRVFNEGMKNHSVIITKKLLEFYTGFDESVSTLVDVGGGIGATLHAITSHHSHIRGVNFDLPHVISEAPPFPGVQHVGGDMFKSVPAGDAILMKWILHDWSDAHCATLLKNCYDALPEKGGKVIVVECVLPVTTDAVPKAQGVFHVDMIMLAHNPGGRERYEREFRDLAKAAGFSGFKATYIYANAWAIEFIK 4ph4 B 2.8 BS01 2UG B 1 F612 I634 K636 Y670 M682 F684 I685 S687 L750 I760 F270 I292 K294 Y328 M340 F342 I343 S345 L408 I418 2.7.1.137 0016301,0016303,0046854 remove_due_to_license_issue IC50=18nM Q8NEB9 25327288 902 SGIRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEPLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHALF 4phu A 2.332 BS01 2YB A 1 P80 V84 F87 Y91 L138 G139 F142 L158 W174 R183 Y2240 R2258 P80 V84 F87 Y91 L130 G131 F134 L150 W166 R175 Y394 R412 E1011 D1020 E215 D224 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 Kd=12.04nM remove_due_to_license_issue O14842,P00720 25043059 2401 MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSAVYALNLGCSDLLLTVSLPLKAVEALASGAWPLPASLCPVFAVAHFAPLYAGGGFLAALSAARYLGAAFPPCYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAGPARFSLSLLLFFLPLAITAFCFVGCLRALARGSNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYGSLTHRRKLRAAWVAGGALLTLLLCVGPYNASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLG 4phv A 2.1 BS01 VAC B 1 D25 G27 A28 D29 V32 G48 P81 V82 D25 G27 A28 D29 V32 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4phv A 2.1 BS02 VAC B 2 D25 G27 A28 D29 V32 G48 V82 D25 G27 A28 D29 V32 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4phv B 2.1 BS01 VAC B 1 D25 G27 A28 D29 V32 I47 G48 V82 D25 G27 A28 D29 V32 I47 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=0.67nM remove_due_to_license_issue P12497 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4phv B 2.1 BS02 VAC B 2 D25 G27 A28 D29 V32 I47 G48 P81 V82 D25 G27 A28 D29 V32 I47 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 ic50=0.67nM remove_due_to_license_issue P12497 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4phw A 2.5 BS02 2W1 A 1 I682 Y683 F686 P702 M703 E711 V712 G715 F719 I229 Y230 F233 P249 M250 E258 V259 G262 F266 3.1.4.17 0004114,0007165,0008081 ic50=0.1nM remove_due_to_license_issue IC50=0.17nM Q9Y233 25062128 805 LPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRG 4pid A 1.59 BS02 2UQ A 1 G52 V53 Q115 A120 C122 G52 V53 Q115 A120 C122 H54 E71 Q115 C122 H54 E71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 remove_due_to_license_issue P03252 25147618 302 MGSSEQELKAIVKDLGCGPYFLGTYDKRFPGFVSPHKLACAIVNTAGRETGGVHWMAFAWNPRSKTCYLFEPFGFSDQRLKQVYQFEYESLLRRSAIASSPDRCITLEKSTQSVQGPNSAACGLFCCMFLHAFANWPQTPMDHNPTMNLITGVPNSMLNSPQVQPTLRRNQEQLYSFLERHSPYFRSHSAQIRSATSFCHLKNM 4pin A 1.9 BS01 AVI A 1 F47 Y56 T163 N166 Y206 E282 S284 F48 Y57 T162 N165 Y205 E281 S283 2.1.1.44 0008168,0008276,0032259,0052699,0052704,0052706 Kd=4uM remove_due_to_license_issue A0R5M8 25404173 401 HMALSLANYLAADSAAEALRRDVRAGLTATQKSLPPKWFYDAVGSDLFDQITRLPEYYPTRTEAQILRTRSAEIISAAGADTLVELGSSEKTRMLLDAMRDAELLRRFIPFDVDAGVLRSAGAAIGAEYPGIEIDAVCGDFEEHLGKIPHVGRRLVVFLGSTIGNLTPAPRAEFLSTLADTLQPGDSLLLGTDLVKDTGRLVRAYDDAAGVTAAFNRNVLAVVNRELSADFDLDAFEHVAKWNSDEERIEMWLRARTAQHVRVAALDLEVDFAAGEEMLTEVSCKFRPENVVAELAEAGLRQTHWWTDPAGDFGLSLAVR 4pio A 1.506 BS02 AVI A 1 Y56 G161 S162 T163 N166 Y206 E282 S284 Y42 G147 S148 T149 N152 Y192 E268 S270 2.1.1.44 0008168,0008276,0032259,0052699,0052704,0052706 Kd=2uM remove_due_to_license_issue A0R5M8 25404173 402 AEALRRDVRAGLTATQKSLPPKWFYDAVGSDLFDQITRLPEYYPTRTEAQILRTRSAEIISAAGADTLVELGSGTSEKTRMLLDAMRDAELLRRFIPFDVDAGVLRSAGAAIGAEYPGIEIDAVCGDFEEHLGKIPHVGRRLVVFLGSTIGNLTPAPRAEFLSTLADTLQPGDSLLLGTDLVKDTGRLVRAYDDAAGVTAAFNRNVLAVVNRELSADFDLDAFEHVAKWNSDEERIEMWLRARTAQHVRVAALDLEVDFAAGEEMLTEVSDKFRPENVVAELAEAGLRQTHWWTDPAGDFGLSLAVR 4piq A 2.07 BS02 3FS A 1 S3 S4 E5 T24 H25 D26 N44 A46 G47 R48 G51 G52 V53 W55 A120 C122 S3 S4 E5 T24 H25 D26 N44 A46 G47 R48 G51 G52 V53 W55 A120 C122 H54 D71 Q115 C122 H54 D71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 remove_due_to_license_issue B9A5C1 25147618 301 SGSSEQELAAIVRDLGCGPYFLGTHDKRFPGFLAGNKLACAIVNTAGRETGGVHWLAFGWNPRSRTCYMFDPFGFSDRRLKQIYSFEYEAMLRRSALALSPDRCLSLEQSTQTVQGPDSAACGLFCCMFLHAFVHWPDRPMDGNPTMNLLTGVPNGMLQSPQVLPTLRRNQEKLYRFLAHHSPYFRSHRAAIEHATAFDKMKQL 4pis A 2.1 BS02 3FU A 1 S1 S4 E5 T24 H25 D26 N44 A46 G47 R48 G51 G52 V53 W55 A120 C122 S1 S4 E5 T24 H25 D26 N44 A46 G47 R48 G51 G52 V53 W55 A120 C122 H54 D71 Q115 C122 H54 D71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 remove_due_to_license_issue B9A5C1 25147618 301 SGSSEQELAAIVRDLGCGPYFLGTHDKRFPGFLAGNKLACAIVNTAGRETGGVHWLAFGWNPRSRTCYMFDPFGFSDRRLKQIYSFEYEAMLRRSALALSPDRCLSLEQSTQTVQGPDSAACGLFCCMFLHAFVHWPDRPMDGNPTMNLLTGVPNGMLQSPQVLPTLRRNQEKLYRFLAHHSPYFRSHRAAIEHATAFDKMKQL 4pji A 2.5 BS01 30W A 1 Y7 R9 K43 Y62 W69 R94 I96 W156 Y7 R9 K42 Y61 W68 R93 I95 W155 ? remove_due_to_license_issue Q95460 25049336 301 RTHSLRYFRLGVSDPIGVPEFISVGYVDSHPITTYDSVTRQKEPRAPWMAENLAPDHWERYTQLLRGWQQMFKVELKRLQRHYNHSGSHTYQRMIGCELLEDGSTTGFLQYAYDGQDFLIFNKDTLSWLAVDNVAHTIKQAWEANQHELLYQKNWLEEECIAWLKRFLEYGKDTLQRTEPPLVRVNRKETFPGVTALFCKAHGFYPPEIYMTWMKNGEEIVQEIDYGDILPSGDGTYQAWASIELLYSCHVEHSGVHMVLQV 4pjt A 2.35 BS01 2YQ A 1 E763 H862 G863 G888 Y889 Y896 S904 Y907 E96 H190 G191 G216 Y217 Y224 S232 Y235 S904 Y907 E988 S232 Y235 E316 2.4.2.-,2.4.2.30 0003950 ic50=0.57nM remove_due_to_license_issue Ki=1.2nM, IC50=0.570000nM, EC50=2.5nM P09874 25195882 1105 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQDSQILDLSNRFYTLIPHDFKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 4pkb A 2.09 BS01 MAY A 1 G36 G37 G38 S77 T78 D215 G12 G13 G14 S53 T54 D191 3.1.1.- 0006629 remove_due_to_license_issue Q8LPW4 25248161 401 LGEMVTVLSIDGGGIRGIIPATILEFLEGQLQEMDNNADARLADYFDVIGGTSTGGLLTAMISTPNENNRPFAAAKEIVPFYFEHGPQIFNPSGQILGPKYDGKYLMQVLQEKLGETRVHQALTEVVISSFDIKTNKPVIFTKSNLANSPELDAKMYDISYSTAAAPTYFPPHYFVTNTSNGDEYEFNLVDGAVATVADPALLSISVATRLAQKDPAFASIRSLNYKKMLLLSLGTGTTSEFDKTYTAKEAATWTAVHWMLVIQKMTDAASSYMTDYYLSTAFQALDSKNNYLRVQENALTGTTTEMDDASEANMELLVQVGENLLKKPVSEDNPETYEEALKRFAKLLSDRKKLRA 4pkr A 2.2 BS01 2ZL A 1 S655 K656 G657 L677 H686 E687 H690 Y728 E735 E739 R742 S374 K375 G376 L396 H405 E406 H409 Y447 E454 E458 R461 H686 E687 H690 Y728 E735 H405 E406 H409 Y447 E454 3.4.24.83 0008237 ic50=15.2uM remove_due_to_license_issue P15917 25372673 801 RYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEELSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4pks A 2.3 BS02 30H A 1 F329 S655 K656 G657 L677 H686 E687 H690 Y728 E735 E739 R742 F63 S365 K366 G367 L387 H396 E397 H400 Y438 E445 E449 R452 H686 E687 H690 Y728 E735 H396 E397 H400 Y438 E445 3.4.24.83 0008237 ic50=15.2uM remove_due_to_license_issue P15917 25372673 802 RYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4pkt A 2.4 BS01 30O A 1 D328 K656 G657 V675 L677 H686 E687 H690 Y728 R742 D64 K377 G378 V396 L398 H407 E408 H411 Y449 R463 H686 E687 H690 Y728 E735 H407 E408 H411 Y449 E456 3.4.24.83 0008237 ic50=14.9uM remove_due_to_license_issue P15917 25372673 801 LSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSSSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINSLV 4pku A 2.4 BS01 30P A 1 S655 K656 G657 V675 L677 H686 E687 H690 Y728 E735 E739 S368 K369 G370 V388 L390 H399 E400 H403 Y441 E448 E452 H686 E687 H690 Y728 E735 H399 E400 H403 Y441 E448 3.4.24.83 0008237 ic50=30uM remove_due_to_license_issue P15917 25372673 801 SRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4pkv A 2.5 BS01 30R A 1 D328 S655 K656 G657 V675 L677 H686 E687 H690 Y728 E735 D65 S392 K393 G394 V412 L414 H423 E424 H427 Y465 E472 H686 E687 H690 Y728 E735 H423 E424 H427 Y465 E472 3.4.24.83 0008237 ic50=5.6uM remove_due_to_license_issue P15917 25372673 801 ALSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEEEKELLNRIQVDSSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINSLV 4pkw A 1.75 BS02 GM6 A 1 D328 F329 V653 H654 S655 K656 G657 H686 E687 H690 Y728 E735 D63 F64 V368 H369 S370 K371 G372 H401 E402 H405 Y443 E450 H686 E687 H690 Y728 E735 H401 E402 H405 Y443 E450 3.4.24.83 0008237 ic50=22.5uM remove_due_to_license_issue P15917 25372673 802 SRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4pl0 A 2.7 BS01 ANP A 1 Y354 S380 G381 S382 G383 K384 S385 T386 Q426 Y346 S372 G373 S374 G375 K376 S377 T378 Q418 ? 0005524,0005886,0015031,0015421,0016020,0016887,0030153,0035672,0043213,0055085,0140359 remove_due_to_license_issue Q9X2W0 24920594 601 LFNYIYSLMDVRGKFLFFSMLFITSLSSIIISISPLILAKITDLLSGSLSNFSYEYLVLLACLYMFCVISNKASVFLFMILQSSLRINMQKKMSLKYLRELYNENITNLSKNNAGYTTQSLNQASNDIYILVRNVSQNILSPVIQLISTIVVVLSTKDWFSAGVFFLYILVFVIFNTRLTGSLASLRKHSMDITLNSYSLLSDTVDNMIAAKKNNALRLISERYEDALTQENNAQKKYWLLSSKVLLLNSLLAVILFGSVFIYNILGVLNGVVSIGHFIMITSYIILLSTPVENIGALLSEIRQSMSSLAGFIQRHAENKATSPSIPFLNMERKLNLSIRELSFSYSDDKKILNSVSLDLFTGKMYSLTGPSGSGKSTLVKIISGYYKNYFGDIYLNDISLRNISDEDLNDAIYYLTQDDYIFMDTLRFNLRLANYDASENEIFKVLKLANLSVVNNEPVSLDTHLINRGNNYSGGQKQRISLARLFLRKPAIIIIDEATSALDYINESEILSSIRTHFPDALIINISHRINLLECSDCVYVLNEGNIVASGHFRDLMVSNEYISGLASVT 4pl0 A 2.7 BS03 ANP B 1 N464 N479 N480 S482 G484 Q485 N456 N471 N472 S474 G476 Q477 ? 0005524,0005886,0015031,0015421,0016020,0016887,0030153,0035672,0043213,0055085,0140359 remove_due_to_license_issue Q9X2W0 24920594 601 LFNYIYSLMDVRGKFLFFSMLFITSLSSIIISISPLILAKITDLLSGSLSNFSYEYLVLLACLYMFCVISNKASVFLFMILQSSLRINMQKKMSLKYLRELYNENITNLSKNNAGYTTQSLNQASNDIYILVRNVSQNILSPVIQLISTIVVVLSTKDWFSAGVFFLYILVFVIFNTRLTGSLASLRKHSMDITLNSYSLLSDTVDNMIAAKKNNALRLISERYEDALTQENNAQKKYWLLSSKVLLLNSLLAVILFGSVFIYNILGVLNGVVSIGHFIMITSYIILLSTPVENIGALLSEIRQSMSSLAGFIQRHAENKATSPSIPFLNMERKLNLSIRELSFSYSDDKKILNSVSLDLFTGKMYSLTGPSGSGKSTLVKIISGYYKNYFGDIYLNDISLRNISDEDLNDAIYYLTQDDYIFMDTLRFNLRLANYDASENEIFKVLKLANLSVVNNEPVSLDTHLINRGNNYSGGQKQRISLARLFLRKPAIIIIDEATSALDYINESEILSSIRTHFPDALIINISHRINLLECSDCVYVLNEGNIVASGHFRDLMVSNEYISGLASVT 4pl0 B 2.7 BS01 ANP A 1 N464 N479 N480 S482 G483 G484 Q485 N461 N476 N477 S479 G480 G481 Q482 ? 0005524,0005886,0015031,0015421,0016020,0016887,0030153,0035672,0043213,0055085,0140359 remove_due_to_license_issue Q9X2W0 24920594 601 KQKNSLFNYIYSLMDVRGKFLFFSMLFITSLSSIIISISPLILAKITDLLSGSLSNFSYEYLVLLACLYMFCVISNKASVFLFMILQSSLRINMQKKMSLKYLRELYNENITNLSKNNAGYTTQSLNQASNDIYILVRNVSQNILSPVIQLISTIVVVLSTKDWFSAGVFFLYILVFVIFNTRLTGSLASLRKHSMDITLNSYSLLSDTVDNMIAAKKNNALRLISERYEDALTQENNAQKKYWLLSSKVLLLNSLLAVILFGSVFIYNILGVLNGVVSIGHFIMITSYIILLSTPVENIGALLSEIRQSMSSLAGFIQRHAENKATSPSIPFLNMERKLNLSIRELSFSYSDDKKILNSVSLDLFTGKMYSLTGPSGSGKSTLVKIISGYYKNYFGDIYLNDISLRNISDEDLNDAIYYLTQDDYIFMDTLRFNLRLANYDASENEIFKVLKLANLSVVNNEPVSLDTHLINRGNNYSGGQKQRISLARLFLRKPAIIIIDEATSALDYINESEILSSIRTHFPDALIINISHRINLLECSDCVYVLNEGNIVASGHFRDLMVSNEYISGLASVT 4pl0 B 2.7 BS02 ANP B 1 Y354 S380 G381 S382 G383 K384 S385 T386 Q426 Y351 S377 G378 S379 G380 K381 S382 T383 Q423 ? 0005524,0005886,0015031,0015421,0016020,0016887,0030153,0035672,0043213,0055085,0140359 remove_due_to_license_issue Q9X2W0 24920594 601 KQKNSLFNYIYSLMDVRGKFLFFSMLFITSLSSIIISISPLILAKITDLLSGSLSNFSYEYLVLLACLYMFCVISNKASVFLFMILQSSLRINMQKKMSLKYLRELYNENITNLSKNNAGYTTQSLNQASNDIYILVRNVSQNILSPVIQLISTIVVVLSTKDWFSAGVFFLYILVFVIFNTRLTGSLASLRKHSMDITLNSYSLLSDTVDNMIAAKKNNALRLISERYEDALTQENNAQKKYWLLSSKVLLLNSLLAVILFGSVFIYNILGVLNGVVSIGHFIMITSYIILLSTPVENIGALLSEIRQSMSSLAGFIQRHAENKATSPSIPFLNMERKLNLSIRELSFSYSDDKKILNSVSLDLFTGKMYSLTGPSGSGKSTLVKIISGYYKNYFGDIYLNDISLRNISDEDLNDAIYYLTQDDYIFMDTLRFNLRLANYDASENEIFKVLKLANLSVVNNEPVSLDTHLINRGNNYSGGQKQRISLARLFLRKPAIIIIDEATSALDYINESEILSSIRTHFPDALIINISHRINLLECSDCVYVLNEGNIVASGHFRDLMVSNEYISGLASVT 4pl3 A 2.9 BS01 31J A 1 F889 Y892 N906 K907 H910 F313 Y316 N330 K331 H334 D688 K690 N693 D711 T734 D129 K131 N134 D152 T163 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue Q9EQY0 25164867 1001 ETRMVIVGKISFCPKDVLGHGAEGTIVYKGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLHQTTSGLAHLHSLNIVHRDLKPHNILLSMPNAHGRIKAMISDFGLCKKLVPGTEGWIAPEMLDNPTYTVDIFSAGCVFYYVISEGYHPFGKSLQRQANILLGACNLDCFHSDKHEDVIARELIEKMIAMDPQQRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKEALDGPIVRQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPVEVQETLGSIPDDFVRYFTSRFPHLLSHTYQAMELCRHERLFQTYYWHE 4pl4 A 3.0 BS01 31K A 1 F889 Y892 N906 K907 H910 F311 Y314 N328 K329 H332 D688 K690 N693 D711 T734 D127 K129 N132 D150 T162 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue Q9EQY0 25164867 1001 RMVIVGKISFCPKDVLGHGAEGTIVYKGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLHQTTSGLAHLHSLNIVHRDLKPHNILLSMPNAHGRIKAMISDFGLCKKLAVPGTEGWIAPEMLSPTYTVDIFSAGCVFYYVISEGYHPFGKSLQRQANILLGACNLDCFHSDKHEDVIARELIEKMIAMDPQQRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKEALDGPIVRQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPVEVQETLGSIPDDFVRYFTSRFPHLLSHTYQAMELCRHERLFQTYYWH 4pl5 A 3.4 BS01 31L A 1 Y892 K907 H910 Y314 K329 H332 D688 K690 N693 D711 T734 D127 K129 N132 D150 T161 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue Q9EQY0 25164867 1001 RMVIVGKISFCPKDVLGHGAEGTIVYKGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLHQTTSGLAHLHSLNIVHRDLKPHNILLSMPNAHGRIKAMISDFGLCKKLVPGTEGWIAPEMLSEPTYTVDIFSAGCVFYYVISEGYHPFGKSLQRQANILLGACNLDCFHSDKHEDVIARELIEKMIAMDPQQRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKEALDGPIVRQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPVEVQETLGSIPDDFVRYFTSRFPHLLSHTYQAMELCRHERLFQTYYWHE 4pm0 A 2.1 BS02 32V A 1 Y211 I363 N365 V380 F384 I412 Q413 F416 Y73 I225 N227 V242 F246 I274 Q275 F278 S169 A250 S31 A112 3.1.4.53 0004114,0007165,0008081 ic50=45nM remove_due_to_license_issue IC50=45nM Q13946 25383422 503 DYNGQAKCMLEKVGNWNFDIFLFDRLTNGNSLVSLTFHLFSLHGLIEYFHLDMMKLRRFLVMIQEDYHSQNPYHNAVHAADVTQAMHCYLKEPKLANSVTPWDILLSLIAAATHDLDHPGVNQPFLIKTNHYLATLYKNTSVLENHHWRSAVGLLRESGLFSHLPLESRQQMETQIGALILATDISRQNEYLSLFRSHLDRGDLCLEDTRHRHLVLQMALKCADICNPCRTWELSKQWSEKVTEEFFHQGDIEKKYHLGVSPLCDRHTESIANIQIGFMTYLVEPLFTEWARFSNTRLSQTMLGHVGLNKASWKGLQR 4pml A 1.87 BS02 3AB A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 E1138 H69 G70 Y98 F99 K105 S106 Y109 E175 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 KEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVGLALAEYVIYRGEQAYPEYLITYQIMRPE 4pmm A 2.0 BS01 31V A 1 A542 K544 E560 F589 Y591 M592 L657 G667 D668 F669 A39 K41 E54 F83 Y85 M86 L151 G161 D162 F163 D650 A652 R654 N655 D668 S677 L689 D144 A146 R148 N149 D162 S171 L183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd=27nM remove_due_to_license_issue IC50=662nM, Kd=27nM P04629 24914455 801 CVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLDKMLVAVKALKESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAHHHH 4pmp A 1.8 BS01 31W A 1 A542 L564 V573 F589 E590 Y591 M592 L657 G667 D668 F669 A38 L56 V65 F81 E82 Y83 M84 L149 G159 D160 F161 D650 A652 R654 N655 D668 S677 L689 D142 A144 R146 N147 D160 S168 L178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd~400nM remove_due_to_license_issue Kd=400nM, IC50=549nM P04629 24914455 801 CVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLKMLVAVKALKSARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRIYSTDYYRVGTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAHHHH 4pms A 2.8 BS01 31X A 1 V524 K544 L564 V573 F589 L657 D668 F669 G670 M671 V24 K41 L58 V67 F83 L151 D162 F163 G164 M165 D650 A652 R654 N655 D668 S677 L689 D144 A146 R148 N149 D162 S171 L181 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=2300nM, Kd=7.9nM P04629 24914455 801 CVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLDKMLVAVKALKESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAHHHH 4pmt A 2.1 BS01 31Y A 1 L516 G517 A542 F589 M592 R599 L657 R673 L16 G17 A38 F76 M79 R86 L144 R158 D650 A652 R654 N655 D668 S677 L689 D137 A139 R141 N142 D155 S162 L171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=997nM remove_due_to_license_issue IC50=997nM P04629 24914455 801 CVHHIKRRDIVLKWELGEGAFGKVFLAECHNLDKMLVAVKALDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFSRDIYSTDYYRVTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAHHHH 4pmw A 2.95 BS01 rna C 0 R74 P77 K78 F80 F84 D93 H271 R275 D381 P382 D387 L388 N389 D390 Y433 Y492 L549 D550 Q551 K553 Y573 E581 M584 R606 H608 Q612 M615 S664 R665 M667 M669 A670 H686 Y694 H696 T698 R702 R741 K745 R746 L776 N777 Q778 Q790 R792 Y794 N796 R26 P29 K30 F32 F36 D45 H106 R110 D216 P217 D222 L223 N224 D225 Y268 Y327 L384 D385 Q386 K388 Y408 E416 M419 R441 H443 Q447 M450 S499 R500 M502 M504 A505 H521 Y529 H531 T533 R537 R576 K580 R581 L611 N612 Q613 Q625 R627 Y629 N631 D381 D387 N389 D390 Y492 R702 D216 D222 N224 D225 Y327 R537 3.1.13.- 0000175,0003723,0004540 remove_due_to_license_issue Q8CI75 25119025 1 ~ 14 IFETYMSKEDVSEGLKRGTLIQGVLRINPKKFHEAFIPSPDGDRDIFIDGVVARNRALNGDLVVVKLLPEKSAKVVYILEKKHSRAATGILKLLFKKYALFSPSDHRVPRIYVPLKDCPQDFMTRPKDFANTLFICRIIDWKEDCNFALGQLAKSLGQAGEIEPETEGILTEYGVDFSDFSSEVLECLPQSLPWTIPPDEVGKRRDLRKDCIFTIDPSTARDLNDALACRRLTDGTFEVGVHIADVSYFVPEGSSLDKVAAERATSVYLVQKVVPMLPRLLCEELCSLNPMTDKLTFSVIWKLTPEGKILEEWFGRTIIRSCTKLSYDHAQSMIENPTEKIPEEELPPISPEHSVEEVHQAVLNLHSIAKQLRRQRFVDGALRLDQLKLAFTLDHETGLPQGCHIYEYRDSNKLVEEFMLLANMAVAHKIFRTFPEQALLRRHPPPQTKMLSDLVEFCDQMGLPMDVSSAGALNKSLTKTFGDDKYSLARKEVLTNMYSRPMQMALYFCSGMLQDQEQFRHYALNVPLYTHFTSPIRRFADVIVHRLLAAALGYSEQPDVEPDTLQKQADHCNDRRMASKRVQELSIGLFFAVLVKESGPLESEAMVMGVLNQAFDVLVLRFGVQKRIYCNALALRSYSFQKVGKKPELTLVWEPDDLEEEPTQQVITIFSLVDVVLQAEATALKYSAILK 4pmw B 2.95 BS01 rna D 0 R74 N76 P77 K78 F80 F84 D93 H271 R275 D381 P382 A385 D387 L388 N389 D390 Y433 Y492 L549 D550 Q551 K553 Y573 E581 M584 R606 H608 Q612 M615 S664 R665 M667 M669 A670 H686 Y694 H696 T698 S699 R702 R741 K745 R746 L776 N777 Q778 Q790 R792 Y794 N796 R26 N28 P29 K30 F32 F36 D45 H106 R110 D216 P217 A220 D222 L223 N224 D225 Y268 Y327 L384 D385 Q386 K388 Y408 E416 M419 R441 H443 Q447 M450 S499 R500 M502 M504 A505 H521 Y529 H531 T533 S534 R537 R576 K580 R581 L611 N612 Q613 Q625 R627 Y629 N631 D381 D387 N389 D390 Y492 R702 D216 D222 N224 D225 Y327 R537 3.1.13.- 0000175,0003723,0004540 remove_due_to_license_issue Q8CI75 25119025 1 ~ 14 IFETYMSKEDVSEGLKRGTLIQGVLRINPKKFHEAFIPSPDGDRDIFIDGVVARNRALNGDLVVVKLLPEKSAKVVYILEKKHSRAATGILKLLFKKYALFSPSDHRVPRIYVPLKDCPQDFMTRPKDFANTLFICRIIDWKEDCNFALGQLAKSLGQAGEIEPETEGILTEYGVDFSDFSSEVLECLPQSLPWTIPPDEVGKRRDLRKDCIFTIDPSTARDLNDALACRRLTDGTFEVGVHIADVSYFVPEGSSLDKVAAERATSVYLVQKVVPMLPRLLCEELCSLNPMTDKLTFSVIWKLTPEGKILEEWFGRTIIRSCTKLSYDHAQSMIENPTEKIPEEELPPISPEHSVEEVHQAVLNLHSIAKQLRRQRFVDGALRLDQLKLAFTLDHETGLPQGCHIYEYRDSNKLVEEFMLLANMAVAHKIFRTFPEQALLRRHPPPQTKMLSDLVEFCDQMGLPMDVSSAGALNKSLTKTFGDDKYSLARKEVLTNMYSRPMQMALYFCSGMLQDQEQFRHYALNVPLYTHFTSPIRRFADVIVHRLLAAALGYSEQPDVEPDTLQKQADHCNDRRMASKRVQELSIGLFFAVLVKESGPLESEAMVMGVLNQAFDVLVLRFGVQKRIYCNALALRSYSFQKVGKKPELTLVWEPDDLEEEPTQQVITIFSLVDVVLQAEATALKYSAILK 4pnc A 1.54 BS01 7NP A 1 C59 Y65 C70 H79 F177 H178 C58 Y64 C69 H78 F176 H177 H79 D97 D108 H171 Q175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 Q174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008235,0046872,0070006 remove_due_to_license_issue C3TPN7 25293447 301 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGQGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHD 4pni A 1.85 BS01 KQQ A 1 L193 F198 V201 A214 T265 M267 N268 G270 D271 L321 R474 T475 L164 F169 V172 A185 T236 M238 N239 G241 D242 L292 R445 T446 D314 K316 E318 N319 D332 A341 T352 D285 K287 E289 N290 D303 A312 T323 2.7.11.14 0001750,0004672,0004674,0004703,0005515,0005524,0005737,0006468,0007165,0007601,0009966,0016020,0022400,0042995,0046777,0050254,0097381 ic50=0.125uM remove_due_to_license_issue IC50=130nM P28327 25238254 601 SRDRKYLARLKLPPLSKCEALRESLDLGFEGMCLEQPIGKRLFQQFLRTHEQHGPALQLWKDIEDYDTADDALRPQKAQALRAAYLEPQAQLFCSFLDAETVARARAGAGDGLFQPLLRAVLAHLGQAPFQEFLDSLYFLRFLQWKWLEAQPMGEDWFLDFRVLGRGGFGEVFACQMKATGKLYACKKLNKKRLKKRKGYQGAMVEKKILAKVHSRFIVSLAYAFETKTDLCLVMTIMNGGDIRYHIYNVDEDNPGFQEPRAIFYTAQIVSGLEHLHQRNIIYRDLKPENVLLDDDGNVRISDLGLAVELKAGQTKTKGYAGTPGFMAPELLLGEEYDFSVDYFALGVTLYEMIAARGPFRARGEKVENKELKQRVLEQAVTYPDKFSPASKDFCEALLQKDPEKRLGFRDGSCDGLRTHPLFRDISWRQLEAGMLTPPFVPDSRTVYAKNIAFEKADTEFFQEFASGTCPIPWQEEMIETGVFGDLNVWRP 4pnk A 2.56 BS01 KZQ A 1 I197 R199 G200 A218 D272 M274 A321 L324 S334 I168 R170 G171 A189 D243 M245 A292 L295 S305 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue P25098 25238254 701 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPREVNATKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 4pnl A 1.5 BS02 DRL A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 E1138 H69 G70 Y98 F99 K105 S106 Y109 E176 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 KEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4pnm A 2.19 BS02 NU1 A 1 H1031 G1032 Y1060 A1062 S1068 Y1071 H70 G71 Y99 A101 S107 Y110 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4pnn A 1.65 BS02 JPZ A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 E1138 H69 G70 Y98 F99 K105 S106 Y109 E176 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 KEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4pnq A 1.85 BS02 32X A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 E1138 H72 G73 Y101 F102 K108 S109 Y112 E179 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 PDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4pnr A 1.71 BS02 G18 A 1 H1031 G1032 Y1050 Y1060 F1061 K1067 S1068 Y1071 H70 G71 Y89 Y99 F100 K106 S107 Y110 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4pns A 1.65 BS02 32Y A 1 H1031 G1032 Y1060 S1068 Y1071 H70 G71 Y97 S105 Y108 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4pnt A 1.6 BS02 IQD A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 E1138 H71 G72 Y99 F100 K106 S107 Y110 E177 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4pnu A 1.9 BS01 2VD A 1 R152 Y154 T172 G174 H175 R176 L177 V247 V360 M362 R147 Y149 T167 G169 H170 R171 L172 V242 V355 M357 0003677,0003887,0006260,0008408,0009360 remove_due_to_license_issue 25970224 405 MKFTVEREHLLKPLQQVSGPLLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4pnw B 2.0 BS01 2VM B 1 Y154 D173 G174 H175 R176 L177 V360 M362 Y154 D173 G174 H175 R176 L177 V360 M362 0003677,0003887,0006260,0008408,0009360 remove_due_to_license_issue 25970224 402 MKFTVEREHLLKPLQQVSGPLGGRPTLPILGNLLLQVADGTLSLTGTDLEMEMVARVALVQPHEPGATTVPARKFFDICRGLPEGAEIAVQLEGERMLVRSGRSRFSLSTLPAADFPNLDDWQSEVEFTLPQATMKRLIEATQFSMAHQDVRYYLNGMLFETEGEELRTVATDGHRLAVCSMPIGQSLPSHSVIVPRKGVIELMRMLDGGDNPLRVQIGSNNIRAHVGDFIFTSKLVDGRFPDYRRVLPKNPDKHLEAGCDLLKQAFARAAILSNEKFRGVRLYVSENQLKITANNPEQEEAEEILDVTYSGAEMEIGFNVSYVLDVLNALKCENVRMMLTDSVSSVQIEDAASQSAAYVVMPM 4po0 A 2.73 BS01 NPS A 1 N391 Y411 K414 V449 L453 R485 F488 S489 N390 Y410 K413 V448 L452 R484 F487 S488 ? 0003677,0005504,0005576,0005615,0005737,0005783,0005794,0008289,0009267,0015643,0019825,0030170,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0140272,1903981 remove_due_to_license_issue G1U9S2 24753230 601 AHKSEIAHRFNDVGEEHFIGLVLITFSQYLQKCPYEEHAKLVKEVTDLAKACVADESAANCDKSLHDIFGDKICALPSLRDTYGDVADCCEKKEPERNECFLHHKDDKPDLPPFARPEADVLCKAFHDDEKAFFGHYLYEVARRHPYFYAPELLYYAQKYKAILTECCEAADKGACLTPKLDALKEKALISAAQERLRCASIQKFGDRAYKAWALVRLSQRFPKADFTDISKIVTDLTKVHKECCHGDLLECADDRADLAKYMCEHQETISSHLKECCDKPILEKAHCIYGLHNDETPAGLPAVAEEFVEDKDVCKNYEEAKDLFLGKFLYEYSRRHPDYSVVLLLRLGKAYEATLKKCCATDDPHACYAKVLDEFQPLVDEPKNLVKQNCELYEQLGDYNFQNALLVRYTKKVPQVSTPTLVEISRSLGKVGSKCCKHPEAERLPCVEDYLSVVLNRLCVLHEKTPVSEKVTKCCSESLVDRRPCFSALGPDETYVPKEFNAETFTFHADICTLPETERKIKKQTALVELVKHKPHATNDQLKTVVGEFTALLDKCCSAEDKEACFAVEGPKLVESSKATLG 4po0 A 2.73 BS02 NPS A 2 R209 A213 G328 L331 G350 R208 A212 G327 L330 G349 ? 0003677,0005504,0005576,0005615,0005737,0005783,0005794,0008289,0009267,0015643,0019825,0030170,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0140272,1903981 remove_due_to_license_issue G1U9S2 24753230 602 AHKSEIAHRFNDVGEEHFIGLVLITFSQYLQKCPYEEHAKLVKEVTDLAKACVADESAANCDKSLHDIFGDKICALPSLRDTYGDVADCCEKKEPERNECFLHHKDDKPDLPPFARPEADVLCKAFHDDEKAFFGHYLYEVARRHPYFYAPELLYYAQKYKAILTECCEAADKGACLTPKLDALKEKALISAAQERLRCASIQKFGDRAYKAWALVRLSQRFPKADFTDISKIVTDLTKVHKECCHGDLLECADDRADLAKYMCEHQETISSHLKECCDKPILEKAHCIYGLHNDETPAGLPAVAEEFVEDKDVCKNYEEAKDLFLGKFLYEYSRRHPDYSVVLLLRLGKAYEATLKKCCATDDPHACYAKVLDEFQPLVDEPKNLVKQNCELYEQLGDYNFQNALLVRYTKKVPQVSTPTLVEISRSLGKVGSKCCKHPEAERLPCVEDYLSVVLNRLCVLHEKTPVSEKVTKCCSESLVDRRPCFSALGPDETYVPKEFNAETFTFHADICTLPETERKIKKQTALVELVKHKPHATNDQLKTVVGEFTALLDKCCSAEDKEACFAVEGPKLVESSKATLG 4po0 A 2.73 BS03 NPS A 3 L529 N541 L544 K545 V548 L528 N540 L543 K544 V547 ? 0003677,0005504,0005576,0005615,0005737,0005783,0005794,0008289,0009267,0015643,0019825,0030170,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0140272,1903981 remove_due_to_license_issue G1U9S2 24753230 603 AHKSEIAHRFNDVGEEHFIGLVLITFSQYLQKCPYEEHAKLVKEVTDLAKACVADESAANCDKSLHDIFGDKICALPSLRDTYGDVADCCEKKEPERNECFLHHKDDKPDLPPFARPEADVLCKAFHDDEKAFFGHYLYEVARRHPYFYAPELLYYAQKYKAILTECCEAADKGACLTPKLDALKEKALISAAQERLRCASIQKFGDRAYKAWALVRLSQRFPKADFTDISKIVTDLTKVHKECCHGDLLECADDRADLAKYMCEHQETISSHLKECCDKPILEKAHCIYGLHNDETPAGLPAVAEEFVEDKDVCKNYEEAKDLFLGKFLYEYSRRHPDYSVVLLLRLGKAYEATLKKCCATDDPHACYAKVLDEFQPLVDEPKNLVKQNCELYEQLGDYNFQNALLVRYTKKVPQVSTPTLVEISRSLGKVGSKCCKHPEAERLPCVEDYLSVVLNRLCVLHEKTPVSEKVTKCCSESLVDRRPCFSALGPDETYVPKEFNAETFTFHADICTLPETERKIKKQTALVELVKHKPHATNDQLKTVVGEFTALLDKCCSAEDKEACFAVEGPKLVESSKATLG 4poh A 2.3 BS02 2VR A 1 I268 A271 A272 Q275 W305 F313 R316 L326 L436 I24 A27 A28 Q31 W61 F69 R72 L82 L192 ? 0003677,0003707,0005634,0006355,0008270 Kd=10nM remove_due_to_license_issue EC50=620nM, Kd=10.0nM P19793 24801499 501 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4poj A 2.0 BS02 2VP A 1 I268 A271 A272 Q275 F313 R316 L326 A327 I345 L436 I24 A27 A28 Q31 F69 R72 L82 A83 I101 L192 ? 0003677,0003707,0005634,0006355,0008270 Kd=8nM remove_due_to_license_issue Kd=8.0nM, EC50=160nM P19793 24801499 501 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4pop A 2.2 BS01 2VY A 1 W34 E84 Y85 H125 W133 N151 W29 E79 Y80 H120 W128 N146 ? 0005886,0015234,0015888,0071934 remove_due_to_license_issue Kd=7.44nM A2RI47 25676607 201 FNVRLLTEIAFMAALAFIISLIPNTVYGWIIVEIACIPILLLSLRRGLTAGLVGGLIWGILSMITGHAYILSLSQAFLEYLVAPVSLGIAGLFRQKTAPLKLAPVLLGTFVAVLLKYFFHFIAGIIFWSQYAWKGWGAVAYSLAVNGISGILTAIAAFVILIIFVKKFPKLFIHSNY 4pov A 2.2 BS01 2VY A 1 W34 E84 Y85 H125 W133 N151 W30 E80 Y81 H121 W129 N147 ? 0005886,0015234,0015888,0071934 remove_due_to_license_issue Kd=7.44nM A2RI47 25676607 201 KFNVRLLTEIAFMAALAFIISLIPNTVYGWIIVEIACIPILLLSLRRGLTAGLVGGLIWGILSMITGHAYILSLSQAFLEYLVAPVSLGIAGLFRQKTAPLKLAPVLLGTFVAVLLKYFFHFIAGIIFWSQYAWKGWGAVAYSLAVNGISGILTAIAAFVILIIFVKKFPKLFIHSNY 4pow A 1.55 BS01 OP1 A 1 E36 Y39 W77 A94 A95 G97 R102 M117 Q165 T168 S169 H170 S207 E9 Y12 W50 A67 A68 G70 R75 M90 Q138 T141 S142 H143 S180 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=0.58uM remove_due_to_license_issue P35120 25299655 303 YKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPMTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASP 4pp0 A 1.57 BS01 OP1 A 1 E36 Y39 W77 A94 A95 G97 R102 Q165 T168 S169 H170 S207 E9 Y12 W50 A67 A68 G70 R75 Q138 T141 S142 H143 S180 ? 0015276,0016020,0030288,0034220,0042597,0071705 remove_due_to_license_issue P35120 25299655 301 YKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPNTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASP 4pp3 A 2.0 BS02 2VZ A 1 I268 A271 A272 Q275 F313 R316 L326 A327 I345 F346 C432 L436 I24 A27 A28 Q31 F69 R72 L82 A83 I101 F102 C188 L192 ? 0003677,0003707,0005634,0006355,0008270 Kd=15nM remove_due_to_license_issue EC50=100nM, Kd=15nM P19793 24801499 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4pp5 A 2.0 BS02 2W0 A 1 I268 A271 A272 Q275 F313 R316 L326 A327 V342 C432 L436 I24 A27 A28 Q31 F69 R72 L82 A83 V98 C188 L192 ? 0003677,0003707,0005634,0006355,0008270 Kd=18nM remove_due_to_license_issue Kd=2240nM, EC50=720nM P19793 24801499 500 EDMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4pp7 A 3.4 BS01 2VX A 1 V471 A481 K483 L505 L514 I527 T529 W531 C532 F583 D594 F595 G596 V24 A34 K36 L58 L67 I80 T82 W84 C85 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=62nM P15056 24675381 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 4pp9 A 2.58 BS01 2VT A 1 I369 K387 A389 F435 F437 M438 E439 G441 L489 I14 K32 A34 F80 F82 M83 E84 G86 L134 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P148 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Q08881 24767842 703 SVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4ppa A 2.67 BS01 2VU A 1 K387 A389 K391 F435 F437 M438 E439 G441 L489 D500 K32 A34 K36 F73 F75 M76 E77 G79 L127 D138 D482 A484 R486 N487 D500 P521 D120 A122 R124 N125 D138 P141 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue IC50=210nM, Ki=1.1nM Q08881 24767842 701 SVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4ppb A 2.82 BS01 2VV A 1 A389 K391 F435 E436 F437 M438 E439 G441 L489 A34 K36 F73 E74 F75 M76 E77 G79 L127 D482 A484 R486 N487 D500 P521 D120 A122 R124 N125 D138 P141 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Ki=0.100000nM, IC50=25nM Q08881 24767842 701 SVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4ppc A 2.95 BS01 2VW A 1 A389 K391 F435 E436 F437 M438 E439 G441 L489 D500 A32 K34 F68 E69 F70 M71 E72 G74 L122 D133 D482 A484 R486 N487 D500 P521 D115 A117 R119 N120 D133 P135 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Ki=0.930000nM Q08881 24767842 701 SVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4ppc A 2.95 BS02 2VW B 1 Q367 I369 V377 Q12 I14 V20 D482 A484 R486 N487 D500 P521 D115 A117 R119 N120 D133 P135 2.7.10.2 0004672,0004713,0004715,0005524,0006468 remove_due_to_license_issue Ki=0.930000nM Q08881 24767842 701 SVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4pqa A 1.78 BS01 X8Z A 1 D101 E135 E136 E164 G325 I349 D100 E134 E135 E163 G324 I348 3.5.1.18 0006526,0008270,0008777,0009014,0009085,0009089,0016787,0019877,0046872,0050897 remove_due_to_license_issue Q9JYL2 26186504 401 TETQSLELAKELISRPSVTPDDRDCQKLLAERLHKIGFAAEELHFGDTKNIWLRRGTKAPVVCFAGHTDVVPTGPVEKWDSPPFEPAERDGRLYGRGAADMKTSIACFVTACERFVAKHPNHQGSIALLITSDEEGDALDGTTKVVDVLKARDELIDYCIVGEPTAVDKLGDMIKNGRRGSLSGNLTVKGKQGHIAYPHLAINPVHTFAPALLELTQEVWDEGNEYFPPTSFQISNINGGTGATNVIPGELNVKFNFRFSTESTEAGLKQRVHAILDKHGVQYDLQWSCSGQPFLTQAGKLTDVARAAIAETCGIEAELSTTGGTSDGRFIKAIAQELIELGPSNATIHQINENVRLNDIPKLSAVYEGILARLL 4pqn A 1.71 BS01 2W6 A 1 I369 A389 F435 E436 F437 M438 E439 H440 G441 L489 I13 A31 F77 E78 F79 M80 E81 H82 G83 L131 D482 A484 R486 N487 D500 P521 D124 A126 R128 N129 D142 P146 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=0.7nM remove_due_to_license_issue IC50=55nM, Ki=0.700000nM Q08881 24918870 701 VIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEASVIHRDLAARNCLVGENQVIKVSDFGFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAAI 4prg A 2.9 BS01 072 A 1 L255 E259 F264 H266 A278 R280 I281 C285 R288 I326 Y327 M329 L333 I341 F360 M364 L49 E53 F58 H60 A72 R74 I75 C79 R82 I120 Y121 M123 L127 I135 F154 M158 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 10339548 1 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 4prj A 2.8 BS01 2VU A 1 R137 L139 A160 K162 L194 L210 E211 Y212 A213 G216 R220 L263 A273 D274 R13 L15 A33 K35 L67 L83 E84 Y85 A86 G89 R93 L136 A146 D147 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=72nM O14965 24918870 401 KRQWALEDFEIGRPLGKGNVYLAREKNSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDSTRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKKVIHRDIKPENLLLGSAGELKIADFGWSVCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQDTYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4ps3 A 2.9 BS01 2WH A 1 W812 E814 K833 Y867 I879 I881 V882 K883 D884 A885 M953 I963 D964 W576 E578 K597 Y631 I643 I645 V646 K647 D648 A649 M717 I727 D728 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=2.0nM P48736 24754609 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEWCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 4ps5 A 1.4 BS01 2TA A 1 W81 P82 F83 V87 L92 L94 N140 I146 W40 P41 F42 V46 L51 L53 N99 I105 ? ic50=0.29uM remove_due_to_license_issue Kd=164nM, IC50=290nM O60885 24568369 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4ps7 A 2.69 BS01 2WJ A 1 W812 I831 Y867 I879 V882 I963 D964 W576 I595 Y631 I643 V646 I727 D728 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=39nM P48736 24754609 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEWCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 4ps8 A 2.99 BS01 2WK A 1 W812 K833 D841 Y867 I879 I881 V882 A885 M953 I963 D964 W576 K597 D605 Y631 I643 I645 V646 A649 M717 I727 D728 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Ki=1.000000nM P48736 24754609 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAKQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEWCDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIARAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLVL 4psb A 1.42 BS01 GA3 A 1 V30 F56 Q67 E69 L83 T139 Y142 V30 F56 Q67 E69 L83 T139 Y142 ? 0004864,0005634,0005737,0006952,0009738,0010331,0010427,0038023,0044373 Kd=23uM remove_due_to_license_issue A0A1S3THR8 25004979 201 MVKEFNTQTELSVRLEALWAVLSKDFITVVPKVLPHIVKDVQLIEGDGGVGTILIFNFLPEVSPSYQREEITEFDESSHEIGLQVIEGGYLSQGLSYYKTTFKLSEIEEDKTLVNVKISYDHDSDIEEKVTPTKTSQSTLMYLRRLERYLSN 4psh A 2.6 BS01 ARG A 1 S16 D18 F19 F57 S74 G75 M76 T77 R82 Q123 T126 T127 D164 S15 D17 F18 F56 S73 G74 M75 T76 R81 Q122 T125 T126 D163 ? 0015276,0016020,0034220 remove_due_to_license_issue Q9WZ62 24832102 301 IDEIKSRGYLLVGLSADFPPFEFVDENGNIVGFDVDLAKEIARRLGVELKIVDMTFDGLIPSLLTKKIDVIISGMTITEERKKVVAFSDPYFDAGQVIVVRKDSDFRPKTYEDLVGKTVAVQIGTTGDIEVSKYDGIKVVRFDKFTDAFLELKRGRADAVVLDSATARAFVAKNPDLVISSGVLSSEQYGIAVRKEDTDLLEFINSVLRELKKSPYDVLIEKWFS 4psq B 2.4 BS01 2WL B 1 F36 L37 M73 M88 Y90 G100 R121 F36 L37 M73 M88 Y90 G100 R121 ? 0001654,0002639,0005501,0005515,0005576,0005615,0006094,0007507,0007601,0016918,0019841,0030277,0030324,0032024,0032526,0034632,0034633,0042572,0042593,0048562,0048706,0048738,0048807,0060044,0060059,0060065,0060068,0060157,0060347,0070062 ic50=0.44uM remove_due_to_license_issue IC50=440nM P02753 24835984 201 ERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIVAEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGNDDHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLARQYRLIVHNGYCD 4ptc A 2.711 BS01 2WE A 1 F67 V70 A83 K85 Y134 V135 P136 R141 D200 F32 V35 A48 K50 Y95 V96 P97 R102 D161 D181 K183 N186 D200 S219 D142 K144 N147 D161 S180 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue IC50=1.1nM P49841 25845281 501 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPH 4pte A 2.033 BS01 2WF A 1 F67 V70 A83 K85 Y134 V135 P136 R141 L188 D200 F32 V35 A48 K50 Y93 V94 P95 R100 L147 D159 D181 K183 N186 D200 S219 D140 K142 N145 D159 S178 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=74nM remove_due_to_license_issue IC50=74nM P49841 25845281 501 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDFKNRELQIMRKLDHCNIVRLRYFFYSSDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 4ptg A 2.361 BS01 2WG A 1 F67 V70 A83 K85 Y134 V135 P136 R141 L188 C199 D200 F32 V35 A48 K50 Y93 V94 P95 R100 L147 C158 D159 D181 K183 N186 D200 S219 D140 K142 N145 D159 S178 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=5.9nM remove_due_to_license_issue IC50=5.9nM P49841 25845281 501 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 4pu3 C 3.39 BS01 dna Q 0 V53 T54 T57 R60 D66 V67 Y68 T71 V35 T36 T39 R42 D48 V49 Y50 T53 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 25 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSAGWY 4pu3 C 3.39 BS02 dna P 0 R37 Q44 K55 K56 I59 Y68 R19 Q26 K37 K38 I41 Y50 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 24 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSAGWY 4pu3 D 3.39 BS01 dna Q 0 R37 T43 Q44 K55 K56 Y68 R19 T25 Q26 K37 K38 Y50 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 25 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSAGWY 4pu3 D 3.39 BS02 dna P 0 T54 T57 R60 D66 V67 Y68 T71 T36 T39 R42 D48 V49 Y50 T53 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 24 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSAGWY 4pu4 C 3.786 BS01 dna Q 0 T55 T58 R61 D67 V68 Y69 T72 T36 T39 R42 D48 V49 Y50 T53 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 25 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSA 4pu4 C 3.786 BS02 dna P 0 T44 Q45 K56 K57 I60 K64 Y69 T25 Q26 K37 K38 I41 K45 Y50 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 24 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSA 4pu4 D 3.786 BS01 dna Q 0 R38 T44 Q45 K57 K64 Y69 R19 T25 Q26 K38 K45 Y50 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 25 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSAQTSDTETNGW 4pu4 D 3.786 BS02 dna P 0 V54 T55 T58 R61 D67 V68 Y69 T72 V35 T36 T39 R42 D48 V49 Y50 T53 ? 0003677 remove_due_to_license_issue Q8EIX4 25056321 1 ~ 24 IMASPLNQQSLGLLIKERRKSAALTQDVAAMLCGVTKKTLIRVEKGEDVYISTVFKILDGLGIDIVSAQTSDTETNGW 4puj A 1.42 BS02 CKR A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 R286 D93 Y97 D140 C142 G213 L215 A216 M244 G245 R270 D102 D280 C318 C320 C323 H349 D93 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=35nM remove_due_to_license_issue P28720 24955548 407 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4puk A 1.49 BS02 2WU A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 D93 Y97 D144 C146 G217 L219 A220 M248 G249 D102 D280 C318 C320 C323 H349 D93 D268 C306 C308 C311 H337 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=52.4nM remove_due_to_license_issue P28720 24955548 405 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4pul A 1.654 BS02 2WU A 1 Y106 D156 C158 G229 L231 A232 M260 G261 Y96 D140 C142 G213 L215 A216 M244 G245 N102 D280 C318 C320 C323 H349 N92 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=146.1nM remove_due_to_license_issue P28720 24955548 403 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTNSGGYQVMSLSSLTKQSEEGVTFKSHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4pum A 1.93 BS02 2WU A 1 D102 Y106 N156 C158 G229 A232 M260 G261 D92 Y96 N143 C145 G216 A219 M247 G248 D102 D280 C318 C320 C323 H349 D92 D267 C305 C307 C310 H336 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=188.1nM remove_due_to_license_issue P28720 24955548 404 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHSRHMLSPERSIEIQHLLGSDIVMAFNECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4puz A 2.085 BS01 CG9 A 1 L377 S379 V385 A400 M448 A451 E452 G454 P455 L501 D512 L15 S17 V23 A38 M81 A84 E85 G87 P88 L134 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7.7nM remove_due_to_license_issue IC50=377nM, EC50=125nM P43405 24779514 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDV 4pv0 A 2.0 BS01 CG4 A 1 V385 A400 A451 E452 G454 P455 K458 L501 V21 A36 A82 E83 G85 P86 K89 L132 D494 A496 R498 N499 D512 K533 D125 A127 R129 N130 D143 K164 2.7.10.2 0004672,0004713,0005524,0006468 Kd=4nM remove_due_to_license_issue IC50=0.840000nM, EC50=175nM, Kd=4.0nM P43405 24779514 701 VYLDRKLLTLEDKELGSFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEG 4pv5 A 2.3 BS02 CBW A 1 R123 K151 R111 K139 Q34 E100 H127 E173 Q22 E88 H115 E161 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 remove_due_to_license_issue Q9CPU0 26279158 202 DETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIAT 4pv5 B 2.3 BS02 CBW A 1 R38 N104 R36 N102 Q34 E100 H127 E173 Q32 E98 H125 E171 4.4.1.5 0004462,0005654,0005829,0005886,0006357,0006749,0008270,0009438,0016829,0019243,0030316,0043066,0046872 remove_due_to_license_issue Q9CPU0 26279158 202 EPQPASSGLTDETAFSCCSDPDPSTKDFLLQQTMLRIKDPKKSLDFYTRVLGLTLLQKLDFPAMKFSLYFLAYEDKNDIPKDKSEKTAWTFSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIEILNPNKIATII 4pv7 A 3.24 BS01 CJP A 1 R125 E205 E206 Y547 S630 Y662 Y666 H740 R86 E166 E167 Y508 S591 Y623 Y627 H701 Y547 S630 Y631 D708 H740 Y508 S591 Y592 D669 H701 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 1000 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 4pvo A 1.48 BS04 SVB A 1 F61 Y67 N233 H263 F31 Y36 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue Q9K2N0 25411887 404 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4pvt A 2.0 BS03 S3C A 1 W87 H118 D120 H196 C221 N233 H263 W56 H85 D87 H148 C167 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue Q9K2N0 25411887 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4pvv A 2.5 BS01 HO4 A 1 S8 D12 G48 V49 N52 F102 F116 Q172 D257 S8 D12 G48 V49 N52 F102 F116 Q172 D254 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 ic50=0.33uM remove_due_to_license_issue P9WID5 25259627 401 MTIAVTGSIATDHLMRFPGRFSEQLLPEHLHKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQLASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 4pvx F 2.18 BS03 YS1 F 1 F99 D103 M106 R112 T167 Q171 K200 D243 K257 F92 D96 M99 R105 T160 Q164 K193 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=12nM P14324 29036218 404 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 4pvy F 2.05 BS03 JD1 F 1 F99 D103 R112 T167 E168 Q171 K200 T201 D243 K257 F92 D96 R105 T160 E161 Q164 K193 T194 D236 K250 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=60nM P14324 29036218 404 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4px6 A 1.6 BS01 2X6 A 1 A400 M448 E449 M450 A451 G454 P455 R498 L501 D512 A35 M78 E79 M80 A81 G84 P85 R128 L131 D142 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K159 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4nM remove_due_to_license_issue IC50=307nM P43405 24726806 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNE 4pxi A 3.2 BS01 dna E 0 T42 G44 F48 T38 G40 F44 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 3 ~ 22 LRAEQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDGRGYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAPVRPPLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQE 4pxi A 3.2 BS02 dna F 0 T31 L32 S33 Y47 A52 K53 T27 L28 S29 Y43 A48 K49 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 1 ~ 22 LRAEQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDGRGYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAPVRPPLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQE 4pxi B 3.2 BS01 dna E 0 T31 Y47 A52 K53 T27 Y43 A48 K49 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 3 ~ 22 LRAEQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDGRGYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAGVPVRPPLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTRTLEPAGREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQET 4pxi B 3.2 BS02 dna F 0 A7 T10 T42 K43 G44 A45 F48 H49 A3 T6 T38 K39 G40 A41 F44 H45 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 1 ~ 22 LRAEQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDGRGYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAGVPVRPPLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTRTLEPAGREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQET 4pxi C 3.2 BS01 dna E 0 L5 R6 A7 T10 T42 K43 G44 A45 F48 H49 L1 R2 A3 T6 T38 K39 G40 A41 F44 H45 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 3 ~ 22 LRAEQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDGRGYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAGVVRPPLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTRVVGREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQET 4pxi C 3.2 BS02 dna F 0 L5 R6 T31 L32 Y47 A52 K53 L1 R2 T27 L28 Y43 A48 K49 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 1 ~ 22 LRAEQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDGRGYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAGVVRPPLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTRVVGREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQET 4pxi D 3.2 BS01 dna E 0 T31 L32 K43 Y47 A52 K53 T24 L25 K36 Y40 A45 K46 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 3 ~ 22 EQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAGVPVRLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTRVAGREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQET 4pxi D 3.2 BS02 dna F 0 T42 G44 A45 T35 G37 A38 ? 0003677,0006355 remove_due_to_license_issue O66122 25092919 1 ~ 22 EQTRATIIGAAADLFDRRGYESTTLSEIVAHAGVTKGALYFHFAAKEDLAHAILEIQSRTSRRLAKDLDYSSLEALMRLTFGMARLCVQGPVLRAGLRLATAGVPVRLPHPFTEWREIATSRLLDAVRQSDVHQDIDVDSVAHTLVCSVVGTRVAGREPRRLAEMWYILIRGMVPVTRRARYVTLAARLEQET 4pxm A 1.9 BS02 EST A 1 E353 L387 F404 G521 H524 L525 E47 L81 F98 G202 H205 L206 ? remove_due_to_license_issue IC50=1.3nM, Kd=0.2nM, EC50=0.75nM, Ki=0.21nM P03372 26836308 2000 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYGLLLEMLDAHRL 4py1 A 2.16 BS01 2YK A 1 L903 K910 V911 A928 K930 M978 L1030 G1040 D1041 L15 K22 V23 A40 K42 M90 L142 G152 D153 D1023 A1025 R1027 N1028 D1041 P1064 D135 A137 R139 N140 D153 P176 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P29597 25113930 1201 PTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHSQHYIHRDLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYQG 4py2 A 2.15 BS01 43E A 1 A11 I12 Y14 D51 H53 G54 M227 Y228 V229 W230 D232 I265 F268 H269 A9 I10 Y12 D49 H51 G52 M225 Y226 V227 W228 D230 I263 F266 H267 I12 H20 H23 D51 S128 D131 G150 W230 I265 I10 H18 H21 D49 S126 D129 G148 W228 I263 6.1.1.10 0000166,0004812,0004825,0005524,0005737,0006412,0006418,0006431 ic50=0.272uM remove_due_to_license_issue Q2YQ76 27500735 601 REKYYITTAIAYPNGKPHIGHAYELIATDAMARFQRLNGMDVYFLTGTDEHGIKMLQSARKEGITPRDLADRNTSAFRRMAEVLNSSNDDYIRTSEERHYKASQAIWQAMVANGDIYKGGYAGWYSVRDEAYYGEEETEVRADGVRYGPQGTPVEWVEEESYFFRLSAYQDKLLDLYENNPGFIMPAERRNEIVSFVKSGLKDLSISRTTFDWGIPVPGDEKHVMYVWVDALTNYITALGYPDTTDERWAYWPANAHIIGKDISRFHAVYWPAFLMSAQLPLPKRVFAHGFLFNRIDPFELVERYGLDQLRYFLMREVPFGQDGSYSHEAIVNRTNADLANDLGNLAQRSLSMIAKNCEGKVPQPGAFSEADKAILDQADAALETARKAMDDQALHLALGAIFAVVAEANRYFAGQEPWALRKTDPARMGTVLYVTAEVLRRVGIMVQPFIPQSAEKLLDILAVPADKRQFADVLASPLAGGTDLPAPQPVFPRY 4py4 A 2.76 BS01 XL2 A 1 H1682 G1683 Y1714 Y1721 S1722 Y1727 H70 G71 Y92 Y99 S100 Y105 2.4.2.- 0003950 remove_due_to_license_issue Q460N5 1901 KQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4py4 B 2.76 BS01 XL2 B 1 H1682 G1683 D1685 Y1701 Y1714 S1722 Y1727 H68 G69 D71 Y87 Y94 S102 Y107 2.4.2.- 0003950 remove_due_to_license_issue Q460N5 1901 QNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 4pyn A 1.2 BS01 SAH A 1 K89 G109 Y111 S115 E133 I134 S162 D184 H185 K45 G65 Y67 S71 E89 I90 S118 D140 H141 D184 K187 D212 N213 E242 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 ic50~30uM remove_due_to_license_issue P22734 25084335 300 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSPDK 4pyo A 2.1 BS01 SAH A 1 G109 Y111 S115 E133 I134 A161 S162 D184 H185 W186 G64 Y66 S70 E88 I89 A116 S117 D139 H140 W141 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 ic50~30uM remove_due_to_license_issue P22734 25084335 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 4pyq A 1.39 BS01 2X1 A 1 I134 N135 P136 W186 D188 I89 N90 P91 W141 D143 D184 K187 D212 N213 E242 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 ic50=4.4uM remove_due_to_license_issue P22734 25084335 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 4pyv A 2.65 BS01 2XF A 1 V30 D32 G34 R74 Y75 T77 P111 F117 D215 G217 V34 D36 G38 R80 Y81 T83 P116 F122 D221 G223 D32 S35 N37 W39 Y75 D215 A218 D36 S39 N41 W43 Y81 D221 A224 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=200nM P00797 25050166 1001 LGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4pyx A 1.8 BS02 V90 A 1 N62 H64 N67 Q92 H94 H96 H119 V121 F131 V143 L198 T199 T200 W209 N59 H61 N64 Q89 H91 H93 H116 V118 F127 V139 L194 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=730nM remove_due_to_license_issue Kd=730nM P00918 25358084 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4pyy A 1.75 BS02 V14 A 1 I91 H94 H96 V121 F131 L198 T199 T200 P201 I88 H91 H93 V118 F127 L194 T195 T196 P197 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=59nM remove_due_to_license_issue Kd=60nM P00918 25358084 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4pzh A 1.06 BS02 V13 A 1 H94 H119 V121 F131 L198 T199 T200 P201 P202 H92 H117 V119 F128 L195 T196 T197 P198 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd<10nM remove_due_to_license_issue Kd=17nM P00918 25358084 305 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4pzv A 1.704 BS01 J1D A 1 V45 F58 N60 L75 K79 R87 W94 R97 D100 D102 I103 K115 L116 T117 H120 F128 V45 F58 N60 L75 K79 R87 W94 R97 D100 D102 I103 K115 L116 T117 H120 F128 R87 R97 D100 D102 K382 R417 R87 R97 D100 D102 K374 R409 2.5.1.15,2.7.6.3 0003848,0004156,0005524,0005829,0009396,0016301,0042558,0044237,0046654,0046656,0046872 Kd=2uM remove_due_to_license_issue Q5NGA7 24975935 501 MQYIIGIGTNIGFTIENIHLAITALESQQNIRIIRKASLYSSKAVLKEDAPKEWDIRFLNTAVKISSSLKPDELLVLLKDIELKIGRDLNAPAWSPRVIDLDILAAEDLILETDKLTIPHKELINRSFALAPLLELSKGWHHPKYVEWDLNIRLKELGEIVKLKQTLANTIRMGIVNLSSDGNFDDNQRKLNLDELIQSGAEIIDIGAESTKPISIEEEFNKLDEFLEYFKSQLANLIYKPLVSIDTRKLEVMQKILAKHHDIIWMINDVECNNIEQKAQLIAKYNKKYVIIHNLGITDRNQYLDKENAIDNVCDYIEQKKQILLKHGIAQQNIYFDIGFGFGKKSDTARYLLENIIEIKRRLELKALVGHSRKPSVLGLAKDSNLATLDRATRELSRKLEKLDIDIIRVHKI 4pzw A 1.8 BS01 2X4 A 1 Q73 G74 L91 D93 Y132 F169 I171 W176 D289 G291 T292 Q17 G18 L35 D37 Y76 F113 I115 W120 D227 G229 T230 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D227 T230 3.4.23.46 0004190,0006508,0016020 ic50=0.11uM remove_due_to_license_issue IC50=20nM P56817 24780121 502 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4pzx A 1.8 BS01 2X5 A 1 Q73 G74 D93 Y132 F169 I171 D289 G291 T292 Q17 G18 D37 Y76 F113 I115 D230 G232 T233 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D230 T233 3.4.23.46 0004190,0006508,0016020 ic50=1uM remove_due_to_license_issue IC50=130nM P56817 24780121 502 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4q06 A 1.15 BS02 V90 A 1 N62 H64 Q92 H94 H96 V121 L197 T198 T199 N60 H62 Q90 H92 H94 V119 L195 T196 T197 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=22nM remove_due_to_license_issue Kd=730nM P00918 25358084 304 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKALQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q07 A 1.15 BS02 V14 A 1 N62 Q67 Q92 H94 H96 H119 V121 L134 L197 T198 T199 N59 Q64 Q89 H91 H93 H116 V118 L131 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=7.3nM remove_due_to_license_issue Kd=60nM P00918 25358084 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVEFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKALQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q08 A 1.07 BS02 V90 A 1 N62 H64 S65 H94 H96 H119 V121 L197 T198 T199 N59 H61 S62 H91 H93 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=500nM remove_due_to_license_issue Kd=730nM P00918 25358084 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFKVEFDDSQDKAVLKGGPLDGTYRLTQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDAGKASQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLNECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q09 A 1.2 BS02 V14 A 1 K67 H94 H96 V121 L197 T198 T199 P200 K64 H91 H93 V118 L194 T195 T196 P197 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=6.7nM remove_due_to_license_issue Kd=60nM P00918 25358084 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFKVEFDDSQDKAVLKGGPLDGTYRLTQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDAGKASQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLNECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q0a C 1.9 BS02 4OA C 1 Y175 L261 S303 S306 W314 H333 Y21 L47 S89 S92 W100 H119 ? 0003677,0004879,0005634,0006355 Kd=0.33uM remove_due_to_license_issue Q9PTN2 24818857 501 MLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEVS 4q0a C 1.9 BS03 4OA C 2 D181 R184 F185 S263 Q267 D27 R30 F31 S49 Q53 ? 0003677,0004879,0005634,0006355 Kd=0.33uM remove_due_to_license_issue Q9PTN2 24818857 502 MLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEVS 4q0k A 1.34 BS01 GA3 A 1 L34 F56 Q68 F103 S140 T141 L34 F56 Q68 F103 S140 T141 ? 0004864,0005634,0005737,0006952,0009738,0009740,0010427,0038023 Kd=13.4uM remove_due_to_license_issue G7J032 25004979 201 MIKEFNTQTTLNVGLEALWAAQSKDITLVVPKVLPNIVKDVQVIEGDGGVGTKLIFNFLPGIAPVNYQREVITEYDELSHTIGLQVVEGGYLNQGLSYYKTTFQFSAISENKTLVNVKISYDHESELIEEKVKPTKTSESTLFYLGQLEKFLLN 4q0l A 2.0 BS02 V14 A 1 K69 Q89 H91 H93 H117 V119 S133 L197 T198 T199 K67 Q87 H89 H91 H115 V117 S131 L195 T196 T197 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=20nM remove_due_to_license_issue Kd=5.3nM O43570 25358084 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4q15 A 2.35 BS02 HFG A 1 F335 E338 P358 T359 E361 R390 F454 T478 H480 W509 G510 F79 E82 P102 T103 E105 R134 F198 T222 H224 W253 G254 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=275nM remove_due_to_license_issue Q8I5R7 27798837 803 ILGITSKKIENFSDWYTQVIVKSELIEYYDISGCYILRPAAYYIWECVQAFFNKEIKKLNVENSYFPLFVTKNKLEKGFSPEVAWVTKYGDSNLPEEIAIRPTSETIMYSVFPKWIRSYRDLPLKLNQWNTVVRWEFKQPTPFIRTREFLWQEGHTAHKNEEEAVKLVFDILDLYRRWYEEYLAVPIIKGIKSEGEKFGGANFTSTAEAFISENGRAIQAATSHYLGTNFAKMFKIEFEDENEVKQYVHQTSWGCTTRSIGIMIMTHGDDKGLVLPPNVSKYKVVIVPIFYTDENAIHSYCKDIEKILKNAQINCVYDDRASYSPGYKFNHWELRGIPIRIEVGPKDLQNNSCVIVRRDNNEKCNVKKESVLLETQQMLVDIHKNLFLKAKKKLDDSIVQVTSFSEVMNALNKKKMVLAPWCEAMKPLCIPLDQPPMPPNMKCFWSGKPAKRWCLFGRSY 4q18 A 2.0 BS01 2XJ A 1 E53 V55 M85 Y86 P89 F96 Q97 F137 S144 E33 V35 M55 Y56 P59 F66 Q67 F107 S114 E53 R128 E33 R98 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=735nM remove_due_to_license_issue IC50=754nM, Ki=735nM P27707 25341194 301 IKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q18 A 2.0 BS02 2XJ A 2 I30 S59 Y86 E196 G199 I200 P201 Y204 I10 S39 Y56 E166 G169 I170 P171 Y174 E53 R128 E33 R98 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=735nM remove_due_to_license_issue IC50=754nM, Ki=735nM P27707 25341194 302 IKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q19 A 2.09 BS01 2XL A 1 E53 V55 Y86 P89 Q97 F137 Y204 E33 V35 Y55 P58 Q66 F105 Y172 E53 R128 E33 R96 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=8.9nM remove_due_to_license_issue IC50=19nM, Ki=8.9nM P27707 25341194 301 IKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1a A 1.9 BS01 2XZ A 1 E53 V55 L82 Y86 P89 F96 Q97 D133 F137 S146 Y204 E34 V36 L52 Y56 P59 F66 Q67 D103 F107 S116 Y174 E53 R128 E34 R98 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=0.5nM remove_due_to_license_issue IC50=1.2nM, Ki=0.500000nM P27707 25341194 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1b A 2.15 BS01 2Y0 A 1 E53 V55 L82 M85 Y86 Q97 D133 F137 N140 S144 Y204 E34 V36 L51 M54 Y55 Q66 D102 F106 N109 S113 Y173 E53 R128 E34 R97 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=1.9nM remove_due_to_license_issue IC50=12nM, Ki=1.9nM P27707 25341194 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1c A 2.0 BS01 2XM A 1 E53 V55 Y86 P89 F96 Q97 D133 F137 L141 S144 S146 Y204 E34 V36 Y56 P59 F66 Q67 D103 F107 L111 S114 S116 Y174 E53 R128 E34 R98 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=2nM remove_due_to_license_issue IC50=0.900000nM, Ki=2.0nM P27707 25341194 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1d A 2.0 BS01 2Y1 A 1 E53 V55 L82 Y86 P89 Q97 D133 F137 L141 S144 Y204 E34 V36 L53 Y57 P60 Q68 D104 F108 L112 S115 Y175 E53 R128 E34 R99 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=16.6nM remove_due_to_license_issue IC50=10.0nM, Ki=17nM P27707 25341194 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1e A 1.85 BS01 2Y8 A 1 E53 M85 Q97 D133 F137 L141 S144 Y204 E34 M56 Q68 D104 F108 L112 S115 Y175 E53 R128 E34 R99 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=6.8nM remove_due_to_license_issue P27707 25341194 301 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1f A 2.1 BS02 2XN A 1 E53 V55 M85 Y86 P89 Q97 D133 F137 N140 S144 Y204 K207 E34 V36 M56 Y57 P60 Q68 D104 F108 N111 S115 Y175 K178 E53 R128 E34 R99 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 Ki=9.2nM remove_due_to_license_issue Ki=9.2nM, IC50=28nM P27707 25341194 302 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNLTMEQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESESMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 4q1n A 2.09 BS01 2Y9 A 1 D32 G34 R74 Y75 S76 T77 P111 A115 F117 V120 I130 D215 G217 A218 I291 D38 G40 R82 Y83 S84 T85 P118 A122 F124 V127 I137 D222 G224 A225 I301 D32 S35 N37 W39 Y75 D215 A218 D38 S41 N43 W45 Y83 D222 A225 3.4.23.15 0004190,0006508 ic50=0.2nM remove_due_to_license_issue IC50=0.200000nM P00797 25050166 404 LTLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4q1s a 2.6 BS01 2YD H 1 L154 K157 N179 L154 K157 N179 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0034515,0043161,0043248,0051603 remove_due_to_license_issue P30657 25038530 301 TQQPIVTGTSVISMKYDNGVIIAADNLGSYGSLLRFNGVERLIPVGDNTVVGISGDISDMQHIERLLKDLVTENAYDNPLADAEEALEPSYIFEYLATVMYQRRSKMNPLWNAIIVAGVQSNGDQFLRYVNLLGVTYSSPTLATGFGAHMANPLLRKVVDRESDIPKTTVQVAEEAIVNAMRVLYYRDARSSRNFSLAIIDKNTGLTFKKNLQVENMKWDFAKDIKGYGTQKI 4q1s H 2.6 BS01 2YD H 1 V137 S140 H141 D157 V137 S140 H141 D157 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25038530 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4q1w A 1.85 BS01 017 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=2pM remove_due_to_license_issue P04585 25091085 104 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLMTQIGCTLNF 4q1w B 1.85 BS01 017 A 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 25091085 104 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLMTQIGCTLNF 4q1x A 1.9 BS01 017 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=7pM remove_due_to_license_issue P04585 25091085 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTILEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4q1x B 1.9 BS01 017 A 1 D25 G27 A28 D30 I50 P81 V82 D25 G27 A28 D30 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 25091085 101 PQITLWKRPLVTIRIGGQLKEALLDTGADDTILEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4q1y A 1.5 BS01 017 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=45pM remove_due_to_license_issue P04585 25091085 106 PQITLWKRPLVTIRIGGQLKEALLDTGADDTIFEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4q1y B 1.5 BS01 017 A 1 D25 A28 D30 I50 P81 D25 A28 D30 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 25091085 106 PQITLWKRPLVTIRIGGQLKEALLDTGADDTIFEEMNLPGKWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4q2k A 2.2 BS01 5BF A 1 C191 S195 S214 W215 G216 S217 S218 C177 S181 S200 W201 G202 S203 S204 H57 D102 M192 G193 D194 S195 G196 H52 D90 M178 G179 D180 S181 G182 3.4.21.1 0004252,0005515,0005576,0006508,0007586,0008236,0097180,0097655 remove_due_to_license_issue P00766 24903745 301 CGVPAIQPVLIVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGVTTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKNDITLLKLSTAASFSQTVSAVCLPSASDDFAAGTTCVTTGWGLTRYANTPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 4q2k A 2.2 BS02 5BF D 1 S186 T222 S223 S172 T208 S209 H57 D102 M192 G193 D194 S195 G196 H52 D90 M178 G179 D180 S181 G182 3.4.21.1 0004252,0005515,0005576,0006508,0007586,0008236,0097180,0097655 remove_due_to_license_issue P00766 24903745 301 CGVPAIQPVLIVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGVTTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKNDITLLKLSTAASFSQTVSAVCLPSASDDFAAGTTCVTTGWGLTRYANTPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 4q3q A 2.001 BS03 ABH A 1 D154 H156 D158 S167 H171 D213 D262 E307 D128 H130 D132 S141 H145 D187 D236 E281 H131 D154 H156 D158 H171 D262 D264 E307 H105 D128 H130 D132 H145 D236 D238 E281 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=1.3uM remove_due_to_license_issue Q6WVP6 25007099 405 KLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3r A 2.169 BS03 XA2 A 1 H131 D154 H156 D158 S167 H171 D213 D262 E307 H105 D128 H130 D132 S141 H145 D187 D236 E281 H131 D154 H156 D158 H171 D262 D264 E307 H105 D128 H130 D132 H145 D236 D238 E281 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.54uM remove_due_to_license_issue Q6WVP6 25007099 407 KLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQT 4q3r B 2.169 BS03 XA2 B 1 D154 H156 D158 N160 S167 H171 D213 D262 E307 D127 H129 D131 N133 S140 H144 D186 D235 E280 H131 D154 H156 D158 H171 D262 D264 E307 H104 D127 H129 D131 H144 D235 D237 E280 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.54uM remove_due_to_license_issue Q6WVP6 25007099 409 KLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHM 4q3s A 2.11 BS03 X7A A 1 H131 D154 H156 D158 S167 H171 D211 D213 D262 E307 H105 D128 H130 D132 S141 H145 D185 D187 D236 E281 H131 D154 H156 D158 H171 D262 D264 E307 H105 D128 H130 D132 H145 D236 D238 E281 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.26uM remove_due_to_license_issue Q6WVP6 25007099 403 KLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3s C 2.11 BS03 X7A C 1 D154 H156 D158 N160 S167 H171 D211 D213 D262 E307 D125 H127 D129 N131 S138 H142 D182 D184 D233 E278 H131 D154 H156 D158 H171 D262 D264 E307 H102 D125 H127 D129 H142 D233 D235 E278 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.26uM remove_due_to_license_issue Q6WVP6 25007099 403 KLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3t A 2.142 BS03 HAR A 1 D154 H156 D158 N160 H171 D213 D262 E307 D129 H131 D133 N135 H146 D188 D237 E282 H131 D154 H156 D158 H171 D262 D264 E307 H106 D129 H131 D133 H146 D237 D239 E282 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.33uM remove_due_to_license_issue Q6WVP6 25007099 405 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q3u A 2.5 BS03 NNH A 1 D154 H156 D158 S167 H171 D213 T276 D129 H131 D133 S142 H146 D188 T251 H131 D154 H156 D158 H171 D262 D264 E307 H106 D129 H131 D133 H146 D237 D239 E282 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 Kd=0.36uM remove_due_to_license_issue Q6WVP6 25007099 405 PKLLYTSANFLGIPTNRGQPKIGTYQGPELIRKSNFFQLVAEDGIQLTDCGDIIPVELNEAEDPQRFGMKWSRSFSLTTLRIAERVEELMKQSNKSTPLVIVGGDHSMATGTILGHAEAKPDLCVLWIDAHGDINTPLNSASGNMHGMPLSFLVKELQDQIPWLDDFEGIKPCLNASNIAYIGLRDLDAHETHDIRKHGIAYFTMLDVDRMGIEAVIKEALLAVNPRLEKAIHLSFDIDALDPLVAPSTGTAVPGGLTLREGLRICEEVSATGKLSVVELAELNPLLGSQEDVLKTQSSAVHILRACLGHCRSGHLPFKVRNLTDQGIMSRAAHMQ 4q46 A 1.8 BS01 GDP A 1 F327 R334 W359 E363 F406 S431 M433 F7 R14 W39 E43 F86 S111 M113 ? 0033650 remove_due_to_license_issue A0A0J9X1Z6 25691568 501 IRQRQRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSKMKLEKLLINSAKKEDMRDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSSDLFDQWGYEESPKASELHGINESMNASDYTLKGVVVTKN 4q46 A 1.8 BS02 GDP B 1 R326 R368 R6 R48 ? 0033650 remove_due_to_license_issue A0A0J9X1Z6 25691568 501 IRQRQRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSKMKLEKLLINSAKKEDMRDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSSDLFDQWGYEESPKASELHGINESMNASDYTLKGVVVTKN 4q4e A 1.9 BS02 BB2 A 1 M260 G261 A262 E264 H297 E298 H301 E320 Y381 R783 R825 M256 G257 A258 E260 H293 E294 H297 E316 Y377 R779 R821 E264 H297 E298 H301 E320 N373 Y381 E260 H293 E294 H297 E316 N369 Y377 3.4.11.2 0004177,0005515,0005886,0006508,0008237,0008270,0042802,0046872 ic50=0.19uM remove_due_to_license_issue P04825 25644575 902 PQAKYRHDYRAPDYQITDIDLTFDLDAQKTVVTAVSQAVRHGASDAPLRLNGEDLKLVSVHINDEPWTAWKEEEGALVISNLPERFTLKIINEISPAANTALEGLYQSGDALCTQCEAEGFRHITYYLDRPDVLARFTTKIIADKIKYPFLLSNGNRVAQGELENGRHWVQWQDPFPKPCYLFALVAGDFDVLRDTFTTRSGREVALELYVDRGNLDRAPWAMTSLKNSMKWDEERFGLEYDLDIYMIVAVDFFNMGAMENKGLNIFNSKYVLARTDTATDKDYLDIERVIGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSSDLGSRAVNRINNVRTMRGLQFAEDASPMAHPIRPDMVIEMNNFYTLTVYEKGAEVIRMIHTLLGEENFQKGMQLYFERHDGSAATCDDFVQAMEDASNVDLSHFRRWYSQSGTPIVTVKDDYNPETEQYTLTISQRTPATPDQAEKQPLHIPFAIELYDNEGKVIPLQKGGHPVNSVLNVTQAEQTFVFDNVYFQPVPALLCEFSAPVKLEYKWSDQQLTFLMRHARNDFSRWDAAQSLLATYIKLNVARHQQGQPLSLPVHVADAFRAVLLDEKIDPALAAEILTLPSVNEMAELFDIIDPIAIAEVREALTRTLATELADELLAIYNANYQSEYRVEHEDIAKRTLRNACLRFLAFGETHLADVLVSKQFHEANNMTDALAALSAAVAAQLPCRDALMQEYDDKWHQNGLVMDKWFILQATSPAANVLETVRGLLQHRSFTMSNPNRIRSLIGAFAGSNPAAFHAEDGSGYLFLVEMLTDLNSRNPQVASRLIEPLIRLKRYDAKRQEKMRAALEQLKGLENLSGDLYEKITKALA 4q4o A 1.35 BS02 2YM A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 D92 Y96 D141 C143 G214 L216 A217 M245 G246 D102 D280 C318 C320 C323 H349 D92 D265 C303 C305 C308 H334 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=34.3nM remove_due_to_license_issue P28720 24960372 406 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4q4p A 1.539 BS02 2YO A 1 Y106 D156 C158 G229 G230 L231 A232 M260 G261 L283 R286 Y96 D137 C139 G210 G211 L212 A213 M241 G242 L264 R267 D102 D280 C318 C320 C323 H349 D92 D261 C299 C301 C304 H330 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=407.4nM remove_due_to_license_issue P28720 24960372 405 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSTKQSEEGVTFKHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4q4q A 1.41 BS02 SAQ A 1 Y106 D156 C158 G229 G230 L231 A232 M260 G261 Y97 D141 C143 G214 G215 L216 A217 M245 G246 D102 D280 C318 C320 C323 H349 D93 D265 C303 C305 C308 H334 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=1638.9nM remove_due_to_license_issue P28720 24960372 406 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4q4r A 1.448 BS02 SQO A 1 Y106 D156 C158 G229 G230 L231 A232 M260 G261 R286 Y96 D137 C139 G210 G211 L212 A213 M241 G242 R267 D102 D280 C318 C320 C323 H349 D92 D261 C299 C301 C304 H330 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=369.2nM remove_due_to_license_issue P28720 24960372 405 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSTKQSEEGVTFKHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4q4s A 1.249 BS02 S98 A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 D92 Y96 D139 C141 G212 L214 A215 M243 G244 D102 D280 C318 C320 C323 H349 D92 D263 C301 C303 C306 H332 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=111.6nM remove_due_to_license_issue Ki=3.5nM P28720 24960372 406 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4q6d A 1.12 BS02 WW3 A 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.0435uM remove_due_to_license_issue P00918 25353386 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q6e A 1.12 BS02 KR5 A 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.667uM remove_due_to_license_issue P00918 25353386 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q6r A 2.4 BS01 30J A 1 L173 I386 Y387 A388 L63 I276 Y277 A278 4.1.2.27 0016830,0019752,0030170 ic50=0.21uM remove_due_to_license_issue IC50=210nM O95470 24809814 903 EYVKALPSQGLSSSAVLEKLKEYSSMDAFWQEGRASGTVYSGEEKLTELLVKAYGDFAWSNPLHPDIFPGLRKIEAEIVRIACSLFNGGPDSCGCVTSGGTESILMACKAYRDLAFEKGIKTPEIVAPQSAHAAFNKAASYFGMKIVRVPLTKMMEVDVRAMRRAISRNTAMLVCSTPQFPHGVIDPVPEVAKLAVKYKIPLHVDACLGGFLIVFMEKAGYPLEHPFDFRVKGVTSISADTHKYGYAPKGSSLVLYSDKKYRNYQFFVDTDWQGGIYASPTIAGSRPGGISAACWAALMHFGENGYVEATKQIIKTARFLKSELENIKGIFVFGNPQLSVIALGSRDFDIYRLSNLMTAKGWNLNQLQFPPSIHFCITLLHARKRVAIQFLKDIRESVTQIMKNPKAKTTGMGAIYGMAQTTVDRNMVAELSSVFLDSLYSTD 4q6r A 2.4 BS02 30J B 1 V538 L541 S542 F545 V428 L431 S432 F435 4.1.2.27 0016830,0019752,0030170 ic50=0.21uM remove_due_to_license_issue IC50=210nM O95470 24809814 602 EYVKALPSQGLSSSAVLEKLKEYSSMDAFWQEGRASGTVYSGEEKLTELLVKAYGDFAWSNPLHPDIFPGLRKIEAEIVRIACSLFNGGPDSCGCVTSGGTESILMACKAYRDLAFEKGIKTPEIVAPQSAHAAFNKAASYFGMKIVRVPLTKMMEVDVRAMRRAISRNTAMLVCSTPQFPHGVIDPVPEVAKLAVKYKIPLHVDACLGGFLIVFMEKAGYPLEHPFDFRVKGVTSISADTHKYGYAPKGSSLVLYSDKKYRNYQFFVDTDWQGGIYASPTIAGSRPGGISAACWAALMHFGENGYVEATKQIIKTARFLKSELENIKGIFVFGNPQLSVIALGSRDFDIYRLSNLMTAKGWNLNQLQFPPSIHFCITLLHARKRVAIQFLKDIRESVTQIMKNPKAKTTGMGAIYGMAQTTVDRNMVAELSSVFLDSLYSTD 4q6r B 2.4 BS01 30J A 1 V538 L541 S542 F545 V429 L432 S433 F436 4.1.2.27 0016830,0019752,0030170 ic50=0.21uM remove_due_to_license_issue IC50=210nM O95470 24809814 903 KEYVKALPSQGLSSSAVLEKLKEYSSMDAFWQEGRASGTVYSGEEKLTELLVKAYGDFAWSNPLHPDIFPGLRKIEAEIVRIACSLFNGGPDSCGCVTSGGTESILMACKAYRDLAFEKGIKTPEIVAPQSAHAAFNKAASYFGMKIVRVPLTKMMEVDVRAMRRAISRNTAMLVCSTPQFPHGVIDPVPEVAKLAVKYKIPLHVDACLGGFLIVFMEKAGYPLEHPFDFRVKGVTSISADTHKYGYAPKGSSLVLYSDKKYRNYQFFVDTDWQGGIYASPTIAGSRPGGISAACWAALMHFGENGYVEATKQIIKTARFLKSELENIKGIFVFGNPQLSVIALGSRDFDIYRLSNLMTAKGWNLNQLQFPPSIHFCITLLHARKRVAIQFLKDIRESVTQIMKNPKAKTTGMGAIYGMAQTTVDRNMVAELSSVFLDSLYSTD 4q6r B 2.4 BS03 30J B 1 L173 I386 Y387 A388 L64 I277 Y278 A279 4.1.2.27 0016830,0019752,0030170 ic50=0.21uM remove_due_to_license_issue IC50=210nM O95470 24809814 602 KEYVKALPSQGLSSSAVLEKLKEYSSMDAFWQEGRASGTVYSGEEKLTELLVKAYGDFAWSNPLHPDIFPGLRKIEAEIVRIACSLFNGGPDSCGCVTSGGTESILMACKAYRDLAFEKGIKTPEIVAPQSAHAAFNKAASYFGMKIVRVPLTKMMEVDVRAMRRAISRNTAMLVCSTPQFPHGVIDPVPEVAKLAVKYKIPLHVDACLGGFLIVFMEKAGYPLEHPFDFRVKGVTSISADTHKYGYAPKGSSLVLYSDKKYRNYQFFVDTDWQGGIYASPTIAGSRPGGISAACWAALMHFGENGYVEATKQIIKTARFLKSELENIKGIFVFGNPQLSVIALGSRDFDIYRLSNLMTAKGWNLNQLQFPPSIHFCITLLHARKRVAIQFLKDIRESVTQIMKNPKAKTTGMGAIYGMAQTTVDRNMVAELSSVFLDSLYSTD 4q7p A 1.65 BS02 3MH A 1 H94 H96 H119 T199 T200 H91 H93 H116 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=48uM remove_due_to_license_issue Ki=48000nM P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q7s A 1.8 BS02 2YU A 1 H94 H96 T199 T200 H91 H93 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=38uM remove_due_to_license_issue Ki=38000nM P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q7v A 1.6 BS02 5MH A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=260uM remove_due_to_license_issue Ki=260000nM P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q7w A 1.45 BS02 6MH A 1 H94 H119 V121 L198 T199 H91 H116 V118 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2300uM remove_due_to_license_issue Ki=2300000nM P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q81 A 1.55 BS02 7MH A 1 H94 H96 H119 L198 T199 T200 H91 H93 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=950uM remove_due_to_license_issue Ki=950000nM P00918 25116076 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q83 A 1.55 BS02 3FH A 1 H94 H96 H119 V121 L198 T199 T200 H91 H93 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=64uM remove_due_to_license_issue Ki=64000nM P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q87 A 1.55 BS02 4FH A 1 H94 H96 L198 T199 T200 H91 H93 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=14uM remove_due_to_license_issue Ki=14000nM P00918 25116076 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q8x A 1.55 BS02 7FH A 1 V121 L198 T200 V118 L194 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=270uM remove_due_to_license_issue Ki=270000nM P00918 25116076 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q8y A 1.45 BS02 HQT A 1 H94 H96 V121 L141 L198 T199 T200 H91 H93 V118 L137 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2300uM remove_due_to_license_issue Ki=2300000nM P00918 25116076 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q90 A 1.54 BS02 4H2 A 1 H94 L198 T200 H91 L194 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7mM remove_due_to_license_issue P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q93 A 2.1 BS01 STL A 1 Y39 G41 L72 H77 Y166 Q170 D173 Y36 G38 L69 H74 Y163 Q167 D170 6.1.1.1 0000166,0004812,0004831,0005524,0006418,0006437 remove_due_to_license_issue P54577 25533949 401 APSPEEKLHLITRNLQEVLGEEKLKEILKERELKIYWGTATTGKPHVAYFVPMSKIADFLKAGCEVTILFADLHAYLDNMKAPWELLELRVSYYENVIKAMLESIGVPLEKLKFIKGTDYQLSKEYTLDVYRLSSVVTQHDSKKAGAEVVKQVEHPLLSGLLYPGLQALDEEYLKVDAQFGGIDQRKIFTFAEKYLPALGYSKRVHLMNPMVPGLTGSKIDLLDRKEDVKKKLKKAFCEPGNVENNGVLSFIKHVLFPLKSEFVILRDEKWGGNKTYTAYVDLEKDFAAEVVHPGDLKNSVEVALNKLLDPIREKFNTPALKKLASAAYP 4q99 A 1.5 BS02 HT4 A 1 H94 V121 T199 T200 W209 H91 V118 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.52uM remove_due_to_license_issue P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q9m A 2.06 BS01 2ZW A 1 M49 Q53 I87 P91 Y98 V99 L102 A129 F143 M33 Q37 I71 P75 Y82 V83 L86 A113 F127 D28 H45 L139 D12 H29 L123 2.5.1.- 0000287,0004659,0005829,0008834,0016094,0016740,0016765,0030145,0045547,0046872 Kd=66nM remove_due_to_license_issue Q8DRB3 25287857 301 TQVPAHIGIIMDGNGRWAKKRMQPRVFGHKAGMEALQTVTKAANKLGVKVITVYAFSTENWTRPDQEVKFIMNLPVEFYDNYVPELHANNVKIQMIGETDRLPKQTFEALTKAEELTKNNTGLILNFALNYGGRAEITQALKLISQDVLDAKINPGDITEELIGNYLFTQHLPKDLRDPDLIIRTSGELRLSNFLPWQGAYSELYFTDTLWPDFDEAALQEAILAYNRRH 4q9o A 2.2 BS01 2ZW A 1 M49 L52 Q53 I87 P91 Y95 Y98 V99 L102 A129 F143 M43 L46 Q47 I81 P85 Y89 Y92 V93 L96 A123 F137 D28 H45 L139 D22 H39 L133 2.5.1.- 0000287,0004659,0005829,0008834,0016094,0016740,0016765,0030145,0045547,0046872 Kd=1.7uM remove_due_to_license_issue Q8DRB3 25287857 301 GSMAVEVEVPTQVPAHIGIIMDGNGRWAKKRMQPRVFGHKAGMEALQTVTKAANKLGVKVITVYAFSTENWTRPDQEVKFIMNLPVEFYDNYVPELHANNVKIQMIGETDRLPKQTFEALTKAEELTKNNTGLILNFALNYGGRAEITQALKLISQDVLDAKINPGDITEELIGNYLFTQHLPKDLRDPDLIIRTSGELRLSNFLPWQGAYSELYFTDTLWPDFDEAALQEAILAYNRRH 4q9s A 2.07 BS01 30G A 1 A452 M499 E500 C502 E506 L553 A37 M84 E85 C87 E91 L138 D546 A548 R550 N551 D564 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 ic50=156uM remove_due_to_license_issue IC50=156000nM Q05397 25000588 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQ 4q9y A 1.55 BS02 M3T A 1 H94 V121 L198 T199 T200 H91 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.1uM remove_due_to_license_issue P00918 25116076 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4q9z A 2.6 BS01 PZW A 1 L386 F391 V394 A407 M458 E459 L461 D508 L511 D522 F664 L12 F17 V20 A33 M84 E85 L87 D134 L137 D148 F290 D504 K506 D508 N509 D522 T542 D130 K132 D134 N135 D148 T168 2.7.11.13 0004672,0004674,0004697,0005524,0006468 remove_due_to_license_issue IC50=55nM Q04759 25000588 801 LKIEDFELHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNEFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPPFRPKVKSPFDCSNFDKEFLNEKPRLSFADRALINSMDQNMFRNFSFMNPGMERLISH 4qaa A 2.7 BS01 KK1 A 1 Y89 K139 W143 T144 Y192 Y97 K147 W151 T152 Y194 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 DYKDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVEAYEDVEVSLNFRKKG 4qaa A 2.7 BS02 KK1 E 1 W53 L112 M114 W61 L120 M122 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 DYKDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVEAYEDVEVSLNFRKKG 4qaa B 2.7 BS01 KK1 B 1 Y89 K139 W143 V183 Y192 Y95 K145 W149 V189 Y194 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 KDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTPEAYEDVEVSLNFRKKG 4qab A 2.984 BS01 KK2 A 1 Y89 W143 Y185 C188 Y192 Y97 W151 Y188 C191 Y195 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 DYKDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qab A 2.984 BS02 KK2 E 1 W53 M114 Y164 W61 M122 Y167 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 DYKDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qab B 2.984 BS01 KK2 A 1 W53 R104 M114 W57 R108 M118 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 DDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qab B 2.984 BS02 KK2 B 1 Y89 W143 Y185 Y192 Y93 W147 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 remove_due_to_license_issue P58154 25006260 301 DDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qac A 2.1 BS01 KK3 A 1 Y89 S142 W143 Y185 Y192 Y97 S150 W151 Y189 Y196 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.0004uM remove_due_to_license_issue P58154 25006260 304 DYKDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qac A 2.1 BS02 KK3 E 1 W53 R104 M114 Y164 W61 R112 M122 Y168 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.0004uM remove_due_to_license_issue P58154 25006260 302 DYKDDDDKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qac B 2.1 BS01 KK3 A 1 W53 R104 M114 Y164 W55 R106 M116 Y164 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.0004uM remove_due_to_license_issue P58154 25006260 304 DKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qac B 2.1 BS02 KK3 B 1 Y89 W143 Y185 Y192 Y91 W145 Y185 Y192 ? 0004888,0005216,0005230,0005576,0006811,0016020,0034220,0043083,0045202,0098794 Kd=0.0004uM remove_due_to_license_issue P58154 25006260 303 DKLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4qag A 1.712 BS03 F95 A 1 D443 E478 D498 S499 H539 D19 E54 D74 S75 H115 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0004523 ic50=4.8uM remove_due_to_license_issue P03366 24840303 603 LWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIR 4qb3 A 0.94 BS01 30M A 1 W81 F83 L94 N140 D144 D145 I146 W40 F42 L53 N99 D103 D104 I105 ? Kd=3.4uM remove_due_to_license_issue Kd=3400nM, Ki=17200nM O60885 24954007 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4qbb A 1.6 BS01 E69 A 1 N46 D49 C51 W52 E96 G97 G98 E147 H148 D164 N18 D21 C23 W24 E68 G69 G70 E119 H120 D136 N46 C51 H148 D163 N18 C23 H120 D135 2.7.7.48,3.4.22.28,3.4.22.46,3.6.1.15 0004197,0016032,0019082 remove_due_to_license_issue P03305 25240326 202 MELTLYNGEKKTFYSRPNNHDNCWLNAILQLFRYVEEPFFDWVYSSPENLTLEAIKQLEDLTGLELHEGGPPALVIWNIKHLLHTGIGTASRPSEVCVVDGTDMCLADFHAGIFLKGQEHAVFACVTSNGWYAIDDEDFYPWTPDPSDVLVFVPYDQEP 4qd6 A 2.45 BS01 30T A 1 A389 V419 F435 F437 M438 E439 H440 G441 L489 A35 V60 F76 F78 M79 E80 H81 G82 L130 D482 A484 R486 N487 D500 P521 D123 A125 R127 N128 D141 P146 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=2.3nM remove_due_to_license_issue Ki=2.3nM Q08881 25455497 701 GSVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTISEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4qd6 A 2.45 BS02 30T B 1 I369 V377 I15 V23 D482 A484 R486 N487 D500 P521 D123 A125 R127 N128 D141 P146 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=2.3nM remove_due_to_license_issue Ki=2.3nM Q08881 25455497 701 GSVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTISEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 4qdk A 1.7 BS01 SAH A 1 F16 Y28 H44 G70 C71 G72 D91 I92 D120 L121 L134 Y140 F10 Y22 H38 G64 C65 G66 D85 I86 D114 L115 L128 Y134 2.1.1.11 0008168,0015979,0015995,0032259,0036068,0046406 remove_due_to_license_issue Q55467 25077963 301 DDKTIVRDYFNSTGFDRWRRIYGDGQVNFVQKDIRVGHQQTVDSVVAWLVADGNLPGLLVCDAGCGVGSLSIPLAQAGALVYGSDISEKMVGEAQQKAQEVLAYGNQPTFMTQDLAQLGGKYDTVICLDVLIHYPTEEASAMISHLASLADRRLILSFAPKTLGLTVLKKIGGLFPGRAYQHKEADIRKILGDNGFSIARTGMTSTRFYYSRILEAVRS 4qei A 2.875 BS01 rna C 0 D72 R76 Q82 G88 G89 S91 I280 D545 Q547 R548 L567 S568 N570 S596 S597 S599 G601 R602 Y604 A605 R606 E609 T617 D619 F620 T631 R633 M638 Q640 F672 Q675 D9 R13 Q19 G25 G26 S28 I175 D427 Q429 R430 L449 S450 N452 S478 S479 S481 G483 R484 Y486 A487 R488 E491 T499 D501 F502 T513 R515 M520 Q522 F554 Q557 2.7.7.-,6.1.1.14 0000166,0004812,0004820,0005524,0005737,0006418,0006426 remove_due_to_license_issue P41250 26797133 1 ~ 71 IVDRAKMGDTLKRRFFYDQAFAIYGGVSGLYDFGPVGCALKNNIIQTWRQHFIQEEQILEIDCTMLTPEPVLKTSGHVDKFADFMVKDVKNGERFRADHLLKAHLQKLQQELADLFVNFNLMFKTFIGPGGNMPGYLRPETAQGIFLNFKRLLEFNQGKLPFAAAQIGNSFRNEISPRSGLIRVREFTMAEIEHFVDPSEKDHPKFQNVADLHLYLYSAKAQVSGQSARKMRLGDAVEQGVINNTVLGYFIGRIYLYLTKVGISPDKLRFRQHMEDCWDAESKTSYGWIEIVGCADRSCYDLSCHARATKVPLVAEKPLKEPKTVNVVQFEPSKGAIGKAYKKDAKLVMEYLAICDECYITEMEMLLNEKGEFTIETQLTKDMINVKRFQKTLYVEEVVPNVIEPSFGLGRIMYTVFEHTFHVREGDEQRTFFSFPAVVAPFKCSVLPLSQNQEFMPFVKELSEALTRHGVSHKVDDSSGSIGRRYARTDEIGVAFGVTIDFDTVNKTPHTATLRDRDSMRQIRAEISELPSIVQDLANGNITWADVEARYPLFEGQETGKK 4qer A 1.2 BS01 STL A 1 L2 F5 G30 C45 H48 D49 L2 F5 G29 C44 H47 D48 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 remove_due_to_license_issue P59071 25541253 202 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 4qev A 1.8 BS01 31O A 1 W370 P371 F372 Y428 N429 V435 W25 P26 F27 Y83 N84 V90 ? remove_due_to_license_issue Kd=1470nM P25440 25323695 501 LSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGAHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 4qew A 1.7 BS01 31P A 1 W370 P371 F372 Y386 Y428 N429 V435 W27 P28 F29 Y43 Y85 N86 V92 ? remove_due_to_license_issue P25440 25323695 503 GKLSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGAHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 4qf7 A 1.48 BS01 C0R A 1 L2 F5 G6 A18 I19 Y22 S23 G30 L2 F5 G6 A17 I18 Y21 S22 G29 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 remove_due_to_license_issue P59071 25541253 201 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 4qf8 A 1.65 BS01 SPD A 1 A18 C29 G30 C45 H48 D49 A17 C28 G29 C44 H47 D48 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 remove_due_to_license_issue P59071 25541253 201 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 4qf9 A 2.28 BS01 35K A 1 Y16 Y61 P88 L89 T90 R95 T192 S193 Y216 Y12 Y57 P84 L85 T86 R91 T188 S189 Y212 ? 0015276,0016020 Ki=37.1uM remove_due_to_license_issue P22756 25856736 301 TLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGN 4qfg C 3.46 BS01 AMP C 1 H150 T199 I203 A204 V224 S225 I311 S313 S315 D316 H122 T171 I175 A176 V196 S197 I276 S278 S280 D281 ? 0004672,0004679,0005515,0005524,0005634,0005737,0005829,0006110,0006633,0010628,0016208,0019887,0019901,0031588,0031669,0032991,0042149,0043531,0043609,0044877,0045722,0051170 remove_due_to_license_issue P80385 25066137 401 SSVYTTFMKSHRCYDLIPTSSKLVVFDTSLQVKKAFFALVTNGVRAAPLWDSKKQSFVGMLTITDFINILHRYYKSALVQIYELEEHKIETWREVYLQPLVCISPNASLFDAVSSLIRNKIHRLPVIDPESGNTLYILTHKRILKFLKLFITEFPKPEFMSKSLEELQIGTYANIAMVRTTTPVYVALGIFVQHRVSALPVVDEKGRVVDIYSKFDVINLAAEKTYNNLDVSVTKALQHRLKCYLHETLEAIINRLVEAEVHRLVVVDEHDVVKGIVSLSDILQALV 4qfl A 1.749 BS02 PHE A 1 T48 G50 R383 Y385 T20 G22 R355 Y357 ? 0015833,0030288,0043190,0055085,1904680 remove_due_to_license_issue A7Y7W1 25605306 602 QGLVYCAEANPVSFNPQVTTTGSTIDIIANQLYDRLISIDPVTAEFKSELATDWKISKDGKSVTFTLRKGVKFHTTAYFTPTREFNADDVIFTFSRLFDVYNPYHFVGDANYPYFQSVGIDQLIRKIVRVSDHQVRFELFNAESSFLANMATDFAVVLSKEYAMALKANNQENLFDQYPVGTGPYIYKEYRRDHLVRFYKNADYWKHEVALEQLVYDITPNGTTRIAKILTKECDVTAHPSSAQLSILAQRDDINVERETNLNIGYWAFNTERPPFDNLKVRQALVHAIDIEKIMQAVYYGNGLRARSILPPTSWAFEPQKNMPIFDPQLAKKLLTEAGYEKGFDMSIWAMPVSRIYNPNARKMAELMQSDLRKIGVNVNIVEYEWNTFIQRIGEHRHDSVLLGWAADTPDPDNFFSPLLSCTATFSGKNPANWCNPEFDLLLTKALDTTDLNLRKQYYDAAQSMIIEQLPLYPIAHGMRFQASSADVEGITLGPFGAISLANARKK 4qfn A 2.297 BS02 GLU A 1 T48 T49 G50 R383 Y385 K457 T20 T21 G22 R355 Y357 K429 ? 0015833,0030288,0043190,0055085,1904680 remove_due_to_license_issue A7Y7W1 25605306 602 QGLVYCAEANPVSFNPQVTTTGSTIDIIANQLYDRLISIDPVTAEFKSELATDWKISKDGKSVTFTLRKGVKFHTTAYFTPTREFNADDVIFTFSRLFDVYNPYHFVGDANYPYFQSVGIDQLIRKIVRVSDHQVRFELFNAESSFLANMATDFAVVLSKEYAMALKANNQENLFDQYPVGTGPYIYKEYRRDHLVRFYKNADYWKHEVALEQLVYDITPNGTTRIAKILTKECDVTAHPSSAQLSILAQRDDINVERETNLNIGYWAFNTERPPFDNLKVRQALVHAIDIEKIMQAVYYGNGLRARSILPPTSWAFEPQKNMPIFDPQLAKKLLTEAGYEKGFDMSIWAMPVSRIYNPNARKMAELMQSDLRKIGVNVNIVEYEWNTFIQRIGEHRHDSVLLGWAADTPDPDNFFSPLLSCTATFSGKNPANWCNPEFDLLLTKALDTTDLNLRKQYYDAAQSMIIEQLPLYPIAHGMRFQASSADVEGITLGPFGAISLANARKK 4qfo A 2.304 BS01 MET A 1 T48 I53 W433 A434 D436 T20 I25 W405 A406 D408 ? 0015833,0030288,0043190,0055085,1904680 remove_due_to_license_issue A7Y7W1 25605306 601 QGLVYCAEANPVSFNPQVTTTGSTIDIIANQLYDRLISIDPVTAEFKSELATDWKISKDGKSVTFTLRKGVKFHTTAYFTPTREFNADDVIFTFSRLFDVYNPYHFVGDANYPYFQSVGIDQLIRKIVRVSDHQVRFELFNAESSFLANMATDFAVVLSKEYAMALKANNQENLFDQYPVGTGPYIYKEYRRDHLVRFYKNADYWKHEVALEQLVYDITPNGTTRIAKILTKECDVTAHPSSAQLSILAQRDDINVERETNLNIGYWAFNTERPPFDNLKVRQALVHAIDIEKIMQAVYYGNGLRARSILPPTSWAFEPQKNMPIFDPQLAKKLLTEAGYEKGFDMSIWAMPVSRIYNPNARKMAELMQSDLRKIGVNVNIVEYEWNTFIQRIGEHRHDSVLLGWAADTPDPDNFFSPLLSCTATFSGKNPANWCNPEFDLLLTKALDTTDLNLRKQYYDAAQSMIIEQLPLYPIAHGMRFQASSADVEGITLGPFGAISLANARKK 4qfo A 2.304 BS02 LEU A 1 G50 R383 Y385 I418 W433 G22 R355 Y357 I390 W405 ? 0015833,0030288,0043190,0055085,1904680 remove_due_to_license_issue A7Y7W1 25605306 602 QGLVYCAEANPVSFNPQVTTTGSTIDIIANQLYDRLISIDPVTAEFKSELATDWKISKDGKSVTFTLRKGVKFHTTAYFTPTREFNADDVIFTFSRLFDVYNPYHFVGDANYPYFQSVGIDQLIRKIVRVSDHQVRFELFNAESSFLANMATDFAVVLSKEYAMALKANNQENLFDQYPVGTGPYIYKEYRRDHLVRFYKNADYWKHEVALEQLVYDITPNGTTRIAKILTKECDVTAHPSSAQLSILAQRDDINVERETNLNIGYWAFNTERPPFDNLKVRQALVHAIDIEKIMQAVYYGNGLRARSILPPTSWAFEPQKNMPIFDPQLAKKLLTEAGYEKGFDMSIWAMPVSRIYNPNARKMAELMQSDLRKIGVNVNIVEYEWNTFIQRIGEHRHDSVLLGWAADTPDPDNFFSPLLSCTATFSGKNPANWCNPEFDLLLTKALDTTDLNLRKQYYDAAQSMIIEQLPLYPIAHGMRFQASSADVEGITLGPFGAISLANARKK 4qfp A 1.903 BS01 VAL A 1 T48 G50 W433 A434 D436 T20 G22 W405 A406 D408 ? 0015833,0030288,0043190,0055085,1904680 remove_due_to_license_issue A7Y7W1 25605306 601 QGLVYCAEANPVSFNPQVTTTGSTIDIIANQLYDRLISIDPVTAEFKSELATDWKISKDGKSVTFTLRKGVKFHTTAYFTPTREFNADDVIFTFSRLFDVYNPYHFVGDANYPYFQSVGIDQLIRKIVRVSDHQVRFELFNAESSFLANMATDFAVVLSKEYAMALKANNQENLFDQYPVGTGPYIYKEYRRDHLVRFYKNADYWKHEVALEQLVYDITPNGTTRIAKILTKECDVTAHPSSAQLSILAQRDDINVERETNLNIGYWAFNTERPPFDNLKVRQALVHAIDIEKIMQAVYYGNGLRARSILPPTSWAFEPQKNMPIFDPQLAKKLLTEAGYEKGFDMSIWAMPVSRIYNPNARKMAELMQSDLRKIGVNVNIVEYEWNTFIQRIGEHRHDSVLLGWAADTPDPDNFFSPLLSCTATFSGKNPANWCNPEFDLLLTKALDTTDLNLRKQYYDAAQSMIIEQLPLYPIAHGMRFQASSADVEGITLGPFGAISLANARKK 4qfp A 1.903 BS02 THR A 1 G50 R383 Y385 G22 R355 Y357 ? 0015833,0030288,0043190,0055085,1904680 remove_due_to_license_issue A7Y7W1 25605306 602 QGLVYCAEANPVSFNPQVTTTGSTIDIIANQLYDRLISIDPVTAEFKSELATDWKISKDGKSVTFTLRKGVKFHTTAYFTPTREFNADDVIFTFSRLFDVYNPYHFVGDANYPYFQSVGIDQLIRKIVRVSDHQVRFELFNAESSFLANMATDFAVVLSKEYAMALKANNQENLFDQYPVGTGPYIYKEYRRDHLVRFYKNADYWKHEVALEQLVYDITPNGTTRIAKILTKECDVTAHPSSAQLSILAQRDDINVERETNLNIGYWAFNTERPPFDNLKVRQALVHAIDIEKIMQAVYYGNGLRARSILPPTSWAFEPQKNMPIFDPQLAKKLLTEAGYEKGFDMSIWAMPVSRIYNPNARKMAELMQSDLRKIGVNVNIVEYEWNTFIQRIGEHRHDSVLLGWAADTPDPDNFFSPLLSCTATFSGKNPANWCNPEFDLLLTKALDTTDLNLRKQYYDAAQSMIIEQLPLYPIAHGMRFQASSADVEGITLGPFGAISLANARKK 4qfr A 3.34 BS02 32J A 1 G19 K29 K31 I46 K51 D88 F90 G11 K21 K23 I38 K43 D80 F82 D139 K141 E143 N144 D157 S176 D131 K133 E135 N136 D149 S168 2.7.11.1,2.7.11.26,2.7.11.31 0000785,0002842,0003682,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005737,0005829,0006006,0006325,0006338,0006468,0006633,0006695,0006914,0008284,0008610,0009410,0009411,0009631,0010332,0010508,0010628,0010629,0014823,0016055,0016324,0016607,0017148,0019395,0030424,0030425,0031000,0031588,0031669,0032007,0032991,0033554,0034599,0035175,0035402,0035403,0035979,0042149,0042542,0042557,0042593,0042752,0043025,0043066,0043627,0044022,0044023,0044024,0044025,0044877,0045722,0045821,0045893,0046321,0046326,0046627,0046872,0047322,0048511,0048643,0050321,0050870,0050995,0055089,0060627,0061744,0061762,0062028,0070050,0070301,0070507,0071277,0071333,0071361,0071380,0071456,0071466,0072354,0072371,0072518,0097009,0106310,0140823,0140855,0140857,1903109,1903829,1903944,1903955,1904179,1904262,1904428,1905691,1990044,1990244,2000758 remove_due_to_license_issue P54645 25066137 606 GRVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFKWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDDSHTIEFFEMCANLIKILAQ 4qfr B 3.34 BS01 32J A 1 R83 R107 D108 V113 R5 R29 D30 V35 ? remove_due_to_license_issue P80386 25066137 606 PTVFRWTGGGKEVYLSGSFNNWSKLPLTRDQNNFVAILDLPEGEHQYKFFVDGQWTHDPSEPIVTSQLGTVNNIIQVKKTDFEVFDALMVDSQKAPPILPPHLLQVILNKSCDPALLPEPNHVMLNHLYALSIKDGVMVLSATHRYKKKYVTTLLYKPI 4qfs A 3.55 BS02 32H A 1 K29 K31 I46 K51 D88 F90 K21 K23 I38 K43 D80 F82 D139 K141 E143 N144 D157 S176 D131 K133 E135 N136 D149 S168 2.7.11.1,2.7.11.26,2.7.11.31 0000785,0002842,0003682,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005737,0005829,0006006,0006325,0006338,0006468,0006633,0006695,0006914,0008284,0008610,0009410,0009411,0009631,0010332,0010508,0010628,0010629,0014823,0016055,0016324,0016607,0017148,0019395,0030424,0030425,0031000,0031588,0031669,0032007,0032991,0033554,0034599,0035175,0035402,0035403,0035979,0042149,0042542,0042557,0042593,0042752,0043025,0043066,0043627,0044022,0044023,0044024,0044025,0044877,0045722,0045821,0045893,0046321,0046326,0046627,0046872,0047322,0048511,0048643,0050321,0050870,0050995,0055089,0060627,0061744,0061762,0062028,0070050,0070301,0070507,0071277,0071333,0071361,0071380,0071456,0071466,0072354,0072371,0072518,0097009,0106310,0140823,0140855,0140857,1903109,1903829,1903944,1903955,1904179,1904262,1904428,1905691,1990044,1990244,2000758 remove_due_to_license_issue P54645 25066137 602 GRVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFKWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDDSHTIEFFEMCANLIKILAQ 4qfs B 3.55 BS01 32H A 1 R83 D108 V113 R5 D30 V35 ? remove_due_to_license_issue P80386 25066137 602 PTVFRWTGGGKEVYLSGSFNNWSKLPLTRDQNNFVAILDLPEGEHQYKFFVDGQWTHDPSEPIVTSQLGTVNNIIQVKKTDFEVFDALMVDSQKAPPILPPHLLQVILNKCDPALLPEPNHVMLNHLYALSIKDGVMVLSATHRYKKKYVTTLLYKPI 4qg3 A 2.0 BS01 rna B 0 H3 G4 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 P133 R134 D166 K167 T168 H172 S211 Y213 T217 M218 V219 S221 H3 G4 K5 R6 Y7 A35 K36 F37 T40 E42 H44 K46 P133 R134 D166 K167 T168 H172 S211 Y213 T217 M218 V219 S221 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 25664749 2105 ~ 2184 PKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTMVPSVRINPHS 4qg7 A 1.67 BS01 32K A 1 E37 R48 L52 F66 R70 R92 S96 S97 Y100 Q101 E36 R47 L51 F65 R69 R91 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=10nM remove_due_to_license_issue Q6GJI9 24828090 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKNDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEKI 4qga A 1.94 BS01 31Z A 1 E37 R48 L52 F66 S69 R70 R92 S96 S97 Y100 Q101 E36 R47 L51 F65 S68 R69 R91 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=12nM remove_due_to_license_issue Q6GJI9 24828090 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKNDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEK 4qgd A 1.8 BS01 PZZ A 1 L2 L3 F5 G6 A18 I19 S23 G30 L2 L3 F5 G6 A17 I18 S22 G29 Y28 G30 G32 H48 D49 Y52 Y73 D99 Y27 G29 G31 H47 D48 Y51 Y64 D89 3.1.1.4 0004623,0005509,0005543,0005576,0006644,0016042,0016787,0035821,0042130,0046872,0047498,0047499,0050482,0090729 remove_due_to_license_issue P59071 25541253 201 SLLEFGKMILEETGKLAIPSYSSYGCYCGWGGKGTPKDATDRCCFVHDCCYGNLPDCNPKSDRYKYKRVNGAIVCEKGTSCENRICECDKAAAICFRQNLNTYSKKYMLYPDFLCKGELKC 4qge A 2.0 BS01 35O A 1 M365 L420 Y424 A452 Q453 F456 M181 L236 Y240 A268 Q269 F272 3.1.4.35 0004114,0004115,0004117,0005737,0005783,0005794,0005886,0007165,0008081,0010613,0016787,0019933,0032587,0042383,0042995,0046068,0046069,0046872,0047555,0048101,0048471 Ki=0.5nM remove_due_to_license_issue H2QL32 25432025 601 KYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQKK 4qgf A 1.83 BS01 32B A 1 E37 R48 L52 F66 S69 R70 R92 S97 Y100 Q101 E36 R47 L51 F65 S68 R69 R91 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=69nM remove_due_to_license_issue Q6GJI9 24828090 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEKI 4qgg A 1.62 BS01 32C A 1 E37 R48 L52 F66 S69 R70 R92 S96 S97 Y100 Q101 E36 R47 L51 F65 S68 R69 R91 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=1nM remove_due_to_license_issue Q6GJI9 24828090 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEKI 4qgh A 1.78 BS01 32E A 1 E37 R48 L52 F66 R70 S97 Y100 Q101 E36 R47 L51 F65 R69 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=1nM remove_due_to_license_issue Q6GJI9 24828090 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKNDQEDLKFHEKVIEGYQEIIHNQRFKSVNADQPLENVVEDTYQTIIKYLEKI 4qgh B 1.78 BS01 32E B 1 E37 R48 L52 F66 R70 R92 S96 S97 Y100 Q101 E36 R47 L51 F65 R69 R91 S95 S96 Y99 Q100 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0046940 ic50=1nM remove_due_to_license_issue Q6GJI9 24828090 301 SAFITFEGPEGSGKTTVINEVYHRLVKDYDVIMTREPGGVPTGEEIRKIVLEGNDMDIRTEAMLFAASRREHLVLKVIPALKEGKVVLCDRYIDSSLAYQGYARGIGVEEVRALNEFAINGLYPDLTIYLNVSAEVGRERIIKRLDQEDLKFHEKVIEGYQEIIHNESQRFKSVNADQPLENVVEDTYQTIIKYLEKI 4qgi A 1.896 BS01 ROC A 1 D25 G27 A28 D29 D30 T48 G49 I50 D25 G27 A28 D29 D30 T48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 25513833 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMITGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNMLTQIGCTLNF 4qgi B 1.896 BS01 ROC A 1 D25 G27 G49 I50 P81 I84 D25 G27 G49 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P0C6F2 25513833 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMITGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNMLTQIGCTLNF 4qhc A 1.899 BS01 33V A 1 S84 S116 I117 E182 N186 G252 T253 S42 S74 I75 E140 N144 G210 T211 S84 K87 S142 E182 K250 T253 S42 K45 S100 E140 K208 T211 3.5.2.6 0005576,0005886,0008800,0016787,0017001,0030655,0042597,0046677 remove_due_to_license_issue P9WKD3 26237118 401 DLADRFAELERRYDARLGVYVPATGTTAAIEYRADERFAFCSTFKAPLVAAVLHQNPLTHLDKLITYTSDDIRSISPVAQQHVQTGMTIGQLCDAAIRYSDGTAANLLLADLGGPGGGTAAFTGYLRSLGDTVSRLDAEEPELNRDPPGDERDTTTPHAIALVLQQLVLGNALPPDKRALLTDWMARNTTGAKRIRAGFPADWKVIDKTGTGDYGRANDIAVVWSPTGVPYVVAVMSDRAGGGYDAEPREALLAEAATCVAGVLA 4qhp A 1.6 BS01 32Q A 1 Q115 E117 M256 G257 A258 M259 E260 H293 E294 H297 E316 D323 Y377 Q114 E116 M255 G256 A257 M258 E259 H292 E293 H296 E315 D322 Y376 E260 H293 E294 H297 E316 N369 Y377 E259 H292 E293 H296 E315 N368 Y376 3.4.11.2 0004177,0006508,0008237,0008270,0046872 Ki=9nM remove_due_to_license_issue Q9JYV4 25192493 901 SKTVHYLKDYQTPAYHILKTDLHFDINEPQTVVKSRLTVEPQRVGEPLVLDGSAKLLSVKINGAAADYVLEGETLTIAGVPSERFTVEVETEILPAENKSLMGLYASGGNLFTQCEPEGFRKITFYIDRPDVMSKFTTTIVADKKRYPVLLSNGNKIDGGEFSDGRHWVKWEDPFSKPSYLFALVAGDLAVTEDYFTTMSGRNVKIEFYTTEADKPKVGFAVESLKNAMKWDETRFGLEYDLDIFMVVAVGDFNMGAMENKGLNIFNTKFVLADSRTATDTDFEGIESVVGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSGDRASRAVRRIENIRLLRQHQFPEDAGPTAHPVRPASYEEMNNFYTMTVYEKGAEVVRMYHTLLGEEGFQKGMKLYFQRHDGQAVTCDDFRAAMADANGINLDQFALWYSQAGTPVLEAEGRLKNNIFELTVKQTVPPTPDMTDKQPMMIPVKVGLLNRNGEAVAFDYQGKRATEAVLLLTEAEQTFLLEGVTEAVVPSLLRGFSAPVHLNYPYSDDDLLLLLAHDSDAFTRWEAAQTLYRRAVAANLATLSDGVELPKHEKLLAAVEKVISDDLLDNAFKALLLGVPSEAELWDGAENIDPLRYHQAREALLDTLAVHFLPKWHELNRQAAKQENQSYEYSPEAAGWRTLRNVCRAFVLRADPAHIETVAEKYGEMAQNMTHEWGILSAVNGNESDTRNRLLAQFADKFSDDALVMDKYFALVGSSRRSDTLQQVRTALQHPKFSLENPNKARSLIGSFSRNVPHFHAEDGSGYRFIADKVIEIDRFNPQVAARLVQAFNLCNKLEPHRKNLVKQALQRIRAQEGLSKDVGEIVGKILD 4qht A 2.559 BS01 ANP A 1 M131 V132 S161 G162 G164 K165 E166 V167 L312 H315 R319 V348 R349 M2 V3 S32 G33 G35 K36 E37 V38 L183 H186 R190 V219 R220 ? 0005524,0006355,0008134,0016887 remove_due_to_license_issue A0A0H3AHP1 25688103 401 HMVVADTKSLKLLALADKVAKTDANVMILGPSGSGKEVMSRYIHNASPRKEGPFIAINCAAIPDNMLEATLFGYEKGAFTGAVQACPGKFEQAQGGTILLDEISEMDLNLQAKLLRVLQEREVERLGSRKSIKLDVRVLATSNRDLKQYVQAGHFREDLYYRLNVFPLTWPALCERKDDIEPLANHLIERHCKKLGLPVPSIAPNAITKLLNYPWPGNVRELDNVVQRALILSENGHIQSEHILLE 4qht B 2.559 BS01 ANP B 1 M131 V132 S161 G162 S163 G164 K165 V167 L312 R319 V348 R349 M2 V3 S32 G33 S34 G35 K36 V38 L183 R190 V219 R220 ? 0005524,0006355,0008134,0016887 remove_due_to_license_issue A0A0H3AHP1 25688103 401 HMVVADTKSLKLLALADKVAKTDANVMILGPSGSGKEVMSRYIHNASPRKEGPFIAINCAAIPDNMLEATLFGYEKGAFTGAVQACPGKFEQAQGGTILLDEISEMDLNLQAKLLRVLQEREVERLGSRKSIKLDVRVLATSNRDLKQYVQAGHFREDLYYRLNVFPLTWPALCERKDDIEPLANHLIERHCKKLGLPVPSIAPNAITKLLNYPWPGNVRELDNVVQRALILSENGHIQSEHILL 4qi2 A 3.0 BS01 rna E 0 R188 R219 K220 S238 K239 T240 Q247 Y250 R251 E262 D263 S264 S265 R16 R47 K48 S66 K67 T68 Q75 Y78 R79 E90 D91 S92 S93 2.3.2.27 remove_due_to_license_issue Q4VGL6 25026077 3 ~ 21 HQNPQQLSSNLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRTYEALRREHDSQIVQIAMEAGLRIAPDQWSSLLYGDQSHKSHMQSIIDKLQ 4qi2 B 3.0 BS01 rna F 0 R188 R219 K220 S238 K239 T240 Q247 Y250 R251 E262 D263 S264 S265 R16 R47 K48 S66 K67 T68 Q75 Y78 R79 E90 D91 S92 S93 2.3.2.27 remove_due_to_license_issue Q4VGL6 25026077 4 ~ 21 HQNPQQLSSNLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRTYEALRREHDSQIVQIAMEAGLRIAPDQWSSLLYGDQSHKSHMQSIIDKLQ 4qi2 C 3.0 BS01 rna G 0 W184 R188 F194 R219 K220 S238 K239 T240 Q247 Y250 R251 E262 D263 S264 W11 R15 F21 R46 K47 S65 K66 T67 Q74 Y77 R78 E89 D90 S91 2.3.2.27 remove_due_to_license_issue Q4VGL6 25026077 4 ~ 22 QNPQQLSSNLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRTYEALRREHDSQIVQIAMEAGLRIAPDQWSSLLYGDQSHKSHMQSIIDKLQ 4qi2 D 3.0 BS01 rna H 0 W184 R188 F194 R219 K220 S238 K239 T240 Q247 Y250 R251 S253 E262 D263 S264 S265 W13 R17 F23 R48 K49 S67 K68 T69 Q76 Y79 R80 S82 E91 D92 S93 S94 2.3.2.27 remove_due_to_license_issue Q4VGL6 25026077 4 ~ 21 QHQNPQQLSSNLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRTYEALRREHDSQIVQIAMEAGLRIAPDQWSSLLYGDQSHKSHMQSIIDKLQ 4qij A 2.2 BS01 1HA A 1 V57 R58 A60 F61 K95 S103 G104 G105 D106 Q107 Y115 L134 I136 W157 G161 T184 D185 S190 V44 R45 A47 F48 K82 S90 G91 G92 D93 Q94 Y102 L121 I123 W144 G148 T171 D172 S177 G105 R110 Y115 R130 H135 G161 S164 D185 S190 D192 G193 A279 Y287 G92 R97 Y102 R117 H122 G148 S151 D172 S177 D179 G180 A266 Y274 4.1.3.36 0005886,0008935,0009234,0016829,0034214 Kd=2.9uM remove_due_to_license_issue P9WNP5 25372686 401 ALSDNPFDAKAWRLVDGFDDLTDITYHRHVDDATVRVAFNRPEVRNAFRPHTVDELYRVLDHARMSPDVGVVLLTGNGPSPKDGGWAFCSGGDQRIRGRSGYQYASGDTADTVDVARAGRLHILEVQRLIRFMPKVVICLVNGWAAGGGHSLHVVCDLTLASREYARFKQTDADVGSFDGGYGSAYLARQVGQKFAREIFFLGRTYTAEQMHQMGAVNAVAEHAELETVGLQWAAEINAKSPQAQRMLKFAFNLLDDGLVGQQLFAGEATRLAYMTDEAVEGRDAFLQKRPPDWSPFPRYF 4qij A 2.2 BS02 1HA F 1 F299 K302 F286 K289 G105 R110 Y115 R130 H135 G161 S164 D185 S190 D192 G193 A279 Y287 G92 R97 Y102 R117 H122 G148 S151 D172 S177 D179 G180 A266 Y274 4.1.3.36 0005886,0008935,0009234,0016829,0034214 Kd=2.9uM remove_due_to_license_issue P9WNP5 25372686 401 ALSDNPFDAKAWRLVDGFDDLTDITYHRHVDDATVRVAFNRPEVRNAFRPHTVDELYRVLDHARMSPDVGVVLLTGNGPSPKDGGWAFCSGGDQRIRGRSGYQYASGDTADTVDVARAGRLHILEVQRLIRFMPKVVICLVNGWAAGGGHSLHVVCDLTLASREYARFKQTDADVGSFDGGYGSAYLARQVGQKFAREIFFLGRTYTAEQMHQMGAVNAVAEHAELETVGLQWAAEINAKSPQAQRMLKFAFNLLDDGLVGQQLFAGEATRLAYMTDEAVEGRDAFLQKRPPDWSPFPRYF 4qij F 2.2 BS01 1HA A 1 F299 K302 F283 K286 G105 R110 Y115 R130 H135 G161 S164 D185 S190 D192 G193 A279 Y287 G89 R94 Y99 R114 H119 G145 S148 D169 S174 D176 G177 A263 Y271 4.1.3.36 0005886,0008935,0009234,0016829,0034214 Kd=2.9uM remove_due_to_license_issue P9WNP5 25372686 401 DNPFDAKAWRLVDGFDDLTDITYHRHVDDATVRVAFNRPEVRNAFRPHTVDELYRVLDHARMSPDVGVVLLTGNGPSPKDGGWAFCSGGDQRIRGRSGYQYASGDTADTVDVARAGRLHILEVQRLIRFMPKVVICLVNGWAAGGGHSLHVVCDLTLASREYARFKQTDADVGSFDGGYGSAYLARQVGQKFAREIFFLGRTYTAEQMHQMGAVNAVAEHAELETVGLQWAAEINAKSPQAQRMLKFAFNLLDDGLVGQQLFAGEATRLAYMTDEAVEGRDAFLQKRPPDWSPFPRYF 4qij F 2.2 BS02 1HA F 1 E56 V57 R58 A60 K95 S103 G104 G105 D106 Q107 Y115 I136 L137 W157 G161 T184 D185 V188 S190 E40 V41 R42 A44 K79 S87 G88 G89 D90 Q91 Y99 I120 L121 W141 G145 T168 D169 V172 S174 G105 R110 Y115 R130 H135 G161 S164 D185 S190 D192 G193 A279 Y287 G89 R94 Y99 R114 H119 G145 S148 D169 S174 D176 G177 A263 Y271 4.1.3.36 0005886,0008935,0009234,0016829,0034214 Kd=2.9uM remove_due_to_license_issue P9WNP5 25372686 401 DNPFDAKAWRLVDGFDDLTDITYHRHVDDATVRVAFNRPEVRNAFRPHTVDELYRVLDHARMSPDVGVVLLTGNGPSPKDGGWAFCSGGDQRIRGRSGYQYASGDTADTVDVARAGRLHILEVQRLIRFMPKVVICLVNGWAAGGGHSLHVVCDLTLASREYARFKQTDADVGSFDGGYGSAYLARQVGQKFAREIFFLGRTYTAEQMHQMGAVNAVAEHAELETVGLQWAAEINAKSPQAQRMLKFAFNLLDDGLVGQQLFAGEATRLAYMTDEAVEGRDAFLQKRPPDWSPFPRYF 4qip A 2.0 BS01 SDS A 1 F58 F62 F64 M139 T142 F58 F62 F64 M139 T142 ? 0004864,0005634,0005737,0006952,0009738,0010427,0038023 remove_due_to_license_issue P15494 25517162 201 GVFNYETETTSVIPAARLFKAFILDGDNLFPKVAPQAISSVENIEGNGGPGTIKKISFPEGFPFKYVKDRVDEVDHTNFKYNYSVIEGGPIGDTLEKISNEIKIVATPDGGSILKISNKYHTKGDHEVKAEQVKASKEMGETLLRAVESYLLAHSDAYN 4qip A 2.0 BS02 SDS A 2 T9 F22 K54 D69 Y81 I102 G140 E141 T9 F22 K54 D69 Y81 I102 G140 E141 ? 0004864,0005634,0005737,0006952,0009738,0010427,0038023 remove_due_to_license_issue P15494 25517162 202 GVFNYETETTSVIPAARLFKAFILDGDNLFPKVAPQAISSVENIEGNGGPGTIKKISFPEGFPFKYVKDRVDEVDHTNFKYNYSVIEGGPIGDTLEKISNEIKIVATPDGGSILKISNKYHTKGDHEVKAEQVKASKEMGETLLRAVESYLLAHSDAYN 4qir A 1.701 BS01 379 A 1 E117 M256 G257 A258 M259 E260 H293 E294 H297 E316 D323 N369 Y372 Y377 E114 M253 G254 A255 M256 E257 H290 E291 H294 E313 D320 N366 Y369 Y374 E260 H293 E294 H297 E316 N369 Y377 E257 H290 E291 H294 E313 N366 Y374 3.4.11.2 0004177,0006508,0008237,0008270,0046872 Ki=112nM remove_due_to_license_issue Q9JYV4 25192493 901 TVHYLKDYQTPAYHILKTDLHFDINEPQTVVKSRLTVEPQRVGEPLVLDGSAKLLSVKINGAAADYVLEGETLTIAGVPSERFTVEVETEILPAENKSLMGLYASGGNLFTQCEPEGFRKITFYIDRPDVMSKFTTTIVADKKRYPVLLSNGNKIDGGEFSDGRHWVKWEDPFSKPSYLFALVAGDLAVTEDYFTTMSGRNVKIEFYTTEADKPKVGFAVESLKNAMKWDETRFGLEYDLDIFMVVAVGDFNMGAMENKGLNIFNTKFVLADSRTATDTDFEGIESVVGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSGDRASRAVRRIENIRLLRQHQFPEDAGPTAHPVRPASYEEMNNFYTMTVYEKGAEVVRMYHTLLGEEGFQKGMKLYFQRHDGQAVTCDDFRAAMADANGINLDQFALWYSQAGTPVLEAEGRLKNNIFELTVKQTVPPTPDMTDKQPMMIPVKVGLLNRNGEAVAFDYQGKRATEAVLLLTEAEQTFLLEGVTEAVVPSLLRGFSAPVHLNYPYSDDDLLLLLAHDSDAFTRWEAAQTLYRRAVAANLATLSDGVELPKHEKLLAAVEKVISDDLLDNAFKALLLGVPSEAELWDGAENIDPLRYHQAREALLDTLAVHFLPKWHELNRQAAKQENQSYEYSPEAAGWRTLRNVCRAFVLRADPAHIETVAEKYGEMAQNMTHEWGILSAVNGNESDTRNRLLAQFADKFSDDALVMDKYFALVGSSRRSDTLQQVRTALQHPKFSLENPNKARSLIGSFSRNVPHFHAEDGSGYRFIADKVIEIDRFNPQVAARLVQAFNLCNKLEPHRKNLVKQALQRIRAQEGLSKDVGEIVGKILD 4qiy A 1.3 BS02 WWX A 1 N62 N67 I91 H94 H96 V135 L198 T199 T200 P202 N59 N64 I88 H91 H93 V131 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=50nM remove_due_to_license_issue P00918 25758852 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4qiz A 1.55 BS02 WWX A 1 S64 N69 Q94 H96 H98 F133 L200 T201 V202 P204 S59 N64 Q89 H91 H93 F128 L195 T196 V197 P199 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=7.1nM remove_due_to_license_issue Q8N1Q1 25758852 304 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 4qj0 A 1.55 BS02 WWX A 1 N64 S67 H91 H117 V119 L197 T198 T199 N62 S65 H89 H115 V117 L195 T196 T197 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=48nM remove_due_to_license_issue O43570 25758852 303 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFS 4qjm A 1.75 BS02 V1F A 1 N62 H64 N67 I91 Q92 H94 H96 H119 F131 L198 T199 T200 P201 N59 H61 N64 I88 Q89 H91 H93 H116 F127 L194 T195 T196 P197 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=6.7nM remove_due_to_license_issue P00918 25758852 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4qjo A 1.8 BS02 V1F A 1 Q89 H91 H93 H117 A129 L197 T198 T199 P200 Q87 H89 H91 H115 A127 L195 T196 T197 P198 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=40nM remove_due_to_license_issue O43570 25758852 303 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4qjp B 1.62 BS02 V1F B 1 S64 H66 N69 H96 H121 V123 F133 L200 T201 V202 P204 S59 H61 N64 H91 H116 V118 F128 L195 T196 V197 P199 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=2.5nM remove_due_to_license_issue Q8N1Q1 25758852 303 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 4qjr A 2.4 BS02 PIZ A 1 L265 L306 Q339 A340 G341 L344 L429 Y436 K440 L48 L89 Q122 A123 G124 L127 L212 Y219 K223 ? 0003677,0004879 Kd=80nM remove_due_to_license_issue Q13285 25288771 501 SGGPNVPELILQLLQLEPDEDQVRARILGSLQEPTKSRPDQPAAFGLLCRMADQTFISIVDWARRCMVFKELEVADQMTLLQNCWSELLVFDHIYRQVQHGKEGSILLVTGQEVELTTVATQAGSLLHSLVLRAQELVLQLLALQLDRQEFVCLKFIILFSLDLKFLNNHILVKDAQEKANAALLDYTLCHYPHSGDKFQQLLLCLVEVRALSMQAKEYLYHKHLGNEMPRNNLLIEMLQAKQT 4qju A 2.16 BS01 dna C 0 R58 G60 P63 Q64 I71 R58 G60 P63 Q64 I71 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q99U17 25478845 1 ~ 21 MNKTDLINAVAEQADLTKKEAGSAVDAVFESIQNSLAKGEKVQLIGFGNFEVRERAARKGRNPQTGKEIDIPASKVPAFKAGKALKDAVK 4qju A 2.16 BS02 dna D 0 A56 K59 R61 P63 E68 A56 K59 R61 P63 E68 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q99U17 25478845 1 ~ 21 MNKTDLINAVAEQADLTKKEAGSAVDAVFESIQNSLAKGEKVQLIGFGNFEVRERAARKGRNPQTGKEIDIPASKVPAFKAGKALKDAVK 4qju B 2.16 BS01 dna C 0 R55 A56 K59 R61 P63 K83 R55 A56 K59 R61 P63 K83 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q99U17 25478845 1 ~ 21 MNKTDLINAVAEQADLTKKEAGSAVDAVFESIQNSLAKGEKVQLIGFGNFEVRERAARKGRNPQTGKEIDIPASKVPAFKAGKALKDAVK 4qju B 2.16 BS02 dna D 0 Q43 G46 N49 R55 R58 G60 R61 P63 Q64 I69 I71 G82 Q43 G46 N49 R55 R58 G60 R61 P63 Q64 I69 I71 G82 ? 0003677,0005829,0030261,0030527 remove_due_to_license_issue Q99U17 25478845 1 ~ 21 MNKTDLINAVAEQADLTKKEAGSAVDAVFESIQNSLAKGEKVQLIGFGNFEVRERAARKGRNPQTGKEIDIPASKVPAFKAGKALKDAVK 4qjw A 1.55 BS02 WWO A 1 Q89 H91 H93 H117 A129 S130 L197 T198 T199 P200 Q87 H89 H91 H115 A127 S128 L195 T196 T197 P198 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=16nM remove_due_to_license_issue O43570 25758852 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4qjx A 1.95 BS02 WWO A 1 S64 H66 N69 H96 H98 F133 L200 T201 V202 S59 H61 N64 H91 H93 F128 L195 T196 V197 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=52nM remove_due_to_license_issue Kd=0.013000nM Q8N1Q1 25758852 304 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 4qk4 A 2.81 BS02 PIK A 1 F262 L265 C266 S303 L306 V307 L344 L429 A433 Y436 L437 H439 F45 L48 C49 S86 L89 V90 L127 L212 A216 Y219 L220 H222 ? 0003677,0004879 remove_due_to_license_issue Q13285 25288771 501 SGGPNVPELILQLLQLEPDEDQVRARILGSLQEPTKSRPDQPAAFGLLCRMADQTFISIVDWARRCMVFKELEVADQMTLLQNCWSELLVFDHIYRQVQHGKEGSILLVTGQEVELTTVATQAGSLLHSLVLRAQELVLQLLALQLDRQEFVCLKFIILFSLDLKFLNNHILVKDAQEKANAALLDYTLCHYPHSGDKFQQLLLCLVEVRALSMQAKEYLYHKHLGNEMPRNNLLIEMLQAKQT 4qkd A 1.35 BS02 AKG A 1 X110 H121 D123 Y165 H177 R197 S199 R203 X94 H105 D107 Y149 H161 R181 S183 R187 1.14.11.- 0005515,0005739,0005759,0006631,0006974,0010883,0012501,0046872,0051213,1902445 remove_due_to_license_issue Q9BT30 25122757 302 MWVRGSGPSVLSRLQDAAVVRPGFLSTAEEETLSRELEPELRRRRYEYDHWDAAIHGFRETEKSRWSEASRAILRRVQAAAFGPQTLLSSVHVLDLEARGYIKPHVDSIKFCGATIAGLSLLSPSVMRLVHTQEPGEWLELLLEPGSLYILRGSARYDFSHEILRDEESFFGERRIPRGRRISVICRSLP 4qkx A 3.3 BS01 35V A 1 C1093 W1109 D1113 V1114 C1191 F1193 S1203 S1207 N1312 Y1316 C236 W252 D256 V257 C334 F336 S346 S350 N424 Y428 E876 D885 E19 D28 3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue P00720,P07550 25006259 1403 DAENLYFQGNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYAADEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAACILTKTWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLQKFALKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 4ql1 A 1.5 BS01 35Q A 1 S49 S50 A65 S91 D107 F133 P173 Y191 C261 S19 S20 A35 S61 D77 F103 P143 Y161 C231 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue Kd=30nM P61964 26167872 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 4ql8 A 2.1 BS01 JAD A 1 L704 N705 L707 W741 M742 M745 M749 F764 M780 F876 T877 L34 N35 L37 W71 M72 M75 M79 F94 M110 F199 T200 ? ic50=0.7nM remove_due_to_license_issue EC50=0.500000nM, IC50=0.700000nM P10275 25121964 1001 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFH 4qlc A 3.503 BS01 dna I 0 Y41 R42 T45 R63 R83 F84 Q85 R116 V117 T118 M120 Y4 R5 T8 R26 R46 F47 Q48 R79 V80 T81 M83 ? 0000785,0000786,0003677,0005515,0005634,0005694,0005700,0006334,0030527,0031492,0035059,0046982 remove_due_to_license_issue P02299 26212454 1 ~ 166 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 4qlc A 3.503 BS02 dna J 0 H39 R40 Y41 G44 V46 A47 R49 R63 K64 L65 P66 R69 H2 R3 Y4 G7 V9 A10 R12 R26 K27 L28 P29 R32 ? 0000785,0000786,0003677,0005515,0005634,0005694,0005700,0006334,0030527,0031492,0035059,0046982 remove_due_to_license_issue P02299 26212454 1 ~ 166 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 4qlc B 3.503 BS01 dna I 0 T30 R36 R45 T6 R12 R21 ? 0000228,0000786,0003676,0003677,0005515,0005634,0005694,0006334,0030527,0035059,0046982 remove_due_to_license_issue P84040 26212454 1 ~ 166 NIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4qlc B 3.503 BS02 dna J 0 R35 R45 I46 S47 G48 R78 K79 T80 R11 R21 I22 S23 G24 R54 K55 T56 ? 0000228,0000786,0003676,0003677,0005515,0005634,0005694,0006334,0030527,0035059,0046982 remove_due_to_license_issue P84040 26212454 1 ~ 166 NIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4qlc C 3.503 BS01 dna I 0 K14 R16 R28 R31 R76 K1 R3 R15 R18 R63 ? 0000786,0003677,0005515,0005634,0005694,0005700,0005704,0006325,0006334,0007526,0030527,0031507,0046982 remove_due_to_license_issue P84051 26212454 1 ~ 166 KSRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLPK 4qlc C 3.503 BS02 dna J 0 R28 R34 R41 V42 G43 A44 T75 R76 R15 R21 R28 V29 G30 A31 T62 R63 ? 0000786,0003677,0005515,0005634,0005694,0005700,0005704,0006325,0006334,0007526,0030527,0031507,0046982 remove_due_to_license_issue P84051 26212454 1 ~ 166 KSRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLPK 4qlc D 3.503 BS01 dna I 0 K29 R30 Y39 S52 S53 R83 S84 T85 K1 R2 Y11 S24 S25 R55 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0006325,0030527,0044877,0046982 remove_due_to_license_issue P02283 26212454 1 ~ 166 KRKESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4qlc D 3.503 BS02 dna J 0 R30 K31 S33 Y37 R2 K3 S5 Y9 ? 0000786,0003677,0005515,0005634,0005694,0006325,0030527,0044877,0046982 remove_due_to_license_issue P02283 26212454 1 ~ 166 KRKESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4qlc E 3.503 BS01 dna I 0 H39 R40 Y41 G44 V46 R49 K56 R63 K64 L65 P66 R69 R83 H2 R3 Y4 G7 V9 R12 K19 R26 K27 L28 P29 R32 R46 ? 0000785,0000786,0003677,0005515,0005634,0005694,0005700,0006334,0030527,0031492,0035059,0046982 remove_due_to_license_issue P02299 26212454 1 ~ 166 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 4qlc E 3.503 BS02 dna J 0 Y41 R42 P43 T45 R63 R83 F84 Q85 R116 V117 T118 M120 Y4 R5 P6 T8 R26 R46 F47 Q48 R79 V80 T81 M83 ? 0000785,0000786,0003677,0005515,0005634,0005694,0005700,0006334,0030527,0031492,0035059,0046982 remove_due_to_license_issue P02299 26212454 1 ~ 166 PHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 4qlc F 3.503 BS01 dna I 0 R45 I46 S47 G48 R78 K79 T80 R23 I24 S25 G26 R56 K57 T58 ? 0000228,0000786,0003676,0003677,0005515,0005634,0005694,0006334,0030527,0035059,0046982 remove_due_to_license_issue P84040 26212454 1 ~ 166 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4qlc F 3.503 BS02 dna J 0 T30 P32 R36 R45 T8 P10 R14 R23 ? 0000228,0000786,0003676,0003677,0005515,0005634,0005694,0006334,0030527,0035059,0046982 remove_due_to_license_issue P84040 26212454 1 ~ 166 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4qlc G 3.503 BS01 dna I 0 R28 R34 R41 V42 G43 A44 T75 R76 R16 R22 R29 V30 G31 A32 T63 R64 ? 0000786,0003677,0005515,0005634,0005694,0005700,0005704,0006325,0006334,0007526,0030527,0031507,0046982 remove_due_to_license_issue P84051 26212454 1 ~ 166 AKSRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4qlc G 3.503 BS02 dna J 0 A13 R16 R28 R31 R41 R76 A1 R4 R16 R19 R29 R64 ? 0000786,0003677,0005515,0005634,0005694,0005700,0005704,0006325,0006334,0007526,0030527,0031507,0046982 remove_due_to_license_issue P84051 26212454 1 ~ 166 AKSRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4qlc H 3.503 BS01 dna I 0 K31 S33 Y37 K4 S6 Y10 ? 0000786,0003677,0005515,0005634,0005694,0006325,0030527,0044877,0046982 remove_due_to_license_issue P02283 26212454 1 ~ 166 RKRKESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4qlc H 3.503 BS02 dna J 0 K29 Y39 S52 S53 S84 T85 K2 Y12 S25 S26 S57 T58 ? 0000786,0003677,0005515,0005634,0005694,0006325,0030527,0044877,0046982 remove_due_to_license_issue P02283 26212454 1 ~ 166 RKRKESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4qlc U 3.503 BS01 dna I 0 H25 T27 Y28 R42 S46 Q48 R74 K85 G91 S92 H4 T6 Y7 R21 S25 Q27 R53 K64 G70 S71 ? 0000786,0003677,0006334,0030527 remove_due_to_license_issue P02259 26212454 1 ~ 166 SASHPTYSEMIAAAIRAEKSRGGSSRQSIQKYIKSHYKVGHNADLQIKLSIRRLLAAGVLKQTKGVGASGSFRLAK 4qlc U 3.503 BS02 dna J 0 R47 L66 K69 R73 A89 S90 R94 R26 L45 K48 R52 A68 S69 R73 ? 0000786,0003677,0006334,0030527 remove_due_to_license_issue P02259 26212454 1 ~ 166 SASHPTYSEMIAAAIRAEKSRGGSSRQSIQKYIKSHYKVGHNADLQIKLSIRRLLAAGVLKQTKGVGASGSFRLAK 4qlq H 2.4 BS01 38N H 1 T1 S20 T21 Q22 C31 G47 T48 A49 T52 G168 T1 S20 T21 Q22 C31 G47 T48 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25006746 303 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qls K 2.8 BS02 37Y K 1 T1 A20 T21 V31 G47 A49 S131 Y170 T1 A20 T21 V31 G47 A49 S131 Y170 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25006746 303 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4qls L 2.8 BS01 37Y K 1 D126 E132 D126 E132 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25006746 303 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qlt K 2.8 BS02 39V K 1 T1 A20 T21 V31 K33 G47 A49 S96 Y170 T1 A20 T21 V31 K33 G47 A49 S96 Y170 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25006746 303 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4qlt L 2.8 BS01 39V K 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25006746 303 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qlu K 2.8 BS02 38X K 1 T1 R19 A20 T21 G47 G48 A49 Y170 T1 R19 A20 T21 G47 G48 A49 Y170 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25006746 303 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4qlu L 2.8 BS01 38X K 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25006746 303 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qlv K 2.9 BS02 39Q K 1 T1 A20 T21 V31 K33 G47 A49 Y170 T1 A20 T21 V31 K33 G47 A49 Y170 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25006746 303 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4qlv L 2.9 BS01 39Q K 1 D126 S130 D126 S130 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25006746 303 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qme A 1.601 BS01 37B A 1 Q115 E117 M256 G257 A258 M259 E260 H293 E294 H297 E316 D323 Y377 Q114 E116 M255 G256 A257 M258 E259 H292 E293 H296 E315 D322 Y376 E260 H293 E294 H297 E316 N369 Y377 E259 H292 E293 H296 E315 N368 Y376 3.4.11.2 0004177,0006508,0008237,0008270,0046872 Ki=302nM remove_due_to_license_issue Q9JYV4 25192493 901 SKTVHYLKDYQTPAYHILKTDLHFDINEPQTVVKSRLTVEPQRVGEPLVLDGSAKLLSVKINGAAADYVLEGETLTIAGVPSERFTVEVETEILPAENKSLMGLYASGGNLFTQCEPEGFRKITFYIDRPDVMSKFTTTIVADKKRYPVLLSNGNKIDGGEFSDGRHWVKWEDPFSKPSYLFALVAGDLAVTEDYFTTMSGRNVKIEFYTTEADKPKVGFAVESLKNAMKWDETRFGLEYDLDIFMVVAVGDFNMGAMENKGLNIFNTKFVLADSRTATDTDFEGIESVVGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSGDRASRAVRRIENIRLLRQHQFPEDAGPTAHPVRPASYEEMNNFYTMTVYEKGAEVVRMYHTLLGEEGFQKGMKLYFQRHDGQAVTCDDFRAAMADANGINLDQFALWYSQAGTPVLEAEGRLKNNIFELTVKQTVPPTPDMTDKQPMMIPVKVGLLNRNGEAVAFDYQGKRATEAVLLLTEAEQTFLLEGVTEAVVPSLLRGFSAPVHLNYPYSDDDLLLLLAHDSDAFTRWEAAQTLYRRAVAANLATLSDGVELPKHEKLLAAVEKVISDDLLDNAFKALLLGVPSEAELWDGAENIDPLRYHQAREALLDTLAVHFLPKWHELNRQAAKQENQSYEYSPEAAGWRTLRNVCRAFVLRADPAHIETVAEKYGEMAQNMTHEWGILSAVNGNESDTRNRLLAQFADKFSDDALVMDKYFALVGSSRRSDTLQQVRTALQHPKFSLENPNKARSLIGSFSRNVPHFHAEDGSGYRFIADKVIEIDRFNPQVAARLVQAFNLCNKLEPHRKNLVKQALQRIRAQEGLSKDVGEIVGKILD 4qmm A 1.852 BS01 35R A 1 I30 G31 K32 A51 L102 G105 L151 I22 G23 K24 A43 L94 G97 L143 D144 K146 A148 N149 D162 D171 T182 D136 K138 A140 N141 D154 D163 T174 2.7.11.1 0004672,0005524,0006468 ic50=0.46uM remove_due_to_license_issue Q9Y6E0 27135311 401 GLPGMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAE 4qmn A 2.091 BS01 DB8 A 1 I30 A51 I52 K53 I97 M99 Y101 L102 L151 D162 I16 A37 I38 K39 I83 M85 Y87 L88 L137 D148 D144 K146 A148 N149 D162 D171 T182 D130 K132 A134 N135 D148 D157 T168 2.7.11.1 0004672,0005524,0006468 ic50=0.003uM remove_due_to_license_issue Kd=380nM, IC50=3.9nM Q9Y6E0 27135311 401 NLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmo A 1.898 BS01 34L A 1 I30 K32 A51 M99 Y101 L102 L151 I22 K24 A43 M91 Y93 L94 L143 D144 K146 A148 N149 D162 D171 T182 D136 K138 A140 N141 D154 D163 T174 2.7.11.1 0004672,0005524,0006468 ic50=0.019uM remove_due_to_license_issue Q9Y6E0 27135311 402 GLPGMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAE 4qmp A 2.0 BS01 DKI A 1 I30 G31 K32 G33 V38 A51 Y101 L102 G105 D109 L151 D162 Y291 I22 G23 K24 G25 V30 A43 Y93 L94 G97 D101 L143 D154 Y283 D144 K146 A148 N149 D162 D171 T182 D136 K138 A140 N141 D154 D163 T174 2.7.11.1 0004672,0005524,0006468 ic50=0.014uM remove_due_to_license_issue Q9Y6E0 27135311 402 GLPGMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmq A 1.769 BS01 34U A 1 I30 A51 M99 E100 Y101 L102 D109 A148 L151 D162 I22 A43 M91 E92 Y93 L94 D101 A140 L143 D154 D144 K146 A148 N149 D162 D171 T182 D136 K138 A140 N141 D154 D163 T174 2.7.11.1 0004672,0005524,0006468 ic50=0.26uM remove_due_to_license_issue Q9Y6E0 27135311 401 GLPGMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qms A 1.883 BS01 1N1 A 1 A51 K53 M99 Y101 L102 G103 L151 D162 A37 K39 M85 Y87 L88 G89 L137 D148 D144 K146 A148 N149 D162 D171 T182 D130 K132 A134 N135 D148 D157 T168 2.7.11.1 0004672,0005524,0006468 ic50=7.4uM remove_due_to_license_issue Kd=>10000nM Q9Y6E0 27135311 401 NLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmt A 1.5 BS01 H1N A 1 I30 G31 G33 V38 A51 M99 Y101 L102 G103 G104 L151 Y291 I16 G17 G19 V24 A37 M85 Y87 L88 G89 G90 L137 Y277 D144 K146 A148 N149 D162 D171 T182 D130 K132 A134 N135 D148 D157 T168 2.7.11.1 0004672,0005524,0006468 ic50=0.01uM remove_due_to_license_issue Q9Y6E0 27135311 401 NLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQS 4qmu A 1.546 BS01 SKE A 1 K32 V38 A51 M99 Y101 L102 D109 L151 D162 Y291 K21 V27 A40 M88 Y90 L91 D98 L140 D151 Y280 D144 K146 A148 N149 D162 D171 T182 D133 K135 A137 N138 D151 D160 T171 2.7.11.1 0004672,0005524,0006468 ic50=1.3uM remove_due_to_license_issue Kd=180nM Q9Y6E0 27135311 401 GMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmv A 2.4 BS01 34W A 1 E28 I30 V38 E100 L102 G105 L151 Y291 E19 I21 V29 E91 L93 G96 L142 Y282 D144 K146 A148 N149 D162 D171 T182 D135 K137 A139 N140 D153 D162 T173 2.7.11.1 0004672,0005524,0006468 ic50=0.023uM remove_due_to_license_issue Q9Y6E0 27135311 401 LPGMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmw A 1.6 BS01 KS1 A 1 A51 K53 E70 T83 M99 L102 L151 A161 D162 A40 K42 E59 T72 M88 L91 L140 A150 D151 D144 K146 A148 N149 D162 D171 T182 D133 K135 A137 N138 D151 D160 T171 2.7.11.1 0004672,0005524,0006468 ic50=0.086uM remove_due_to_license_issue Q9Y6E0 27135311 401 GMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmx A 1.882 BS01 H8H A 1 I30 K32 A51 K53 M99 Y101 L102 I19 K21 A40 K42 M88 Y90 L91 D144 K146 A148 N149 D162 D171 T182 D133 K135 A137 N138 D151 D160 T171 2.7.11.1 0004672,0005524,0006468 ic50=11uM remove_due_to_license_issue Q9Y6E0 27135311 401 GMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQS 4qmy A 1.883 BS01 STU A 1 G31 F35 M99 E100 Y101 L102 L151 D162 G21 F25 M89 E90 Y91 L92 L141 D152 D144 K146 A148 N149 D162 D171 T182 D134 K136 A138 N139 D152 D161 T172 2.7.11.1 0004672,0005524,0006468 ic50=0.004uM remove_due_to_license_issue Q9Y6E0 27135311 401 PGMQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qmz A 1.88 BS01 B49 A 1 I30 A51 M99 E100 Y101 L102 L151 Y291 I18 A39 M87 E88 Y89 L90 L139 Y279 D144 K146 A148 N149 D162 D171 T182 D132 K134 A136 N137 D150 D159 T170 2.7.11.1 0004672,0005524,0006468 ic50=0.21uM remove_due_to_license_issue Kd=63nM Q9Y6E0 27135311 401 MQNLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQS 4qn7 A 2.302 BS02 G39 A 1 R36 D69 I141 R143 R211 N213 R290 Y324 R36 D69 I141 R143 R211 N213 R290 Y324 D69 E196 R211 R290 Y324 D69 E196 R211 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0055036 ic50=0.84nM remove_due_to_license_issue Q20R18 24899180 508 NYLMLNKSLCKVEGWVVVAKDNAIRFGESEQIIVTREPYVSCDPLGCKMYALHQGTTIRNKHSNGTIHDRTAFRGLISTPLGSPPIVSNSDFLCVGWSSTSCHDGIGRMTICVQGNNDNATATVYYDRRLTTTIKTWAGNILRTQESECVCHNGTCVVIMTDGSASSQAYTKVLYFHKGLVIKEEALKGSARHIEECSCYGHNSKVTCVCRDNWQGANRPVIEIDMNAMEHTSQYLCTGVLTDTSRPSDKSIGDCNNPITGSPGAPGVKGFGFLDSGNTWLGRTISPRSRSGFEMLKIPNAGTDPNSRITERQEIVDNNNWSGYSGSFIDYWDESSECYNPCFYVELIRGRPEEAKYVWWTSNSLVALCGSPVPVGSGSFPDGAQIQYFS 4qn9 A 2.652 BS03 DXC A 1 W218 K221 C222 W151 K154 C155 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 504 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNN 4qn9 A 2.652 BS04 DXC A 2 Y159 M160 Y92 M93 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 505 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNN 4qn9 A 2.652 BS05 DXC B 2 W218 R257 W151 R190 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 607 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNN 4qn9 B 2.652 BS01 DXC A 1 Y159 M160 Y92 M93 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 504 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNND 4qn9 B 2.652 BS02 DXC A 2 W218 K221 W151 K154 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 505 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNND 4qn9 B 2.652 BS03 DXC B 1 Y188 R257 Y121 R190 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 601 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNND 4qn9 B 2.652 BS06 DXC B 3 K256 L259 K189 L192 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 608 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNND 4qn9 B 2.652 BS07 DXC B 4 G161 P162 A348 G94 P95 A281 3.1.4.54 0000139,0001523,0001659,0005634,0005635,0005654,0005737,0005768,0005769,0005794,0008270,0009395,0016020,0016787,0030868,0031901,0032052,0042622,0042734,0042802,0045211,0046872,0048874,0050729,0070062,0070290,0070291,0070292,0090336,0098686,0098793 remove_due_to_license_issue Q6IQ20 25684574 610 SKKGKDGRFVNPWPTWKNPSIPNSSVPSSKEELDKELPVLKPYFITNPEEAGVREAGLRVTWLGHATVMVEMDELIFLTDPIFSSRASPSQYMGPKRFRRSPCTISELPPIDAVLISHNHYDHLDYNSVIALNERFGNELRWFVPLGLLDWMQKCGCENVIELDWWEENCVPGHDKVTFVFTPSQHWCKRTLMDDNKVLWGSWSVLGPWNRFFFAGDTGYCPAFEEIGKRFGPFDLAAIPIGAYEPRWFMKYQHVDPEEAVRIHTDVQTKKSMAIHWGTFALANEHYLEPPVKLNEALERYGLNAEDFFVLKHGESRYLNND 4qna A 1.849 BS01 X11 A 1 I30 T83 M99 E100 Y101 L102 I16 T69 M85 E86 Y87 L88 D144 K146 A148 N149 D162 D171 T182 D130 K132 A134 N135 D148 D157 T168 2.7.11.1 0004672,0005524,0006468 ic50=0.023uM remove_due_to_license_issue Q9Y6E0 27135311 401 NLKADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQS 4qnb A 1.996 BS01 1B0 A 1 N53 L56 N57 Q63 M66 K70 T107 Y130 N53 L56 N57 Q63 M66 K70 T107 Y130 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0016032 Kd=0.26uM remove_due_to_license_issue P12497 25518861 301 PIVQNLQGQMVHQCISPRTLNAWVKVVEEKAFSPEVIPMFSALSCGATPQDLNTMLNTVGGHQAAMQMLKETINEEAAEWDRLHPVHAGPIAPGQMREPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYSPTSILDIRQGPKEPFRDYVDRFYKTLRAEQASQEVTETLLVQNANPDCKTILKALGPGATLEEMMTACQ 4qnu A 2.6 BS01 GEK A 1 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 K91 K110 G130 D152 P153 F157 I181 M196 G197 Y200 R315 2.5.1.- 0002098,0006400,0008033,0016740,0016765 remove_due_to_license_issue A1AC32 25855808 401 MIDFGNFYSLIAKNHLSHWLETLPAQIANWQREQQHGLFKQWSNAVEFLPEIKPYRLDLLHSVTAESEEPLSAGQIKRIETLMRNLMPWRKGPFSLYGVNIDTEWRSDWKWDRVLPHLSDLTGRTILDVGCGSGYHMWRMIGAGAHLAVGIDPTQLFLCQFEAVRKLLGNDQRAHLLPLGIEQLPALKAFDTVFSMGVLYHRRSPLEHLWQLKDQLVNEGELVLETLVIDGDENTVLVPGDRYAQMRNVYFIPSALALKNWLKKCGFVDIRIADVSVTTTEEQRRTEWMVTESLADFLDPHDPGKTVEGYPAPKRAVLIARKP 4qo4 A 1.7 BS01 35S A 1 L54 F55 G58 I61 M62 F86 V93 K94 H96 I99 Y100 L37 F38 G41 I44 M45 F65 V72 K73 H75 I78 Y79 2.3.2.27 0005634,0043066,0051726 ic50=0.005uM remove_due_to_license_issue Q00987 25147610 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4qo9 A 2.2 BS01 627 A 1 I30 A51 K53 M99 E100 Y101 L102 G103 G104 L151 Y291 I13 A34 K36 M82 E83 Y84 L85 G86 G87 L134 Y274 D144 K146 A148 N149 D162 D171 T182 D127 K129 A131 N132 D145 D154 T165 2.7.11.1 0004672,0005524,0006468 ic50=0.16uM remove_due_to_license_issue Q9Y6E0 27135311 404 ADPEELFTKLEKIGKGSFGEVFKGIDNRTQKVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSPYVTKYYGSYLKDTKLWIIMEYLGGGSALDLLEPGPLDETQIATILREILKGLDYLHSEKKIHRDIKAANVLLSEHGEVKLADFGVAGQLTDTQIKRNTFVGTPFWMAPEVIKQSAYDSKADIWSLGITAIELARGEPPHSELHPMKVLFLIPKNNPPTLEGNYSKPLKEFVEACLNKEPSFRPTAKELLKHKFILRNAKKTSYLTELIDRYKRWKAEQ 4qoc A 1.7 BS01 35T A 1 L54 G58 I61 M62 Y67 V93 K94 H96 I99 Y100 L36 G40 I43 M44 Y49 V75 K76 H78 I81 Y82 2.3.2.27 0005634,0043066,0051726 ic50=0.12nM remove_due_to_license_issue IC50=0.100000nM Q00987 25042256 201 IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4qp1 A 2.7 BS01 EMU A 1 E33 A52 Q105 D106 M108 L156 E22 A41 Q94 D95 M97 L145 D149 K151 S153 N154 D167 T190 D138 K140 S142 N143 D156 T179 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue P28482 26338362 401 EMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFDDLPKEKLKELIFEETARFQPGYRS 4qp2 A 2.23 BS01 36R A 1 I31 A52 D106 M108 I20 A41 D95 M97 D149 K151 S153 N154 D167 T190 D138 K140 S142 N143 D156 T173 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Kd=940uM remove_due_to_license_issue Kd=940000nM P28482 26338362 401 EMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHYVATRWYRAPEIMLNYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFLDDLPKEKLKELIFEETARFQPGYRS 4qp6 A 3.1 BS01 36N A 1 A52 Q105 D106 M108 L156 A41 Q94 D95 M97 L145 D149 K151 S153 N154 D167 T190 D138 K140 S142 N143 D156 T173 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue Kd=343000nM P28482 26338362 401 EMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHYVATRWYRAPEIMLNYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGYRS 4qp7 A 2.249 BS01 363 A 1 A52 Q105 D106 L107 M108 K114 L156 A40 Q93 D94 L95 M96 K102 L144 D149 K151 S153 N154 D167 T190 D137 K139 S141 N142 D155 T170 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=5.9uM remove_due_to_license_issue IC50=5900nM P28482 26338362 401 MVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 4qp8 A 2.446 BS01 362 A 1 Y36 A52 Q105 D106 L107 M108 T110 K114 L156 Y25 A41 Q94 D95 L96 M97 T99 K103 L145 D149 K151 S153 N154 D167 T190 D138 K140 S142 N143 D156 T168 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.28uM remove_due_to_license_issue IC50=280nM P28482 26338362 401 EMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVAEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 4qp9 A 2.001 BS01 35X A 1 I31 Y36 A52 Q105 D106 M108 K114 L156 I19 Y24 A40 Q93 D94 M96 K102 L144 D149 K151 S153 N154 D167 T190 D137 K139 S141 N142 D155 T170 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.071uM remove_due_to_license_issue IC50=71nM P28482 26338362 401 MVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQPG 4qpa A 2.85 BS01 35W A 1 G32 A50 K52 Q103 D104 M106 K112 L154 C164 G20 A38 K40 Q91 D92 M94 K100 L142 C152 D147 K149 S151 N152 D165 T188 D135 K137 S139 N140 D153 T173 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue IC50=37nM P28482 26338362 401 EMVRFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 4qpd A 2.1 BS01 THG A 1 Q88 F89 I90 I104 G115 A116 D138 G140 L141 D142 Y200 K205 Q88 F89 I90 I104 G115 A116 D138 G140 L141 D142 Y200 K205 H106 D142 H106 D142 1.5.1.6 0003824,0009058 remove_due_to_license_issue E3NZ06 25849409 402 MKIAVIGQSLFGQEVYKELKNEGHMIVGVFTIPDKDGKVDPLAIEAEKDGVPVFKFPRWRLKGKAITEVVDQYKAVGAELNVLPFCSQFIPMEVIDHPKHGSIIYHPSLLPRHRGASAINWTLIHGDKKGGFTVFWADDGLDTGPILLQRECDVEPNDNVNSIYKRFLFPEGVKGMVEAVRLIATGKAPRIKQPEEGATYECIQKKENSKIDWNQPAEAIHNWIRGNDRVPGAWAEIDGKSVSFYGSTLLENDHFSSNGQPLEIPGASRAALVTKNGLVLFGNDGKMLLVKNLQFEDGKMIPGSQYFK 4qpl A 1.9 BS01 V3L A 1 K61 Y107 G109 R110 W114 Y116 I139 Y144 Q153 R161 R163 K175 G179 K32 Y78 G80 R81 W85 Y87 I110 Y115 Q124 R132 R134 K146 G150 2.3.2.27 0008270,0016055,0061630,0072572 Kd=39nM remove_due_to_license_issue Q9CZW6 25327252 201 SLTVPECAICLQTCVHPVSLPCKHVFCYLCVKGASWLGKRCALCRQEIPEDFLDKPTLLSPEELKAASRGNGEYAWYYEGRNGWWQYDERTSRELEDAFSKGKKNTEMLIAGFLYVADLENMVQYRRNEHGRRRKIKRDIIDIPKKGVAGLRL 4qpq A 3.106 BS01 dna P 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHE 4qpq A 3.106 BS02 dna Q 0 K3 S34 F35 S36 A37 K2 S33 F34 S35 A36 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHE 4qpq B 3.106 BS01 dna P 0 S34 F35 S36 S33 F34 S35 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq B 3.106 BS02 dna Q 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq C 3.106 BS01 dna P 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq C 3.106 BS02 dna Q 0 K3 S34 F35 S36 A37 K2 S33 F34 S35 A36 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq D 3.106 BS01 dna P 0 S34 F35 S36 S33 F34 S35 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq D 3.106 BS02 dna Q 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq E 3.106 BS01 dna P 0 K3 S34 F35 S36 A37 K2 S33 F34 S35 A36 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHE 4qpq E 3.106 BS02 dna Q 0 N5 Y7 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHE 4qpq F 3.106 BS01 dna P 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq F 3.106 BS02 dna Q 0 S34 F35 S36 S33 F34 S35 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEAQ 4qpq G 3.106 BS01 dna P 0 K3 S34 F35 S36 K2 S33 F34 S35 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHE 4qpq G 3.106 BS02 dna Q 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHE 4qpq H 3.106 BS01 dna P 0 K3 N5 Y7 K2 N4 Y6 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEA 4qpq H 3.106 BS02 dna Q 0 S34 F35 S36 S33 F34 S35 ? 0003677 remove_due_to_license_issue P10026 25284757 1 ~ 28 AKVNLYISNDAYEKINAIIEKRRQEGAREKDVSFSATASMLLELGLRVHEA 4qps A 1.8 BS01 37Q A 1 L828 V836 A853 M902 Y904 L905 C909 R953 N954 L956 D967 L15 V22 A39 M78 Y80 L81 C85 R129 N130 L132 D143 A949 A951 R953 N954 D967 A125 A127 R129 N130 D143 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue P52333 25552479 1201 PTIFEERHLKYISQLGKGNGSVELCRYDPLGDNTGALVAVKQLDQQRDFQREIQILKALHSDFIVKYRGVSYSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 4qq5 A 2.203 BS01 37O A 1 L478 E480 C482 F483 E525 I539 L555 C557 A558 A559 G561 L624 D635 F636 L32 E34 C36 F37 E74 I88 L104 C106 A107 A108 G110 L160 D171 F172 D617 A619 R621 N622 D635 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 25317566 801 QDPLLAGLVSLDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVILECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLALPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 4qqb A 2.8 BS01 rna P 0 N130 Y131 Q134 D138 R139 Y142 R146 A147 R155 M157 R158 Y160 K161 G163 S165 F166 G167 Y168 F170 K194 R195 K197 A201 R202 G204 V238 N241 L243 F256 R258 E290 N8 Y9 Q12 D16 R17 Y20 R24 A25 R33 M35 R36 Y38 K39 G41 S43 F44 G45 Y46 F48 K72 R73 K75 A79 R80 G82 V116 N119 L121 F134 R136 E168 ? 0003676,0003723,1990904 remove_due_to_license_issue P19339 25209665 4 ~ 20 SNTNLIVNYLPQDMTDRELYALFRAIGPINTCRIMRDYKTGYSFGYAFVDFTSEMDSQRAIKVLNGITVRNKRLKVSYARPGGESIKDTNLYVTNLPRTITDDQLDTIFGKYGSIVQKNILRDKLTGRPRGVAFVRYNKREEAQEAISALNNVIPEGGSQPLSVRLAEE 4qqb B 2.8 BS01 rna C 0 N130 Y131 Q134 D138 R139 Y142 R146 R155 M157 R158 Y160 K161 G163 Y164 F166 Y168 F170 K194 R195 K197 A201 R202 G204 Y214 V238 N241 L243 R252 F256 R258 N8 Y9 Q12 D16 R17 Y20 R24 R33 M35 R36 Y38 K39 G41 Y42 F44 Y46 F48 K72 R73 K75 A79 R80 G82 Y92 V116 N119 L121 R130 F134 R136 ? 0003676,0003723,1990904 remove_due_to_license_issue P19339 25209665 4 ~ 20 SNTNLIVNYLPQDMTDRELYALFRAIGPINTCRIMRDYKTGYSFGYAFVDFTSEMDSQRAIKVLNGITVRNKRLKVSYARPGGESIKDTNLYVTNLPRTITDDQLDTIFGKYGSIVQKNILRDKLTGRPRGVAFVRYNKREEAQEAISALNNVIPEGGSQPLSVRLAEE 4qqb X 2.8 BS01 rna P 0 K13 L15 H16 S17 Y18 F20 R29 F31 H33 R59 K13 L15 H16 S17 Y18 F20 R29 F31 H33 R59 ? 0003676 remove_due_to_license_issue B7Z0E2 25209665 4 ~ 20 GAMATRETGIIEKLLHSYGFIQCCERQARLFFHFSQFSGNIDHLKIGDPVEFEMTYDRRTGKPIASQVSKIA 4qqb Y 2.8 BS01 rna C 0 K13 L15 H16 S17 Y18 F20 R29 F31 H33 K62 K13 L15 H16 S17 Y18 F20 R29 F31 H33 K62 ? 0003676 remove_due_to_license_issue B7Z0E2 25209665 4 ~ 20 GAMATRETGIIEKLLHSYGFIQCCERQARLFFHFSQFSGNIDHLKIGDPVEFEMTYDRRTGKPIASQVSKIA 4qqc A 2.4 BS01 37O A 1 L473 E475 C477 F478 I534 V550 C552 A553 L619 D630 L31 E33 C35 F36 I87 V103 C105 A106 L159 D170 D612 A614 R616 N617 D630 D152 A154 R156 N157 D170 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 25349422 801 DPLLAGLVSLDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 4qr3 A 1.374 BS01 BNJ A 1 W81 P82 V87 L92 I146 W40 P41 V46 L51 I105 ? ic50=1.4uM remove_due_to_license_issue IC50=1400nM O60885 25559428 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4qr4 A 1.28 BS01 BNK A 1 P82 V87 L92 I146 P41 V46 L51 I105 ? ic50=0.25uM remove_due_to_license_issue IC50=250nM O60885 25559428 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4qr5 A 1.41 BS01 BNM A 1 W81 P82 Q85 L92 I146 W40 P41 Q44 L51 I105 ? ic50=0.06uM remove_due_to_license_issue IC50=60nM O60885 25559428 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4qrc A 1.901 BS01 0LI A 1 L473 A501 K503 E520 M524 V550 C552 A553 L603 C608 I609 H610 R611 L619 A629 D630 F631 L633 L20 A48 K50 E67 M71 V97 C99 A100 L150 C155 I156 H157 R158 L166 A176 D177 F178 L180 D612 A614 R616 N617 D630 R650 D159 A161 R163 N164 D177 R197 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=8.0nM P22455 25317566 802 LPLDPLWEFPRDRLVLGKPLGEGAFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPDLSPDGPRSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 4qrh B 1.65 BS01 0O2 B 1 G16 V17 G18 K19 S39 R43 Y55 E74 Y78 Y83 G84 E103 I104 E105 G15 V16 G17 K18 S38 R42 Y54 E73 Y77 Y82 G83 E102 I103 E104 2.7.4.8 0004385,0005524,0005737,0005829,0006163,0016301,0046037,0046710 Ki=7uM remove_due_to_license_issue A0A0J9X1Z9 25661490 303 DNEKGLLIVLSGPSGVGKGTVRKRIFEDPSTSYKYSISMTTRQMREGEVDGVDYFFKTRDAFEALIKDDQFIEYAEYVGNYYGTPVQYVKDTMDEGHDVFLEIEVEGAKQVRKKFPDALFIFLAPPSLEHLNEARKEVEMMNLYDYVVVNDEVELAKNRIQCIVEAEHLKRERVEAKYRKMILEAK 4qsh A 2.51 BS02 2BA A 1 Y722 Y749 A753 S756 Y653 Y680 A684 S687 K710 K641 0003824,0004736,0005524,0006090,0006094,0046872 remove_due_to_license_issue 25215494 2003 HMMNRIKKVLVANRGEIAIRVMRACTELKIKTVAIYSQEDTGSFHRYKSDEAYLVGAGKKPIDAYLDIENIIEIAKESGADAIHPGYGFLSENIEFARRCEQEGIIFVGPKSKHLDMFGDKIKAKEQALLADIPVIVMNPKHIEVQILGDTHGNIVHLFERDCSIQRRHQKVVEVAPCNAITSELRNRICDAAVKLMKNVDYINAGTVEFLVEGDDFYFIEVNPRVQVEHTITEMITGIDIVQSQLFIADGYALHDQLVAIPKQEDIHIHGSAIQSRITTEDPLNNFMPDTGRVDTYRSTGGFGVRLDAGNGFQGTVVTPFYDSLLVKLCTWGMTFEQATRKMRRNLIEFRIRGVKTNIPFLLNVVRHPDFASGNYNTSFIDTTPELFKFPHIRDRGTKTLRYIGNVTVNGFPGIKHRDKPVYAEPRLPKIPYGSQISPGTKQILDAKGPEGVVDWVKKQEEVLLTDTTLRDAHQSLLATRVRSKDIFQIADAMAHLLPNMFSFEMWGGATFDVAYRFLNEDPWVRLETLRKQIPNVMFQMLLRGANAVGYKNYPDNVIREFVKQSAQSGVDVFRVFDSLNWIKGMEVSIDAVREAGKIVEAAICYTGDIDDDTRTKYTIDYYKDMAKELVAQGTHILGIKDMAGLLKPQAAYRLIGELKDTVDVPIHLHTHDTSGNGIYTYAAAVSAGVDIVDVASSAMSGATSQPSMTGLYYGLVNGNRQTNLDAQNSQIINHYWEDVRHYYKDFDNALNSPQTEVYIHEMPGGQYTNLQQQAIAVGLGDRWDEVKEMYTVVNQMFGDIVKVTPSSKVVGDLALFMVQNELSEEDVYEKGDTIDFPDSVIEFFMGEIGQPYGGFPEKLQKLVLKGRTPLTDRPGALMEPVNFVEVKAELKEKMGYEPTEKDVISYILYPKVFLDYQEMINKYGDVTVLDTPTFYKGMRLGETIEVELEKGKILLIKLNSIGEPIADGTRVIYFELNGQPREINIQDMNVQARRKIDTTNPEHVGATMTGSVIQVVVKKGDSVKKGDPLLITEAMKMETTIQAPFDGEVSSIYVSDGDTIESGDLLIEVNR 4qsh D 2.51 BS01 2BA A 1 Y722 Y749 A753 S756 Y654 Y681 A685 S688 K710 K642 0003824,0004736,0005524,0006090,0006094,0046872 remove_due_to_license_issue 25215494 2003 MMNRIKKVLVANRGEIAIRVMRACTELKIKTVAIYSQEDTGSFHRYKSDEAYLVGAGKKPIDAYLDIENIIEIAKESGADAIHPGYGFLSENIEFARRCEQEGIIFVGPKSKHLDMFGDKIKAKEQALLADIPVIPCVMNPKHIEVQILGDTHGNIVHLFERDCSIQRRHQKVVEVAPCNAITSELRNRICDAAVKLMKNVDYINAGTVEFLVEGDDFYFIEVNPRVQVEHTITEMITGIDIVQSQLFIADGYALHDQLVAIPKQEDIHIHGSAIQSRITTEDPLNNFMPDTGRVDTYRSTGGFGVRLDAGNGFQGTVVTPFYDSLLVKLCTWGMTFEQATRKMRRNLIEFRIRGVKTNIPFLLNVVRHPDFASGNYNTSFIDTTPELFKFPHIRDRGTKTLRYIGNVTVNGFPGIKHRDKPVYAEPRLPKIPYGSQISPGTKQILDAKGPEGVVDWVKKQEEVLLTDTTLRDAHQSLLATRVRSKDIFQIADAMAHLLPNMFSFEMWGGATFDVAYRFLNEDPWVRLETLRKQIPNVMFQMLLRGANAVGYKNYPDNVIREFVKQSAQSGVDVFRVFDSLNWIKGMEVSIDAVREAGKIVEAAICYTGDIDDDTRTKYTIDYYKDMAKELVAQGTHILGIKDMAGLLKPQAAYRLIGELKDTVDVPIHLHTHDTSGNGIYTYAAAVSAGVDIVDVASSAMSGATSQPSMTGLYYGLVNGNRQTNLDAQNSQIINHYWEDVRHYYKDFDNALNSPQTEVYIHEMPGGQYTNLQQQAIAVGLGDRWDEVKEMYTVVNQMFGDIVKVTPSSKVVGDLALFMVQNELSEEDVYEKGDTIDFPDSVIEFFMGEIGQPYGGFPEKLQKLVLKGRTPLTDRPGALMEPVNFVEVKAELKEKMGYEPTEKDVISYILYPKVFLDYQEMINKYGDVTVLDTPTFYKGMRLGETIEVELEKGKILLIKLNSIGEPIADGTRVIYFELNGQPREINIQDMNVARRKIDTTNPEHVGATMTGSVIQVVVKKGDSVKKGDPLLITEAMKMETTIQAPFDGEVSSIYVSDGDTIESGDLLIEVNR 4qsk A 2.7 BS01 2BA A 1 Y722 Y749 A753 S756 Y654 Y681 A685 S688 K710 K642 0003824,0004736,0005524,0006090,0006094,0046872 remove_due_to_license_issue 25215494 2000 MMNRIKKVLVANRGEIAIRVMRACTELKIKTVAIYSQEDTGSFHRYKSDEAYLVGAGKKPIDAYLDIENIIEIAKESGADAIHPGYGFLSENIEFARRCEQEGIIFVGPKSKHLDMFGDKIKAKEQALLADIPVIPCVMNPKHIEVQILGDTHGNIVHLFERDCSIQRRHQKVVEVAPCNAITSELRNRICDAAVKLMKNVDYINAGTVEFLVEGDDFYFIEVNPRVQVEHTITEMITGIDIVQSQLFIADGYALHDQLVAIPKQEDIHIHGSAIQSRITTEDPLNNFMPDTGRVDTYRSTGGFGVRLDAGNGFQGTVVTPFYDSLLVKLCTWGMTFEQATRKMRRNLIEFRIRGVKTNIPFLLNVVRHPDFASGNYNTSFIDTTPELFKFPHIRDRGTKTLRYIGNVTVNGFPGIKHRDKPVYAEPRLPKIPYGSQISPGTKQILDAKGPEGVVDWVKKQEEVLLTDTTLRDAHQSLLATRVRSKDIFQIADAMAHLLPNMFSFEMWGGATFDVAYRFLNEDPWVRLETLRKQIPNVMFQMLLRGANAVGYKNYPDNVIREFVKQSAQSGVDVFRVFDSLNWIKGMEVSIDAVREAGKIVEAAICYTGDIDDDTRTKYTIDYYKDMAKELVAQGTHILGIKDMAGLLKPQAAYRLIGELKDTVDVPIHLHTHDTSGNGIYTYAAAVSAGVDIVDVASSAMSGATSQPSMTGLYYGLVNGNRQTNLDAQNSQIINHYWEDVRHYYKDFDNALNSPQTEVYIHEMPGGQYTNLQQQAIAVGLGDRWDEVKEMYTVVNQMFGDIVKVTPSSKVVGDLALFMVQNELSEEDVYEKGDTIDFPDSVIEFFMGEIGQPYGGFPEKLQKLVLKGRTPLTDRPGALMEPVNFVEVKAELKEKMGYEPTEKDVISYILYPKVFLDYQEMINKYGDVTVLDTPTFYKGMRLGETIEVELEKGKILLIKLNSIGEPIADGTRVIYFELNGQPREINIQDMNVQARRKIDTTNPEHVGATMTGSVIQVVVKKGDSVKKGDPLLITEAMKMETTIQAPFDGEVSSIYVSDGDTIESGDLLIEVNR 4qsm A 3.0 BS01 38K A 1 D52 V53 A96 G97 R99 N115 I116 F119 D51 V52 A95 G96 R98 N114 I115 F118 R106 D166 R169 H193 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 remove_due_to_license_issue IC50=4800nM P00338 25664730 501 ATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQFH 4qsu A 1.9 BS01 TDR A 1 V1013 N1064 I1074 V35 N86 I96 3.6.1.- remove_due_to_license_issue Q6PL18 1210 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4qsw A 1.8 BS01 38T A 1 V1008 D1014 E1017 N1064 I1074 V30 D36 E39 N86 I96 3.6.1.- remove_due_to_license_issue Q6PL18 1207 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4qsx A 1.93 BS01 38S A 1 V1008 Y1063 N1064 I1074 V30 Y85 N86 I96 3.6.1.- remove_due_to_license_issue Q6PL18 1207 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4qt0 A 3.2 BS01 38Q A 1 D52 V53 A96 G97 R99 I116 F119 D51 V52 A95 G96 R98 I115 F118 R106 D166 R169 H193 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 remove_due_to_license_issue P00338 25664730 501 ATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQFH 4qt1 A 2.4 BS01 3C9 A 1 L828 G829 K830 V836 A853 Y904 L905 L956 L15 G16 K17 V23 A40 Y85 L86 L137 D949 A951 R953 N954 D967 D130 A132 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM remove_due_to_license_issue IC50=7.0nM P52333 25262541 1201 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGS 4qt2 A 1.44 BS01 RAP A 1 Y44 D56 F65 G72 E73 V74 I75 W78 Y101 Y38 D50 F59 G66 E67 V68 I69 W72 Y95 Y44 F55 D56 I75 Y101 F118 Y38 F49 D50 I69 Y95 F112 5.2.1.8 0003755 ic50=0.48uM remove_due_to_license_issue Q8I4V8 26057671 202 FEKVELTADGGVIKTILKKGDEGEENIPKKGNEVTVHYVGKLESTGKVFDSSFDRNVPFKFHLEQGEVIKGWDICVSSMRKNEKCLVRIESMYGYGDEGCGESIPGNSVLLFEIELLSFREL 4qta A 1.45 BS01 38Z A 1 I31 A35 Y36 A52 K54 I56 Y64 T68 E71 Q105 D106 M108 E109 T110 K114 L156 C166 D167 I22 A26 Y27 A43 K45 I47 Y55 T59 E62 Q96 D97 M99 E100 T101 K105 L147 C157 D158 D149 K151 S153 N154 D167 T190 D140 K142 S144 N145 D158 T167 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Kd=0.233uM remove_due_to_license_issue P28482 25195011 411 GPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADTRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 4qtb A 1.4 BS01 38Z A 1 A52 Y53 A69 K71 I73 Y81 R84 T85 E88 Q122 D123 M125 E126 T127 K131 L173 C183 D184 A29 Y30 A46 K48 I50 Y58 R61 T62 E65 Q99 D100 M102 E103 T104 K108 L150 C160 D161 D166 K168 S170 N171 D184 T207 D143 K145 S147 N148 D161 T184 2.7.11.24 0000165,0001784,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005635,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005829,0005856,0005886,0005901,0005925,0006351,0006468,0006915,0006974,0007254,0008286,0009887,0010759,0014032,0014044,0016020,0016310,0019233,0019902,0030278,0030509,0030641,0030878,0031143,0031281,0031663,0032206,0032496,0032872,0033554,0034198,0035556,0038083,0038133,0042473,0042552,0042770,0042802,0043330,0045944,0048009,0048538,0050804,0051216,0051403,0051493,0060020,0060324,0060425,0060440,0061308,0070161,0070371,0070374,0070498,0070849,0071260,0071356,0072584,0090170,0098792,0098978,0106310,0120041,0140297,1904262,1904417,2000641 Kd=0.213uM remove_due_to_license_issue P27361 25195011 418 VPGEVEMVKGQPFDVGPRYTQLQYIGEGAYGMVSSAYDHVRKTRVAIKKISPFEHQTYCQRTLREIQILLRFRHENVIGIRDILRASTLEAMRDVYIVQDLMETDLYKLLKSQQLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLINTTCDLKICDFGLARIADPEHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINMKARNYLQSLPSKTKVAWAKLFPKSDSKALDLLDRMLTFNPNKRITVEEALAHPYLEQYYDPTDEPVAEEPFTFAMELDDLPKERLKELIFQETARFQPG 4qtc A 1.4 BS01 38Z A 1 I490 G491 E492 A509 Y580 G585 S586 A587 G608 L656 I686 I22 G23 E24 A41 Y112 G117 S118 A119 G140 L188 I218 2.7.11.1 0004672,0005524,0006468 Kd=0.297uM remove_due_to_license_issue Q8TF76 25195011 804 QKGPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 4qtd A 1.5 BS01 38Z A 1 V40 A53 M108 L110 M111 D112 A113 N114 C116 Q117 Q120 S155 N156 L168 V35 A48 M103 L105 M106 D107 A108 N109 C111 Q112 Q115 S150 N151 L163 D151 K153 N156 D169 T188 D146 K148 N151 D164 T180 2.7.11.24 0004672,0004707,0005524,0006468 ic50=1080nM remove_due_to_license_issue P45983 25195011 424 RDNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTSFMMTPYVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDL 4qtl A 1.8 BS02 WWO A 1 N62 Q92 H94 H96 H119 V121 F131 L198 T199 T200 N59 Q89 H91 H93 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=120nM remove_due_to_license_issue Kd=6.1nM P00918 25758852 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4qtn A 2.8 BS01 NNR A 1 C53 V54 V57 Q171 W182 W185 N189 C52 V53 V56 Q170 W181 W184 N188 ? 0005886,0016020,0034257,0034258,0042802,0070207 remove_due_to_license_issue D2ZZC1 301 GSLAWWKRELFGGWTHFEAVWLLMFLGIQAVVFVFNPDSWLASVAAVTGILCVVFVGKGKISNYLFGLISVSLYAYVSYTFKLYGEMMLNLLVYVPVQFVGFAMWRKHMALGETAETEEVKAKALTVRQWLLVVAASVVGTSVYIEWLHHLGSALPTLDGVTVVVSIVAQVLMILRYREQWALWIVVNILTISLWAVAWFKNGETSLPLLLMYVMYLCNSVYGYINWTKLVKRHS 4quo A 1.65 BS01 3DZ A 1 Q115 E117 M256 G257 A258 M259 E260 V290 H293 E294 H297 E316 Y377 Q113 E115 M254 G255 A256 M257 E258 V288 H291 E292 H295 E314 Y375 E260 H293 E294 H297 E316 N369 Y377 E258 H291 E292 H295 E314 N367 Y375 3.4.11.2 0004177,0006508,0008237,0008270,0046872 Ki=12nM remove_due_to_license_issue Q9JYV4 25192493 901 KTVHYLKDYQTPAYHILKTDLHFDINEPQTVVKSRLTVEPQRVGEPLVLDGSAKLLSVKINGAAADYVLEGETLTIAGVPSERFTVEVETEILPAENKSLMGLYASGGNLFTQCEPEGFRKITFYIDRPDVMSKFTTTIVADKKRYPVLLSNGNKIDGGEFSDGRHWVKWEDPFSKPSYLFALVAGDLAVTEDYFTTMSGRNVKIEFYTTEADKPKVGFAVESLKNAMKWDETRFGLEYDLDIFMVVAVGDFNMGAMENKGLNIFNTKFVLADSRTATDTDFEGIESVVGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSGDRASRAVRRIENIRLLRQHQFPEDAGPTAHPVRPASYEEMNNFYTMTVYEKGAEVVRMYHTLLGEEGFQKGMKLYFQRHDGQAVTCDDFRAAMADANGINLDQFALWYSQAGTPVLEAEGRLKNNIFELTVKQTVPPTPDMTDKQPMMIPVKVGLLNRNGEAVAFDYQGKRATEAVLLLTEAEQTFLLEGVTEAVVPSLLRGFSAPVHLNYPYSDDDLLLLLAHDSDAFTRWEAAQTLYRRAVAANLATLSDGVELPKHEKLLAAVEKVISDDLLDNAFKALLLGVPSEAELWDGAENIDPLRYHQAREALLDTLAVHFLPKWHELNRQAAKQENQSYEYSPEAAGWRTLRNVCRAFVLRADPAHIETVAEKYGEMAQNMTHEWGILSAVNGNESDTRNRLLAQFADKFSDDALVMDKYFALVGSSRRSDTLQQVRTALQHPKFSLENPNKARSLIGSFSRNVPHFHAEDGSGYRFIADKVIEIDRFNPQVAARLVQAFNLCNKLEPHRKNLVKQALQRIRAQEGLSKDVGEIVGKILD 4quo A 1.65 BS03 3DZ A 2 N156 P175 F176 R203 D242 L243 D244 N154 P173 F174 R201 D240 L241 D242 E260 H293 E294 H297 E316 N369 Y377 E258 H291 E292 H295 E314 N367 Y375 3.4.11.2 0004177,0006508,0008237,0008270,0046872 Ki=12nM remove_due_to_license_issue Q9JYV4 25192493 908 KTVHYLKDYQTPAYHILKTDLHFDINEPQTVVKSRLTVEPQRVGEPLVLDGSAKLLSVKINGAAADYVLEGETLTIAGVPSERFTVEVETEILPAENKSLMGLYASGGNLFTQCEPEGFRKITFYIDRPDVMSKFTTTIVADKKRYPVLLSNGNKIDGGEFSDGRHWVKWEDPFSKPSYLFALVAGDLAVTEDYFTTMSGRNVKIEFYTTEADKPKVGFAVESLKNAMKWDETRFGLEYDLDIFMVVAVGDFNMGAMENKGLNIFNTKFVLADSRTATDTDFEGIESVVGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSGDRASRAVRRIENIRLLRQHQFPEDAGPTAHPVRPASYEEMNNFYTMTVYEKGAEVVRMYHTLLGEEGFQKGMKLYFQRHDGQAVTCDDFRAAMADANGINLDQFALWYSQAGTPVLEAEGRLKNNIFELTVKQTVPPTPDMTDKQPMMIPVKVGLLNRNGEAVAFDYQGKRATEAVLLLTEAEQTFLLEGVTEAVVPSLLRGFSAPVHLNYPYSDDDLLLLLAHDSDAFTRWEAAQTLYRRAVAANLATLSDGVELPKHEKLLAAVEKVISDDLLDNAFKALLLGVPSEAELWDGAENIDPLRYHQAREALLDTLAVHFLPKWHELNRQAAKQENQSYEYSPEAAGWRTLRNVCRAFVLRADPAHIETVAEKYGEMAQNMTHEWGILSAVNGNESDTRNRLLAQFADKFSDDALVMDKYFALVGSSRRSDTLQQVRTALQHPKFSLENPNKARSLIGSFSRNVPHFHAEDGSGYRFIADKVIEIDRFNPQVAARLVQAFNLCNKLEPHRKNLVKQALQRIRAQEGLSKDVGEIVGKILD 4qvc D 1.99 BS01 rna G 0 Y25 N28 G29 I30 K31 Y20 N23 G24 I25 K26 ? 0003723,0006355 remove_due_to_license_issue C1IFD2 25670676 1 ~ 4 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4qvd D 1.972 BS01 rna H 0 Y25 N28 G29 I30 K31 T61 Y20 N23 G24 I25 K26 T56 ? 0003723,0006355 remove_due_to_license_issue C1IFD2 25670676 4 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4qvd E 1.972 BS01 rna H 0 I30 K31 L32 Q33 Q52 I25 K26 L27 Q28 Q47 ? 0003723,0006355 remove_due_to_license_issue C1IFD2 25670676 4 ~ 7 SLQDPFLNALRRERVPVSIYLVNGIKLQGQIESFDQFVILLKNTVSQMVYKHAISTVVPS 4qvi A 1.9 BS01 rna B 0 M0 H3 G4 K5 R6 Y7 A35 K36 T40 E42 H44 K46 R134 D166 T168 H172 S211 Y213 T215 T217 L218 G219 S221 M1 H4 G5 K6 R7 Y8 A36 K37 T41 E43 H45 K47 R135 D167 T169 H173 S212 Y214 T216 T218 L219 G220 S222 ? 0000049,0003723,0003735,0005840,0006412,0006417,0015934,0019843,1990904 remove_due_to_license_issue P27150 25664749 2105 ~ 2184 MPKHGKRYRALLEKVDPNKIYTIDEAAHLVKELATAKFDETVEVHAKLGIDPRRSDQNVRGTVSLPHGLGKQVRVLAIAKGEKIKEAEEAGADYVGGEEIIQKILDGWMDFDAVVATPDVMGAVGSKLGRILGPRGLLPNPKAGTVGFNIGEIIREIKAGRIEFRNDKTGAIHAPVGKASFPPEKLADNIRAFIRALEAHKPEGAKGTFLRSVYVTTTLGPSVRINPHS 4qvl H 2.8 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvm H 2.8 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvm I 2.8 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qvn H 2.9 BS01 BO2 H 1 T1 S20 T21 Q22 G47 A49 T1 S20 T21 Q22 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvp H 2.3 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvp I 2.3 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qvq H 2.6 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvq I 2.6 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qvv H 2.8 BS01 BO2 H 1 T1 S20 T21 Q22 G47 A49 T1 S20 T21 Q22 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvv I 2.8 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qvw H 3.0 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvw I 3.0 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qvx A 2.1 BS01 3CQ A 1 E96 F97 Y101 R102 F105 S106 L108 N136 G138 R139 A142 S145 F146 A149 Y195 E36 F37 Y41 R42 F45 S46 L48 N76 G78 R79 A82 S85 F86 A89 Y135 ? 0042981 Ki<0.01nM remove_due_to_license_issue Ki=<0.010000nM Q07817 25313317 301 SQSNRELVVDFLSYKLSQKGYGMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKKMQVLVSRIAAWMATYLNDHLEPWIQENGGWATFVELYG 4qvy H 2.51 BS01 BO2 H 1 T1 S20 T21 Q22 K33 G47 A49 T1 S20 T21 Q22 K33 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qvy I 2.51 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qw0 H 2.9 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qw0 I 2.9 BS01 BO2 H 1 D124 C128 D124 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qw1 H 2.9 BS01 BO2 H 1 T1 S20 T21 Q22 G47 A49 T1 S20 T21 Q22 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qw3 H 2.9 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qw4 H 2.8 BS01 3BV H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw4 H 2.8 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw4 Z 2.8 BS01 3BV Y 1 R101 H108 D126 P127 R101 H108 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qw5 H 3.0 BS01 3BV H 1 T1 S20 T21 G47 T48 A49 G168 T1 S20 T21 G47 T48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw5 H 3.0 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw5 Z 3.0 BS01 3BV Y 1 R101 H108 D126 P127 V128 R101 H108 D126 P127 V128 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qw6 H 2.9 BS01 3BV H 1 T1 S20 T21 G47 T48 A49 G168 T1 S20 T21 G47 T48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw6 H 2.9 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw6 Z 2.9 BS01 3BV Y 1 R101 H108 D126 P127 V128 R101 H108 D126 P127 V128 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qw7 H 2.7 BS01 3BV H 1 T1 S20 T21 G47 T48 A49 S129 T1 S20 T21 G47 T48 A49 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw7 H 2.7 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qw7 I 2.7 BS01 3BV H 1 D124 I126 D124 I126 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qw7 Z 2.7 BS01 3BV Y 1 H108 D126 P127 V128 H108 D126 P127 V128 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwf H 3.0 BS01 3BV H 1 T1 S20 T21 G47 A49 G168 T1 S20 T21 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwf H 3.0 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwf Z 3.0 BS01 3BV Y 1 R101 H108 D126 P127 V128 R101 H108 D126 P127 V128 ? 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwg H 2.6 BS01 3BV H 1 T1 S20 T21 G47 A49 S129 T1 S20 T21 G47 A49 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwg H 2.6 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwg I 2.6 BS01 3BV H 1 D124 L125 D124 L125 ? 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qwg Z 2.6 BS01 3BV Y 1 H108 D126 P127 H108 D126 P127 ? 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwi H 2.6 BS01 3BV H 1 T1 S20 T21 G47 T48 A49 T1 S20 T21 G47 T48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwi H 2.6 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwi I 2.6 BS01 3BV H 1 D124 I126 C128 D124 I126 C128 ? 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qwi Z 2.6 BS01 3BV Y 1 R101 H108 D126 P127 V128 R101 H108 D126 P127 V128 ? 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwj H 2.9 BS01 3BV H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwj H 2.9 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwj I 2.9 BS01 3BV H 1 D124 I126 D124 I126 ? 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qwj Z 2.9 BS01 3BV Y 1 H108 D126 P127 V128 H108 D126 P127 V128 ? 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwk H 2.8 BS01 3BV H 1 T1 S20 T21 A46 G47 A49 T1 S20 T21 A46 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwk H 2.8 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwk Z 2.8 BS01 3BV Y 1 R101 H108 D126 P127 R101 H108 D126 P127 ? 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwl H 2.6 BS01 3BV H 1 T1 S20 T21 A46 G47 T48 A49 T1 S20 T21 A46 G47 T48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwl H 2.6 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwl I 2.6 BS01 3BV H 1 D124 I126 D124 I126 ? 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qwl Z 2.6 BS01 3BV Y 1 R101 H108 D126 P127 R101 H108 D126 P127 ? 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwr H 2.9 BS01 3BV H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwr H 2.9 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qwr I 2.9 BS01 3BV H 1 D124 L125 I126 C128 D124 L125 I126 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 25599643 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 4qwr Z 2.9 BS01 3BV Y 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qws H 3.0 BS01 3BV H 1 T1 S20 T21 G47 T48 A49 G168 T1 S20 T21 G47 T48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qws H 3.0 BS02 3BV N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qws Z 3.0 BS01 3BV Y 1 R101 H108 D126 P127 V128 R101 H108 D126 P127 V128 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25599643 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4qwu H 3.0 BS01 BO2 H 1 T1 S20 T21 G47 A49 T1 S20 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 4qwx H 2.9 BS01 04C H 1 T1 S20 T21 Q22 G47 A49 T52 G168 T1 S20 T21 Q22 G47 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qxj H 2.8 BS01 04C H 1 T1 S20 T21 G47 A49 T52 G168 T1 S20 T21 G47 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qxo A 1.88 BS01 1YE A 1 S162 Y163 Y167 T263 P264 T267 S9 Y10 Y14 T110 P111 T114 ? 0002218,0032481 Kd=3.12uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFRDMLPQQNIDRAGIKNRVYSNSVYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxq A 2.42 BS01 1YE A 1 A162 Y163 Y167 T263 T267 A9 Y10 Y14 T110 T114 ? 0002218,0032481 Kd=1.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxq A 2.42 BS02 1YE B 1 G166 I235 R238 G13 I82 R85 ? 0002218,0032481 Kd=1.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxq B 2.42 BS01 1YE A 1 G166 R238 G13 R85 ? 0002218,0032481 Kd=1.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxq B 2.42 BS02 1YE B 1 A162 T263 P264 T267 A9 T110 P111 T114 ? 0002218,0032481 Kd=1.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxr A 2.37 BS01 1YE A 1 A162 Y167 T263 P264 T267 A9 Y14 T110 P111 T114 ? 0002218,0032481 Kd=0.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTIDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxr A 2.37 BS02 1YE B 1 G166 R238 G13 R85 ? 0002218,0032481 Kd=0.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTIDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxr B 2.37 BS01 1YE A 1 G166 R238 G13 R85 ? 0002218,0032481 Kd=0.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTIDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxr B 2.37 BS02 1YE B 1 A162 T263 T267 A9 T110 T114 ? 0002218,0032481 Kd=0.99uM remove_due_to_license_issue Q86WV6 25199835 401 SVAHGLAWAYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTIDRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLITLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 4qxs F 1.9 BS02 WC1 F 1 K57 N59 R60 S205 F206 F239 D243 K347 K48 N50 R51 S196 F197 F230 D234 K338 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.1uM remove_due_to_license_issue IC50=1100nM P14324 25630225 403 YAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 4qy3 A 1.5 BS02 3G1 A 1 G6 Y7 G8 F231 N232 E236 E239 G3 Y4 G5 F227 N228 E232 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.15uM remove_due_to_license_issue P00918 25407638 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4qye A 2.05 BS01 3DL A 1 L15 V23 K38 L84 Y86 C87 E91 L137 D148 L13 V21 K36 L75 Y77 C78 E82 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.2uM remove_due_to_license_issue IC50=1200nM O14757 25453805 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS 4qyg A 1.75 BS01 3DW A 1 L15 A36 K38 L84 Y86 C87 L137 D148 L13 A34 K36 L75 Y77 C78 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.0041uM remove_due_to_license_issue IC50=>10000nM O14757 25453805 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 4qyh A 1.9 BS01 3DX A 1 L15 A36 L84 E85 Y86 C87 E91 L137 D148 L13 A34 L75 E76 Y77 C78 E82 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.0013uM remove_due_to_license_issue IC50=1.3nM, EC50=98nM O14757 25453805 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 4qyy A 1.65 BS01 3G7 A 1 A33 Y34 A50 K52 I54 Y62 R65 E69 Q103 D104 L105 M106 L154 D165 A21 Y22 A38 K40 I42 Y50 R53 E57 Q91 D92 L93 M94 L142 D153 D147 K149 S151 N152 D165 T188 D135 K137 S139 N140 D153 T176 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 Kd=0.05uM remove_due_to_license_issue P63086 25313996 401 RGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKLDDLPKEKLKELIFEETARFQ 4qz0 H 3.0 BS01 04C H 1 T1 S20 T21 Q22 G47 T48 A49 T52 G168 T1 S20 T21 Q22 G47 T48 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz1 H 3.0 BS01 04C H 1 T1 S20 T21 Q22 G47 A49 G168 T1 S20 T21 Q22 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz2 H 2.7 BS01 04C H 1 T1 S20 T21 Q22 G47 A49 T52 G168 T1 S20 T21 Q22 G47 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz3 H 2.8 BS01 04C H 1 T1 S20 T21 C31 G47 T48 A49 G168 T1 S20 T21 C31 G47 T48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz4 H 3.0 BS01 04C H 1 T1 S20 T21 Q22 G47 T48 A49 T52 G168 T1 S20 T21 Q22 G47 T48 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz5 H 2.8 BS01 04C H 1 T1 S20 T21 C31 G47 A49 T52 G168 T1 S20 T21 C31 G47 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz6 H 2.9 BS01 04C H 1 T1 S20 T21 G47 T48 A49 G168 T1 S20 T21 G47 T48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qz7 H 2.8 BS01 04C H 1 T1 T21 A46 G47 T48 A49 T52 G168 T1 T21 A46 G47 T48 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qzs A 1.45 BS01 JQ1 A 1 W81 P82 L92 X97 X139 N140 I146 M149 W40 P41 L51 X56 X98 N99 I105 M108 ? Kd=89nM remove_due_to_license_issue O60885 25290579 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4qzw H 3.0 BS01 04C H 1 T1 S20 T21 Q22 G47 A49 T52 G168 T1 S20 T21 Q22 G47 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4qzx H 2.6 BS01 04C H 1 T1 S20 T21 Q22 G47 A49 T52 G168 T1 S20 T21 Q22 G47 A49 T52 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 25599643 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 4r02 K 2.5 BS01 3E5 K 1 T1 T21 M45 A46 G47 A49 S131 T1 T21 M45 A46 G47 A49 S131 T1 D17 R19 K33 G47 S131 D168 S171 T1 D17 R19 K33 G47 S131 D168 S171 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25087721 301 TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4r02 L 2.5 BS01 3E5 K 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 25087721 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 4r06 A 2.22 BS01 3E7 A 1 I281 F282 G284 C285 R288 S289 H323 Y327 L330 V339 I341 M364 H449 L453 Y473 I58 F59 G61 C62 R65 S66 H100 Y104 L107 V116 I118 M141 H226 L230 Y250 ? 0003677,0004879,0005634,0006355 Kd=565nM remove_due_to_license_issue IC50=7nM P37231 26579553 501 PESADLRALAKHLYDSYIKSFPLTKAKARAILTTTDKSPFVIYDMNSLMMGEEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKD 4r07 A 2.0 BS03 UCG A 1 K314 V315 E340 I341 D343 H373 R375 H469 T471 R472 P473 L474 K267 V268 E293 I294 D296 H326 R328 H398 T400 R401 P402 L403 ? 0002224,0004888,0006955,0016020 Kd=4.8uM remove_due_to_license_issue Q9NR97 25599397 902 RSYPCDEKVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPTDFEFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSALETKTTTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 4r0a A 1.9 BS01 URI A 1 Y348 K350 G351 Y353 F405 R429 Y305 K307 G308 Y310 F362 R386 ? 0002224,0004888,0006955,0016020 Kd=55uM remove_due_to_license_issue Q9NR97 25599397 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLEFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSALETKTTTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSL 4r0i A 1.9 BS02 3KM A 1 D189 S190 C191 Q192 S195 V213 W215 G216 D217 G219 C220 D185 S186 C187 Q188 S191 V210 W212 G213 D214 G215 C216 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 Ki=0.3uM remove_due_to_license_issue Q9Y5Y6 25556099 900 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 4r17 K 2.1 BS01 3K4 K 1 T2 D17 K33 G130 S131 Y170 S171 T1 D16 K32 G129 S130 Y169 S170 D17 R19 K33 G47 S131 D168 S171 D16 R18 K32 G46 S130 D167 S170 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25244435 301 TTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4r18 K 2.4 BS01 ABA K 1 T2 D17 K33 G130 S131 Y170 S171 T1 D16 K32 G129 S130 Y169 S170 D17 R19 K33 G47 S131 D168 S171 D16 R18 K32 G46 S130 D167 S170 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P30656 25244435 301 TTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPFLLGTMAGGAADCQFWETWLGSQCRLHELREKERISVAAASKILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGTRLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRSILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVKEEEGSFNNVIG 4r1v A 1.2 BS01 3E8 A 1 I1084 A1108 L1140 P1158 Y1159 M1160 K1161 G1163 D1164 R1208 M1211 A1221 D1222 Y1230 I30 A54 L86 P102 Y103 M104 K105 G107 D108 R152 M155 A165 D166 Y174 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A187 2.7.10.1 0004672,0004713,0005524,0006468 ic50<1nM remove_due_to_license_issue IC50=<100nM P08581 25736998 1401 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 4r1y A 2.0 BS01 3EH A 1 I1084 A1108 P1158 Y1159 M1160 D1164 R1208 N1209 M1211 A1221 D1222 Y1230 I23 A41 P79 Y80 M81 D85 R129 N130 M132 A142 D143 Y151 D1204 A1206 R1208 N1209 D1222 A1243 D125 A127 R129 N130 D143 A162 2.7.10.1 0004672,0004713,0005524,0006468 ic50=400nM remove_due_to_license_issue IC50=400nM P08581 25736998 1401 LVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLIHCAVKSLNSQFLTEGIIMKDFSHPNVLSLLGICLSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4r22 B 2.6 BS01 dna G 0 S15 I16 G17 R28 R31 R43 R49 S9 I10 G11 R22 R25 R37 R43 ? 0003677,0003700,0006355 remove_due_to_license_issue G2RUZ1 25691471 0 ~ 20 SYRDKKVMSIGIVKELTGLSERQIRYYEKRSLLFPDRTNTGIRKYSFSDVERLMDIADRIEEGVQTSEIRTELAKKDEARKM 4r3b A 1.366 BS02 3GE A 1 S70 N132 E166 T167 N170 G236 A237 S45 N107 E141 T142 N145 G211 A212 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 25536850 302 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 4r3c A 2.06 BS02 3GF A 1 V38 A51 K53 L104 V105 T106 M109 S154 L167 V35 A48 K50 L101 V102 T103 M106 S151 L164 D150 K152 N155 D168 T185 D147 K149 N152 D165 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Ki=100nM, IC50=230nM Q16539 25676389 402 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4r3c A 2.06 BS03 3GF A 2 E22 R23 T44 E19 R20 T41 D150 K152 N155 D168 T185 D147 K149 N152 D165 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue Ki=100nM, IC50=230nM Q16539 25676389 403 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 4r3i A 1.8 BS01 rna B 0 K361 S362 N363 N367 W377 S378 L380 P381 V382 R404 E405 W428 M434 K472 I473 G474 R475 D476 K18 S19 N20 N24 W34 S35 L37 P38 V39 R61 E62 W85 M91 K129 I130 G131 R132 D133 ? 0003723 remove_due_to_license_issue Q96MU7 25242552 1 ~ 5 GTSKLKYVLQDARFFLIKSNNHENVSLAKAKGVWSTLPVNEKKLNLAFRSARSVILIFSVRESGKFQGFARLSSESHHGGSPIHWVLPAGMSAKMLGGVFKIDWICRRELPFTKSAHLTNPWNEHKPVKIGRDGQEIELECGTQLCLLFPPDESIDLYQVIHKM 4r3w A 1.91 BS02 A2P A 1 G9 T11 G12 A13 A36 S37 R39 S40 T57 A72 T76 G161 M162 G8 T10 G11 A12 A35 S36 R38 S39 T56 A71 T75 G160 M161 0004073,0008652,0009086,0009088,0009089,0009097,0016620,0046983,0050661,0051287 Ki=1mM remove_due_to_license_issue 25478842 406 GYTVAVVGATGAVGAQMIKMLEESTLPIDKIRYLASARSAGKSLKFKDQDITIEETTETAFEGVDIALFSAGSSTSAKYAPYAVKAGVVVVDNTSYFRQNPDVPLVVPEVNAHALDAHNGIIACPNCSTIQMMVALEPVRQKWGLDRIIVSTYQAVSGAGMGAILETQRELREVLNDGVKPCDLHAEILPSGGDKKHYPIAFNALPQIDVFTDNDYTYEEMKMTKETKKIMEDDSIAVSATCVRIPVLSAHSESVYIETKEVAPIEEVKAAIAAFPGAVLEDDVAHQIYPQAINAVGSRDTFVGRIRKDLDAEKGIHMWVVSDNLLKGAAWNSVQIAETLHERGLVRPTAELKFELK 4r4c A 1.4 BS01 3HS A 1 R31 I33 T34 R41 R43 S55 M57 A59 T60 N85 V93 I95 R34 I36 T37 R44 R46 S58 M60 A62 T63 N88 V96 I98 ? 0003677,0005634,0006260 remove_due_to_license_issue Kd=2900nM P27694 25699140 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4r4e B 2.57 BS01 dna D 0 G15 R26 R29 R41 N45 R46 R47 G15 R26 R29 R41 N45 R46 R47 ? 0003677,0003700,0006355 remove_due_to_license_issue P37582 25691471 9 ~ 17 MSDNIRRSMPLFPIGIVMQLTELSARQIRYYEENGLIFPARTEGNRRLFSFHDVDKLLEIKHLIEQGVNMAGIKQILAKAEAEP 4r4e B 2.57 BS02 dna E 0 S24 R26 Q27 Y30 R46 S24 R26 Q27 Y30 R46 ? 0003677,0003700,0006355 remove_due_to_license_issue P37582 25691471 2 ~ 9 MSDNIRRSMPLFPIGIVMQLTELSARQIRYYEENGLIFPARTEGNRRLFSFHDVDKLLEIKHLIEQGVNMAGIKQILAKAEAEP 4r4i A 1.4 BS01 3HV A 1 R31 I33 T34 R41 R43 S55 A59 T60 N85 I95 R34 I36 T37 R44 R46 S58 A62 T63 N88 I98 ? 0003677,0005634,0006260 remove_due_to_license_issue Kd=0.540000nM P27694 25699140 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4r4o A 1.33 BS01 3HW A 1 I33 R41 R43 S55 M57 A59 N85 V93 M97 I36 R44 R46 S58 M60 A62 N88 V96 M100 ? 0003677,0005634,0006260 remove_due_to_license_issue Kd=1.5nM P27694 25699140 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4r4q A 1.35 BS01 3HZ A 1 I33 R41 R43 S55 M57 A59 T60 N85 L87 R91 V93 I95 I34 R42 R44 S56 M58 A60 T61 N86 L88 R92 V94 I96 ? 0003677,0005634,0006260 remove_due_to_license_issue P27694 25699140 201 HMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4r4t A 1.28 BS01 3J0 A 1 I33 T34 R41 R43 S55 M57 A59 T60 V93 I95 I35 T36 R43 R45 S57 M59 A61 T62 V95 I97 ? 0003677,0005634,0006260 remove_due_to_license_issue Kd=0.550000nM P27694 25699140 201 SHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 4r55 A 1.8 BS01 dna B 0 K24 W26 L28 Y44 R46 K22 W24 L26 Y42 R44 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 101 ~ 108 SGKKPVKVKTPAGKEAELVPEKVWALGRVKIGLFKDPETGKYFRHKLPDDYPI 4r55 A 1.8 BS02 dna C 0 V31 R46 H47 K48 V29 R44 H45 K46 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 109 ~ 116 SGKKPVKVKTPAGKEAELVPEKVWALGRVKIGLFKDPETGKYFRHKLPDDYPI 4r56 A 2.3 BS01 dna C 0 K24 W26 L28 A29 P30 K31 L40 Y49 R51 K23 W25 L27 A28 P29 K30 L39 Y48 R50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 101 ~ 108 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 4r56 A 2.3 BS02 dna D 0 V36 R51 H52 K53 V35 R50 H51 K52 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 109 ~ 116 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 4r56 A 2.3 BS03 dna F 0 K37 P59 I60 K36 P58 I59 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 109 ~ 116 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 4r56 B 2.3 BS01 dna E 0 K24 W26 L28 A29 P30 K31 L40 Y49 R51 K23 W25 L27 A28 P29 K30 L39 Y48 R50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 101 ~ 108 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 4r56 B 2.3 BS02 dna F 0 V36 R51 H52 K53 V35 R50 H51 K52 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 25555709 109 ~ 116 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 4r59 A 1.65 BS02 3J3 A 1 L91 H94 V121 L197 T198 W208 L89 H92 V119 L195 T196 W206 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=11nM remove_due_to_license_issue P00918 25254302 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4r5a A 1.64 BS02 3J4 A 1 W5 N62 H64 Q92 H94 H119 L198 T199 T200 P201 W5 N62 H64 Q92 H94 H119 L197 T198 T199 P200 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2nM remove_due_to_license_issue P00918 25254302 303 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4r5b A 1.5 BS02 3J4 A 1 N62 Q92 H94 F131 L198 T199 T200 N62 Q92 H94 F130 L197 T198 T199 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=185nM remove_due_to_license_issue P00918 25254302 303 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4r5g B 3.4501 BS01 3JE B 1 L392 T395 P396 L399 A503 S504 L15 T18 P19 L22 A126 S127 ? 0005524,0140662 remove_due_to_license_issue P0A6Y8 25148104 701 MHHHHHHIEGRVLLLDVTPLSLGIETMGGVMTTLIAKNTTIPTKHSQVFSTAEDNQSAVTIHVLQGERKRAADNKSLGQFNLDGINPAPRGMPQIEVTFDIDADGILHVSAKDKNSGKEQKITIKASSGLNEDEIQKMVRDAEANAEADRKFEELVQTRNQGDHLLHSTRKQVEEDDKTAIESALTALETALKGKAAIEAKMQELAQVS 4r5n A 1.8 BS01 3J9 A 1 G72 Q73 G74 L91 D93 Y132 F169 I171 W176 D289 G291 G13 Q14 G15 L32 D34 Y73 F110 I112 W117 D223 G225 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=76nM remove_due_to_license_issue IC50=60nM P56817 25411915 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4r5t A 1.98 BS02 R5T A 1 E319 V459 G460 A461 H496 E497 H500 E519 Y575 Y580 E124 V264 G265 A266 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=0.8uM remove_due_to_license_issue Ki=0.800000nM O96935 25299353 1112 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4r5v A 2.1 BS02 R5V A 1 V459 G460 A461 M462 E463 R489 H496 E497 H500 E519 Y575 Y580 V264 G265 A266 M267 E268 R294 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=0.7uM remove_due_to_license_issue Ki=0.700000nM O96935 25299353 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4r5w A 2.84 BS01 XAV A 1 D766 N767 H862 G863 Y896 F897 K903 S904 Y907 D106 N107 H200 G201 Y234 F235 K241 S242 Y245 S904 Y907 E988 S242 Y245 E326 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=120nM, Kd=620nM P09874 28001384 1106 MKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKTAH 4r5x A 1.85 BS02 R5X A 1 E319 V459 G460 A461 M462 R489 H496 E497 H500 E519 Y575 Y580 M1034 E123 V263 G264 A265 M266 R293 H300 E301 H304 E323 Y379 Y384 M838 E463 H496 E497 H500 E519 E572 Y580 E267 H300 E301 H304 E323 E376 Y384 3.4.11.- 0006508,0008237,0008270 Ki=5.5uM remove_due_to_license_issue Ki=5.5nM O96935 25299353 1107 KIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4r5y A 3.5 BS01 3K3 A 1 V471 A481 K483 E501 L505 I527 T529 W531 C532 F583 D594 V23 A33 K35 E53 L57 I79 T81 W83 C84 F135 D146 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S149 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=23nM P15056 26208524 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 4r6e A 2.2 BS01 3JD A 1 D766 H862 G863 Y889 Y896 F897 K903 S904 Y907 D106 H202 G203 Y229 Y236 F237 K243 S244 Y247 S904 Y907 E988 S244 Y247 E328 2.4.2.-,2.4.2.30 0003950 ic50=132nM remove_due_to_license_issue IC50=132nM, Ki=3.2nM, EC50=31000nM P09874 28001384 1101 MKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 4r6t A 2.6 BS04 R5T A 1 K386 M392 D459 E461 L487 G489 A577 K297 M303 D370 E372 L398 G400 A488 K386 R463 K297 R374 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue Ki=0.030000nM Q8IL11 25299353 1007 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4r6v A 2.353 BS01 FI3 A 1 L473 G474 E475 C477 F478 K503 E520 I534 L550 C552 A553 G556 E560 L619 A629 D630 F631 L31 G32 E33 C35 F36 K56 E73 I87 L103 C105 A106 G109 E113 L159 A169 D170 F171 D612 A614 R616 N617 D630 D152 A154 R156 N157 D170 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 25349422 801 DPLLAGLVSLDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVILECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLAPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 4r6w A 1.5894 BS02 SAH A 1 Y19 I36 S37 G63 D85 I86 I111 R127 H132 Y11 I28 S29 G55 D77 I78 I103 R119 H124 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 Kd=5.4uM remove_due_to_license_issue Q8IDQ9 25288796 302 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRAAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4r6x A 2.5534 BS02 SAH A 1 Y19 Y35 I36 S37 G63 S64 D85 I86 D110 I111 R127 A128 A129 H132 Y11 Y27 I28 S29 G55 S56 D77 I78 D102 I103 R119 A120 A121 H124 2.1.1.103 0000139,0000234,0005737,0005794,0006656,0008168,0008654,0009058,0016020,0032259 remove_due_to_license_issue Q8IDQ9 25288796 502 SDKTFLENNQYTDEGVKVYEFIFGENYISSGGLEATKKILSDIELNENSKVLDIGSGLGGGCMYINEKYGAHTHGIDICSNIVNMANERVSGNNKIIFEANDILTKEFPENNFDLIYSRAAILHLSLENKNKLFQKCYKWLKPTGTLLITDYCATEKENWDDEFKEYVKQRKYTLITVEEYADILTACNFKNVVSKDLSDYWNQLLEVEHKYLHENKEEFLKLFSEKKFISLDDGWSRKIKDSKRKMQRWGYFKATKN 4r73 A 1.6 BS01 G6P A 1 R34 S37 G59 Y103 S148 G149 T150 G185 I186 H205 D206 E229 Q269 R36 S39 G61 Y105 S150 G151 T152 G187 I188 H207 D208 E231 Q271 ? 0015888,0030288,0030975,0030976 Kd=23nM remove_due_to_license_issue A3N294 26295949 401 GSKGRLVIYCSATNVMCENAAKTFEQKYDVKTSFIRNGSGSTFAKIEAEKNNPQADVWYGGTLDPQSQAGELGLLEAYRSPNIDQIMPKFQDPAKVKGNLSSAVYIGILGFAVNTERLKKLGIEKIPQCWNDLTDPKLKGEIQIADPQSSGTAYTAIATFAQLWGEDKAFDYFKHLHPNISQYTKSGITPARNAARGETTVGIGFLHDYALEKEQGAPLEMVVPCEGTGYELGGVSILKGARNLDNAKLFVDFALSKEGQETAWKKGQALQTLTNTTAEQSPLAFDLTKLKLIDYDFEKYGASDERKRLINKWVDEIKLAK 4r74 A 1.93 BS01 F6P A 1 T11 S37 G59 Y103 S148 G149 T150 G185 I186 H205 D206 E229 T12 S38 G60 Y104 S149 G150 T151 G186 I187 H206 D207 E230 ? 0015888,0030288,0030975,0030976 Kd=8nM remove_due_to_license_issue A3N294 26295949 401 SKGRLVIYCSATNVMCENAAKTFEQKYDVKTSFIRNGSGSTFAKIEAEKNNPQADVWYGGTLDPQSQAGELGLLEAYRSPNIDQIMPKFQDPAKVKGNLSSAVYIGILGFAVNTERLKKLGIEKIPQCWNDLTDPKLKGEIQIADPQSSGTAYTAIATFAQLWGEDKAFDYFKHLHPNISQYTKSGITPARNAARGETTVGIGFLHDYALEKEQGAPLEMVVPCEGTGYELGGVSILKGARNLDNAKLFVDFALSKEGQETAWKKGQALQTLTNTTAEQSPLAFDLTKLKLIDYDFEKYGASDERKRLINKWVDEIKLA 4r75 A 1.278 BS01 S7P A 1 T11 G36 S37 G59 T60 Y103 S148 G149 T150 G185 H205 D206 E229 T11 G36 S37 G59 T60 Y103 S148 G149 T150 G185 H205 D206 E229 ? 0015888,0030288,0030975,0030976 Kd=57nM remove_due_to_license_issue A3N294 26295949 401 KGRLVIYCSATNVMCENAAKTFEQKYDVKTSFIRNGSGSTFAKIEAEKNNPQADVWYGGTLDPQSQAGELGLLEAYRSPNIDQIMPKFQDPAKVKGNLSSAVYIGILGFAVNTERLKKLGIEKIPQCWNDLTDPKLKGEIQIADPQSSGTAYTAIATFAQLWGEDKAFDYFKHLHPNISQYTKSGITPARNAARGETTVGIGFLHDYALEKEQGAPLEMVVPCEGTGYELGGVSILKGARNLDNAKLFVDFALSKEGQETAWKKGQALQTLTNTTAEQSPLAFDLTKLKLIDYDFEKYGASDERKRLINKWVDEIKLA 4r76 A 2.5 BS04 R5X A 1 K374 D379 D459 E461 L487 T488 G489 L492 A577 K286 D291 D371 E373 L399 T400 G401 L404 A489 K386 R463 K298 R375 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.014uM remove_due_to_license_issue Ki=0.014000nM Q8IL11 25299353 1004 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4r76 F 2.5 BS04 R5X F 1 D379 M392 F398 N457 D459 E461 L487 T488 G489 L492 D285 M298 F304 N363 D365 E367 L393 T394 G395 L398 K386 R463 K292 R369 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.014uM remove_due_to_license_issue Ki=0.014000nM Q8IL11 25299353 1004 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4r7m A 2.85 BS04 3MW A 1 K374 D379 M392 M396 N457 D459 E461 L487 T488 G489 K287 D292 M305 M309 N370 D372 E374 L400 T401 G402 K386 R463 K299 R376 3.4.11.1,3.4.13.- 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue Ki=0.011000nM Q8IL11 25299353 1006 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4r8y A 1.9 BS01 3KO A 1 D93 Y132 I171 D289 G291 D36 Y75 I114 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=0.64uM remove_due_to_license_issue Ki=640nM P56817 25455483 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4r91 A 1.58 BS01 3KT A 1 D93 Y132 F169 D289 G291 D36 Y75 F112 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=430nM remove_due_to_license_issue Ki=430nM P56817 25455483 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4r92 A 1.71 BS01 3KU A 1 D93 Y132 K168 F169 F170 R189 D289 G291 D37 Y76 K112 F113 F114 R133 D233 G235 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 Ki=39nM remove_due_to_license_issue Ki=39nM P56817 25455483 501 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4r93 A 1.71 BS01 779 A 1 D93 Y132 K168 F169 I171 D289 G291 D36 Y75 K111 F112 I114 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=16nM remove_due_to_license_issue Ki=16nM P56817 25455483 503 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4r95 A 1.99 BS01 3KW A 1 D93 Y132 K168 F169 R189 D289 G291 D36 Y75 K111 F112 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=22nM remove_due_to_license_issue P56817 25455483 503 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4ra1 A 1.75 BS01 ALX A 1 S53 N54 Y145 W178 Y375 Y376 W418 S419 N420 T430 E434 E510 S22 N23 Y114 W147 Y344 Y345 W387 S388 N389 T399 E403 E479 ? 0015833,0030288,0042597,0043190,0055085,1904680 Kd=0.43uM remove_due_to_license_issue Q52012 26244338 601 RRALRLGVNGLPNSLEPVNAISNVGPRIVNQIFDTLIARDFFAKGAPGNAIDLVPALAESWERIDEKSVRFKLRQKVMFHDGVELTADDVAYTFSSERLWGPEAIKKIPLGKSYSLDFDEPVVEDKYTVTLRTKTPSYLIETFVASWMSRIVPKEYYKKLGAVDFGNKPVGTGPYKFVEFVAGDRVVLEANDAYWGPKPTASKITYQIVAEPATRVAGLISGEYDIITTLTPDDIQLINSYPDLETRGTLIENFHMFTFNMNQEVFKDKKLRRALALAVNRPIMVEALWKKQASIPAGFNFPNYGETFDPKRKAMEYNVEEAKRLVKESGYDGTPITYHTMGNYYANAMPALMMMIEMWKQIGVNVVMKTYAPGSFPPDNQTWMRNWSNGQWMTDAYATIVPEFGPNGQVQKRWGWKAPAEFNELCQKVTVLPNGKERFDAYNRMRDIFEEEAPAVILYQPYDVYAARKDVHWKPVSFEMMEFRNNLSFG 4ra5 A 2.61 BS01 3L0 A 1 L386 G387 K388 V394 A407 M458 E459 D508 L511 D522 F664 F668 L13 G14 K15 V21 A34 M85 E86 D135 L138 D149 F291 F295 D504 K506 D508 N509 D522 T542 D131 K133 D135 N136 D149 T169 2.7.11.13 0004672,0004674,0004697,0005524,0006468 remove_due_to_license_issue IC50=4.0nM Q04759 25254961 801 KLKIEDFELHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNEFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPPFRPKVKSPFDCSNFDKEFLNEKPRLSFADRALINSMDQNMFRNFSFMNPGMERLISH 4rab A 2.264 BS01 3L3 A 1 D137 T138 G139 T141 K165 F186 V187 D193 D118 T119 G120 T122 K146 F167 V168 D174 E133 D134 D137 F186 R199 E114 D115 D118 F167 R180 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.04uM remove_due_to_license_issue P00492 25494538 301 PGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYK 4rab C 2.264 BS01 3L3 C 1 D137 T138 G139 K140 T141 K165 F186 V187 D193 D123 T124 G125 K126 T127 K151 F172 V173 D179 E133 D134 D137 F186 R199 E119 D120 D123 F172 R185 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.04uM remove_due_to_license_issue P00492 25494538 301 PGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4rac A 2.05 BS01 3L4 A 1 K68 G69 D137 T138 G139 T141 K165 F186 V187 D193 R199 K65 G66 D124 T125 G126 T128 K152 F173 V174 D180 R186 E133 D134 D137 F186 R199 E120 D121 D124 F173 R186 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.03uM remove_due_to_license_issue P00492 25494538 301 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4rac C 2.05 BS01 3L4 C 1 K68 G69 I135 D137 T138 G139 T141 K165 F186 V187 D193 R199 K63 G64 I121 D123 T124 G125 T127 K151 F172 V173 D179 R185 E133 D134 D137 F186 R199 E119 D120 D123 F172 R185 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.03uM remove_due_to_license_issue P00492 25494538 301 GVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKDIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4rad A 2.0 BS01 3L5 A 1 I135 D137 T138 G139 T141 K165 F186 V187 I118 D120 T121 G122 T124 K148 F166 V167 E133 D134 D137 F186 R199 E116 D117 D120 F166 R179 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 25494538 301 PGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4rad C 2.0 BS01 3L5 C 1 K68 I135 D137 T138 G139 T141 K165 F186 V187 D193 K65 I122 D124 T125 G126 T128 K152 F173 V174 D180 E133 D134 D137 F186 R199 E120 D121 D124 F173 R186 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 25494538 301 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKY 4rak A 2.04 BS01 652 A 1 F271 T272 L274 A275 S278 M312 T316 R319 F329 L330 L345 I353 F54 T55 L57 A58 S61 M95 T99 R102 F112 L113 L128 I136 ? 0003677,0004879,0006629 Ki=14nM remove_due_to_license_issue EC50=250nM, Ki=14nM P55055 25435151 503 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRKLPPLLSEIW 4ran A 2.549 BS01 3L6 A 1 D137 T138 G139 T141 K165 F186 V187 D193 D121 T122 G123 T125 K149 F170 V171 D177 E133 D134 D137 F186 R199 E117 D118 D121 F170 R183 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 25494538 301 RSPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKVIGGDSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4rao A 1.871 BS01 3L7 A 1 K68 G69 D137 T138 G139 K140 T141 K165 F186 V187 R199 K68 G69 D118 T119 G120 K121 T122 K146 F167 V168 R180 E133 D134 D137 F186 R199 E114 D115 D118 F167 R180 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=1uM remove_due_to_license_issue P00492 25494538 301 ATRSPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSRSIPMTVDFIRLKLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYK 4rao C 1.871 BS01 3L7 C 1 K68 G69 I135 D137 T138 G139 T141 K165 F186 V187 D193 R199 K65 G66 I121 D123 T124 G125 T127 K151 F172 V173 D179 R185 E133 D134 D137 F186 R199 E119 D120 D123 F172 R185 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=1uM remove_due_to_license_issue P00492 25494538 301 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4raq A 2.53 BS01 3L8 A 1 K68 G69 R100 I136 D137 T138 G139 T141 K165 F186 V187 D193 R199 K65 G66 R97 I117 D118 T119 G120 T122 K146 F167 V168 D174 R180 E133 D134 D137 F186 R199 E114 D115 D118 F167 R180 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 25494538 301 SPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4raq C 2.53 BS01 3L8 C 1 K68 D137 T138 G139 T141 K165 F186 V187 D193 R199 K64 D119 T120 G121 T123 K147 F167 V168 D174 R180 E133 D134 D137 F186 R199 E115 D116 D119 F167 R180 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue P00492 25494538 301 PGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYKA 4rbo A 3.3 BS01 dna B 0 Y119 Y136 K140 Q144 R147 M148 K151 Y20 Y37 K41 Q45 R48 M49 K52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q9H9S0 25825768 1 ~ 12 TVFSSTQLCVLNDRFQRQKYLSLQQMQELSNILNLSYKQVKTWFQNQRMKSKRWQ 4rbo A 3.3 BS02 dna C 0 T100 F102 K137 Q138 W142 N145 T1 F3 K38 Q39 W43 N46 ? 0000981,0003677,0006355 remove_due_to_license_issue Q9H9S0 25825768 1 ~ 12 TVFSSTQLCVLNDRFQRQKYLSLQQMQELSNILNLSYKQVKTWFQNQRMKSKRWQ 4rbo D 3.3 BS01 dna E 0 Y119 Y136 Q144 R147 M148 K151 Y20 Y37 Q45 R48 M49 K52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q9H9S0 25825768 1 ~ 12 TVFSSTQLCVLNDRFQRQKYLSLQQMQELSNILNLSYKQVKTWFQNQRMKSKRW 4rbo D 3.3 BS02 dna F 0 F102 K137 W142 N145 F3 K38 W43 N46 ? 0000981,0003677,0006355 remove_due_to_license_issue Q9H9S0 25825768 1 ~ 12 TVFSSTQLCVLNDRFQRQKYLSLQQMQELSNILNLSYKQVKTWFQNQRMKSKRW 4rcd A 1.9 BS01 3LL A 1 G11 G13 L30 D32 Y71 W76 F108 I118 R128 D228 G230 G13 G15 L32 D34 Y73 W78 F110 I120 R130 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.7nM remove_due_to_license_issue IC50=0.700000nM P56817 25363711 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4rce A 2.4 BS01 3LN A 1 G11 Q12 G13 L30 D32 Y71 F108 I118 D228 G230 G13 Q14 G15 L32 D34 Y73 F110 I120 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=2nM remove_due_to_license_issue IC50=25nM P56817 25389560 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4rcf A 1.78 BS01 3LO A 1 G11 Q12 G13 L30 D32 Y71 W76 F108 R128 D228 G230 G13 Q14 G15 L32 D34 Y73 W78 F110 R130 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=4nM remove_due_to_license_issue IC50=4.1nM P56817 25389560 404 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 4rcg A 2.6 BS01 GDP A 1 S271 A272 G274 K275 T276 N277 W501 F502 G514 F515 S264 A265 G267 K268 T269 N270 W487 F488 G500 F501 R81 Y220 K229 H249 S271 C273 D296 R389 R74 Y213 K222 H242 S264 C266 D289 R382 4.1.1.32 0004611,0004613,0005525,0005576,0005737,0005829,0005886,0006094,0006107,0009274,0010106,0016831,0017076,0019543,0030145,0033993,0042594,0046327,0046872,0052572,0071333 remove_due_to_license_issue P9WIH3 25798914 701 GLDTAPTNHQGLLSWVEEVAELTQPDRVVFTDGSEEEFQRLCDQLVEAGTFIRLNPEKHKNSYLALSDPSDVARVESRTYICSAKEIDAGPTNNWMDPGEMRSIMKDLYRGCMRGRTMYVVPFCMGPLGAEDPKLGVEITDSEYVVVSMRTMTRMGKAALEKMGDDGFFVKALHSVGAPLEPGQKDVAWPCSETKYITHFPETREIWSYGSGYGGNALLGKKCYSLRIASAMAHDEGWLAEHMLILKLISPENKAYYFAAAFPSACGKTNLAMLQPTIPGWRAETLGDDIAWMRFGKDGRLYAVNPEFGFFGVAPGTNWKSNPNAMRTIAAGNTVFTNVALTDDGDVWWEGLEGDPQHLIDWKGNDWYFRETETNAAHPNSRYCTPMSQCPILAPEWDDPQGVPISGILFGGRRKTTVPLVTEARDWQHGVFIGATLGSEQTANVRRDPMAMLPFLGYNVGDYFQHWINLGKHADEAKLPKVFFVNWFRRGDDGRFLWPGFGENSRVLKWIVDRIEHKAGGATTPIGTVPAVEDLDLDGLDVDAADVAAALAVDADEWRQELPLIEEWLQFVGEKLPTGVKDEFDALKERLG 4rcj A 1.6 BS01 rna B 0 K395 S396 Y397 D401 W411 C412 N441 G442 W465 K469 W470 N504 S505 R506 D507 K31 S32 Y33 D37 W47 C48 N77 G78 W101 K105 W106 N140 S141 R142 D143 ? 0003723 remove_due_to_license_issue Q9BYJ9 26318451 1 ~ 5 HPVLEKLKAAHSYNPKEFEWNLKSGRVFIIKSYSEDDIHRSIKYSIWCSTEHGNKRLDSAFRCMSSKGPVYLLFSVNGSGHFCGVAEMKSPVDYGTSAGVWSQDKWKGKFDVQWIFVKDVPNNQLRHIRLENNDNKPVTNSRDTQEVPLEKAKQVLKIISSYKHTTSIFDDFAHYEKRQEEEEVVRKE 4rcm A 1.8 BS01 rna D 0 K161 S163 H167 W177 S178 W231 Y237 D274 K22 S24 H28 W38 S39 W92 Y98 D135 ? 0003723 remove_due_to_license_issue Q06390 26318451 3 GSAAIIPPWLNIPENSRFFVIKSSSLKHVKRSFYNGIWSSTHFGNKRLSEAYKKLNSGAKVFLFFSINTSGRFCGVAEMVSDLKMDLDTSIWEDEQKYGKAFKVRWVIVRDINNRSLKRFLIPSNEMKPITHSRDTQEIPYSIGISIINLFKTQDSDIFSFLDE 4rcm B 1.8 BS01 rna E 0 K161 S163 H167 W177 S178 T180 W231 Y237 D274 K20 S22 H26 W36 S37 T39 W90 Y96 D133 ? 0003723 remove_due_to_license_issue Q06390 26318451 3 AAIIPPWLNIPENSRFFVIKSSSLKHVKRSFYNGIWSSTHFGNKRLSEAYKKLNSGAKVFLFFSINTSGRFCGVAEMVSDLKMDLDTSIWEDEQKYGKAFKVRWVIVRDINNRSLKRFLIPSNEMKPITHSRDTQEIPYSIGISIINLFKTQDIFSFLD 4rd0 A 1.713 BS01 GDP A 1 A19 G21 K22 T23 T24 N149 K150 D152 S184 L186 A18 G20 K21 T22 T23 N148 K149 D151 S183 L185 A19 K22 T23 T46 H97 A18 K21 T22 T45 H96 3.6.5.3 0000049,0001731,0003743,0003746,0003924,0005515,0005525,0006412,0006413,0006414,0016787,0046872,1990606 Kd=0.24uM remove_due_to_license_issue Q980A5 25690901 501 AWPKVQPEVNIGVVGHVAHGKTTLVQAITGIWTSKHSEELKRGMTIKLGYAETNIGVCESCKKPEAYVTEPSCKSCGSDDEPKFLRRISFIDAPGHEVLMATMLSGAALMDGAILVVAANEPFPQPQTREHFVALGIIGVKNLIIVQNKVDVVSKEEALSQYRQIKQFTKGTWAENVPIIPVSALHKINIDSLIEGIEEYIKTPYRDLSQKPVMLVIRSFDVNKPGTQFNELKGGVIGGSIIQGLFKVDQEIKVLPGLRVEKQGKVSYEPIFTKISSIRFGDEEFKEAKPGGLVAIGTYLDPSLTKADNLLGSIITLADAEVPVLWNIRIKYNLLERVVGAKEMLKVDPIRAKETLMLSVGSSTTLGIVTSVKKDEIEVELRRPVAVWSNNIRTVISRQIAGRWRMIGWGLVEI 4rd0 A 1.713 BS03 GDP A 2 F221 V223 K225 K234 S278 R280 A296 F220 V222 K224 K233 S277 R279 A295 A19 K22 T23 T46 H97 A18 K21 T22 T45 H96 3.6.5.3 0000049,0001731,0003743,0003746,0003924,0005515,0005525,0006412,0006413,0006414,0016787,0046872,1990606 Kd=0.24uM remove_due_to_license_issue Q980A5 25690901 503 AWPKVQPEVNIGVVGHVAHGKTTLVQAITGIWTSKHSEELKRGMTIKLGYAETNIGVCESCKKPEAYVTEPSCKSCGSDDEPKFLRRISFIDAPGHEVLMATMLSGAALMDGAILVVAANEPFPQPQTREHFVALGIIGVKNLIIVQNKVDVVSKEEALSQYRQIKQFTKGTWAENVPIIPVSALHKINIDSLIEGIEEYIKTPYRDLSQKPVMLVIRSFDVNKPGTQFNELKGGVIGGSIIQGLFKVDQEIKVLPGLRVEKQGKVSYEPIFTKISSIRFGDEEFKEAKPGGLVAIGTYLDPSLTKADNLLGSIITLADAEVPVLWNIRIKYNLLERVVGAKEMLKVDPIRAKETLMLSVGSSTTLGIVTSVKKDEIEVELRRPVAVWSNNIRTVISRQIAGRWRMIGWGLVEI 4rd3 A 1.69 BS01 GDP A 1 D19 G21 K22 T23 T24 N149 K150 D152 S184 L186 D18 G20 K21 T22 T23 N148 K149 D151 S183 L185 D19 K22 T23 T46 A97 D18 K21 T22 T45 A96 3.6.5.3 0000049,0001731,0003743,0003746,0003924,0005515,0005525,0006412,0006413,0006414,0016787,0046872,1990606 remove_due_to_license_issue Q980A5 25690901 502 AWPKVQPEVNIGVVGHVDHGKTTLVQAITGIWTSKHSEELKRGMTIKLGYAETNIGVCESCKKPEAYVTEPSCKSCGSDDEPKFLRRISFIDAPGAEVLMATMLSGAALMDGAILVVAANEPFPQPQTREHFVALGIIGVKNLIIVQNKVDVVSKEEALSQYRQIKQFTKGTWAENVPIIPVSALHKINIDSLIEGIEEYIKTPYRDLSQKPVMLVIRSFDVNKPGTQFNELKGGVIGGSIIQGLFKVDQEIKVLPGLRVEKQGKVSYEPIFTKISSIRFGDEEFKEAKPGGLVAIGTYLDPSLTKADNLLGSIITLADAEVPVLWNIRIKYNLLERVVGAKEMLKVDPIRAKETLMLSVGSSTTLGIVTSVKKDEIEVELRRPVAVWSNNIRTVISRQIAGRWRMIGWGLVEI 4rd3 A 1.69 BS03 GDP A 2 F221 V223 K234 S278 R280 A296 G298 F220 V222 K233 S277 R279 A295 G297 D19 K22 T23 T46 A97 D18 K21 T22 T45 A96 3.6.5.3 0000049,0001731,0003743,0003746,0003924,0005515,0005525,0006412,0006413,0006414,0016787,0046872,1990606 remove_due_to_license_issue Q980A5 25690901 504 AWPKVQPEVNIGVVGHVDHGKTTLVQAITGIWTSKHSEELKRGMTIKLGYAETNIGVCESCKKPEAYVTEPSCKSCGSDDEPKFLRRISFIDAPGAEVLMATMLSGAALMDGAILVVAANEPFPQPQTREHFVALGIIGVKNLIIVQNKVDVVSKEEALSQYRQIKQFTKGTWAENVPIIPVSALHKINIDSLIEGIEEYIKTPYRDLSQKPVMLVIRSFDVNKPGTQFNELKGGVIGGSIIQGLFKVDQEIKVLPGLRVEKQGKVSYEPIFTKISSIRFGDEEFKEAKPGGLVAIGTYLDPSLTKADNLLGSIITLADAEVPVLWNIRIKYNLLERVVGAKEMLKVDPIRAKETLMLSVGSSTTLGIVTSVKKDEIEVELRRPVAVWSNNIRTVISRQIAGRWRMIGWGLVEI 4rd6 A 1.944 BS01 GDP A 1 D19 G21 K22 T23 T24 N149 K150 D152 S184 L186 D18 G20 K21 T22 T23 N139 K140 D142 S174 L176 D19 K22 T23 H97 D18 K21 T22 H87 3.6.5.3 0000049,0001731,0003743,0003746,0003924,0005515,0005525,0006412,0006413,0006414,0016787,0046872,1990606 Kd=0.52uM remove_due_to_license_issue Q980A5 25690901 501 AWPKVQPEVNIGVVGHVDHGKTTLVQAITGIWTSKHSKLGYAETNIGVCESCKKPEAYVTEPSCKSCGSDDEPKFLRRISFIDAPGHEVLMATMLSGAALMDGAILVVAANEPFPQPQTREHFVALGIIGVKNLIIVQNKVDVVSKEEALSQYRQIKQFTKGTWAENVPIIPVSALHKINIDSLIEGIEEYIKTPYRDLSQKPVMLVIRSFDVNKPGTQFNELKGGVIGGSIIQGLFKVDQEIKVLPGLRVEKQGKVSYEPIFTKISSIRFGDEEFKEAKPGGLVAIGTYLDPSLTKADNLLGSIITLADAEVPVLWNIRIKYNLLERVVGAKEMLKVDPIRAKETLMLSVGSSTTLGIVTSVKKDEIEVELRRPVAVWSNNIRTVISRQIAGRWRMIGWGLVEI 4rdn A 2.1 BS01 6MD A 1 K416 S417 Y418 D422 W432 C433 W486 W491 D528 K17 S18 Y19 D23 W33 C34 W87 W92 D129 ? 0003723 remove_due_to_license_issue Q9Y5A9 25412658 601 ENLYFQHMKHGRVFIIKSYSEDDIHRSIKYNIWCSTEHGNKRLDAAYRSMNGKGPVYLLFSVNGSGHFCGVAEMKSAVDYNTCAGVWSQDKWKGRFDVRWIFVKDVPNSQLRHIRLENNENKPVTNSRDTQEVPLEKAKQVLKIIASYK 4re2 A 2.0 BS01 MVL A 1 Q32 H133 N178 E179 Y318 W361 E389 W436 E443 W444 F452 Q36 H137 N182 E183 Y322 W365 E393 W440 E447 W448 F456 R89 H133 E179 C182 N316 Y318 E389 R93 H137 E183 C186 N320 Y322 E393 3.2.1.25 0004553,0004565,0005975,0008422,0033907 remove_due_to_license_issue A2YPH1 501 APFTYWLNPEIYDAGGLSRRAFPEGFVFGTAASAYQVEGMAKQGGRGPSIWDAFIEKPGTIPNNATADVTVDEYHRYKEDVNIMKNMGFDAYRFSISWSRIFPNGTGMVNQEGVDYYNRLIDYMVKKGIKPYANLYHYDLPLALHEQYLGWLSPNIVEAFADYADFCFQTFGDRVKDWFTFNEPRCVAALGYDNGFHAPGRCSGCDAGGNSTTEPYLAAHHLILSHAAAVKRYREKYQLYQKGRIGILLDFVWYEPFSDSNADRAAAQRARDFHLGWFLDPIIHGRYPYSMLEIVKDRMPTFSDEESRMVKDSIDYVGINHYTSFYMKDPGPWNLTPTSYQDDWHVGFAYERNGVPIGAQANSYWLYIVPWGINKAVTYVKETYGNPTMILSENGMDQPGNVSITQGVHDTVRIRYYRNYITELKKAIDDGAKVIGYFAWSLLDNFEWRLGYTSRFGIVYVDYKTLKRYPKDSAFWFKNMLS 4re3 A 2.55 BS01 GIM A 1 Q32 H133 E179 Y318 W361 E389 W436 E443 F452 Q37 H138 E184 Y323 W366 E394 W441 E448 F457 R89 H133 E179 C182 N316 Y318 E389 R94 H138 E184 C187 N321 Y323 E394 3.2.1.25 0004553,0004565,0005975,0008422,0033907 remove_due_to_license_issue A2YPH1 507 AAPFTYWLNPEIYDAGGLSRRAFPEGFVFGTAASAYQVEGMAKQGGRGPSIWDAFIEKPGTIPNNATADVTVDEYHRYKEDVNIMKNMGFDAYRFSISWSRIFPNGTGMVNQEGVDYYNRLIDYMVKKGIKPYANLYHYDLPLALHEQYLGWLSPNIVEAFADYADFCFQTFGDRVKDWFTFNEPRCVAALGYDNGFHAPGRCSGCDAGGNSTTEPYLAAHHLILSHAAAVKRYREKYQLYQKGRIGILLDFVWYEPFSDSNADRAAAQRARDFHLGWFLDPIIHGRYPYSMLEIVKDRMPTFSDEESRMVKDSIDYVGINHYTSFYMKDPGPWNLTPTSYQDDWHVGFAYERNGVPIGAQANSYWLYIVPWGINKAVTYVKETYGNPTMILSENGMDQPGNVSITQGVHDTVRIRYYRNYITELKKAIDDGAKVIGYFAWSLLDNFEWRLGYTSRFGIVYVDYKTLKRYPKDSAFWFKNMLS 4re4 A 2.29 BS01 IFM A 1 Q32 H133 E179 Y318 E389 W436 E443 W444 F452 Q37 H138 E184 Y323 E394 W441 E448 W449 F457 R89 H133 E179 C182 N316 Y318 E389 R94 H138 E184 C187 N321 Y323 E394 3.2.1.25 0004553,0004565,0005975,0008422,0033907 remove_due_to_license_issue A2YPH1 501 AAPFTYWLNPEIYDAGGLSRRAFPEGFVFGTAASAYQVEGMAKQGGRGPSIWDAFIEKPGTIPNNATADVTVDEYHRYKEDVNIMKNMGFDAYRFSISWSRIFPNGTGMVNQEGVDYYNRLIDYMVKKGIKPYANLYHYDLPLALHEQYLGWLSPNIVEAFADYADFCFQTFGDRVKDWFTFNEPRCVAALGYDNGFHAPGRCSGCDAGGNSTTEPYLAAHHLILSHAAAVKRYREKYQLYQKGRIGILLDFVWYEPFSDSNADRAAAQRARDFHLGWFLDPIIHGRYPYSMLEIVKDRMPTFSDEESRMVKDSIDYVGINHYTSFYMKDPGPWNLTPTSYQDDWHVGFAYERNGVPIGAQANSYWLYIVPWGINKAVTYVKETYGNPTMILSENGMDQPGNVSITQGVHDTVRIRYYRNYITELKKAIDDGAKVIGYFAWSLLDNFEWRLGYTSRFGIVYVDYKTLKRYPKDSAFWFKNMLS 4re9 A 2.908 BS02 3M9 A 1 H108 H112 F115 S128 N139 F820 R824 Y831 H66 H70 F73 S86 N97 F778 R782 Y789 E111 E69 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 26394692 1102 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLEHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 4res A 3.408 BS04 BUF A 1 E117 D121 L125 G319 V322 A323 F783 T797 I800 E97 D101 L105 G299 V302 A303 F763 T777 I780 D369 D710 D714 D349 D690 D694 7.2.2.13 0000166,0002028,0005215,0005391,0005515,0005524,0005886,0005890,0006813,0006814,0006883,0008556,0010248,0016020,0016323,0016887,0030007,0030424,0030955,0031402,0036376,0042383,0042470,0042995,0046872,0051117,0055085,0086009,1902600,1990573 remove_due_to_license_issue P05024 25624492 2001 KERDMDELKKEVSMDDHKLSLDELHRKYGTDLSRGLTPARAAEILARDGPNALTPPPTTPEWVKFCRQLFGGFSMLLWIGAILCFLAYGIQAATEEEPQNDNLYLGVVLSAVVIITGCFSYYQEAKSSKIMESFKNMVPQQALVIRNGEKMSINAEEVVVGDLVEVKGGDRIPADLRIISANGCKVDNSSLTGESEPQTRSPDFTNENPLETRNIAFFSTNCVEGTARGIVVYTGDRTVMGRIATLASGLEGGQTPIAAEIEHFIHIITGVAVFLGVSFFILSLILEYTWLEAVIFLIGIIVANVPEGLLATVTVCLTLTAKRMARKNCLVKNLEAVETLGSTSTICSDKTGTLTQNRMTVAHMWSDNQIHEADTTENQSGVSFDKTSATWLALSRIAGLCNRAVFQANQENLPILKRAVAGDASESALLKCIELCCGSVKEMRERYTKIVEIPFNSTNKYQLSIHKNPNTAEPRHLLVMKGAPERILDRCSSILIHGKEQPLDEELKDAFQNAYLELGGLGERVLGFCHLFLPDEQFPEGFQFDTDDVNFPLDNLCFVGLISMIDPPRAAVPDAVGKCRSAGIKVIMVTGDHPITAKAIAKGVGIISEGNETVEDIAARLNIPVSQVNPRDAKACVVHGSDLKDMTSEQLDDILKYHTEIVFARTSPQQKLIIVEGCQRQGAIVAVTGDGVNDSPASKKADIGVAMGIAGSDVSKQAADMILLDDNFASIVTGVEEGRLIFDNLKKSIAYTLTSNIPEITPFLIFIIANIPLPLGTVTILCIDLGTDMVPAISLAYEQAESDIMKRQPRNPKTDKLVNEQLISMAYGQIGMIQALGGFFTYFVILAENGFLPIHLLGLRVNWDDRWINDVEDSYGQQWTYEQRKIVEFTCHTPFFVTIVVVQWADLVICKTRRNSVFQQGMKNKILIFGLFEETALAAFLSYCPGMGVALRMYPLKPTWWFCAFPYSLLIFVYDEVRKLIIRRRPGGWVEKETYY 4ret A 4.0 BS07 DGX A 1 D121 N122 L125 E312 G319 V322 A323 F783 L793 R880 D101 N102 L105 E292 G299 V302 A303 F763 L773 R860 D369 D710 D714 D349 D690 D694 7.2.2.13 0000166,0002028,0005215,0005391,0005515,0005524,0005886,0005890,0006813,0006814,0006883,0008556,0010248,0016020,0016323,0016887,0030007,0030424,0030955,0031402,0036376,0042383,0042470,0042995,0046872,0051117,0055085,0086009,1902600,1990573 remove_due_to_license_issue P05024 25624492 1107 KERDMDELKKEVSMDDHKLSLDELHRKYGTDLSRGLTPARAAEILARDGPNALTPPPTTPEWVKFCRQLFGGFSMLLWIGAILCFLAYGIQAATEEEPQNDNLYLGVVLSAVVIITGCFSYYQEAKSSKIMESFKNMVPQQALVIRNGEKMSINAEEVVVGDLVEVKGGDRIPADLRIISANGCKVDNSSLTGESEPQTRSPDFTNENPLETRNIAFFSTNCVEGTARGIVVYTGDRTVMGRIATLASGLEGGQTPIAAEIEHFIHIITGVAVFLGVSFFILSLILEYTWLEAVIFLIGIIVANVPEGLLATVTVCLTLTAKRMARKNCLVKNLEAVETLGSTSTICSDKTGTLTQNRMTVAHMWSDNQIHEADTTENQSGVSFDKTSATWLALSRIAGLCNRAVFQANQENLPILKRAVAGDASESALLKCIELCCGSVKEMRERYTKIVEIPFNSTNKYQLSIHKNPNTAEPRHLLVMKGAPERILDRCSSILIHGKEQPLDEELKDAFQNAYLELGGLGERVLGFCHLFLPDEQFPEGFQFDTDDVNFPLDNLCFVGLISMIDPPRAAVPDAVGKCRSAGIKVIMVTGDHPITAKAIAKGVGIISEGNETVEDIAARLNIPVSQVNPRDAKACVVHGSDLKDMTSEQLDDILKYHTEIVFARTSPQQKLIIVEGCQRQGAIVAVTGDGVNDSPASKKADIGVAMGIAGSDVSKQAADMILLDDNFASIVTGVEEGRLIFDNLKKSIAYTLTSNIPEITPFLIFIIANIPLPLGTVTILCIDLGTDMVPAISLAYEQAESDIMKRQPRNPKTDKLVNEQLISMAYGQIGMIQALGGFFTYFVILAENGFLPIHLLGLRVNWDDRWINDVEDSYGQQWTYEQRKIVEFTCHTPFFVTIVVVQWADLVICKTRRNSVFQQGMKNKILIFGLFEETALAAFLSYCPGMGVALRMYPLKPTWWFCAFPYSLLIFVYDEVRKLIIRRRPGGWVEKETYY 4rfc A 1.645 BS02 3O1 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.7nM remove_due_to_license_issue Ki=5.7nM P00918 25358036 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rfd A 1.631 BS02 3O5 A 1 H94 H96 H119 L197 T198 T199 H91 H93 H116 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8.9nM remove_due_to_license_issue P00918 25358036 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rfd A 1.631 BS03 3O5 A 2 H4 W5 H10 N11 H15 W16 D19 H1 W2 H7 N8 H12 W13 D16 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8.9nM remove_due_to_license_issue P00918 25358036 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rfm A 2.1 BS01 3P6 A 1 I369 F374 A389 K391 F435 E436 F437 M438 E439 H440 G441 L489 I14 F19 A34 K36 F80 E81 F82 M83 E84 H85 G86 L134 D482 A484 R486 N487 D500 P521 D127 A129 R131 N132 D145 P152 2.7.10.2 0004672,0004713,0004715,0005524,0006468 Ki=0.00009uM remove_due_to_license_issue IC50=4.0nM, Ki=0.090000nM Q08881 25844760 701 SVIDPSELTFVQEIGSGQFGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEASVIHRDLAARNCLVGENQVIKVSDFGMTRFPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAAIAAS 4rfr B 1.5 BS01 RHN B 1 N120 Y122 L128 D133 I143 S145 F154 W178 H187 I189 R204 N206 T208 N107 Y109 L115 D120 I130 S132 F141 W165 H174 I176 R191 N193 T195 1.14.11.33 0005515,0005737,0005829,0006281,0006307,0008198,0035513,0035515,0035516,0042245,0046872,0051213,0070989,0072702 Kd=0.29uM remove_due_to_license_issue P05050 27015802 301 PLAAGAVILRRFAFNAAEQLIRDINDVASQSPFRQMVTPGGYTMSVAMTNCGHLGWTTHRQGYLYSPIDPQTNKPWPAMPQSFHNLCQRAATAAGYPDFQPDACLINRYAPGAKLSLHQDKDEPDLRAPIVSVSLGLPAIFQFGGLKRNDPLKRLLLEHGDVVVWGGESRLFYHGIQPLKAGFHPLTIDCRYNLTFRQAGK 4rfy A 1.7 BS01 3OU A 1 G411 F413 V416 A428 K430 Y476 M477 A478 G480 N526 L528 D539 Y551 G16 F18 V21 A33 K35 Y81 M82 A83 G85 N131 L133 D144 Y156 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=100nM remove_due_to_license_issue Q06187 25466710 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4rfz A 1.17 BS01 3OV A 1 L408 G411 Q412 V416 A428 K430 Y476 M477 A478 G480 N526 L528 D539 S543 Y551 L13 G16 Q17 V21 A33 K35 Y81 M82 A83 G85 N131 L133 D144 S148 Y156 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=40nM remove_due_to_license_issue IC50=40nM Q06187 25466710 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4rg0 A 2.5 BS01 3P0 A 1 L408 G411 V416 A428 K430 Y476 M477 A478 G480 N526 L528 D539 L13 G16 V21 A33 K35 Y81 M82 A83 G85 N131 L133 D144 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=50nM remove_due_to_license_issue IC50=50nM Q06187 25466710 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4rhu A 2.573 BS01 3QE A 1 S127 G128 T130 K154 F175 V176 D182 S105 G106 T108 K132 F153 V154 D160 E122 D123 D126 F175 R188 E100 D101 D104 F153 R166 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 remove_due_to_license_issue P9WHQ9 25915781 301 QTAELYPGDIKSVLLTAEQIQARIAELGEQIGNDYRETTGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSYSGVVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVHANVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVYQ 4rhu B 2.573 BS01 3QE B 1 G67 V124 D126 S127 G128 T130 K154 F175 V176 D182 R188 G52 V102 D104 S105 G106 T108 K132 F151 V152 D158 R164 E122 D123 D126 F175 R188 E100 D101 D104 F151 R164 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 remove_due_to_license_issue P9WHQ9 25915781 301 AELYPGDIKSVLLTAEQIQARIAELGEQIGNDYRELSATTGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSYGVVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVNVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVYQ 4rhx A 2.0322 BS01 3QF A 1 K66 G67 V90 D126 S127 G128 T130 K154 F175 V176 L181 D182 R188 K50 G51 V74 D106 S107 G108 T110 K134 F155 V156 L161 D162 R168 E122 D123 D126 F175 R188 E102 D103 D106 F155 R168 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 Ki=1.6uM remove_due_to_license_issue P9WHQ9 25915781 301 ELYPGDIKSVLLTAEQIQARIAELGEQIGNDYRELSATTGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSYGSSGVVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVHANVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVY 4rhx B 2.0322 BS01 3QF B 1 K66 G67 V90 D126 S127 G128 T130 K154 F175 V176 L181 D182 R188 K49 G50 V73 D99 S100 G101 T103 K127 F148 V149 L154 D155 R161 E122 D123 D126 F175 R188 E95 D96 D99 F148 R161 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 Ki=1.6uM remove_due_to_license_issue P9WHQ9 25915781 301 AELYPGDIKSVLLTAEQIQARIAELGEQIGNDYRSATTGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVHANVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVYQ 4rhx D 2.0322 BS01 3QF D 1 K66 G67 V90 D126 S127 G128 T130 K154 F175 V176 D182 R188 K49 G50 V73 D99 S100 G101 T103 K127 F148 V149 D155 R161 E122 D123 D126 F175 R188 E95 D96 D99 F148 R161 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 Ki=1.6uM remove_due_to_license_issue P9WHQ9 25915781 301 LYPGDIKSVLLTAEQIQARIAELGEQIGNDYRELSATTGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVHANVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVY 4rhy A 2.3196 BS02 3QG A 1 K66 G67 V125 D126 S127 G128 T130 K154 F175 V176 R188 K45 G46 V96 D97 S98 G99 T101 K125 F146 V147 R159 E122 D123 D126 F175 R188 E93 D94 D97 F146 R159 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 Ki=1.13uM remove_due_to_license_issue P9WHQ9 25915781 303 ELYPGDIKSVLLTAEQIQARIAELGEQIGNDYREGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSYVVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVHANVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVY 4rhy B 2.3196 BS02 3QG B 1 K66 G67 V125 D126 S127 G128 T130 K154 F175 V176 R188 K44 G45 V97 D98 S99 G100 T102 K126 F147 V148 R160 E122 D123 D126 F175 R188 E94 D95 D98 F147 R160 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006177,0006178,0006188,0016757,0032263,0032264,0043101,0046100,0046872,0052657 Ki=1.13uM remove_due_to_license_issue P9WHQ9 25915781 303 ELYPGDIKSVLLTAEQIQARIAELGEQIGNDYRGQDLLLITVLKGAVLFVTDLARAIPVPTQFEFMAVSSYGGVVRILKDLDRDIHGRDVLIVEDVVDSGLTLSWLSRNLTSRNPRSLRVCTLLRKPDAVHANVEIAYVGFDIPNDFVVGYGLDYDERYRDLSYIGTLDPRVY 4ri9 A 2.9 BS01 dna S 0 E675 R706 H742 K794 S795 R952 N980 E297 R328 H364 K410 S411 R558 N586 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 0 ~ 10 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 A 2.9 BS02 dna X 0 S473 Q492 K493 S104 Q123 K124 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 1 ~ 12 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 A 2.9 BS03 dna Z 0 Y374 R420 R424 K425 Y436 T573 V577 R581 Y5 R51 R55 K56 Y67 T195 V199 R203 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 11 ~ 22 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 A 2.9 BS04 dna Y 0 R679 H681 R710 L713 Q717 R749 R752 R982 R301 H303 R332 L335 Q339 R371 R374 R588 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 8 ~ 14 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 B 2.9 BS01 dna U 0 Y374 R420 R424 K425 Y436 T573 V577 R581 Y5 R51 R55 K56 Y67 T195 V199 R203 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 11 ~ 22 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 B 2.9 BS02 dna V 0 K433 S473 A474 Q492 K493 K64 S104 A105 Q123 K124 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 1 ~ 12 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 B 2.9 BS03 dna W 0 E675 R706 R710 H742 K794 R952 G956 K986 E297 R328 R332 H364 K410 R558 G562 K592 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 0 ~ 10 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4ri9 B 2.9 BS04 dna T 0 R679 H681 R710 L713 Q717 R749 R982 R301 H303 R332 L335 Q339 R371 R588 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 8 ~ 14 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rib A 3.25 BS01 dna X 0 Y374 R420 R424 K425 Y436 T573 Y5 R51 R55 K56 Y67 T195 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 0 ~ 19 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rib A 3.25 BS02 dna U 0 E675 R706 R710 P757 R955 G956 G957 D960 N980 D981 E297 R328 R332 P379 R561 G562 G563 D566 N586 D587 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 0 ~ 19 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rib A 3.25 BS03 dna Y 0 K433 S473 Q492 K493 T573 K64 S104 Q123 K124 T195 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 1 ~ 12 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rib A 3.25 BS04 dna W 0 R679 H681 R710 Q717 H718 R749 R752 R982 R301 H303 R332 Q339 H340 R371 R374 R588 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 1 ~ 7 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCKSVFVMVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rib B 3.25 BS01 dna U 0 Y374 R420 R424 K425 Y436 Y5 R51 R55 K56 Y67 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 0 ~ 19 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCPQRKSVFVMEAGEAADPTTVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rib B 3.25 BS02 dna V 0 K433 S473 A474 K493 K64 S104 A105 K124 3.1.21.-,3.1.4.1 0003676,0004518,0016788,0036297 remove_due_to_license_issue Q9Y2M0 25430771 1 ~ 12 TGHPYYLRSFLVVLKTVLENEDDMLLFDEQEKGIVTKFYQLSATGQKLYVRLFQRKLSWIKMTKLEYEEIALDLTPVIEELTNAGFLQTESELQELSEVLELLSAPELKSLAKTFHLANPNGQKQQLVDAFLKLAKQRSVIGAVILKRAKALAGQSVRICKGPRAVFSRILLLFSLTDSMEDEDAACGGQGQLSTVLLVNLGRMEFPSYTINRKTHIFQDRDDLIRYAAATHMLSDISSAMANGNWEEAKELAQCAKRDWNRLKNHPSLRCHEDLPLFLRCFTVGWIYTRILSRFVEILQRLHMYEEAVRELESLLSQRIYCPDSRGRWWDRLALNLHQHLKRLEPTIKCITEGLADPEVRTGHRLSLYQRAVRLRESPSCKKFKHLFQQLPEMAVQDVKHVTITGRLCPQRKSVFVMEAGEAADPTTVLCSVEELALAHYRRSGFDQGIHGEGSTFSTLYGLLLWDIIFMDGIPDVFRNACQAFPLDLCTDSFFTSRRPALEARLQLIHDAPEESLRAWVAATWHEQEGRVASLVSWDRFTSLQQAQDLVSCLGGPVLSGVCRHLAADFRHCRGGLPDLVVWNSQSRHFKLVEVKGPNDRLSHKQMIWLAELQKLGAEVEVCHVVAV 4rio A 2.69 BS01 3QX A 1 G829 A853 M902 E903 Y904 L905 G908 N954 L956 G15 A39 M88 E89 Y90 L91 G94 N140 L142 D949 A951 R953 N954 D967 D135 A137 R139 N140 D153 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1.000000nM P52333 25453808 4000 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 4riu A 1.651 BS02 3QR A 1 L91 H94 H96 H119 V121 V131 L198 T199 T200 L89 H92 H94 H117 V119 V128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 25614109 305 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4riv A 1.631 BS02 LSA A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=5950nM P00918 25614109 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4riv A 1.631 BS03 LSA A 2 G6 Y7 G8 F231 G3 Y4 G5 F227 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=5950nM P00918 25614109 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rj3 A 1.63 BS01 3QS A 1 I10 A31 K33 F80 L83 H84 D86 L134 D145 I10 A31 K33 F73 L76 H77 D79 L127 D138 D127 K129 Q131 N132 D145 T158 T165 D120 K122 Q124 N125 D138 T151 T158 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=93nM remove_due_to_license_issue IC50=93nM P24941 25383627 302 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPH 4rj4 A 2.78 BS01 3QW A 1 L718 F723 V726 A743 K745 M766 C775 M790 Q791 M793 L844 T854 L22 F27 V30 A47 K49 M67 C76 M91 Q92 M94 L145 T155 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 25383627 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKEATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEDMDDVVDADEYLI 4rj5 A 3.1 BS01 3QY A 1 L718 A743 K745 E762 M790 M793 G796 L844 L22 A47 K49 E62 M90 M93 G96 L144 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 25383627 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKETSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYDMDDVVDADEYLIP 4rj6 A 2.7 BS01 3R0 A 1 L718 G719 A743 E762 M790 Q791 M793 L844 D855 L22 G23 A47 E62 M90 Q91 M93 L144 D155 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 25383627 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKETSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYDMDDVVDADEYLI 4rj7 A 2.55 BS01 3R1 A 1 L718 F723 V726 A743 K745 M793 G796 L844 L22 F27 V30 A47 K49 M92 G95 L143 D837 A839 R841 N842 D855 D136 A138 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=101nM P00533 25383627 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKESPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFDMDDVVDADEYLI 4rj8 A 2.5 BS01 3QS A 1 L718 G719 V726 A743 K745 C775 M790 Q791 M793 L844 T854 D855 L22 G23 V30 A47 K49 C75 M90 Q91 M93 L144 T154 D155 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 Ki=17nM remove_due_to_license_issue Ki=553nM P00533 25383627 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEDMDDVVDADEYLI 4rkg A 2.5 BS01 dna I 0 C525 R526 C527 R543 P545 C3 R4 C5 R14 P16 2.3.2.27 0061630,0072487 remove_due_to_license_issue P50534 25452275 1 ~ 12 PKCRCGITTCRNSRCPCYKSYNSCAGCHCVGCKNPHK 4rkg B 2.5 BS01 dna I 0 C525 R526 C527 N534 R543 P545 C4 R5 C6 N13 R22 P24 2.3.2.27 0061630,0072487 remove_due_to_license_issue P50534 25452275 1 ~ 12 KPKCRCGISGSSNTLTTCRNSRCPCYKSYNSCAGCHCVGCKNPHKE 4rkx A 1.59 BS01 3S9 A 1 C192 V193 S280 G281 S282 Q332 G333 V334 C47 V48 S135 G136 S137 Q187 G188 V189 C192 H340 W357 C47 H195 W212 3.4.22.10 0006508,0008234 Ki=8uM remove_due_to_license_issue A0A0M3KKW7 26132413 502 QPVVKSLLNSKGIHYNQGNPYNLLTPVIEKVKPGEQSFVGQHAATGCVATATAQIMKYHNYPNKGLKDYTYTLSSNNPYFNHPKNLFAAISTRQYNWNNILPTYSGRESNVQKMAISELMADVGISVDMDYGPSSGSAGSSRVQRALKENFGYNQSVHQINRSDFSKQDWEAQIDKELSQNQPVYYQGVGKVGGHAFVIDGADGRNFYHVNWGWGGVSDGFFRLDALNPSALGTGGGAGGFNGYQSAVVGIKPL 4rlk A 1.24 BS01 E91 A 1 V45 I66 K68 V95 F113 Y115 V116 N118 M163 I174 D175 V39 I60 K62 V89 F107 Y109 V110 N112 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue P28523 25449433 406 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAENS 4rll A 1.85 BS01 E91 A 1 L45 V66 K68 F113 M163 I174 D175 L44 V65 K67 F112 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 25449433 402 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 4rlp A 2.79 BS01 72B A 1 L97 G98 K99 G100 V105 A121 L172 Y174 L175 E179 E222 M225 T235 L13 G14 K15 G16 V21 A37 L72 Y74 L75 E79 E122 M125 T135 D218 K220 E222 N223 D236 T256 D118 K120 E122 N123 D136 T145 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P23443 25356520 401 KIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKRNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPL 4rlt A 2.049 BS01 FSE A 1 C61 G64 Y65 Q68 Q86 Q89 L91 N125 T140 L142 C61 G64 Y65 Q68 Q86 Q89 L91 N125 T140 L142 4.2.1.59 0005515,0005886,0006633,0016836,0019171 Kd=10.9uM remove_due_to_license_issue P9WFK1 26081470 201 VALSADIVGMHYRYPDHYEVEREKIREYAVAVQNDDAWYFEEDGAAELGYKGLLAPLTFICVFGYKAQAAFFKHANIATAEAQIVQVDQVLKFEKPIVAGDKLYCDVYVDSVREAHGTQIIVTKNIVTNEEGDLVQETYTTLAGRAGGEGFSDGA 4rlu A 2.198 BS01 HCC A 1 C61 G64 Y65 Q68 Q86 Q89 N125 T138 T140 C61 G64 Y65 Q68 Q86 Q89 N125 T138 T140 4.2.1.59 0005515,0005886,0006633,0016836,0019171 remove_due_to_license_issue P9WFK1 26081470 201 VALSADIVGMHYRYPDHYEVEREKIREYAVAVQNDDAWYFEEDGAAELGYKGLLAPLTFICVFGYKAQAAFFKHANIATAEAQIVQVDQVLKFEKPIVAGDKLYCDVYVDSVREAHGTQIIVTKNIVTNEEGDLVQETYTTLAGRAEGFSDG 4rlw A 2.196 BS01 BUN A 1 C61 G64 Y65 Q68 Q86 Q89 N125 T138 T140 L142 C61 G64 Y65 Q68 Q86 Q89 N125 T138 T140 L142 4.2.1.59 0005515,0005886,0006633,0016836,0019171 remove_due_to_license_issue P9WFK1 26081470 201 VALSADIVGMHYRYPDHYEVEREKIREYAVAVQNDDAWYFEEDGAAELGYKGLLAPLTFICVFGYKAQAAFFKHANIATAEAQIVQVDQVLKFEKPIVAGDKLYCDVYVDSVREAHGTQIIVTKNIVTNEEGDLVQETYTTLAGRAGEGFSDG 4rn0 A 1.761 BS01 L6G A 1 Y100 H143 F152 D178 H180 F208 M274 Y306 Y81 H124 F133 D159 H161 F189 M255 Y287 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=255nM remove_due_to_license_issue IC50=255nM Q9BY41 25793284 501 LVPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 4rn0 A 1.761 BS03 L6G B 1 P273 Y306 P254 Y287 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=255nM remove_due_to_license_issue IC50=255nM Q9BY41 25793284 501 LVPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 4rn1 A 2.18 BS02 L8G A 1 Y100 H143 F152 H180 F208 Y306 Y83 H126 F135 H163 F191 Y289 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue Q9BY41 25793284 404 LVPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 4rn1 A 2.18 BS03 L8G B 1 F152 Y306 F135 Y289 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue Q9BY41 25793284 404 LVPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVVI 4rn2 A 2.39 BS02 L7G A 1 H143 F152 H180 F208 Y306 H115 F124 H152 F180 Y278 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=1500nM remove_due_to_license_issue IC50=1491nM Q9BY41 25793284 404 VPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQSIEYGLTEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 4rn2 A 2.39 BS03 L7G B 1 K33 P273 Y306 K19 P245 Y278 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=1500nM remove_due_to_license_issue IC50=1491nM Q9BY41 25793284 404 VPVYIYSPEYVSMCDSLAKIPKRADMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQSIEYGLTEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 4rn4 A 1.53 BS02 3T7 A 1 I91 Q92 H94 H96 H119 F130 L197 T198 T199 I89 Q90 H92 H94 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=114nM remove_due_to_license_issue P00918 25581127 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rn6 A 3.0 BS01 15U A 1 H57 Y60A W60D W148 W215 G216 H74 Y78 W81 W179 W252 G253 H57 D102 E192 G193 D194 A195 G196 H74 D130 E227 G228 D229 A230 G231 3.4.21.5 0004252,0005509,0005576,0006508,0007596 remove_due_to_license_issue P00734 23467412 301 EADCGLRPLFEKKSLEDKTERELLESYIDGRIVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTAPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDAGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 4rpn D 2.272 BS01 PCI D 1 S104 F106 F151 F167 E169 Y171 H206 F231 P248 V275 S16 F18 F63 F79 E81 Y83 H118 F143 P160 V187 ? Kd=110nM remove_due_to_license_issue P52679 25397598 401 RFDPGTSNRNFRIAASDFGQALMLPRLYATLEETAPQVRVTGVNLRHGPLVEELESGSIDIAFGGFPTLSAGIKTQTLFREEYVCVMRQSHPALTHGLDLEAFRQCRHIIVTAHEFNHVHEQVEARLLELLPPESIRFTTENFLVSAVIAEETDVILTIPSRLARWFANRGGLTIFPVPIELPSIEVKQYWHERYDKDPGNIWLRRVIAKIGFQNPPA 4rpn D 2.272 BS02 PCI D 2 F106 A109 L110 P113 R114 R250 L251 W254 F18 A21 L22 P25 R26 R162 L163 W166 ? Kd=110nM remove_due_to_license_issue P52679 25397598 402 RFDPGTSNRNFRIAASDFGQALMLPRLYATLEETAPQVRVTGVNLRHGPLVEELESGSIDIAFGGFPTLSAGIKTQTLFREEYVCVMRQSHPALTHGLDLEAFRQCRHIIVTAHEFNHVHEQVEARLLELLPPESIRFTTENFLVSAVIAEETDVILTIPSRLARWFANRGGLTIFPVPIELPSIEVKQYWHERYDKDPGNIWLRRVIAKIGFQNPPA 4rpn D 2.272 BS03 PCI C 2 V236 E240 V148 E152 ? Kd=110nM remove_due_to_license_issue P52679 25397598 402 RFDPGTSNRNFRIAASDFGQALMLPRLYATLEETAPQVRVTGVNLRHGPLVEELESGSIDIAFGGFPTLSAGIKTQTLFREEYVCVMRQSHPALTHGLDLEAFRQCRHIIVTAHEFNHVHEQVEARLLELLPPESIRFTTENFLVSAVIAEETDVILTIPSRLARWFANRGGLTIFPVPIELPSIEVKQYWHERYDKDPGNIWLRRVIAKIGFQNPPA 4rpo A 1.95 BS01 T6C A 1 S104 F106 F151 F167 E169 H206 F231 P248 S16 F18 F63 F79 E81 H118 F143 P160 ? Kd=22.8nM remove_due_to_license_issue P52679 25397598 401 RFDPGTSNRNFRIAASDFGQALMLPRLYATLEETAPQVRVTGVNLRHGPLVEELESGSIDIAFGGFPTLSAGIKTQTLFREEYVCVMRQSHPALTHGLDLEAFRQCRHIIVTAHEFNHVHEQVEARLLELLPPESIRFTTENFLVSAVIAEETDVILTIPSRLARWFANRGGLTIFPVPIELPSIEVKQYWHERYDKDPGNIWLRRVIAKIGFQNPPAE 4rpv A 3.05 BS01 3UR A 1 F49 A65 K67 L120 E121 N172 L174 D186 F17 A33 K35 L88 E89 N140 L142 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 25597005 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4rqk A 1.55 BS02 R1S A 1 K115 I118 I119 V127 R131 T148 F149 L155 K42 I45 I46 V54 R58 T75 F76 L82 D205 K207 E209 N210 D223 T245 D132 K134 E136 N137 D150 T172 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Kd=1500nM O15530 25518860 404 PRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 4rqv A 1.502 BS02 R2S A 1 K115 I118 I119 V124 T128 R131 T148 L155 F157 K45 I48 I49 V54 T58 R61 T78 L85 F87 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T175 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 25518860 406 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 4rr6 A 1.88 BS01 A3S A 1 A19 V42 Y75 A76 A88 F112 G113 W114 A19 V42 Y75 A76 A88 F112 G113 W114 6.1.1.3 0004829,0005524,0005737,0008270 Kd=1uM remove_due_to_license_issue Q9YFY3 26113036 500 MRLLYLHADRFEYKTVKPALKNPPDPPGEASFGEALVVFTTVEDGDGPQTVMYAASDIASHSSRLKVTTVILYPYAHLSSRLAKPMAAHKRLIELEGALRTKFPGHVHRAPFGWYKSFSIACKGHPLAELSRSFTE 4rra A 1.7 BS01 A3T A 1 V42 P74 Y75 L82 A88 F112 G113 W114 Y115 V42 P74 Y75 L82 A88 F112 G113 W114 Y115 6.1.1.3 0004829,0005524,0005737,0008270 Kd=13.4uM remove_due_to_license_issue Q9YFY3 26113036 201 MRLLYLHADRFEYKTVKPALKNPPDPPGEASFGEALVVFTTVEDGDGPQTVMYAASDIASHSSRLKVTTVILYPYAHLSSRLAKPMAAHKRLIELEGALRTKFPGHVHRAPFGWYKSFSIACKGHPLAELSRSFTE 4rrf A 1.7 BS01 A3S A 1 I25 V46 P81 Y82 A83 H84 L89 A95 F118 G119 W120 Y121 I21 V42 P77 Y78 A79 H80 L85 A91 F114 G115 W116 Y117 6.1.1.3 0004829,0005524,0005737,0008270 Kd=239.2uM remove_due_to_license_issue Q58597 26113036 501 MKMLLIHSDYLEFEAKEKTKIAEETENLKGKLDECLACFIAVEREDENNPEGTAIGAVEEIEKVANQLKVNNIVVYPYAHLSSDLSSPETAVKVLKDIESILKERGYNVLRAPFGWYKAFKISCKGHPLSELSRKIVA 4rrf D 1.7 BS01 A3S D 1 I25 V46 Y82 L89 A95 F118 G119 I21 V42 Y78 L85 A91 F114 G115 6.1.1.3 0004829,0005524,0005737,0008270 Kd=239.2uM remove_due_to_license_issue Q58597 26113036 201 MKMLLIHSDYLEFEAKEKTKIAEETENLKGKLDECLACFIAVEREDENNPEGTAIGAVEEIEKVANQLKVNNIVVYPYAHLSSDLSSPETAVKVLKDIESILKERGYNVLRAPFGWYKAFKISCKGHPLSELSRKIVAK 4rrg A 1.93 BS01 A3T A 1 I25 V46 Y82 A83 H84 A95 F118 G119 I21 V42 Y78 A79 H80 A91 F114 G115 6.1.1.3 0004829,0005524,0005737,0008270 Kd=1538.5uM remove_due_to_license_issue Q58597 26113036 501 MKMLLIHSDYLEFEAKEKTKIAEETENLKGKLDECLACFIAVEREDENNPEGTAIGAVEEIEKVANQLKVNNIVVYPYAHLSSDLSSPETAVKVLKDIESILKERGYNVLRAPFGWYKAFKISCKGHPLSELSRKIVA 4rrg B 1.93 BS01 A3T B 1 V46 Y82 H84 L89 S90 A95 F118 Y121 V42 Y78 H80 L85 S86 A91 F114 Y117 6.1.1.3 0004829,0005524,0005737,0008270 Kd=1538.5uM remove_due_to_license_issue Q58597 26113036 201 MKMLLIHSDYLEFEAKEKTKIAEETENLKGKLDECLACFIAVEREDENNPEGTAIGAVEEIEKVANQLKVNNIVVYPYAHLSSDLSSPETAVKVLKDIESILKERGYNVLRAPFGWYKAFKISCKGHPLSELSRKIVA 4rrn A 1.8 BS01 3UW A 1 G72 Q73 G74 L91 D93 Y132 F169 I171 W176 D289 G291 G13 Q14 G15 L32 D34 Y73 F110 I112 W117 D223 G225 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=48nM remove_due_to_license_issue IC50=12nM P56817 25411915 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4rro A 1.8 BS01 3UX A 1 G72 Q73 G74 L91 D93 Y132 F169 I171 W176 I179 D289 G291 G13 Q14 G15 L32 D34 Y73 F110 I112 W117 I120 D223 G225 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=26nM remove_due_to_license_issue IC50=26nM P56817 25411915 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4rrq A 1.79 BS01 A3S A 1 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 6.1.1.3 0004829,0005524,0005737,0008270 remove_due_to_license_issue Q9UZ14 26113036 500 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYMAFKISCKGHPLAELSRTIVP 4rrq B 1.79 BS01 A3S B 1 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 M121 A19 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 M121 6.1.1.3 0004829,0005524,0005737,0008270 remove_due_to_license_issue Q9UZ14 26113036 501 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYMAFKISCKGHPLAELSRTIVPEEARVE 4rrr A 1.86 BS01 A3T A 1 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 V45 P80 F81 A82 A94 F117 G118 Y119 Y120 6.1.1.3 0004829,0005524,0005737,0008270 remove_due_to_license_issue Q9UZ14 26113036 201 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYMAFKISCKGHPLAELSRTIVPEE 4rrr B 1.86 BS01 A3T B 1 L20 V45 P80 F81 A82 L88 A94 F117 G118 Y119 Y120 L20 V45 P80 F81 A82 L88 A94 F117 G118 Y119 Y120 6.1.1.3 0004829,0005524,0005737,0008270 remove_due_to_license_issue Q9UZ14 26113036 201 MRVLLIHSDYIEYEVKDKALKNPEPISEDMKRGRMEEVLVAFISVEKVDEKNPEEVSLKAIEEISKVAEQVKAENVFVYPFAHLSSELAKPSVAMDILNRVYQGLKERGFNVGKAPFGYYMAFKISCKGHPLAELSRTIVPE 4rrs A 1.8 BS01 3UY A 1 G72 Q73 G74 L91 D93 Y132 F169 I171 I179 D289 G291 G13 Q14 G15 L32 D34 Y73 F110 I112 I120 D223 G225 D93 S96 N98 A100 Y132 D289 T292 D34 S37 N39 A41 Y73 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=210nM remove_due_to_license_issue IC50=130nM P56817 25411915 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4rs0 A 2.807 BS01 IBP A 1 R120 V349 Y355 G526 A527 R89 V318 Y324 G495 A496 Q203 H207 L384 Y385 H388 G526 S530 Q172 H176 L353 Y354 H357 G495 S499 1.14.99.1 0001516,0001525,0004601,0004666,0005515,0005634,0005637,0005640,0005737,0005783,0005789,0005901,0006979,0007566,0007612,0007613,0008217,0008284,0008285,0009410,0009624,0009750,0010042,0010269,0010575,0016020,0016702,0019371,0019899,0020037,0030216,0030282,0031394,0031622,0031915,0032227,0032310,0032355,0032496,0032991,0033138,0033280,0034097,0034605,0034612,0035633,0042127,0042307,0042633,0042803,0043005,0043065,0043066,0045429,0045786,0045907,0045986,0045987,0046697,0046872,0048661,0050873,0051213,0051384,0051926,0051968,0070542,0071222,0071260,0071284,0071318,0071456,0071471,0071498,0071636,0090050,0090271,0090336,0090362,0098869,0150077,1902219,1905375,1990776,2000117 remove_due_to_license_issue IC50=860nM Q05769 25825493 706 ANPCCSNPCQNRGECMSTGFDQYKCDCTRTGFYGENCTTPEFLTRIKLLLKPTPNTVWYILTHFKGVWNIVNNIPFLRSLIMKYVLTSRSYLIDSPPTYNVHYGYKSWEAFSNLSYYTRALPPVADDCPTPMGVKGNKELPDSKEVLEKVLLRREFIPDPQGSNMMFAFFAQHFTHQFFKTDHKRGPGFTRGLGHGVDLNHIYGETLDRQHKLRLFKDGKLKYQVIGGEVYPPTVKDTQVEMIYPPHIPENLQFAVGQEVFGLVPGLMMYATIWLREHNRVCDILKQEHPEWGDEQLFQTSRLILIGETIKIVIEDYVQHLSGYHFKLKFDPELLFNQQFQYQNRIASEFNTLYHWHPLLPDTFNIEDQEYSFKQFLYNNSILLEHGLTQFVESFTRQIAGRVAGGRNVPIAVQAVAKASIDQSREMKYQSLNEYRKRFSLKPYTSFEELTGEKEMAAELKALYSDIDVMELYPALLVEKPRPDAIFGETMVELGAPFSLKGLMGNPICSPQYWKPSTFGGEVGFKIINTASIQSLICNNVKGCPFTSFNVQDPQPT 4rsc A 1.8 BS02 A3V A 1 F61 F103 V134 T147 E148 N194 F59 F101 V114 T127 E128 N174 3.1.1.64,5.3.3.22 0001523,0001786,0001895,0003834,0004744,0005634,0005737,0005783,0005789,0005886,0006629,0007601,0016020,0016702,0016787,0016853,0031210,0042572,0042574,0042802,0046872,0050251,0050908,0052884,0052885,1901612,1901827 ic50=232nM remove_due_to_license_issue IC50=<1000nM Q28175 25894083 603 SQVEHPAGGYKKLFETVEELSSPLTAHVTGRIPLWLTGSLLRCGPGLFEVGSEPFYHLFDGQALLHKFDFKEGHVTYHRRFIRTDAYVRAMTEKRIVITEFGTCAFEVTDNALVNIYPVGEDYYACTETNFITKVNPETLETIKQVDLCNYVSVNGATAHPHIENDGTVYNIGNCFIAYNIVKIPPLQADKEDPISKSEIVVQFPCSDRFKPSYVHSFGLTPNYIVFVETPVKINLFKFLSSGANYMDCFESNETMGVWLHIADKKRKKYINNKYRTSPFNLFHHINTYEDHEFLIVDLCCWKGFEFVYNYLYLANLRENWEEVKKNARKAPQPEVRRYVLPLNIDKADTGKNLVTLPNTTATAILCSDETIWLEPEVLFSGPRQAFEFPQINYQKYGGKPYTYAYGLGLNHFVPDRLCKLNVKTKETWVWQEPDSYPSEPIFVSHPDALEEDDGVVLSVVVSPGAGQKPAYLLILNAKDLSEVARAEVEINIPVTFHGLFKKS 4rse A 2.39 BS02 A6V A 1 F61 F103 T147 E148 N194 Y275 F60 F102 T129 E130 N176 Y252 3.1.1.64,5.3.3.22 0001523,0001786,0001895,0003834,0004744,0005634,0005737,0005783,0005789,0005886,0006629,0007601,0016020,0016702,0016787,0016853,0031210,0042572,0042574,0042802,0046872,0050251,0050908,0052884,0052885,1901612,1901827 ic50=396nM remove_due_to_license_issue Q28175 25894083 603 SSQVEHPAGGYKKLFETVEELSSPLTAHVTGRIPLWLTGSLLRCGPGLFEVGSEPFYHLFDGQALLHKFDFKEGHVTYHRRFIRTDAYVRAMTEKRIVITEFGTCAFPEVTDNALVNIYPVGEDYYACTETNFITKVNPETLETIKQVDLCNYVSVNGATAHPHIENDGTVYNIGNCFIAYNIVKIPPLQADKEDPISKSEIVVQFPCSDRFKPSYVHSFGLTPNYIVFVETPVKINLFKFLSSWSLWGANYMDCFESNETMGVWLHIADKKRKKYINNKYRTSPFNLFHHINTYEDHEFLIVDLCCWKGFEFVYNYLYLANLRENWEEVKKNARKAPQPEVRRYVLPLNIDKADTGKNLVTLPNTTATAILCSDETIWLEPEVLFSGPRQAFEFPQINYQKYGGKPYTYAYGLGLNHFVPDRLCKLNVKTKETWVWQEPDSYPSEPIFVSHPDALEEDDGVVLSVVVSPGAGQKPAYLLILNAKDLSEVARAEVEINIPVTFHGLFKKS 4rsk A 2.1 BS01 U3P A 1 H12 K41 N44 T45 H119 F120 H12 K41 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Kd=47.4uM remove_due_to_license_issue Ki=78500nM P61823 9860854 125 KETAAAAFEAQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACANGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 4rss A 1.83 BS01 4MG A 1 A400 M448 M450 A451 G454 P455 R498 L501 D512 A37 M83 M85 A86 G89 P90 R133 L136 D147 D494 A496 R498 N499 D512 K533 D129 A131 R133 N134 D147 K168 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.7nM remove_due_to_license_issue IC50=56nM P43405 26384287 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEAPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV 4rt0 A 1.8 BS01 C2E A 1 E14 A15 R17 R21 R95 E1 A2 R4 R8 R82 2.4.1.33 0035438 Kd=3.13uM remove_due_to_license_issue Q9HY69 25817996 201 EAQRQFARVKLPARIRYIGANREGVDARLLDLSAGGFAFTASGAPIQPGDLYKGKMLFQVDSISFSLEVEFQVRSVDPASRRVGCEFQNLKPREVAALRYLITSYLAGE 4rt0 A 1.8 BS02 C2E A 2 R17 Q18 R21 D44 S46 G48 G49 F50 A51 R87 R95 G97 C98 E99 R4 Q5 R8 D31 S33 G35 G36 F37 A38 R74 R82 G84 C85 E86 2.4.1.33 0035438 Kd=3.13uM remove_due_to_license_issue Q9HY69 25817996 202 EAQRQFARVKLPARIRYIGANREGVDARLLDLSAGGFAFTASGAPIQPGDLYKGKMLFQVDSISFSLEVEFQVRSVDPASRRVGCEFQNLKPREVAALRYLITSYLAGE 4rt1 A 1.7 BS01 C2E A 1 A15 Q16 R17 Q18 R21 D44 S46 G48 G49 F50 A51 R87 G97 C98 E99 A2 Q3 R4 Q5 R8 D31 S33 G35 G36 F37 A38 R74 G84 C85 E86 2.4.1.33 0035438 Kd=0.73uM remove_due_to_license_issue Q9HY69 25817996 201 EAQRQFARVKLPARIRYIGANREGVDARLLDLSAGGFAFTASGAPIQPGDLYKGKMLFQVDSISFSLEVEFQVRSVDPASRAVGCEFQNLKPREVAALRYLITSYLAG 4ruu A 1.4 BS01 RET A 1 F16 T53 Y60 L77 K108 F16 T53 Y60 L77 K108 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 23224553 201 TRDQNGTWEMESNENFEGYMKALDIDFATRKIAVRLTQTLVIDQDGDNFKTKTTSTFRNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 4rux A 1.14 BS02 3W3 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=12nM remove_due_to_license_issue Ki=12nM P00918 25766630 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rux A 1.14 BS03 3W3 A 2 D180 G183 D176 G179 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=12nM remove_due_to_license_issue Ki=12nM P00918 25766630 309 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ruy A 1.14 BS02 3W6 A 1 H94 H96 H119 L198 T199 T200 H91 H93 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=12.8nM remove_due_to_license_issue Ki=13nM P00918 25766630 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ruy A 1.14 BS03 3W6 A 2 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=12.8nM remove_due_to_license_issue Ki=13nM P00918 25766630 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ruz A 1.63 BS02 3W8 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=23nM P00918 25766630 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ruz A 1.63 BS03 3W8 A 2 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=23nM P00918 25766630 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4rvk A 1.85 BS01 3XK A 1 L15 A36 K38 L84 E85 Y86 C87 G90 L137 D148 L13 A34 K36 L75 E76 Y77 C78 G81 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=13.5nM remove_due_to_license_issue EC50=425nM, IC50=14nM O14757 25988399 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 4rvl A 1.85 BS01 3XL A 1 L15 A36 K38 L84 E85 C87 G90 E91 L137 D148 L13 A28 K30 L69 E70 C72 G75 E76 L122 D133 D130 K132 E134 N135 D148 T170 D115 K117 E119 N120 D133 T155 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=41.7nM remove_due_to_license_issue EC50=>5000nM, IC50=42nM O14757 25988399 301 VPFVEDWDLVQTLGVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 4rvm A 1.86 BS01 3X7 A 1 T14 L15 A36 K38 L84 E85 Y86 C87 L137 D148 T12 L13 A34 K36 L75 E76 Y77 C78 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1.000000nM, EC50=53nM O14757 25988399 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 4rvr A 1.98 BS01 3WQ A 1 W1887 P1888 P1892 V1893 V1898 I1950 W32 P33 P37 V38 V43 I95 ? remove_due_to_license_issue Kd=60nM, IC50=430nM Q9UIF8 25799074 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKVS 4rvt A 2.4 BS01 3XM A 1 V31 Y36 A52 E106 F107 C108 G109 L160 V170 V18 Y23 A39 E89 F90 C91 G92 L143 V153 D153 K155 Q157 N158 D171 T191 D136 K138 Q140 N141 D154 T163 2.7.11.1 0004672,0005524,0006468 ic50=1.9uM remove_due_to_license_issue O95819 25908259 401 DLSSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEEIKLEINMLKKYSHHRNIATYYGAFIKKSPPGHDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVNTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRT 4rwj A 2.489 BS01 66T A 1 L484 G485 F489 A512 K514 E531 M535 I545 V561 A564 S565 G567 L630 D641 L28 G29 F33 A56 K58 E75 M79 I89 V105 A108 S109 G111 L174 D185 D623 A625 R627 N628 D641 D167 A169 R171 N172 D185 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=2nM remove_due_to_license_issue P11362 25686244 801 MAGVSEYELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQ 4rwk A 2.982 BS01 66T A 1 L484 V492 A512 A564 S565 G567 L630 D641 L28 V36 A56 A108 S109 G111 L174 D185 D623 A625 R627 N628 D641 D167 A169 R171 N172 D185 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 25686244 801 MAGVSEYELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIMEYASKGNLREYLQARRPPGLEYSYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQ 4rwl B 2.193 BS01 3ZC B 1 L484 A512 K514 E531 M535 V561 E562 Y563 A564 L630 D641 F642 L27 A52 K54 E71 M75 V101 E102 Y103 A104 L157 D168 F169 D623 A625 R627 N628 D641 D150 A152 R154 N155 D168 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=8nM remove_due_to_license_issue IC50=18nM P11362 25686244 801 AGVSEYELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQ 4rww A 1.6 BS01 2BA A 1 I7 G34 F36 L37 V91 Q92 G94 I7 G34 F36 L37 V91 Q92 G94 ? remove_due_to_license_issue Q8Y3Y7 25693966 2001 MKLIFAIVQDQDSNRLSDALTKGNFGATKLATTGGFLKAGNTTFIIGTEDERVEDALAIIKENCKAREQMMTPSASLGVTVDTYVPYPIEVQVGGATVFVMPVESFHHFLEHH 4rww A 1.6 BS02 2BA A 2 M1 E49 D50 E51 R52 M1 E49 D50 E51 R52 ? remove_due_to_license_issue Q8Y3Y7 25693966 2002 MKLIFAIVQDQDSNRLSDALTKGNFGATKLATTGGFLKAGNTTFIIGTEDERVEDALAIIKENCKAREQMMTPSASLGVTVDTYVPYPIEVQVGGATVFVMPVESFHHFLEHH 4rww A 1.6 BS03 2BA C 1 G26 A27 T28 G47 H108 G26 A27 T28 G47 H108 ? remove_due_to_license_issue Q8Y3Y7 25693966 2001 MKLIFAIVQDQDSNRLSDALTKGNFGATKLATTGGFLKAGNTTFIIGTEDERVEDALAIIKENCKAREQMMTPSASLGVTVDTYVPYPIEVQVGGATVFVMPVESFHHFLEHH 4rww B 1.6 BS01 2BA A 1 G26 A27 T28 G47 H108 G26 A27 T28 G47 H102 ? remove_due_to_license_issue Q8Y3Y7 25693966 2001 MKLIFAIVQDQDSNRLSDALTKGNFGATKLATTGGFLKAGNTTFIIGTEDERVEDALAIIKENCKAREQMMTPTVDTYVPYPIEVQVGGATVFVMPVESFHHFLEH 4rww B 1.6 BS02 2BA B 1 I7 G34 F36 L37 V91 Q92 G94 T97 I7 G34 F36 L37 V85 Q86 G88 T91 ? remove_due_to_license_issue Q8Y3Y7 25693966 2001 MKLIFAIVQDQDSNRLSDALTKGNFGATKLATTGGFLKAGNTTFIIGTEDERVEDALAIIKENCKAREQMMTPTVDTYVPYPIEVQVGGATVFVMPVESFHHFLEH 4rx5 A 1.356 BS01 3YO A 1 L408 T410 G411 F413 V416 K430 Y476 M477 A478 G480 L528 D539 L15 T17 G18 F20 V23 K37 Y83 M84 A85 G87 L135 D146 D521 A523 R525 N526 D539 F559 D128 A130 R132 N133 D146 F166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=3.0nM Q06187 26675441 706 SWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 4rx7 A 1.8 BS01 3YV A 1 L377 A400 M448 E449 A451 G454 P455 R498 L501 D512 L15 A38 M83 E84 A86 G89 P90 R133 L136 D147 D494 A496 R498 N499 D512 K533 D129 A131 R133 N134 D147 K168 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5nM remove_due_to_license_issue IC50=104nM P43405 25633741 703 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHH 4rx8 A 1.59 BS01 3YX A 1 L377 A400 M448 M450 A451 G454 P455 R498 L501 S511 D512 L14 A37 M80 M82 A83 G86 P87 R130 L133 S143 D144 D494 A496 R498 N499 D512 K533 D126 A128 R130 N131 D144 K164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=35nM remove_due_to_license_issue IC50=367nM, Kd=0.640000nM P43405 25633741 703 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHH 4rx9 A 1.75 BS01 3YT A 1 L377 A400 M448 E449 A451 P455 R498 L501 D512 L15 A35 M78 E79 A81 P85 R128 L131 D142 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K162 2.7.10.2 0004672,0004713,0005524,0006468 ic50=13nM remove_due_to_license_issue IC50=178nM P43405 25633741 702 VYLDRKLLTLEDKELGFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHHH 4rxa A 2.2 BS01 3F2 A 1 K57 N59 R60 L62 T63 V66 F239 D243 G343 K347 K46 N48 R49 L51 T52 V55 F226 D230 G323 K327 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K46 F86 D91 D95 R100 D162 K187 F226 D230 D231 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.8uM remove_due_to_license_issue IC50=1.8e+3nM P14324 25815158 1001 QEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQIKENYGQVAVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 4rxc A 2.31 BS01 HRX A 1 D103 R112 Q172 K212 D92 R101 Q161 K199 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H87 D92 D96 R101 D164 K199 F238 D242 D243 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50~33uM remove_due_to_license_issue Q86C09 25815158 401 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPRLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKR 4rxc A 2.31 BS04 HRX A 2 F251 Q252 D255 F238 Q239 D242 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H87 D92 D96 R101 D164 K199 F238 D242 D243 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50~33uM remove_due_to_license_issue Q86C09 25815158 405 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPRLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKR 4rxc B 2.31 BS01 HRX B 1 D103 R112 Q172 Y216 D93 R102 Q162 Y203 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K199 F238 D242 D243 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50~33uM remove_due_to_license_issue Q86C09 25815158 401 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKR 4rxc B 2.31 BS04 HRX B 2 F251 Q252 D255 K269 F238 Q239 D242 K256 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K199 F238 D242 D243 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50~33uM remove_due_to_license_issue Q86C09 25815158 405 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKR 4rxd A 2.0 BS03 RIS A 1 D103 R112 Q172 K212 T213 D255 K269 D91 R100 Q160 K200 T201 D243 K257 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K45 H86 D91 D95 R100 D163 K200 F239 D243 D244 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=300nM remove_due_to_license_issue Q86C09 25815158 1404 MQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 4rxd C 2.0 BS01 RIS C 1 D103 R112 Q172 K212 T213 D255 K269 D93 R102 Q162 K202 T203 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=300nM remove_due_to_license_issue Q86C09 25815158 1600 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 4rxe A 2.5 BS01 3YQ A 1 D103 D107 R112 K212 Y216 D255 K269 D94 D98 R103 K203 Y207 D246 K260 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H89 D94 D98 R103 D166 K203 F242 D246 D247 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=230nM remove_due_to_license_issue Q86C09 25815158 3001 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSLDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 4ryc A 2.45 BS01 3ZK A 1 T12 Q13 V30 D32 G34 Y75 S76 T77 P111 L114 A115 F117 Q128 L213 D215 G217 A218 T17 Q18 V35 D37 G39 Y82 S83 T84 P117 L120 A121 F123 Q134 L220 D222 G224 A225 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y82 D222 A225 3.4.23.15 0004190,0006508 ic50=0.08uM remove_due_to_license_issue IC50=80nM P00797 25782742 1001 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4ryg A 2.65 BS01 3ZJ A 1 T12 Q13 Y14 V30 D32 G34 Y75 S76 T77 P111 F117 V120 L213 D215 G217 A218 I291 T17 Q18 Y19 V35 D37 G39 Y82 S83 T84 P117 F123 V126 L220 D222 G224 A225 I301 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y82 D222 A225 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=8.0nM P00797 25782742 1001 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4ryl A 2.1 BS01 3ZG A 1 K392 H393 R396 V420 E422 T466 A467 K150 H151 R154 V178 E180 T224 A225 D253 E346 E355 H496 D11 E104 E113 H254 2.1.1.319 0016274,0018216 Kd=53nM remove_due_to_license_issue IC50=91nM, EC50=2000nM O60678 25728001 601 HYGIHEEMLKDKIRTESYRDFIYQNPHIFKDKVVLDVGCGTGILSMFAAKAGAKKVLGVDQSEILYQAMDIIRLNKLEDTITLIKGKIEEVHLPVEKVDVIISEWMGYFLLFESMLDSVLYAKNKYLAKGGSVYPDICTISLVAVSDVNKHADRIAFWDDVYGFKMSCMKKAVIPEAVVEVLDPKTLISEPCGIKHIDCHTTSISDLEFSSDFTLKITRTSMCTAIAGYFDIYFEKNCHNRVVFSTGPQSTKTHWKQTVFLLEKPFSVKAGEALKGKVTVHKSLTVTLTLNNSTQTYGLQ 4rz1 A 2.6 BS01 3ZN A 1 T12 Q13 V30 D32 G34 Y75 S76 T77 P111 L114 F117 L213 D215 G217 A218 I291 T17 Q18 V35 D37 G39 Y82 S83 T84 P117 L120 F123 L220 D222 G224 A225 I301 D32 S35 N37 W39 Y75 D215 A218 D37 S40 N42 W44 Y82 D222 A225 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=80nM P00797 25754490 1001 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4s04 A 3.2 BS01 dna C 0 T151 K153 Y179 T187 N188 R210 T151 K153 Y179 T187 N188 R210 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 A 3.2 BS02 dna D 0 H195 R198 T208 R210 G211 Y214 H195 R198 T208 R210 G211 Y214 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 B 3.2 BS01 dna C 0 T151 K153 Y179 P185 T187 N188 T189 V192 H193 R210 T151 K153 Y179 P185 T187 N188 T189 V192 H193 R210 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 B 3.2 BS02 dna D 0 H195 K203 T208 R210 G211 Y214 H195 K203 T208 R210 G211 Y214 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 E 3.2 BS01 dna G 0 T151 P152 K153 Y179 T187 N188 H193 R210 T151 P152 K153 Y179 T187 N188 H193 R210 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 E 3.2 BS02 dna H 0 H195 R198 K203 T208 R210 Y214 H195 R198 K203 T208 R210 Y214 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 F 3.2 BS01 dna G 0 T151 K153 Y179 A186 T187 N188 T189 H193 R210 T151 K153 Y179 A186 T187 N188 T189 H193 R210 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s04 F 3.2 BS02 dna H 0 E191 H195 T208 R210 G211 Y214 E191 H195 T208 R210 G211 Y214 ? 0000156,0000160,0000976,0003677,0005829,0006355,0032993,0046872 remove_due_to_license_issue A0A0R4I965 26564787 1 ~ 25 MKILVIEDDALLLQGLILAMQSEGYVCDGVSTAHEAALSLASNHYSLIVLDLGLPDEDGLHFLSRMRREKMTQPVLILTARDTLEDRISGLDTGADDYLVKPFALEELNARIRALLRRHNNQGDNEISVGNLRLNVTRRLVWLGETALDLTPKEYALLSRLMMKAGSPVHREILYNDIYSGDNEPATNTLEVHIHNLREKIGKSRIRTVRGFGYMLANN 4s0n A 1.501 BS01 dna E 0 G69 Y72 Y73 Y93 D94 H110 K112 K113 F142 G14 Y17 Y18 Y38 D39 H55 K57 K58 F87 2.3.2.27,3.6.4.- 0003676,0008270,0016818 remove_due_to_license_issue Q14527 26051180 5 ~ 10 DSVLFGSLRGHVVGLRYYTGVVNNNEMVALQRDPNNPYDKNAIKVNNVNGNQVGHLKKELAGALAYIMDNKLAQIEGVVPFGANNAFTMPLHMTFWGKEENRKAVSDQLKKHGFKLGPAPKT 4s0n B 1.501 BS01 dna F 0 R71 Y72 Y73 N91 Y93 D94 H110 K112 K113 F142 R16 Y17 Y18 N36 Y38 D39 H55 K57 K58 F87 2.3.2.27,3.6.4.- 0003676,0008270,0016818 remove_due_to_license_issue Q14527 26051180 7 ~ 10 DSVLFGSLRGHVVGLRYYTGVVNNNEMVALQRDPNNPYDKNAIKVNNVNGNQVGHLKKELAGALAYIMDNKLAQIEGVVPFGANNAFTMPLHMTFWGKEENRKAVSDQLKKHGFKLGPAPKTLGF 4s0n C 1.501 BS01 dna G 0 G69 Y72 Y73 Y93 D94 H110 K113 G19 Y22 Y23 Y43 D44 H60 K63 2.3.2.27,3.6.4.- 0003676,0008270,0016818 remove_due_to_license_issue Q14527 26051180 7 ~ 10 GPGSVDSVLFGSLRGHVVGLRYYTGVVNNNEMVALQRDPNNPYDKNAIKVNNVNGNQVGHLKKELAGALAYIMDNKLAQIEGVVPFGANNAFTMPLHMTFWGKEENRKAVSDQLKKHGFKLGPA 4s0n D 1.501 BS01 dna E 0 S62 H147 P173 S12 H97 P123 2.3.2.27,3.6.4.- 0003676,0008270,0016818 remove_due_to_license_issue Q14527 26051180 5 ~ 10 GPGSVDSVLFGSLRGHVVGLRYYTGVVNNNEMVALQRDPNNPYDKNAIKVNNVNGNQVGHLKKELAGALAYIMDNKLAQIEGVVPFGANNAFTMPLHMTFWGKEENRKAVSDQLKKHGFKLGPAPK 4s0n D 1.501 BS02 dna H 0 V68 G69 Y72 Y73 Y93 D94 H110 K112 K113 V18 G19 Y22 Y23 Y43 D44 H60 K62 K63 2.3.2.27,3.6.4.- 0003676,0008270,0016818 remove_due_to_license_issue Q14527 26051180 7 ~ 10 GPGSVDSVLFGSLRGHVVGLRYYTGVVNNNEMVALQRDPNNPYDKNAIKVNNVNGNQVGHLKKELAGALAYIMDNKLAQIEGVVPFGANNAFTMPLHMTFWGKEENRKAVSDQLKKHGFKLGPAPK 4s1g A 2.1 BS01 43T A 1 D104 Y149 S150 T151 P184 D292 G294 H367 D37 Y82 S83 T84 P117 D225 G227 H300 D104 S107 N109 W111 Y149 D292 A295 D37 S40 N42 W44 Y82 D225 A228 3.4.23.15 0004190,0006508 Ki=0.6nM remove_due_to_license_issue P00797 25728416 502 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4s2i A 1.6 BS01 NXL A 1 C69 S70 N104 S130 N132 N170 T235 G236 S237 C42 S43 N77 S103 N105 N143 T208 G209 S210 S70 K73 S130 E166 K234 S237 S43 K46 S103 E139 K207 S210 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue G3G192 27622530 301 ADVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTD 4s3f A 1.7 BS01 43W A 1 M29 R56 D87 R110 R141 N145 K204 T231 R260 S262 M26 R53 D84 R107 R138 N142 K201 T228 R257 S259 1.17.7.3 0005506,0008299,0016114,0016491,0019288,0044237,0046429,0046872,0051539,0141197 ic50=580nM remove_due_to_license_issue Q5SLI8 25868383 902 MRRPTPTVYVGRVPIGGAHPIAVQSMTNTPTRDVEATTAQVLELHRAGSEIVRLTVNDEEAAKAVPEIKRRLLAEGAEVPLVGDFHFNGHLLLRKYPKMAEALDKFRINPGTLGRGRHKDEHFAEMIRIAMDLGKPVRIGANWGSLDPALLTELMDRNARRPEPKSAHEVVLEALVESAVRAYEAALEMGLGEDKLVLSAKVSKARDLVWVYRELARRTQAPLHLGLTEAGMGVKGIVASAAALAPLLLEGIGDTIRVSLTPAPGEPRTKEVEVAQEILQALGLRAFAPEVTSCPGCGRTTSTFFQELAEEVSRRLKERLPEWRARYPGVEELKVAVMGCVVNGPGESKHAHIGISLPGAGEEPKAPVYADGKLLTILKGEGIAEEFLRLVEDYVKTRFAP 4std A 2.15 BS01 BFS A 1 Y30 Y50 V75 L76 V108 S129 I151 F158 F162 G165 Y22 Y42 V67 L68 V100 S121 I143 F150 F154 G157 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=47pM remove_due_to_license_issue Ki=47nM P56221 10382670 173 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFGDK 4std B 2.15 BS01 BFS B 1 Y30 Y50 V75 L76 V108 S129 N131 P149 F162 G165 Y22 Y42 V67 L68 V100 S121 N123 P141 F154 G157 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=47pM remove_due_to_license_issue Ki=47nM P56221 10382670 174 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFGDK 4tim B 2.4 BS01 2PG B 1 N11 K13 H95 I172 G173 G211 S213 L232 G234 G235 N10 K12 H94 I171 G172 G210 S212 L231 G233 G234 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=6.9mM remove_due_to_license_issue P04789 1895291 300 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 4tju A 1.57 BS02 CNQ A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 I1075 E1138 H69 G70 Y97 F98 K104 S105 Y108 I112 E175 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 KEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tjw A 1.7 BS02 P34 A 1 H1031 G1032 Y1050 G1053 G1056 Y1060 F1061 K1067 S1068 Y1071 I1075 E1138 H69 G70 Y88 G91 G94 Y98 F99 K105 S106 Y109 I113 E176 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=2951nM Q9H2K2 25286857 1202 KEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4tjy A 1.9 BS02 3GN A 1 H1031 G1032 Y1060 F1061 K1067 S1068 Y1071 E1138 H70 G71 Y99 F100 K106 S107 Y110 E177 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tk0 A 1.65 BS02 32Z A 1 H1031 G1032 G1053 Y1060 F1061 K1067 Y1071 I1075 E1138 H70 G71 G92 Y99 F100 K106 Y110 I114 E177 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tk5 A 2.02 BS02 UHB A 1 H1031 G1032 S1033 F1035 I1039 F1044 D1045 H1048 A1049 G1058 Y1060 S1068 Y1071 H72 G73 S74 F76 I80 F85 D86 H89 A90 G99 Y101 S109 Y112 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 PDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tkf A 2.6 BS02 33C A 1 H1031 S1033 F1035 A1038 G1043 F1044 D1045 H1048 Y1050 I1059 Y1060 Y1071 H70 S72 F74 A77 G82 F83 D84 H87 Y89 I98 Y99 Y110 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=31nM Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tkg A 1.95 BS02 09L A 1 H1031 G1032 I1039 H1048 Y1050 I1059 Y1060 F1061 S1068 Y1071 I1075 E1138 H70 G71 I78 H87 Y89 I98 Y99 F100 S107 Y110 I114 E177 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=2340nM Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4tki A 2.15 BS02 33E A 1 H1031 G1032 Y1050 Y1060 S1068 Y1071 H70 G71 Y89 Y99 S107 Y110 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1202 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tki A 2.15 BS03 33E A 2 F1035 A1038 I1039 H1048 F74 A77 I78 H87 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1203 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tki A 2.15 BS04 33E A 3 K999 C1001 N1002 K1003 W1006 Y1148 E1150 K38 C40 N41 K42 W45 Y187 E189 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 25286857 1204 DKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRP 4tln A 2.3 BS06 LNO A 1 N112 A113 H142 E143 H146 E166 R203 H231 N112 A113 H142 E143 H146 E166 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=190uM remove_due_to_license_issue Kd=190546nM P00800 7317361 322 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 4tlr A 1.86 BS01 33H A 1 L419 R422 M423 H475 S476 Y477 I482 R501 W528 L419 R422 M423 H475 S476 Y477 I482 R501 W528 0003723,0003968,0039694 ic50=0.003uM remove_due_to_license_issue 24986660 601 SMSYTWTGALITPCAAEETKLPINALSNSLLRHHNLVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSL 4tmf A 2.05 BS01 JS2 A 1 L124 W125 S126 R127 L145 E146 D156 W189 S220 T221 F222 E226 L77 W78 S79 R80 L98 E99 D109 W142 S173 T174 F175 E179 E146 T221 E226 E99 T174 E179 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue P28907 25226087 401 QTWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFDTSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVEVHNLQPEKVQTLEAWVIHGRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKNPEDSSC 4tmk A 1.98 BS01 T5A A 1 E12 G13 G15 K16 T17 R39 E40 L55 F74 R78 R100 S104 T105 Y108 Q109 R149 R153 I159 E11 G12 G14 K15 T16 R38 E39 L54 F73 R77 R99 S103 T104 Y107 Q108 R148 R152 I158 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0015949,0016301,0042803,0046940 Kd=20nM remove_due_to_license_issue P0A720 9826650 214 RSKYIVIEGLEGAGKTTARNVVVETLEQLGIRDMVFTREPGGTQLAEKLRSLLLDIKSVGDEVITDKAEVLMFYAARVQLVETVIKPALANGTWVIGDRHDLSTQAYQGGGRGIDQHMLATLRDAVLGDFRPDLTLYLDVTPEVGLKRARARGELDRIEQESFDFFNRTRARYLELAAQDKSIHTIDATQPLEAVMDAIRTTVTHWVKEL 4tmn E 1.7 BS01 0PK E 1 N112 A113 F114 W115 H142 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 W115 H142 E143 H146 Y157 E166 L202 R203 H231 3.4.24.27 0004222,0006508 Ki=0.068nM remove_due_to_license_issue Ki=99999999999999nM P00800 3442675 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 4tmr A 2.7 BS02 99S A 1 L124 G128 H129 L130 V141 T183 N354 K355 N356 T357 C364 R371 L124 G128 H129 L130 V141 T183 N354 K355 N356 T357 C364 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tmr A 2.7 BS03 99S B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tmr B 2.7 BS01 99S A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tmr B 2.7 BS03 99S B 1 L124 G128 H129 L130 V141 T183 N356 C364 R371 L124 G128 H129 L130 V141 T183 N356 C364 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tmu A 2.4 BS01 dna B 0 L74 I75 N96 S97 E124 R125 W154 F158 R159 P223 L224 S245 R246 R259 H267 A268 T293 V294 R315 W347 M432 G433 A442 N443 N444 R446 H489 S490 L71 I72 N93 S94 E121 R122 W151 F155 R156 P220 L221 S242 R243 R256 H264 A265 T290 V291 R312 W344 M429 G430 A439 N440 N441 R443 H486 S487 5.6.2.4 0003676,0003678,0004386,0005524,0006260,0006281,0006310,0009432,0043138 remove_due_to_license_issue A7MQK9 25831501 3 ~ 33 AEVYSQETLAKQVLQETFGYQQFRPGQATIIDAVLEGRDCLVVMPTGGGKSLCYQIPALVKTGLTIVVSPLISLMKDQVDQLLANGVAAACLNSTQSREEQQAVLAGCRTGQVRLLYIAPERLMMDNFIDTLGYWDLAMVAVDEAHCISQWGHDFRPEYAALGQLRARFPAVPFMALTATADDTTRRDIVRLLGLDDPLIEISSFDRPNIRYMLMEKFKPLDQLMRYVQEQRGKSGIIYCNSRAKVEDTAARLQSRGISAAAYHAGLEHEVRASVQEKFQRDDLQIVVATVAFGMGINKPNVRFVVHFDIPRNIESYYQETGRAGRDGLPAEAMLFYDPADMAWLRRCLEEKAPGPLQDIERHKLNAMGAFAEAQTCRRLVLLNYFGEGRQAPCGNCDICLDPPRRYDGLVDAQKALSAIARVEQRFGMGYVVEVLRGANNQRIRELGHDKLKVYGIGRDQSQEHWVSVIRQLIHLGVVTQNIAQHSALQLTEAARPFLRGEAPLMLAVPR 4tn2 A 2.7 BS01 33J A 1 L419 R422 M423 H475 S476 Y477 I482 L497 W528 L413 R416 M417 H469 S470 Y471 I476 L491 W522 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue P26663 24986660 900 ASYTWTGALITPCAAEESKLPINALSNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGVQEDAASLRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLFQGPAASQLDLSGWFVAGYSGGDIYHSLSRA 4tn4 A 2.2 BS02 33G A 1 L124 G127 G128 T183 N354 K355 N356 L124 G127 G128 T183 N354 K355 N356 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 503 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tn4 A 2.2 BS04 33G B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 503 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tn4 B 2.2 BS02 33G A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 503 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tn4 B 2.2 BS04 33G B 1 L124 G128 T183 N354 K355 R371 L124 G128 T183 N354 K355 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 25785478 503 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 4tpk A 2.7 BS02 3F9 A 1 I69 D70 W82 G117 F329 Y332 I67 D68 W80 G115 F327 Y330 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0004104 remove_due_to_license_issue IC50=21nM, Ki=2.7nM P06276 25226236 615 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 4tpm A 2.77 BS01 35E A 1 L665 T675 I682 Y683 P702 M703 E711 V712 G715 F719 L212 T222 I229 Y230 P249 M250 E258 V259 G262 F266 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=2.4nM Q9Y233 25456383 2009 LPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVI 4tpp A 2.65 BS02 35D A 1 I682 Y683 P702 M703 E711 G715 Q716 F719 I230 Y231 P250 M251 E259 G263 Q264 F267 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=2.6nM Q9Y233 25456383 1011 TLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIR 4tpt A 2.6 BS01 35H A 1 K360 I363 M380 V388 L403 L442 H449 A468 D469 F470 L472 R474 K31 I34 M51 V59 L74 L113 H120 A139 D140 F141 L143 R145 D451 N453 H455 N456 D469 N509 D122 N124 H126 N127 D140 N157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=92nM P53671 25589930 701 DLIHGEVLGKGFFGQAIKVTHKATGKVMVMKELIRCDEETQKTFLTEVKVMRSLDHPNVLKFIGVLYKDKKLNLLTEYIEGGTLKDFLRSMDPFPWQQKVRFAKGIASGMAYLHSMCIIHRDLNSHNCLIKLDKTVVVADFGLSRLIVKKRYTVVGNPYWMAPEMLNGKSYDETVDIFSFGIVLCEIIGQVYADPDCLPRTLDFGLNVKLFWEKFVPTDCPPAFFPLAAICCRLEPESRPAFSKLEDSFEALSLYLGELGIPLPAELEELDHTVSMQYG 4tpt B 2.6 BS01 35H B 1 K360 L362 I363 M380 V388 T405 H449 A468 D469 F470 L472 R474 K31 L33 I34 M51 V59 T76 H120 A139 D140 F141 L143 R145 D451 N453 H455 N456 D469 N509 D122 N124 H126 N127 D140 N154 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=92nM P53671 25589930 701 DLIHGEVLGKGFFGQAIKVTHKATGKVMVMKELIRCDEETQKTFLTEVKVMRSLDHPNVLKFIGVLYKDKKLNLLTEYIEGGTLKDFLRSMDPFPWQQKVRFAKGIASGMAYLHSMCIIHRDLNSHNCLIKLDKTVVVADFGLSRLIVYTVVGNPYWMAPEMLNGKSYDETVDIFSFGIVLCEIIGQVYADPDCLPRTLDFGLNVKLFWEKFVPTDCPPAFFPLAAICCRLEPESRPAFSKLEDSFEALSLYLGELGIPLPAELEELDHTVSMQYGL 4tpw A 1.5 BS02 33R A 1 F47 K49 N59 R61 I63 H78 F15 K17 N27 R29 I31 H46 ? 0003723,0003743,0005737,0006413 Kd=20.5uM remove_due_to_license_issue P06730 25049413 302 HYIKHPLQNRWALWFFKNDKSKTWQANLRLISKFDTVEDFWALYNHIQLSSNLMPGCDYSLFKDGIEPMWEDEKNKRGGRWLITLNKQQRRSDLDRFWLETLLCLIGESFDDYSDDVCGAVVNVRAKGDKIAIWTTECENREAVTHIGRVYKERLGLPPKIVIGYQSHADTATKSGSTTKNRFVV 4tq3 A 2.4076 BS01 GPP A 1 R22 S64 F65 N68 L88 Y139 K146 R8 S50 F51 N54 L70 Y121 K128 ? 0005886,0016020,0016740,0016765,0046872 Kd=3.2uM remove_due_to_license_issue O28625 25051182 401 SKYLRLLRPVAWLCFLLPYAVGFGFGITPNASLQHAVLGLLSFAFWMAFSFTINALYDRDVDRLHDGLNLSMQPLVTGEISVREAWLYCIAFLALSLATAAAINEKFFLAMLGANIIGYVYSAPPRFKAWPVMDVICNALAAVLAFYAGLSIGGAEVPIAIYPAAFFLAATFYIPTAVSDYEFDKKAGLKNTPVFFGPERALKSLYPLSAITVILWAYVFLMAERIEIKVISPLIIAYTLIYTFIINSRWDGEKLNVSPNLILTPFGIISALFIAYGFAVISV 4tqn A 1.7 BS01 UL4 A 1 L1109 P1110 V1115 L1120 I1122 N1168 R1173 V1174 L26 P27 V32 L37 I39 N85 R90 V91 2.3.1.-,2.3.1.48 Kd=0.77uM remove_due_to_license_issue IC50=8700nM, Kd=670nM Q92793 26125948 1201 IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQS 4trc A 2.4 BS01 ADE A 1 I97 D99 W148 F149 I96 D98 W147 F148 D95 D96 D99 D94 D95 D98 2.4.2.- 0000166,0016757 remove_due_to_license_issue Q97W95 25790177 301 QKIPVKVVTWDEIVSLSTKLAEKIKADEYNVNVIVAIARGGLVPARLVADVLGVFDILSIKIEHWIETASHTPEAKVKYPFKVDLSDKNVLIIDDITDTGDSIELARKYVMENFRPTEVKTATLQYIKPAAKIIPDYYAEEIVSWAWFMYPWNYWEDEINLVNKILIERKTKDIDINELKRNFVESYGIENPPISLDKILTEMKRRKIV 4ts1 A 2.5 BS01 TYR A 1 Y34 G36 D78 Y169 Q173 D176 Q195 Y34 G36 D78 Y169 Q173 D176 Q195 T40 H45 H48 K82 R86 Q173 D194 K230 K233 T234 T40 H45 H48 K82 R86 Q173 D194 K228 K231 T232 6.1.1.1 0000166,0004812,0004831,0005524,0006418,0006437 Kd=11.6uM remove_due_to_license_issue P00952 3612807 320 MDLLAELQWRGLVNQTTDEDGLRKLLNEERVTLYCGFDPTADSLHIGHLATILTMRRFQQAGHRPIALVGGATGLIGDPSGKKSERTLNAKETVEAWSARIKEQLGRFLDFEADGNPAKIKNNYDWIGPLDVITFLRDVGKHFSVNYMMAKESVQSRIETGISFTEFSYMMLQAYDFLRLYETEGCRLQIGGSDQWGNITAGLELIRKTKGRAFGLTIPLVTKADGTKFGKTESGTIWLDKEKTSPYEFYQFWINTDDRDVIRYLKYFTFLSKEEIEALEQELREAPEKRAAQKTLAEEVTKLVHGEEALRQAIRYA 4tsx A 1.94 BS01 LF0 A 1 Q95 L102 T124 T125 A128 A129 W132 Q41 L48 T70 T71 A74 A75 W78 ? 0003676,0015074 Kd=10.3uM remove_due_to_license_issue F2WR39 25421939 301 DCSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGIPESMNKELKKIIGQVRDQAETLKTAVQMAVFIHNKKRKGGGGYSAGERIVDIIATDIQ 4tte A 1.8 BS01 36Z A 1 V1008 P1012 N1064 I1074 V30 P34 N86 I96 3.6.1.- Kd=202uM remove_due_to_license_issue Q6PL18 25486442 1204 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4ttv A 2.8 BS01 BC9 A 1 G387 H388 R442 Y540 D564 L567 H590 G67 H68 R122 Y220 D244 L247 H270 C413 R442 Q460 D462 H464 K543 H590 C93 R122 Q140 D142 H144 K223 H270 6.1.1.3 0000166,0004812,0004829,0005524,0005737,0006418,0006435 remove_due_to_license_issue P26639 26271225 801 SDHRKIGRDQELYFFHELSPGSCFFLPKGAYIYNALIEFIRSEYRKRGFQEVVTPNIFNSRLWMTSGHWQHYSENMFSFEVEKELFALKPMNCPGHCLMFDHRPRSWRELPLRLADFGVLHRNELSGALTGLTRVRRFQQDDAHIFCAMEQIEDEIKGCLDFLRTVYSVFGFSFKLNLSTRPEKFLGDIEVWDQAEKQLENSLNEFGEKWELNSGDGAFYGPKIDIQIKDAIGRYHQCATIQLDFQLPIRFNLTYVSHDGDDKKRPVIVHRAILGSVERMIAILTENYGGKWPFWLSPRQVMVVPVGPTCDEYAQKVRQQFHDAKFMADIDLDPGCTLNKKIRNAQLAQYNFILVVGEKEKISGTVNIRTRDNKVHGERTISETIERLQQLKEFRSKQAEEEF 4tu4 A 1.73 BS01 37N A 1 R1007 V1008 V1013 D1014 E1017 Y1063 N1064 I1074 R29 V30 V35 D36 E39 Y85 N86 I96 3.6.1.- Kd=175uM remove_due_to_license_issue Q6PL18 25486442 1204 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4tuh A 1.8 BS01 38H A 1 A93 E96 F97 Y101 R102 F105 S106 L108 T109 L130 N136 G138 R139 A142 S145 F146 A149 Y195 A41 E44 F45 Y49 R50 F53 S54 L56 T57 L78 N84 G86 R87 A90 S93 F94 A97 Y143 ? 0042981 remove_due_to_license_issue Ki=0.380000nM, EC50=60nM Q07817 24944740 301 PLGSMSQSNRELVVDFLSYKLSQKGYSWSQMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 4tun A 1.925 BS01 MVH A 1 E35 N44 D52 Q57 N59 W63 A107 W108 E35 N44 D52 Q57 N59 W63 A107 W108 E35 N46 D48 S50 D52 N59 E35 N46 D48 S50 D52 N59 3.2.1.17 0003796,0005515,0005576,0005615,0005737,0005783,0016231,0016798,0016998,0031640,0042742,0042802,0050829,0050830,0051672 remove_due_to_license_issue P00698 24969463 201 KVFGRCELAAAMKRHGLDNYRGYSLGNWVCAAKFESNFNTQATNRNTDGSTDYGILQINSRWWCNDGRTPGSRNLCNIPCSALLSSDITASVNCAKKIVSDGNGMNAWVAWRNRCKGTDVQAWIRGCRL 4tuw A 2.902 BS01 rna D 0 R225 D226 R38 D39 ? 0003723,0003729 remove_due_to_license_issue Q9VAN6 25002523 1 ~ 26 SSYTEADPAILSRRQKQIDYGKNTAAYERYVEMVPRTRDHPREPNKYGKYSRRAFDGLVKIWRKSLHIYDP 4tuw A 2.902 BS02 rna C 0 S185 K200 Y204 N207 Y237 S238 R239 R240 A241 G244 L245 K247 I248 R250 H254 S1 K16 Y20 N23 Y50 S51 R52 R53 A54 G57 L58 K60 I61 R63 H67 ? 0003723,0003729 remove_due_to_license_issue Q9VAN6 25002523 1 ~ 28 SSYTEADPAILSRRQKQIDYGKNTAAYERYVEMVPRTRDHPREPNKYGKYSRRAFDGLVKIWRKSLHIYDP 4tuw B 2.902 BS01 rna D 0 R197 Y204 N207 Y237 S238 R239 R240 A241 G244 L245 K247 R250 H254 R12 Y19 N22 Y49 S50 R51 R52 A53 G56 L57 K59 R62 H66 ? 0003723,0003729 remove_due_to_license_issue Q9VAN6 25002523 1 ~ 26 SYTEADPAILSRRQKQIDYGKNTAAYERYVEMVPKTRDHPREPNKYGKYSRRAFDGLVKIWRKSLHIYDP 4tux A 3.08 BS01 rna C 0 R197 K200 Y204 N207 Y237 S238 R239 R240 A241 L245 K247 R250 H254 R12 K15 Y19 N22 Y51 S52 R53 R54 A55 L59 K61 R64 H68 ? 0003723,0003729 remove_due_to_license_issue Q9VAN6 25002523 1 ~ 25 SYTEADPAILSRRQKQIDYGKNTAAYERYVEMVPKDERTRHPRTPNKYGKYSRRAFDGLVKIWRKSLHIYD 4tux B 3.08 BS01 rna D 0 R197 Y204 N207 Y237 S238 R239 R240 A241 L245 K247 I248 R250 K251 H254 R12 Y19 N22 Y48 S49 R50 R51 A52 L56 K58 I59 R61 K62 H65 ? 0003723,0003729 remove_due_to_license_issue Q9VAN6 25002523 1 ~ 26 SYTEADPAILSRRQKQIDYGKNTAAYERYVEMVPKDEHPRTPNKYGKYSRRAFDGLVKIWRKSLHIY 4tv3 A 2.85 BS01 ML9 A 1 R770 I800 K802 D810 Y836 V851 Q859 M922 I932 D933 R627 I657 K659 D667 Y693 V708 Q716 M772 I782 D783 2.7.11.1,2.7.1.137,2.7.1.153 0016301,0046854 remove_due_to_license_issue IC50=8.3nM, Ki=0.57nM P42336 25043846 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRKSLWVINSALRIKILCATYVNVNDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREAGFSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDRVPFVLTQDFLIVISTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDA 4tvj A 2.1 BS01 09L A 1 E335 H428 G429 R444 Y455 Y462 F463 S470 Y473 E113 H206 G207 R222 Y233 Y240 F241 S248 Y251 K264 A265 I289 F305 T307 S470 Y473 E558 K42 A43 I67 F83 T85 S248 Y251 E336 2.4.2.-,2.4.2.30 0003950 ic50=251nM remove_due_to_license_issue IC50=2.8nM, Kd=0.280000nM Q9UGN5 28001384 601 DLGTENLYFQSMDLRVQELIKLICNVQAMEEMMMEMKYNTKKAPLGKLTVAQIKAGYQSLKKIEDCIRAGQHGRALMEACNEFYTRIPHDFGLRTPPLIRTQKELSEKIQLLEALGDIEIAIKLVKTELQSPEHPLDQHYRNLHCALRPLDHESYEFKVISQYLQSTHAPTHSDYTMTLLDLFEVEKDGEKEAFREDLHNRMLLWHGSRMSNWVGILSHGLRIAHPEAPITGYMFGKGIYFADMSSKSANYCFASRLKNTGLLLLSEVALGQCNELLEANPKAEGLLQGKHSTKGLGKMAPSSAHFVTLNGSTVPLGPASDTGILNPDGYTLNYNEYIVYNPNQVRMRYLLKVQFNF 4tw6 A 1.4 BS01 37L A 1 Y57 K60 D68 F77 G84 Q85 V86 I87 W90 Y113 K121 Y45 K48 D56 F65 G72 Q73 V74 I75 W78 Y101 K109 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=61000nM remove_due_to_license_issue Q13451 25436518 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4tw7 A 1.25 BS01 37K A 1 Y57 K60 D68 F77 G84 Q85 V86 I87 W90 Y113 F130 Y45 K48 D56 F65 G72 Q73 V74 I75 W78 Y101 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=26nM remove_due_to_license_issue Q13451 25436518 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4tw8 A 3.003 BS01 37M A 1 Y57 G59 D68 E85 V86 I87 W90 Y113 K121 I122 F130 Y37 G39 D48 E65 V66 I67 W70 Y93 K101 I102 F110 Y57 F67 D68 I87 Y113 F130 Y37 F47 D48 I67 Y93 F110 5.2.1.8 0003755 remove_due_to_license_issue Q02790 25436518 301 EGVDISPKQDEGVLKVIKREGTGTEMPMIGDRVFVHYTGWLLDGTKFDSSLDRKDKFSFDLGKGEVIKAWDIAIATMKVGEVCHITCKPEYAYGSAGSPPKIPPNATLVFEVELFEFKGEDLTEEEDGGIIRRIQTRGEGYAKPNEGAIVEVALEGYYKDKLFDQRELRFEIGEGENLDLPYGLERAIQRMEKGEHSIVYLKPSYAFGSVGKEKFQIPPNAELKYELHLKSFEKA 4tw9 A 2.4 BS01 386 A 1 I15 A36 Y56 M82 L85 G86 P87 D91 L135 I14 A35 Y55 M81 L84 G85 P86 D90 L134 D128 K130 D127 K129 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.02uM remove_due_to_license_issue P48730 25191940 1010 ELRVGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAAKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF 4tw9 B 2.4 BS01 386 B 1 I23 A36 Y56 M82 L85 G86 P87 D91 L135 L293 I23 A36 Y56 M82 L85 G86 P87 D91 L135 L287 D128 K130 D128 K130 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.02uM remove_due_to_license_issue P48730 25191940 1007 MELRVGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF 4twc A 1.7 BS01 37J A 1 A36 Y56 L85 G86 P87 D91 L92 L135 L293 A35 Y55 L84 G85 P86 D90 L91 L134 L291 D128 K130 D127 K129 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=22nM P48730 22331384 1007 ELRVGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF 4twd A 3.2 BS01 377 A 1 F133 Y175 F188 F123 Y165 F178 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue P0C7B7 25199693 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENADNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYASYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 4twd E 3.2 BS01 377 E 1 E131 Y175 F188 E121 Y165 F178 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue P0C7B7 25199693 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENADNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYASYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 4twp A 2.4 BS01 AXI A 1 L248 Y253 A269 K271 E316 F317 M318 G321 L370 D381 L16 Y21 A37 K39 E79 F80 M81 G84 L133 D144 D363 A365 R367 N368 D381 P402 D126 A128 R130 N131 D144 P165 2.7.10.2 0004672,0004713,0005524,0006468 Ki=100pM remove_due_to_license_issue P00519 25686603 601 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSIS 4tww A 2.42 BS01 3A7 A 1 H41 M49 F140 L141 N142 G143 S144 C145 H163 E166 D187 I188 H41 M49 F140 L141 N142 G143 S144 C145 H163 E166 D187 I188 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=63uM remove_due_to_license_issue IC50=63000nM P0C6X7 25614110 401 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDIQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 4tww B 2.42 BS01 3A7 B 1 M49 F140 L141 N142 G143 S144 C145 H163 E166 M49 F140 L141 N142 G143 S144 C145 H163 E166 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=63uM remove_due_to_license_issue IC50=63000nM P0C6X7 25614110 401 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDIQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 4twy A 1.6 BS01 3BL A 1 H41 T45 A46 M49 F140 L141 G143 C145 E166 H41 T45 A46 M49 F140 L141 G143 C145 E166 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue IC50=108000nM P0C6X7 25614110 401 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDIQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 4tx6 A 1.9 BS01 38B A 1 Y34 G123 A124 D172 E174 Q230 Y232 W312 Y6 G95 A96 D144 E146 Q202 Y204 W284 3.2.1.14 0004553,0005975 ic50=2.6uM remove_due_to_license_issue B0Y2Y2 25063338 401 SNLAIYWGQGPNQLRLSHFCQETSLDIINIGFINYFPDMSPGHWPGSNFGNQCDGSVYVTNDGVVTKLLSGCHQIMEDIPICQAAGKKVLLSIGGAYPPDQSILSEDSAVAFATFLWGAFGPVAEGWEGPRPFGDVVVDGFDFDIEHNGGFGYATMVNTFRQYFNQVPERKFYLSAAPQCIIPDAQLSDAIFNAAFDFIWIQYYNTAACSAKSFIDTSLGTFNFDAWVTVLKASASKDAKLYVGLPASETAANQGYYLTPDEVESLVSTYMDRYPDTFGGIMLWEATASENNQIDGAPYADHMKDILLH 4txc A 1.951 BS01 38G A 1 L19 A40 K42 E64 I77 L93 V96 E143 N144 M146 D161 L18 A39 K41 E63 I76 L92 V95 E142 N143 M145 D160 V27 D139 K141 E143 N144 D161 T180 V26 D138 K140 E142 N143 D160 T179 2.7.11.1 0004672,0005524,0006468 Kd=0.24uM remove_due_to_license_issue P53355 25382253 301 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 4txe A 1.8 BS01 38F A 1 Y32 Q35 F60 A110 D155 E157 A187 F210 Q212 Y214 W285 Y8 Q11 F36 A86 D131 E133 A163 F186 Q188 Y190 W261 3.2.1.14 0004553,0005975 ic50=2.4uM remove_due_to_license_issue P29029 25063338 401 ANTNIAVYWGQNSAGTQESLATYCESSDADIFLLSFLNQFPTLGLNFANACSDTFSDGLLHCTQIAEDIETCQSLGKKVLLSLGGASGSYLFSDDSQAETFAQTLWDTFGEGTGASERPFDSAVVDGFDFDIENNNEVGYSALATKLRTLFAEGTKQYYLSAAPQCPYPDASVGDLLENADIDFAFIQFYNNYCSVSGQFNWDTWLTYAQTVSPNKNIKLFLGLPGSASAAGSGYISDTSLLESTIADIASSSSFGGIALWDASQAFSNELNGEPYVEILKNLLTSAS 4ty1 A 2.7 BS01 38W A 1 G47 V52 A65 K67 L120 E121 V126 L174 I185 D186 G15 V20 A33 K35 L88 E89 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 remove_due_to_license_issue IC50=1.578nM P11309 25599837 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4ty6 A 1.85 BS02 39D A 1 H40 C42 H57 I151 D189 A190 C191 K192 G193 S195 T213 H27 C29 H44 I141 D182 A183 C184 K185 G186 S188 T206 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=30nM remove_due_to_license_issue P03951 25405503 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4ty7 A 2.09 BS01 39F A 1 R39 H40 L41 C42 H57 Y143 I151 D189 A190 C191 K192 G193 S195 T213 W215 R26 H27 L28 C29 H44 Y134 I141 D182 A183 C184 K185 G186 S188 T206 W208 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.3nM remove_due_to_license_issue P03951 25405503 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4ty8 A 2.78 BS01 3AV A 1 P197 C366 S368 Y448 P187 C356 S358 Y438 2.7.7.48,3.6.4.13 0000166,0001172,0003689,0003723,0003968,0004386,0006338,0006508,0008236,0016020,0016887,0034062,0039694,0061775,0140584,0140588,0140665,0140849 remove_due_to_license_issue D0PY27 25666181 601 SMSYTWTGALITPCAAEESKLPNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPISGWFVAGYSGGDIYH 4ty9 A 2.78 BS01 3B0 A 1 E361 N369 S371 E481 E351 N359 S361 E471 2.7.7.48,3.6.4.13 0000166,0001172,0003689,0003723,0003968,0004386,0006338,0006508,0008236,0016020,0016887,0034062,0039694,0061775,0140584,0140588,0140665,0140849 remove_due_to_license_issue D0PY27 25666181 601 SMSYTWTGALITPCAAEESKLPNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPLSSMFVAGYSGGDIYH 4tya A 2.94 BS01 3AE A 1 C366 S368 L384 M414 Y448 C356 S358 L374 M404 Y438 2.7.7.48,3.6.4.13 0000166,0001172,0003689,0003723,0003968,0004386,0006338,0006508,0008236,0016020,0016887,0034062,0039694,0061775,0140584,0140588,0140665,0140849 remove_due_to_license_issue D0PY27 25666181 601 SMSYTWTGALITPCAAEESKLPNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPISGWFVAGYSGGDIYH 4tyb A 2.93 BS01 3B1 A 1 C366 M414 Y415 Y448 C356 M404 Y405 Y438 2.7.7.48,3.6.4.13 0000166,0001172,0003689,0003723,0003968,0004386,0006338,0006508,0008236,0016020,0016887,0034062,0039694,0061775,0140584,0140588,0140665,0140849 remove_due_to_license_issue D0PY27 25666181 601 SMSYTWTGALITPCAAEESKLPNSLLRHHNMVYATTSRSAGLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSAKSKFGYGAKDVRNLSSKAVNHIHSVWKDLLEDTVTPIDTTIMAKNEVFCVQRKPARLIVFPDLGVRVCEKMALYDVVSTLPQVVMGSSYGFQYSPGQRVEFLVNTWKSKKNPMGFSYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIKSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKASAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAASLRVFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVKTKLKLTPIPSGWFVAGYSGGDIYH 4tyl A 1.85 BS01 39O A 1 V1008 V1013 Y1063 N1064 I1074 V30 V35 Y85 N86 I96 3.6.1.- Kd=600uM remove_due_to_license_issue Kd=600000nM Q6PL18 25314628 1203 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4tyo A 1.75 BS01 39X A 1 H59 L61 K63 C113 S115 L122 Q131 F134 S154 H157 H9 L11 K13 C63 S65 L72 Q81 F84 S104 H107 H59 C113 Q131 S154 H157 H9 C63 Q81 S104 H107 5.2.1.8 0003755 Ki=0.08uM remove_due_to_license_issue Q13526 25091930 201 EPARVRCSHLLVKHSQSRRPSSWRQEQITRTQEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 4tyt A 1.799 BS03 S3C A 1 W89 H118 D120 H179 C198 N210 H240 W50 H79 D81 H140 C159 N171 H201 H116 H118 D120 H179 C198 K201 N210 H240 H77 H79 D81 H140 C159 K162 N171 H201 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.02uM remove_due_to_license_issue IC50=80nM P04190 25411887 303 EKTVIKNTGTISISQLNKNVWVHTELGSAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 4tz2 A 1.7 BS01 39R A 1 V1008 F1009 Y1021 M1029 I1056 N1064 I1074 V30 F31 Y43 M51 I78 N86 I96 3.6.1.- Kd=350uM remove_due_to_license_issue Q6PL18 25314628 1205 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4tz8 A 2.15 BS01 39U A 1 V1008 V1013 I1074 V30 V35 I96 3.6.1.- Kd=500uM remove_due_to_license_issue Kd=500000nM Q6PL18 25314628 1204 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 4u01 A 2.8 BS02 39W A 1 F43 H57 D79 D81 V132 K136 G137 S139 F154 R155 A156 A157 F43 H57 D79 D81 V132 K136 G137 S139 F154 R155 A156 A157 H57 D81 G137 S139 H57 D81 G137 S139 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue Q9WMX2 26410074 301 APITAYSQQTRGLLGCIITSLTGRDRNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMRAS 4u03 A 2.041 BS05 TLL A 1 R40 R108 F109 W110 T111 Q116 Y137 F204 Y238 L240 D260 K262 R38 R106 F107 W108 T109 Q114 Y135 F202 Y216 L218 D238 K240 2.7.7.- 0005524,0005525,0005575,0009117,0009190,0009405,0016779,0046872,0050922,0051607,0052621,0140701 ic50=1.69uM remove_due_to_license_issue Q9KVG7 25201413 505 MTWNFHQYYTNRNDGLMGKLVLTDEEKNNLKALRKIIRLRTRDVFEEAKGIAKAVKKSALTFEIIQEKVSTTQIKHLSDSEQREVAKLIYEMDDDARDEFLGLTPRFWTQGSFQYDTLNRPFQPGQEMDIDDGTYMPMPIFESEPKIGHSLLILLVDASLKSLVAENHGWKFEAKQTCGRIKIEAEKTHIDVPMYAIPKDEFQKKQIALEANRSFYELDSENVNLALREGDRKWINSDPKIVEDWFNDSCIRIGKHLRKVCRFMKAWRDAQWDVGGPSSISLMAATVNILDSVAHDASDLGETMKIIAKHLPSEFARGVESPDSTDEKPLFPPSYKHGPREMDIMSKLERLPEILSSAESADSKSEALKKINMAFGNRVTNSELIVLAK 4u0e A 2.043 BS01 1B0 A 1 N53 L56 N57 Q63 M66 K70 T107 Y130 N50 L53 N54 Q60 M63 K67 T102 Y125 ? 0016032 Kd=0.12uM remove_due_to_license_issue P12493 25356722 302 PIVQNQMVHQCISPRTLNAWVKVVEEKAFSPEVIPMFSALSCGATPQDLNTMLNTVGGHQAAMQMLKETINEEAAEWDRLHPVHPIAPGQMREPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYSPTSILDIRQGPKEPFRDYVDRFYKTLRAEQASQETETLLVQNANPDCKTILKALGPGATLEEMMTACQ 4u0f A 2.22 BS01 3A8 A 1 N53 L56 N57 K70 I73 N74 T107 N50 L53 N54 K67 I70 N71 T101 ? 0016032 Kd=1.2uM remove_due_to_license_issue P12493 25356722 302 PIVQNQMVHQCISPRTLNAWVKVVEEKAFSPEVIPMFSALSCGATPQDLNTMLNTVGGHQAAMQMLKETINEEAAEWDRLHPVHIAPGQMREPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYSPTSILDIRQGPKEPFRDYVDRFYKTLRAETLLVQNANPDCKTILKALGPGATLEEMMTACQ 4u0i A 2.0 BS01 0LI A 1 L595 A621 V622 K623 E640 T670 Y672 C673 I789 H790 R791 L799 C809 D810 F811 L31 A54 V55 K56 E73 T103 Y105 C106 I153 H154 R155 L163 C173 D174 F175 D792 R796 N797 D810 D156 R160 N161 D174 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50<11nM remove_due_to_license_issue IC50=1.7nM P10721 25239608 1001 GNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFICSLALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISESTN 4u0m A 2.3 BS04 TLL A 1 R36 R40 R108 F109 W110 Y137 F204 E239 L240 D260 K262 R34 R38 R106 F107 W108 Y135 F202 E215 L216 D236 K238 2.7.7.- 0005524,0005525,0005575,0009117,0009190,0009405,0016779,0046872,0050922,0051607,0052621,0140701 remove_due_to_license_issue Q9KVG7 25201413 504 MTWNFHQYYTNRNDGLMGKLVLTDEEKNNLKALRKIIRLRTRDVFEEAKGIAKAVKKSALTFEIIQEKVSTTQIKHLSDSEQREVAKLIYEMDDDARDEFLGLTPRFWTQGSFQYDTLNRPFQPGQEMDIDDGTYMPMPIFESEPKIGHSLLILLVDASLKSLVAENHGWKFEAKQTCGRIKIEAEKTHINVPMYAIPKDEFQKKQIALEANRYELDSENVNLALREGDRKWINSDPKIVEDWFNDSCIRIGKHLRKVCRFMKAWRDAQWDVGGPSSISLMAATVNILDSVAHDASDLGETMKIIAKHLPSEFARGVESPDSTDEKPLFPPSYKHGPREMDIMSKLERLPEILSSAESADSKSEALKKINMAFGNRVTNSELIVLAK 4u0n A 2.102 BS02 TLL A 1 K37 R40 R108 F109 W110 D205 D224 K226 K35 R38 R106 F107 W108 D203 D222 K224 2.7.7.- 0140701 remove_due_to_license_issue Q9KVG7 25201413 402 MTWNFHQYYTNRNDGLMGKLVLTDEEKNNLKALRKIIRLRTRDVFEEAKGIAKAVKKSALTFEIIQEKVSTTQIKHLSDSEQREVAKLIYEMDDDARDEFLGLTPRFWTQGSFQYDTLNRPFQPGQEMDIDDGTYMPMPIFESEPKIGHSLLILLVDASLKSLVAENHGWKFEAKQTCGRIKIEAEKTHIDVPMYAIPKDELDSENVNLALREGDRKWINSDPKIVEDWFNDSCIRIGKHLRKVCRFMKAWRDAQWDVGGPSSISLMAATVNILDSVAHDASDLGETMKIIAKHLPSEFARGVESPDSTDEKPLFPPSYKHGPREMDIMSKLERLPEILSSAESADSKSEALKKINMAFGNRVTNSELIVLAK 4u0s A 2.49 BS01 ADP A 1 H319 V360 H363 D367 G368 N369 G370 R371 Y399 Y400 N407 H209 V250 H253 D257 G258 N259 G260 R261 Y289 Y290 N297 2.7.7.108,3.1.4.- Kd=0.158uM remove_due_to_license_issue Q9BVA6 25435325 501 AALNQALEMKRQGKREKAQKLFMHALKMDPDFVDALTEFGIFSEEDKDIIQADYLYTRALTISPYHEKALVNRDRTLPLVEEIDQRYFSIIDSKVKKVMSINSALRRVMEETYYHHIYHTVAIGGNTLTLSEIRHILETRYAVPGKSLEEQNEVIGMHAAMKYINTTLVSRIGSVTISDVLEIHRRVLGYVDPVEAGRFRTTQVLVGHHIPPHPQDVEKQMQEFVQWLNSEEAMNLHPVEFAALAHYKLVYIHPFIDGNGRTSRLLMNLILMQAGYPPITIRKEQRSDYYHVLEAANEGDVRPFIRFIAKCTETTLDTLLFAT 4u0u A 2.98 BS01 ADP A 1 E234 V316 V360 D367 G368 N369 G370 R371 Y400 N407 E127 V209 V253 D260 G261 N262 G263 R264 Y293 N300 2.7.7.108,3.1.4.- remove_due_to_license_issue Q9BVA6 25435325 503 AALNQALEMKRQGKREKAQKLFMHALKMDPDFVDALTEFGIFSEEDKDIIQADYLYTRALTISPYHEKALVNRDRTLPLVEEIDQRYFSIIDSKVKKVMSIPKGNSALRRVMEETYYHHIYHTVAIEGNTLTLSEIRHILETRYAVPGKSLEEQNEVIGMHAAMKYINTTLVSRIGSVTISDVLEIHRRVLGYVDPVEAGRFRTTQVLVGHHIPPHPQDVEKQMQEFVQWLNSEEAMNLHPVEFAALAHYKLVYIHPFIDGNGRTSRLLMNLILMQAGYPPITIRKEQRSDYYHVLEAANEGDVRPFIRFIAKCTETTLDTLLFATTEYSVALP 4u0w A 2.001 BS01 16G A 1 S88 F89 T90 R133 R135 E145 S165 I166 Y167 Q183 I209 R211 E222 Y228 S89 F90 T91 R134 R136 E146 S166 I167 Y168 Q184 I210 R212 E223 Y229 ? 0003677,0003700,0006355,0045892 Kd=1mM remove_due_to_license_issue O34817 25564531 301 HMNINKQSPIPIYYQIMEQLKTQIKNGELQPDMPLPSEREYAEQFGISRMTVRQALSNLVNEGLLYRLKGRGTFVSKPKMEQALQGLTSFTEDMKSRGMTPGSRLIDYQLIDSTEELAAILGCGHPSSIHKITRVRLANDIPMAIESSHIPFELAGELNESHFQSSIYDHIERYNSIPISRAKQELEPSAATTEEANILGIQKGAPVLLIKRTTYLQNGTAFEHAKSVYRGDRYTFVHYMDRL 4u0w B 2.001 BS01 16G B 1 S88 F89 T90 R133 R135 E145 S165 I166 Y167 I209 R211 E222 Y228 S89 F90 T91 R134 R136 E146 S166 I167 Y168 I210 R212 E223 Y229 ? 0003677,0003700,0006355,0045892 Kd=1mM remove_due_to_license_issue O34817 25564531 301 HMNINKQSPIPIYYQIMEQLKTQIKNGELQPDMPLPSEREYAEQFGISRMTVRQALSNLVNEGLLYRLKGRGTFVSKPKMEQALQGLTSFTEDMKSRGMTPGSRLIDYQLIDSTEELAAILGCGHPSSIHKITRVRLANDIPMAIESSHIPFELAGELNESHFQSSIYDHIERYNSIPISRAKQELEPSAATTEEANILGIQKGAPVLLIKRTTYLQNGTAFEHAKSVYRGDRYTFVHYMDRL 4u0x B 2.03 BS01 ZXM B 1 S64 Y150 G314 S315 T316 R340 S64 Y150 G314 S315 T316 R340 S64 K67 Y150 E272 K312 S315 S64 K67 Y150 E272 K312 S315 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 25380506 401 NTPKDQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 4u1b A 1.89 BS03 Q08 A 1 F198 C203 H212 D229 D240 H303 H310 E336 E367 F109 C114 H123 D140 D151 H214 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=4.9uM remove_due_to_license_issue Ki=4900nM P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u2y A 2.483 BS01 RZM A 1 K264 S279 W281 Q324 Y357 D359 R392 D394 N395 E423 D480 K534 Y535 K250 S265 W267 Q310 Y343 D345 R378 D380 N381 E409 D466 K520 Y521 2.4.99.16 0004553,0004556,0005975,0009313,0016757,0016758,0030979 remove_due_to_license_issue Q9L1K2 26245983 701 PTVVGRIPVLDVRPVVQRGRRPAKAVTGESFEVSATVFREGHDAVGANVVLRDPRGRPGPWTPMRELAPGTDRWGATVTAGETGTWSYTVEAWGDPVTTWRHHARIKIPAGLDTDLVLEEGARLYERAAADVPGREDRRELLAAVDALRDESRPAASRLAAALTPQVDAVLARHPLRDLVTSSDPLPLLVERERALYGAWYEFFPRSEGTPHTPHGTFRTAARRLPAIAAMGFDVVYLPPIHPIGTTHRKGRNNTLSATGDDVGSPWAIGSPEGGHDSIHPALGTLDDFDHFVTEAGKLGLEIALDFALQCSPDHPWVHKHPEWFHHRPDGTIAHAENPPKKYQDIYPIAFDADPDGLATETVRILRHWMDHGVRIFRVDNPHTKPVAFWERVIADINGTDPDVIFLAEAFTRPAMMATLAQIGFQQSYTYFTWRNTKQELTEYLTELSGEAASYMRPNFFANTPDILHAYLQHGGRPAFEVRAVLAATLSPTWGIYSGYELCENTPLREGSEEYLDSEKYQLKPRDWTRAAREGTTIAPLVTRLNTIRRENPALRQLRDLHFHPTDKEEVIAYSKRQGSNTVLVVVNLDPRHTQEATVSLDMPQLGLDWHESVPVRDELTGETYHWGRANYVRLEPGRTPAHVCTVLR 4u3f C 3.2312 BS03 Y52 C 1 M125 A126 F129 Y132 G143 A144 I147 K270 P271 E272 Y274 F275 M125 A126 F129 Y132 G143 A144 I147 K270 P271 E272 Y274 F275 H202 S206 K228 D229 E272 H202 S206 K228 D229 E272 ? 0005737,0005739,0005743,0006122,0006979,0008121,0009055,0016020,0016491,0020037,0022904,0045275,0046872,1902600 remove_due_to_license_issue P18946 503 MAPNIRKSHPLLKMINNSLIDLPAPSNISAWWNFGSLLAVCLMTQILTGLLLAMHYTADTSLAFSSVAHTCRNVQYGWLIRNLHANGASFFFICIFLHIGRGLYYGSYLYKETWNTGVILLLTLMATAFVGYVLPWGQMSFWGATVITNLFSAIPYIGHTLVEWAWGGFSVDNPTLTRFFALHFLLPFAIAGITIIHLTFLHESGSNNPLGISSDSDKIPFHPYYSFKDILGLTLMLTPFLTLALFSPNLLGDPENFTPANPLVTPPHIKPEWYFLFAYAILRSIPNKLGGVLALAASVLILFLIPFLHKSKQRTMTFRPLSQTLFWLLVANLLILTWIGSQPVEHPFIIIGQMASLSYFTILLILFPTIGTLENKMLNY 4u43 A 2.18 BS01 3D8 A 1 V31 V39 A52 C108 L160 V170 D171 V18 V26 A39 C95 L147 V157 D158 D153 K155 Q157 N158 D171 T191 D140 K142 Q144 N145 D158 T167 2.7.11.1 0004672,0005524,0006468 Kd=48uM remove_due_to_license_issue Kd=48000nM O95819 25139565 401 DLSSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEDEEEEIKLEINMLKKYSHHRNIATYYGAFIKKSPPGHDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVNTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTRK 4u44 A 2.43 BS01 3D9 A 1 V31 V39 A52 K54 M105 C108 G111 L160 D171 V20 V28 A41 K43 M91 C94 G97 L146 D157 D153 K155 Q157 N158 D171 T191 D139 K141 Q143 N144 D157 T167 2.7.11.1 0004672,0005524,0006468 ic50=0.008uM remove_due_to_license_issue IC50=8.0nM O95819 25139565 403 DIDLSSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEDEEEEIKLEINMLKKYSHHRNIATYYGAFIKKSHDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVSATFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTR 4u45 A 2.58 BS03 3DC A 1 V31 V39 A52 M105 C108 G111 L160 V170 D171 V20 V28 A41 M92 C95 G98 L147 V157 D158 D153 K155 Q157 N158 D171 T191 D140 K142 Q144 N145 D158 T169 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O95819 25139565 403 DIDLSSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEDEEEEIKLEINMLKKYSHHRNIATYYGAFIKKSPPDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVSANTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTRK 4u4s A 1.9 BS01 3C1 A 1 P494 S729 K730 G731 P102 S214 K215 G216 ? 0015276,0016020 Kd=1200uM remove_due_to_license_issue P19491 25375781 801 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDEC 4u4s A 1.9 BS03 3C1 B 1 P494 F495 M496 P102 F103 M104 ? 0015276,0016020 Kd=1200uM remove_due_to_license_issue P19491 25375781 801 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDEC 4u4s B 1.9 BS01 3C1 A 1 P494 F495 M496 L751 P105 F106 M107 L239 ? 0015276,0016020 Kd=1200uM remove_due_to_license_issue P19491 25375781 801 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 4u4s B 1.9 BS02 3C1 B 1 P494 S729 K730 G731 P105 S217 K218 G219 ? 0015276,0016020 Kd=1200uM remove_due_to_license_issue P19491 25375781 801 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 4u4x A 1.56 BS01 3C2 A 1 P494 S497 S729 K730 G731 P105 S108 S217 K218 G219 ? 0015276,0016020 Kd=9.8uM remove_due_to_license_issue P19491 25375781 801 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 4u4x A 1.56 BS03 3C2 B 1 P494 F495 M496 S497 P105 F106 M107 S108 ? 0015276,0016020 Kd=9.8uM remove_due_to_license_issue P19491 25375781 801 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 4u4x B 1.56 BS01 3C2 A 1 P494 F495 M496 S497 P102 F103 M104 S105 ? 0015276,0016020 Kd=9.8uM remove_due_to_license_issue P19491 25375781 801 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECG 4u4x B 1.56 BS02 3C2 B 1 P494 S497 S729 K730 G731 P102 S105 S214 K215 G216 ? 0015276,0016020 Kd=9.8uM remove_due_to_license_issue P19491 25375781 801 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECG 4u54 A 2.41 BS01 3C5 A 1 N361 E396 W399 N403 N288 E323 W326 N330 ? Kd=8.7mM remove_due_to_license_issue P52293 25899172 501 VNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFSV 4u58 A 2.56 BS01 3C6 A 1 N361 A364 E396 W399 N403 N290 A293 E325 W328 N332 ? remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5j A 2.26 BS01 RXT A 1 G276 V281 M341 A390 N391 L393 D404 G18 V23 M83 A132 N133 L135 D146 D386 R388 A390 N391 D404 F424 D128 R130 A132 N133 D146 F158 2.7.10.2 0004672,0004713,0005524,0006468 ic50=2.92uM remove_due_to_license_issue P00523 25197973 601 AWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4u5l A 2.53 BS01 3D6 A 1 V321 T322 G323 N361 A364 E396 W399 N403 V250 T251 G252 N290 A293 E325 W328 N332 ? remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5n A 2.31 BS01 3D4 A 1 V321 G323 K353 E354 W357 S360 N361 E396 W399 N403 V250 G252 K282 E283 W286 S289 N290 E325 W328 N332 ? Kd=3.3mM remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5o A 2.0 BS01 3D5 A 1 V321 S360 N361 E396 W399 N403 V250 S289 N290 E325 W328 N332 ? Kd=3.8mM remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5s A 2.12 BS01 3D0 A 1 D280 G281 N319 V321 T322 W357 N361 E396 W399 N403 D209 G210 N248 V250 T251 W286 N290 E325 W328 N332 ? Kd=3.9mM remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5s A 2.12 BS02 3D0 A 2 W142 N146 S149 G150 T155 Q181 W184 N188 D192 N228 W231 N235 W71 N75 S78 G79 T84 Q110 W113 N117 D121 N157 W160 N164 ? Kd=3.9mM remove_due_to_license_issue P52293 25899172 502 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5t A 3.301 BS01 3CG A 1 R20 R27 R19 R26 ? 0003700,0006355,0006357 remove_due_to_license_issue Q10587 22851716 101 DPDLEIRAAFLEKENTALRTEVAELRKEVGRCKNIVS 4u5u A 1.96 BS01 3D2 A 1 N361 A364 E396 W399 N403 N290 A293 E325 W328 N332 ? Kd=1.3mM remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5u A 1.96 BS02 3D2 A 2 W357 E396 W286 E325 ? Kd=1.3mM remove_due_to_license_issue P52293 25899172 502 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5v A 1.968 BS01 RH2 A 1 N361 E396 W399 N403 N290 E325 W328 N332 ? Kd=0.9mM remove_due_to_license_issue P52293 25899172 501 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u5v A 1.968 BS02 RH2 A 2 E354 E396 E283 E325 ? Kd=0.9mM remove_due_to_license_issue P52293 25899172 502 GTVNWSVEDIVKGINSNNLESQLQATQAARKLLSREKQPPIDNIIRAGLIPKFVSFLGKTDCSPIQFESAWALTNIASGTSEQTKAVVDGGAIPAFISLLASPHAHISEQAVWALGNIAGDGSAFRDLVIKHGAIDPLLALLAVPDLSTLACGYLRNLTWTLSNLCRNKNPAPPLDAVEQILPTLVRLLHHNDPEVLADSCWAISYLTDGPNERIEMVVKKGVVPQLVKLLGATELPIVTPALRAIGNIVTGTDEQTQKVIDAGALAVFPSLLTNPKTNIQKEATWTMSNITAGRQDQIQQVVNHGLVPFLVGVLSKADFKTQKEAAWAITNYTSGGTVEQIVYLVHCGIIEPLMNLLSAKDTKIIQVILDAISNIFQAAEKLGETEKLSIMIEECGGLDKIEALQRHENESVYKASLNLIEKYFS 4u69 A 1.6 BS03 Q07 A 1 H212 D229 D240 H303 F309 H310 E336 E367 H123 D140 D151 H214 F220 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=54.8uM remove_due_to_license_issue Ki=54800nM P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u6c A 1.91 BS03 Q06 A 1 F198 C203 H212 D229 D240 H303 F309 H310 E336 W353 E367 F109 C114 H123 D140 D151 H214 F220 H221 E247 W264 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=9.9uM remove_due_to_license_issue P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u6e A 1.9 BS03 Q02 A 1 P192 C203 H212 D229 D240 F309 H310 E336 E367 P103 C114 H123 D140 D151 F220 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=111.6uM remove_due_to_license_issue Ki=111600nM P53582 25699713 403 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u6r A 2.5 BS01 3E4 A 1 V586 A597 K599 E612 L616 I642 C645 E651 D711 F712 V26 A37 K39 E52 L56 I82 C85 E91 D151 F152 D688 K690 N693 D711 T734 D128 K130 N133 D151 T174 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue IC50=14nM O75460 25589933 1001 TSVVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCKKLAVGRHSFSRRSGVPGTEGWIAPEMLSEDCKENPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPAEVRETLGTLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFH 4u6w A 1.83 BS03 Q08 A 1 S191 P192 H212 D229 T231 D240 H303 M309 H310 E336 W353 E367 S102 P103 H123 D140 T142 D151 H214 M220 H221 E247 W264 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 remove_due_to_license_issue Ki=4900nM P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u6z A 1.8 BS03 Q07 A 1 F198 C203 H212 D229 D240 H310 E336 W353 E367 F109 C114 H123 D140 D151 H221 E247 W264 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=3.9uM remove_due_to_license_issue Ki=54800nM P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u70 A 1.6 BS03 Q04 A 1 P192 Y195 F198 C203 H212 D229 D240 H303 H310 E336 E367 P103 Y106 F109 C114 H123 D140 D151 H214 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=9.5uM remove_due_to_license_issue Ki=>500000nM P53582 25699713 403 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u71 A 1.8 BS03 Q03 A 1 P192 Y195 C203 H212 D229 D240 M309 H310 E336 E367 P103 Y106 C114 H123 D140 D151 M220 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=6uM remove_due_to_license_issue Ki=>500000nM P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u73 A 1.8 BS03 Q02 A 1 P192 H212 D229 D240 H303 H310 E336 E367 P103 H123 D140 D151 H214 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 Ki=6.6uM remove_due_to_license_issue Ki=111600nM P53582 25699713 404 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 4u79 A 2.23 BS01 3EL A 1 V78 K93 R107 E111 I124 L144 M146 M149 Q155 D207 V33 K48 R62 E66 I79 L99 M101 M104 Q110 D162 D189 K191 N194 D207 T226 D144 K146 N149 D162 T170 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 25589933 501 VDNQFYSVEVGDSTFTVLKRYQNLKPIGSGGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPLDEREHTIEEWKELIYKEVMN 4u7o A 2.395 BS01 AN2 A 1 N514 Y518 I547 V555 F560 R561 V562 G572 G574 G576 L577 F603 N143 Y147 I176 V184 F189 R190 V191 G196 G198 G200 L201 F227 2.7.13.3 0000155,0000160,0000166,0004721,0005886,0007165,0016020,0016036,0016301,0016310,0016772 remove_due_to_license_issue A0A0M3KKX3 28994408 701 VTEQQKIDNDRKQFVSNVSHELRTPLTSLRSYIEALSDGAWKDPEVAPGFLKVTQEETDRMIRMINELLSLSRMDSGTTRVDMELVNINEMFNYVLDRFDMILKKDDNPAKYYTIKREFTKRDLWVEIDTDKFTQVLDNIMNNAIKYSPDGGVVTCRLLETHNQVIISISDQGLGIPRADLGHVFDRFFRVDKQGGTGLGLAISKEVVQMLGGRIWVDSVEGKGSTFYISLPYE 4u7q A 1.7 BS01 3EM B 1 R8 D25 D30 G48 I50 T80 P81 I84 R8 D25 D30 G48 I50 T80 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 25751579 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4u7q B 1.7 BS01 3EM B 1 D25 G27 D29 D30 G49 I50 V82 I84 D25 G27 D29 D30 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=180pM remove_due_to_license_issue P04585 25751579 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4u7v A 1.38 BS01 3EN B 1 D25 G48 G49 I50 P81 V82 I84 D25 G48 G49 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 25751579 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4u7v B 1.38 BS01 3EN B 1 D25 G27 A28 G48 G49 I50 D25 G27 A28 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.2uM remove_due_to_license_issue P04585 25751579 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 4u82 A 1.66 BS01 FPS A 1 M32 D33 G34 N35 G36 R37 R46 H50 A76 R84 F99 F148 M14 D15 G16 N17 G18 R19 R28 H32 A58 R66 F81 F130 D33 H50 L144 D15 H32 L126 2.5.1.- 0000287,0004659,0005829,0008834,0016094,0016740,0016765,0030145,0045547,0046872 ic50=1.9uM remove_due_to_license_issue P60477 25574764 302 LDSSNIPEHIAIIMDGNGRWAKKRKMPRIKGHYEGMQTIKKITRIASDIGVKYLTLYAFSTENWSRPESEVNYIMNLPVNFLKTFLPELIEKNVKVETIGFTDKLPKSTIEAINNAKEKTANNTGLKLIFAINYGGRAELVHSIKNMFDELHQQGLNSDIIDETYINNHLMTKDYPDPELLIRTSGEQRISNFLIWQVSYSEFIFNQKLWPDFDEDELIKCIKIYQSRQRRFGGLS 4u8t A 2.7 BS01 rna O 0 K184 S185 S186 H190 W200 S201 Y205 R209 N230 A231 W254 R259 Y260 N276 T293 N294 R296 D297 K20 S21 S22 H26 W36 S37 Y41 R45 N66 A67 W90 R93 Y94 N110 T127 N128 R130 D131 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGSRYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLDDD 4u8t A 2.7 BS02 rna R 0 F204 Y205 F40 Y41 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGSRYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLDDD 4u8t B 2.7 BS01 rna P 0 K184 S185 S186 H190 W200 S201 T203 Y205 R209 N230 A231 W254 Y260 N276 T293 N294 S295 R296 D297 K20 S21 S22 H26 W36 S37 T39 Y41 R45 N66 A67 W90 Y92 N108 T125 N126 S127 R128 D129 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLDD 4u8t B 2.7 BS02 rna Q 0 F204 Y205 F40 Y41 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLDD 4u8t C 2.7 BS01 rna P 0 F204 Y205 F40 Y41 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGSRYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t C 2.7 BS02 rna Q 0 K184 S185 S186 H190 W200 S201 T203 Y205 R209 N230 A231 W254 R259 Y260 N276 T293 N294 R296 D297 K20 S21 S22 H26 W36 S37 T39 Y41 R45 N66 A67 W90 R93 Y94 N110 T127 N128 R130 D131 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGSRYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t C 2.7 BS03 rna R 0 R209 R296 R45 R130 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGSRYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t D 2.7 BS01 rna O 0 R209 R296 R45 R128 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYEQSEVQSFLD 4u8t D 2.7 BS02 rna S 0 F204 Y205 F40 Y41 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYEQSEVQSFLD 4u8t D 2.7 BS03 rna T 0 K184 S185 S186 H190 W200 S201 Y205 R209 N230 A231 W254 Y260 N276 T293 N294 S295 R296 D297 K20 S21 S22 H26 W36 S37 Y41 R45 N66 A67 W90 Y92 N108 T125 N126 S127 R128 D129 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYEQSEVQSFLD 4u8t E 2.7 BS01 rna P 0 R209 R296 R45 R128 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t E 2.7 BS02 rna S 0 K184 S186 H190 W200 S201 Y205 R209 N230 A231 W254 Y260 N276 T293 N294 S295 R296 D297 K20 S22 H26 W36 S37 Y41 R45 N66 A67 W90 Y92 N108 T125 N126 S127 R128 D129 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t E 2.7 BS03 rna T 0 F204 Y205 F40 Y41 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t F 2.7 BS01 rna O 0 F204 Y205 F40 Y41 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t F 2.7 BS02 rna Q 0 R209 R296 R45 R128 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8t F 2.7 BS03 rna R 0 K184 S185 S186 H190 W200 S201 Y205 R209 N230 A231 W254 Y260 N276 T293 N294 S295 R296 D297 K20 S21 S22 H26 W36 S37 Y41 R45 N66 A67 W90 Y92 N108 T125 N126 S127 R128 D129 ? 0003723 remove_due_to_license_issue C5E1V0 25201973 -3 ~ 3 GAIIPPWIHVPDHSRFFVIKSSSLEHVKKSFYNGIWSSTFYGNKRLSEAYESLPQGAKIYLLFSVNASGRFCGVAEMSSNLREDLDTSIWGYRHAFKVRWIVVRDVHNRSLKQFLIPANDMKPVTNSRDTQEIPATISKSILKLFKYVQSFLD 4u8w A 1.3 BS01 G10 A 1 D25 G27 A28 D30 G48 G49 V82 I84 D25 G27 A28 D30 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.0058nM remove_due_to_license_issue P03366 25336073 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4u8w B 1.3 BS01 G10 A 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 25336073 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4u93 A 1.55 BS01 990 A 1 A55 M98 L107 F138 V150 A39 M82 L91 F122 V134 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.013uM remove_due_to_license_issue IC50=13nM P07900 25368984 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4ual A 1.71 BS01 3FV A 1 R84 A103 K105 M153 D154 Y155 Y156 D204 L207 D218 R86 A105 K107 M155 D156 Y157 Y158 D206 L209 D220 D200 K202 N205 D218 T239 D202 K204 N207 D220 T238 2.7.11.1 0004672,0004674,0005524,0006468 Ki=4nM remove_due_to_license_issue Q9Y5S2 25288205 501 GGSSAKVRLKKLEQLLLDGPWRNESALSVETLLDVLVCLYTECSHSALRRDKYVAEFLEWAKPFTQLVKEMQLHREDFEIIKVIGRGAFGEVAVVKMKNTERIYAMKILNKWEMLKRAETACFREERDVLVNGDCQWITALHYAFQDENHLYLVMDYYVGGDLLTLLSKFEDKLPEDMARFYIGEMVLAIDSIHQLHYVHRDIKPDNVLLDVNGHIRLADFGSCLKMNDDGTVVAVGTPDYISPEILQAMEDGKYGPECDWWSLGVCMYEMLYGETPFYAESLVETYGKIMNHEERFQFPSHVTDVSEEAKDLIQRLICSRERRLGQNGIEDFKKHAFFEGLNWENIRNLEAPYIPDVSSPSDTSNFDVILPPHTGFSGLHLPFIGFTFTTESCFSDRGSLKS 4uat A 1.3 BS01 XBP A 1 D8 V9 N10 E17 H20 T49 G50 G51 R54 H75 K78 T115 T116 T117 S118 D8 V9 N10 E17 H20 T49 G50 G51 R54 H75 K78 T115 T116 T117 S118 D8 V9 N10 T16 T47 T115 T116 K151 E175 D176 D8 V9 N10 T16 T47 T115 T116 K151 E175 D176 3.1.3.- 0000287,0005998,0016787,0046872 remove_due_to_license_issue P95649 27246049 301 MIEAILFDVNGTLAETEELHRRAFNETFAALGVDWFWDREEYRELLTTTGGKERIARFLRHQKGDPAPLPIADIHRAKTERFVALMAEGEIALRPGIADLIAEAKRAGIRLAVATTTSLPNVEALCRACFGHPAREIFDVIAAGDMVAEKKPSPDIYRLALRELDVPPERAVALEDSLNGLRAAKGAGLRCIVSPGFYTRHEEFAGADRLLDSFAELGGLAGLDL 4uau A 1.45 BS01 XBP A 1 D8 V9 N10 E17 H20 T49 G50 G51 R54 H75 K78 T115 T116 T117 S118 D8 V9 N10 E17 H20 T49 G50 G51 R54 H75 K78 T115 T116 T117 S118 D8 V9 N10 T16 T47 T115 T116 K151 E175 D176 D8 V9 N10 T16 T47 T115 T116 K151 E175 D176 3.1.3.- 0000287,0005998,0016787,0046872 remove_due_to_license_issue P95649 27246049 301 MIEAILFDVNGTLAETEELHRRAFNETFAALGVDWFWDREEYRELLTTTGGKERIARFLRHQKGDPAPLPIADIHRAKTERFVALMAEGEIALRPGIADLIAEAKRAGIRLAVATTTSLPNVEALCRACFGHPAREIFDVIAAGDMVAEKKPSPDIYRLALRELDVPPERAVALEDSLNGLRAAKGAGLRCIVSPGFYTRHEEFAGADRLLDSFAELGGLAGLDLT 4uc5 A 2.19 BS02 PHE A 1 Q153 A156 L181 S182 F211 S213 Q150 A153 L178 S179 F208 S210 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 remove_due_to_license_issue Q9K169 26794122 1354 HYPTDDIKIKEVKELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMAR 4uc5 B 2.19 BS02 PHE B 1 Q153 A156 L181 S182 S213 Q150 A153 L178 S179 S210 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 remove_due_to_license_issue Q9K169 26794122 1352 HYPTDDIKIKEVKELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMAR 4ucc A 2.05 BS01 ZKW A 1 M50 E128 S131 R132 Y135 R150 H151 M20 E98 S101 R102 Y105 R120 H121 ? 0003723,0019013 Kd=48uM remove_due_to_license_issue P03418 26246564 301 DSIDTPNYDVQKHINKLCGMLLITEDANHKFTGLIGMLYAMSRLGREDTIKILRDAGYHVKANGVDVTTHRQDINGKEMKFEVLTLASLTTEIQINIEIESRKSYKKMLKEMGEVAPEYRHDSPDCGMIILCIAALVITKLAAGDRSGLTAVIRRANNVLKNEMKRYKGLLPKDIANSFYEVFEKHPHFIDVFVHFGIAQSSTRGGSRVEGIFAGLFMNAYGL 4ucd A 2.66 BS01 M81 A 1 S131 R132 Y135 R150 H151 S100 R101 Y104 R119 H120 ? 0003723,0019013 remove_due_to_license_issue P03418 26246564 1301 SIDTPNYDVQKHINKLCGMLLITEDANHKFTGLIGMLYAMSRLGREDTIKILRDAGYHVKANGVDVTTHRQDINGKEMKFEVLTLASLTTEIQINIEIESRKSYKKMLKEMGEVAPEYRHDSPDCGMIILCIAALVITKLAAGRSGLTAVIRRANNVLKNEMKRYKGLLPKDIANSFYEVFEKHPHFIDVFVHFGIAQSSTGGSRVEGIFAGLFMNAYGL 4uce A 2.95 BS01 MZS A 1 S131 R132 Y135 R150 H151 S100 R101 Y104 R119 H120 ? 0003723,0019013 remove_due_to_license_issue P03418 26246564 301 SIDTPNYDVQKHINKLCGMLLITEDANHKFTGLIGMLYAMSRLGREDTIKILRDAGYHVKANGVDVTTHRQDINGKEMKFEVLTLASLTTEIQINIEIESRKSYKKMLKEMGEVAPEYRHDSPDCGMIILCIAALVITKLARSGLTAVIRRANNVLKNEMKRYKGLLPKDIANSFYEVFEKHPHFIDVFVHFGIAQSSTRGGSRVEGIFAGLFMNAYG 4uco A 2.5 BS01 D41 A 1 L80 L82 P115 L117 R137 E174 Y226 V289 K291 L80 L82 P115 L117 R137 E174 Y226 V289 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 1318 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFP 4ucr A 2.15 BS02 JCF A 1 L82 E114 L117 E174 Y226 V289 K291 L82 E114 L117 E174 Y226 V289 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 1319 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFP 4ucs A 1.9 BS02 9MJ A 1 L82 E114 K116 L117 Y226 V289 K291 L82 E114 K116 L117 Y226 V289 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 1319 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFP 4uct A 2.1 BS02 5U1 A 1 L82 E114 Y226 V289 K291 L82 E114 Y226 V289 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 1320 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFPA 4ucu A 2.1 BS01 8HC A 1 L80 L82 E114 Y226 K291 L80 L82 E114 Y226 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 1319 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFPA 4ucv A 2.6 BS02 I6G A 1 L80 L82 E114 E174 Y226 K291 L80 L82 E114 E174 Y226 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 1320 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFPA 4uda A 2.03 BS02 DEX A 1 L769 N770 A773 Q776 M807 S810 F829 M845 F941 C942 T945 L32 N33 A36 Q39 M70 S73 F92 M108 F200 C201 T204 ? Ki=6.3nM remove_due_to_license_issue IC50=33nM, Ki=7.2nM P08235 26602186 1985 PVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLSSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHR 4udb A 2.36 BS02 CV7 A 1 L766 L769 N770 A773 Q776 M807 L810 F829 M845 M852 F941 C942 T945 L27 L30 N31 A34 Q37 M68 L71 F90 M106 M113 F202 C203 T206 ? Ki=0.18nM remove_due_to_license_issue P08235 26602186 1987 SPVMVLENIEPEIVYAGYDPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHR 4ufd H 1.429 BS03 S49 H 1 H57 Y60A W60D N98 L99 D189 A190 E192 V213 S214 W215 G216 G219 C220 H43 Y47 W50 N95 L96 D192 A193 E195 V218 S219 W220 G221 G223 C224 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 26762840 1251 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4ufe H 1.593 BS03 3ZD H 1 Y60A W60D N98 L99 I174 D189 A190 E192 S195 V213 S214 W215 G216 E217 G219 Y47 W50 N95 L96 I172 D192 A193 E195 S198 V218 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 26762840 1249 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4uff H 1.55 BS03 6V2 H 1 Y60A W60D N98 L99 D189 A190 S195 V213 S214 W215 G216 E217 G219 C220 Y47 W50 N95 L96 D192 A193 S198 V218 S219 W220 G221 E222 G223 C224 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 26762840 1248 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 4ufg H 1.65 BS03 D6J H 1 H57 Y60A W60D N98 L99 I174 D189 A190 E192 S195 V213 S214 W215 G216 E217 G219 H43 Y47 W50 N95 L96 I172 D192 A193 E195 S198 V218 S219 W220 G221 E222 G223 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 26762840 1249 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 4ufh A 2.16 BS01 GIF A 1 G48 T93 E182 E258 S261 W291 Y303 R380 G24 T69 E158 E234 S237 W267 Y279 R356 3.2.1.46 0004336,0006683 Ki=380nM remove_due_to_license_issue P54818 26029356 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGQRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4ufi A 2.4 BS01 AGK A 1 G48 T93 E182 E258 S261 W291 Y303 R380 G24 T69 E158 E234 S237 W267 Y279 R356 3.2.1.46 0004336,0006683 Ki=630nM remove_due_to_license_issue P54818 26029356 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGQRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4ufj A 2.2 BS01 IF7 A 1 G48 T93 W135 N181 E182 E258 S261 W291 Y303 R380 G24 T69 W111 N157 E158 E234 S237 W267 Y279 R356 3.2.1.46 0004336,0006683 Ki=52uM remove_due_to_license_issue P54818 26029356 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4ufk A 2.402 BS01 LDU A 1 G48 T93 W135 E258 S261 W291 Y303 R380 G24 T69 W111 E234 S237 W267 Y279 R356 3.2.1.46 0004336,0005739,0005764,0006665,0006683,0016020,0016042,0016798,0042552 Ki=130uM remove_due_to_license_issue P54818 26029356 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4ufl A 2.4 BS01 DZX A 1 G48 T93 E182 Y238 E258 S261 W291 Y303 R380 W524 G24 T69 E158 Y214 E234 S237 W267 Y279 R356 W497 3.2.1.46 0004336,0005739,0005764,0006665,0006683,0016020,0016042,0016798,0042552 Ki=2.3mM remove_due_to_license_issue P54818 26029356 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGQRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4ufm A 2.4 BS01 DGJ A 1 G48 T93 W135 N181 E182 E258 S261 W291 Y303 R380 G24 T69 W111 N157 E158 E234 S237 W267 Y279 R356 3.2.1.46 0004336,0005739,0005764,0006665,0006683,0016020,0016042,0016798,0042552 Ki=190uM remove_due_to_license_issue P54818 26029356 1001 GAYVLDDSDGLGREFDGIGAVSGGGATSRLLVNYPEPYRSEILDYLFKPNFGASLHILKVEIGGDGQTTDGTEPSHMHYELDENYFRGYEWWLMKEAKKRNPDIILMGLPWSFPGWLGKGFSWPYVNLQLTAYYVVRWILGAKHYHDLDIDYIGIWNERPFDANYIKELRKMLDYQGLQRVRIIASDNLWEPISSSLLLDQELWKVVDVIGAHYPGTYTVWNAKMSGKKLWSSEDFSTINSNVGAGCWSRILNQNYINGNMTSTIAWNLVASYYEELPYGRSGLMTAQEPWSGHYVVASPIWVSAHTTQFTQPGWYYLKTVGHLEKGGSYVALTDGLGNLTIIIETMSHQHSMCIRPYLPYYNVSHQLATFTLKGSLREIQELQVWYTKLGRLHFKQLDTLWLLDGSGSFTLELEEDEIFTLTTLTTGRKGSYPPPPSSKPFPTNYKDDFNVEYPLFSEAPNFADQTGVFEYYMNNEDREHRFTLRQVLNQRPITWAADASSTISVIGDHHWTNMTVQCDVYIETPRSGGVFIAGRVNKGGILIRSATGVFFWIFANGSYRVTADLGGWITYASGHADVTAKRWYTLTLGIKGYFAFGMLNGTILWKNVRVKYPGHGWAAIGTHTFEFAQFDNFRVEAAR 4ufu A 2.1 BS02 2ZI A 1 H1031 G1032 F1035 Y1050 Y1060 F1061 A1062 S1068 Y1071 E1138 H80 G81 F84 Y99 Y109 F110 A111 S117 Y120 E185 2.4.2.-,2.4.2.30 0003950 ic50=10nM remove_due_to_license_issue IC50=10nM Q9H2K2 27163581 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4ufy A 1.7 BS02 M3W A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 E1138 H80 G81 Y99 Y109 A111 S117 Y120 E185 2.4.2.-,2.4.2.30 0003950 ic50=7nM remove_due_to_license_issue IC50=6.7nM Q9H2K2 27163581 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4ufz A 2.33 BS01 IA7 A 1 S81 L82 A121 R137 E174 Y226 V289 K291 S81 L82 A121 R137 E174 Y226 V289 K291 E114 K116 D118 Y226 K315 E114 K116 D118 Y226 K315 6.5.1.2 0003911 remove_due_to_license_issue P43813 26463129 1318 MTNIQTQLDNLRKTLRQYEYEYHVLDNPSVPDSEYDRLFHQLKALELEHPEFLTSDSPTQRVGAKPLSGFSQIRHEIPMLSLDNAFSDAEFNAFVKRIEDRLILLPKPLTFCCEPKLDGLAVSILYVNGELTQAATRGDGTTGEDITANIRTIRNVPLQLLTDNPPARLEVRGEVFMPHAGFERLNKYALEHNEKTFANPRNAAAGSLRQLDPNITSKRPLVLNAYGIGIAEGVDLPTTHYARLQWLKSIGIPVNPEIRLCNGADEVLGFYRDIQNKRSSLGYDIDGTVLKINDIALQNELGFISKAPRWAIAYKFP 4uhg A 1.7 BS02 SZ5 A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=540nM remove_due_to_license_issue IC50=540nM Q9H2K2 27163581 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4ui3 A 2.0 BS02 06R A 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 I1075 H80 G81 Y99 Y109 A111 K116 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=133nM remove_due_to_license_issue IC50=133nM Q9H2K2 27163581 2115 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4ui4 B 2.4 BS02 RJN B 1 H1031 G1032 Y1050 Y1060 A1062 K1067 S1068 Y1071 H80 G81 Y99 Y109 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=45nM remove_due_to_license_issue IC50=45nM Q9H2K2 27163581 2117 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4ui5 B 1.65 BS02 BJ4 B 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=167nM remove_due_to_license_issue IC50=167nM Q9H2K2 27163581 2116 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4ui6 B 1.8 BS01 ECZ B 1 H1031 G1032 S1033 F1035 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 S82 F84 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=87nM remove_due_to_license_issue IC50=87nM Q9H2K2 27163581 2114 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4ui7 A 1.8 BS02 VT3 A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=44nM remove_due_to_license_issue IC50=44nM Q9H2K2 27163581 2116 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 4ui8 B 2.05 BS02 IY5 B 1 H1031 G1032 P1034 F1035 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 P83 F84 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=25nM remove_due_to_license_issue Q9H2K2 27163581 2116 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 4uia A 2.18 BS03 FH9 A 1 H69 R127 N144 R145 Y198 Y248 D255 F279 H64 R122 N139 R140 Y194 Y244 D251 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=0.19uM remove_due_to_license_issue P09955 25990761 1313 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGIHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLSIHSYSQHIVYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTLYLAPGGGDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHLY 4uib A 1.94 BS03 GWX A 1 H69 R127 N144 R145 T164 Y198 S207 Y248 D255 E270 F279 H64 R122 N139 R140 T159 Y194 S203 Y244 D251 E266 F275 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 ic50=0.001uM remove_due_to_license_issue P09955 25990761 1318 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGIHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLSIHSYSQHIVYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTLYLAPGGGDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHLY 4uil H 2.853 BS01 QI9 H 1 W33 S59 E99 S106 F109 W33 S59 E99 S106 F109 remove_due_to_license_issue 26282540 1223 AVQLQESGTVLARPGASVKMSCKASGYTFTSYWMHWVKQRPGQGLEWIGAIYPGNSDTSYNQKFKGKAKLTAVTSTSTAYMELSSLTNEDSAVYYCTRERGLYYGSSSFDYWGQGTTLTVSSAETTPPSVYPLAPGTSSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSQTVTCNVAHPASSTKVDKKIVPR 4uil L 2.853 BS01 QI9 H 1 G91 N92 T93 L94 P96 G91 N92 T93 L94 P96 remove_due_to_license_issue 26282540 1223 DIVMTQTTSSLSASLGDRVTISCRASQDISNYLSWYQQKPDGTVKVLIYYTSKLHSGVPSRFSGSGSGTDYSLTISNLEQEDIATYFCQQGNTLPPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 4uin H 2.5 BS01 QI9 H 1 W33 T50 E99 G106 R107 F109 W33 T50 E99 G106 R107 F109 Kd=24nM remove_due_to_license_issue 26282540 1226 EVQLQQSGTVLARPGASVKMSCEASGYTFTSYWMHWLKKRPGQGLEWIGTIYPGNSDSSYNQRFKGKAKLTAVTSTSTAYMELSSLTNEDSAVYYCTRERGLYYGGRSFDYWGQGTTLTVSSAKTTPPSVYPLAPGSNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLESDLYTLSSSVTVPSSPRPSETVTCNVAHPASSTKVDKKIVPRDCG 4uin L 2.5 BS01 QI9 H 1 G91 L94 G91 L94 remove_due_to_license_issue 26282540 1226 DIQMTQTTSSLSASLGDRVTISCRASQDISNYLTWYQQKPDGTVKLLIYYTSKLHSGVPSRFSGSGSGTDYSLTISNLEQEDVANYFCQQGNSLPPTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 4uit A 1.3 BS01 N1D A 1 F44 V49 I53 A54 Y99 N100 R101 Y106 F23 V28 I32 A33 Y78 N79 R80 Y85 ? ic50=0.00000001M remove_due_to_license_issue Q9H8M2 25856009 1123 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 4uiu A 1.64 BS01 TVU A 1 F44 F45 V49 I53 Y99 N100 R101 T104 Y106 F23 F24 V28 I32 Y78 N79 R80 T83 Y85 ? ic50=0.00000001M remove_due_to_license_issue Q9H8M2 25856009 1123 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 4uiv A 1.72 BS01 XZB A 1 F44 F45 V49 I53 A54 Y99 N100 R101 Y106 F23 F24 V28 I32 A33 Y78 N79 R80 Y85 ? ic50=0.00000001M remove_due_to_license_issue Q9H8M2 25856009 1124 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 4uiw A 1.73 BS01 H1B A 1 F44 F45 V49 I53 Y99 N100 R101 Y106 F23 F24 V28 I32 Y78 N79 R80 Y85 ? ic50=0.00000001M remove_due_to_license_issue Q9H8M2 25856009 1124 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 4uix A 1.58 BS01 TVU A 1 W81 P82 F83 L92 L94 N140 K141 D144 W39 P40 F41 L50 L52 N98 K99 D102 ? ic50=0.00000001M remove_due_to_license_issue O60885 25856009 1171 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHKFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4uiy A 1.3 BS01 5V2 A 1 W81 P82 V87 L92 N140 K141 D144 I146 W40 P41 V46 L51 N99 K100 D103 I105 ? ic50=0.00000001M remove_due_to_license_issue O60885 25856009 1172 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4uiz A 1.19 BS01 N1D A 1 W81 P82 L92 L94 Y139 N140 W40 P41 L51 L53 Y98 N99 ? ic50=0.00001995M remove_due_to_license_issue O60885 25856009 1171 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4uj1 A 1.768 BS02 NVX A 1 G50 G55 R56 V57 A70 K72 E121 Y122 E170 L173 T183 D184 G37 G42 R43 V44 A57 K59 E108 Y109 E157 L160 T170 D171 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 26578105 1351 SVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4uj2 A 2.019 BS02 NVV A 1 G50 T51 G52 G55 V57 A70 K72 E121 E170 L173 T183 D184 F327 G37 T38 G39 G42 V44 A57 K59 E108 E157 L160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 26578105 1351 SVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4uj9 A 1.87 BS02 S3N A 1 G50 T51 G52 F54 G55 R56 V57 A70 K72 L74 M120 E121 Y122 E170 N171 L173 T183 D184 F327 G41 T42 G43 F45 G46 R47 V48 A61 K63 L65 M111 E112 Y113 E161 N162 L164 T174 D175 F318 D166 K168 E170 N171 D184 T201 D157 K159 E161 N162 D175 T192 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 26578105 1351 SEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4uja A 1.93 BS02 4L7 A 1 G50 T51 G52 G55 R56 V57 A70 K72 E121 Y122 E170 L173 T183 D184 G38 T39 G40 G43 R44 V45 A58 K60 E109 Y110 E158 L161 T171 D172 D166 K168 E170 N171 D184 T201 D154 K156 E158 N159 D172 T189 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 26578105 1351 ESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4ujb A 1.949 BS02 8BQ A 1 G50 T51 G52 R56 V57 A70 K72 M120 E121 Y122 E170 L173 T183 D184 F327 G47 T48 G49 R53 V54 A67 K69 M117 E118 Y119 E167 L170 T180 D181 F324 D166 K168 E170 N171 D184 T201 D163 K165 E167 N168 D181 T198 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 26578105 1351 AAAKKGSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4um1 A 2.83 BS01 09P A 1 Y89 W143 Y192 Y89 W143 Y188 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=2.2nM P58154 26180047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 4um1 A 2.83 BS02 09P E 1 H104 Q112 T114 H104 Q112 T114 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=2.2nM P58154 26180047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKK 4um1 B 2.83 BS01 09P A 1 W53 H104 T114 W53 H104 T114 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=2.2nM P58154 26180047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4um1 B 2.83 BS02 09P B 1 Y89 W143 Y185 C188 Y192 Y89 W143 Y180 C183 Y187 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=2.2nM P58154 26180047 211 LDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4um3 P 2.703 BS01 09R P 1 Y89 W143 Y185 C187 Y192 Y88 W142 Y180 C182 Y187 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=1.3nM P58154 26180047 301 LDRADILYNIRQTSRPDVIPTQRRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGR 4um3 P 2.703 BS02 09R T 1 W53 H104 Q112 T114 W52 H103 Q111 T113 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=1.3nM P58154 26180047 301 LDRADILYNIRQTSRPDVIPTQRRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGR 4um3 Q 2.703 BS01 09R P 1 W53 H104 Q112 T114 W50 H101 Q109 T111 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=1.3nM P58154 26180047 301 LDRADILYNIRQTSRPDVIPTQPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4um3 Q 2.703 BS02 09R Q 1 Y89 W143 Y185 C187 C188 Y192 Y86 W140 Y176 C178 C179 Y183 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=1.3nM P58154 26180047 301 LDRADILYNIRQTSRPDVIPTQPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLAHVVSDGEVQYTPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKG 4uma A 1.76 BS02 GZ3 A 1 R94 K99 G165 A166 R167 K188 R236 H270 R78 K83 G149 A150 R151 K172 R220 H254 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Ki=3.9uM remove_due_to_license_issue Q9K169 25245459 1351 ELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMAR 4uma B 1.76 BS02 GZ3 B 1 R94 K99 G165 A166 R167 K188 R236 H270 R78 K83 G149 A150 R151 K172 R220 H254 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Ki=3.9uM remove_due_to_license_issue Q9K169 25245459 1351 ELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMAR 4umb A 2.17 BS02 0V5 A 1 R94 K99 A166 R167 K188 R236 H270 R79 K84 A151 R152 K173 R221 H255 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Ki=99uM remove_due_to_license_issue Q9K169 25245459 1353 KELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMARA 4umb B 2.17 BS02 0V5 B 1 R94 K99 P100 G165 A166 R167 K188 R236 H270 R78 K83 P84 G149 A150 R151 K172 R220 H254 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Ki=99uM remove_due_to_license_issue Q9K169 25245459 1351 ELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMAR 4umc A 2.34 BS02 PEQ A 1 R94 K99 G165 R167 K188 R236 H270 R79 K84 G150 R152 K173 R221 H255 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Ki=360uM remove_due_to_license_issue Q9K169 25245459 1352 KELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMAR 4umc B 2.34 BS02 PEQ B 1 R94 K99 G165 A166 R167 K188 R236 H270 R78 K83 G149 A150 R151 K172 R220 H254 2.5.1.54 0003849,0005737,0008652,0009058,0009073,0009423,0016740,0046872 Ki=360uM remove_due_to_license_issue Q9K169 25245459 1352 ELLPPIAHLYELPISKEASGLVHRTRQEISDLVHGRDKRLLVIIGPCSIHDPKAALEYAERLLKLRKQYENELLIVMRVYFEKPRTTVGWKGLINDPHLDGTFDINFGLRQARSLLLSLNNMGMPASTEFLDMITPQYYADLISWGAIGARTTESQVHRELASGLSCPVGFKNGTDGNLKIAIDAIGAASHSHHFLSVTKAGHSAIVHTGGNPDCHVILRGGKEPNYDAEHVSEAAEQLRAAGVTDKLMIDCSHANSRKDYTRQMEVAQDIAAQLEQDGGNIMGVMVESHLVEGRQDKPEVYGKSITDACIGWGATEELLALLAGANKKRMARA 4umj A 1.85 BS03 BFQ A 1 S79 D83 R94 M153 Q157 K180 S78 D82 R93 M152 Q156 K175 2.5.1.10 0004659,0005737,0008299,0016740,0046872 ic50=2.7uM remove_due_to_license_issue Q9HWY4 25760619 1297 IAAYQARCQARVDAALDALFVAPREELQRLYEAMRYSVMNGGKRVRPLLAYAACEALGGAPQRADAAACAVELIHAYSLVHDDLPAMDDDDLRRGQPTTHRAFDEATAILAADGLQALAFEVLADTRRNPQEHAVCLEMLTRLARAAGSAGMVGGQAIDLGSLDQAALEVMHRHKTGALIEASVRLGALASGRAEPASLAALERYAEAIGLAFQVQDDILDVPTYPALLGLEAAKGYALELRDLALAALDGFPPSADPLRQLARYIVER 4umj A 1.85 BS04 BFQ A 2 F218 D222 F213 D217 2.5.1.10 0004659,0005737,0008299,0016740,0046872 ic50=2.7uM remove_due_to_license_issue Q9HWY4 25760619 1298 IAAYQARCQARVDAALDALFVAPREELQRLYEAMRYSVMNGGKRVRPLLAYAACEALGGAPQRADAAACAVELIHAYSLVHDDLPAMDDDDLRRGQPTTHRAFDEATAILAADGLQALAFEVLADTRRNPQEHAVCLEMLTRLARAAGSAGMVGGQAIDLGSLDQAALEVMHRHKTGALIEASVRLGALASGRAEPASLAALERYAEAIGLAFQVQDDILDVPTYPALLGLEAAKGYALELRDLALAALDGFPPSADPLRQLARYIVER 4umj B 1.85 BS03 BFQ B 1 S79 D83 R94 Q157 K180 S80 D84 R95 Q158 K181 2.5.1.10 0004659,0005737,0008299,0016740,0046872 ic50=2.7uM remove_due_to_license_issue Q9HWY4 25760619 1294 SMIAAYQARCQARVDAALDALFVAPREELQRLYEAMRYSVMNGGKRVRPLLAYAACEALGGAPQRADAAACAVELIHAYSLVHDDLPAMDDDDLRRGQPTTHRAFDEATAILAADGLQALAFEVLADTRRNPQEHAVCLEMLTRLARAAGSAGMVGGQAIDLGSVGVALDQAALEVMHRHKTGALIEASVRLGALASGRAEPASLAALERYAEAIGLAFQVQDDILDVPTYPALLGLEAAKGYALELRDLALAALDGFPPSADPLRQLARYIV 4umq A 2.6 BS01 B5S A 1 I17 A38 K40 E57 L61 C70 L86 E87 Y88 C89 P90 L139 I149 D150 I13 A34 K36 E53 L57 C66 L82 E83 Y84 C85 P86 L135 I145 D146 D132 K134 E136 N137 D150 S171 D128 K130 E132 N133 D146 S152 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589925 1334 DELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4umr A 3.0 BS01 QBB A 1 I17 V25 L27 A38 Y88 C89 P90 L139 I12 V20 L22 A33 Y83 C84 P85 L134 D132 K134 E136 N137 D150 S171 D127 K129 E131 N132 D145 S151 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=160000nM Q14680 25589925 1334 ELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4umt A 1.98 BS01 47W A 1 A38 E57 L61 A129 H130 L139 I149 D150 F151 A36 E55 L59 A127 H128 L137 I147 D148 F149 D132 K134 E136 N137 D150 S171 D130 K132 E134 N135 D148 S154 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589926 1335 DYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4umu A 2.02 BS01 0V0 A 1 A38 E57 L61 I69 C89 L139 L148 I149 D150 F151 A36 E55 L59 I67 C87 L137 L146 I147 D148 F149 D132 K134 E136 N137 D150 S171 D130 K132 E134 N135 D148 S154 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 25589926 1334 DYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDTAAALVAKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 4und A 2.2 BS01 2YQ A 1 E763 H862 G863 Y889 Y896 S904 Y907 E109 H208 G209 Y235 Y242 S250 Y253 S904 Y907 E988 S250 Y253 E334 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Ki=1.2nM, IC50=0.570000nM, EC50=2.5nM P09874 28001384 2011 NLYFQSMKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 4unn A 2.5 BS01 QZZ A 1 D9 P37 M66 F70 R74 R95 S99 N100 Y103 S104 R107 D9 P37 M66 F70 R74 R95 S99 N100 Y103 S104 R107 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 ic50=0.42uM remove_due_to_license_issue IC50=420nM P9WKE1 25486447 1210 VLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAP 4unp A 2.3 BS01 TXW A 1 F70 R74 N100 Y103 F70 R74 N100 Y103 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 Kd=590uM remove_due_to_license_issue IC50=590000nM P9WKE1 25486447 1211 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAPP 4unq A 2.3 BS01 H6D A 1 P37 F70 R74 R95 S99 N100 Y103 S104 R107 P37 F70 R74 R95 S99 N100 Y103 S104 R107 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 ic50=0.24uM remove_due_to_license_issue P9WKE1 25486447 1210 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAEDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAP 4unr A 1.98 BS01 QZE A 1 D9 P37 L52 F70 R74 R95 N100 Y103 S104 R107 D9 P37 L52 F70 R74 R95 N100 Y103 S104 R107 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 ic50=0.002uM remove_due_to_license_issue IC50=2.0nM P9WKE1 25486447 1211 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAEDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAP 4uns A 2.18 BS01 QZ3 A 1 D9 P37 Y39 F70 R74 R95 N100 Y103 D9 P37 Y39 F70 R74 R95 N100 Y103 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 ic50=0.2uM remove_due_to_license_issue IC50=200nM P9WKE1 25486447 1210 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAEDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAP 4uof A 2.102 BS01 DAT A 1 L54 F59 R87 T93 V111 N114 L54 F59 R87 T93 V111 N114 K11 Y51 N114 H117 E128 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0006183,0006228,0006241,0009142,0016301,0046872 remove_due_to_license_issue A5J299 25195883 1152 MVRERTFIAVKPDGVQRGLIGEIIKRFEAKGFKLAGMKYIQASEDLLKQHYIDLADKPFYPGLCKYMSSGPVVAMCWEGTGVVKTARVMMGETRPADSKPGTIRGDFCIEVGRNIIHGSDSVESANKEIALWFKPEELVSWTQTNESWIYE 4uof B 2.102 BS01 DAT B 1 L54 F59 L63 R87 T93 V111 L54 F59 L63 R87 T93 V111 K11 Y51 N114 H117 E128 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0006183,0006228,0006241,0009142,0016301,0046872 remove_due_to_license_issue A5J299 25195883 1152 MVRERTFIAVKPDGVQRGLIGEIIKRFEAKGFKLAGMKYIQASEDLLKQHYIDLADKPFYPGLCKYMSSGPVVAMCWEGTGVVKTARVMMGETRPADSKPGTIRGDFCIEVGRNIIHGSDSVESANKEIALWFKPEELVSWTQTNESWIYE 4uoh B 2.007 BS01 ADP B 1 K11 L54 F59 L63 R87 T93 V111 N114 K11 L54 F59 L63 R87 T93 V111 N114 K11 Y51 N114 H117 E128 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0006183,0006228,0006241,0009142,0016301,0046872 remove_due_to_license_issue A5J299 25195883 1152 MVRERTFIAVKPDGVQRGLIGEIIKRFEAKGFKLAGMKYIQASEDLLKQHYIDLADKPFYPGLCKYMSSGPVVAMCWEGTGVVKTARVMMGETRPADSKPGTIRGDFCIEVGRNIIHGSDSVESANKEIALWFKPEELVSWTQTNESWIYE 4uoh C 2.007 BS01 ADP C 1 K11 L54 F59 R87 T93 V111 N114 K11 L54 F59 R87 T93 V111 N114 K11 Y51 N114 H117 E128 K11 Y51 N114 H117 E128 2.7.4.6 0004550,0005524,0006183,0006228,0006241,0009142,0016301,0046872 remove_due_to_license_issue A5J299 25195883 1152 MVRERTFIAVKPDGVQRGLIGEIIKRFEAKGFKLAGMKYIQASEDLLKQHYIDLADKPFYPGLCKYMSSGPVVAMCWEGTGVVKTARVMMGETRPADSKPGTIRGDFCIEVGRNIIHGSDSVESANKEIALWFKPEELVSWTQTNESWIYE 4up5 A 1.65 BS03 94W A 1 A332 F354 T359 D380 A7 F29 T34 D55 ? Kd=2.5mM remove_due_to_license_issue Q86UU0,Q9BRQ0 25323450 1385 GVYPCGACRSEVNDDQDAILCEASCQKWFHRECTGMTESAYGLLTTEASAVWACDLCVYVFTTHLANTAAEAVLQGRADSILAYH 4ura A 2.23 BS02 LEL A 1 Y132 Y177 F185 H188 K206 K241 Y129 Y174 F182 H185 K203 K238 G170 Y177 H188 E190 H276 S288 G167 Y174 H185 E187 H273 S285 1.14.11.66,1.14.11.69 ic50=0.00000316uM remove_due_to_license_issue O75164 26682034 4000 ESETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAE 4urk A 2.9 BS01 A82 A 1 M804 W812 I831 Y867 I879 V882 M953 I963 D964 M560 W568 I587 Y623 I635 V638 M709 I719 D720 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=1090nM P48736 25042253 2092 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 4url A 2.29 BS01 XAM A 1 I46 N49 E53 D76 R79 M81 H86 T92 I96 L100 H101 G103 T168 I29 N32 E36 D59 R62 M64 H69 T75 I79 L83 H84 G86 T137 0003677,0003918,0005524,0006265 ic50=500nM remove_due_to_license_issue 24992706 2000 EGLEAVRKRPGMYIGSTDKRGLHHLVYEIVDNSVDEVLNGYGNEIDVTINKDGSISIEDNGRGMPTGIHKSGKPTVEVIFTVLHAGHGVGASVVNALSEWLEVEIHRDGNIYHQSFKNGGSPSSGLVKKGKTKKTGTKVTFKPDDTIFKASTSFNFDVLSERLQESAFLLKNLKITLNDLRSGKERQEHYHYEEGIKEFVSYVNEGKEVLHDVATFSGEANGIEVDVAFQYNDQYSESILSFVNNVRTKDGGTHEVGFKTAMTRVFNDYARRINELKTDKNLDGNDIREGLTAVVSVRIPEELLQFKSKLGTSEARSAVDSVVADKLPFYLEEKGQLSKSLVKKAIKAQQAREAARKAREDARS 4urm A 2.94 BS01 XAM A 1 N54 E58 D81 R84 I86 Q91 K93 M94 H107 A108 G109 G110 T173 I175 N30 E34 D57 R60 I62 Q67 K69 M70 H83 A84 G85 G86 T136 I138 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue P0A0K8 24992706 2000 LEAARKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTVLHAGGKGVGSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYEG 4urn A 2.3 BS01 NOV A 1 N49 E53 R79 M81 P82 I96 R138 N33 E37 R63 M65 P66 I80 R103 0003677,0003918,0005524,0006265 remove_due_to_license_issue 24992706 2000 LEGLEAVRKRPGMYIGSTDKRGLHHLVYEIVDNSVDEVLNGYGNEIDVTINKDGSISIEDNGRGMPTGIHKSGKPTVEVIFTVLVGASVVNALSEWLEVEIHRDGNIYHQSFKNGGSPSSGLVKKGKTKKTGTKVTFKPDDTIFKASTSFNFDVLSERLQESAFLLKNLKITLNDLRSGKERQEHYHY 4uro A 2.59 BS01 NOV A 1 N54 S55 E58 D81 R84 I86 P87 D89 I102 R144 N29 S30 E33 D56 R59 I61 P62 D64 I77 R100 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue IC50=41nM P0A0K8 24992706 2000 EAARKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTVGVGSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYEG 4uru S 2.83 BS01 6W2 S 1 M878 N879 Y884 F890 L901 H905 M285 N286 Y291 F297 L308 H312 ? 0005085,0007264 remove_due_to_license_issue Q07889 25695162 2046 MRLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4urv S 2.58 BS01 UMK S 1 M878 N879 Y884 D887 F890 L901 M283 N284 Y289 D292 F295 L306 ? 0005085,0007264 remove_due_to_license_issue Q07889 25695162 2047 RLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4urw S 2.76 BS01 DXO S 1 M878 D887 F890 K898 L901 H905 M286 D295 F298 K306 L309 H313 ? 0005085,0007264 remove_due_to_license_issue Q07889 25695162 2046 QMRLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4urx S 2.49 BS02 HXY S 1 V852 V883 Y884 L886 F890 V259 V290 Y291 L293 F297 ? 0005085,0007264 Kd=1.3mM remove_due_to_license_issue Q07889 25695162 2047 QMRLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPESAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIASSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4ury R 2.47 BS01 RV1 R 1 K5 L6 D54 L56 Y71 T74 K6 L7 D55 L57 Y72 T75 3.6.5.2 0003924,0005525,0007165,0016020 Kd=6mM remove_due_to_license_issue P01112 25695162 1167 HMTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHQYREQIKRVKDSDDVPMVLVGNKCDLAARTVESRQAQDLARSYGIPYIETSAKTRQGVEDAFYTLVREIRQH 4ury S 2.47 BS01 RV1 R 1 S908 H911 Y912 S312 H315 Y316 ? 0005085,0007264 Kd=6mM remove_due_to_license_issue Q07889 25695162 1167 QMRLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4ury S 2.47 BS02 RV1 S 1 R786 E864 V1040 P1042 R190 E268 V444 P446 ? 0005085,0007264 Kd=6mM remove_due_to_license_issue Q07889 25695162 2046 QMRLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4urz R 2.24 BS01 VJP R 1 K5 L6 D54 L56 T74 K6 L7 D55 L57 T75 3.6.5.2 0003924,0005525,0007165,0016020 Kd=3mM remove_due_to_license_issue P01112 25695162 1167 HMTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHQYREQIKRVKDSDDVPMVLVGNKCDLAARTVESRQAQDLARSYGIPYIETSAKTRQGVEDAFYTLVREIRQH 4urz S 2.24 BS01 VJP R 1 S908 D910 H911 S317 D319 H320 ? 0005085,0007264 remove_due_to_license_issue Q07889 25695162 1167 MRLPSADVYRFAEPDSEENIIFEENMQPKAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 4us3 A 2.098 BS01 TRP A 1 S25 A26 L29 G30 Y108 F230 T231 S233 M236 S327 L328 S18 A19 L22 G23 Y101 F223 T224 S226 M229 S320 L321 ? 0016020 Kd=4.8uM remove_due_to_license_issue Q9KDT3 25282149 601 GREQWASRLGFILAAMGSAVGLGNIWRFSYVTGENGGAAFLLVYLGFIALIGIPIVLAEFTIGRRAQSDAVGSFEKLAPGKPWKVAGLMGVAAGFLILSFYGVIAGWILFYLFNYITGQLWSAPAEGFGGFFEGFIANPTLPLFWQALFMIATIWIVAIGVKKGIERSNKILMPLLGVLLIALAIYSLTLGGAKEGLAFLFSPDWSALKDPGVYLAAISQAFFTLSLGMGALITYGSYVSKDSRLPGAAVSVAGLDTAFAIIAGIMIFPAVFALGLSPSGGPGLVFVVLPDIFDSIRLGPIVGIAFFILLGAAALSSAVSLLEVPVAYFMRKFDWSRKQAAITLGVIITLLGIPSSLSFGVLGEVTIIPGLNIFDSVDFIASSVFLPLGGMIIALFIGWGWKTSDALAESDLTDSVWGKLWILSLRFIAPIAILIVFLSAF 4us4 A 2.6 BS01 TRP A 1 S25 A26 G28 G30 Y108 F230 T231 S233 M236 L328 S9 A10 G12 G14 Y92 F214 T215 S217 M220 L312 ? 0016020 remove_due_to_license_issue Q9KDT3 25282149 601 GFILAAMGSAVGLGNIWRFSYVTGENGGAAFLLVYLGFIALIGIPIVLAEFTIGRRAQSDAVGSFEKLAPGKPWKVAGLMGVAAGFLILSFYGVIAGWILFYLFNYITGQLWSAPAEGFGGFFEGFIANPTLPLFWQALFMIATIWIVAIGVKKGIERSNKILMPLLGVLLIALAIYSLTLGGAKEGLAFLFSPDWSALKDPGVYLAAISQAFFTLSLGMGALITYGSYVSKDSRLPGAAVSVAGLDTAFAIIAGIMIFPAVFALGLSPSGGPGLVFVVLPDIFDSIRLGPIVGIAFFILLGAAALSSAVSLLEVPVAYFMRKFDWSRKQAAITLGVIITLLGIPSSLSFGVLGEVTIIPGLNIFDSVDFIASSVFLPLGGMIIALFIGWGWKTSDALAESDLTDSVWGKLWILSLRFIAPIAILIVFLSAFQ 4usi A 1.45 BS02 AKG A 1 V53 G54 Q56 G58 K76 G105 V49 G50 Q52 G54 K65 G94 0006808,0030234 Kd=38.9uM remove_due_to_license_issue 25416954 1153 SIQCDLSAFPGVKFFRIEAIFRPWRLPFVIDTLSKYGIRGLTNTPVKGVGVQGGSEFGPSNLVDKEKLDIVVSRAQVDAVVRLVAASAYTGEIGDGKIFVHPVAEVVRIRTAETG 4usj A 2.85 BS01 ARG A 1 K210 E284 I285 S287 E289 G290 G292 M294 K194 E268 I269 S271 E273 G274 G276 M278 K41 G44 G76 G77 R98 D196 D216 K255 K25 G28 G60 G61 R82 D180 D200 K239 2.7.2.8 0003991,0005524,0005737,0006526,0016301 remove_due_to_license_issue Q9SCL7 25416954 301 DYRVEILSESLPFIQKFRGKTIVVKYGGAAMTSPELKSSVVSDLVLLACVGLRPILVHGGGPDINRYLKQLNIPAEFRDGLRVTDATTMEIVSMVLVGKVNKNLVSLINAAGATAVGLSGHDGRLLTARPVPNSAQLGFVGEVARVDPSVLRPLVDYGYIPVIASVAADDSGQAYNINADTVAGELAAALGAEKLILLTDVAGILENKEDPSSLIKEIDIKGVKKMIEDGKVAGGMIPKVKCCIRSLAQGVKTASIIDGRRQHSLLHEIMSDEGAGTMITG 4usj B 2.85 BS01 ARG B 1 F33 K210 K232 E284 I285 S287 E289 G290 M294 F17 K194 K216 E268 I269 S271 E273 G274 M278 K41 G44 G77 D196 K255 K25 G28 G61 D180 K239 2.7.2.8 0003991,0005524,0005737,0006526,0016301 remove_due_to_license_issue Q9SCL7 25416954 301 DYRVEILSESLPFIQKFRGKTIVVKYGGAAMTSPELKSSVVSDLVLLACVGLRPILVHGGGPDINRYLKQLNIPAEFRDGLRVTDATTMEIVSMVLVGKVNKNLVSLINAAGATAVGLSGHDGRLLTARPVPNSAQLGFVGEVARVDPSVLRPLVDYGYIPVIASVAADDSGQAYNINADTVAGELAAALGAEKLILLTDVAGILENKEDPSSLIKEIDIKGVKKMIEDGKVAGGMIPKVKCCIRSLAQGVKTASIIDGRRQHSLLHEIMSDEGAGTMITG 4usw A 2.05 BS01 ATP A 1 D47 S49 G50 T52 A97 G98 D99 F338 L345 V406 N412 D47 S49 G50 T52 A97 G98 D99 F330 L337 V397 N403 4.6.1.1 0009190,0035556 Kd=2.03mM remove_due_to_license_issue Q96PN6 25040695 1471 MNTPKEEFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTE 4uuh A 2.52 BS02 T40 A 1 H1184 G1185 H1201 Y1203 Y1213 F1214 A1215 K1220 S1221 Y1224 E1291 H80 G81 H97 Y99 Y109 F110 A111 K116 S117 Y120 E181 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 3000 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPYAEYVIYRGEQAYPEYLITYQIMKPE 4uuq A 2.36 BS01 64D A 1 S132 M133 L158 N162 S165 L215 G220 L223 L224 C252 S117 M118 L143 N147 S150 L200 G205 L208 L209 C237 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 remove_due_to_license_issue Q99685 25560837 1306 SPRRTPQSIPYQDLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTA 4uv8 A 2.8 BS01 D69 A 1 G285 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 F538 A539 V590 L625 P626 W756 S760 Y761 G800 E801 A809 T810 V811 A814 G115 G117 S119 L137 E138 A139 R140 G145 R146 G160 A161 M162 V163 F368 A369 V420 L455 P456 W586 S590 Y591 G630 E631 A639 T640 V641 A644 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 25173853 900 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 4uv9 A 3.0 BS01 D70 A 1 G285 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 T335 F538 A589 V590 L625 P626 W751 W756 S760 Y761 G800 E801 A809 T810 V811 A814 G115 G117 S119 L137 E138 A139 R140 G145 R146 G160 A161 M162 V163 T165 F368 A419 V420 L455 P456 W581 W586 S590 Y591 G630 E631 A639 T640 V641 A644 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 25173853 900 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 4uva A 2.9 BS01 D73 A 1 G285 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 F538 A589 V590 L625 P626 W751 W756 S760 Y761 G800 E801 A809 T810 V811 G115 G117 S119 L137 E138 A139 R140 G145 R146 G160 A161 M162 V163 F368 A419 V420 L455 P456 W581 W586 S590 Y591 G630 E631 A639 T640 V641 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 25173853 900 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 4uvb A 2.8 BS01 D51 A 1 G285 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 A539 A589 V590 L625 P626 W756 S760 Y761 G800 E801 A809 T810 V811 A814 G115 G117 S119 L137 E138 A139 R140 G145 R146 G160 A161 M162 V163 A369 A419 V420 L455 P456 W586 S590 Y591 G630 E631 A639 T640 V641 A644 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 25173853 900 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 4uvc A 3.1 BS01 D52 A 1 G285 G287 S289 L307 E308 A309 R310 G315 R316 G330 A331 M332 V333 V590 L625 P626 K661 W751 W756 S760 Y761 G800 E801 A809 T810 V811 G115 G117 S119 L137 E138 A139 R140 G145 R146 G160 A161 M162 V163 V420 L455 P456 K491 W581 W586 S590 Y591 G630 E631 A639 T640 V641 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 25173853 900 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 4uvu A 1.95 BS01 U1T A 1 H1031 G1032 F1035 A1049 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 F84 A98 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=1200nM remove_due_to_license_issue Q9H2K2 26189030 2162 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4uvv A 1.9 BS01 W8L A 1 H1031 G1032 S1033 Y1050 Y1060 F1061 A1062 S1068 Y1071 E1138 H80 G81 S82 Y99 Y109 F110 A111 S117 Y120 E185 2.4.2.-,2.4.2.30 0003950 ic50=32nM remove_due_to_license_issue Q9H2K2 26189030 2162 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4uvw A 2.1 BS02 NYJ A 1 H1031 G1032 S1033 Y1060 A1062 S1068 Y1071 H80 G81 S82 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=19nM remove_due_to_license_issue Q9H2K2 26189030 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4uvx A 1.95 BS02 H2W A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=11nM remove_due_to_license_issue Q9H2K2 26189030 2166 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4uvy A 1.95 BS02 SGW A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 E1138 H80 G81 Y99 Y109 A111 S117 Y120 E185 2.4.2.-,2.4.2.30 0003950 ic50=5.5nM remove_due_to_license_issue Q9H2K2 26189030 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4uw1 A 3.37 BS02 92R A 1 H1184 G1185 Y1203 Y1213 A1215 Y1224 E1291 H80 G81 Y99 Y109 A111 Y120 E187 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue O95271 3000 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKP 4uwf A 2.99 BS01 EUT A 1 F612 P618 I634 K636 Y670 M682 Q683 F684 I685 I760 F289 P295 I311 K313 Y347 M359 Q360 F361 I362 I437 2.7.1.137 0016301,0046854 remove_due_to_license_issue IC50=7.0nM Q8NEB9 25402320 4000 LKPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEINSAEIDSSQIITSPLLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHALFAA 4uwg A 2.7 BS01 RBQ A 1 F612 P618 I634 Y670 M682 Q683 F684 I685 L750 I760 F287 P293 I309 Y345 M357 Q358 F359 I360 L425 I435 2.7.1.137 0016301,0046854 remove_due_to_license_issue IC50=7.0nM Q8NEB9 25402320 1873 LKPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEAEIDSSQIITSPLPLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHA 4uwh A 1.93 BS01 JXM A 1 F612 P618 I634 K636 Y670 M682 Q683 F684 I685 L750 I760 F293 P299 I315 K317 Y351 M363 Q364 F365 I366 L431 I441 2.7.1.137 0016301,0046854 ic50=3nM remove_due_to_license_issue IC50=3.0nM Q8NEB9 25402320 1876 DLKPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEPINSAEIDSSQIITSPLPNLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHALFAA 4uwk A 2.83 BS01 UJB A 1 F612 P618 I634 K636 Y670 M682 Q683 I685 I760 D761 F287 P293 I309 K311 Y345 M357 Q358 I360 I435 D436 2.7.1.137 0016301,0046854 remove_due_to_license_issue Q8NEB9 25402320 1872 KPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEAEIDSSQIITSPLPNLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHA 4uwl A 2.8 BS01 7A5 A 1 F612 S614 P618 I634 Y670 M682 Q683 F684 I685 I760 D761 F286 S288 P292 I308 Y344 M356 Q357 F358 I359 I434 D435 2.7.1.137 0016301,0046854 remove_due_to_license_issue IC50=82nM Q8NEB9 25402320 1872 LKPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLEEIDSSQIITSPLPLEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLFKSALMPAQLFFKTEDGGKYPVIFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFMQFIQSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHA 4ux4 A 1.8 BS01 E9L A 1 H1031 G1032 Y1050 Y1060 F1061 A1062 S1068 Y1071 E1138 H80 G81 Y99 Y109 F110 A111 S117 Y120 E185 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 26026769 2162 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 4ux5 A 2.4 BS01 dna C 0 T52 K62 K80 Q82 G86 K87 Q89 G90 T91 T37 K47 K65 Q67 G71 K72 Q74 G75 T76 ? 0003677 remove_due_to_license_issue G4NA99 25550425 1 ~ 14 GPGIYSATYSGIPVYEYQFGLKEHVMRRRVDDWINATHILKAAGFDKPARTRILEREVQKDQHEKVQGGYGKYQGTWIPLEAGEALAHRNNIFDRLRPIFEFSPGPDSPPPAP 4ux5 A 2.4 BS02 dna D 0 S23 D61 G83 G84 Y85 S10 D46 G68 G69 Y70 ? 0003677 remove_due_to_license_issue G4NA99 25550425 1 ~ 14 GPGIYSATYSGIPVYEYQFGLKEHVMRRRVDDWINATHILKAAGFDKPARTRILEREVQKDQHEKVQGGYGKYQGTWIPLEAGEALAHRNNIFDRLRPIFEFSPGPDSPPPAP 4ux5 B 2.4 BS01 dna C 0 Y22 S23 R67 G84 Y85 P128 Y9 S10 R52 G69 Y70 P113 ? 0003677 remove_due_to_license_issue G4NA99 25550425 1 ~ 14 GPGIYSATYSGIPVYEYQFGLKEHVMRRRVDDWINATHILKAAGFDKPARTRILEREVQKDQHEKVQGGYGKYQGTWIPLEAGEALAHRNNIFDRLRPIFEFSPGPDSPPPAP 4ux5 B 2.4 BS02 dna D 0 K62 G86 Q89 K47 G71 Q74 ? 0003677 remove_due_to_license_issue G4NA99 25550425 1 ~ 14 GPGIYSATYSGIPVYEYQFGLKEHVMRRRVDDWINATHILKAAGFDKPARTRILEREVQKDQHEKVQGGYGKYQGTWIPLEAGEALAHRNNIFDRLRPIFEFSPGPDSPPPAP 4ux6 B 3.0 BS04 YWO B 1 Q257 P344 F363 G365 W366 Y367 E371 Q150 P237 F256 G258 W259 Y260 E264 C194 R197 W366 E371 C87 R90 W259 E264 1.14.13.39 0004517,0006809,0020037 remove_due_to_license_issue P29477 21398123 1499 SCLGSIMNPKSLTRGPRDKPTPLEELLPHAIEFINQYYGSFKEAKIEEHLARLEAVTKEIETTGTYQLTLDELIFATKMAWRNAPRCIGRIQWSNLQVFDARNCSTAQEMFQHICRHILYATNNGNIRSAITVFPQRSDGKHDFRLWNSQLIRYAGYQMPDGTIRGDAATLEFTQLCIDLGWKPRYGRFDVLPLVLQADGQDPEVFEIPPDLVLEVTMEHPKYEWFQELGLKWYALPAVANMLLEVGGLEFPACPFNGWYMGTEIGVRDFCDTQRYNILEEVGRRMGLETHTLASLWKDRAVTEINVAVLHSFQKQNVTIMDHHTASESFMKHMQNEYRARGGCPADWIWLVPPVSGSITPVFHQEMLNYVLSPFYYYQIEPWKTHIWQ 4uxb A 3.22 BS01 P34 A 1 H862 G863 G888 Y889 Y896 S904 Y907 H182 G183 G208 Y209 Y216 S224 Y227 S904 Y907 E988 S224 Y227 E301 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=110nM, Kd=110nM, EC50=20nM P09874 28001384 2011 MKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQDSQILDLSNRFYTLIPHDPLLNNADSVQAKAEMLDNLLDIEVAYSLLRDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHANAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHSKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 4uxh A 2.4 BS01 T5A A 1 M13 F14 G16 K17 T18 T19 M22 K39 Y46 E85 Q87 F88 L111 D114 Y115 F120 T151 Q160 L162 G164 Y169 M11 F12 G14 K15 T16 T17 M20 K37 Y44 E79 Q81 F82 L105 D108 Y109 F114 T145 Q154 L156 G158 Y163 2.7.1.21 0004797,0005524 ic50=1.1uM remove_due_to_license_issue Q4QC75 25978379 1180 RGRIELIIGPMFAGKTTELMRRVKREIHARRSCFVIKYSKDTRYDEHNVALMLRAQAAVSQLTEVRDTWKRFDVLAIDEGQFFSDLVDFCNTAADAGKVVMVSALDGDYRRKPFGQICELVPYCEAVDKLTAVCMMCHEQPACFTRRTVNVEQQELIGGADMYIATCRECYSK 4uxj E 3.0 BS02 TTP E 1 M13 F14 G16 K17 T18 E85 F88 L111 D114 Y115 T151 Q160 L162 G164 Y169 M11 F12 G14 K15 T16 E76 F79 L102 D105 Y106 T142 Q151 L153 G155 Y160 2.7.1.21 0004797,0005524 remove_due_to_license_issue Q4QC75 25978379 1181 RGRIELIIGPMFAGKTTELMRRVKREIHARRSCFVIKYSKDTRYDEHNVASAQAAVSQLTEVRDTWKRFDVLAIDEGQFFSDLVDFCNTAADAGKVVMVSALDGDYRRKPFGQICELVPYCEAVDKLTAVCMMCHEQPACFTRRTVNVEQQELIGGADMYIATCRECYSK 4uxl A 2.4 BS01 5P8 A 1 L1951 A1978 L2026 M2029 G2032 L2086 G2101 K2228 S2229 L18 A45 L93 M96 G99 L153 G168 K287 S288 D2079 A2081 R2083 N2084 D2102 E2120 D146 A148 R150 N151 D169 E179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki<0.025nM remove_due_to_license_issue P08922 25733882 3230 IENLPAFPREKLTLRLLLGSGAFGEVYEGTAVDILGVGSGEIKVAVKTLKKGSTDQEKIEFLKEAHLMSKFNHPNILKQLGVCLLNEPQYIILELMEGGDLLTYLRKARMATFYGPLLTLVDLVDLCVDISKGCVYLERMHFIHRDLAARNCLVSVKDYTSPRIVKIGDFGLARDIYKEGLLPVRWMAPESLMDGIFTTQSDVWSFGILIWEILTLGHQPYPAHSNLDVLNYVQTGGRLEPPRNCPDDLWNLMTQCWAQEPDQRPTFHRIQDQLQLFRNFFLNSIYKS 4uxq A 1.85 BS01 0LI A 1 L473 V481 A501 K503 E520 M524 I527 I534 V550 A553 I609 H610 R611 L619 I628 A629 D630 F631 L22 V30 A50 K52 E69 M73 I76 I83 V99 A102 I145 H146 R147 L155 I164 A165 D166 F167 D612 A614 R616 N617 D630 D641 R650 D148 A150 R152 N153 D166 D177 R186 2.7.10.1 0004672,0004713,0005524,0006468 Kd=16nM remove_due_to_license_issue IC50=8.0nM P22455 25465127 1752 LDLPLDPLWEFPRDRLVLGKPLGEGAFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 4uy1 A 2.2 BS02 TJM A 1 L5 P17 Y20 G28 H46 D47 L5 P17 Y20 G28 H46 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 ic50=20uM remove_due_to_license_issue IC50=20000nM O15496 25316315 1130 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKC 4uyd A 1.37 BS01 V1T A 1 P82 L92 N140 I146 P40 L50 N98 I104 ? ic50=79.4uM remove_due_to_license_issue IC50=79433nM O60885 25408830 1171 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4uye A 1.65 BS01 9F9 A 1 I652 F653 E655 V657 P658 E661 N708 F714 I24 F25 E27 V29 P30 E33 N80 F86 ? Kd=9.54nM remove_due_to_license_issue IC50=79nM P55201 25408830 1739 QLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAE 4uyf A 1.6 BS01 73B A 1 W97 P98 K107 L108 N156 I162 W27 P28 K37 L38 N86 I92 ? Kd=4.4nM remove_due_to_license_issue IC50=158nM, Kd=25nM P25440 25249180 1191 NPGRVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQELVV 4uyf A 1.6 BS02 73B C 1 N77 Q80 H83 K84 N7 Q10 H13 K14 ? Kd=4.4nM remove_due_to_license_issue IC50=158nM, Kd=25nM P25440 25249180 1183 NPGRVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQELVV 4uyg A 2.5 BS01 73B A 1 W370 P371 V376 L381 N429 V435 M438 W24 P25 V30 L35 N83 V89 M92 ? Kd=4.4nM remove_due_to_license_issue IC50=158nM, Kd=25nM P25440 25249180 1456 SEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 4uyh A 1.73 BS01 9S3 A 1 W97 P98 K107 L108 N156 I162 W23 P24 K33 L34 N82 I88 ? ic50=0.00000001M remove_due_to_license_issue IC50=501nM P25440 25249180 1184 VTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQE 4uyn A 1.9 BS01 Y3M A 1 G140 V147 A160 K162 L178 V182 Q185 L208 L210 Y212 A213 G216 L263 F275 G16 V23 A36 K38 L52 V56 Q59 L82 L84 Y86 A87 G90 L137 F149 D256 K258 E260 N261 D274 D130 K132 E134 N135 D148 2.7.11.1 0004672,0005524,0006468 ic50=4nM remove_due_to_license_issue O14965 25369539 1392 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 4uzb A 2.865 BS01 dna C 0 H1011 P1012 R1013 Y1014 P1033 Y1066 K1070 W1122 L1128 A1129 G1130 H2 P3 R4 Y5 P24 Y57 K61 W113 L119 A120 G121 ? 0003677,0042025 remove_due_to_license_issue Q9QR71 25947153 2 ~ 21 PHPRYQQPPVPYRQIDDCPAKARPQHIFYQQFLGKDGRRDPKCQWEFAVIFWGNDPYGLKKLSQAFQFGGVKAGPVSCLPHPGPDQSPITYCVYVYCQNAATSKKVQMARLEWEASHPLAGNLQSSIVSFDDPLPLT 4uzb A 2.865 BS02 dna D 0 P1012 R1013 Y1014 Q1015 K1030 K1069 P3 R4 Y5 Q6 K21 K60 ? 0003677,0042025 remove_due_to_license_issue Q9QR71 25947153 -21 ~ -2 PHPRYQQPPVPYRQIDDCPAKARPQHIFYQQFLGKDGRRDPKCQWEFAVIFWGNDPYGLKKLSQAFQFGGVKAGPVSCLPHPGPDQSPITYCVYVYCQNAATSKKVQMARLEWEASHPLAGNLQSSIVSFDDPLPLT 4uzb B 2.865 BS01 dna C 0 H1011 R1013 K1030 Y1066 H2 R4 K21 Y57 ? 0003677,0042025 remove_due_to_license_issue Q9QR71 25947153 2 ~ 21 PHPRYQQPPVPYRQIDDCPAKARPQHIFYQQFLGKDGRRDPKCQWEFAVIFWGNDPYGLKKLSQAFQFGGVKAGPVSCLPHPGPDQSPITYCVYVYCQNAATSKKVQMARLEWEASHPLAGNLQSSIVSFDDPLPLT 4uzb B 2.865 BS02 dna D 0 P1012 Q1015 P3 Q6 ? 0003677,0042025 remove_due_to_license_issue Q9QR71 25947153 -21 ~ -2 PHPRYQQPPVPYRQIDDCPAKARPQHIFYQQFLGKDGRRDPKCQWEFAVIFWGNDPYGLKKLSQAFQFGGVKAGPVSCLPHPGPDQSPITYCVYVYCQNAATSKKVQMARLEWEASHPLAGNLQSSIVSFDDPLPLT 4uzd A 3.2 BS01 QMN A 1 V147 K162 L178 Q185 L194 L208 L210 Y212 A213 A273 F275 V21 K36 L52 Q59 L68 L82 L84 Y86 A87 A147 F149 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=0.600000nM, EC50=106nM O14965 25369539 1389 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4uzd B 3.2 BS01 QMN B 1 K141 V147 A160 K162 L178 Q185 L194 L208 E211 Y212 A213 A273 F275 G276 K17 V23 A36 K38 L54 Q61 L70 L84 E87 Y88 A89 A149 F151 G152 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T161 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=0.600000nM, EC50=106nM O14965 25369539 1390 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 4uzh A 2.0 BS01 JVE A 1 L139 V147 A160 E211 Y212 A213 N242 L263 A273 S391 L16 V24 A37 E88 Y89 A90 N119 L140 A150 S251 D256 K258 E260 N261 D274 D133 K135 E137 N138 D151 2.7.11.1 0004672,0005524,0006468 ic50=9800nM remove_due_to_license_issue IC50=9800nM O14965 25369539 1392 MKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 4v01 A 2.33 BS01 0LI A 1 A512 K514 E531 M534 M535 I545 V561 Y563 A564 I620 H621 L630 I639 A640 D641 A42 K44 E61 M64 M65 I75 V91 Y93 A94 I136 H137 L146 I155 A156 D157 D623 A625 R627 N628 D641 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 25465127 1776 LPEDPRWELPRDRLVLGKPLGGQVVLAEAIGLDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4v04 A 2.12 BS01 0LI A 1 V492 A512 K514 E531 M534 V561 Y563 A564 L614 C619 I620 H621 R622 L630 I639 A640 D641 G643 L644 V27 A47 K49 E66 M69 V96 Y98 A99 L147 C152 I153 H154 R155 L163 I172 A173 D174 G176 L177 D623 A625 R627 N628 D641 D156 A158 R160 N161 D174 0004672,0004713,0005007,0005524,0006468 Kd=7.7nM remove_due_to_license_issue 25465127 1772 YELPEDPRWELPRDRLVLGKPLGEGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4v05 A 2.57 BS01 66T A 1 L484 F489 A512 K514 E531 V561 Y563 A564 S565 G567 L630 D641 L21 F26 A49 K51 E68 V98 Y100 A101 S102 G104 L156 D167 D623 A625 R627 N628 D641 D149 A151 R153 N154 D167 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue 25465127 1769 ELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4v0i A 2.54 BS01 J82 A 1 F751 M752 P758 W760 I777 Y813 E826 V827 V828 M900 I910 D911 F504 M505 P511 W513 I530 Y566 E579 V580 V581 M646 I656 D657 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 27144736 1500 KKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPVSNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNQPFSIELIVQAGLFHGNEMLCKTDISVCDLPRMARLCFALYADCPIAWANLMLFDYKDQLKTGERCLYMWPSLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLTAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRES 4v1f A 1.697 BS01 BQ1 A 1 G62 E65 A66 F69 G62 E65 A66 F69 0015078,0015986,0033177,0045263,1902600 remove_due_to_license_issue 26601184 1087 MELDPNALITAGALIGGGLIMGGGAIGAGIGDGIAGNALISGIARQPEAQGRLFTPFFITVGLVEAAYFINLAFMALFVFATPGLQ 4v1f A 1.697 BS02 BQ1 B 1 A67 I70 A67 I70 0015078,0015986,0033177,0045263,1902600 remove_due_to_license_issue 26601184 1087 MELDPNALITAGALIGGGLIMGGGAIGAGIGDGIAGNALISGIARQPEAQGRLFTPFFITVGLVEAAYFINLAFMALFVFATPGLQ 4v24 A 1.8 BS01 GYR A 1 F259 I260 V263 D264 F278 L347 L354 M358 F374 F389 H397 F167 I168 V171 D172 F186 L249 L256 M260 F276 F291 H299 2.3.1.-,2.7.1.91 0000287,0001568,0001727,0003376,0003677,0005515,0005516,0005524,0005634,0005654,0005737,0005768,0005829,0005886,0005905,0006473,0006629,0006670,0006954,0007420,0008283,0008284,0008289,0008481,0010008,0010800,0010803,0016020,0016301,0016407,0017050,0019722,0030100,0030139,0030148,0030307,0030335,0031398,0031901,0032651,0032740,0034612,0035556,0035924,0038036,0043066,0043231,0045202,0045766,0045840,0045931,0045987,0046512,0046521,0048146,0050764,0051092,0051721,0070301,0071363,0071897,0090520,0098793,0150077,1900060,1900745,1901224,1903978,1905364 Ki=4.3nM remove_due_to_license_issue Ki=3.6nM, IC50=28nM, Kd=5.0nM Q9NYA1 25516793 1450 PRGVLPRPCRVLVLLNPRGGKGKALQLFRSHVQPLLAEAEISFTLMLTERRNHARELVRSEELGRWDALVVMSGDGLMHEVVNGLMERPDWETAIQKPLCSLPAGSGNALAASLNHYAGYEQVTNEDLLTNCTLLLCRRLLSPMNLLSLHTASGLRLFSVLSLAWGFIADVDLESEKYRRLGEMRFTLGTFLRLAALRTYRGRLAYLPVGRVGSKTPASGPVDAHLVPLEEPVPSHWTVVPDEDFVLVLALLHSHLGSEMFAAPMGRCAAGVMHLFYVRAGVSRAMLLRLFLAMEKGRHMEYECPYLVYVPVVAFRLEPKDGKGVFAVDGELMVSEAVQGQVHPNYFWMVS 4v25 A 2.6 BS02 SZ6 A 1 K246 N247 R250 A251 D282 G284 G286 V287 T346 K232 N233 R236 A237 D268 G270 G272 V273 T323 H239 E243 K246 N247 H225 E229 K232 N233 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 remove_due_to_license_issue IC50=80nM Q15119 25404640 1369 GSAPKYIEHFSKFSPSPLSMKQFLDFGSACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTAPPLAGFGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVY 4v27 A 1.9 BS01 MAN A 1 H63 R295 E333 H335 E336 H33 R265 E303 H305 E306 3.2.1.130 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 25487964 500 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 4v27 A 1.9 BS02 IFM A 1 Y46 W126 H154 E156 Y195 Y252 E336 Y16 W96 H124 E126 Y165 Y222 E306 3.2.1.130 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 25487964 501 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 4vgc C 2.1 BS02 SRD C 1 S190 M192 S195 V213 S214 W215 G216 S217 S40 M42 S45 V63 S64 W65 G66 S67 M192 G193 D194 S195 G196 M42 G43 D44 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 9425066 358 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 4w4s A 2.0 BS01 B29 A 1 I36 L68 L71 F72 D75 S165 I166 A167 R204 N207 I275 Y280 R281 I36 L68 L71 F72 D75 S165 I166 A167 R204 N207 I264 Y269 R270 ? ic50=9.5uM remove_due_to_license_issue Q45222 25269599 401 MIQTERAVQQVLEWGRSLTGFADEHAVEAVRGGQYILQRIHPSLRGTSARTGRDPQDETLIVTFYRELALLFWLDDCNDLGLISPEQLAAVEQALGQGVPCALPGFEGCAVLRASLATLAYDRRDYAQLLDDTRCYSAALRAGHAQAVAAERWSYAEYLHNGIDSIAYANVFCCLSLLWGLDMATLRARPAFRQVLRLISAIGRLQNDLHDNAVILLLQRYPAMPVVEFLNDELAGHTRMLHRVMAEERFPAPWGPLIEAMAAIRVQYYR 4w4v A 2.01 BS01 3H8 A 1 I70 G73 Q75 V78 A91 K93 I124 L144 M146 L148 M149 D150 A151 L206 I26 G29 Q31 V34 A47 K49 I80 L100 M102 L104 M105 D106 A107 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 ic50=866nM remove_due_to_license_issue IC50=866nM P53779 25623238 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDQLDEREHTIEEWKELIYKEVMN 4w4w A 1.9 BS01 3HJ A 1 I70 A91 K93 I124 L144 M146 L148 M149 D150 A151 L206 I26 A47 K49 I80 L100 M102 L104 M105 D106 A107 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T180 2.7.11.24 0004672,0004707,0005524,0006468 ic50=6630nM remove_due_to_license_issue P53779 25623238 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQLDEREHTIEEWKELIYKEVMN 4w4x A 2.65 BS01 3HN A 1 I70 G73 Q75 V78 K93 I124 L144 M146 L148 M149 D150 A151 L206 I26 G29 Q31 V34 K49 I80 L100 M102 L104 M105 D106 A107 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue P53779 25623238 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPLDEREHTIEEWKELIYKEVMN 4w4y A 2.3 BS01 3HQ A 1 I70 G73 V78 K93 L144 M146 L148 M149 D150 A151 L206 I26 G29 V34 K49 L100 M102 L104 M105 D106 A107 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 ic50=3034nM remove_due_to_license_issue P53779 25623238 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPLDEREHTIEEWKELIYKEVMN 4w52 A 1.5001 BS01 BNZ A 1 L84 V87 A99 V111 L118 L84 V87 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=175uM remove_due_to_license_issue P00720 25847998 200 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKNL 4w53 A 1.56 BS01 MBN A 1 V87 A99 V111 L118 V87 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=102uM remove_due_to_license_issue Kd=102000nM P00720 25847998 200 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKNL 4w54 A 1.7901 BS01 PYJ A 1 A99 L118 A99 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=68uM remove_due_to_license_issue P00720 25847998 200 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKNL 4w55 A 1.6401 BS01 3H0 A 1 V87 Y88 A99 V111 L118 V87 Y88 A99 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=18uM remove_due_to_license_issue P00720 25847998 200 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKNL 4w57 A 1.6801 BS01 N4B A 1 V87 A99 M102 V111 L118 V87 A99 M102 V111 L118 E11 D20 E11 D20 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 Kd=14uM remove_due_to_license_issue P00720 25847998 200 MNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNCNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRCAAINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKNL 4w5j A 1.65 BS01 AP5 A 1 P9 G10 G12 K13 G14 T15 T31 G32 F35 R36 I53 E57 V59 T64 G86 Y87 R89 Q93 R124 R128 T137 F138 H139 F142 R156 R167 I197 P9 G10 G12 K13 G14 T15 T31 G32 F35 R36 I53 E57 V59 T64 G86 Y87 R89 Q93 R124 R128 T137 F138 H139 F142 R155 R166 I196 K13 R89 R128 R156 R167 K13 R89 R128 R155 R166 2.7.4.3 0004017,0005524,0005737,0006139,0009165,0016301,0016776,0019205,0044209,0046940,0050145 remove_due_to_license_issue Q04ML5 25372811 302 MNLLIMGLPGAGKGTQAAKIVEQFHVAHISTGDMFRAAMANQTEMGVLAKSYIDKGELVPDEVTNGIVKERLSQDDIKETGFLLDGYPRTIEQAHALDKTLAELGIELEGIINIEVNPDSLLERLSGRIIHRVTGETFHKVFNPPVYKEEDYYQREDDKPETVKRRLDVNIAQGEPIIAHYRAKGLVHDIEGNQDINDVFSDIEKVLTNLK 4w7p A 2.8 BS01 3J7 A 1 I82 V90 A103 K105 E154 Y155 M156 D160 D202 D216 I77 V85 A98 K100 E146 Y147 M148 D152 D194 D208 D198 K200 N203 D216 T237 D190 K192 N195 D208 T229 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=32nM Q13464 25248678 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEETFPIPKAFVGNQLPFVGFTYYSNRRY 4w7t A 1.8 BS01 3JC A 1 N51 A55 M98 N106 F138 N35 A39 M82 N90 F122 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.9uM remove_due_to_license_issue P07900 25368984 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4w97 A 1.6 BS01 UCA A 1 Y108 Q109 N128 Q131 R159 R162 D163 W166 Y106 Q107 N126 Q129 R157 R160 D161 W164 ? 0000976,0003677,0003700,0006355 Kd=0.08uM remove_due_to_license_issue P9WMB9 25406313 301 RVAGQVNSRRGELLELAAAMFAERGLRATTVRDIADGAGILSGSLYHHFASKEEMVDELLRGFLDWLFARYRDIVDSTANPLERLQGLFMASFEAIEHHHAQVVIYQDEAQRLASQPRFSYIEDRNKQQRKMWVDVLNQGIEEGYFRPDLDVDLVYRFIRDTTWVSVRWYRPGGPLTAQQVGQQYLAIVLGGITKE 4w9c C 2.2 BS01 3JG C 1 W88 Y98 I109 H110 S111 Y112 H115 W117 W27 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=22.2uM remove_due_to_license_issue Kd=22200nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9d C 2.2 BS01 3JK C 1 W88 Y98 I109 H110 S111 Y112 H115 W117 W27 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=10.2uM remove_due_to_license_issue Kd=10200nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9e C 2.6 BS01 3JT C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue Kd=7090nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9f C 2.1 BS01 3JU C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=3.27uM remove_due_to_license_issue Kd=3270nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQ 4w9g C 2.7 BS01 3JV C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue Kd=6530nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9h C 2.1 BS01 3JF C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=0.185uM remove_due_to_license_issue Kd=185nM, IC50=696nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9i C 2.4 BS01 3JS C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=1.1uM remove_due_to_license_issue Kd=1100nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9j C 2.2 BS01 3JH C 1 N67 W88 F91 Y98 I109 H110 S111 Y112 H115 W117 N6 W27 F30 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=0.588uM remove_due_to_license_issue Kd=588nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9k C 2.1 BS01 3JO C 1 R69 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 R8 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=0.291uM remove_due_to_license_issue Kd=291nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9l C 2.2 BS01 3JJ C 1 N67 W88 F91 Y98 I109 H110 S111 Y112 H115 W117 N6 W27 F30 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=9.52uM remove_due_to_license_issue Kd=9520nM P40337 25166285 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 4w9n A 1.84 BS01 TCL B 1 F1766 L1780 I1784 F1791 F233 L241 I245 F252 1.1.1.100,1.3.1.39,2.3.1.38,2.3.1.39,2.3.1.41,2.3.1.85,3.1.2.14,4.2.1.59 0016491 remove_due_to_license_issue P49327 25301948 1905 HAFVSTLTRGDLSSIRWVCSRHAQPTCPGAQLCTVYYASLNFRDIMLATGKLSPDAIPGKWTSQDSLLGMEFSGRDASGKRVMGLVPAKGLATSVLLSPDFLWDVPSNWTLEEAASVPVVYSTAYYALVVRGRVRPGETLLIHSGSGGVGQAAIAIALSLGCRVFTTVGSAEKRAYLQARFPQLDSTSFANSRSFEQHVLWHTGGKGVDLVLNSLAEEKLQASVRCLATHGRFLEIGKFDLGMAIFLKNVTFHGVLLDAFFNESSADWREVWALVQAGIRDGVVRPLKCTVFHGAQVEDAFRYMAQGKHIGKVVVQVLAEEPE 4w9n B 1.84 BS01 TCL B 1 F1766 L1780 F1791 F222 L231 F242 1.1.1.100,1.3.1.39,2.3.1.38,2.3.1.39,2.3.1.41,2.3.1.85,3.1.2.14,4.2.1.59 0016491 ic50=54.7uM remove_due_to_license_issue P49327 25301948 1905 HAFVSTLTRGDLSSIRWVCAQLCTVYYASLNFRDIMLATGKLSPDAIPGKWTSQDSLLGMEFSGRDASGKRVMGLVPAKGLATSVLLSPDFLWDVPSNWTLEEAASVPVVYSTAYYALVVRGRVRPGETLLIHSGSGGVGQAAIAIALSLGCRVFTTVGSAEKRAYLQARFPQLDSTSFANSSFEQHVLWHTGGKGVDLVLNSLAEEKLQASVRCLATHGRFLEIGKFDLLGMAIFLKNVTFHGVLLDAFFNESSADWREVWALVQAGIRDGVVRPLKCTVFHGAQVEDAFRYMAQGKHIGKVVVQVLAEE 4w9o A 1.27 BS01 3JQ A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 S118 F130 Y41 F51 D52 F61 G68 Q69 V70 I71 W74 Y97 S102 F114 Y57 F67 D68 I87 Y113 F130 Y41 F51 D52 I71 Y97 F114 5.2.1.8 0003755 remove_due_to_license_issue Q13451 25412894 201 TVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKG 4w9p A 1.5 BS01 3JR A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 S118 F130 Y39 F49 D50 F59 G66 Q67 V68 I69 W72 Y95 S100 F112 Y57 F67 D68 I87 Y113 F130 Y39 F49 D50 I69 Y95 F112 5.2.1.8 0003755 remove_due_to_license_issue Q13451 25412894 201 TEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKG 4w9q A 1.08 BS01 3JP A 1 Y57 F67 D68 F77 G84 Q85 V86 I87 W90 Y113 S118 K121 F130 Y45 F55 D56 F65 G72 Q73 V74 I75 W78 Y101 S106 K109 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 remove_due_to_license_issue Q13451 25412894 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4w9s A 1.8 BS03 3K1 A 1 K34 A37 I38 H41 E80 D108 E119 K134 K39 A42 I43 H46 E85 D113 E124 K139 3.1.-.- 0003723,0039694 ic50=0.15uM remove_due_to_license_issue P13166 25225968 304 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4w9w A 1.72 BS01 YDJ A 1 A77 Y132 C133 G136 N185 L187 C197 A39 Y94 C95 G98 N147 L149 C159 D180 K182 N185 D198 N208 T226 D142 K144 N147 D160 N170 T188 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9NSY1 26853940 401 VGVRVFAVGRHQVTLEESLAEGGFSTVFLVRTHGGIRCALKRMYVNNMPDLNVCKREITIMKELSGHKNIVGYLDCAVNSISDNVWEVLILMEYCRAGQVVNQMNKKLQTGFTEPEVLQIFCDTCEAVARLHQCKTPIIHRDLKVENILLNDGGNYVLCDFGSATNKFLNPQKDGVNVVEEEIKKYTTLSYRAPEMINLYGGKPITTKADIWALGCLLYKLCFFTLPFGESQVAICDGNFTIPDNSRYSRNIHCLIRFMLEPDPEHRPDIFQVSYFAFKFAAADCPVSNINNSSIPSALPEPMTAS 4w9w A 1.72 BS02 YDJ A 2 N289 Y313 F314 F318 N251 Y275 F276 F280 D180 K182 N185 D198 N208 T226 D142 K144 N147 D160 N170 T188 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9NSY1 26853940 402 VGVRVFAVGRHQVTLEESLAEGGFSTVFLVRTHGGIRCALKRMYVNNMPDLNVCKREITIMKELSGHKNIVGYLDCAVNSISDNVWEVLILMEYCRAGQVVNQMNKKLQTGFTEPEVLQIFCDTCEAVARLHQCKTPIIHRDLKVENILLNDGGNYVLCDFGSATNKFLNPQKDGVNVVEEEIKKYTTLSYRAPEMINLYGGKPITTKADIWALGCLLYKLCFFTLPFGESQVAICDGNFTIPDNSRYSRNIHCLIRFMLEPDPEHRPDIFQVSYFAFKFAAADCPVSNINNSSIPSALPEPMTAS 4w9x A 2.14 BS01 3JW A 1 A58 E59 G60 S63 A77 V109 M130 C133 Q137 E184 N185 L187 D198 A20 E21 G22 S25 A39 V71 M89 C92 Q96 E142 N143 L145 D156 D180 K182 N185 D198 N208 T226 D138 K140 N143 D156 N166 T184 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9NSY1 26853940 403 VGVRVFAVGRHQVTLEESLAEGGFSTVFLVRTHGGIRCALKRMYVNNMPDLNVCKREITIMKELSGHKNIVGYLDCAVNSISWEVLILMEYCRAGQVVNQMNKKQTGFTEPEVLQIFCDTCEAVARLHQCKTPIIHRDLKVENILLNDGGNYVLCDFGSATNKFLNPQKDGVNVVEEEIKKYTTLSYRAPEMINLYGGKPITTKADIWALGCLLYKLCFFTLPFGESQVAICDGNFTIPDNSRYSRNIHCLIRFMLEPDPEHRPDIFQVSYFAFKFAAADCPVSNINNSSIPSALPEPMT 4wa9 B 2.2 BS01 AXI B 1 Y253 V256 A269 K271 E316 F317 M318 G321 L370 A380 F382 Y21 V24 A37 K39 E84 F85 M86 G89 L138 A148 F150 D363 A365 R367 N368 D381 P402 D131 A133 R135 N136 D149 P170 2.7.10.2 0004672,0004713,0005524,0006468 Ki=3800pM remove_due_to_license_issue P00519 25686603 9000 DKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEK 4waf A 2.39 BS01 3K6 A 1 W780 M800 K802 Y836 I848 V850 V851 S854 M922 I932 D933 W743 M763 K765 Y799 I811 V813 V814 S817 M878 I888 D889 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue IC50=>10000nM P42336 25589927 1101 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRISSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIMFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLVHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTTKMDWIFHT 4wag A 3.407 BS01 3K7 A 1 I562 K564 E572 Y598 I610 P612 V613 L678 D689 I226 K228 E236 Y262 I274 P276 V277 L342 D353 2.7.1.67 0016301,0046854 remove_due_to_license_issue Q9UBF8 25897704 801 LLRLFESKLFDISMAISYLYNSKEPGVQAYIGNRLFCFRNEDVDFYLPQLLNMYIHMDEDVGDAIKPYIVHRCRQSINFSLQCALLLGAYSSDMSFSSPVRLAPEREFIKSLMAIGKRLATLPTKEQKTQRLISELSLLNHKLPARVWLPTAGFDHHVVRVPHTQAVVLNSKDKAPYLIYVEVLECENFDTTSVPARIPEWQEKVRRIREGSPYGHLPNWRLLSVIVKCGDDLRQELLAFQVLKQLQSIWEQERVPLWIKPYKILVISADSGMIEPVVNAVSIHQVKKQSQLSLLDYFLQEHGSYTTEAFLSAQRNFVQSCAGYCLVCYLLQVKDRHNGNILLDAEGHIIHIDFGFILSSSPRNLGFETSAFKLTTEFVDVMGGLDGDMFNYYKMLMLQGLIAARKHMDKVVQIVEIMQQGSQLPCFHGSSTIRNLKERFHMSMTEEQLQLLVEQMVDGSMR 4wbg A 1.9 BS01 AZR A 1 S65 Q121 Y151 Y223 I292 T313 G314 S315 S59 Q115 Y145 Y215 I284 T301 G302 S303 S65 K68 M107 E109 F122 Y151 G157 E272 K312 S315 S59 K62 M101 E103 F116 Y145 G151 E264 K300 S303 3.5.2.6 0008800,0016787,0017001,0030288,0046677,0046872 remove_due_to_license_issue Q51578 26055361 1001 DPLRPVVDASIQPLLKEHRIPGMAVAVLKDGKAHYFNYGVANRESGASVSEQTLFEIGSVSKTLTATLGAYAVVKGAMQLDDKASRHAPWLKGSVFDSITMGELATYSAGGLPLQFPEEVDSSEKMRAYYRQWAPVYSPGSHRQYSNPSIGLFGHLAASSLKQPFAQLMEQTLLPGLGMHHTYVNVPKQAMASYAYGYSKEDKPIRVGMLADEAYGIKTSSADLLAFVKANIGGVDDKALQQAISLTHKGHYSVGGMTQGLGWESYAYPVTEQTLLAGNSAKVILEANPTAAPRQVLFNKTGSSNGFGAYVAFVPARGIGIVMLANRNYPIPARVKAAHAILAQLAG 4wbo A 2.81 BS01 ANW A 1 L193 A214 M267 L321 A478 L166 A187 M240 L294 A451 D314 K316 E318 N319 D332 A341 T352 D287 K289 E291 N292 D305 A314 T325 2.7.11.14 0001750,0004672,0004674,0004703,0005515,0005524,0005737,0006468,0007165,0007601,0009966,0016020,0022400,0042995,0046777,0050254,0097381 remove_due_to_license_issue P28327 25340299 601 PASRDRKYLARLKLPPLSKCEALRESLDLGFEGMCLEQPIGKRLFQQFLRTHEQHGPALQLWKDIEDYDTADDALRPQKAQALRAAYLEPQAQLFCSFLDAETVARARAGAGDGLFQPLLRAVLAHLGQAPFQEFLDSLYFLRFLQWKWLEAQPMGEDWFLDFRVLGRGGFGEVFACQMKATGKLYACKKLNKKRLKKRKGYQGAMVEKKILAKVHSRFIVSLAYAFETKTDLCLVMTIMNGGDIRYHIYNVDEDNPGFQEPRAIFYTAQIVSGLEHLHQRNIIYRDLKPENVLLDDDGNVRISDLGLAVELKAGQTKTKGYAGTPGFMAPELLLGEEYDFSVDYFALGVTLYEMIAARGPFRARGEKVENKELKQRVLEQAVTYPDKFSPASKDFCEALLQKDPEKRLGFRDGSCDGLRTHPLFRDISWRQLEAGMLTPPFVPDSRTVYAKNIKGVAFEKADTEFFQEFASGTCPIPWQEEMIETGVFGDLNVWRP 4wcf A 1.93 BS02 3KN A 1 S95 F97 Y174 P210 S94 F96 Y155 P191 R14 D161 Y174 K178 R13 D142 Y155 K159 ? 0000166,0016491,0047040 remove_due_to_license_issue O76290 28983525 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 4wcu A 2.35 BS01 3KQ A 1 M273 D318 I336 F340 M357 Q369 F372 F432 Q433 M184 D229 I247 F251 M268 Q280 F283 F326 Q327 3.1.4.53 0004114,0007165,0008081 ic50=3nM remove_due_to_license_issue IC50=3.0nM Q08499 24984230 500 DVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPTEKFQFEL 4wet A 1.63 BS01 WEF A 1 H32 L40 Q164 T168 M171 F174 H31 L39 Q163 T167 M170 F173 1.8.4.2 0015036,0016491,0042597,0046872 Kd=444uM remove_due_to_license_issue A0A0H2UL03 25556635 201 QYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 4wey A 1.55 BS01 EG6 B 1 H32 F36 T168 M171 F174 H32 F36 T168 M171 F174 1.8.4.2 0015036,0016491,0042597,0046872 remove_due_to_license_issue A0A0H2UL03 25556635 202 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 4wf2 A 2.31 BS01 BTX A 1 S89 T90 Q112 R116 G117 R118 R121 K122 W123 F124 Y132 K183 G186 I187 A205 G206 N208 S87 T88 Q110 R114 G115 R116 R119 K120 W121 F122 Y130 K181 G184 I185 A199 G200 N202 R118 K183 R317 R116 K181 R301 6.3.4.15 0000976,0003676,0003677,0004077,0005515,0005524,0005737,0006355,0006768,0009102,0009374,0016874,0017053,0036211,0042803 remove_due_to_license_issue Ki=87nM, Kd=1.5nM P06709 25746672 501 DNTVPLKLIALLANGEFHSGEQLGETLGMSRAAINKHIQTLRDWGVDVFTVPGKGYSLPEPIQLLNAKQILGQLDGGSVAVLPVIDSTNQYLLDRIGELKSGDACIAEYQQAGRGRRGRKWFSPFGANLYLSMFWRLEQAPAAAIGLSLVIGIVMAEVLRKLGADKVRVKWPNDLYLQDRKLAGILVELTDAAQIVIGAGINMAMGWITLQEAGINLDRNTLAAMLIRELRAALELFEQEGLAPYLSRWEKLDNFINRPVKLIIGDKEIFGISRGIDKQGALLLEQDGIIKPWMGGEISLRSAE 4wf4 B 1.7 BS01 WF4 B 1 H32 L40 T168 M171 F174 H32 L40 T168 M171 F174 1.8.4.2 0015036,0016491,0042597,0046872 Kd=777uM remove_due_to_license_issue A0A0H2UL03 25556635 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 4wf6 A 2.6521 BS02 407 A 1 S655 K656 G657 L658 V675 L677 H686 E687 H690 Y728 E735 E739 S382 K383 G384 L385 V402 L404 H413 E414 H417 Y455 E462 E466 H686 E687 H690 Y728 E735 H413 E414 H417 Y455 E462 3.4.24.83 0008237 remove_due_to_license_issue IC50=1600nM P15917 26492514 802 SRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEEEKELLNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4wgi A 1.85 BS03 3M6 A 1 A227 F228 M231 F254 R263 I264 T266 L267 F270 K302 A419 F420 M423 F446 R455 I456 T458 L459 F462 K494 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0042981,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q07820 25516789 402 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYEDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGAGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4wh7 A 1.62 BS01 8H8 A 1 L398 R485 R488 L25 R112 R115 3.1.3.48 0004725,0006470,1902751 ic50>5mM remove_due_to_license_issue P30305 25423142 607 DHRELIGDYSKAFLLQTVDGKHQDLKYISPETMVALLTGKFSNIVDKFVIVDCRYPYEYEGGHIKTAVNLPLERDAESFLLKSPIAPCSLDKRVILIFHSEFSSERGPRMCRFIRERDRAVNDYPSLYYPEMYILKGGYKEFFPQHPNFCEPQDYRPMNHEAFKDELKTFRLKTRSWA 4wh9 A 1.5 BS01 3M8 A 1 D397 L398 C484 R485 R488 R492 D23 L24 C110 R111 R114 R118 3.1.3.48 0004725,0006470,1902751 ic50=2.2mM remove_due_to_license_issue P30305 25423142 601 HRELIGDYSKAFLLQTVDGKHQDLKYISPETMVALLTGKFSNIVDKFVIVDCRYPYEYEGGHIKTAVNLPLERDAESFLLKSPIAPCSLDKRVILIFHSEFSSERGPRMCRFIRERDRAVNDYPSLYYPEMYILKGGYKEFFPQHPNFCEPQDYRPMNHEAFKDELKTFRLKTRSWA 4whq A 1.78 BS01 3N8 A 1 R167 E168 R167 E168 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 25548185 302 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 4whr A 1.58 BS01 3N8 A 1 R167 E168 R167 E168 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 25548185 301 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 4whs A 1.35 BS01 3N8 A 1 R167 E168 R167 E168 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 25548185 301 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 4whs A 1.35 BS02 3N8 B 1 P15 Y16 P15 Y16 Y79 V114 M122 H125 N127 Y79 V114 M122 H125 N127 1.13.11.3 0003824,0005506,0008199,0009056,0016702,0018578,0042952,0051213 remove_due_to_license_issue P00436 25548185 603 PIELLPETPSQTAGPYVHIGLALEAAGNPTRDQEIWNRLAKPDAPGEHILLLGQVYDGNGHLVRDSFLEVWQADANGEYQDAYNLENAFNSFGRTATTFDAGEWTLHTVKPGVVNNAAGVPMAPHINISLFARGINIHLHTRLYFDDEAQANAKCPVLNLIEQPQRRETLIAKRCEVDGKTAYRFDIRIQGEGETVFFDF 4whz A 1.79 BS01 3NL A 1 I70 A91 K93 I124 L144 M146 L148 M149 D150 A151 L206 I26 A47 K49 I80 L100 M102 L104 M105 D106 A107 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T177 2.7.11.24 0004672,0004707,0005524,0006468 ic50<1nM remove_due_to_license_issue IC50=<1.000000nM P53779 25393557 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPREHTIEEWKELIYKEVMN 4wi1 A 1.65 BS01 3O6 A 1 Y266 A291 R403 E404 I474 T513 I516 G517 M521 Y25 A47 R107 E108 I178 T217 I220 G221 M225 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=5uM remove_due_to_license_issue Q8I5R7 27798837 801 AHHHHHHSNILGITSKKIENFSDWYTQVIVKSELIEYYGCYILRPAAYYIWECVQAFFNKEIKKLNVENSYFPLFVTSETIMYSVFPKWIRSYRDLPLKLNQWNTVREFLWQEGHTAHKNEEEAVKLVFDILDLYRRWYEEYLAVPIIKGIKSEGEKFGGANFTSTAEAFISENGRAIQAATSHYLGTNFAKMFKIEFEDENEVKQYVHQTSWGCTTRSIGIMIMTHGDDKGLVLPPNVSKYKVVIVPIFYKTTDENAIHSYCKDIEKILKNAQINCVYDDRASYSPGYKFNHWELRGIPIRIEVGPKDLQNNSCVIVRRDNNEKCNVKKESVLLETQQMLVDIHKNLFLKAKKKLDDSIVQVTSFSEVMNALNKKKMVLAPWCEDIATEEEIKKETQRLSSGAMKPLCIPLDQPPMPPNMKCFWSGKPAKRWCLFGRSY 4wiv A 1.56 BS01 3P2 A 1 W81 F83 V87 L92 N140 I146 W40 F42 V46 L51 N99 I105 ? Kd=550nM remove_due_to_license_issue IC50=637nM, Kd=550nM O60885 25314271 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4wk1 A 1.98 BS01 2BA A 1 I7 G34 F36 L37 T97 F99 I15 G42 F44 L45 T80 F82 ? 0046872 Kd=109nM remove_due_to_license_issue A0A0H2WXZ7 25435171 201 GLVPRGSHMKMIIAIVQDQDSQELADQLVKNNFRATKLATTGGFLRAGNTTFLCGVNDDRVDEILSVINQTCGNEVGGATVFVMPVDAFHQF 4wk7 A 1.24 BS05 3PQ A 1 T329 L330 G331 F357 H361 E362 H371 V390 A392 P393 V394 M395 T108 L109 G110 F136 H140 E141 H150 V167 A169 P170 V171 M172 3.4.24.82 0004222,0006508,0008237 ic50=74nM remove_due_to_license_issue IC50=74nM O75173 25415648 505 SRFVETLVVADDKMAAFHGAGLKRYLLTVMAAAAKAFKHPSIRNPVSLVVTRLVILGPQVGPSAAQTLRSFCAWQRGLNTPEDSDPDHFDTAILFTRQDLCGVSTCDTLGMADVGTVCDPARSCAIVEDDGLQSAFTAAHELGHVFNMLHDNSKPCISLNGPLSRHVMAPVMAHVDPEEPWSPCSARFITDFLDNGYGHCLLDKPEAPL 4wkb A 1.37 BS01 TDI A 1 I50 S76 A77 G78 F152 V153 E173 M174 E175 D198 F208 I50 S76 A77 G78 F152 V153 E173 M174 E175 D198 F208 3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509 Ki=2.7pM remove_due_to_license_issue A5F5R2 25806409 301 MKIGIIGAMQQEVAILKDLIEDVQEVNQAGCTFYSGQIQGVDVVLLQSGIGKVSAALGTALLISQYAPDVVINTGSAGGFDASLNVGDVVISSEVRHHDADVTAFGYEIGQMAGQPAAFKADEKLMTVAEQALAQLPNTHAVRGLICTGDAFVCTAERQQFIRQHFPSVVAVEMEASAIAQTCHQFKVPFVVVRAISDVADKESPLSFEEFLPLAAKSSSAMVLKMVELLKENLYFQ 4wkb B 1.37 BS01 TDI B 1 I50 S76 A77 G78 F152 V153 E173 M174 E175 D198 F208 I50 S76 A77 G78 F152 V153 E173 M174 E175 D198 F208 3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509 Ki=2.7pM remove_due_to_license_issue A5F5R2 25806409 301 MKIGIIGAMQQEVAILKDLIEDVQEVNQAGCTFYSGQIQGVDVVLLQSGIGKVSAALGTALLISQYAPDVVINTGSAGGFDASLNVGDVVISSEVRHHDADVTAFGYEIGQMAGQPAAFKADEKLMTVAEQALAQLPNTHAVRGLICTGDAFVCTAERQQFIRQHFPSVVAVEMEASAIAQTCHQFKVPFVVVRAISDVADKESPLSFEEFLPLAAKSSSAMVLKMVELLKENLYFQ 4wkc A 1.64 BS01 BIG A 1 M9 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 M9 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0046124 Ki=0.21pM remove_due_to_license_issue A7ZHQ1 25806409 301 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAHG 4wke A 1.62 BS05 3PU A 1 T329 L330 G331 M332 H361 E362 H371 V390 A392 P393 V394 M395 T110 L111 G112 M113 H142 E143 H152 V169 A171 P172 V173 M174 3.4.24.82 0004222,0006508,0008237 ic50=8nM remove_due_to_license_issue IC50=8.0nM O75173 25415648 508 LSRFVETLVVADDKMAAFHGAGLKRYLLTVMAAAAKAFKHPSIRNPVSLVVTRLVILEGPQVGPSAAQTLRSFCAWQRGLNTPEDSDPDHFDTAILFTRQDLCGVSTCDTLGMADVGTVCDPARSCAIVEDDGLQSAFTAAHELGHVFNMLHDNSKPCISLNGPLSRHVMAPVMAHVDPEEPWSPCSARFITDFLDNGYGHCLLDKPEAPLHLP 4wki A 1.6 BS05 3PW A 1 T329 L330 G331 H361 E362 H371 V390 A392 P393 V394 M395 T110 L111 G112 H142 E143 H152 V169 A171 P172 V173 M174 3.4.24.82 0004222,0006508,0008237 ic50=5nM remove_due_to_license_issue IC50=3.0nM O75173 25415648 506 SLSRFVETLVVADDKMAAFHGAGLKRYLLTVMAAAAKAFKHPSIRNPVSLVVTRLVILGPQVGPSAAQTLRSFCAWQRGLNTPEDSDPDHFDTAILFTRQDLCGVSTCDTLGMADVGTVCDPARSCAIVEDDGLQSAFTAAHELGHVFNMLHDNSKPCISLNGPLSRHVMAPVMAHVDPEEPWSPCSARFITDFLDNGYGHCLLDKPEAPLHLP 4wkn A 2.0 BS01 TDI A 1 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=0.19nM remove_due_to_license_issue Q9ZMY2 26494017 301 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4wkp A 1.58 BS01 3QA A 1 I52 A79 G80 F153 V154 E173 M174 E175 D198 A200 F208 I52 A79 G80 F153 V154 E173 M174 E175 D198 A200 F208 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q9ZMY2 26494017 301 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4wkp A 1.58 BS02 3QA B 1 F107 H109 P115 F107 H109 P115 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q9ZMY2 26494017 301 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4wkp B 1.58 BS01 3QA A 1 F107 H109 P115 F107 H109 P115 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q9ZMY2 26494017 301 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4wkp B 1.58 BS02 3QA B 1 I52 A79 G80 F153 V154 E173 M174 E175 D198 F208 I52 A79 G80 F153 V154 E173 M174 E175 D198 F208 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q9ZMY2 26494017 301 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4wkt C 1.782 BS01 BUB C 1 S217 H239 T285 V286 N485 S1 H23 T69 V70 N269 S217 S1 3.5.1.97 0016787,0017000 Ki=0.00055M remove_due_to_license_issue Q9I194 25290020 801 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIREAA 4wku B 2.0 BS01 3QJ B 1 S217 H239 F240 T285 V286 S1 H23 F24 T69 V70 S217 H239 V286 N485 T695 S1 H23 V70 N269 T479 3.5.1.97 0016787,0017000 remove_due_to_license_issue Q9I194 25290020 801 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIREAA 4wkv C 2.1434 BS01 3QK C 1 S217 H239 F240 L266 T285 V286 S1 H23 F24 L50 T69 V70 S217 S1 3.5.1.97 0016787,0017000 remove_due_to_license_issue Q9I194 25290020 801 SNAIAVGSERSADGKGMLLANPHFPWNGAMRFYQMHLTIPGRLDVMGASLPGLPVVNIGFSRHLAWTHTVDTSSHFTLYRLALDPKDPRRYLVDGRSLPLEEKSVAIEVRGADGKLSRVEHKVYQSIYGPLVVWPGKLDWNRSEAYALRDANLENTRVLQQWYSINQASDVADLRRRVEALQGIPWVNTLAADEQGNALYMNQSVVPYLKPELIPACAIPQLVAEGLPALQGQDSRCAWSRDPAAAQAGITPAAQLPVLLRRDFVQNSNDSAWLTNPASPLQGFSPLVSQEKPIGPRARYALSRLQGKQPLEAKTLEEMVTANHVFSADQVLPDLLRLCRDNQGEKSLARACAALAQWDRGANLDSGSGFVYFQRFMQRFAELDGAWKEPFDAQRPLDTPQGIALDRPQVATQVRQALADAAAEVEKSGIPDGARWGDLQVSTRGQERIAIPGGDGHFGVYNAIQSVRKGDHLEVVGGTSYIQLVTFPEEGPKARGLLAFSQSSDPRSPHYRDQTELFSRQQWQTLPFSDRQIDADPQLQRLSIREAA 4wlb A 1.702 BS02 3QQ A 1 Q286 L287 C320 H323 M365 R367 A368 F378 I400 H479 Q27 L28 C61 H64 M106 R108 A109 F119 I141 H220 ? 0003677,0004879,0005634,0006355 ic50=0.18uM remove_due_to_license_issue IC50=180nM, EC50=520nM P51449 25453817 601 GSAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 4wm9 A 2.4 BS01 NXL A 1 S81 W115 S128 L168 S219 G220 W221 M223 R261 S51 W85 S98 L138 S189 G190 W191 M193 R229 S81 K84 S128 Y133 W167 W221 S51 K54 S98 Y103 W137 W191 ? 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 25406838 301 FHISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 4wmc A 2.3 BS01 NXL A 1 S70 S118 V120 T209 G210 Y211 R250 S42 S90 V92 T181 G182 Y183 R222 S70 K73 S118 Y123 W157 Y211 S42 K45 S90 Y95 W129 Y183 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 remove_due_to_license_issue Q6XEC0 25406838 301 EWQENKSWNAHFQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 4wmu A 1.55 BS03 19H A 1 A227 F228 L246 M250 F254 R263 T266 L267 F270 G271 I294 A423 F424 L442 M446 F450 R459 T462 L463 F466 G467 I490 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 Kd=0.18uM remove_due_to_license_issue P0AEX9,Q07820 25909780 402 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 4wmv A 2.4 BS03 3R4 A 1 F228 M231 R263 T266 L267 F270 F421 M424 R456 T459 L460 F463 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 Kd=93uM remove_due_to_license_issue P0AEX9,Q07820 25909780 404 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4wmx A 2.0 BS03 3R7 A 1 F228 M231 M250 V253 L267 F270 F423 M426 M445 V448 L462 F465 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 Kd=14.1uM remove_due_to_license_issue P0AEX9,Q07820 25909780 402 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 4wmy A 1.601 BS04 3S6 A 1 N260 H263 E274 Y297 N230 H233 E244 Y267 ? 0001934,0005509,0005515,0005576,0005615,0005886,0009624,0030246,0031526,0042802,0043235,0045121,0046326,0046872,0070062,0070207,0070492,0098552 Kd=85nM remove_due_to_license_issue Q8WWA0 26148048 404 CSSSPSLPRSCKEIKDECPSAFDGLYFLRTENGVIYQTFCDMTSGGGGWTLVASVHENDMRGKCTVGDRWSSQQGSKAVYPEGDGNWANYNTFGSAEAATSDDYKNPGYYDIQAKDLGIWHVPNKSPMQHWRNSSLLRYRTDTGFLQTLGHNLFGIYQKYPVKYGEGKCWTDNGPVIPVVYDFGDAQKTASYYSPYGQREFTAGFVQFRVFNNERAANALCAGMRVTGCNTEHHCIGGGGYFPEASPQQCGDFSGFDWSGYGTHVGYSSSREITEAAVLLFYR 4wn0 A 2.2 BS05 G3P A 1 N289 H292 E303 W326 N224 H227 E238 W261 ? 0005509,0005576,0005615,0030133,0030141,0030246,0031410,0034214,0046872,0070492 ic50=0.6mM remove_due_to_license_issue Q5PPM0 26755729 409 GYRSCNEIKSSDSRAPDGIYTLATEDGESYQTFCDMTTNGGGWTLVASVHENNMFGKCTVGDRWSTQQGNMLQNPEGDGNWANYATFGLPEGATSDDYKNPGYYDIEAKNLALWHVPNKTPMVMWRNSSILRYRTQNGFLTEEGGNLFELYKKYPVKYDIGKCLADNGPAVPVVYDLGSAEKTASLYSPNGRSEFTPGFVQFRAVNSERATLALCAGVKVKGCNVEHHCIGGGGYIPEGSPRQCGDFAALDWDGYGTNLGWSASKQIIEAAVMLFYR 4wn1 A 3.13 BS02 3SJ A 1 Y524 L635 L675 Y693 F696 M713 E721 V722 Q726 F729 Y78 L189 L229 Y247 F250 M267 E275 V276 Q280 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Q9Y233 25515954 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 4wnk A 2.42 BS01 453 A 1 G193 K194 G195 F197 G198 V200 A213 K215 M230 I265 M266 E315 N316 L318 D329 G170 K171 G172 F174 G175 V177 A190 K192 M207 I242 M243 E292 N293 L295 D306 D311 K313 E315 N316 D329 E338 T348 D288 K290 E292 N293 D306 E315 T325 2.7.11.16 0004672,0004674,0004703,0005524,0005634,0005737,0005886,0006468,0006915,0007165,0008289,0009966,0016055,0043066,0046777 ic50=0.38uM remove_due_to_license_issue P43249 26032411 701 KGKSKKWKEILKFPHINQCEDLRRTIDRDYCSLCDKQPVGRLLFRQFCETRPGLESYIQFLDSVAEYEVTPDEKLGEKGKEIMTKYLTPKSPVFITQVGRDLVSQTEEKLLQKPCKELFSACVQSVHDYLRGEPFHEYLDSMYFDRFLQWKWLERQPVTKNTFRQYRVLGKGGFGEVCACQVRATGKMYACKRLEKKRIKKRKGESMALNEKQILEKVNSRFVVNLAYAYETKDALCLVLTIMNGGDLKFHIYNMGNPGFEEERALFYAAEILCGLEDLHHENIVYRDLKPENILLDDYGHIRISDLGLAVKIPEGDLIRGRVGTVGYMAPEVLNNQRYGLSPDYWGLGCLIYEMIEGQSPFRGRKEKVKREEVDRRVLETEEVYSHKFSEEAKSICKMLLTKDAKQRLGCQEEGAAEVKRHPFFRNMNFKRLEAGMLDPPFVPDPRAVYHTDDDFYSKFSTGSVPIPWQSEMIETECFKELNVFGPHGTLSPDLNRSH 4wnm A 2.5 BS01 3RT A 1 L377 A400 M448 M450 A451 G454 P455 K458 N499 L501 S511 D512 L18 A41 M85 M87 A88 G91 P92 K95 N136 L138 S148 D149 D494 A496 R498 N499 D512 K533 D131 A133 R135 N136 D149 K170 2.7.10.2 0004672,0004713,0005524,0006468 Ki=18nM remove_due_to_license_issue P43405 26756335 701 VYEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNH 4wno A 1.56 BS01 3RF A 1 I22 V30 A44 M92 E93 Y94 C95 G98 L145 D165 I15 V23 A37 M85 E86 Y87 C88 G91 L138 D158 D138 K140 Q142 N143 D165 S184 D131 K133 Q135 N136 D158 S177 2.7.11.1 0004672,0004674,0005524,0006468,0010506 ic50=160nM remove_due_to_license_issue O75385 25551253 401 TETVGKFEFSRKDLIGHGAFAVVFKGRHRAAHDLEVAVKCINKKNLAKSQTLLGKEIKILKELKHENIVALYDFQEMANSVYLVMEYCNGGDLADYLHAMRTLSEDTIRLFLQQIAGAMRLLHSKGIIHRDLKPQNILLSNPAGRRANPNSIRVKIADFGFARYLQSNMMAATLCGSPMYMAPEVIMSQHYDGKADLWSIGTIVYQCLTGKAPFQASSPQDLRLFYEKNKTLVPTIPRETSAPLRQLLLALLQRNHKDRMDFDEFFHHPFLDA 4wnp A 1.88 BS01 3RJ A 1 I22 A44 M92 E93 Y94 C95 G98 Q142 N143 L145 I16 A38 M86 E87 Y88 C89 G92 Q136 N137 L139 D138 K140 Q142 N143 D165 S184 D132 K134 Q136 N137 D159 S178 2.7.11.1 0004672,0004674,0005524,0006468,0010506 ic50=8nM remove_due_to_license_issue O75385 25551253 303 GTETVGKFEFSRKDLIGHGAFAVVFKGRHRAAHDLEVAVKCINKKNLAKSQTLLGKEIKILKELKHENIVALYDFQEMANSVYLVMEYCNGGDLADYLHAMRTLSEDTIRLFLQQIAGAMRLLHSKGIIHRDLKPQNILLSNPAGRRANPNSIRVKIADFGFARYLQSNMMAATLCGSPMYMAPEVIMSQHYDGKADLWSIGTIVYQCLTGKAPFQASSPQDLRLFYEKNKTLVPTIPRETSAPLRQLLLALLQRNHKDRMDFDEFFHHPFLDA 4wop A 2.393 BS01 CTP A 1 G12 V13 G14 K15 T16 V17 E108 G169 G199 A200 G12 V13 G14 K15 T16 V17 E108 G169 G199 A200 T11 G12 K15 T16 K37 T41 G54 E108 T11 G12 K15 T16 K37 T41 G54 E108 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 Kd=17.2uM remove_due_to_license_issue P9WPQ5 25801336 301 ATILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 4wov A 1.8 BS01 3SM A 1 L595 G596 V640 Y689 V690 G693 P694 L741 L16 G17 V35 Y84 V85 G88 P89 L136 N734 R738 N739 D759 N129 R133 N134 D154 2.7.10.2 0004672,0005524,0006468 ic50=72nM remove_due_to_license_issue P29597 25762719 901 SFHRVDQKEITQLSHLGQGTRTNVYEGRLRELRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLTRL 4wp7 A 1.8 BS01 3SR A 1 G125 T129 F171 G294 Y297 C302 I304 G458 V460 A462 G118 T122 F164 G287 Y290 C295 I297 G451 V453 A455 N170 K193 E269 C303 E400 E477 N163 K186 E262 C296 E393 E470 1.2.1.19,1.2.1.28,1.2.1.3,1.2.1.36 0000166,0001523,0001758,0004029,0005096,0005497,0005515,0005737,0005829,0006081,0006629,0009449,0016491,0016620,0018479,0019145,0030392,0030424,0036438,0042572,0042995,0045202,0051287,0070062,0106373,0110095,0120163 ic50=0.8uM remove_due_to_license_issue IC50=800nM, Ki=720nM P00352 25634381 602 DLPVLLTDLKIQYTKIFINNEWHDSVSGKKFPVFNPATEEELCQVEEGDKEDVDKAVKAARQAFQIGSPWRTMDASERGRLLYKLADLIERDRLLLATMESMNGGKLYSNAYLSDLAGCIKTLRYCAGWADKIQGRTIPIDGNFFTYTRHEPIGVCGQIIPWNFPLVMLIWKIGPALSCGNTVVVKPAEQTPLTALHVASLIKEAGFPPGVVNIVPGYGPTAGAAISSHMDIDKVAFTGSTEVGKLIKEAAGKSNLKRVTLELGGKSPCIVLADADLDNAVEFAHHGVFYHQGQCCIAASRIFVEESIYDEFVRRSVERAKKYILGNPLTPGVTQGPQIDKEQYDKILDLIESGKKEGAKLECGGGPWGNKGYFVQPTVFSNVTDEMRIAKEEIFGPVQQIMKFKSLDDVIKRANNTFYGLSAGVFTKDIDKAITISSALQAGTVWVNCYGVVSAQCPFGGFKMSGNGRELGEYGFHEYTEVKTVTVKISQKNS 4wpf A 2.202 BS02 3SN A 1 Q286 L287 W317 C320 L324 A368 F378 L391 Q23 L24 W54 C57 L61 A105 F115 L128 ? 0003677,0004879,0005634,0006355 ic50=0.25uM remove_due_to_license_issue EC50=69nM, IC50=249nM P51449 25815138 601 YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTE 4wpn A 1.95 BS01 3ST A 1 F171 H293 G294 Y297 C302 I304 G458 V460 F164 H286 G287 Y290 C295 I297 G451 V453 N170 K193 E269 C303 E400 E477 N163 K186 E262 C296 E393 E470 1.2.1.19,1.2.1.28,1.2.1.3,1.2.1.36 0000166,0001523,0001758,0004029,0005096,0005497,0005515,0005737,0005829,0006081,0006629,0009449,0016491,0016620,0018479,0019145,0030392,0030424,0036438,0042572,0042995,0045202,0051287,0070062,0106373,0110095,0120163 ic50=0.21uM remove_due_to_license_issue IC50=210nM, Ki=96nM P00352 25634381 601 DLPVLLTDLKIQYTKIFINNEWHDSVSGKKFPVFNPATEEELCQVEEGDKEDVDKAVKAARQAFQIGSPWRTMDASERGRLLYKLADLIERDRLLLATMESMNGGKLYSNAYLNDLAGCIKTLRYCAGWADKIQGRTIPIDGNFFTYTRHEPIGVCGQIIPWNFPLVMLIWKIGPALSCGNTVVVKPAEQTPLTALHVASLIKEAGFPPGVVNIVPGYGPTAGAAISSHMDIDKVAFTGSTEVGKLIKEAAGKSNLKRVTLELGGKSPCIVLADADLDNAVEFAHHGVFYHQGQCCIAASRIFVEESIYDEFVRRSVERAKKYILGNPLTPGVTQGPQIDKEQYDKILDLIESGKKEGAKLECGGGPWGNKGYFVQPTVFSNVTDEMRIAKEEIFGPVQQIMKFKSLDDVIKRANNTFYGLSAGVFTKDIDKAITISSALQAGTVWVNCYGVVSAQCPFGGFKMSGNGRELGEYGFHEYTEVKTVTVKISQKNS 4wq2 A 1.64 BS01 3SU A 1 L124 V127 H131 Q175 L29 V32 H36 Q80 F164 G187 I189 F69 G92 I94 ? 0005509 ic50=0.5uM remove_due_to_license_issue P04632 28757975 301 EEVRQFRRLFAQLAGDDMEVSATELMNILNKVVTRHPDLKTDGFGIDTCRSMVAVMDSDTTGKLGFEEFKYLWNNIKRWQAIYKQFDTDRSGTICSSELPGAFEAAGFHLNEHLYNMIIRRYSDESGNMDFDNFISCLVRLDAMFRAFKSLDKDGTGQIQVNIQEWLQLTMYS 4wq3 A 1.79 BS05 3SU A 1 L104 I123 V127 R130 H131 F164 W168 L9 I28 V32 R35 H36 F69 W73 F164 G187 I189 F69 G92 I94 ? 0005509 ic50=0.1uM remove_due_to_license_issue P04632 28757975 305 EEVRQFRRLFAQLAGDDMEVSATELMNILNKVVTRHPDLKTDGFGIDTCRSMVAVMDSDTTGKLGFEEFKYLWNNIKRWQAIYKQFDTDRSGTICSSELPGAFEAAGFHLNEHLYNMIIRRYSDESGNMDFDNFISCLVRLDAMFRAFKSLDKDGTGQIQVNIQEWLQLTMYS 4wq3 A 1.79 BS06 3SU A 2 L124 V127 W168 K172 Q175 L29 V32 W73 K77 Q80 F164 G187 I189 F69 G92 I94 ? 0005509 ic50=0.1uM remove_due_to_license_issue P04632 28757975 306 EEVRQFRRLFAQLAGDDMEVSATELMNILNKVVTRHPDLKTDGFGIDTCRSMVAVMDSDTTGKLGFEEFKYLWNNIKRWQAIYKQFDTDRSGTICSSELPGAFEAAGFHLNEHLYNMIIRRYSDESGNMDFDNFISCLVRLDAMFRAFKSLDKDGTGQIQVNIQEWLQLTMYS 4wr7 A 1.5 BS02 3TV A 1 F91 H94 H96 H119 A135 L198 T199 H200 F89 H92 H94 H117 A133 L196 T197 H198 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T197 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=0.002nM remove_due_to_license_issue Kd=0.033nM P00915 26079542 302 PDWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 4wr8 B 2.6 BS01 3TX C 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Ki=590nM, Kd=260nM P14174 25697265 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4wr8 C 2.6 BS01 3TX C 1 P1 M2 K32 P33 Y36 H62 I64 V106 F113 P1 M2 K32 P33 Y36 H62 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Ki=590nM, Kd=260nM P14174 25697265 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4wrb A 1.81 BS01 3TW A 1 P1 M2 K32 P33 Y36 S63 I64 V106 F113 P1 M2 K32 P33 Y36 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=0.65uM remove_due_to_license_issue Ki=570nM P14174 25697265 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4wrb C 1.81 BS01 3TW A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Ki=570nM P14174 25697265 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 4wri A 1.4 BS01 OKA A 1 R44 F48 M58 R61 H65 S107 S108 T110 L131 M150 Q167 V184 R185 R41 F45 M55 R58 H62 S104 S105 T107 L128 M147 Q164 V181 R182 ? remove_due_to_license_issue Q2MHR1 25965326 201 LKEPSAHWCRKMRTVFRPWDVEGGSKGYVTEEVFKDGVQRRLEKFPELAPTKDKMYERSHRHWVNHCNLGVKMPEGYRLTESQYVQNAWLLIHSPDFEASLKESSQTFWEGIDREKKGYITKEEATKLGIRVTKDPNLKSTGIFEAMDEKNTGRITFEDTLKAQLFFFTDQDNTTHPFNYVRGALVD 4wrs A 2.2 BS01 3U1 A 1 L44 G45 F49 A65 E121 R122 V126 D128 E171 L174 I185 L12 G13 F17 A33 E89 R90 V94 D96 E139 L142 I153 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.4nM remove_due_to_license_issue IC50=0.400000nM P11309 25597005 403 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4wsj A 1.64 BS01 3U3 A 1 H66 E87 W88 H135 H136 Y178 D229 R262 W316 H32 E53 W54 H101 H102 Y144 D195 R228 W282 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A3I4 29142681 503 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAK 4wsk A 1.92 BS01 3U2 A 1 H66 E87 W88 H135 H136 Y178 D229 R262 E288 H32 E53 W54 H101 H102 Y144 D195 R228 E254 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 remove_due_to_license_issue Q8A3I4 29142681 503 EIPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAKGTKSIY 4wsy A 2.3 BS01 3U5 A 1 L44 F49 A65 E121 R122 V126 L174 I185 D186 L12 F17 A33 E89 R90 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.017uM remove_due_to_license_issue P11309 25616902 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4wt2 A 1.42 BS01 3UD A 1 V14 L54 I61 M62 V93 K94 H96 I99 Y100 V9 L49 I56 M57 V88 K89 H91 I94 Y95 2.3.2.27 0005634,0043066,0051726 Kd=38pM remove_due_to_license_issue IC50=0.600000nM, Kd=257nM Q00987 25384157 201 MSVPTDGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4wt6 A 2.3 BS01 3U6 A 1 G45 F49 A65 E121 V126 L174 I185 D186 G13 F17 A33 E89 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.012uM remove_due_to_license_issue IC50=111nM P11309 25616902 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4wtu A 1.85 BS01 3UT A 1 G11 Q12 G13 L30 D32 S35 Y71 W76 F108 I118 R128 D228 G230 G13 Q14 G15 L32 D34 S37 Y73 W78 F110 I120 R130 D220 G222 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.3nM remove_due_to_license_issue IC50=3.0nM P56817 25699151 407 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4wu4 A 2.3 BS01 dna H 0 K177 S181 N191 R192 K39 S43 N53 R54 remove_due_to_license_issue 25897118 -102 ~ -86 MVLHEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLAK 4wu4 B 2.3 BS01 dna G 0 N162 K174 K177 S181 N191 R192 N24 K36 K39 S43 N53 R54 remove_due_to_license_issue 25897118 -86 ~ -102 MVLHEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLAK 4wu4 B 2.3 BS02 dna H 0 T146 R148 I171 T172 K174 T175 H179 T8 R10 I33 T34 K36 T37 H41 remove_due_to_license_issue 25897118 -102 ~ -86 MVLHEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLAK 4wul A 2.4 BS01 dna H 0 S161 N162 K177 S181 L184 N191 R192 S21 N22 K37 S41 L44 N51 R52 remove_due_to_license_issue 25897118 -124 ~ -99 LHEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLA 4wul A 2.4 BS02 dna C 0 T146 R148 I171 T172 K174 T175 T178 H179 T6 R8 I31 T32 K34 T35 T38 H39 remove_due_to_license_issue 25897118 -99 ~ -124 LHEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLA 4wul B 2.4 BS01 dna H 0 T146 R148 I171 T172 K174 T175 T178 H179 T5 R7 I30 T31 K33 T34 T37 H38 remove_due_to_license_issue 25897118 -124 ~ -99 HEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLA 4wul B 2.4 BS02 dna C 0 S161 N162 N191 R192 S20 N21 N50 R51 remove_due_to_license_issue 25897118 -99 ~ -124 HEDLTNREHEILMLIAQGKSNQEIADELFITLKTVKTHVSNILAKLDVDNRTQAAIYAFQHGLA 4wup A 1.75 BS02 3UF A 1 H94 H96 H119 L198 T199 H200 W209 H90 H92 H115 L194 T195 H196 W205 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=0.15nM remove_due_to_license_issue Kd=790nM P00915 26079542 302 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 4wuy A 1.63 BS01 3UJ A 1 K145 I149 N180 C181 N182 G183 F184 T185 Y240 Y258 K141 I145 N176 C177 N178 G179 F180 T181 Y236 Y254 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 ic50<15nM remove_due_to_license_issue IC50=<15nM Q9NRG4 25825497 501 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLGFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKAEAIRDMVRYARNVIEEFRELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIESH 4wvl A 2.41 BS01 3US A 1 D161 G163 S164 V169 E186 K187 D222 F223 F239 N241 S268 D145 G147 S148 V153 E170 K171 D206 F207 F223 N225 S252 2.1.1.360 0031151,0051726 remove_due_to_license_issue Q8TEK3 25397901 401 KLELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMEDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNNYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLKNPKLREEQEAARRRQQR 4ww6 A 1.06 BS02 3TV A 1 H94 H119 V121 F131 V143 L198 T199 T200 H91 H116 V118 F127 V139 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.062nM remove_due_to_license_issue Kd=0.91nM P00918 26079542 306 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ww6 A 1.06 BS03 3TV A 2 H4 W5 H10 H15 D19 H1 W2 H7 H12 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.062nM remove_due_to_license_issue Kd=0.91nM P00918 26079542 307 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4ww8 A 1.42 BS02 VD9 A 1 H91 H117 L197 T198 T199 H89 H115 L195 T196 T197 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=0.067nM remove_due_to_license_issue Kd=400nM O43570 26079542 305 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 4wwn A 2.7 BS01 3VC A 1 V803 M804 P810 W812 I831 Y867 E880 T886 M953 I963 V557 M558 P564 W566 I585 Y621 E634 T640 M707 I717 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 25469863 1203 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAIDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKETVSLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNHPIALPKHQEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 4wwo A 2.3 BS01 3VD A 1 K802 M804 P810 W812 I831 Y867 I879 E880 M953 I963 K543 M545 P551 W553 I572 Y608 I620 E621 M690 I700 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=0.038uM remove_due_to_license_issue P48736 25469863 1205 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGSFNADKLTSATNPDKENSMSISILLDNAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 4wwp A 2.4 BS01 3VE A 1 K802 M804 P810 W812 I831 Y867 I879 E880 I881 V882 M953 I963 K545 M547 P553 W555 I574 Y610 I622 E623 I624 V625 M696 I706 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 ic50=0.12uM remove_due_to_license_issue P48736 25469863 1204 QAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEETVSLWDCDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCGKKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDNEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 4wx4 A 1.03 BS02 3VF A 1 S1 S3 S4 E5 T24 H25 D26 N44 G47 R48 G51 G52 V53 W55 A120 C122 S1 S3 S4 E5 T24 H25 D26 N44 G47 R48 G51 G52 V53 W55 A120 C122 H54 D71 Q115 C122 H54 D71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 remove_due_to_license_issue B9A5C1 25571794 301 SGSSEQELAAIVRDLGCGPYFLGTHDKRFPGFLAGNKLACAIVNTAGRETGGVHWLAFGWNPRSRTCYMFDPFGFSDRRLKQIYSFEYEAMLRRSALALSPDRCLSLEQSTQTVQGPDSAACGLFCCMFLHAFVHWPDRPMDGNPTMNLLTGVPNGMLQSPQVLPTLRRNQEKLYRFLAHHSPYFRSHRAAIEHATAFDKM 4wx6 A 2.15 BS02 3VK A 1 G2 S3 S4 E5 T24 D26 N44 A46 R48 G51 G52 V53 H54 W55 F73 Y84 C122 G2 S3 S4 E5 T24 D26 N44 A46 R48 G51 G52 V53 H54 W55 F73 Y84 C122 H54 D71 Q115 C122 H54 D71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 remove_due_to_license_issue B9A5C1 25571794 301 SGSSEQELAAIVRDLGCGPYFLGTHDKRFPGFLAGNKLACAIVNTAGRETGGVHWLAFGWNPRSRTCYMFDPFGFSDRRLKQIYSFEYEAMLRRSALALSPDRCLSLEQSTQTVQGPDSAACGLFCCMFLHAFVHWPDRPMDGNPTMNLLTGVPNGMLQSPQVLPTLRRNQEKLYRFLAHHSPYFRSHRAAIEHATAFDKMKQL 4wx7 A 2.4 BS02 3VJ A 1 G2 S3 E5 T24 H25 D26 N44 G47 R48 G51 G52 V53 H54 W55 C122 G2 S3 E5 T24 H25 D26 N44 G47 R48 G51 G52 V53 H54 W55 C122 H54 D71 Q115 C122 H54 D71 Q115 C122 3.4.22.39 0003677,0004197,0006508,0008234,0042025,0044423 remove_due_to_license_issue B9A5C1 25571794 301 SGSSEQELAAIVRDLGCGPYFLGTHDKRFPGFLAGNKLACAIVNTAGRETGGVHWLAFGWNPRSRTCYMFDPFGFSDRRLKQIYSFEYEAMLRRSALALSPDRCLSLEQSTQTVQGPDSAACGLFCCMFLHAFVHWPDRPMDGNPTMNLLTGVPNGMLQSPQVLPTLRRNQEKLYRFLAHHSPYFRSHRAAIEHATAFDKMKQL 4wxi A 2.6 BS01 3VM A 1 R39 H40 C42 H57 Y143 I151 D189 A190 C191 K192 G193 S195 T213 W215 R26 H27 C29 H44 Y134 I141 D182 A183 C184 K185 G186 S188 T206 W208 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 25592713 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4wy1 A 1.98 BS01 3VO A 1 L30 D32 Y71 F108 W115 D228 G230 L32 D34 Y73 F110 W117 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=5.1uM remove_due_to_license_issue IC50=5100nM P56817 25695670 4000 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQTDESRSHHHH 4wy3 A 1.89 BS01 3X5 A 1 H41 M49 F140 L141 G143 C145 H163 M165 E166 D187 I188 Q189 H41 M49 F140 L141 G143 C145 H163 M165 E166 D187 I188 Q189 H41 G143 C145 H41 G143 C145 2.1.1.-,2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.4.22.69,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=240uM remove_due_to_license_issue IC50=240000nM P0C6X7 25614110 401 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDTVYCPRHVICTAEDMLNPNYEDLLIRKSNHSFLVQAGNVQLRVIGHSMQNCLLRLKVDTSNPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNHTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGKFYGPFVDIQTAQAAGTDTTITLNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCAALKELLQNGMNGRTILGSTILEDEFTPFDVVRQCSGVTFQ 4wy6 A 2.1 BS01 3VP A 1 D32 Y71 F108 W115 D228 G230 D36 Y75 F112 W119 D223 G225 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=1.07uM remove_due_to_license_issue IC50=1070nM P56817 25695670 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4wyo B 2.89 BS01 3W2 B 1 V1923 R1954 F1956 L2025 E2026 G2029 E2032 V444 R475 F477 L546 E547 G550 E553 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 4000 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFAQDLAKKIRSDHDNAIDGLSEVTDDKEKLLKTLKL 4wyo B 2.89 BS02 3W2 C 1 A1761 L1762 K1764 V1765 A282 L283 K285 V286 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 4000 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFAQDLAKKIRSDHDNAIDGLSEVTDDKEKLLKTLKL 4wyo C 2.89 BS01 3W2 B 1 A1761 L1762 V1765 A270 L271 V274 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 4000 WLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKSLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGNAIDGLSEVIKMLSTDDKEKLLKTLK 4wyo C 2.89 BS02 3W2 C 1 V1923 R1954 F1956 G1958 L2025 E2026 G2029 E2032 V432 R463 F465 G467 L534 E535 G538 E541 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 4000 WLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKSLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGNAIDGLSEVIKMLSTDDKEKLLKTLK 4wyp A 1.502 BS01 AMP A 1 K41 P42 H119 F120 K41 P42 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Kd=440uM remove_due_to_license_issue P61823 26655472 401 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVGCEGNPYVPVHFDASV 4wyy A 1.28 BS01 3VT A 1 S90 Q146 Y177 N179 Y249 T343 G344 S345 S62 Q118 Y149 N151 Y221 T315 G316 S317 S90 K93 Y177 E299 K342 S345 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 27622821 406 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLE 4wyz A 1.449 BS01 U3P A 1 H12 K41 N44 T45 F120 H13 K42 N45 T46 F121 H12 K41 H119 F120 D121 H13 K42 H120 F121 D122 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Kd=50uM remove_due_to_license_issue Ki=78500nM P61823 26655472 401 MKETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVGCEGNPYVPVHFDASV 4wz4 A 1.05 BS01 3VU A 1 S90 Q146 Y177 N179 Y249 T343 G344 S345 S62 Q118 Y149 N151 Y221 T315 G316 S317 S90 K93 Y177 E299 K342 S345 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 27622821 402 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLE 4wz5 A 1.6 BS01 3VU A 1 S67 W102 S115 V117 L155 G207 F208 S209 R250 S47 W82 S95 V97 L135 G187 F188 S189 R230 S67 K70 S115 F120 W154 F208 S47 K50 S95 F100 W134 F188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0042597,0046677,0071555 remove_due_to_license_issue P14489 27622821 303 SITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNDLARASKEYLPASTFKIPNAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLTLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLYLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKETEVYFFAFNMDIDNESKLPLRKSIPTKIMESEGII 4wz6 A 2.05 BS01 ATP A 1 W401 V440 T460 G461 G463 K464 T465 S466 Q493 W13 V33 T53 G54 G56 K57 T58 S59 Q86 5.6.1.6 0005524,0016887 Kd=1.4uM remove_due_to_license_issue P13569 26444971 701 TTEVVMENVTAFWEEGFGELFEKAKQSLLGTPVLKDINFKIERGQLLAVAGSTGAGKTSLLMMIMGELEPSEGKIKHSGRISFCSQNSWIMPGTIKENIIGVSYDEYRYRSVIKACQLEEDISKFAEKDNIVLGITLSGGQRARISLARAVYKDADLYLLDSPFGYLDVLTEKEIFESCVCKLMANKTRILVTSKMEHLKKADKILILHEGSSYFYGTFSELQNLRPDFSSKLMSFDQFSAERRNSILTETLHRFSLE 4wz8 B 2.23 BS01 3W7 B 1 V1923 R1954 F1956 L2025 E2026 G2029 V444 R475 F477 L546 E547 G550 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 4wz8 B 2.23 BS02 3W7 C 1 A1761 L1762 K1764 V1765 A282 L283 K285 V286 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 4wz8 C 2.23 BS01 3W7 B 1 A1761 K1764 A268 K271 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 2301 QPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKSLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKL 4wz8 C 2.23 BS02 3W7 C 1 V1923 R1954 F1956 L2025 E2026 E2028 G2029 V430 R461 F463 L532 E533 E535 G536 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 25423286 2301 QPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKSLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVGEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKL 4wzv A 1.65 BS01 E40 A 1 L187 L188 A189 H190 A191 H226 E227 H230 D235 H236 L243 Y245 P246 M247 Y248 L76 L77 A78 H79 A80 H115 E116 H119 D124 H125 L132 Y134 P135 M136 Y137 H226 E227 H230 H236 H115 E116 H119 H125 3.4.24.35 0004222,0006508,0008237,0008270,0031012 ic50=0.43nM remove_due_to_license_issue IC50=0.430000nM P14780 26263024 301 GDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4wzv A 1.65 BS07 E40 B 1 Y245 P246 Y134 P135 H226 E227 H230 H236 H115 E116 H119 H125 3.4.24.35 0004222,0006508,0008237,0008270,0031012 ic50=0.43nM remove_due_to_license_issue IC50=0.430000nM P14780 26263024 301 GDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4wzw A 2.9516 BS01 dna B 0 R268 H362 V455 R140 H234 V327 ? 0003723 remove_due_to_license_issue Q15397 25512524 1 ~ 14 KTNYDIVVRAKQMWEILRRKDCDKEKRVKLMSDLQKLIQGKIKTIAFAHDSTRVIQCYIQYGNEEQRKQAFEELRDDLVELSKAKYSRNIVKKFLMYGSKPQIAEIIRSFKGHVRKMLRHAEASAIVEYAYNDKAILEQRNMLTEELYGNTFQLYKSADHPTLDKVLEVQPEKLELIMDEMKQILTPMAQKEAVIKHSLVHKVFLDFFTYAPPKLRSEMIEAIREAVVYLAHTHDGARVAMHCLWHGTPKDRKVIVKTMKTYVEKVANGQYSHLVLLAAFDCIDDTKLVKQIIISEIISSLPSIVNDKYGRKVLLYLLSPRDPAHTVREIIEVLQKGDGNAHSKKDTEVRRRELLESISPALLSYLQEHAQEVVLDKSACVLVSDILGSATGDVQPTMNAIASLAATGLHPLHIAEHPAGHLVLKWLIEQDKKMKENGREGCFAKTLVEHVGMKNLKSWASVNRGAIILSSLLQSCDLEVANKVKAALKSLIPTLEKGIEILLEK 4x0f A 3.22 BS02 ROL A 1 Y405 T579 I582 S614 Q615 F618 Y159 T333 I336 S368 Q369 F372 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q07343 25775568 804 VTPFAQVLASLRSVRNNFTLEELDWALDQLETIQTYRSVSEMASNKFKRMLNRELTHLSEMSRCGNQVSEYISNTFLDKSRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTAIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHADIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHAADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMADKHTACVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIP 4x0f B 3.22 BS02 ROL B 1 Y405 T579 I582 M583 F586 Q615 F618 Y162 T336 I339 M340 F343 Q372 F375 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q07343 25775568 803 TPFAQVLASLRSVRNNFTIESYQKLAMETLEELDWALDQLETIQTYRSVSEMASNKFKRMLNRELTHLSEMSRCGNQVSEYISNTFLDTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTAIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHADIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHAADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMADKHTACVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQAMIP 4x0u A 1.95 BS01 3W9 A 1 F168 V172 C302 F166 V170 C299 N167 K190 E268 C302 E399 N165 K188 E266 C299 E396 1.2.1.3,1.2.1.31,1.2.1.8 0004029,0004043,0005515,0005634,0005737,0005739,0005759,0005829,0006081,0007605,0008802,0016491,0016620,0019285,0042426,0042802,0070062 remove_due_to_license_issue P49419 25554827 601 TLLINQPQYAWLKELGLREENEGVYNGSWGGRGEVITTYCPANNEPIARVRQASVADYEETVKKAREAWKIWADIPAPKRGEIVRQIGDALREKIQVLGSLVSLEMGKILVEGVGEVQEYVDICDYAVGLSRMIGGPILPSERSGHALIEQWNPVGLVGIITAFNFPVAVYGWNNAIAMICGNVCLWKGAPTTSLISVAVTKIIAKVLEDNKLPGAICSLTCGGADIGTAMAKDERVNLLSFTGSTQVGKQVGLMVQERFGRSLLELGNNAIIAFEDADLSLVVPSALFAAVGTAGQRCTTARRLFIHESIHDEVVNRLKKAYAQIRVGNPWDPNVLYGPLHTKQAVSMFLGAVEEAKKEGGTVVYGGKVMDRPGNYVEPTIVTGLGHDASIAHTETFAPILYVFKFKNEEEVFAWNNEVKQGLSSSIFTKDLGRIFRWLGPKGSDCGIVNVNISDAWKQYMRRSTCTINYQGIKFQ 4x0z C 1.85 BS01 GAL G 1 I61 S62 I37 S38 ? 0005198,0019028 remove_due_to_license_issue P90498 25855729 3 EVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNKDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTTLMNVHSNGQATHDNGAAKPVQGTSFHFFSVGGEALELQGVVFNYRTTYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x0z C 1.85 BS02 SIA G 1 L54 K59 S60 N264 S266 S268 Q270 L30 K35 S36 N232 S234 S236 Q238 ? 0005198,0019028 remove_due_to_license_issue P90498 25855729 4 EVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNKDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTTLMNVHSNGQATHDNGAAKPVQGTSFHFFSVGGEALELQGVVFNYRTTYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x11 A 2.3 BS01 SIA A 1 L54 K59 S60 N264 S266 S268 Q270 L29 K34 S35 N231 S233 S235 Q237 ? 0005198,0019028 remove_due_to_license_issue P90498 25855729 301 VLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNKDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTTLMNVHSNGQATHDNGAAKPVQGTSFHFFSVGGEALELQGVVFNYRTTYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x11 B 2.3 BS01 SIA B 1 K59 S60 N123 N264 S266 S268 K35 S36 N91 N232 S234 S236 ? 0005198,0019028 remove_due_to_license_issue P90498 25855729 301 EVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNKDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTTLMNVHSNGQATHDNGAAKPVQGTSFHFFSVGGEALELQGVVFNYRTTYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x13 B 2.0 BS01 SIA F 1 L54 K59 S60 N264 S266 S268 Q270 L30 K35 S36 N232 S234 S236 Q238 ? 0005198,0019028 remove_due_to_license_issue P90498 25855729 5 EVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNKDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTTLMNVHSNGQATHDNGAAKPVQGTSFHFFSVGGEALELQGVVFNYRTTYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x13 C 2.0 BS01 SIA G 1 L54 K59 S60 N264 S266 S268 Q270 L31 K36 S37 N233 S235 S237 Q239 ? 0005198,0019028 remove_due_to_license_issue P90498 25855729 5 VEVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNKDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTTLMNVHSNGQATHDNGAAKPVQGTSFHFFSVGGEALELQGVVFNYRTTYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x14 B 2.3 BS01 GAL F 1 S60 I61 S37 I38 ? 0005198,0019028 remove_due_to_license_issue P03089 25855729 3 VEVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNRDMLPCYSVARIPLPNLNILMWEAVTLKTEVIGVTSLMNVHSNGQATHDNGAGKPVQGTSFHFFSVGGEALELQGVLFNYRTKYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x14 B 2.3 BS02 SIA F 1 L54 K59 S60 N264 S266 S268 Q270 L31 K36 S37 N234 S236 S238 Q240 ? 0005198,0019028 remove_due_to_license_issue P03089 25855729 4 VEVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNRDMLPCYSVARIPLPNLNILMWEAVTLKTEVIGVTSLMNVHSNGQATHDNGAGKPVQGTSFHFFSVGGEALELQGVLFNYRTKYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x14 C 2.3 BS01 GAL G 1 S60 S62 S36 S38 ? 0005198,0019028 remove_due_to_license_issue P03089 25855729 4 EVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNRDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTSLMNVHSNGQATHDNGAGKPVQGTSFHFFSVGGEALELQGVLFNYRTKYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x14 C 2.3 BS02 SIA G 1 L54 K59 S60 N264 S266 S268 Q270 L30 K35 S36 N232 S234 S236 Q238 ? 0005198,0019028 remove_due_to_license_issue P03089 25855729 5 EVLEVKTGVDSITEVECFLTPEMGDPDEHLRGFSKSISISDTFESDSPNRDMLPCYSVARIPLPNLILMWEAVTLKTEVIGVTSLMNVHSNGQATHDNGAGKPVQGTSFHFFSVGGEALELQGVLFNYRTKYPDGTIFPKNATVQSQVMNTEHKAYLDKNKAYPVECWVPDPTRNENTRYFGTLTGGENVPPVLHITNTATTVLLDEFGVGPLCKGDNLYLSAVDVCGMFTNRSGSQQWRGLSRYFKVQLRKRRVK 4x1f A 2.0 BS01 3WF A 1 D205 L206 M243 S247 F251 H407 R410 M425 D47 L48 M85 S89 F93 H244 R247 M262 ? 0003677,0004879,0006355 Kd=10.8nM remove_due_to_license_issue O75469 26333997 501 GLTEEQRMMIRELMDAQMKTFDTTFSHFKNFRLPGVEAAKWSQVRKDLCSLKVSLQLRGEDGSVWNYKPPADSGGKEIFSLLPHMADMSTYMFKGIISFAKVISYFRDLPIEDQISLLKGAAFELCQLRFNTVFNAETGTWECGRLSYCLEDQQLLLEPMLKFHYMLKKLQLHEEEYVLMQAISLFSPDRPGVLQHRVVDQLQEQFAITLKSYIECNRPQPAHRFLFLKIMAMLTELRSINAQHTQRLLRIQDIHPFATPLMQELFGITGS 4x21 A 1.95 BS01 3WH A 1 V78 A91 M146 M149 D150 A151 N152 Q155 L206 V33 A46 M101 M104 D105 A106 N107 Q110 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T167 2.7.11.24 0004672,0004707,0005524,0006468 Kd=36nM remove_due_to_license_issue P53779 26505827 501 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIDEREHTIEEWKELIYKEVMN 4x23 A 3.5 BS01 dna I 0 R42 T45 R83 F84 Q85 S86 R116 V117 T118 R3 T6 R44 F45 Q46 S47 R77 V78 T79 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 2 ~ 147 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIE 4x23 A 3.5 BS02 dna J 0 Y41 G44 V46 A47 R49 R63 K64 L65 P66 R69 R83 Y2 G5 V7 A8 R10 R24 K25 L26 P27 R30 R44 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 1 ~ 146 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIE 4x23 B 3.5 BS01 dna I 0 T30 P32 R36 R45 T7 P9 R13 R22 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 2 ~ 147 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 B 3.5 BS02 dna J 0 R35 R45 I46 S47 R78 K79 T80 R12 R22 I23 S24 R55 K56 T57 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 1 ~ 146 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 C 3.5 BS01 dna I 0 R16 R19 R28 R31 R41 R76 R2 R5 R14 R17 R27 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 2 ~ 147 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 C 3.5 BS02 dna J 0 R34 R41 V42 A44 K74 T75 R76 R20 R27 V28 A30 K60 T61 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 1 ~ 146 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 D 3.5 BS01 dna I 0 Y39 G50 I51 S53 S84 T85 Y8 G19 I20 S22 S53 T54 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 2 ~ 147 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4x23 D 3.5 BS02 dna J 0 E32 S33 I36 Y37 E1 S2 I5 Y6 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 1 ~ 146 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4x23 E 3.5 BS01 dna I 0 R40 Y41 R42 G44 V46 A47 R49 R63 K64 L65 P66 R69 R83 R1 Y2 R3 G5 V7 A8 R10 R24 K25 L26 P27 R30 R44 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 2 ~ 147 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIEGGL 4x23 E 3.5 BS02 dna J 0 R42 T45 R63 R72 R83 F84 Q85 S86 R116 V117 T118 R3 T6 R24 R33 R44 F45 Q46 S47 R77 V78 T79 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 1 ~ 146 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIEGGL 4x23 F 3.5 BS01 dna I 0 R35 R45 I46 S47 G48 R78 K79 T80 R12 R22 I23 S24 G25 R55 K56 T57 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 2 ~ 147 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 F 3.5 BS02 dna J 0 T30 P32 R36 R45 T7 P9 R13 R22 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 1 ~ 146 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 G 3.5 BS01 dna I 0 R28 R41 V42 A44 K74 T75 R76 R14 R27 V28 A30 K60 T61 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 2 ~ 147 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 G 3.5 BS02 dna J 0 R16 G27 R28 R31 R41 R76 R2 G13 R14 R17 R27 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 1 ~ 146 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 H 3.5 BS01 dna I 0 E32 I36 Y37 E1 I5 Y6 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 2 ~ 147 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4x23 H 3.5 BS02 dna J 0 Y39 G50 I51 S53 R83 S84 T85 Y8 G19 I20 S22 R52 S53 T54 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 1 ~ 146 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4x23 K 3.5 BS01 dna S 0 R40 R42 P43 T45 R63 R72 R83 F84 Q85 S86 R116 V117 T118 R1 R3 P4 T6 R24 R33 R44 F45 Q46 S47 R77 V78 T79 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 2 ~ 147 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIE 4x23 K 3.5 BS02 dna T 0 R40 Y41 R42 G44 V46 A47 R63 K64 L65 P66 R69 R83 R1 Y2 R3 G5 V7 A8 R24 K25 L26 P27 R30 R44 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 1 ~ 146 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIE 4x23 L 3.5 BS01 dna S 0 T30 P32 R36 R45 T7 P9 R13 R22 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 2 ~ 147 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 L 3.5 BS02 dna T 0 R35 R45 I46 R78 K79 T80 R12 R22 I23 R55 K56 T57 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 1 ~ 146 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 M 3.5 BS01 dna S 0 R16 R31 R76 R2 R17 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 2 ~ 147 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 M 3.5 BS02 dna T 0 R28 R34 R41 V42 A44 K74 T75 R76 R14 R20 R27 V28 A30 K60 T61 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 1 ~ 146 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 N 3.5 BS01 dna S 0 Y39 G50 I51 S53 S84 T85 Y8 G19 I20 S22 S53 T54 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 2 ~ 147 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4x23 N 3.5 BS02 dna T 0 E32 I36 Y37 E1 I5 Y6 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 1 ~ 146 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSS 4x23 O 3.5 BS01 dna S 0 R40 Y41 R42 P43 G44 T45 V46 A47 K56 R63 K64 L65 P66 R69 R83 R1 Y2 R3 P4 G5 T6 V7 A8 K17 R24 K25 L26 P27 R30 R44 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 2 ~ 147 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIEGGL 4x23 O 3.5 BS02 dna T 0 R42 P43 T45 R63 R72 R83 F84 Q85 S86 R116 V117 T118 R3 P4 T6 R24 R33 R44 F45 Q46 S47 R77 V78 T79 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02299 23723239 1 ~ 146 RYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGIEGGL 4x23 P 3.5 BS01 dna S 0 R35 R45 I46 S47 R78 K79 T80 R12 R22 I23 S24 R55 K56 T57 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 2 ~ 147 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 P 3.5 BS02 dna T 0 T30 P32 R36 R45 T7 P9 R13 R22 ? 0003677,0030527,0046982 remove_due_to_license_issue P84040 23723239 1 ~ 146 DNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 4x23 Q 3.5 BS01 dna S 0 R28 R34 R41 V42 G43 A44 K74 T75 R76 R14 R20 R27 V28 G29 A30 K60 T61 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 2 ~ 147 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 Q 3.5 BS02 dna T 0 R16 R28 R31 R41 R76 R2 R14 R17 R27 R62 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P84051 23723239 1 ~ 146 SRSNRAGLQFPVGRIHRLLRKGNYAERVGAGAPVYLAAVMEYLAAEVLELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLSGVTIAQGGVLPNIQAVLLP 4x23 R 3.5 BS01 dna S 0 E32 I36 Y37 E1 I5 Y6 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 2 ~ 147 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYT 4x23 R 3.5 BS02 dna T 0 Y39 I51 S53 R83 S84 T85 Y8 I20 S22 R52 S53 T54 ? 0000786,0003677,0030527,0046982 remove_due_to_license_issue P02283 23723239 1 ~ 146 ESYAIYIYKVLKQVHPDTGISSKAMSIMNSFVNDIFERIAAEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYT 4x24 A 1.5 BS01 TDI A 1 M9 I50 S76 A77 G78 F152 I153 E173 M174 E175 D198 F208 M9 I50 S76 A77 G78 F152 I153 E173 M174 E175 D198 F208 3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509 Ki=166pM remove_due_to_license_issue A5F5R2 25806409 301 MKIGIIGAMQQEVAILKDLIEDVQEVNQAGCTFYSGQIQGVDVVLLQSGIGKVSAALGTALLISQYAPDVVINTGSAGGFDASLNVGDVVISSEVRHHDADVTAFGYEIGQMPGQPAAFKADEKLMTVAEQALAQLPNTHAVRGLICTGDAFICTAEGQQFIRQHFPSVVAVEMEASAIAQTCHQFKVPFVVVRAISDVADKESPLSFEEFLPLAAKSSSAMVLKMVELLKENLYFQ 4x24 B 1.5 BS01 TDI B 1 M9 I50 S76 A77 G78 F152 I153 E173 M174 E175 D198 F208 M9 I50 S76 A77 G78 F152 I153 E173 M174 E175 D198 F208 3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509 Ki=166pM remove_due_to_license_issue A5F5R2 25806409 301 MKIGIIGAMQQEVAILKDLIEDVQEVNQAGCTFYSGQIQGVDVVLLQSGIGKVSAALGTALLISQYAPDVVINTGSAGGFDASLNVGDVVISSEVRHHDADVTAFGYEIGQMPGQPAAFKADEKLMTVAEQALAQLPNTHAVRGLICTGDAFICTAEGQQFIRQHFPSVVAVEMEASAIAQTCHQFKVPFVVVRAISDVADKESPLSFEEFLPLAAKSSSAMVLKMVELLKENLYFQ 4x2i A 1.2 BS01 3X0 A 1 W81 P82 L92 Y139 N140 I146 M149 W41 P42 L52 Y99 N100 I106 M109 ? ic50=0.35uM remove_due_to_license_issue O60885 26985289 202 GSTNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4x2l A 2.55 BS01 3WP A 1 D32 Y71 F108 W115 D228 G230 D36 Y75 F112 W119 D221 G223 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=36000nM P56817 25695670 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4x2s A 4.21 BS01 ASP A 1 S276 S277 S278 T314 G354 V355 P356 G357 A358 G359 R397 T398 S265 S266 S267 T303 G343 V344 P345 G346 A347 G348 R386 T387 ? 0005283,0005886,0006865,0015108,0015183,0015293,0015501,0016020,0035725,0042802,0046872,0046942,0070207,0070778,0140009,1902476 remove_due_to_license_issue O59010 25652997 501 VLQKILIGLILGAIVGLILGHYGYAHAVHTYVKPFGDLFVRLLKMLVMPIVFASLVVGAASISPARLGRVGVKIVVYYLLTSAFAVTLGIIMARLFNPGAGIHLAVGGQQFQPHQAPPLVHILLDIVPTNPFGALANGQVLPTIFFAIILGIAITYLMNSENEKVRKSAETLLDAINGLAEAMYKIVNGVMQYAPIGVFALIAYVMAEQGVHVVGELAKVTAAVYVGLTLQILLVYFVLLKIYGIDPISFIKHAKDAMLTAFVTSSSSGTLPVTMRVAKEMGISEGIYSFTLPLGATINMDGTALYQGVATFFIANALGSHLTVGQQLTIVLTAVLASIGTAGVPGAGAIMLAMVLHSVGLPLTDPNVAAAYAMILGIDAILDRGRTMVNVTGDLTGTAIVAKTE 4x3r A 1.86 BS04 686 A 1 K207 R210 E424 L428 R463 R511 G518 N519 R536 W541 Y552 H553 K699 Y700 K153 R156 E370 L374 R409 R457 G464 N465 R482 W487 Y495 H496 K639 Y640 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 Ki=0.0086nM remove_due_to_license_issue Ki=0.008600nM Q04609 25923815 1320 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 4x3t A 2.14 BS01 45E A 1 F11 W32 W35 Y39 E43 H47 F7 W28 W31 Y35 E39 H43 ? 0035102 Kd=28.9uM remove_due_to_license_issue Q8VDS3 25660273 101 HMGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEERDRA 4x3t B 2.14 BS01 45E B 1 M6 F11 W32 W35 Y39 T41 E43 H47 M2 F7 W28 W31 Y35 T37 E39 H43 ? 0035102 Kd=28.9uM remove_due_to_license_issue Q8VDS3 25660273 101 HMGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEERD 4x3u A 1.63 BS01 SVR B 1 R20 W32 W35 Y39 S40 T41 W42 E46 H47 R10 W22 W25 Y29 S30 T31 W32 E36 H37 ? 0035102 remove_due_to_license_issue Q8VDS3 25660273 101 FAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEERDRA 4x3u B 1.63 BS01 SVR B 1 R20 R22 W32 W35 Y39 S40 T41 W42 H47 R11 R13 W23 W26 Y30 S31 T32 W33 H38 ? 0035102 ic50=8.1uM remove_due_to_license_issue Q8VDS3 25660273 101 VFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEE 4x3u B 1.63 BS02 SVR B 2 R20 V21 R11 V12 ? 0035102 ic50=8.1uM remove_due_to_license_issue Q8VDS3 25660273 102 VFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEE 4x47 A 2.0 BS01 DAN A 1 R257 D282 D339 T557 R575 R637 Y677 W698 R23 D48 D105 T323 R341 R403 Y443 W464 0004308 ic50=1.41mM remove_due_to_license_issue 26154892 801 GAMADIGSNIFYAGDATKSNYFRIPSLLALDSGTVIAAADARYGGTHDAKSKINTAFAKSTDGGKTWGQPTLPLKFDDYVAKNIDWPRDSVGKNVQIQGSASYIDPVLLEDKETHRVFLFADMMPAGIGSSNASVGSGFKEVDGKKYLKLHWKDDAAGTYDYSVRENGTIYNDTTNSATEYSVDGEYNLYKNGNAMLCKQYDYNFEGTKLLETQTDTDVNMNVFYKDADFKVFPTTYLAMKYSDDEGETWSDLQIVSTFKPEESKFLVLGPGVGKQIANGEHAGRLIVPLYSKSSAELGFMYSDDHGNNWTYVEADQNTGGATAEAQIVEMPDGSLKTYLRTGSGYIAQVMSTDGGETWSERVPLTEIATTGYGTQLSVINYSQPVDGKPAILLSAPNATNGRKNGKIWIGLISETGNSGKDKYSVDWKYCYSVDTPQMGYSYSCLTELPDGEIGLLYEKYDSWSRNELHLKNILKYERFNIDELKVQP 4x48 A 1.89 BS03 XPF C 1 K493 P494 S497 S729 K730 L751 N754 K101 P102 S105 S214 K215 L236 N239 ? 0015276,0016020 remove_due_to_license_issue P19491 25905800 804 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4x48 C 1.89 BS03 XPF C 1 P494 S729 K730 G731 N754 P101 S213 K214 G215 N238 ? 0015276,0016020 remove_due_to_license_issue P19491 25905800 804 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4x49 A 2.01 BS01 G39 A 1 R257 D282 D339 S364 R575 R637 Y677 W698 R23 D48 D105 S130 R341 R403 Y443 W464 0004308 ic50=0.0296mM remove_due_to_license_issue 26154892 801 GAMADIGSNIFYAGDATKSNYFRIPSLLALDSGTVIAAADARYGGTHDAKSKINTAFAKSTDGGKTWGQPTLPLKFDDYVAKNIDWPRDSVGKNVQIQGSASYIDPVLLEDKETHRVFLFADMMPAGIGSSNASVGSGFKEVDGKKYLKLHWKDDAAGTYDYSVRENGTIYNDTTNSATEYSVDGEYNLYKNGNAMLCKQYDYNFEGTKLLETQTDTDVNMNVFYKDADFKVFPTTYLAMKYSDDEGETWSDLQIVSTFKPEESKFLVLGPGVGKQIANGEHAGRLIVPLYSKSSAELGFMYSDDHGNNWTYVEADQNTGGATAEAQIVEMPDGSLKTYLRTGSGYIAQVMSTDGGETWSERVPLTEIATTGYGTQLSVINYSQPVDGKPAILLSAPNATNGRKNGKIWIGLISETGNSGKDKYSVDWKYCYSVDTPQMGYSYSCLTELPDGEIGLLYEKYDSWSRNELHLKNILKYERFNIDELKVQP 4x50 A 2.0 BS01 3X8 A 1 F1 I13 N46 Y48 D54 Q133 N135 Y137 D140 F1 I13 N46 Y48 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=17.7nM remove_due_to_license_issue P08191 25940742 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4x5p A 0.997 BS01 3XJ A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 Y137 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=6.2nM remove_due_to_license_issue P08191 25940742 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4x5q A 1.12 BS01 3XN A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 Y137 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 Y137 D140 ? 0007155,0009289 remove_due_to_license_issue P08191 25940742 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4x5r A 1.65 BS01 3XO A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 ? 0007155,0009289 Kd=14nM remove_due_to_license_issue P08191 25940742 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4x5y A 1.59 BS01 3XW A 1 S155 L177 S178 H181 F238 Y276 M278 M322 Y323 E363 E366 S134 L156 S157 H160 F217 Y255 M257 M301 Y302 E342 E345 ? 0005634 Kd=9.3nM remove_due_to_license_issue IC50=15nM, Kd=10.0nM O00255 25817203 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMKK 4x5z A 1.86 BS01 3XY A 1 S155 L177 S178 H181 F238 Y276 M278 M322 Y323 E363 S134 L156 S157 H160 F217 Y255 M257 M301 Y302 E342 ? 0005634 Kd=23.6nM remove_due_to_license_issue Kd=24nM O00255 25817203 605 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 4x60 A 2.35 BS02 3XV A 1 L319 F327 E435 E444 V503 F577 S578 W579 F580 L307 F315 E423 E432 V491 F565 S566 W567 F568 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 Kd<1nM remove_due_to_license_issue IC50=47nM O14744 25915199 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 4x61 A 2.85 BS02 3XV A 1 Y304 L319 F327 E444 V503 F577 S578 W579 F580 Y292 L307 F315 E432 V491 F565 S566 W567 F568 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 remove_due_to_license_issue IC50=47nM O14744 25915199 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 4x63 A 3.05 BS02 3XV A 1 Y304 L312 L319 F327 K333 E444 V503 F577 S578 W579 F580 Y292 L300 L307 F315 K321 E432 V491 F565 S566 W567 F568 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 remove_due_to_license_issue IC50=47nM O14744 25915199 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 4x68 A 1.68 BS01 OP0 A 1 S90 Q146 Y177 Y249 T343 G344 S345 S60 Q116 Y147 Y219 T313 G314 S315 S90 K93 Y177 E299 K342 S345 S60 K63 Y147 E269 K312 S315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 26089439 401 MDRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGL 4x68 B 1.68 BS01 OP0 B 1 S90 Q146 Y177 Y249 T343 G344 S345 S60 Q116 Y147 Y219 T313 G314 S315 S90 K93 Y177 E299 K342 S345 S60 K63 Y147 E269 K312 S315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P24735 26089439 401 MDRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGL 4x69 A 1.42 BS01 OP0 A 1 S70 N104 S130 N132 N170 T235 G236 S237 S43 N77 S103 N105 N143 T208 G209 S210 S70 K73 S130 E166 K234 S237 S43 K46 S103 E139 K207 S210 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q47066 26089439 301 NSVQQQLEALEKSSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKQSESDKHLLNQRVEIKKSDLVNYNPIAEKHVNGTMTLAELGAAALQYSDNTAMNKLIAHLGGPDKVTAFARSLGDETFRLDRTEPTLNTAIPGDPRDTTTPLAMAQTLKNLTLGKALAETQRAQLVTWLKGNTTGSASIRAGLPKSWVVGDKTGSGDYGTTNDIAVIWPENHAPLVLVTYFTQPEQKAERRRDILAAAAKIVTHGF 4x6i A 1.87 BS01 3Y1 A 1 G65 G66 Y67 N161 G65 G66 Y67 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 Ki=10nM remove_due_to_license_issue Ki=10.0nM P43235 26280490 301 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 4x6j A 1.59 BS01 3Y2 A 1 G23 C25 G65 G66 Y67 N161 G23 C25 G65 G66 Y67 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 26280490 307 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 4x6k A 1.94 BS01 3XR A 1 R257 D282 I338 D339 R575 R637 Y677 R19 D44 I100 D101 R337 R399 Y439 0004308 ic50=0.00487mM remove_due_to_license_issue 26154892 802 ADISNIFYAGDATKSNYFRIPSLLALDSGTVIAAADARYGGTHDAKSKINTAFAKSTDGGKTWGQPTLPLKFDDYVAKNIDWPRDSVGKNVQIQGSASYIDPVLLEDKETHRVFLFADMMPAGIGSSNASVGSGFKEVDGKKYLKLHWKDDAAGTYDYSVRENGTIYNDTTNSATEYSVDGEYNLYKNGNAMLCKQYDYNFEGTKLLETQTDTDVNMNVFYKDADFKVFPTTYLAMKYSDDEGETWSDLQIVSTFKPEESKFLVLGPGVGKQIANGEHAGRLIVPLYSKSSAELGFMYSDDHGNNWTYVEADQNTGGATAEAQIVEMPDGSLKTYLRTGSGYIAQVMSTDGGETWSERVPLTEIATTGYGTQLSVINYSQPVDGKPAILLSAPNATNGRKNGKIWIGLISETGNSGKDKYSVDWKYCYSVDTPQMGYSYSCLTELPDGEIGLLYEKYDSWSRNELHLKNILKYERFNIDELKVQP 4x6m A 2.4 BS01 3Y3 A 1 R39 H40 C42 H57 Y143 I151 D189 A190 C191 K192 G193 S195 T213 S214 W215 G218 G226 V227 Y228 R26 H27 C29 H44 Y134 I141 D182 A183 C184 K185 G186 S188 T206 S207 W208 G211 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=5.8nM remove_due_to_license_issue Ki=5.8nM P03951 25728130 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4x6n A 2.1 BS02 3Y5 A 1 R39 H40 C42 H57 Y143 I151 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 Y228 R26 H27 C29 H44 Y134 I141 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=1.5nM remove_due_to_license_issue Ki=1.5nM P03951 25728130 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4x6o A 2.1 BS01 3Y4 A 1 R39 H40 L41 C42 H57 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 Y228 R26 H27 L28 C29 H44 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=1.9nM remove_due_to_license_issue IC50=3.60nM P03951 25728130 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4x6p A 1.93 BS01 3YU A 1 H40 H57 Y143 I151 D189 A190 C191 K192 G193 S195 W215 G216 G218 C219 G226 V227 Y228 H27 H44 Y134 I141 D182 A183 C184 K185 G186 S188 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=5nM remove_due_to_license_issue Ki=5.0nM P03951 25728130 302 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYTDSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQ 4x6x A 1.8 BS01 S74 A 1 F267 D335 W336 P361 I363 Y383 F387 M419 Y466 V498 L499 M503 H524 W525 F38 D106 W107 P132 I134 Y154 F158 M190 Y237 V269 L270 M274 H295 W296 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F38 H105 D106 W107 N130 N149 Y154 Y237 D267 H295 3.1.3.76,3.3.2.10 0003824 ic50=2.3nM remove_due_to_license_issue IC50=2.3nM P34913 25800114 601 TSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD 4x6y A 2.1 BS01 S94 A 1 F267 D335 W336 M339 Y383 L408 Y466 L499 M503 H524 F38 D106 W107 M110 Y154 L179 Y237 L270 M274 H295 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F38 H105 D106 W107 N130 N149 Y154 Y237 D267 H295 3.1.3.76,3.3.2.10 0003824 remove_due_to_license_issue IC50=18nM P34913 25800114 601 TSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD 4x7h A 2.0 BS01 3Z2 A 1 L599 A620 K622 E639 I886 M888 C891 K893 H935 F944 G954 D955 L15 A36 K38 E55 I85 M87 C90 K92 H134 F143 G153 D154 N937 K939 N942 D955 T987 N136 K138 N141 D154 T157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=42nM Q9NZJ5 25587754 1101 YISRYLTDFEPIQCLGRGGFGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEAPPKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRNLKPSNIFFTMDDVVKVGDFGTKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDLDFPGKT 4x7i A 1.77 BS01 3YS A 1 S10 Q12 G13 L30 D32 S35 Y71 F108 D228 G230 T231 T232 S15 Q17 G18 L35 D37 S40 Y76 F113 D233 G235 T236 T237 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=20nM P56817 25609634 401 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMDCGYN 4x7j A 2.3 BS01 3Z1 A 1 A620 K622 L643 M888 C891 G954 D955 F956 A36 K38 L59 M87 C90 G153 D154 F155 N937 K939 N942 D955 N136 K138 N141 D154 2.7.11.1 0004672,0005524,0006468 ic50=41nM remove_due_to_license_issue IC50=1200nM, EC50=310nM Q9NZJ5 25587754 1101 YISRYLTDFEPIQCLGRGGFGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEAPPKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRNLKPSNIFFTMDDVVKVGDFGLVKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDLDFPGKT 4x7k A 1.8 BS01 3Z3 A 1 A620 K622 E639 L643 V652 I886 M888 C891 G954 D955 F956 A36 K38 E55 L59 V68 I85 M87 C90 G153 D154 F155 N937 K939 N942 D955 T987 N136 K138 N141 D154 T160 2.7.11.1 0004672,0005524,0006468 ic50=4nM remove_due_to_license_issue Q9NZJ5 25587754 1101 YISRYLTDFEPIQCLGRGGFGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEAPPKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRNLKPSNIFFTMDDVVKVGDFGLVTTKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDLDFPGKTV 4x7l A 1.9 BS01 3Z4 A 1 A620 K622 E639 L643 V652 I886 M888 C891 G954 D955 F956 A36 K38 E55 L59 V68 I85 M87 C90 G153 D154 F155 N937 K939 N942 D955 T987 N136 K138 N141 D154 T160 2.7.11.1 0004672,0005524,0006468 ic50=9nM remove_due_to_license_issue IC50=1300nM, EC50=200nM Q9NZJ5 25587754 1101 YISRYLTDFEPIQCLGRGGFGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEAPPKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRNLKPSNIFFTMDDVVKVGDFGLVTTKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDLDFPGKTV 4x7n A 2.35 BS01 3Z5 A 1 A620 K622 E639 L643 V652 I886 M888 C891 G954 D955 F956 A36 K38 E55 L59 V68 I84 M86 C89 G152 D153 F154 N937 K939 N942 D955 T987 N135 K137 N140 D153 T159 2.7.11.1 0004672,0005524,0006468 ic50=6nM remove_due_to_license_issue IC50=>50000nM, EC50=400nM Q9NZJ5 25587754 1101 YISRYLTDFEPIQCLGRGGFGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEAPKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRNLKPSNIFFTMDDVVKVGDFGLVTTKLYMSPEQIHGNSYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDLDFPGKTV 4x7o A 2.65 BS01 3Z6 A 1 V640 L643 A644 V652 Y654 I886 M888 C891 F944 D955 V54 L57 A58 V66 Y68 I83 M85 C88 F141 D152 N937 K939 N942 D955 T987 N134 K136 N139 D152 T155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9NZJ5 25587754 1101 YISRYLTDFEPIQCLGRGGVVFEAKNKVDDCNYAIKRIRLPNRELAREKVMREVKALAKLEHPGIVRYFNAWLEAPPKVYLYIQMQLCRKENLKDWMNGRCTIEERERSVCLHIFLQIAEAVEFLHSKGLMHRNLKPSNIFFTMDDVVKVGDFGTKLYMSPEQIHYSHKVDIFSLGLILFELLYPFSTQMERVRTLTDVRNLKFPPLFTQKYPCEYVMVQDMLSPSPMERPEAINIIENAVFEDLD 4x7q B 2.33 BS01 3YR B 1 F43 V46 A59 K61 E117 R118 A122 D124 E167 L170 I181 D182 F16 V19 A32 K34 E73 R74 A78 D80 E123 L126 I137 D138 D163 K165 N168 D182 T200 D119 K121 N124 D138 T156 2.7.11.1 0000082,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0006338,0006468,0006915,0007346,0008285,0008637,0009615,0010508,0016236,0016239,0035175,0035402,0035403,0035979,0043066,0043123,0044022,0044023,0044024,0044025,0045893,0050821,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=14nM remove_due_to_license_issue IC50=14nM Q9P1W9 25575657 401 AFEAEYRLGPLLGKGFGTVFAGHRLTDRLQVAIKVIPRCPLEVALLWKVGAGGGHPGVIRLLDWFETFMLVLERPLPAQDLFDYITEKGPLGEGPSRCFFGQVVAAIQHCHSRGVVHRDIKDENILIDLRRGCAKLIDFGSGALLHDEPYTDFDGTRVYSPPEWISRHQYHALPATVWSLGILLYDMVCGDIPFERDQEILEAELHFPAHVSPDCCALIRRCLAPKPSSRPSLEEILLDPWMQ 4x8g A 3.29 BS05 3Z0 A 1 H471 D473 E474 A581 F582 F583 P584 N585 N588 F634 V643 H416 D418 E419 A526 F527 F528 P529 N530 N533 F579 V586 D350 H471 D473 A645 D310 H416 D418 A588 3.5.3.15 0004668,0005509,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0006338,0016787,0019827,0032991,0036211,0042802,0043687,0045087,0046872,0140794,0140795,0140796,0140797,0140798,0140809,0140810,0140811 remove_due_to_license_issue Q9UM07 25622091 705 QGTLIRVTPEQPTHAVCVLGTLTQLDICSSAPEDCTSFSINASPGVVVDIASTWPLDPGVEVTLTMKVASGSTGDQKVQISYYPVKALLYLTGVEISLCADITRTGKVKPTAVKDQRTWTWGPCGQGAILLVNCDRDNLESSAMDCEDDEVLDSEDLQDMSLMTLSTKTPKDFFTNHTLVLHVARSEMDKVRVFQATKCSVVLGPKWPSHYLMVPGGKHNMDFYVEALAFPDTDFPGLITLTISLLDTSNLELPEAVVFQDSVVFRVAPWIMTPNTQPPQEVYACFENEDFLKSVTTLAMKAKCKLTIQDEMEIGYIQAPHKTLPVVFDSPRKRVMGPDFGYVTRISGLDSFGNLEVSPPVTVRGKEYPLGRILFGDSCYPSNDSRQMHQALQDFLSAQQVQAPVKLYSDWLSVGHVDEFLSFVPAPDRKGFRLLLASPRSCYKLFQEQQNEGHGEALLFEGIKKKKQQKIKNILSNKTLREHNSFVERCIDWNRELLKRELGLAESDIIDIPQLFKLKEFSKAEAFFPNMVNMLVLGKHLGIPKPFGPVINGRCCLEEKVCSLLEPLGLQCTFINDFFTYHIGEVHAGTNVRRKPFSFKWWNMVP 4x8o A 2.1 BS01 AP5 A 1 G10 G12 K13 G14 T15 T31 G32 L35 R36 M53 K57 L58 V59 V64 R88 Q92 R119 R123 V132 Y133 H134 F137 R156 R167 V202 G10 G12 K13 G14 T15 T31 G32 L35 R36 M53 K57 L58 V59 V64 R88 Q92 R119 R123 V132 Y133 H134 F137 R156 R167 V202 K13 R88 R123 R156 R167 K13 R88 R123 R156 R167 2.7.4.3 0000287,0004017,0004550,0005515,0005524,0005737,0005829,0006139,0006172,0009123,0009132,0009165,0015951,0016208,0016301,0016776,0019205,0044209,0046083,0046940,0050145 Kd=250nM remove_due_to_license_issue P69441 26138143 301 MRIILLGAPGAGKGTQAQFIMEKYGIPQISTGDMLRAAVKSGSELGKQAKDIMDAGKLVTDELVIALVKERIAQEDCRNGFLLDGFPRTIPQADAMKEAGINVDYVLEFDVPDELIVDRIVGRRVHAPSGRVYHVKFNPPKVEGKDDVTGEELTTRKDDQEETVRKRLVEWHQMTAPLIGYYSKEAEAGNTKYAKVDGTKPVAEVRADLEKILG 4x8s H 2.1 BS01 3Z7 H 1 D189 S190 K192 V213 W215 G216 G219 G226 V227 Y228 D181 S182 K184 V205 W207 G208 G210 G218 V219 Y220 3.4.21.21 0004252,0006508 Ki=13mM remove_due_to_license_issue Ki=13000000nM P08709 25764119 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4x8t H 2.2 BS01 3Z8 H 1 D189 S190 K192 S195 S214 W215 G216 G219 C220 D182 S183 K185 S188 S207 W208 G209 G211 C212 3.4.21.21 0004252,0006508 Ki=8.9mM remove_due_to_license_issue Ki=8900000nM P08709 25764119 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4x8u H 2.1 BS01 3ZB H 1 D189 S190 K192 V213 W215 G219 G226 V227 Y228 D183 S184 K186 V207 W209 G212 G220 V221 Y222 3.4.21.21 0004252,0006508 Ki=3.5mM remove_due_to_license_issue Ki=3500000nM P08709 25764119 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4x8v H 2.5 BS01 3Z9 H 1 H57 K60A G97 T99 D189 S190 K192 S195 S214 W215 G216 G219 H41 K45 G85 T87 D186 S187 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=130nM remove_due_to_license_issue Ki=130nM P08709 25764119 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4x9j A 1.412 BS01 dna B 0 R114 R118 E121 R124 R142 R146 H149 H153 T156 R174 E177 R180 R13 R17 E20 R23 R41 R45 H48 H52 T55 R73 E76 R79 ? remove_due_to_license_issue P18146 25999311 1 ~ 11 ERPYACPVESCDRRFSRSDELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLR 4x9j A 1.412 BS02 dna C 0 D120 D148 K179 D19 D47 K78 ? remove_due_to_license_issue P18146 25999311 51 ~ 61 ERPYACPVESCDRRFSRSDELTRHIRIHTGQKPFQCRICMRNFSRSDHLTTHIRTHTGEKPFACDICGRKFARSDERKRHTKIHLR 4xaq A 2.21 BS01 40F A 1 R57 R61 S143 Y144 S145 A166 S167 T168 Y216 D295 K377 R36 R40 S99 Y100 S101 A122 S123 T124 Y172 D251 K333 ? 0004930,0007186,0016020 Ki=71.7nM remove_due_to_license_issue Ki=72nM, EC50=5.1nM, IC50=5.6nM Q14416 25602126 601 AKKVLTLEGDLVLGGLFPVHQKGGPAEDCGPVNEHRGIQRLEAMLFALDRINRDPHLLPGVRLGAHILDSCSKDTHALEQALDFVRASLTAITGVIGGSYSDVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFFQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFELEARARNISVATSEKVGRAMSRAAFEGVVRALLQKPSARVAVLFTRSEDARELLAASQRLNASFTWVASDGWGALEEVVAGSEGAAEGAITIELASYPISDFASYFQSLDPWNNSRNPWFREFWEQRFRCSFRQRDCAAHSLRAVPFEQESKIMFVVNAVYAMAHALHNMHRALCPNTTRLCDAMRPVNGRRLYKDFVLNVKFDAPFRPADTHNEVRFDRFGDGIGRYNIFTYLRAGSGRYRYQKVGYWAEGLTLDTSLIPW 4xar A 2.26 BS01 40F A 1 R64 R68 S149 Y150 S151 A172 S173 T174 Y222 D301 G302 K389 R35 R39 S98 Y99 S100 A121 S122 T123 Y171 D250 G251 K331 ? 0004930,0007186,0016020 Ki=107nM remove_due_to_license_issue EC50=38nM, Ki=93nM Q14832 25602126 601 RREIKIEGDLVLGGLFPINEKGTGTEECGRINEDRGIQRLEAMLFAIDEINKDDYLLPGVKLGVHILDTCSRDTYALEQSLEFVRASLLLIAGVIGGSYSSVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFYQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFEQEARLRNISIATAEKVGRSNIRKSYDSVIRELLQKPNARVVVLFMRSDDSRELIAAASRANASFTWVASDGWGAQESIIKGSEHVAYGAITLELASQPVRQFDRYFQSLNPYNNHRNPWFRDFWEQKFQCSLRVCDKHLAIDSSNYEQESKIMFVVNAVYAMAHALHKMQRTLCPNTTKLCDAMKILDGKKLYKDYLLKINFTAPDADSIVKFDTFGDGMGRYNVFNFQNVGGKYSYLKVGHWAETLSLDVNSIHWSRNSVPTSE 4xas A 2.35 BS01 40H A 1 R57 R61 S143 Y144 S145 A166 T168 Y216 R271 D295 K377 R35 R39 S97 Y98 S99 A120 T122 Y170 R225 D249 K331 ? 0004930,0007186,0016020 Ki=260nM remove_due_to_license_issue Q14416 25602126 601 KKVLTLEGDLVLGGLFPVHQKGGPAEDCGPVNEHRGIQRLEAMLFALDRINRDPHLLPGVRLGAHILDSCSKDTHALEQALDFVRASTAITGVIGGSYSDVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFFQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFELEARARNISVATSEKVGRAMSRAAFEGVVRALLQKPSARVAVLFTRSEDARELLAASQRLNASFTWVASDGWGALEEVVAGSEGAAEGAITIELASYPISDFASYFQSLDPWNNSRNPWFREFWEQRFRCSFRQRDCAAHSLRAVPFEQESKIMFVVNAVYAMAHALHNMHRALCPNTTRLCDAMRPVNGRRLYKDFVLNVKFDAPFRPADTHNEVRFDRFGDGIGRYNIFTYLRAGGRYRYQKVGYWAEGLTLDTSLIPW 4xbb A 1.85 BS01 3ZR A 1 H30 E54 Q110 T134 C139 A158 A159 A160 H32 E56 Q112 T126 C131 A150 A151 A152 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 25761614 201 HMAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 4xbd A 1.45 BS01 M40 A 1 H30 E54 Q110 R112 T134 C139 H157 A158 A159 A160 H32 E56 Q112 R114 T127 C132 H150 A151 A152 A153 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 25761614 201 HMAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGTIPGDCGAPYVHKRGNDWVVCGVHAAATNTVVCAVQA 4xbo A 2.6 BS01 SAH A 1 T79 S80 A81 G114 R115 I134 S142 L143 A148 T79 S80 A81 G114 R115 I134 S142 L143 A148 2.1.1.200 0002128,0003723,0005737,0005829,0006396,0008033,0008168,0008173,0032259,0042803,0160206 remove_due_to_license_issue P0AE01 26202969 301 MLQNIRIVLVETSHTGNMGSVARAMKTMGLTNLWLVNPLVKPDSQAIALAAGASDVIGNAHIVDTLDEALAGCSLVVGTSARSRTLPWPMLDPRECGLKSVAEAANTPVALVFGRERVGLTNEELQKCHYHVAIAANPEYSSLNLAMAVQVIAYEVRMAWLATQTPYPLVDDLERFYGHLEQTLLATGFIRENHPGQVMNKLRRLFTRARPESQELNILRGILASIEQ 4xbo B 2.6 BS01 SAH B 1 T79 S80 A81 F113 G114 R115 G119 I134 S142 L143 A148 T72 S73 A74 F106 G107 R108 G112 I127 S135 L136 A141 2.1.1.200 0002128,0003723,0005737,0005829,0006396,0008033,0008168,0008173,0032259,0042803,0160206 remove_due_to_license_issue P0AE01 26202969 301 MLQNIRIVLVETSHTGNMGSVARAMKTMGLTNLWLVNPLVKPAAGASDVIGNAHIVDTLDEALAGCSLVVGTSARSRTLPWPMLDPRECGLKSVAEAANTPVALVFGRERVGLTNEELQKCHYHVAIAANPEYSSLNLAMAVQVIAYEVRMAWLATQENETPYPLVDDLERFYGHLEQTLLATGFIRENHPGQVMNKLRRLFTRARPESQELNILRGILASIEQQN 4xcb A 1.6 BS02 HY0 A 1 R51 E87 H102 K137 W232 E234 D249 E254 R54 E90 H105 K140 W235 E237 D252 E257 ? 0016491,0046872 remove_due_to_license_issue Q2MFS1 26240321 303 LHMVPALTREQLYIFDTTGFLVIPGVFGSGEVESFRSELERLDTVDPGFPRTRRYPDLPAASPVFARLALDDRLLAPVRDVVNQPLRLLEGYGLRRTKDSVLYLHGGNSELLDLGDRQVGRDLSITHTYHDGKLYCPYVKALVYLSDIQSPEDGSFCYVQGSHKANFPLLRERAERGENTSLVDSGFPTLSDVFVRSGDVLLLNEALMHGTRRKLTEGDRLLTAFGYGPTFFTEWRELDAETADLRGAGYVDHDVEEDFV 4xct A 1.3 BS01 N73 A 1 L187 A189 L222 H226 E227 H230 H236 L243 Y245 P246 M247 Y248 L75 A77 L110 H114 E115 H118 H124 L131 Y133 P134 M135 Y136 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 ic50=6.7nM remove_due_to_license_issue P14780 26263024 301 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4xcu A 1.71 BS01 40M A 1 K503 E520 M524 V550 C552 A553 G556 L619 A629 D630 K48 E65 M69 V95 C97 A98 G101 L155 A165 D166 D612 A614 R616 N617 D630 R650 D148 A150 R152 N153 D166 R186 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 25776529 1002 DLPLDPLWEFPRDRLVLGKPLGEGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAVSH 4xe0 A 2.434 BS01 40L A 1 M752 P758 W760 I777 Y813 E826 V828 T833 N836 M900 I910 M552 P558 W560 I577 Y613 E626 V628 T633 N636 M700 I710 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=19nM remove_due_to_license_issue O35904 25631052 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILEYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRE 4xe1 A 1.8 BS03 IL5 A 1 H94 H119 F131 L198 T199 T200 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=77.3nM remove_due_to_license_issue P00918 25733161 305 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4xg3 A 2.3 BS01 X3G A 1 L377 V385 A400 M448 M450 A451 G454 P455 K458 R498 L501 D512 L15 V18 A33 M76 M78 A79 G82 P83 K86 R126 L129 D140 D494 A496 R498 N499 D512 K533 D122 A124 R126 N127 D140 K161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=17.5nM remove_due_to_license_issue P43405 27504936 701 VYLDRKLLTLEDKELGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV 4xg4 A 2.3 BS01 X4G A 1 L377 V385 A400 M448 M450 A451 G454 P455 R498 N499 L501 D512 L15 V23 A38 M81 M83 A84 G87 P88 R131 N132 L134 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 ic50=21.5nM remove_due_to_license_issue P43405 27504936 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 4xg6 A 2.4 BS01 X6G A 1 L377 V385 A400 M448 A451 G454 R498 L501 D512 L15 V23 A38 M86 A89 G92 R136 L139 D150 D494 A496 R498 N499 D512 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=9.7nM remove_due_to_license_issue IC50=7.3nM P43405 27504936 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNL 4xg7 A 1.76 BS01 X7G A 1 L377 A400 M448 M450 A451 G454 P455 R498 L501 D512 L14 A32 M78 M80 A81 G84 P85 R128 L131 D142 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=32.6nM remove_due_to_license_issue IC50=20nM P43405 27504936 701 YLDRKLLTLEDKELGTVKKGYYQMKKVVKTVAVKILKNEAPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNL 4xg8 A 2.4 BS01 X8G A 1 L377 A400 M448 M450 A451 P455 R498 L501 D512 L12 A31 M74 M76 A77 P81 R124 L127 D138 D494 A496 R498 N499 D512 D120 A122 R124 N125 D138 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.9nM remove_due_to_license_issue IC50=11.1nM P43405 27504936 700 DRKLLTLEDKELGSGGTVKKGYYQMVVKTVAVKILDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 4xg9 A 2.91 BS01 X9G A 1 L377 V385 A400 M448 M450 A451 G454 P455 R498 N499 L501 D512 L15 V23 A38 M81 M83 A84 G87 P88 R131 N132 L134 D145 D494 A496 R498 N499 D512 D127 A129 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1nM P43405 27504936 700 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYD 4xh6 A 2.04 BS01 HUL A 1 L44 A65 K67 I104 L120 I185 D186 L12 A33 K35 I72 L88 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=2.71uM remove_due_to_license_issue IC50=2710nM P11309 26275107 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4xhe A 1.9 BS01 40P A 1 Y93 W147 V148 Y188 Y195 Y101 W155 V156 Y196 Y203 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 YKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4xhe A 1.9 BS02 40P B 1 T36 Y55 I118 T44 Y63 I126 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 YKDDDDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4xhe E 1.9 BS01 40P A 1 Y55 I118 S167 Y58 I121 S170 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4xhe E 1.9 BS02 40P E 1 Y93 W147 V148 Y195 Y96 W150 V151 Y198 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 DKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 4xhk B 1.9 BS01 3YR B 1 L44 F49 A65 K67 E121 R122 V126 L174 I185 D186 L13 F18 A34 K36 E86 R87 V91 L139 I150 D151 N172 D186 L193 N137 D151 L158 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=5nM remove_due_to_license_issue IC50=5.0nM P11309 25575657 401 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 4xhl A 3.01 BS01 CKI A 1 I15 I23 A36 L85 D91 L135 I148 I11 I14 A27 L76 D82 L126 I139 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P29295 27491543 401 VGRKFRIGRKIGDIYHGTNLISGEEVAIRLESIRSRHPQLDYESRVYRYLSGGVGIPFIRWFGREGEYNAMVIDLLGPSLEDLFNYCHRRFSFKTVIMLALQMFCRIQYIHGRSFIHRDIKPDNFLMGVGRRGSTVHVIDFGLSKKYRDFNTHRHIPYRENKSLTGTARYASVNTHLGIEQSRRDDLESLGYVLIYFCKGSLPWQGLKATTKKQKYDRIMEKKLNVSVETLCSGLPLEFQEYMAYCKNLKFDEKPDYLFLARLFKDLSIKLEYHNDHLFDWTMLRYTKAMTFNKIKLLAMKKFPTHFHYYKNEDKHNPSPEEIKQQTILN 4xic A 2.69 BS01 dna B 0 K2 R5 Y25 R31 Q50 R53 M54 K57 K1 R4 Y24 R30 Q49 R52 M53 K56 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 0 ~ 14 KRGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xic A 2.69 BS02 dna C 0 R3 R5 Q6 Y8 R43 I47 N51 R2 R4 Q5 Y7 R42 I46 N50 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 23 ~ 37 KRGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xic D 2.69 BS01 dna E 0 R5 T7 Y25 R28 R31 Q50 R53 M54 R1 T3 Y21 R24 R27 Q46 R49 M50 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 0 ~ 14 RQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xic D 2.69 BS02 dna F 0 R5 Q6 Y8 Q44 I47 N51 R1 Q2 Y4 Q40 I43 N47 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 23 ~ 37 RQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xid A 2.701 BS01 dna B 0 R3 R5 Y25 R28 R31 K46 Q50 R53 K57 R1 R3 Y23 R26 R29 K44 Q48 R51 K55 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 0 ~ 14 RGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xid A 2.701 BS02 dna C 0 R3 R5 Q6 Y8 I47 N51 R1 R3 Q4 Y6 I45 N49 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 24 ~ 38 RGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xid A 2.701 BS03 dna F 0 R28 R29 R30 R26 R27 R28 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 24 ~ 38 RGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xid D 2.701 BS01 dna E 0 R5 T7 Y25 R28 R31 K46 Q50 R53 M54 R1 T3 Y21 R24 R27 K42 Q46 R49 M50 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 0 ~ 14 RQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xid D 2.701 BS02 dna F 0 R5 Q6 Y8 I47 N51 K55 R1 Q2 Y4 I43 N47 K51 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 26331260 24 ~ 38 RQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 4xii A 2.7 BS01 40V A 1 N68 I69 D70 W82 G116 G117 E197 S198 W231 F329 Y332 H438 N66 I67 D68 W80 G114 G115 E195 S196 W229 F327 Y330 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue IC50=215nM P06276 26116179 1001 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 4xip A 1.7 BS01 40W A 1 M98 F138 Y139 W162 M83 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=235nM remove_due_to_license_issue Ki=235nM P07900 25677667 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4xiq A 1.84 BS01 40Y A 1 N51 M98 L107 F138 Y139 W162 N36 M83 L92 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=86nM remove_due_to_license_issue Ki=86nM P07900 25677667 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 4xir A 1.7 BS01 40X A 1 M98 L107 F138 Y139 W162 T184 M83 L92 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=115nM remove_due_to_license_issue Ki=115nM P07900 25677667 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4xit A 1.86 BS01 40Z A 1 K58 M98 L107 F138 Y139 W162 T184 K43 M83 L92 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Ki=41nM remove_due_to_license_issue P07900 25677667 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4xj0 A 2.58 BS01 41B A 1 E33 G37 V39 A52 K54 Q105 D106 M108 T110 K114 N154 L156 D167 E22 G26 V28 A41 K43 Q94 D95 M97 T99 K103 N143 L145 D156 D149 K151 S153 N154 D167 T190 D138 K140 S142 N143 D156 T179 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue IC50=3.9nM, Ki=0.600000nM P28482 25603482 401 EMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQPGYRS 4xjr A 3.0 BS02 OEL A 1 R192 T193 E276 Y319 Y337 E409 R424 R502 Y530 R52 T53 E133 Y176 Y194 E266 R281 R359 Y387 3.2.1.18 0004308,0019031,0019058,0046789 remove_due_to_license_issue P08492 25676091 606 RITHDVGIKPLNPDDFWRCTSGLPSLMKTPKIRLMPGPGLLAMPTTVDGCVRTPSLVINDLIYAYTSNLITRGCQDIGKSYQVLQIGIITVNVPDLNPRISHTFNINDNRKSCSLALLNTDVYQLCSTPKVDERSDYASSGIEDIVLDIVNHDGSISTTRFKNNNISFDQPYAALYPSVGPGIYYKGKIIFLGYGGLEHPINENAICNTTGCPGKTQRDCNQASHSPWFSDRRMVNSIIVVDKGLNSIPKLKVWTISMRQNYWGSEGRLLLLGNKIYIYTRSTSWHSKLQLGIIDITDYSDIRIKWTWHNVLSRPGNNECPWGHSCPDGCITGVYTDAYPLNPTGSIVSSVILDSQKSRVNPVITYSTATERVNELAIRNKTLSAGYTTTSCITHYNKGYCFHIVEINHKSLDTFQPMLFKTEIPKSCS 4xjs A 2.8 BS01 733 A 1 E146 D155 S186 W189 D219 S220 T221 E101 D110 S141 W144 D174 S175 T176 E146 T221 E226 E101 T176 E181 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue IC50=76nM P28907 26267483 401 WRQQWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFATSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVEVHNLQPEKVQTLEAWVIHGSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCV 4xjt A 2.6 BS01 41Z A 1 W125 E146 D155 S186 W189 K190 T221 W80 E101 D110 S141 W144 K145 T176 E146 T221 Q226 E101 T176 Q181 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue IC50=7200nM P28907 26267483 401 WRQQWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFATSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVQVHNLQPEKVQTLEAWVIHGSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKN 4xk9 A 2.2 BS01 41J A 1 Y93 W147 V148 Y188 Y195 Y95 W149 V150 Y190 Y197 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 KLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4xk9 E 2.2 BS01 41J A 1 T36 Y55 I118 T40 Y59 I122 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4xk9 E 2.2 BS02 41J E 1 Y93 W147 V148 Y188 C191 Y195 Y97 W151 V152 Y192 C195 Y199 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 26004441 301 DDKLHSQANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKADSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGATCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 4xkb A 1.501 BS01 DE9 A 1 R113 W183 W189 W192 F196 N211 Q212 L213 R105 W175 W181 W184 F188 N203 Q204 L205 ? 0046906 remove_due_to_license_issue P72583 25958236 300 DNLTELSQQLKQLTAIAALAEMGEGGQGILLDYLAKNVPLEKPVLAVGNVYQTLRNLEQETITTQLQRNYPTGIFPLQSAQGIDYLPLQEALGSQDFETADEITRDKLCELAGPGASQRQWLYFTEVEKFPALDLHTINALWWLHSNGNFGFSVQRRLWLASGKEFTKLWPKIGWKSGNVWTRWPKGFTWDLSAPQGHLPLLNQLRGVRVAESLYRHPVWSQYGW 4xkc A 2.0 BS01 MD9 A 1 R113 W183 W189 W192 F196 N211 Q212 L213 R105 W175 W181 W184 F188 N203 Q204 L205 ? 0046906 remove_due_to_license_issue P72583 25958236 300 NLTELSQQLHKQLTAIAALAEMGEGGQGILLDYLAKNVPLEKPVLAVGNVYQTLRNLEQETITTQLQRNYPTGIFPLQSAQGIDYLPLQEALGSQDFETADEITRDKLCELAGPGASQRQWLYFTEVEKFPALDLHTINALWWLHSNGNFGFSVQRRLWLASGKEFTKLWPKIGWKSGNVWTRWPKGFTWDLSAPQGHLPLLNQLRGVRVAESLYRHPVWSQYGW 4xkx A 1.8 BS01 43K A 1 G11 Q12 G13 L30 D32 G34 S35 Y71 F108 I118 R128 Y198 D228 G230 G13 Q14 G15 L32 D34 G36 S37 Y73 F110 I120 R130 Y189 D219 G221 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.9nM remove_due_to_license_issue IC50=21nM P56817 25613679 405 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4xm6 A 2.352 BS01 41R A 1 K656 G657 L668 G674 V675 L677 G683 H686 E687 Y728 E735 K366 G367 L378 G384 V385 L387 G393 H396 E397 Y438 E445 H686 E687 H690 Y728 E735 H396 E397 H400 Y438 E445 3.4.24.83 0008237 ic50=90uM remove_due_to_license_issue P15917 26578066 801 SRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSLSTEEKEFLKKLQIDLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4xm7 A 2.7 BS01 41S A 1 S655 K656 G657 L668 L677 G683 H686 E687 H690 Y728 S388 K389 G390 L401 L410 G416 H419 E420 H423 Y461 H686 E687 H690 Y728 E735 H419 E420 H423 Y461 E468 3.4.24.83 0008237 remove_due_to_license_issue P15917 26578066 801 LSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDEEEKELLNRIQVDSSNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINSL 4xm8 A 2.7 BS01 41T A 1 S655 K656 G657 G674 V675 L677 N679 G683 H686 E687 H690 Y728 E735 S379 K380 G381 G398 V399 L401 N403 G407 H410 E411 H414 Y452 E459 H686 E687 H690 Y728 E735 H410 E411 H414 Y452 E459 3.4.24.83 0008237 remove_due_to_license_issue P15917 26578066 801 SRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSSTEEKEFLKKLQIDIRDSLSEEEKELLNPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 4xmb A 2.428 BS01 41P A 1 Y334 S363 G364 R380 N414 R415 I461 S508 G509 Y525 Q530 S555 A556 F577 S602 G603 Y11 S40 G41 R57 N91 R92 I138 S185 G186 Y202 Q207 S232 A233 F254 S279 G280 ? Kd=44nM remove_due_to_license_issue Ki=53nM, IC50=44nM, Kd=44nM, EC50=12000nM Q14145 26363505 701 VGRLIYTAGGYFRQSLSYLEAYNPSDGTWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVT 4xmo A 1.75 BS01 46G A 1 I1084 A1108 Y1159 M1160 D1164 R1208 N1209 M1211 A1221 D1222 Y1230 I34 A52 Y103 M104 D108 R152 N153 M155 A165 D166 Y174 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A187 2.7.10.1 0004672,0004713,0005524,0006468 ic50=2nM remove_due_to_license_issue IC50=3.0nM P08581 25699405 1401 VHIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 4xmr A 1.3 BS01 ILE A 1 Y118 K149 W151 Y167 D169 T170 D196 Y82 K109 W111 Y127 D129 T130 D156 ? remove_due_to_license_issue Q0P864 26457436 301 GIDPFTKTSLYESTLKNQTDLLKVTQSTVEDFRSTNQSFTRALEKDIANLPYQSLITEENIINNVGPILKYYRHSINALNVYLGLNNGKVLLSQKSMPELRDDLDIKTKDWYQEALKTNDIFVTPAYLDTVLKQYVITYSKAIYKDGKIIGVLGVDIPSEDLQNLVAKTPGNTFLFDQKNKIFAATNKELLNPSIDHSPVLNAYKLNGDNNFFSYKLNNEERLGACTKVFAYTACITESADIINK 4xnv A 2.2 BS01 BUR A 1 F62 F66 L102 T103 P105 A106 F119 M123 L126 Q127 F24 F28 L64 T65 P67 A68 F81 M85 L88 Q89 ? 0004930,0005506,0007186,0007200,0009055,0016020,0030168,0043448,0045028,0046872,0090075 Ki=161nM remove_due_to_license_issue P00268,P47900 25822790 1101 SFKCALTKTGFQFYYLPAVYILVFIIGFLGNSVAIWMFVFHMKPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDAMCKLQRFIFHVNLYGSILFLTCISAHRYSGVVYPKSLGRLKKKNAICISVLVWLIVVVAISPILFYSGTGVRKNKTITCYDTTSDEYLRSYFIYSMCTTVAMFCVPLVLILGCYGLIVRALIYKMKKYTCTVCGYIYNPEDGDPDNGVNPGTDFKDIVCPLCGVGKDQFEEVEEPLRRKSIYLVIIVLTVFAVSYIPFHVMKTMNLRARLDFQTPAMCAFNDRVYATYQVTRGLASLNSCVNPILYFLAGDTFRRR 4xnw A 2.7 BS01 2ID A 1 C42 L44 K46 R195 D204 T205 N283 R287 Q291 N299 Y303 Y306 R310 C5 L7 K9 R158 D167 T168 N295 R299 Q303 N311 Y315 Y318 R322 ? 0004930,0005506,0007186,0007200,0009055,0016020,0030168,0043448,0045028,0046872,0090075 remove_due_to_license_issue P00268,P47900 25822790 1101 SSFKCALTKTGFQFYYLPAVYILVFIIGFLGNSVAIWMFVFHMKPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDAMCKLQRFIFHVNLYGSILFLTCISAHRYSGVVYPLKSLGRLKKKNAICISVLVWLIVVVAISPILFYSGTGVRKNKTITCYDTTSDEYLRSYFIYSMCTTVAMFCVPLVLILGCYGLIVRALIYKMKKYTCTVCGYIYNPEDGDPDNGVNPGTDFKDIPDDWVCPLCGVGKDQFEEVEEPLRRKSIYLVIIVLTVFAVSYIPFHVMKTMNLRARLDFQTPAMCAFNDRVYATYQVTRGLASLNSCVNPILYFLAGDTFRRR 4xo8 A 1.698 BS01 KGM A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 ? 0007155,0009289 Kd=1.1nM remove_due_to_license_issue P08191 26948702 501 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4xoc A 1.42 BS01 KGM A 1 F1 I13 N46 Y48 D54 Q133 N135 D140 F1 I13 N46 Y48 D54 Q133 N135 D140 0007155,0009289 Kd=3nM remove_due_to_license_issue 26948702 501 FACKTANGTAIPIGGGSANVYVNLAPAVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSSFSGTVKYNGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 4xoe A 2.4 BS02 KGM A 1 F1 N46 Y48 T51 D54 Q133 N135 Y137 D140 F1 N46 Y48 T51 D54 Q133 N135 Y137 D140 0007155,0009289 Kd=9.9uM remove_due_to_license_issue 26948702 301 FACKTANGTAIPIGGGSANVYVNLAPAVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSSFSGTVKYNGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPTGGCDVSARDVTVTLPDYPGSVPIPLTVYCAKSQNLGYYLSGTTADAGNSIFTNTASFSPAQGVGVQLTRNGTIIPANNTVSLGAVGTSAVSLGLTANYARTGGQVTAGNVQSIIGVTFVYQ 4xpj A 2.605 BS01 LPY B 1 K88 W99 K79 W90 ? 0005102 remove_due_to_license_issue P01139 26144237 201 GEFSVCDSVSVWVGDKTTATDIKGKEVTVLAEVNINNSVFRQYFFETKCRASNPVESGCRGIDSKHWNSYCTTTHTFVKALTTDEKQAAWRFIRIDTACVCVLSR 4xpj B 2.605 BS01 LPY B 1 F49 R50 Y52 W99 F39 R40 Y42 W89 ? 0005102 remove_due_to_license_issue P01139 26144237 201 EFSVCDSVSVWVGDKTTATDIKGKEVTVLAEVNINNSVFRQYFFETKCRASNPVESGCRGIDSKHWNSYCTTTHTFVKALTTDEKQAAWRFIRIDTACVCVLSRK 4xqa A 1.4072 BS02 423 B 1 Y308 Y312 P317 D318 K345 Y127 Y131 P136 D137 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4xqa B 1.4072 BS01 423 B 1 Y308 Y312 P317 D318 P320 S344 K345 Y127 Y131 P136 D137 P139 S163 K164 ? 0007155,0019028,0019058,0019062 Kd=10.3uM remove_due_to_license_issue Q64823 26177934 401 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4xqa C 1.4072 BS01 423 B 1 Y308 Y312 P317 D318 S344 K345 Y126 Y130 P135 D136 S162 K163 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 TRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4xqb A 1.597 BS01 425 A 1 Y308 Y312 P317 S344 K345 Y127 Y131 P136 S163 K164 ? 0007155,0019028,0019058,0019062 Kd=163.4uM remove_due_to_license_issue Q64823 26177934 401 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4xqb B 1.597 BS01 425 A 1 Y312 P317 S344 K345 Y132 P137 S164 K165 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 YDTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4xqb C 1.597 BS01 425 A 1 Y312 P317 S344 K345 Y131 P136 S163 K164 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue Q64823 26177934 401 DTRTLWTTPDTSPNCTIAQDKDSKLTLVLTKCGSQILANVSLIVVAGKYHIINNKTNPKIKSFTIKLLFNKNGVLLDNSNLGKAYWNFRSGNSNVSTAYEKAIGFMPNLVAYPKPSNSKKYARDIVYGTIYLGGKPDQPAVIKTTFNQETGCEYSITFNFSWSKTYENVEFETTSFTFSYIAQE 4xqu A 3.25 BS01 GAL G 1 R137 Q226 R128 Q219 ? 0019031,0019064,0046789 remove_due_to_license_issue A0A059T4A1 25766296 2 DKICLGHHAVANGTIVKTLTNEQEEVTNATETVESTGINRLCMKGRKHKDLGNCHPIGMLIGTPACDLHLTGMWDTLIERENAIAYCYPGATVNVEALRQKIMESGGINKISTGFTYGSSINSAGTTRACMRNGGNSFYAELKWLVSKSKGQNFPQTTNTYRNTDTAEHLIMWGIHHPSSTQEKNDLYGTQSLSISVGSSTYRNNFVPVVGARPQVNGQSGRIDFHWTLVQPGDNITFSHNGGLIAPSRVSKLIGRGLGIQSDAPIDNNCESKCFWRGGSINTRLPFQNLSPRTVGQCPKYVNRRSLMLATGMRNVPE 4xqu A 3.25 BS02 SIA G 1 Y98 T135 T136 R137 W153 H183 E190 Q226 Y88 T126 T127 R128 W144 H176 E183 Q219 ? 0019031,0019064,0046789 remove_due_to_license_issue A0A059T4A1 25766296 3 DKICLGHHAVANGTIVKTLTNEQEEVTNATETVESTGINRLCMKGRKHKDLGNCHPIGMLIGTPACDLHLTGMWDTLIERENAIAYCYPGATVNVEALRQKIMESGGINKISTGFTYGSSINSAGTTRACMRNGGNSFYAELKWLVSKSKGQNFPQTTNTYRNTDTAEHLIMWGIHHPSSTQEKNDLYGTQSLSISVGSSTYRNNFVPVVGARPQVNGQSGRIDFHWTLVQPGDNITFSHNGGLIAPSRVSKLIGRGLGIQSDAPIDNNCESKCFWRGGSINTRLPFQNLSPRTVGQCPKYVNRRSLMLATGMRNVPE 4xrq A 1.95 BS01 1B0 A 1 N53 L56 N57 Q63 M66 K70 T107 Y130 N53 L56 N57 Q63 M66 K70 T107 Y130 ? 0016032 Kd=0.232uM remove_due_to_license_issue P12493 26109731 301 PIVQNLQGQMVHQCISPRTLNAWVKVVEEKAFSPEVIPMFAALSCGATPQDLNTMLNTVGGHQAAMHMLKETINEEAAEWDRLHPVHAGPIAPGQMREPRGSDIAGTTSTLQEQIGWMTHNPPIPVGEIYKRWIILGLNKIVRMYSPTSILDIRQGPKEPFRDYIDRFYKTIRAEQASQEATETLLVQNANPDCKTILKALGPGATLEEMMTACQ 4xs2 A 2.73 BS01 42P A 1 V200 A211 K213 Y262 Y264 M265 G268 S269 A315 L318 D329 V36 A47 K49 Y93 Y95 M96 G99 S100 A146 L149 D160 D311 K313 A315 N316 D329 T351 D142 K144 A146 N147 D160 T178 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue Q9NWZ3 25870132 501 TRFHSFSFYELKNVTNNFDERPISVNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4xsx C 3.708 BS01 42S C 1 P552 S642 P550 S640 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue A7ZUK1 26195788 1401 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4xsx D 3.708 BS01 42S C 1 P750 I755 L770 F773 P743 I748 L763 F766 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0008270,0016779,0034062,0042793,0046872 remove_due_to_license_issue A7ZUK2 26195788 1401 LKAQTKTEEFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRRAAG 4xsy C 4.007 BS01 42T C 1 H551 P552 S642 H549 P550 S640 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue A7ZUK1 26195788 1401 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4xsy D 4.007 BS01 42T C 1 K749 P750 I755 F773 K742 P743 I748 F766 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0008270,0016779,0034062,0042793,0046872 remove_due_to_license_issue A7ZUK2 26195788 1401 LKAQTKTEEFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRRAAG 4xsz C 3.683 BS01 42U C 1 D444 P552 Y555 E641 S642 D442 P550 Y553 E639 S640 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0016779,0032549,0034062,0042793 remove_due_to_license_issue A7ZUK1 26195788 1401 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4xsz D 3.683 BS01 42U C 1 K749 P750 I755 I774 K742 P743 I748 I767 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0006351,0006360,0006366,0006383,0008270,0016779,0034062,0042793,0046872 remove_due_to_license_issue A7ZUK2 26195788 1401 LKAQTKTEEFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRRAAG 4xt2 A 1.698 BS01 43L A 1 H248 M252 Y281 M289 S292 H293 L296 V302 S304 Y307 M309 G323 H15 M19 Y48 M56 S59 H60 L63 V69 S71 Y74 M76 G90 ? Kd=63nM remove_due_to_license_issue Kd=63nM, IC50=112nM Q99814 26226049 401 GEFKGLDSKTFLSEHSMDMKFTYCDDRITELIGYHPEELLGRSAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGGYVWLETQGTVIYNPRNLQPQCIMCVNYVLSEIEK 4xt9 A 2.25 BS02 43V A 1 Q286 L287 C320 L324 R364 M365 R367 A368 V376 F377 F388 I400 F401 Q22 L23 C56 L60 R100 M101 R103 A104 V112 F113 F124 I136 F137 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=158nM, EC50=3162nM P51449 26277758 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 4xta A 2.5 BS01 DIF A 1 R288 S289 A292 M329 L330 I341 R67 S68 A71 M108 L109 I120 ? 0003677,0004879,0005634,0006355 ic50=3.7uM remove_due_to_license_issue P37231 26445566 501 SADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDLHPLLQEIY 4xtt A 2.708 BS01 2BA A 1 I163 D167 R169 A170 I176 P191 I31 D35 R37 A38 I44 P59 ? 0006813,0008324,0098655 remove_due_to_license_issue A0A0M3KL06 25957408 301 ASASVLDYLELADEHSIVELKATEKMAGQSIIDLDIRAQYGINIIAIKRGKEFIISPNPNINLEIGDILIMIGHDNDLNRFEKNI 4xtt B 2.708 BS01 2BA A 1 I163 I164 D167 R169 I176 P191 I31 I32 D35 R37 I44 P59 ? 0006813,0008324,0098655 remove_due_to_license_issue A0A0M3KL06 25957408 301 ASASVLDYLELADEHSIVELKATEKMAGQSIIDLDIRAQYGINIIAIKRGKEFIISPNPNINLEIGDILIMIGHDNDLNRFEKNI 4xtv A 1.45001 BS01 44K A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 I83 N130 K138 I142 V155 G156 N158 V166 D167 A170 S37 T38 N39 Q62 G65 R66 G67 R68 R71 G72 W73 A74 I82 N129 K137 I141 V154 G155 N157 V165 D166 A169 R69 K138 R68 K137 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.54nM remove_due_to_license_issue I6YFP0 26299766 301 TDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHL 4xtw A 2.30014 BS01 44M A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 W74 A75 I83 N130 K138 G141 I142 V155 G156 N158 V166 D167 A170 S38 T39 N40 Q63 G66 R67 G68 R69 R72 W74 A75 I83 N130 K138 G141 I142 V155 G156 N158 V166 D167 A170 R69 K138 R266 R69 K138 R266 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.933nM remove_due_to_license_issue I6YFP0 26299766 301 VTDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 4xtx A 2.3001 BS01 590 A 1 S38 T39 Q63 G66 R67 G68 R69 R72 G73 W74 A75 K138 G141 I142 V155 G156 N158 V166 D167 A170 S38 T39 Q63 G66 R67 G68 R69 R72 G73 W74 A75 K138 G141 I142 V155 G156 N158 V166 D167 A170 R69 K138 R266 R69 K138 R266 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.027nM remove_due_to_license_issue I6YFP0 26299766 301 VTDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 4xty A 1.80003 BS01 44L A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 I83 N130 K138 G141 I142 V155 G156 N158 V166 D167 A170 S37 T38 N39 Q62 G65 R66 G67 R68 R71 G72 W73 A74 I82 N129 K137 G140 I141 V154 G155 N157 V165 D166 A169 R69 K138 R68 K137 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.614nM remove_due_to_license_issue I6YFP0 26299766 301 TDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHL 4xtz A 1.90001 BS01 594 A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 I83 K138 G141 I142 V155 G156 N158 V166 D167 A170 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 I83 K138 G141 I142 V155 G156 N158 V166 D167 A170 R69 K138 R266 R69 K138 R266 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.153nM remove_due_to_license_issue I6YFP0 26299766 301 VTDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 4xu0 A 1.6 BS01 44N A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 I83 K138 G141 I142 V155 G156 N158 V166 D167 S37 T38 N39 Q62 G65 R66 G67 R68 R71 G72 W73 A74 I82 K137 G140 I141 V154 G155 N157 V165 D166 R69 K138 R266 R68 K137 R265 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.769nM remove_due_to_license_issue I6YFP0 26299766 301 TDRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 4xu1 A 1.70001 BS01 44O A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 W74 A75 I83 K138 G141 I142 V155 G156 N158 V166 D167 A170 S36 T37 N38 Q61 G64 R65 G66 R67 R70 W72 A73 I81 K136 G139 I140 V153 G154 N156 V164 D165 A168 R69 K138 R67 K136 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.324nM remove_due_to_license_issue I6YFP0 26299766 301 DRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIAVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHL 4xu2 A 1.85003 BS01 44Q A 1 S38 T39 N40 Q63 G66 R67 G68 R69 R72 G73 W74 A75 K138 I142 V155 G156 N158 V166 D167 S36 T37 N38 Q61 G64 R65 G66 R67 R70 G71 W72 A73 K134 I138 V151 G152 N154 V162 D163 R69 K138 R266 R67 K134 R262 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.592nM remove_due_to_license_issue I6YFP0 26299766 300 DRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 4xu3 A 2.24268 BS01 44R A 1 S38 T39 N40 Q63 G66 R67 R69 R72 G73 W74 A75 K138 I142 V155 G156 N158 V166 D167 A170 S36 T37 N38 Q61 G64 R65 R67 R70 G71 W72 A73 K135 I139 V152 G153 N155 V163 D164 A167 R69 K138 R266 R67 K135 R263 6.3.4.15 0004077,0005524,0005737,0008284,0009374,0016874,0032991,0036211,0042803 Kd=0.315nM remove_due_to_license_issue I6YFP0 26299766 301 DRDRLRPPLDERSLRDQLIGAGSGWRQLDVVAQTGSTNADLLARAASGADIDGVVLIAEHQTAGRGRHGRGWAATARAQIILSVGVRVVDVPVQAWGWLSLAAGLAVLDSVAPLIVPPAETGLKWPNDVLARGGKLAGILAEVAQPFVVLGVGLNVTQAPEEVDPDATSLLDLGVAAPDRNRIASRLLRELEARIIQWRNANPQLAADYRARSLTIGSRVRVELPGGQDVVGIARDIDDQGRLCLDVGGRTVVVSAGDVVHLR 4xua A 1.75 BS01 43C A 1 W1887 P1888 L1890 L1891 V1893 N1894 V1898 I1950 W32 P33 L35 L36 V38 N39 V43 I95 ? ic50=26uM remove_due_to_license_issue Q9UIF8 25719566 2005 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 4xub A 1.98 BS01 43D A 1 W1887 P1888 F1889 L1891 V1893 N1894 L1897 I1950 W32 P33 F34 L36 V38 N39 L42 I95 ? ic50=1.07uM remove_due_to_license_issue Q9UIF8 25719566 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 4xuc A 1.8 BS01 43G A 1 W88 K194 N220 C223 L248 E249 W41 K147 N173 C176 L201 E202 D191 K194 D219 N220 E249 D144 K147 D172 N173 E202 2.1.1.6 0000287,0006584,0008171,0016206 ic50=1100nM remove_due_to_license_issue IC50=47nM P21964 25815153 301 NLLAGDTKEQRILNHVLQHAEPGNAQSVLEAIDTYCEQKEWAMNVGDKKGKIVDAVIQEHQPSVLLELGAYCGYSAVRMARLLSPGARLITIEINPDCAAITQRMVDFAGVKDKVTLVVGASQDIIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVICPGAPDFLAHVRGSSCFECTHYQSFLEYREVVDGLEKAIYKGP 4xue B 2.3 BS01 43J B 1 M90 D191 W193 K194 N220 E249 M40 D141 W143 K144 N170 E199 D191 K194 D219 N220 E249 D141 K144 D169 N170 E199 2.1.1.6 0000287,0006584,0008171,0016206 ic50>5000nM remove_due_to_license_issue IC50=170nM P21964 25815153 301 AGDTKEQRILNHVLQHAEPGNAQSVLEAIDTYCEQKEWAMNVGDKKGKIVDAVIQEHQPSVLLELGAYCGYSAVRMARLLSPGARLITIEINPDCAAITQRMVDFAGVKDKVTLVVGASQDIIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVICPGAPDFLAHVRGSSCFECTHYQSFLEYREVVDGLEKAIYKGP 4xue B 2.3 BS04 43J A 1 L64 R151 L14 R101 D191 K194 D219 N220 E249 D141 K144 D169 N170 E199 2.1.1.6 0000287,0006584,0008171,0016206 ic50>5000nM remove_due_to_license_issue IC50=170nM P21964 25815153 301 AGDTKEQRILNHVLQHAEPGNAQSVLEAIDTYCEQKEWAMNVGDKKGKIVDAVIQEHQPSVLLELGAYCGYSAVRMARLLSPGARLITIEINPDCAAITQRMVDFAGVKDKVTLVVGASQDIIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVICPGAPDFLAHVRGSSCFECTHYQSFLEYREVVDGLEKAIYKGP 4xuh A 2.22 BS01 SFI A 1 F264 R280 I281 C285 I341 S342 F58 R67 I68 C72 I128 S129 ? 0003677,0004879,0005634,0006355 ic50=1.87uM remove_due_to_license_issue EC50=800nM P37231 26445566 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4xuh A 2.22 BS02 SFI A 2 F282 C285 H323 Y327 F360 F363 M364 H449 L469 Y473 F69 C72 H110 Y114 F147 F150 M151 H236 L256 Y260 ? 0003677,0004879,0005634,0006355 ic50=1.87uM remove_due_to_license_issue EC50=800nM P37231 26445566 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4xum A 2.4 BS01 IMN A 1 F282 C285 S289 H323 F360 F363 H449 Y473 F65 C68 S72 H106 F143 F146 H232 Y256 ? 0003677,0004879,0005634,0006355 ic50=21.3uM remove_due_to_license_issue EC50=50000nM P37231 26445566 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4xum A 2.4 BS02 IMN A 2 E259 R280 I281 C285 I341 S342 M348 E53 R63 I64 C68 I124 S125 M131 ? 0003677,0004879,0005634,0006355 ic50=21.3uM remove_due_to_license_issue EC50=50000nM P37231 26445566 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 4xuz A 1.5 BS01 4D6 A 1 C44 S45 K48 N79 S105 N107 P142 N145 T210 G211 S212 G213 C43 S44 K47 N78 S104 N106 P141 N144 T209 G210 S211 G212 S45 K48 S105 E141 K209 S212 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue S5LVN3 25782055 312 TADVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTDGL 4xv1 A 2.47 BS01 904 A 1 I463 A481 L505 L514 T529 Q530 W531 C532 D594 I15 A30 L53 L62 T77 Q78 W79 C80 D140 D576 K578 N580 N581 D594 S616 D122 K124 N126 N127 D140 S145 2.7.11.1 0004672,0005524,0006468 ic50=0.0042uM remove_due_to_license_issue IC50=16nM P15056 26466569 801 DWEIPDGQITVGQRIGSGTVYKGKWHGDVAVKMLNVAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGSGSILWMAPEVIRNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVNCPKRMKRLMAECLKKKRDERPSFPRILAEIEE 4xv2 A 2.5 BS01 P06 A 1 G464 V471 A481 K483 L505 L514 F516 T529 W531 C532 F583 G593 D594 F595 G16 V23 A33 K35 L55 L64 F66 T79 W81 C82 F133 G143 D144 F145 D576 K578 N580 N581 D594 S616 D126 K128 N130 N131 D144 S148 2.7.11.1 0004672,0005524,0006468 ic50=0.00539uM remove_due_to_license_issue IC50=1.000000nM, EC50=529nM P15056 26466569 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 4xv2 B 2.5 BS01 P06 B 1 S465 V471 A481 K483 L505 L514 F516 T529 W531 C532 F583 G593 D594 F595 S18 V24 A34 K36 L58 L67 F69 T82 W84 C85 F134 G144 D145 F146 D576 K578 N580 N581 D594 S616 D127 K129 N131 N132 D145 S149 2.7.11.1 0004672,0005524,0006468 ic50=0.00539uM remove_due_to_license_issue IC50=1.000000nM, EC50=529nM P15056 26466569 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASEFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 4xv3 A 2.8 BS01 P02 A 1 V471 A481 L505 L514 T529 W531 F583 D594 F595 V21 A31 L53 L62 T77 W79 F131 D142 F143 D576 K578 N580 N581 D594 S616 D124 K126 N128 N129 D142 S147 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 26466569 801 DDWEIPDGQITVGQRIGSGTVYKGKWHGDVAVKMLNVPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGSGSILWMAPEVIRNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEEL 4xv9 A 2.0 BS01 1OO A 1 V471 A481 K483 L505 L514 T529 W531 C532 H574 F583 I592 G593 D594 F595 V24 A34 K36 L58 L67 T82 W84 C85 H127 F136 I145 G146 D147 F148 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S155 2.7.11.1 0004672,0005524,0006468 ic50=0.19uM remove_due_to_license_issue P15056 26466569 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLALSGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARELS 4xwk A 3.5 BS01 4C8 A 1 Y303 F310 F331 F724 F728 F755 Y274 F281 F302 F633 F637 F664 7.6.2.1,7.6.2.2 0001666,0001890,0005524,0005737,0005886,0007565,0007595,0007623,0008559,0009410,0009914,0010046,0014070,0015562,0016020,0016324,0016887,0022857,0031526,0031667,0032355,0032496,0032570,0033189,0033280,0033762,0035633,0036146,0042626,0042910,0043215,0045177,0045332,0046581,0046686,0046865,0050892,0055085,0060856,0071217,0071222,0071236,0071312,0071356,0071392,0071475,0071548,0071549,0090554,0090555,0097068,0097305,0097327,0099038,0099040,0140115,0140326,0140328,0140359,1902065,1902396,1903416,1904057,1904148,1904446,1904478,1905231,1905232,1905233,1905235,1905237,1990961,1990962,1990963,2001025 remove_due_to_license_issue P21447 27152359 1301 KPAVSVLTMFRYAGWLDRLYMLVGTLAAIIHGVALPLMMLIFGDMTDSFASVGQVSKQSTQMSEADKRAMFAKLEEEMTTYAYYYTGIGAGVLIVAYIQVSFWCLAAGRQIHKIRQKFFHAIMNQEIGWFDVHDVGELNTRLTDDVSKINEGIGDKIGMFFQAMATFFGGFIIGFTRGWKLTLVILAISPVLGLSAGIWAKILSSFTDKELHAYAKAGAVAEEVLAAIRTVIAFGGQKKELERYNNNLEEAKRLGIKKAITANISMGAAFLLIYASYALAFWYGTSLVISKEYSIGQVLTVFFSVLIGAFSVGQASPNIEAFANARGAAYEVFKIIDNKPSIDSFSKSGHKPDNIQGNLEFKNIHFSYPSRKEVQILKGLNLKVKSGQTVALVGNSGCGKSTTVQLMQRLYDPLDGMVSIDGQDIRTINVRYLREIIGVVSQEPVLFATTIAENIRYGREDVTMDEIEKAVKEANAYDFIMKLPHQFDTLVGERGAQLSGGQKQRIAIARALVRNPKILLLDEATSALDTESEAVVQAALDKAREGRTTIVIAHRLSTVRNADVIAGFDGGVIVEQGNHDELMREKGIYFKLVMTQTPPASFWRILKLNSTEWPYFVVGIFCAIINGGLQPAFSVIFSKVVGVFTNGGPPETQRQNSNLFSLLFLILGIISFITFFLQGFTFGKAGEILTKRLRYMVFKSMLRQDVSWFDDPKNTTGALTTRLANDAAQVKGATGSRLAVIFQNIANLGTGIIISLIYGWQLTLLLLAIVPIIAIAGVVEMKMLSGQALKDKKELEGSGKIATEAIENFRTVVSLTREQKFETMYAQSLQIPYRNAMKKAHVFGITFSFTQAMMYFSYAACFRFGAYLVTQQLMTFENVLLVFSAIVFGAMAVGQVSSFAPDYAKATVSASHIIRIIEKTPEIDSYSTQGLKPNMLEGNVQFSGVVFNYPTRPSIPVLQGLSLEVKKGQTLALVGSSGCGKSTVVQLLERFYDPMAGSVFLDGKEIKQLNVQWLRAQLGIVSQEPILFDCSIAENIAYGDNSRVVSYEEIVRAAKEANIHQFIDSLPDKYNTRVGDKGTQLSGGQKQRIAIARALVRQPHILLLDEATSALDTESEKVVQEALDKAREGRTCIVIAHRLSTIQNADLIVVIQNGKVKEHGTHQQLLAQKGIYFSMVSVQAGA 4xx3 A 2.4 BS01 70X A 1 T84 Q85 Y86 V102 D104 Y149 T151 D292 T293 G294 A295 S296 T17 Q18 Y19 V35 D37 Y82 T84 D225 T226 G227 A228 S229 D104 S107 N109 W111 Y149 D292 A295 D37 S40 N42 W44 Y82 D225 A228 3.4.23.15 0004190,0006508 Ki=56nM remove_due_to_license_issue Ki=56nM P00797 25728416 502 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4xx4 A 2.4 BS01 70Y A 1 D104 Y149 T151 P184 A188 D292 G294 A295 S296 M369 D37 Y82 T84 P117 A121 D225 G227 A228 S229 M302 D104 S107 N109 W111 Y149 D292 A295 D37 S40 N42 W44 Y82 D225 A228 3.4.23.15 0004190,0006508 Ki=44nM remove_due_to_license_issue Ki=44nM P00797 25728416 502 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 4xx9 A 1.4 BS02 RF4 A 1 K76 K115 I118 V127 R131 T148 L155 F157 K6 K45 I48 V57 R61 T78 L85 F87 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T175 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Kd=8000nM, EC50=2000nM O15530 26443011 402 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 4xx9 A 1.4 BS03 RF4 A 2 R172 G278 L279 R102 G208 L209 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T175 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Kd=8000nM, EC50=2000nM O15530 26443011 403 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 4xxs A 1.86 BS01 SI5 A 1 D32 G34 S35 Y71 F108 W115 R128 D228 G230 D37 G39 S40 Y76 F113 W120 R133 D224 G226 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D224 T227 3.4.23.46 0004190,0006508,0016020 ic50=52nM remove_due_to_license_issue IC50=4.0nM P56817 25781223 401 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIP 4xy2 A 2.03 BS02 490 A 1 L635 I692 Y693 F696 P712 M713 V722 G725 Q726 F729 L177 I234 Y235 F238 P254 M255 V264 G267 Q268 F271 3.1.4.17 0004114,0007165,0008081 ic50=8nM remove_due_to_license_issue Q9Y233 25960322 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 4xy8 A 1.7 BS01 43U A 1 F44 F47 V49 I53 N100 Y106 F23 F26 V28 I32 N79 Y85 ? Kd=397nM remove_due_to_license_issue Q9H8M2 25703523 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 4xy9 A 1.83 BS01 43U A 1 W81 P82 F83 Q85 L92 N140 I146 W40 P41 F42 Q44 L51 N99 I105 ? Kd=4651nM remove_due_to_license_issue O60885 25703523 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4xya A 2.05 BS01 43S A 1 W81 P82 V87 L92 N140 I146 W40 P41 V46 L51 N99 I105 ? Kd=1370nM remove_due_to_license_issue O60885 25703523 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4xyc A 3.3 BS01 2K9 A 1 Y125 F228 H274 S276 W278 K357 A358 R360 Y117 F220 H266 S268 W270 K349 A350 R352 D50 E129 E131 E215 E223 H272 R343 E362 R364 D51 E121 E123 E207 E215 H264 R335 E354 R356 6.3.1.2 0003824,0004356,0005524,0005737,0006542,0016020,0016874,0019740,0046872 remove_due_to_license_issue P9WN38 25770781 900 KTPDDVFKLAKDEKVEYVDVRFCDLPGIMQHFTIPASAFDKSVFDDGLAFDGHESDMLLLPDPETARIDPFRAAKTLNINFFVHDPFTLEPYSRDPRNIARKAENYLISTGIADTAYFGAEAEFYIFDSVSFDSRANGSFYEVDAISGWWNTGAATEADGSPNRGYKVRHKGGYFPVAPNDQYVDLRDKMLTNLINSGFILEKGHHEVGSGGQAEINYQFNSLLHAADDMQLYKYIIKNTAWQNGKTVTFMPKPLFGDNGSGMHCHQSLWKDGAPLMYDETGYAGLSDTARHYIGGLLHHAPSLLAFTNPTVNSYKRLVPGYEAPINLVYSQRNRSACVRIPITGSNPKAKRLEFRSPDSSGNPYLAFSAMLMAGLDGIKNKIEPQAPVDKDLYELPPEEAASIPQTPTQLSDVIDRLEADHEYLTEGGVFTNDLIETWISFKRENEIEPVNIRPHPYEFALYYDV 4xyf A 1.85 BS01 44X A 1 I1084 A1108 Y1159 M1160 G1163 D1164 R1208 N1209 M1211 A1221 D1222 Y1230 I33 A52 Y103 M104 G107 D108 R152 N153 M155 A165 D166 Y174 D1204 A1206 R1208 N1209 D1222 A1243 D148 A150 R152 N153 D166 A187 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1.000000nM P08581 25699405 1401 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 4y0a A 1.911 BS01 SKM A 1 M27 D50 F73 R74 G96 G97 L136 R153 M17 D40 F63 R64 G86 G87 L126 R143 2.7.1.71 0000287,0004765,0005524,0005737,0005829,0008652,0009073,0009423,0016301,0019752,0046872 remove_due_to_license_issue A0A0M3KL09 26249354 201 PSKAFETLPNIYLVGPMGAGKTTVGRHLAELLGREFLDSDHEIERKTGATIPWIFEKEGEVGFRTRETVVLNELTSRKALVLATGGGAITQAPNREFLKQRGIVVYLYTPVELQLQRTYRDKNRPLLQVENPEQKLRDLLKIRDPLYREVAHYTIETNQGAARDLAQKILQLILSNKLK 4y16 A 2.6 BS02 48G A 1 S28 W63 M69 F70 Y73 S76 D80 W133 D153 G155 T156 T159 L163 F171 S23 W58 M64 F65 Y68 S71 D75 W128 D148 G150 T151 T154 L158 F166 ? remove_due_to_license_issue P11609 26018083 301 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 4y16 C 2.6 BS01 48G A 1 P28 N30 R94 G95 P28 N30 R94 G95 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,P01848 26018083 301 TQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKDFACANAFNNSIIPEDTFFPS 4y24 A 2.32 BS01 TD2 A 1 V31 H44 R48 D54 N61 W68 E71 R73 G124 V30 H43 R47 D53 N60 W67 E70 R72 G123 ? 0002317,0003723,0005515,0005576,0005615,0005737,0005788,0005829,0005886,0006915,0007165,0030246,0030395,0031295,0042981,0043065,0043123,0043236,0045445,0046598,0048018,0050729,0062023,0070062,0098609,1990724,2000329,2001200 Kd=0.22uM remove_due_to_license_issue P09382 27416897 201 CGLVASNLNLKPGECLRVRGEVAPDAKSFVLNLGKDSNNLCLHFNPRFNAHGDANTIVCNSKDGGAWGTEQREAVFPFQPGSVAEVCITFDQANLTVKLPDGYEFKFPNRLNLEAINYMAADGDFKIKCVAFD 4y29 A 1.98 BS02 CTI A 1 I281 C285 R288 L330 L353 M364 I62 C66 R69 L111 L134 M145 ? 0003677,0004879,0005634,0006355 ic50=566nM remove_due_to_license_issue IC50=566nM P37231 26183621 501 SADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 4y2b A 2.2 BS02 EPK A 1 Y211 N365 L401 I412 Q413 F416 Y73 N227 L263 I274 Q275 F278 S169 A250 H301 L302 E371 W376 S377 S31 A112 H163 L164 E233 W238 S239 3.1.4.53 0004114,0007165,0008081 ic50=4.4nM remove_due_to_license_issue IC50=4.4nM Q13946 25866242 503 DYNGQAKCMLEKVGNWNFDIFLFDRLTNGNSLVSLTFHLFSLHGLIEYFHLDMMKLRRFLVMIQEDYHSQNPYHNAVHAADVTQAMHCYLKEPKLANSVTPWDILLSLIAAATHDLDHPGVNQPFLIKTNHYLATLYKNTSVLENHHWRSAVGLLRESGLFSHLPLESRQQMETQIGALILATDISRQNEYLSLFRSHLDRGDLCLEDTRHRHLVLQMALKCADICNPCRTWELSKQWSEKVTEEFFHQGDIEKKYHLGVSPLCDRHTESIANIQIGFMTYLVEPLFTEWARFSNTRLSQTMLGHVGLNKASWKGLQR 4y2j A 2.15 BS02 49G A 1 D335 W336 Y383 L408 Y466 W525 D334 W335 Y382 L407 Y465 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=800uM remove_due_to_license_issue IC50=800000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2p A 2.05 BS02 3C5 A 1 F267 D335 Y383 Y466 H524 W525 F266 D334 Y382 Y465 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=2200uM remove_due_to_license_issue IC50=2200000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2q A 2.4 BS02 49N A 1 F267 D335 Y383 L408 M419 Y466 H524 W525 F266 D334 Y382 L407 M418 Y465 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=1200uM remove_due_to_license_issue IC50=1200000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2s A 2.3 BS02 49P A 1 F267 Y383 F497 V498 H524 F266 Y382 F496 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=52uM remove_due_to_license_issue IC50=52000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2t A 2.4 BS02 49Q A 1 D335 W336 S374 I375 Y383 Y466 D334 W335 S373 I374 Y382 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=150uM remove_due_to_license_issue IC50=79000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2u A 2.75 BS01 49R A 1 F267 D335 W336 Y383 L408 Y466 F266 D334 W335 Y382 L407 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=580000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2v A 2.4 BS02 4A5 A 1 D335 Y383 V498 H524 D334 Y382 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=91uM remove_due_to_license_issue IC50=91000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2x A 2.5 BS02 4A0 A 1 D335 W336 Y383 Q384 Y466 D334 W335 Y382 Q383 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.51uM remove_due_to_license_issue IC50=510nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y2y A 2.3 BS01 49Z A 1 F267 D335 W336 M339 Y383 L408 Y466 L499 H524 W525 F266 D334 W335 M338 Y382 L407 Y465 L498 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=9uM remove_due_to_license_issue IC50=9000nM P34913 25862210 602 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 4y38 A 1.1 BS01 0A9 A 1 D35 Y79 D219 G221 T222 D35 Y79 D219 G221 T222 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Kd=4mM remove_due_to_license_issue P11838 27139825 411 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4y3j A 1.31 BS01 HIC A 1 Y79 D81 F116 G221 T222 T223 Y79 D81 F116 G221 T222 T223 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Kd=6.8mM remove_due_to_license_issue P11838 27139825 415 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4y3y A 1.346 BS01 DCL A 1 D35 G37 Y79 G80 F194 D219 D35 G37 Y79 G80 F194 D219 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Kd=4.5mM remove_due_to_license_issue P11838 27139825 412 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4y46 A 2.04 BS01 4F2 A 1 I70 A91 M146 M149 A151 Q155 L206 I26 A47 M102 M105 A107 Q111 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T180 2.7.11.24 0004672,0004707,0005524,0006468 ic50=11nM remove_due_to_license_issue IC50=11nM P53779 25893042 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDQLDEREHTIEEWKELIYKEVMN 4y4g A 1.439 BS01 GGB A 1 D35 Y79 D81 S83 D219 G221 D35 Y79 D81 S83 D219 G221 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 remove_due_to_license_issue P11838 27139825 411 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4y4j A 1.03 BS01 LNR A 1 D35 Y79 D81 S83 F116 G221 D35 Y79 D81 S83 F116 G221 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Kd=3.4mM remove_due_to_license_issue P11838 27139825 412 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4y4v A 2.04 BS01 DAL A 1 K107 E110 G111 G154 H155 K93 E96 G97 G140 H141 ? 0008360,0009252,0016740,0071555 Kd=224uM remove_due_to_license_issue O25255 26306031 401 LNASDRLLEIMRLYQKQGLEMVGQKLDSYLADKSFWAEELQNKDTDFGYYQNKQFLFVANKSKPSLEFYEIENNMLKKINSSKALVGSKKGDKTLEGDLATPIGVYRITQKLERLDQYYGVLAFVTNYPNLYDTLKKRTGHGIWVHGMPLNGDRNELNTKGCIAIENPLLSSYDKVLKGEKAFLITYEDKFFPSTKEELSMILSSLFQWKEAWARGDFERYMRFYNPNFTRYDGMKFNAFKEYKKRVFAKNEKKNIAFSSINVIPYPNSQNKRLFYVVFDQDYKAYQHNKLSYSSNSQKELYIEIENNQVSIIMEK 4y4v A 2.04 BS02 DAL A 2 Y133 G156 W158 C176 Y119 G142 W144 C162 ? 0008360,0009252,0016740,0071555 Kd=224uM remove_due_to_license_issue O25255 26306031 402 LNASDRLLEIMRLYQKQGLEMVGQKLDSYLADKSFWAEELQNKDTDFGYYQNKQFLFVANKSKPSLEFYEIENNMLKKINSSKALVGSKKGDKTLEGDLATPIGVYRITQKLERLDQYYGVLAFVTNYPNLYDTLKKRTGHGIWVHGMPLNGDRNELNTKGCIAIENPLLSSYDKVLKGEKAFLITYEDKFFPSTKEELSMILSSLFQWKEAWARGDFERYMRFYNPNFTRYDGMKFNAFKEYKKRVFAKNEKKNIAFSSINVIPYPNSQNKRLFYVVFDQDYKAYQHNKLSYSSNSQKELYIEIENNQVSIIMEK 4y59 A 1.22 BS01 T21 A 1 S27 Y43 S45 V47 N49 A50 W79 A86 S88 W92 W108 D128 S13 Y29 S31 V33 N35 A36 W65 A72 S74 W78 W94 D114 ? 0009374 Kd=5.8uM remove_due_to_license_issue P22629 26261872 200 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKP 4y59 D 1.22 BS01 T21 D 1 S27 Y43 W79 A86 W92 W108 D128 S13 Y29 W65 A72 W78 W94 D114 ? 0009374 Kd=5.8uM remove_due_to_license_issue P22629 26261872 200 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKP 4y5d A 1.2 BS01 MT6 A 1 S27 Y43 S45 V47 N49 W79 A86 S88 W108 L110 D128 S13 Y29 S31 V33 N35 W65 A72 S74 W94 L96 D114 ? 0009374 Kd=1.2uM remove_due_to_license_issue P22629 26261872 200 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKPS 4y5d B 1.2 BS01 MT6 B 1 Y43 W79 A86 S88 W92 W108 D128 Y29 W65 A72 S74 W78 W94 D114 ? 0009374 Kd=1.2uM remove_due_to_license_issue P22629 26261872 200 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKPS 4y5d D 1.2 BS01 MT6 D 1 S27 Y43 S45 W79 A86 S88 W92 W108 D128 S13 Y29 S31 W65 A72 S74 W78 W94 D114 ? 0009374 Kd=1.2uM remove_due_to_license_issue P22629 26261872 200 AGITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKPS 4y5h A 2.055 BS01 519 A 1 I70 A91 M146 M149 Q155 L206 I26 A47 M102 M105 Q111 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T180 2.7.11.24 0004672,0004707,0005524,0006468 ic50=15nM remove_due_to_license_issue IC50=15nM P53779 25893042 501 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTASFMMTPYVVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQLDEREHTIEEWKELIYKEVMN 4y5s A 2.543 BS01 AKG A 1 Q130 H133 H209 G211 R222 L226 Q123 H126 H202 G204 R215 L219 1.14.11.38 0005575,0051213,1902181 remove_due_to_license_issue Q4WAW9 26524521 401 DSKPQLQRLAADADVDRMCRLLEEDGAFILKGLLPFDVVESFNRELDVQMAIPPPKGERLLADKYPPHFKYVPNVATTCPTFRNTVLINPVIHAICEAYFQRTGDYWLSAAFLREIESGMPAQPFHRDDATHPLMHYQPLEAPPVSLSVIFPLTEFTEENGATEVILGSHRWTEVGTPERDQAVLATMDPGDVLIVRQRVVHAGGGNRTTAGKPRRVVLAYFNSVQLTPFETYRTMPREMVESMTVLGQRMLGWRTMKPSDPNIVGINLIDDKRLENVLQLKAADSPAL 4y5w A 3.104 BS01 dna M 0 K288 K374 H415 K132 K204 H242 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGETRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCERKGTESVTEEKCAVLFSASFTLGLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 4y5w A 3.104 BS02 dna N 0 R370 S378 V379 V414 R200 S208 V209 V241 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGETRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCERKGTESVTEEKCAVLFSASFTLGLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 4y5w B 3.104 BS01 dna E 0 K374 H415 K203 H241 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGAPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCERKGTESVTEEKCAVLFSASFTLGPPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 4y5w B 3.104 BS02 dna F 0 R370 V379 V414 R199 V208 V240 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGAPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCERKGTESVTEEKCAVLFSASFTLGPPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 4y5w C 3.104 BS01 dna M 0 R370 V379 V414 R200 V203 V234 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGAPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCSVTEEKCAVLFSASFTLGPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGGRGYVPATIKMTVE 4y5w C 3.104 BS02 dna N 0 K288 H415 K131 H235 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGAPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCSVTEEKCAVLFSASFTLGPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGGRGYVPATIKMTVE 4y5w D 3.104 BS01 dna E 0 R370 V379 R203 V210 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGAPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCEGTESVTEEKCAVLFSASFTLGPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGGRGYVPATIKMTVE 4y5w D 3.104 BS02 dna F 0 K288 H415 K134 H242 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 22 KFKTGLRRLQHRVGEIHLLREALQKEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLGAPAKPPLVRADMVTEKQARETGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCEGTESVTEEKCAVLFSASFTLGPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGGRGYVPATIKMTVE 4y60 C 1.75 BS01 dna A 0 R5 N8 F10 A31 S34 K35 W41 K42 Y72 R73 R6 N9 F11 A32 S35 K36 W42 K43 Y73 R74 ? remove_due_to_license_issue P43680 26939885 0 ~ 16 GLRIRRPMNAFMVWAKDERKRLAQQNPDLHNAVLSKMLGKAWKELNTAEKRPFVEEAERLRVQHLRDHPNYKYRPR 4y60 C 1.75 BS02 dna B 0 R2 R4 R5 M7 M11 K15 R18 N30 Y72 R75 R3 R5 R6 M8 M12 K16 R19 N31 Y73 R76 ? remove_due_to_license_issue P43680 26939885 0 ~ 16 GLRIRRPMNAFMVWAKDERKRLAQQNPDLHNAVLSKMLGKAWKELNTAEKRPFVEEAERLRVQHLRDHPNYKYRPR 4y62 A 1.6 BS02 48E A 1 F121 I123 Y126 W181 S185 D211 V212 D213 H301 F57 I59 Y62 W113 S117 D143 V144 D145 H233 H233 G266 W300 E303 A343 H165 G198 W232 E235 A275 2.4.1.37,2.4.1.40 0000139,0000166,0003823,0004380,0004381,0005576,0005794,0005975,0006486,0016020,0016757,0016758,0030145,0030259,0031982,0032580,0046872 remove_due_to_license_issue P16442 402 SLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVP 4y63 A 1.3 BS02 48O A 1 F121 I123 Y126 W181 V184 R188 D211 V212 D213 F58 I60 Y63 W118 V121 R125 D148 V149 D150 H233 G266 W300 E303 A343 H170 G203 W237 E240 A280 2.4.1.37,2.4.1.40 0000139,0000166,0003823,0004380,0004381,0005576,0005794,0005975,0006486,0016020,0016757,0016758,0030145,0030259,0031982,0032580,0046872 remove_due_to_license_issue P16442 402 VSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAVP 4y64 A 1.6 BS02 48C A 1 F121 I123 Y126 V184 D211 V212 D213 F58 I60 Y63 V121 D148 V149 D150 H233 G266 W300 E303 A343 H170 G203 W237 E240 A280 2.4.1.37,2.4.1.40 0000139,0000166,0003823,0004380,0004381,0005576,0005794,0005975,0006486,0016020,0016757,0016758,0030145,0030259,0031982,0032580,0046872 remove_due_to_license_issue P16442 402 VSLPRMVYPQPKVLTPCRKDVLVVTPWLAPIVWEGTFNIDILNEQFRLQNTTIGLTVFAIKKYVAFLKLFLETAEKHFMVGHRVHYYVFTDQPAAVPRVTLGTGRQLSVLEVRAYKRWQDVSMRRMEMISDFCERRFLSEVDYLVCVDVDMEFRDHVGVEILTPLFGTLHPGFYGSSREAFTYERRPQSQAYIPKDEGDFYYGGAFFGGSVQEVQRLTRACHQAMMVDQANGIEAVWHDESHLNKYLLRHKPTKVLSPEYLWDQQLLGWPAVLRKLRFTAV 4y67 A 1.6 BS01 RC5 A 1 S232 E233 S269 S270 W296 S306 N311 K312 H341 P358 D359 S156 E157 S193 S194 W220 S230 N235 K236 H265 P282 D283 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.117uM remove_due_to_license_issue Q8IKG4 25781377 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 4y6m A 2.27 BS01 48Q A 1 I32 D34 G36 V78 T114 I123 Y192 D214 G216 T217 S218 I300 I32 D34 G36 V78 T114 I123 Y192 D214 G216 T217 S218 I300 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue P46925 26625296 501 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 4y6p A 1.9 BS01 R77 A 1 S232 E233 S269 S270 W296 M298 S306 N311 K312 P358 D359 S156 E157 S193 S194 W220 M222 S230 N235 K236 P282 D283 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.069uM remove_due_to_license_issue Q8IKG4 25781377 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 4y6r A 1.9 BS01 RF7 A 1 S232 E233 S269 S270 W296 T303 S306 N311 K312 S156 E157 S193 S194 W220 T227 S230 N235 K236 1.1.1.267 0008299,0030604,0046872,0070402 ic50=3.3uM remove_due_to_license_issue Q8IKG4 25781377 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 4y6s A 2.1 BS02 48S A 1 S232 E233 S269 S270 W296 M298 T303 S306 N311 K312 S156 E157 S193 S194 W220 M222 T227 S230 N235 K236 1.1.1.267 0008299,0030604,0046872,0070402 ic50=9.3uM remove_due_to_license_issue Q8IKG4 25781377 502 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 4y73 A 2.14 BS01 XPY A 1 M192 E194 V200 A211 Y262 M265 G268 A315 L318 D329 M30 E32 V38 A49 Y100 M103 G106 A153 L156 D167 D311 K313 A315 N316 D329 T351 D149 K151 A153 N154 D167 T184 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=0.3nM remove_due_to_license_issue IC50=0.300000nM Q9NWZ3 26101574 1000 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4y79 A 2.1 BS03 4O6 A 1 E97 T98 F174 A190 Q192 W215 G216 G219 G226 I227 Y228 E83 T84 F162 A180 Q182 W205 G206 G208 G216 I217 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 Ki=11nM remove_due_to_license_issue Ki=11nM P00742 17338508 303 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4y83 A 2.89 BS01 49B A 1 W132 I144 R146 V152 A165 K167 M207 G210 G213 S214 E217 V260 D270 W49 I61 R63 V69 A82 K84 M124 G127 G130 S131 E134 V177 D187 D253 K255 N258 D270 T290 D170 K172 N175 D187 T207 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue P41279 25918157 401 LSSVRYGTVEDLLAFANHRPQESGILLNMVITPQNGRYQIDSDVLLIPWKLTYRNIGSDFIPRGAFGKVYLAQDIKTKKRMACKLIPVDQFKPSDVEIQACFRHENIAELYGAVLWGETVHLFMEAGEGGSVLEKLESCGPMREFEIIWVTKHVLKGLDFLHSKKVIHHDIKPSNIVFMSTKAVLVDFGLSVQMTEDVYFPKDLRGTEIYMSPEVILCRGHSTKADIYSLGATLIHMQTGTPPWVKRYYLYIIHKQAPPLEDIADDCSPGMRELIEASLERNPNHRPRAADLLKHEALN 4y85 A 2.33 BS01 499 A 1 W132 F143 P145 V152 A165 K167 E208 G210 G213 S214 E217 V260 V269 D270 W52 F60 P62 V69 A82 K84 E125 G127 G130 S131 E134 V177 V186 D187 D253 K255 N258 D270 T290 D170 K172 N175 D187 T207 2.7.11.25 0004672,0005524,0006468 ic50=13nM remove_due_to_license_issue P41279 25918157 401 LSSVRYGTVEDLLAFANHISNTPQESGILLNMVITPQNGRYQIDSDVLLIPWKLTYRNIFIPRGAFGKVYLAQDIKTKKRMACKLIPVDQFKPSDVEIQACFRHENIAELYGAVLWGETVHLFMEAGEGGSVLEKLESCGPMREFEIIWVTKHVLKGLDFLHSKKVIHHDIKPSNIVFMSTKAVLVDFGLSVQMTEDVYFPKDLRGTEIYMSPEVILCRGHSTKADIYSLGATLIHMQTGTPPWVKRYPRSAYPSYLYIIHKQAPPLEDIADDCSPGMRELIEASLERNPNHRPRAADLLKHEALNP 4y87 A 3.1 BS01 49E A 1 L420 Y424 A452 Q453 F456 L236 Y240 A268 Q269 F272 3.1.4.35 0004114,0004115,0004117,0005515,0005654,0005737,0005783,0005794,0005829,0005886,0007165,0008081,0010613,0016787,0019933,0032587,0042383,0042995,0043204,0046068,0046069,0046872,0047555,0048101,0048471,1900273,2000178 remove_due_to_license_issue O76083 26316540 601 KYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQKK 4y8c A 2.7 BS01 49D A 1 M365 L420 L421 Y424 M442 A452 Q453 F456 M181 L236 L237 Y240 M258 A268 Q269 F272 3.1.4.35 0004114,0004115,0004117,0005515,0005654,0005737,0005783,0005794,0005829,0005886,0007165,0008081,0010613,0016787,0019933,0032587,0042383,0042995,0043204,0046068,0046069,0046872,0047555,0048101,0048471,1900273,2000178 remove_due_to_license_issue IC50=6.00nM O76083 26316540 601 KYLLSPETIEALRKPTFDVWLWEPNEMLSCLEHMYHDLGLVRDFSINPVTLRRWLFCVHDNYRNNPFHNFRHCFCVAQMMYSMVWLCSLQEKFSQTDILILMTAAICHDLDHPGYNNTYQINARTELAVRYNDISPLENHHCAVAFQILAEPECNIFSNIPPDGFKQIRQGMITLILATDMARHAEIMDSFKEKMENFDYSNEEHMTLLKMILIKCCDISNEVRPMEVAEPWVDCLLEEYFMQSDREKSEGLPVAPFMDRDKVTKATAQIGFIKFVLIPMFETVTKLFPMVEEIMLQPLWESRDRYEELKRIDDAMKELQKK 4y8d A 2.1 BS01 49J A 1 A67 K69 T123 C126 K127 G128 L180 A41 K43 T97 C100 K101 G102 L154 D173 K175 N178 D191 D147 K149 N152 D165 2.7.11.1 0004672,0005524,0006468 Kd=0.0089uM remove_due_to_license_issue Kd=8.9nM O14976 25822739 401 DFVGQTVELGELRLRVRRVLAEGGFAFVYEAQDVGSGREYALKRLLSNEEEKNRAIIQEVCFMKKLSGHPNIVQFCSAASIGKEESDTGQAEFLLLTELCKGQLVEFLKKMESRGPLSCDTVLKIFYQTCRAVQHMHRQKPPIIHRDLKVENLLLSNQGTIKLCDFGSATTISHYPYSNFPIGEKQDIWALGCILYLLCFRQHPFSIPPHDTQYTVFHSLIRAMLQVNPEERLSIAEVVHQLQEIAAARNVNPKSPITELLE 4y8x A 1.9 BS01 4GR A 1 R39 H40 L41 H57 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 Y228 R26 H27 L28 H44 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 26005539 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4y8y A 2.6 BS01 4D5 A 1 R39 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 W215 G216 G218 C219 G226 Y228 R26 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 W208 G209 G211 C212 G219 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 26005539 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4y8z A 2.2 BS01 4CE A 1 R39 H40 L41 H57 Y58B I151 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 V227 R26 H27 L28 H44 Y47 I141 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue Ki=0.040000nM P03951 26005539 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 4y94 A 2.4 BS01 IHP A 1 K36 K52 K29 K45 2.7.10.2 0035556 Kd=238nM remove_due_to_license_issue Q3ZC95 25699547 501 ATVILESIFLKRSSPLNFKKRLFLLTVQKLSYYEYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIPEESSETEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQIL 4y94 A 2.4 BS02 IHP A 2 K12 S14 R28 K53 K11 S13 R21 K46 2.7.10.2 0035556 Kd=238nM remove_due_to_license_issue Q3ZC95 25699547 502 ATVILESIFLKRSSPLNFKKRLFLLTVQKLSYYEYDFERGRRGSKKGSIDVEKITCVETVVPEKNPPPERQIPEESSETEQISIIERFPYPFQVVYDEGPLYVFSPTEELRKRWIHQLKNVIRYNSDLVQKYHPCFWIDGQYLCCSQTAKNAMGCQIL 4ya8 A 3.301 BS01 49W A 1 D34 G36 Y77 V78 S79 F111 T114 I123 Y192 D214 G216 T217 S218 I290 I300 D34 G36 Y77 V78 S79 F111 T114 I123 Y192 D214 G216 T217 S218 I290 I300 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue P46925 26625296 400 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 4yab A 1.9 BS03 4CN A 1 A923 V928 V932 N980 A95 V100 V104 N152 2.3.2.27 ic50=8.5uM remove_due_to_license_issue IC50=8500nM O15164 26061247 1103 SPNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4yad A 1.73 BS03 4A7 A 1 P929 Y935 F979 N980 P101 Y107 F151 N152 2.3.2.27 ic50=2.5uM remove_due_to_license_issue O15164 26061247 1103 PNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4yas A 2.0 BS01 CLX A 1 T11 S80 W128 F210 H235 T10 S79 W127 F209 H234 T11 S80 C81 D207 H235 K236 T10 S79 C80 D206 H234 K235 4.1.2.47 0009694,0009696,0016829,0047606,0052891,0052892,0080030,0080031,0080032 remove_due_to_license_issue P52704 10548044 300 AFAHFVLIHTICHGAWIWHKLKPLLEALGHKVTALDLAASGVDPRQIEEIGSFDEYSEPLLTFLEALPPGEKVILVGESCGGLNIAIAADKYCEKIAAAVFHNSVLPDTEHCPSYVVDKLMEVFPDWKDTTYFTYTKDGKEITGLKLGFTLLRENLYTLCGPEEYELAKMLTRKGSLFQNILAKRPFFTKEGYGSIKKIYVWTDQDEIFLPEFQLWQIENYKPDKVYKVEGGDHKLQLTKTKEIAEILQEVADTYN 4yat A 2.18 BS03 4A8 A 1 L922 A923 F924 V928 P929 N980 L90 A91 F92 V96 P97 N147 2.3.2.27 ic50=9.3uM remove_due_to_license_issue IC50=9300nM O15164 26061247 1103 PNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4yax A 2.25 BS01 4AE A 1 L922 A923 V928 P929 V932 F979 N980 V986 L96 A97 V102 P103 V106 F153 N154 V160 2.3.2.27 ic50=1.5uM remove_due_to_license_issue IC50=730nM O15164 26061247 1101 SPNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPSKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4yay A 2.9 BS01 ZD7 A 1 Y35 W84 S105 V108 S109 A163 R167 F182 P285 I288 Y129 W178 S199 V202 S203 A257 R261 F272 P361 I364 ? 0004930,0004945,0005506,0007186,0009055,0016020,0019229,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P30556 25913193 1201 DLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLILNSSDCPKAGRHNYIFVMIPTLYSIIFVVGIFGNSLVVIVIYFYMKLKTVASVFLLNLALADLCFLLTLPLWAVYTAMEYRWPFGNYLCKIASASVSFNLYASVFLLTCLSIDRYLAIVHPMKSRLRRTMLVAKVTCIIIWLLAGLASLPAIIHRNVFFIITVCAFHYETLPIGLGLTKNILGFLFPFLIILTSYTLIWKALKKNDDIFKIIMAIVLFFFFSWIPHQIFTFLDVLIQLGIIRDCRIADIVDTAMPITICIAYFNNCLNPLFYGFLGKKFKRYFLQLL 4yb5 A 2.24 BS01 HIS A 1 G247 V248 R250 T252 M267 V268 G239 V240 R242 T244 M259 V260 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 304 TRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLAHDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4yb5 E 2.24 BS01 HIS A 1 H232 S288 L290 H223 S279 L281 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 304 TRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQELKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLAHDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4yb5 E 2.24 BS02 HIS E 1 G247 V248 R250 T252 M267 V268 G238 V239 R241 T243 M258 V259 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 303 TRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQELKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLAHDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4yb6 A 1.98 BS01 AMP A 1 L170 S172 S173 G174 T176 L167 S169 S170 G171 T173 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 301 NTRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQENKFQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLAHDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4yb6 D 1.98 BS01 AMP D 1 C104 L170 S172 S173 G174 T176 C100 L166 S168 S169 G170 T172 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 301 TRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQENKFQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLAHDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4yb7 B 2.2 BS02 ATP B 1 Q12 G15 R16 L17 R54 D55 N75 G102 Y103 C104 S172 Q9 G12 R13 L14 R51 D52 N72 G99 Y100 C101 S169 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 303 NTRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQENKFQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLAHDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4yb7 C 2.2 BS03 ATP C 1 Q12 G15 R16 R54 D55 N75 C104 L170 S172 Q9 G12 R13 R51 D52 N72 C101 L167 S169 2.4.2.17 0000105,0000287,0003879,0005524,0005737,0016757,0046872 remove_due_to_license_issue Q5HSJ4 27191057 304 NTRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQENKFQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARESKYIMLHAPKEKLDKIQALLPGVERPTILPLDEKNVALHMVSKENLFWETMEALKEEGASSILVLPIEKMLK 4ybi A 1.84 BS01 4B2 A 1 G13 L30 D32 Y71 F108 W115 I118 D228 G230 G17 L34 D36 Y75 F112 W119 I122 D232 G234 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=239nM remove_due_to_license_issue IC50=270nM, EC50=300nM P56817 22090477 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVASQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4ybj A 2.61 BS01 4A9 A 1 L273 A293 K295 E310 M314 I336 T338 Y340 M341 S342 G344 L393 V402 A403 D404 F405 L15 A33 K35 E50 M54 I76 T78 Y80 M81 S82 G84 L133 V142 A143 D144 F145 D386 R388 A390 N391 D404 D126 R128 A130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 26895387 601 AWEIPRESLRLEVKLGQGGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4ybk A 2.5 BS01 4B7 A 1 L273 A293 K295 M314 I336 T338 Y340 M341 S342 G344 L393 D404 F405 L18 A38 K40 M59 I81 T83 Y85 M86 S87 G89 L138 D149 F150 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F157 2.7.10.2 0004672,0004713,0005524,0006468 Kd=15nM remove_due_to_license_issue P00523 26895387 601 AKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 4ybm B 1.46 BS01 4BJ B 1 Y936 T947 R951 M958 Y100 T111 R115 M122 2.3.2.27 ic50=0.14uM remove_due_to_license_issue EC50=3900nM, IC50=140nM O15164 26061247 1101 NEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4ybm B 1.46 BS02 4BJ B 2 L922 A923 V928 P929 F979 N980 V986 L86 A87 V92 P93 F143 N144 V150 2.3.2.27 ic50=0.14uM remove_due_to_license_issue EC50=3900nM, IC50=140nM O15164 26061247 1102 NEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4ybs A 1.83 BS03 4BK A 1 A923 F924 V928 F979 N980 E985 V986 A95 F96 V100 F151 N152 E157 V158 2.3.2.27 ic50=0.057uM remove_due_to_license_issue EC50=1300nM, IC50=<10nM O15164 26061247 1103 PNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4ybt A 1.82 BS03 4BV A 1 A923 F924 V928 P929 F979 N980 E985 V986 A95 F96 V100 P101 F151 N152 E157 V158 2.3.2.27 ic50=0.1uM remove_due_to_license_issue O15164 26061247 1104 PNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4yc0 A 1.5 BS01 5OF A 1 Y72 R117 G118 S142 T143 A150 F153 Y54 R99 G100 S124 T125 A132 F135 2.4.2.31 0000166,0005576,0016757,0016779,0035821,0090729,0106274 Ki=74uM remove_due_to_license_issue A3UNN4 26352925 301 GPFDAIKQPNRSEEEVTQLAEDFKDWSKASNGWRYSFITANEKEAVEDFSISGYQTANDYLRATDTSTWGVAGADARQYIRTVKSALNKLPKYKGTAYRGTWVKLSLLNKLEEGDVLVEPAFTSTSTLPEVAKRFSVVHPNSPQRLKRVLFEVKINQGGHTIAGLSEYSKEAEVLFAPNAHFRITQIERTSNHTYIGVETVKASAVKNTQKYNLYSGEEVEA 4yc8 A 2.9 BS01 4B7 A 1 L248 A269 K271 F283 A287 M290 I313 T315 M318 T319 Y320 G321 L370 F382 L16 A31 K33 F41 A45 M48 I71 T73 M76 T77 Y78 G79 L128 F140 D363 A365 R367 N368 D381 P402 D121 A123 R125 N126 D139 P160 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00519 26895387 601 DKWEMERTDITMKHKLEVYEGVWKKYSLTVAVKTLMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESS 4yc9 A 1.82 BS03 4C1 A 1 A923 F924 Q925 D926 V928 V932 F979 N980 A97 F98 Q99 D100 V102 V106 F153 N154 2.3.2.27 Kd=1.3nM remove_due_to_license_issue Kd=31nM, IC50=7.6nM, EC50=50nM O15164 26061247 1104 SPNEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPSKKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 4ycl A 3.25 BS01 CZA A 1 L61 V62 L98 N101 A102 L311 L61 V62 L98 N101 A102 L311 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 17389383 1003 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 4ycm A 3.2 BS01 7BS A 1 Q56 D59 N101 G105 K246 Q250 L253 I307 P308 L311 P312 I315 Q56 D59 N101 G105 K246 Q250 L253 I307 P308 L311 P312 I315 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue Ki=19nM P04191 25957767 1004 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 4ycn A 3.5 BS01 7BL A 1 N101 V104 G105 Q250 L253 L311 P312 I315 N101 V104 G105 Q250 L253 L311 P312 I315 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue Ki=17nM P04191 25957767 1004 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 4ycu A 2.1 BS01 KRS A 1 E325 H331 N332 F335 N497 G550 R553 E254 H260 N261 F264 N426 G479 R482 R323 E325 T330 H331 E494 N497 R553 R252 E254 T259 H260 E423 N426 R482 2.7.7.-,6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 remove_due_to_license_issue IC50=>20000nM Q15046 26074468 601 DPNQYYKIRSQAIHQLKVNGEDPYPHKFHVDISLTDFIQKYSHLQPGDHLTDITLKVAGRIHAKRASGGKLIFYDLRGEGVKLQVMANSRNYKSEEEFIHINNKLRRGDIIGVQGNPGKTKKGELSIIPYEITLLSPCLHMLPHLHFGLKDKETRYRQRYLDLILNDFVRQKFIIRSKIITYIRSFLDELGFLEIETPMMNIIPGGAVAKPFITYHNELDMNLYMRIAPELYHKMLVVGGIDRVYEIGRQFRNEGIDLTHNPEFTTCEFYMAYADYHDLMEITEKMVSGMVKHITGSYKVTYHPDGPEGQAYDVDFTPPFRRINMVEELEKALGMKLPETNLFETEETRKILDDICVAKAVECPPPRTTARLLDKLVGEFLEVTCINPTFICDHPQIMSPLAKWHRSKEGLTERFELFVMKKEICNAYTELNDPMRQRQLFEEQAKAKAAGDDEAMFIDENFCTALEYGLPPTAGWGMGIDRVAMFLTDSNNIKEVLLFPAMKPE 4ycv A 3.406 BS01 KRS A 1 H338 N339 F342 E500 V501 R559 H256 N257 F260 E418 V419 R463 R330 E332 T337 H338 E500 N503 R559 R248 E250 T255 H256 E418 N421 R463 6.1.1.6 0000049,0000166,0003676,0004812,0004824,0005524,0005737,0005829,0006418,0006430 remove_due_to_license_issue W7JP72 26074468 601 VDPRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSAQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKYGLKDTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFKLLDSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRP 4ycw A 2.9 BS04 KRS A 1 R323 E325 H331 N332 F335 E494 I495 C496 N497 G550 R553 R249 E251 H257 N258 F261 E420 I421 C422 N423 G476 R479 R323 E325 T330 H331 E494 N497 R553 R249 E251 T256 H257 E420 N423 R479 2.7.7.-,6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 remove_due_to_license_issue IC50=>20000nM Q15046 602 DPNQYYKIRSQAIHQLKVNGEDPYPHKFHVDISLTDFIQKYSHLQPGDHLTDITLKVAGRIHAKRASGGKLIFYDLRGEGVKLQVMANSRNYKSEEEFIHINNKLRRGDIIGVQGNPGKTKKGELSIIPYEITLLSPCLHMLPHLLKDKETRYRQRYLDLILNDFVRQKFIIRSKIITYIRSFLDELGFLEIETPMMNIIPGGAVAKPFITYHNELDMNLYMRIATELYHKMLVVGGIDRVYEIGRVFRNEGIDLTHNPEFTSCEFYMAYADYHDLMEITEKMVSGMVKHITGSYKVTYHPDGPEGQAYDVDFTPPFRRINMVEELEKALGMKLPETNLFETEETRKILDDICVAKAVECPPPRTTARLLDKLVGEFLEVTCINPTFICDHPQIMSPLAKWHRSKEGLTERFELFVMKKEICNAYTELNDPMRQRQLFEEQAKAKAAGDDEAMFIDENFCTALEYGLPPTAGWGMGIDRVAMFLTDSNNIKEVLLFPAMKP 4ydf A 2.804 BS01 4B1 A 1 D32 D36 M37 G58 A59 W98 D32 D36 M37 G58 A59 W98 ? 0004190,0006508,0008233,0046872 remove_due_to_license_issue Q82134 26000468 201 PVIPLDPARRPVIKAQVDTQTSHPKTIEALLDTGADMTVIPIALFSSNTPLKNTSVLGAGGQTQDHFKLTSLPVLIRLPFRTTPIVLTSCLVDTKNNWAIIGRDALQQCQGVLYLP 4ydf B 2.804 BS01 4B1 A 1 D32 M37 L57 G58 A59 W98 D32 M37 L57 G58 A59 W98 ? 0004190,0006508,0008233,0046872 remove_due_to_license_issue Q82134 26000468 201 PVIPLDPARRPVIKAQVDTQTSHPKTIEALLDTGADMTVIPIALFSSNTPLKNTSVLGAGGQTQDHFKLTSLPVLIRLPFRTTPIVLTSCLVDTKNNWAIIGRDALQQCQGVLYLP 4ydg A 3.25 BS01 G3G B 1 D32 W98 D32 W90 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0004190,0006508 remove_due_to_license_issue P03362 26000468 201 PVIPLDPARRPVIKAQVDTQTSHPKTIEALLDTGADMTVIPIALFSSNTPLKNTTQDHFKLTSLPVLIRLPFRTTPIVLTSCLVDTKNNWAIIGRDALQQCQGVLYLP 4ydg B 3.25 BS01 G3G B 1 D32 G34 A35 D36 M37 W98 D32 G34 A35 D36 M37 W93 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- 0004190,0006508 remove_due_to_license_issue P03362 26000468 201 PVIPLDPARRPVIKAQVDTQTSHPKTIEALLDTGADMTVIPIALFSSNTPLKNTSVLTQDHFKLTSLPVLIRLPFRTTPIVLTSCLVDTKNNWAIIGRDALQQCQGVLYLP 4ydn A 1.35 BS01 2WN A 1 X15 A108 L110 S117 T118 X6 A99 L101 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 26051248 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4ydn B 1.35 BS01 2WN B 1 M13 L17 T106 S117 T118 M4 L8 T97 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 26051248 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 4ydq A 2.3 BS02 HFG A 1 F335 E338 V339 P358 T359 E361 R390 F454 T478 H480 W509 G510 F82 E85 V86 P105 T106 E108 R137 F201 T225 H227 W256 G257 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 Kd~300nM remove_due_to_license_issue Q8I5R7 25817387 802 MAITSKKIENFSDWYTQVIVKSELIEYYDISGCYILRPAAYYIWECVQAFFNKEIKKLNVENSYFPLFVTKNKLEKEKNHGFSPEVAWVTKYGDSNLPEEIAIRPTSETIMYSVFPKWIRSYRDLPLKLNQWNTVVRWEFKQPTPFIRTREFLWQEGHTAHKNEEEAVKLVFDILDLYRRWYEEYLAVPIIKGIKSEGEKFGGANFTSTAEAFISENGRAIQAATSHYLGTNFAKMFKIEFEDENEVKQYVHQTSWGCTTRSIGIMIMTHGDDKGLVLPPNVSKYKVVIVPIFYKTTDENAIHSYCKDIEKILKNAQINCVYDDRASYSPGYKFNHWELRGIPIRIEVGPKDLQNNSCVIVRRDNNEKCNVKKESVLLETQQMLVDIHKNLFLKAKKKLDDSIVQVTSFSEVMNALNKKKMVLAPWCEDIATEEEIKKETQRLSLNQSGAMKPLCIPLDQPPMPPNMKCFWSGKPAKRWCLFGRSY 4ydq B 2.3 BS02 HFG B 1 F335 P358 T359 E361 R390 F454 T478 H480 W509 G510 F76 P99 T100 E102 R131 F195 T219 H221 W250 G251 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 Kd~300nM remove_due_to_license_issue Q8I5R7 25817387 802 MAITSKKIENFSDWYTQVIVKSELIEYYDISGCYILRPAAYYIWECVQAFFNKEIKKLNVENSYFPLFVTKNKLEFSPEVAWVTKYGDSNLPEEIAIRPTSETIMYSVFPKWIRSYRDLPLKLNQWNTVVRWEFKQPTPFIRTREFLWQEGHTAHKNEEEAVKLVFDILDLYRRWYEEYLAVPIIKGIKSEGEKFGGANFTSTAEAFISENGRAIQAATSHYLGTNFAKMFKIEFEDENEVKQYVHQTSWGCTTRSIGIMIMTHGDDKGLVLPPNVSKYKVVIVPIFYKTTDENAIHSYCKDIEKILKNAQINCVYDDRASYSPGYKFNHWELRGIPIRIEVGPKDLQNNSCVIVRRDNNEKCNVKKESVLLETQQMLVDIHKNLFLKAKKKLDDSIVQVTSFSEVMNALNKKKMVLAPWCEDIATEEEIKKETQRLTLSGAMKPLCIPLDQPPMPPNMKCFWSGKPAKRWCLFGRSY 4ye3 A 1.35 BS01 G04 B 1 D25 G27 A28 N30 V82 D25 G27 A28 N30 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 26010498 201 PQITLWKRPFVTVKVGGQLKEALLDTGADNTIFEDINLPGRWKPKMVGGIGGFLKVREYDQVPIEIAGHKVIGTVLVGPTPVNVIGRDTMTQIGATLNF 4ye3 B 1.35 BS01 G04 B 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.3nM remove_due_to_license_issue P03366 26010498 201 PQITLWKRPFVTVKVGGQLKEALLDTGADNTIFEDINLPGRWKPKMVGGIGGFLKVREYDQVPIEIAGHKVIGTVLVGPTPVNVIGRDTMTQIGATLNF 4yes B 1.5 BS04 45S B 1 H406 W413 A563 C564 S568 V588 S589 W590 G591 G593 G601 F602 H43 W50 A193 C194 S198 V218 S219 W220 G221 G223 G231 F232 H406 D462 E565 G566 D567 S568 G569 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=9.6nM remove_due_to_license_issue P00734 26005532 704 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 4yff A 3.07 BS01 4CV A 1 I469 A488 K490 T539 Y541 I542 H592 L595 D606 I25 A44 K46 T88 Y90 I91 H141 L144 D155 D588 N590 H592 N593 D606 N627 D137 N139 H141 N142 D155 N165 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=<10.0nM Q59H18 26355916 801 ILLLRAGLPSHFHLQLSEIEFHEIIGSGSFGKVYKGRCRNKIVAIKRYRSDVDMFCREVSILCQLNHPCVIQFVGACLNDPSQFAIVTQYISGGSLFSLLHEQKRILDLQSKLIIAVDVAKGMEYLHNLTQPIIHRDLNSHNILLYEDGHAVVADFGESRFLQSNLRWMAPEVFTQCTRYTIKADVFSYALCLWEILTGEIPFAHLKPAAAAADMAYHHIRPPIGYSIPKPISSLLIRGWNACPEGRPEFSEVVMKLEECLCNI 4yfi A 2.7 BS01 4CW A 1 I469 V477 A488 K490 T539 Y541 I542 L595 D606 I29 V37 A48 K50 T92 Y94 I95 L148 D159 D588 N590 H592 N593 D606 N627 D141 N143 H145 N146 D159 N169 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=500nM, Kd=111nM Q59H18 26355916 801 EKADILLLRAGLPSHFHLQLSEIEFHEIIGSGSFGKVYKGRCRNKIVAIKRYRSDVDMFCREVSILCQLNHPCVIQFVGACLNDPSQFAIVTQYISGGSLFSLLHEQKRILDLQSKLIIAVDVAKGMEYLHNLTQPIIHRDLNSHNILLYEDGHAVVADFGESRFLQGNLRWMAPEVFTQCTRYTIKADVFSYALCLWEILTGEIPFAHLKPAAADMDMAYHHIRPPIGYSIPKPISSLLIRGWNACPEGRPEFSEVVMKLEECLCNI 4ygf A 2.0 BS02 AZM A 1 H110 H112 H129 V131 L190 T191 W201 H89 H91 H108 V110 L169 T170 W180 H85 H110 H112 E116 H129 T191 H64 H89 H91 E95 H108 T170 ? 0004089,0008270,0046872 Ki=21nM remove_due_to_license_issue A0A0M3KL20 26010545 303 KWDYKNKENGPHRWDKLHKDFEVCKSGKSQSPINIEHYYHTQDKADLQFKYAASKPKAVFFTHHTLKASFEPTNHINYRGHDYVLDNVHFHAPMEFLINNKTRPLSAHFVHKDAKGRLLVLAIGFEEGKENPNLDPILEGIQKKQNFKEVALDAFLPKSINYYHFNGSLTAPPCTEGVAWFVIEEPLEVSAKQLAEIKKRMKNSPNQRPVQPDYNTVIIKSSAETR 4ygi A 2.6 BS01 dna B 0 Y378 R379 S391 Q392 G394 S413 G415 Y416 D418 Y428 T429 Q431 Y486 Y17 R18 S30 Q31 G33 S52 G54 Y55 D57 Y67 T68 Q70 Y112 2.1.1.-,2.1.1.367 remove_due_to_license_issue O82175 26841909 1 ~ 10 QIIGTVPGVEVGDEFQYRMELNLLGIHRPSQSGIDYMKDDGGELVATSIVSSGGYNDVLDNSDVLIYTGQGGNVGKKEPPKDQQLVTGNLALKNSINKKNPVRVIRGIKKNYVYDGLYLVEEYWEETGSHGKLVFKFKLRRIPGQPELPW 4yh3 A 1.6 BS01 Y80 A 1 W81 P82 L92 L94 Y139 N140 I146 W40 P41 L51 L53 Y98 N99 I105 ? ic50=26uM remove_due_to_license_issue IC50=26000nM O60885 26022843 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEET 4yh4 A 1.33 BS01 Y81 A 1 W81 P82 L92 L94 N140 I146 M149 W40 P41 L51 L53 N99 I105 M108 ? ic50=26uM remove_due_to_license_issue IC50=26000nM O60885 26022843 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 4yha A 2.2 BS02 MZM A 1 N108 H110 H112 H129 V131 L190 T191 W201 N88 H90 H92 H109 V111 L168 T169 W179 H85 H110 H112 E116 H129 T191 H65 H90 H92 E96 H109 T169 ? 0004089,0008270,0046872 Ki=225nM remove_due_to_license_issue A0A0M3KL20 26010545 303 TKWDYKNKENGPHRWDKLHKDFEVCKSGKSQSPINIEHYYHTQDKADLQFKYAASKPKAVFFTHHTLKASFEPTNHINYRGHDYVLDNVHFHAPMEFLINNKTRPLSAHFVHKDAKGRLLVLAIGFEEGKENPNLDPILEGIQKKFKEVALDAFLPKSINYYHFNGSLTAPPCTEGVAWFVIEEPLEVSAKQLAEIKKRMKNSPNQRPVQPDYNTVIIKSSAETR 4yhf A 2.2 BS01 4C9 A 1 V416 A428 K430 M449 V458 I472 T474 Y476 M477 G480 C481 N484 S538 D539 F540 L542 V26 A38 K40 M59 V68 I82 T84 Y86 M87 G90 C91 N94 S148 D149 F150 L152 D521 A523 R525 N526 D539 F559 D131 A133 R135 N136 D149 F169 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 26006010 701 GYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4yhm H 2.16 BS01 4CC H 1 D31 Y33 H35 E50 N52 R54 Y103 Y105 F106 D31 Y33 H35 E50 N52 R54 Y103 Y105 F106 Kd=173pM remove_due_to_license_issue 26047352 301 QVQLVQSGAEVKKPGASVKVSCKASGYTFTDYYMHWVRQAPGQGLEWMGETNPRNGGTTYNEKFKGKATMTRDTSTSTAYMELSSLRSEDTAVYYCTIGTSGYDYFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 4yhm L 2.16 BS01 4CC H 1 E39 A96 Y101 E39 A96 Y101 remove_due_to_license_issue 26047352 301 DIVMTQTPLSLSVTPGQPASISCRSSQSIVHSDGNIYLEWYLQKPGQSPKLLIYKVSYRFSGVPDRFSGSGSGTGFTLKISRVEAEDVGVYYCFQASHVPYTFGGGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 4yho H 1.82 BS01 4CC H 1 D31 Y33 H35 E50 N52 R54 W103 D104 Y105 F106 D31 Y33 H35 E50 N52 R54 W103 D104 Y105 F106 Kd=18pM remove_due_to_license_issue 26047352 301 QVQLVQSGAEVKKPGASVKVSCKASGYTFTDYYMHWVRQAPGQGLEWMGETNPRNGGTTYNEKFKGKATMTRDTSTSTAYMELSSLRSEDTAVYYCTIGTSGWDYFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 4yho L 1.82 BS01 4CC H 1 E39 A96 E39 A96 remove_due_to_license_issue 26047352 301 DIVMTQTPLSLSVTPGQPASISCRSSQSIVHSDGNIYLEWYLQKPGQSPKLLIYKVSYRFSGVPDRFSGSGSGTDFTLKISRVEAEDVGVYYCFQASHVPYTFGQGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 4yhq A 1.3 BS01 G10 A 1 D25 G27 D29 N30 G48 G49 I50 D25 G27 D29 N30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.7nM remove_due_to_license_issue P03366 26010498 201 PQITLWKRPFVTVKVGGQLKEALLDTGADNTIFEDINLPGRWKPKMVGGIGGFLKVREYDQVPIEIAGHKVIGTVLVGPTPVNVIGRDTMTQIGATLNF 4yhq B 1.3 BS01 G10 A 1 D25 A28 N30 I32 V82 D25 A28 N30 I32 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 26010498 201 PQITLWKRPFVTVKVGGQLKEALLDTGADNTIFEDINLPGRWKPKMVGGIGGFLKVREYDQVPIEIAGHKVIGTVLVGPTPVNVIGRDTMTQIGATLNF 4yht A 3.05 BS01 4EF A 1 I462 V470 A480 K482 T528 W530 C531 G533 N579 F582 D593 I15 V23 A33 K35 T81 W83 C84 G86 N132 F135 D146 D575 K577 N579 N580 D593 S615 D128 K130 N132 N133 D146 S155 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.600000nM P15056 27246618 1002 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHTNETKFEMTKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKGSILWMAPEVIRMQDPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPTFPQILASIETLAR 4yhw A 3.25 BS01 rna E 0 P350 R353 F354 K357 K361 S364 R371 D374 R399 G439 W440 F441 M442 Q457 P16 R19 F20 K23 K27 S30 R37 D40 R65 G105 W106 F107 M108 Q123 ? 0000398,0046540 remove_due_to_license_issue Q03338 26161500 64 ~ 90 TVYHCKVFQFKNLQNPKIRFKLKMNSKELSLKGLCLRIRDDGPGIIIVVGNEKSCKFYENLVMKRIKWNEDFELHTNTGDIKMDMHNNSISKTWEGYLQDCKFKGWFMKVCNDQDSLLRTLGQFDSEHFYSPV 4yhw B 3.25 BS01 rna F 0 P350 K351 R353 F354 K357 K361 R371 D374 G439 W440 F441 M442 Q457 P16 K17 R19 F20 K23 K27 R37 D40 G105 W106 F107 M108 Q123 ? 0000398,0046540 remove_due_to_license_issue Q03338 26161500 64 ~ 90 TVYHCKVFQFKNLQNPKIRFKLKMNSKELSLKGLCLRIRDDGPGIIIVVGNEKSCKFYENLVMKRIKWNEDFELHTNTGDIKMDMHNNSISKTWEGYLQDCKFKGWFMKVCNDQDSLLRTLGQFDSEHFYSPV 4yih A 1.82 BS02 2O2 A 1 D12 F18 F44 L45 R47 Y65 L102 L103 R132 D9 F15 F41 L42 R44 Y62 L99 L100 R129 D10 D12 D145 D7 D9 D142 3.1.3.- 0000166,0000255,0005634,0005737,0005739,0005829,0006204,0006249,0008252,0008253,0009117,0009223,0009264,0016311,0016787,0016791,0019103,0042802,0043605,0046050,0046055,0046074,0046079,0046872,0050483,0070062 remove_due_to_license_issue Q8TCD5 203 SVRVLVDMDGVLADFEAGLLRGFRRRFPEEPHVPLEQRRGFLAREQYRALRPDLADKVASVYEAPGFFLDLEPIPGALDAVREMNDLPDTQVFICTSPLLKYHHCVGEKYRWVEQHLGPQFVERIILTRDKTVVLGDLLIDDKDTVRGQEETPSWEHILFTCCHNRHLVLPPTRRRLLSWSDNWREILDSKR 4yih B 1.82 BS02 2O2 B 1 D12 F18 F44 L45 A46 R47 Y65 L102 L103 R132 D9 F15 F41 L42 A43 R44 Y62 L99 L100 R129 D10 D12 D145 D7 D9 D142 3.1.3.- 0000166,0000255,0005634,0005737,0005739,0005829,0006204,0006249,0008252,0008253,0009117,0009223,0009264,0016311,0016787,0016791,0019103,0042802,0043605,0046050,0046055,0046074,0046079,0046872,0050483,0070062 remove_due_to_license_issue Q8TCD5 203 SVRVLVDMDGVLADFEAGLLRGFRRRFPEEPHVPLEQRRGFLAREQYRALRPDLADKVASVYEAPGFFLDLEPIPGALDAVREMNDLPDTQVFICTSPLLKYHHCVGEKYRWVEQHLGPQFVERIILTRDKTVVLGDLLIDDKDTVRGQEETPSWEHILFTCCHNRHLRRRLLSWSDNWREILDSKR 4yik A 1.483 BS02 2O2 A 1 D41 D43 F49 F75 W76 V77 W96 S131 I133 K134 R163 D15 D17 F23 F49 W50 V51 W70 S105 I107 K108 R137 D41 D43 D176 D15 D17 D150 3.1.3.- 0008253,0009264 remove_due_to_license_issue Q9NPB1 306 SNAASGGRALRVLVDMDGVLADFEGGFLRKFRARFPDQPFIALEDRRGFWVSEQYGRLRPGLSEKAISIWESKNFFFELEPLPGAVEAVKEMASLQNTDVFICTSPIKMFKYCPYEKYAWVEKYFGPDFLEQIVLTRDKTVVSADLLIDDRPDITGAEPTPSWEHVLFTACHNQHLQLQPPRRRLHSWADDWKAILDSKRP 4yir A 3.0501 BS01 dna W 0 R129 C131 N134 S437 V438 Q439 H472 R494 Q495 F556 F597 F599 T604 V605 P607 R4 C6 N9 S312 V313 Q314 H347 R369 Q370 F423 F464 F466 T471 V472 P474 ? 0003677,0003684,0005634,0006289 remove_due_to_license_issue P14736 25562780 1 ~ 24 RTSRNCSSNEERKRRKYFHMLYLVCLMVHGFIRNEWINSKRLSRKLSNLVPEKVFELLHPQKDEELPLRSTRKLLDGLKKCMELWQKHWKITKKYDNEGLYMRTWKEIEMSANNKRKFKTLKRSDFLRAVSKGHGDPDISVQGFVAMLRACNVNARLIMSCQPPDFTNMKIDTSLNGNNAYKDMVKYPIFWCEVWDKFSKKWITVDPVNLKTIEQVRLHSKLAPKGVACCERNMLRYVIAYDRKYGCRDVTRRYAQWMNSKVRKRRITKDDFGEKWFRKVITALHHRKRTKIDDYEDQYFFRRDESEGIPDSVQDLKNHPYYVLEQDIKQTQIVKPGCKECGYLKVHGKVGKVLKVYAKRDIADLKSARQWYMNGRILKTGSRCKKVIKRTEEEDERLYSFEDTELYIPPLASASGEITKNTFGNIEVFAPTMIPGNCCLVENPVAIKAARFLGVEFAPAVTSFKFERGSTVKPVLSGIVVAKWLREAIETAIDGIEFI 4yir A 3.0501 BS02 dna Y 0 N130 N293 M294 K295 N443 F599 E600 R601 N5 N168 M169 K170 N318 F466 E467 R468 ? 0003677,0003684,0005634,0006289 remove_due_to_license_issue P14736 25562780 1 ~ 24 RTSRNCSSNEERKRRKYFHMLYLVCLMVHGFIRNEWINSKRLSRKLSNLVPEKVFELLHPQKDEELPLRSTRKLLDGLKKCMELWQKHWKITKKYDNEGLYMRTWKEIEMSANNKRKFKTLKRSDFLRAVSKGHGDPDISVQGFVAMLRACNVNARLIMSCQPPDFTNMKIDTSLNGNNAYKDMVKYPIFWCEVWDKFSKKWITVDPVNLKTIEQVRLHSKLAPKGVACCERNMLRYVIAYDRKYGCRDVTRRYAQWMNSKVRKRRITKDDFGEKWFRKVITALHHRKRTKIDDYEDQYFFRRDESEGIPDSVQDLKNHPYYVLEQDIKQTQIVKPGCKECGYLKVHGKVGKVLKVYAKRDIADLKSARQWYMNGRILKTGSRCKKVIKRTEEEDERLYSFEDTELYIPPLASASGEITKNTFGNIEVFAPTMIPGNCCLVENPVAIKAARFLGVEFAPAVTSFKFERGSTVKPVLSGIVVAKWLREAIETAIDGIEFI 4yjn A 2.6 BS01 UW4 A 1 L57 G58 V65 A78 M112 L126 Y131 I194 L198 L15 G16 V23 A36 M70 L84 Y89 I152 L156 D174 K176 E178 N179 D195 T214 D132 K134 E136 N137 D153 T172 ? 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue IC50=12nM Q9BJF5 26693272 601 STAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 4yk5 A 1.42 BS01 4DV A 1 P124 S127 Y130 T131 Q134 P118 S121 Y124 T125 Q128 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=0.96uM remove_due_to_license_issue IC50=3nM O14684 25961169 201 VMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 4ykj A 1.401 BS01 ALA A 1 F63 D91 S93 R98 R144 H145 E188 F59 D87 S89 R94 R140 H141 E184 ? 0015276,0016020,0034220,0046872 Ki=37uM remove_due_to_license_issue A0A0R4I973 26460032 301 LIGRHLRLGSVEEQPFMFFATEGCEGNDCWSGMVNDMVVKLSEDLGFTYEYIQPDDRKFGALNKTTNEWNGMIRDLLDDKTDMIAIDLSTNSARKSAIDYSFPFMDAGIKAVVKGEGTTLNQVLELLDQDKYKWGVIGSRHPETLLKTHRDSRYSRLVDEGVELKDLNHAIETLRGGLFVFIDEGPVLAHNLISDCDVFSVGEEFQSFEYAFGLPKDSPYKSLIDSHLLKFREEGFIDILWEKWSSG 4ykk A 1.38 BS02 DSN A 1 F63 D91 S93 R98 R144 H145 E188 F60 D88 S90 R95 R141 H142 E185 ? 0015276,0016020,0034220,0046872 Ki=1.7mM remove_due_to_license_issue A0A0R4I973 26460032 302 NLIGRHLRLGSVEEQPFMFFATEGCEGNDCWSGMVNDMVVKLSEDLGFTYEYIQPDDRKFGALNKTTNEWNGMIRDLLDDKTDMIAIDLSTNSARKSAIDYSFPFMDAGIKAVVKGEGTTLNQVLELLDQDKYKWGVIGSRHPETLLKTHRDSRYSRLVDEGVELKDLNHAIETLRGGLFVFIDEGPVLAHNLISDCDVFSVGEEFQSFEYAFGLPKDSPYKSLIDSHLLKFREEGFIDILWEKWSS 4ykn A 2.9 BS01 4EL A 1 R1770 M1772 S1774 K1802 Y1836 I1848 V1851 Q1859 S1919 M1922 I1932 D1933 R928 M930 S932 K960 Y994 I1006 V1009 Q1017 S1077 M1080 I1090 D1091 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue P27986,P42336 26005528 2101 AEWYWGDISREEVNEKLRDTADGTFLVRDYTLTLRKGGNNKLIKIFHYGFSDPLTVVELINHYRNKLDVKLLYPVYNTQFQEKSREYDRLYEEYTRTSQEIQMKRTAIEAFNETIKIFEEQCQTQERYSKEYIEKFKREGNEKEIQRIMHNYDKLKSRISEIIDSRRRLEEDLKKQAAEYREIDKRMNSIKPDLIQLRKTRDQYLWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRSTKSLWVINSALRIKILCATYVNVNIIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSRELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGGLKGALQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKKKERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWT 4ykn A 2.9 BS02 4EL A 2 W1328 V1329 H1495 R1577 W510 V511 H672 R735 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue P27986,P42336 26005528 2102 AEWYWGDISREEVNEKLRDTADGTFLVRDYTLTLRKGGNNKLIKIFHYGFSDPLTVVELINHYRNKLDVKLLYPVYNTQFQEKSREYDRLYEEYTRTSQEIQMKRTAIEAFNETIKIFEEQCQTQERYSKEYIEKFKREGNEKEIQRIMHNYDKLKSRISEIIDSRRRLEEDLKKQAAEYREIDKRMNSIKPDLIQLRKTRDQYLWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRSTKSLWVINSALRIKILCATYVNVNIIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSRELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGGLKGALQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKKKERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWT 4ykn A 2.9 BS03 4EL A 3 W1328 Y1392 E1494 H1495 W1498 R1577 W510 Y572 E671 H672 W675 R735 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue P27986,P42336 26005528 2103 AEWYWGDISREEVNEKLRDTADGTFLVRDYTLTLRKGGNNKLIKIFHYGFSDPLTVVELINHYRNKLDVKLLYPVYNTQFQEKSREYDRLYEEYTRTSQEIQMKRTAIEAFNETIKIFEEQCQTQERYSKEYIEKFKREGNEKEIQRIMHNYDKLKSRISEIIDSRRRLEEDLKKQAAEYREIDKRMNSIKPDLIQLRKTRDQYLWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRSTKSLWVINSALRIKILCATYVNVNIIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSRELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGGLKGALQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKKKERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWT 4yl0 A 1.52 BS01 4DZ A 1 P124 S127 T131 P120 S123 T127 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=1.59uM remove_due_to_license_issue IC50=1nM O14684 25961169 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 4yl1 A 1.41 BS01 4U8 A 1 P124 S127 V128 T131 L135 P120 S123 V124 T127 L131 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=2.58uM remove_due_to_license_issue IC50=216nM O14684 25961169 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 4yl3 A 1.41 BS01 4U9 A 1 P124 S127 V128 T131 P118 S121 V122 T125 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=3.94uM remove_due_to_license_issue O14684 25961169 201 VMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 4ylj A 2.58 BS01 4E1 A 1 F170 V173 K188 F238 L241 L294 D307 F36 V39 K54 F104 L107 L160 D173 D287 K289 N292 D307 S324 D153 K155 N158 D173 S190 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=6.0nM Q13627 25730262 505 VYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDGKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 4ylk A 1.4 BS01 4E2 A 1 K167 F170 V173 K188 F238 L241 L294 D307 K34 F37 V40 K55 F105 L108 L161 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 ic50=0.18uM remove_due_to_license_issue IC50=180nM Q13627 25730262 519 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 4yll A 1.4 BS01 4E3 A 1 K167 F170 K188 F238 L241 L294 D307 K34 F37 K55 F105 L108 L161 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 ic50=0.12uM remove_due_to_license_issue IC50=120nM Q13627 25730262 515 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 4ylu A 2.1 BS01 R30 A 1 M25 H41 L49 F143 C148 H166 M168 E169 D190 K191 Q192 M25 H41 L49 F143 C148 H166 M168 E169 D190 K191 Q192 H41 G146 C148 H41 G146 C148 3.4.19.12 0008233,0019082 remove_due_to_license_issue V9TU12 26055715 401 SGLVKMSHPSGDVEACMVQVTCGSMTLNGLWLDNTVWCPRHVMCPADQLSDPNYDALLISMTNHSFSVQKHIGAPANLRVVGHAMQGTLLKLTVDVANPSTPAYTFTTVKPGAAFSVLACYNGRPTGTFTVVMRPNYTIKGSFLCGSCGSVGYTKEGSVINFCYMHQMELANGTHTGSAFDGTMYGAFMDKQVHQVQLTDKYCSVNVVAWLYAAILNGCAWFVKPNRTSVVSFNEWALANQFTEFVGTQSVDMLAVKTGVAIEQLLYAIQQLYTGFQGKQILGSTMLEDEFTPEDVNMQIMGVV 4ylu B 2.1 BS01 R30 B 1 M25 H41 L49 F143 L144 C148 H166 M168 E169 D190 K191 M25 H41 L49 F143 L144 C148 H166 M168 E169 D190 K191 H41 G146 C148 H41 G146 C148 3.4.19.12 0008233,0019082 remove_due_to_license_issue V9TU12 26055715 401 SGLVKMSHPSGDVEACMVQVTCGSMTLNGLWLDNTVWCPRHVMCPADQLSDPNYDALLISMTNHSFSVQKHIGAPANLRVVGHAMQGTLLKLTVDVANPSTPAYTFTTVKPGAAFSVLACYNGRPTGTFTVVMRPNYTIKGSFLCGSCGSVGYTKEGSVINFCYMHQMELANGTHTGSAFDGTMYGAFMDKQVHQVQLTDKYCSVNVVAWLYAAILNGCAWFVKPNRTSVVSFNEWALANQFTEFVGTQSVDMLAVKTGVAIEQLLYAIQQLYTGFQGKQILGSTMLEDEFTPEDVNMQIMG 4ym2 A 2.1 BS01 BGC E 1 R240 E259 R55 E74 ? 0030246 remove_due_to_license_issue P56470 26077389 1 PTFNPPVPYFGRLQGGLTARRTIIIKGYVPPTGKSFAINFKVGSSGDIALHINPRMGNGTVVRNSLLNGSWGSEEKKITHNPFGPGQFFDLSIRCGLDRFKVYANGQHLFDFAHRLSAFQRVDTLEIQGDVTLSYVQI 4ym2 A 2.1 BS02 SGA E 1 H236 R240 N249 W256 E259 H51 R55 N64 W71 E74 ? 0030246 remove_due_to_license_issue P56470 26077389 2 PTFNPPVPYFGRLQGGLTARRTIIIKGYVPPTGKSFAINFKVGSSGDIALHINPRMGNGTVVRNSLLNGSWGSEEKKITHNPFGPGQFFDLSIRCGLDRFKVYANGQHLFDFAHRLSAFQRVDTLEIQGDVTLSYVQI 4ymb A 1.93 BS01 4E7 A 1 Y61 P88 T90 R95 V137 T142 E190 S193 Y216 Y58 P85 T87 R92 V134 T139 E187 S190 Y213 ? 0015276,0016020 Ki=0.62uM remove_due_to_license_issue P22756 26200741 301 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGCP 4ymg A 1.899 BS01 SAM A 1 K47 M48 S49 G73 Y75 S79 E98 Y99 P126 A127 D144 A145 N146 Y153 K46 M47 S48 G72 Y74 S78 E97 Y98 P125 A126 D143 A144 N145 Y152 D144 K147 D172 N173 D143 K146 D171 N172 ? 0008168,0008171,0008757,0032259 Kd=21uM remove_due_to_license_issue Q9HGR1 25979334 1001 LGSILPFNEETADRVSAYCEKNSHGIPDALVEHWEWTRTRFPDADKMSSRLQGSWMIFTARDRKPKRILEIGCYSGYSALAWYEGTRDTKAEIVTLEYSPKMIAASREAFKKYGVGDRVKLIEGPAENTLKTLEGEFDLIFVDANKDGYAGYVKTILDQGLLSANGIILCDNVFARGLTIGPDCAPWLNDHVRPYWNGCGQALDKFSAGLMEDPRIDVLLLPVFDGVTQIRWKD 4ymh A 1.876 BS01 SAH A 1 K47 M48 S49 G73 Y75 S79 E98 Y99 A127 D144 N146 K46 M47 S48 G72 Y74 S78 E97 Y98 A126 D143 N145 D144 K147 D172 N173 D143 K146 D171 N172 ? 0008168,0008171,0008757,0032259 Kd=3.2uM remove_due_to_license_issue Q9HGR1 25979334 1001 LGSILPFNEETADRVSAYCEKNSHGIPDALVEHWEWTRTRFPDADKMSSRLQGSWMIFTARDRKPKRILEIGCYSGYSALAWYEGTRDTKAEIVTLEYSPKMIAASREAFKKYGVGDRVKLIEGPAENTLKTLEGEFDLIFVDANKDGYAGYVKTILDQGLLSANGIILCDNVFARGLTIGPDCAPWLNDHVRPYWNGCGQALDKFSAGLMEDPRIDVLLLPVFDGVTQIRWKDGAQRA 4ymj A 2.0 BS01 4EJ A 1 G545 V552 A570 K572 F617 Y619 M620 L686 F698 G19 V26 A44 K46 F91 Y93 M94 L146 F158 D679 R683 N684 D697 S706 D139 R143 N144 D157 S163 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.1uM remove_due_to_license_issue IC50=100nM Q16288 26005534 901 GIHVQHIKRRDIVLKRELGEGAFGKVFLAECYNLSPTKDKMLVAVKALKDPTLAARKDFQREAELLTNLQHEHIVKFYGVCGDGDPLIMVFEYMKHGDLNKFLRAHGPGELGLSQMLHIASQIASGMVYLASQHFVHRDLATRNCLVGANLLVKIGDFGDVYSTDYYRHTMLPIRWMPPESIMYRKFTTESDVWSFGVILWEIFTYGKQPWFQLSNTEVIECITQGRVLERPRVCPKEVYDVMLGCWQREPQQRLNIKEIYKILHALGKAT 4yml A 1.75 BS01 4F0 A 1 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 I50 S76 A77 G78 F151 I152 E172 M173 E174 D197 F207 3.2.2.9 0003824,0005737,0005829,0008782,0008930,0009086,0009116,0009164,0016787,0019284,0019509,0042802,0042803,0046124,0110052 Ki=4.5nM remove_due_to_license_issue P0AF12 26260335 301 MKIGIIGAMEEEVTLLRDKIENRQTISLGGCEIYTGQLNGTEVALLKSGIGKVAAALGATLLLEHCKPDVIINTGSAGGLAPTLKVGDIVVSDEARYHDADVTAFGYEYGQLPGCPAGFKADDKLIAAAEACIAELNLNAVRGLIVSGDAFINGSVGLAKIRHNFPQAIAVEMEATAIAHVCHNFNVPFVVVRAISDVADQQSHLSFDEFLAVAAKQSSLMVESLVQKLAH 4ymq A 2.0 BS01 ZBD A 1 C320 M358 R364 M365 R367 V376 F378 F388 I397 I400 F401 S404 H479 C56 M94 R100 M101 R103 V112 F114 F124 I133 I136 F137 S140 H215 ? 0003677,0004879,0005634,0006355 Kd=1.6uM remove_due_to_license_issue Kd=1600nM, IC50=5700nM P51449 25840886 603 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGKILHRLLQDS 4ymx A 1.481 BS01 ARG A 1 S44 D46 F47 F88 A105 G106 M107 T108 R113 Q152 T155 T156 E193 S8 D10 F11 F52 A69 G70 M71 T72 R77 Q116 T119 T120 E157 ? 0015276,0016020 Kd=79nM remove_due_to_license_issue Q8RCC4 25848002 301 GVIVMGTSADFPPFEFHKVEGGKDEIVGFDIDIANAIAKKLGVKLEIKDMDFKGLIPALQAGRVDMVIAGMTPTAERKKSVDFSDLYYDSRQVVVVKNDSPISKFDDLKVKTIAVQIGTTSEEAAKKIPNVKLKQLNRVSDEFMDLQNGRCDAIVVEDTVAKAYLKEYKDMKILYMDEINNVENGSAVAVAKGNKSLLDVVNEVIKELKQSGEYDKLVDKWFKQ 4ynb A 2.0 BS01 4EH A 1 M11 I53 V79 A80 G81 F154 V155 V173 E174 M175 E176 D199 F209 M10 I52 V78 A79 G80 F153 V154 V172 E173 M174 E175 D198 F208 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=0.043nM remove_due_to_license_issue Q9ZMY2 26494017 301 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4ynd A 2.79 BS04 4GQ A 1 K145 I149 V179 N180 G183 F184 T185 A203 S239 Y240 S257 Y258 K143 I147 V177 N178 G181 F182 T183 A201 S237 Y238 S255 Y256 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 remove_due_to_license_issue IC50=2.8nM Q9NRG4 26101576 504 AEGLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLGFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEI 4yne A 2.0229 BS01 4EK A 1 F521 A542 F589 M592 N655 L657 G667 D668 F25 A44 F86 M89 N152 L154 G164 D165 D650 A652 R654 N655 D668 S677 L689 D147 A149 R151 N152 D165 S169 L177 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=3.0nM P04629 26005534 801 GSGIRVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPDKMLVAVKALKERQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSTDYYRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLD 4ynk A 2.3 BS02 YW2 A 1 Y143 A227 V230 S233 R270 S271 S274 W282 Y291 H301 L309 H393 L410 Y21 A46 V49 S52 R89 S90 S93 W101 Y110 H120 L128 H212 L229 ? 0003677,0004879,0006355 remove_due_to_license_issue P13053 26613420 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNE 4yo6 A 2.32 BS01 4GD A 1 M192 G193 V200 A211 Y262 Y264 M265 G268 S269 M30 G31 V38 A49 Y95 Y97 M98 G101 S102 D311 K313 A315 N316 D329 T351 D144 K146 A148 N149 D162 T181 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=2200nM Q9NWZ3 26101573 501 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4yo8 A 2.1 BS01 4EZ A 1 A80 G81 F154 V155 E174 M175 E176 D199 F209 A87 G88 F161 V162 E181 M182 E183 D206 F216 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=0.03nM remove_due_to_license_issue Q9ZMY2 26494017 301 HENLYFQGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4yo8 B 2.1 BS01 4EZ B 1 A80 F154 V155 E174 M175 E176 D199 A201 F209 A91 F165 V166 E185 M186 E187 D210 A212 F220 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=0.03nM remove_due_to_license_issue Q9ZMY2 26494017 301 HHHHHENLYFQGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 4yog A 2.0 BS01 4F5 A 1 M25 H41 A46 L49 F143 L144 C145 H166 M168 E169 D190 K191 Q192 M25 H41 A46 L49 F143 L144 C145 H166 M168 E169 D190 K191 Q192 H41 G146 C148 H41 G146 C148 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=1.8uM remove_due_to_license_issue P0C6W3 26190463 405 SGLVKMSAPSGAVENCIVQVTCGSMTLNGLWLDNTVWCPRHIMCPADQLTDPNYDALLISKTNHSFIVQKHIGAQANLRVVAHSMVGVLLKLTVDVANPSTPAYTFSTVKPGASFSVLACYNGKPTGVFTVNLRHNSTIKGSFLCGSCGSVGYTENGGVINFVYMHQMELSNGTHTGSSFDGVMYGAFEDKQTHQLQLTDKYCTINVVAWLYAAVLNGCKWFVKPTRVGIVTYNEWALSNQFTEFVGTQSIDMLAHRTGVSVEQMLAAIQSLHAGFQGKTILGQSTLEDEFTPDDVNMQVMGVVMQ 4yog B 2.0 BS01 4F5 B 1 M25 H41 A46 L49 F143 L144 C148 H166 M168 E169 D190 K191 Q192 M25 H41 A46 L49 F143 L144 C148 H166 M168 E169 D190 K191 Q192 H41 G146 C148 H41 G146 C148 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=1.8uM remove_due_to_license_issue P0C6W3 26190463 404 SGLVKMSAPSGAVENCIVQVTCGSMTLNGLWLDNTVWCPRHIMCPADQLTDPNYDALLISKTNHSFIVQKHIGAQANLRVVAHSMVGVLLKLTVDVANPSTPAYTFSTVKPGASFSVLACYNGKPTGVFTVNLRHNSTIKGSFLCGSCGSVGYTENGGVINFVYMHQMELSNGTHTGSSFDGVMYGAFEDKQTHQLQLTDKYCTINVVAWLYAAVLNGCKWFVKPTRVGIVTYNEWALSNQFTEFVGTQSIDMLAHRTGVSVEQMLAAIQSLHAGFQGKTILGQSTLEDEFTPDDVNMQVMGVVMQ 4yoi A 1.82 BS01 4F4 A 1 S24 M25 H41 A46 L49 Y54 F143 L144 C145 C148 H166 M168 E169 D190 K191 Q192 S24 M25 H41 A46 L49 Y54 F143 L144 C145 C148 H166 M168 E169 D190 K191 Q192 H41 G146 C148 H41 G146 C148 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=0.33uM remove_due_to_license_issue P0C6W3 26190463 401 SGLVKMSAPSGAVENCIVQVTCGSMTLNGLWLDNTVWCPRHIMCPADQLTDPNYDALLISKTNHSFIVQKHIGAQANLRVVAHSMVGVLLKLTVDVANPSTPAYTFSTVKPGASFSVLACYNGKPTGVFTVNLRHNSTIKGSFLCGSCGSVGYTENGGVINFVYMHQMELSNGTHTGSSFDGVMYGAFEDKQTHQLQLTDKYCTINVVAWLYAAVLNGCKWFVKPTRVGIVTYNEWALSNQFTEFVGTQSIDMLAHRTGVSVEQMLAAIQSLHAGFQGKTILGQSTLEDEFTPDDVNMQVMGVVMQ 4yoi B 1.82 BS01 4F4 B 1 M25 H41 A46 L49 F143 L144 C148 H166 M168 E169 D190 K191 Q192 M25 H41 A46 L49 F143 L144 C148 H166 M168 E169 D190 K191 Q192 H41 G146 C148 H41 G146 C148 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=0.33uM remove_due_to_license_issue P0C6W3 26190463 401 SGLVKMSAPSGAVENCIVQVTCGSMTLNGLWLDNTVWCPRHIMCPADQLTDPNYDALLISKTNHSFIVQKHIGAQANLRVVAHSMVGVLLKLTVDVANPSTPAYTFSTVKPGASFSVLACYNGKPTGVFTVNLRHNSTIKGSFLCGSCGSVGYTENGGVINFVYMHQMELSNGTHTGSSFDGVMYGAFEDKQTHQLQLTDKYCTINVVAWLYAAVLNGCKWFVKPTRVGIVTYNEWALSNQFTEFVGTQSIDMLAHRTGVSVEQMLAAIQSLHAGFQGKTILGQSTLEDEFTPDDVNMQVMGVVMQ 4yoj A 1.9 BS01 RFM A 1 S24 M25 H41 C44 L49 Y54 F143 L144 C145 C148 H166 M168 E169 D190 K191 S24 M25 H41 C44 L49 Y54 F143 L144 C145 C148 H166 M168 E169 D190 K191 H41 G146 C148 H41 G146 C148 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=0.41uM remove_due_to_license_issue P0C6W3 26190463 401 SGLVKMSAPSGAVENCIVQVTCGSMTLNGLWLDNTVWCPRHIMCPADQLTDPNYDALLISKTNHSFIVQKHIGAQANLRVVAHSMVGVLLKLTVDVANPSTPAYTFSTVKPGASFSVLACYNGKPTGVFTVNLRHNSTIKGSFLCGSCGSVGYTENGGVINFVYMHQMELSNGTHTGSSFDGVMYGAFEDKQTHQLQLTDKYCTINVVAWLYAAVLNGCKWFVKPTRVGIVTYNEWALSNQFTEFVGTQSIDMLAHRTGVSVEQMLAAIQSLHAGFQGKTILGQSTLEDEFTPDDVNMQVMGVVMQ 4yoj B 1.9 BS01 RFM B 1 S24 M25 H41 C44 L49 F143 L144 C145 C148 H166 M168 E169 D190 K191 Q192 S24 M25 H41 C44 L49 F143 L144 C145 C148 H166 M168 E169 D190 K191 Q192 H41 G146 C148 H41 G146 C148 2.1.1.56,2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 ic50=0.41uM remove_due_to_license_issue P0C6W3 26190463 401 SGLVKMSAPSGAVENCIVQVTCGSMTLNGLWLDNTVWCPRHIMCPADQLTDPNYDALLISKTNHSFIVQKHIGAQANLRVVAHSMVGVLLKLTVDVANPSTPAYTFSTVKPGASFSVLACYNGKPTGVFTVNLRHNSTIKGSFLCGSCGSVGYTENGGVINFVYMHQMELSNGTHTGSSFDGVMYGAFEDKQTHQLQLTDKYCTINVVAWLYAAVLNGCKWFVKPTRVGIVTYNEWALSNQFTEFVGTQSIDMLAHRTGVSVEQMLAAIQSLHAGFQGKTILGQSTLEDEFTPDDVNMQVMGVVMQ 4yp1 A 2.65 BS01 2BA A 1 G165 Y166 R237 Y239 P263 G13 Y14 R85 Y87 P111 ? 0002218,0032481 remove_due_to_license_issue Q3TBT3 26171638 401 NVAHGLAWSYYIGYLRLILPGLQARIRMFNQLHNNMLSGAGSRRLYILFPLDCGVPDNLSVVDPNIRFRDMLPQQNIDRAGIKNRVYSNSVYEILENGQPAGVCILEYATPLQTLFAMSQDAKAGFSREDRLEQAKLFCRTLEEILEDVPESRNNCRLIVYQEPFSLSQEVLRHIRQE 4yp1 B 2.65 BS01 2BA A 1 G165 Y166 R237 Y239 P263 G13 Y14 R85 Y87 P111 ? 0002218,0032481 remove_due_to_license_issue Q3TBT3 26171638 401 NVAHGLAWSYYIGYLRLILPGLQARIRMFNQLHNNMLSGAGSRRLYILFPLDCGVPDNLSVVDPNIRFRDMLPQQNIDRAGIKNRVYSNSVYEILENGQPAGVCILEYATPLQTLFAMSQDAKAGFSREDRLEQAKLFCRTLEEILEDVPESRNNCRLIVYQEPTDGNSFSLSQEVLRHIRQ 4yp8 A 2.641 BS01 4GF A 1 M192 G193 E194 V200 A211 Y262 Y264 M265 P266 G268 S269 L318 M29 G30 E31 V37 A48 Y94 Y96 M97 P98 G100 S101 L150 D311 K313 A315 N316 D329 T351 D143 K145 A147 N148 D161 T179 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=13nM Q9NWZ3 26101573 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4ypf A 2.2 BS02 4FS A 1 P125 W155 R156 E167 H168 P78 W108 R109 E115 H116 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 502 MVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYERRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGVTSDKFAPVCVIVDKMEREEVEAQLAVTVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRGFAVPLDRLV 4yps A 2.1012 BS01 4F6 A 1 L516 G517 V524 A542 F589 M592 R654 L657 L20 G21 V25 A40 F84 M87 R149 L152 D650 A652 R654 N655 D668 S677 L689 D145 A147 R149 N150 D163 S170 L179 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=75nM P04629 26005534 801 GSGIRVHHIKRRDIVLKWELGEGKVFLAECHNLLDKMLVAVKALSESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDMSRDIYSTDYYRVTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPV 4yqh A 2.308 BS03 4F7 A 1 S677 I692 Y693 P712 M713 E721 V722 G725 Q726 F729 S229 I244 Y245 P264 M265 E273 V274 G277 Q278 F281 3.1.4.17 0004114,0007165,0008081 ic50=0.009uM remove_due_to_license_issue IC50=<500nM Q9Y233 25863433 803 SICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4yqm A 2.38 BS01 4G9 A 1 C32 P33 R132 C28 P29 R128 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue Ki=440nM, IC50=130nM P78417 27703239 301 SARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 4yqu A 1.94 BS01 4GB A 1 C32 P33 F34 I131 R132 Y229 C29 P30 F31 I128 R129 Y223 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue P78417 27703239 301 ESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 4yqv A 2.06 BS01 4GG A 1 C32 P33 I131 R183 W222 F225 C28 P29 I127 R179 W218 F221 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue P78417 27703239 500 SARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 4yrc A 2.1 BS02 0P6 A 1 P125 C154 W155 R156 E167 H168 P79 C108 W109 R110 E119 H120 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 502 NMVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYEAITRRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGVTSDKFAPVCVIVDKMEKIPREEVEAQLAVLGLEPTVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRRGFAVPLDRLV 4yrc A 2.1 BS03 0P6 A 2 V383 G433 V335 G385 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 503 NMVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYEAITRRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGVTSDKFAPVCVIVDKMEKIPREEVEAQLAVLGLEPTVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRRGFAVPLDRLV 4yrd A 2.44 BS02 3IT A 1 F262 H288 F297 H337 M351 F234 H260 F269 H309 M323 ? 0046872 Kd=27uM remove_due_to_license_issue A0A0H3JP37 26471247 402 MNIVITGAKGFVGKNLKADLTSTTDHHIFEVHRQTKEEELESALLKADFIVHLAGVGSYLDHVLDILTRNTKKPAILLSSSIEQLLREYAEEYGNTVYIYRWPNLFGKWCKPNYNSVIATFCYKIARNEEIQVNDRNVELTLNYVDDIVAEIKRAIEGTPTIENGVPTVPNVFKVTLGEIVDLLYKFKQSRLDRTLPKLDNLFEKDLYSTYLSYLPSTDFSYPLLMNVDDRGSFTEFIKTPDRGQVSVNISKPGITKGNHWHHTKNEKFLVVSGKGVIRFRHVNDDEIIEYYVSGDKLEVVDIPVGYTHNIENLGDTDMVTIMWVNEMFDPNQPDTYFLEV 4yrg A 2.15 BS02 4HU A 1 P125 C154 W155 R156 R165 E167 H168 P78 C107 W108 R109 R113 E115 H116 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 502 MVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYERRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGTSDKFAPVCVIVDKMPREEVEAQLAVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRGFAVPLDRLV 4yrr A 2.3 BS02 691 A 1 C154 W155 R156 R165 E167 H168 C365 C107 W108 R109 R111 E113 H114 C309 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 502 MVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGVTSDKFAPVCVIVDKMIPREEVEAQLAVLGLEPTVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRGFAVPLDRLV 4yrs A 2.75 BS02 4JS A 1 R156 E167 H168 C365 R109 E118 H119 C316 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 502 MVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYEAITRRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGVTSDKFAPVCVIVDKMEKIPREEVEAQLAVLGLEPTVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRRGFAVPLDRLV 4yrt A 2.05 BS02 781 A 1 R156 R166 E167 H168 C365 V366 R109 R114 E115 H116 C313 V314 6.1.1.21 0004821,0005524,0005737,0006427,0016874 remove_due_to_license_issue Q4DA54 26249349 502 MVETEPVQGCRDFPPEAMRCRRHLFDVFHATAKTFGFEEYDAPVLESEELYIRKAGEEITEQMFNFITKGGHRVALRPEMTPSLARLLLGKGRSLLLPAKWYSIPQCWRYERRREHYQWNMDIVGVKSVSAEVELVCAACWAMRSLGLSSKDVGIKVNSRKVLQTVVEQAGVTSDKFAPVCVIVDKMEKIPREEVEAQLAVLGLEPTVVDAITTTLSLKSIDEIAQRVGEEHEAVKELRQFFEQVEAYGYGDWVLFDASVVRGLAYYTGIVFEGFDREGKFRALCGGGRYDNLLTTYGSPTPIPCAGFGFGDCVIVELLQEKRLLPDIPHVVDDVVIPFDESMRPHALAVLRRLRDAGRSADIILDKKKVVQAFNYADRVGAVRAVLVAPEEWERGEVQVKMLRGFAVPLDRLV 4ys7 A 2.502 BS02 4GK A 1 I692 Y693 F696 P712 M713 G725 Q726 F729 I245 Y246 F249 P265 M266 G278 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=0.001uM remove_due_to_license_issue IC50=<10nM Q9Y233 25863433 803 ASICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4ysl A 1.4618 BS02 GSH A 1 H149 D170 A180 R181 Y214 P260 V261 H149 D170 A180 R181 Y214 P260 V261 ? 0006749,0016787,0046872,0050313,0070813 Kd=1.6uM remove_due_to_license_issue A5VWI3 26082492 302 MIIGNNLHVDAFYDEATSTISYLVMDRETRQCALIDSVLDYDPKSGRTCSASADRLVERVNELNASVRWVLETHVHADHLSAAAYLKEKLGGHTAIGAHITQVQKVFGALFNAEPGFARDGSQFDVLLEDEEGFRIGNLQARALHTPGHTPACMSFMIEDAGEIAVFVGDTLFMPDYGTARCDFPGADARTLYRSIRRLLAFPDQTRLFMCHDYLPGGRDMQYVTTVAEQRASNIHIHQGIDEDSFVAMREARDKTLEMPVLILPSVQVNMRSGQLPPPEANGVSYLKIPLNKL 4ysl B 1.4618 BS02 GSH B 1 H149 D170 F173 A180 R181 Y214 P260 V261 H149 D170 F173 A180 R181 Y214 P260 V261 ? 0006749,0016787,0046872,0050313,0070813 Kd=1.6uM remove_due_to_license_issue A5VWI3 26082492 302 MIIGNNLHVDAFYDEATSTISYLVMDRETRQCALIDSVLDYDPKSGRTCSASADRLVERVNELNASVRWVLETHVHADHLSAAAYLKEKLGGHTAIGAHITQVQKVFGALFNAEPGFARDGSQFDVLLEDEEGFRIGNLQARALHTPGHTPACMSFMIEDAGEIAVFVGDTLFMPDYGTARCDFPGADARTLYRSIRRLLAFPDQTRLFMCHDYLPGGRDMQYVTTVAEQRASNIHIHQGIDEDSFVAMREARDKTLEMPVLILPSVQVNMRSGQLPPPEANGVSYLKIPLNKL 4yt6 H 2.07 BS01 4JY H 1 L41 C42 H57 T99 D102 D189 S190 C191 K192 S195 S214 W215 G216 G219 L25 C26 H41 T87 D90 D186 S187 C188 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=11nM remove_due_to_license_issue Ki=11nM P08709 25881820 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4yt7 H 2.3 BS01 4K1 H 1 C42 H57 K60A T99 D102 D189 S190 K192 S214 W215 G216 G219 C26 H41 K45 T87 D90 D186 S187 K189 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=1.7nM remove_due_to_license_issue Ki=1.7nM P08709 25881820 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4ytc A 2.16 BS01 4HW A 1 L855 V863 A880 M929 E930 Y931 L932 G935 R980 L983 L14 V20 A37 M85 E86 Y87 L88 G91 R136 L139 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue O60674 26230873 4000 TQFEERHLKFLQQLGKGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSARRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4ytf A 1.78 BS01 4HZ A 1 L855 G856 V863 A880 M929 Y931 L932 R980 N981 L983 G993 L14 G15 V20 A37 M84 Y86 L87 R135 N136 L138 G148 D976 A978 R980 N981 D994 S1016 D131 A133 R135 N136 D149 S171 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.007uM remove_due_to_license_issue O60674 26230873 4000 TQFEERHLKFLQQLGKGGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4yth A 2.04 BS01 467 A 1 L855 G856 V863 A880 M929 Y931 L932 N981 L983 D994 L14 G15 V22 A39 M88 Y90 L91 N140 L142 D153 D976 A978 R980 N981 D994 S1016 D135 A137 R139 N140 D153 S175 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.002uM remove_due_to_license_issue O60674 26230873 4000 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4yti A 2.52 BS01 VJK A 1 G856 V863 A880 E930 Y931 L932 R980 N981 L983 G993 D994 G15 V22 A39 E86 Y87 L88 R136 N137 L139 G149 D150 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>10000nM, Ki=13nM O60674 26230873 4000 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 4yur A 2.65 BS01 4J7 A 1 L18 G19 F23 R28 A39 E90 M91 C92 H93 G95 L143 L14 G15 F19 R24 A35 E86 M87 C88 H89 G91 L139 D136 T138 S140 N141 D154 D132 T134 S136 N137 D150 2.7.11.21 0004672,0005524,0006468 remove_due_to_license_issue O00444 25931445 1000 IGEKIEDFKVGNLLGKGSFAGVYRAESIHTGLEVAIKMIDKKAMYKAGMVQRVQNEVKIHCQLKHPSILELYNYFEDSNYVYLVLEMCHNGEMNRYLKNRVKPFSENEARHFMHQIITGMLYLHSHGILHRDLTLSNLLLTRNMNIKIADFGLESDVWSLGCMFYTLLIGRPPFTVKNTLNKVVLADYEMPSFLSIEAKDLIHQLLRRNPADRLSLSSVLDHPFMS 4yuw A 1.97 BS02 4JU A 1 Q64 T169 D171 Q201 Y237 Q64 T169 D171 Q201 Y237 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=1.7uM remove_due_to_license_issue Q4DA73 26327378 302 MPGSELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yux A 1.6 BS02 4JT A 1 I63 Q64 Y73 Q201 T236 I242 I62 Q63 Y72 Q200 T235 I241 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=180uM remove_due_to_license_issue Q4DA73 26327378 502 PGSELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yuy A 1.58 BS02 1SQ A 1 I63 Q64 Y73 Q201 I62 Q63 Y72 Q200 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=460uM remove_due_to_license_issue Q4DA73 26327378 502 PGSELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yuz A 1.97 BS02 4JV B 1 Q22 P238 C239 Q13 P217 C218 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 remove_due_to_license_issue Q4DA73 26327378 302 GWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yuz B 1.97 BS02 4JV B 1 E14 M24 S25 W53 T236 E10 M16 S17 W45 T218 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=9.1uM remove_due_to_license_issue Q4DA73 26327378 302 ELISGGWFREEPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 A 1.95 BS02 4JW B 1 E14 M24 L26 W53 P235 T236 E5 M11 L13 W40 P210 T211 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 remove_due_to_license_issue Q4DA73 26327378 302 GWFREEPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv0 B 1.95 BS02 4JW B 1 E14 Q22 A23 M24 Y237 P238 C239 E10 Q18 A19 M20 Y233 P234 C235 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=530uM remove_due_to_license_issue Q4DA73 26327378 302 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv1 A 1.85 BS02 4K2 B 1 M24 W53 T236 M15 W44 T215 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 remove_due_to_license_issue Q4DA73 26327378 302 GWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv1 B 1.85 BS02 4K2 B 1 E14 W19 Q22 M24 P238 C239 E10 W15 Q18 M20 P232 C233 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=830uM remove_due_to_license_issue Q4DA73 26327378 302 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv2 A 2.17 BS02 4K3 B 2 M24 W53 I63 T236 M20 W49 I59 T220 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 remove_due_to_license_issue Q4DA73 26327378 303 ELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv2 B 2.17 BS02 4K3 B 1 M24 S25 L26 W53 I63 M15 S16 L17 W44 I54 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 remove_due_to_license_issue Q4DA73 26327378 302 GWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 4yv5 A 1.9 BS01 SVR B 1 K7 L10 N17 K7 L10 N16 N28 G30 G32 H48 K49 Y52 Y73 D99 N27 G29 G31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0031640,0035821,0042130,0042742,0047498,0050482,0050832,0090729 Kd=0.6uM remove_due_to_license_issue Q9I834 26457430 207 SLFELGKMILQETGKNPAKSYGVYGCNCGVGGRGKPKDATDRCCYVHKCCYKKLTGCDPKKDRYSYSWKDKTIVCGENNSCLKELCECDKAVAICLRENLDTYNKKYRYNYLKPFCKKADPC 4yv5 A 1.9 BS02 SVR A 1 N114 K115 K116 Y119 Y121 L122 F126 N104 K105 K106 Y109 Y111 L112 F115 N28 G30 G32 H48 K49 Y52 Y73 D99 N27 G29 G31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0031640,0035821,0042130,0042742,0047498,0050482,0050832,0090729 Kd=0.6uM remove_due_to_license_issue Q9I834 26457430 205 SLFELGKMILQETGKNPAKSYGVYGCNCGVGGRGKPKDATDRCCYVHKCCYKKLTGCDPKKDRYSYSWKDKTIVCGENNSCLKELCECDKAVAICLRENLDTYNKKYRYNYLKPFCKKADPC 4yv5 B 1.9 BS01 SVR B 1 N114 K115 K116 Y119 Y121 L122 F126 N104 K105 K106 Y109 Y111 L112 F115 N28 G30 G32 H48 K49 Y52 Y73 D99 N27 G29 G31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0031640,0035821,0042130,0042742,0047498,0050482,0050832,0090729 Kd=0.6uM remove_due_to_license_issue Q9I834 26457430 207 SLFELGKMILQETGKNPAKSYGVYGCNCGVGGRGKPKDATDRCCYVHKCCYKKLTGCDPKKDRYSYSWKDKTIVCGENNSCLKELCECDKAVAICLRENLDTYNKKYRYNYLKPFCKKADPC 4yv5 B 1.9 BS02 SVR A 1 G6 K7 L10 N17 P18 G6 K7 L10 N16 P17 N28 G30 G32 H48 K49 Y52 Y73 D99 N27 G29 G31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0031640,0035821,0042130,0042742,0047498,0050482,0050832,0090729 Kd=0.6uM remove_due_to_license_issue Q9I834 26457430 205 SLFELGKMILQETGKNPAKSYGVYGCNCGVGGRGKPKDATDRCCYVHKCCYKKLTGCDPKKDRYSYSWKDKTIVCGENNSCLKELCECDKAVAICLRENLDTYNKKYRYNYLKPFCKKADPC 4yvc A 3.2 BS01 4KH A 1 I82 G83 R84 F87 V90 A103 K105 M153 M156 D216 I77 G78 R79 F82 V85 A98 K100 M143 M146 D206 D198 K200 N203 D216 T237 D188 K190 N193 D206 T227 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=1100nM Q13464 26039570 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLETFPIPKAFVGNQLPFVGFTYYSNRRY 4yve A 3.4 BS01 4KK A 1 G85 G88 E89 V90 A103 K105 L107 M153 M156 A215 D216 G80 G83 E84 V85 A98 K100 L102 M148 M151 A210 D211 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=100nM Q13464 26039570 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEETFPIPKAFVGNQLPFVGFTYYSNRRY 4yvz A 2.495 BS02 3AT B 1 L39 D75 G76 L94 G106 T107 R108 H109 T111 S127 R128 R130 L33 D69 G70 L88 G100 T101 R102 H103 T105 S121 R122 R124 2.7.7.85 0003677,0004016,0005524,0006281,0016779,0106408 ic50=3uM remove_due_to_license_issue Q9WY43 26014055 401 VPQELIEKIKLISPGTELRKALDDIINANFGALIFLVDDPKKYEDVIQGGFWLDTDFSAEKLYELSKMDGAIVLSEDITKIYYANVHLVPDPTIPTGETGTRHRTAERLAKQTGKVVIAVSRRRNIISLYYKNYKYVVNQVDFLISKVTQAISTLEKYKDNFNKLLSELEVLELENRVTLADVVRTLAKGFELLRIVEEIRPYIVELGEEGRLARMQLRELTEDVDDLLVLLIMDYSSEEVEEETAQNILQDFITRREPSPISISRVLGYDVQQAAQLDDVLVSARGYRLLKTVARIPLSIGYNVVRMFKTLDQISKASVEDLKKVEGIGEKRARAISESISSLKHRKT 4yvz B 2.495 BS01 3AT A 1 L39 D75 G76 L94 G106 T107 R108 H109 T111 S127 R128 R130 L33 D69 G70 L88 G100 T101 R102 H103 T105 S121 R122 R124 2.7.7.85 0003677,0004016,0005524,0006281,0016779,0106408 ic50=3uM remove_due_to_license_issue Q9WY43 26014055 403 VPQELIEKIKLISPGTELRKALDDIINANFGALIFLVDDPKKYEDVIQGGFWLDTDFSAEKLYELSKMDGAIVLSEDITKIYYANVHLVPDPTIPTGETGTRHRTAERLAKQTGKVVIAVSRRRNIISLYYKNYKYVVNQVDFLISKVTQAISTLEKYKDNFNKLLSELEVLELENRVTLADVVRTLAKGFELLRIVEEIRPYIVELGEEGRLARMQLRELTEDVDDLLVLLIMDYSSEEVEEETAQNILQDFITRREPSPISISRVLGYDVQQAAQLDDVLVSARGYRLLKTVARIPLSIGYNVVRMFKTLDQISKASVEDLKKVEGIGEKRARAISESISSLKHRKT 4yw2 A 2.0 BS01 SIA C 1 L128 F149 R151 E159 R161 R237 L46 F67 R69 E77 R79 R155 D315 E584 Y695 D233 E502 Y613 3.2.1.18 0004308,0005737,0005975,0006689,0009313,0016020,0016798,0043231 remove_due_to_license_issue A0A0H2UQE4 26370075 2 ETPVLEKNNVTLTGGGENVTKELKDKFTSGDFTVVIKYNQSSEKGLQALFGISNSKPGQQNSYVDVFLRDNGELGMEARDTSSNKNNLVSRPASVWGKYKQEAVTNTVAVVADSVKKTYSLYANGTKVVEKKVDNFLNIKDIKGIDYYMLGGVKRAGKTAFGFNGTLENIKFFNSALDEETVKKMTTNAVTGHLIYTANDTTGSNYFRIPVLYTFSNGRVFSSIDARYGGTHDFLNKINIATSYSDDNGKTWTKPKLTLAFDDFAPVPLEWPREVGGRDLQISGGATYIDSVIVEKKNKQVLMFADVMPAGVSFREATRKDSGYKQIDGNYYLKLRKQGDTDYNYTIRENGTVYDDRTNRPTEFSVDKNFGIKQNGNYLTVEQYSVSFENNKKTEYRNGTKVHMNIFYKDALFKVVPTNYIAYISSNDHGESWSAPTLLPPIMGLNRNAPYLGPGRGIIESSTGRILIPSYTGKESAFIYSDDNGASWKVKVVPLPSSWSAEAQFVELSPGVIQAYMRTNNGKIAYLTSKDAGTTWSAPEYLKFVSNPSYGTQLSIINYSQLIDGKKAVILSTPNSTNGRKHGQIWIGLINDDNTIDWRYHHDVDYSNYGYSYSTLTELPNHEIGLMFEKFDSWSRNELHMKNVVPYITFKIEDLKKNL 4yw6 A 1.4 BS02 G0P A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 26295304 902 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4yw7 C 1.82 BS01 4J0 C 1 Y36 P38 T39 H50 Q53 D100 T104 N107 Y36 P38 T39 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 Kd=130nM remove_due_to_license_issue Q05097 26295304 201 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4ywa A 1.192 BS02 4J9 A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 Kd=28nM remove_due_to_license_issue Q05097 26295304 202 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4ywa B 1.192 BS01 4J9 A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 26295304 202 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 4yx4 A 1.01 BS02 FB2 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1073.4nM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 26700575 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yx9 A 1.75 BS01 4HY A 1 P155 F164 L174 V175 G270 G271 M272 F275 P131 F140 L150 V151 G246 G247 M248 F251 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? Ki=4.5uM remove_due_to_license_issue A0A0M3KL26 26136396 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSR 4yx9 B 1.75 BS01 4HY B 1 F164 L174 V175 H207 G270 M272 F275 F140 L150 V151 H183 G246 M248 F251 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? Ki=4.5uM remove_due_to_license_issue A0A0M3KL26 26136396 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSR 4yxd B 3.0 BS04 FTN C 1 P169 W173 H216 P161 W165 H208 1.3.5.1 0005515,0005739,0005743,0006099,0006121,0008177,0009055,0009060,0016491,0022904,0031966,0045273,0046872,0048039,0051536,0051537,0051538,0051539 remove_due_to_license_issue Q007T0 26198225 302 PRIKKFAIYRWDPDKTGDKPHMQTYEIDLNNCGPMVLDALIKIKNEIDSTLTFRRSCREGICGSCAMNINGGNTLACTRRIDTNLDKVSKIYPLPHMYVIKDLVPDLSNFYAQYKSIEPYLKKKDESQEGKQQYLQSIEEREKLDGLYECILCACCSTSCPSYWWNGDKYLGPAVLMQAYRWMIDSRDDFTEERLAKLQDPFSLYRCHTIMNCTGTCPKGLNPGKAIAEIKKMMATYKE 4yxd C 3.0 BS02 FTN C 1 I30 W35 M39 S42 R46 I25 W30 M34 S37 R41 ? 0005515,0005739,0005743,0006099,0006121,0009055,0016020,0020037,0045273,0046872 remove_due_to_license_issue D0VWV4 26198225 302 TTAKEEMERFWNKNLGSNRPLSPHITIYRWSLPMAMSICHRGTGIALSAGVSLFGLSALLLPGNFESHLELVKSLCLGPTLIYTAKFGIVFPLMYHTWNGIRHLIWDLGKGLTIPQLTQSGVVVLILTVLSSVGLAAM 4yxd D 3.0 BS02 FTN C 1 D90 Y91 D56 Y57 ? 0005515,0005739,0005740,0005743,0006099,0006121,0016020,0020037,0045273,0046872,0048039 remove_due_to_license_issue A5GZW8 26198225 302 SSKAASLHWTGERVVSVLLLGLLPAAYLNPCSAMDYSLAAALTLHGHWGIGQVVTDYVRGDALQKVAKAGLLALSAFTFAGLCYFNYHDVGICKAVAMLWKL 4yxi A 0.96 BS02 4J8 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=318.8nM remove_due_to_license_issue Ki=320nM, Kd=0.060000nM, IC50=580nM P00918 26700575 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yxi A 0.96 BS03 4J8 A 2 R182 G183 R178 G179 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=318.8nM remove_due_to_license_issue Ki=320nM, Kd=0.060000nM, IC50=580nM P00918 26700575 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yxo A 1.06 BS02 4JC A 1 D180 R182 D176 R178 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=91.4nM remove_due_to_license_issue Ki=0.05nM, Kd=125400nM P00918 26700575 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yxo A 1.06 BS03 4JC A 2 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=91.4nM remove_due_to_license_issue Ki=0.05nM, Kd=125400nM P00918 26700575 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yxu A 1.08 BS02 4JE A 1 W5 H15 W16 D19 W3 H13 W14 D17 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=57.4nM remove_due_to_license_issue Ki=0.03nM, Kd=57800nM P00918 26700575 304 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yxu A 1.08 BS03 4JE A 2 H94 H119 L198 T199 T200 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=57.4nM remove_due_to_license_issue Ki=0.03nM, Kd=57800nM P00918 26700575 305 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yyl A 1.905 BS01 4KN A 1 Y24 H41 E80 R84 D108 E119 K134 Y29 H46 E65 R69 D93 E104 K119 3.1.-.- 0003723,0039694 ic50=9.7uM remove_due_to_license_issue IC50=9700nM P03433 26252962 301 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 4yyl A 1.905 BS02 4KN A 2 T20 K34 A37 I38 H41 G121 V122 Y130 T25 K39 A42 I43 H46 G106 V107 Y115 3.1.-.- 0003723,0039694 ic50=9.7uM remove_due_to_license_issue IC50=9700nM P03433 26252962 302 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 4yyl A 1.905 BS03 4KN A 3 E31 K34 A37 F191 S194 E195 E36 K39 A42 F176 S179 E180 3.1.-.- 0003723,0039694 ic50=9.7uM remove_due_to_license_issue IC50=9700nM P03433 26252962 303 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 4yyt A 1.07 BS01 S2O A 1 W5 W16 D19 W2 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=418.3nM remove_due_to_license_issue Ki=125nM, IC50=3000nM, Kd=392000nM P00918 26700575 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yyt A 1.07 BS02 S2O A 2 D110 K111 K112 D107 K108 K109 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=418.3nM remove_due_to_license_issue Ki=125nM, IC50=3000nM, Kd=392000nM P00918 26700575 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yyt A 1.07 BS03 S2O A 3 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=418.3nM remove_due_to_license_issue Ki=125nM, IC50=3000nM, Kd=392000nM P00918 26700575 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yyt A 1.07 BS04 S2O A 4 N67 E69 I91 Q92 N64 E66 I88 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=418.3nM remove_due_to_license_issue Ki=125nM, IC50=3000nM, Kd=392000nM P00918 26700575 306 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4yz9 A 2.463 BS01 4K7 A 1 A581 K599 C605 A609 E612 V613 I626 L679 H686 D711 A20 K38 C44 A48 E51 V52 I65 L118 H125 D150 D688 K690 N693 D711 T734 D127 K129 N132 D150 T156 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 Ki=200nM remove_due_to_license_issue O75460 26438213 1001 SVVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCGTEGWIAPEMLENPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPAEVRETLGSLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFHE 4yzc A 2.494 BS01 STU A 1 L577 V586 A597 K599 I642 L644 C645 H692 L695 L16 V25 A36 K38 I75 L77 C78 H117 L120 D688 K690 N693 D711 T734 D113 K115 N118 D136 T158 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 ic50=3nM remove_due_to_license_issue O75460 26438213 1001 SVVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPDREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCKKLAVRHSFSRRSGVPGTEGWIAPEMLSCKENPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPAEVRETLGSLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFH 4yzm A 3.0 BS01 4K4 A 1 I1032 G1035 K1055 M1105 E1106 L1107 V1108 P1109 G1111 L1161 I16 G19 K39 M83 E84 L85 V86 P87 G89 L139 D1154 R1156 P1158 N1159 D1177 N1194 D132 R134 P136 N137 D155 N164 2.7.11.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q6XHB2 25897865 1301 RLPTLADNEIEYEKQIGKGGFGLVHKGRLVKDKSVVAIKSLILTEMIEKFQEFQREVFIMSNLNHPNIVKLYGLMHNPPRMVMELVPCGDLYHRLLDKAHPIKWSVKLRLMLDIALGIEYMQNQNPPIVHRDLRSPNILLQSLDENAPVCAKVADFGLSQQLGNFQWMAPETIGAEEYTEKADTYSFAMILYTILTGEGPFDEYSYGKIKFINMIREEGLRPTIPEDCPPRLRNVIELCWSGDPKKRPHFSYIVKELSEL 4yzn A 1.55 BS01 4K5 A 1 I1032 V1108 P1109 G1111 L1161 I14 V85 P86 G88 L138 D1154 R1156 P1158 N1159 D1177 N1194 D131 R133 P135 N136 D154 N171 2.7.11.1 0004672,0004713,0005524,0006468 ic50=15.4uM remove_due_to_license_issue Q6XHB2 25897865 1301 PTLADNEIEYEKQIGKGGFGLVHKGRLVKDKSVVAIKSLILETEMIEKFQEFQREVFIMSNLNHPNIVKLYGLMHNPPRMVMELVPCGDLYHRLLDKAHPIKWSVKLRLMLDIALGIEYMQNQNPPIVHRDLRSPNILLQSLDENAPVCAKVADFGLSQQSVHSVSGLLGNFQWMAPETIGAEEESYTEKADTYSFAMILYTILTGEGPFDEYSYGKIKFINMIREEGLRPTIPEDCPPRLRNVIELCWSGDPKKRPHFSYIVKELSEL 4yzu A 1.41 BS01 4K6 A 1 Y99 F174 S190 C191 Q192 W215 G216 E217 C220 Y86 F162 S180 C181 Q182 W205 G206 E207 C209 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 Ki=9uM remove_due_to_license_issue Ki=9000nM P00740 25937013 301 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGASALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKLT 4z07 A 2.5 BS01 PCG A 1 V165 L172 F181 G182 E183 L184 A185 R192 T193 A194 V74 L81 F90 G91 E92 L93 A94 R101 T102 A103 2.7.11.12 0001932,0004692,0005524,0005952,0008603 remove_due_to_license_issue Q13976 27066748 401 SHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMRTGLIKHTEYMEFLKSVPTFQSLPEEILSKLADVLEETHYENGEYIIRQGARGDTFFIISKGTVNVTREDSPSEDPVFLRTLGKGDWFGEKALQGEDVRTANVIAAEAVTCLVIDRDSFKHLIGGLDDVSNKAY 4z07 A 2.5 BS02 PCG A 2 V283 L296 R297 F305 G306 E307 K308 A309 R316 T317 A318 Y351 V192 L205 R206 F214 G215 E216 K217 A218 R225 T226 A227 Y260 2.7.11.12 0001932,0004692,0005524,0005952,0008603 remove_due_to_license_issue Q13976 27066748 402 SHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMRTGLIKHTEYMEFLKSVPTFQSLPEEILSKLADVLEETHYENGEYIIRQGARGDTFFIISKGTVNVTREDSPSEDPVFLRTLGKGDWFGEKALQGEDVRTANVIAAEAVTCLVIDRDSFKHLIGGLDDVSNKAY 4z07 C 2.5 BS01 PCG C 1 V165 L172 F181 G182 E183 L184 A185 R192 T193 A194 V72 L79 F88 G89 E90 L91 A92 R99 T100 A101 2.7.11.12 0001932,0004692,0005524,0005952,0008603 remove_due_to_license_issue Q13976 27066748 401 VTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMRTGLIKHTEYMEFLKSVPTFQSLPEEILSKLADVLEETHYENGEYIIRQGARGDTFFIISKGTVNVTREDSPSEDPVFLRTLGKGDWFGEKALQGEDVRTANVIAAEAVTCLVIDRDSFKHLIGGLDDVSNKAY 4z07 C 2.5 BS02 PCG C 2 V283 L296 R297 F305 G306 E307 K308 A309 R316 T317 A318 Y351 V190 L203 R204 F212 G213 E214 K215 A216 R223 T224 A225 Y258 2.7.11.12 0001932,0004692,0005524,0005952,0008603 remove_due_to_license_issue Q13976 27066748 402 VTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMRTGLIKHTEYMEFLKSVPTFQSLPEEILSKLADVLEETHYENGEYIIRQGARGDTFFIISKGTVNVTREDSPSEDPVFLRTLGKGDWFGEKALQGEDVRTANVIAAEAVTCLVIDRDSFKHLIGGLDDVSNKAY 4z0k A 1.41 BS01 4LN A 1 Y99 F174 S190 C191 Q192 W215 G216 E219 C220 Y86 F162 S180 C181 Q182 W205 G206 E208 C209 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 Ki=0.462uM remove_due_to_license_issue IC50=507nM P00740 25937013 301 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGASALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKL 4z0q A 1.45 BS02 4K9 A 1 H94 H119 F131 L198 T199 T200 P201 P202 H92 H117 F128 L195 T196 T197 P198 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=6.8nM remove_due_to_license_issue Ki=6.8nM P00918 26276436 1002 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4z16 A 2.9 BS01 4LH A 1 L828 A853 M902 Y904 L905 P906 G908 C909 R911 R953 L956 L15 A40 M84 Y86 L87 P88 G90 C91 R93 R135 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=4.8nM P52333 26258521 2000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYELRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVRPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMALCRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 4z1e A 2.01 BS02 DF5 A 1 H94 H119 F130 L197 T198 T199 P201 H93 H118 F129 L196 T197 T198 P200 H64 H94 H96 E106 H119 T198 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.7nM remove_due_to_license_issue P00918 26276436 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4z1j A 1.27 BS02 4KC A 1 Q92 H94 H119 F130 L197 T198 T199 Q90 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.7nM remove_due_to_license_issue Ki=7.7nM P00918 26276436 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4z1k A 1.35 BS02 4KB A 1 Q92 H94 H119 F130 L197 T198 T199 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=4.7nM remove_due_to_license_issue Ki=4.7nM P00918 26276436 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4z1n A 1.47 BS02 4KD A 1 Q92 H94 H119 F130 L197 T198 T199 Q90 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5.89nM remove_due_to_license_issue Ki=5.9nM P00918 26276436 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4z1q A 1.399 BS01 558 A 1 W81 P82 L92 Y139 N140 I146 W39 P40 L50 Y97 N98 I104 ? ic50=0.015uM remove_due_to_license_issue O60885 26985289 201 TNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4z1s A 1.06 BS01 559 A 1 W81 P82 L92 I146 W41 P42 L52 I106 ? ic50=0.79uM remove_due_to_license_issue O60885 26985289 201 GSTNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 4z22 A 2.62 BS01 4KG A 1 D34 W41 Y77 Y192 D214 F294 I300 D34 W41 Y77 Y192 D214 F294 I300 D34 S37 N39 W41 Y77 D214 T217 D34 S37 N39 W41 Y77 D214 T217 3.4.23.39 0004190,0006508 remove_due_to_license_issue IC50=340nM P46925 26670264 401 SSNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNISLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNHSVGIALAKKNL 4z2b A 1.8 BS01 4LC A 1 Y307 E351 W459 P461 N498 F556 Y147 E191 W299 P301 N338 F396 3.1.13.4,3.1.4.- 0003824 Ki=17.5nM remove_due_to_license_issue Q6L8Q7 26055709 705 PPAFTELQLPRYIMAGFPVCPKLSLEFGDPASSLFRWYKEAKPGAAEPEVGVPSSLSPSSPSSSWTETDVEERVYTPSNADIGLRLKLHCTPGDGQRFGHSRELESVCVVEAGPGTCTFDHRHLYTKKVTEDALIRTVSYNILADTYAQTEFSRTVLYPYCAPYALELDYRQNLIQKELTGYNADVICLQEVDRAVFSDSLVPALEAFGLEGVFRIKQHEGLATFYRKSKFSLLSQHDISFYEALESDPLHKELLEKLVLYPSAQEKVLQRSSVLQVSVLQSTKDSSKRICVANTHLYWHPKGGYIRLIQMAVALAHIRHVSCDLYPGIPVIFCGDFNSTPSTGMYHFVINGSIPEDHEDWASNGEEERCNMSLTHFFKLKSACGEPAYTNYVGGFHGCLDYIFIDLNALEVEQVIPLPSHEEVTTHQALPSVSHPSDHIALVCDLKWK 4z2g A 2.6 BS01 M6V A 1 Y10 F12 Y98 D142 E144 M212 Y214 D215 Y292 K335 W403 Y9 F11 Y97 D141 E143 M211 Y213 D214 Y291 K334 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 26030312 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2g A 2.6 BS02 M6V A 2 D102 F190 F191 W220 E221 F239 D101 F189 F190 W219 E220 F238 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 26030312 502 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2h A 2.35 BS01 M6A A 1 Y10 F12 F51 D142 E144 M212 Y214 D215 Y292 W403 Y9 F11 F50 D141 E143 M211 Y213 D214 Y291 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 ic50=8.3uM remove_due_to_license_issue P11797 26030312 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2i A 2.0 BS01 M6B A 1 Y10 F12 F51 Y98 D142 E144 M212 Y214 Y292 I339 W403 Y9 F11 F50 Y97 D141 E143 M211 Y213 Y291 I338 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 ic50=0.036uM remove_due_to_license_issue P11797 26030312 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2i A 2.0 BS02 M6B A 2 W97 F190 F191 L216 W220 E221 W96 F189 F190 L215 W219 E220 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 ic50=0.036uM remove_due_to_license_issue P11797 26030312 502 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2j A 2.6 BS01 M6G A 1 Y10 F12 Y98 D142 E144 M212 Y214 D215 Y292 W403 Y9 F11 Y97 D141 E143 M211 Y213 D214 Y291 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 26030312 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2j A 2.6 BS02 M6G A 2 W97 D102 F190 F191 W220 E221 W96 D101 F189 F190 W219 E220 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 26030312 502 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2k A 2.3 BS01 M6E A 1 Y10 D142 E144 M212 Y214 D215 W220 D316 Y9 D141 E143 M211 Y213 D214 W219 D315 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 26030312 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z2l A 2.3 BS01 M6F A 1 Y10 F12 F51 D142 E144 M212 Y214 D215 Y292 D316 W403 Y9 F11 F50 D141 E143 M211 Y213 D214 Y291 D315 W402 D140 D142 E144 Y214 D139 D141 E143 Y213 3.2.1.14 0004553,0005576,0005975,0008061,0030246 remove_due_to_license_issue P11797 26030312 501 STRKAVIGYYFIPTNQINNYTETDTSVVPFPVSNITPAKAKQLTHINFSFLDINSNLECAWDPATNDAKARDVVNRLTALKAHNPSLRIMFSIGGWYYSNDLGVSHANYVNAVKTPAARTKFAQSCVRIMKDYGFDGVDIDWEYPQAAEVDGFIAALQEIRTLLNQQTIADGRQALPYQLTIAGAGGAFFLSRYYSKLAQIVAPLDYINLMTYDLAGPWEKITNHQAALFGDAAGPTFYNALREANLGWSWEELTRAFPSPFSLTVDAAVQQHLMMEGVPSAKIVMGVPFYGRAFKGVSGGNGGQYSSHSTPGEDPYPNADYWLVGCDECVRDKDPRIASYRQLEQMLQGNYGYQRLWNDKTKTPYLYHAQNGLFVTYDDAESFKYKAKYIKQQQLGGVMFWHLGQDNRNGDLLAALDRYFNAADYDDSQLDMGTGLRYTGVGPGNLPIMTAPAYVPGTTYAQGALVSYQGYVWQTKWGYITSAPGSDSAWLKVGRLA 4z31 A 2.5 BS01 rna C 0 S312 Q315 S316 D319 S208 Q211 S212 D215 2.3.2.27 remove_due_to_license_issue Q9HBD1 26489670 2 ~ 15 NKHYEVAKKCVEDLALYLKPALSRPMQRKLVTLVNCQLVEEEGRVRAMRAARSLGERTVTELILQHQNPQQLSANLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRSYEALRREHDAQIVHIAMEAGLRISPEQWSSLLYGDLAHKSHMQSIIDKLQSPESFAKSVQELTIVLQRTGDPANLNRLRPHLELLANIDPNPDAVSPTWEQLENAMVAVKTVVHGLVDFIQNYSR 4z31 A 2.5 BS02 rna D 0 R128 P129 R132 K133 R24 P25 R28 K29 2.3.2.27 remove_due_to_license_issue Q9HBD1 26489670 1 ~ 14 NKHYEVAKKCVEDLALYLKPALSRPMQRKLVTLVNCQLVEEEGRVRAMRAARSLGERTVTELILQHQNPQQLSANLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRSYEALRREHDAQIVHIAMEAGLRISPEQWSSLLYGDLAHKSHMQSIIDKLQSPESFAKSVQELTIVLQRTGDPANLNRLRPHLELLANIDPNPDAVSPTWEQLENAMVAVKTVVHGLVDFIQNYSR 4z31 A 2.5 BS03 rna F 0 R185 R187 R216 K217 S235 T237 Q244 Y247 R248 E259 D260 S261 S262 R81 R83 R112 K113 S131 T133 Q140 Y143 R144 E155 D156 S157 S158 2.3.2.27 remove_due_to_license_issue Q9HBD1 26489670 1 ~ 15 NKHYEVAKKCVEDLALYLKPALSRPMQRKLVTLVNCQLVEEEGRVRAMRAARSLGERTVTELILQHQNPQQLSANLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRSYEALRREHDAQIVHIAMEAGLRISPEQWSSLLYGDLAHKSHMQSIIDKLQSPESFAKSVQELTIVLQRTGDPANLNRLRPHLELLANIDPNPDAVSPTWEQLENAMVAVKTVVHGLVDFIQNYSR 4z31 B 2.5 BS01 rna C 0 S312 Q315 S316 D319 S211 Q214 S215 D218 2.3.2.27 remove_due_to_license_issue Q9HBD1 26489670 2 ~ 15 NLGENKHYEVAKKCVEDLALYLKALSRPMQRKLVTLVNCQLVEEEGRVRAMRAARSLGERTVTELILQHQNPQQLSANLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRSYEALRREHDAQIVHIAMEAGLRISPEQWSSLLYGDLAHKSHMQSIIDKLQSPESFAKSVQELTIVLQRTGDPANLNRLRPHLELLANIDPNPDAVSPTWEQLENAMVAVKTVVHGLVDFIQNYS 4z31 B 2.5 BS02 rna D 0 K133 R153 S157 R161 K32 R52 S56 R60 2.3.2.27 remove_due_to_license_issue Q9HBD1 26489670 1 ~ 14 NLGENKHYEVAKKCVEDLALYLKALSRPMQRKLVTLVNCQLVEEEGRVRAMRAARSLGERTVTELILQHQNPQQLSANLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRSYEALRREHDAQIVHIAMEAGLRISPEQWSSLLYGDLAHKSHMQSIIDKLQSPESFAKSVQELTIVLQRTGDPANLNRLRPHLELLANIDPNPDAVSPTWEQLENAMVAVKTVVHGLVDFIQNYS 4z31 B 2.5 BS03 rna E 0 R185 R216 S235 T237 Q244 Y247 R248 D260 S261 S262 R84 R115 S134 T136 Q143 Y146 R147 D159 S160 S161 2.3.2.27 remove_due_to_license_issue Q9HBD1 26489670 1 ~ 15 NLGENKHYEVAKKCVEDLALYLKALSRPMQRKLVTLVNCQLVEEEGRVRAMRAARSLGERTVTELILQHQNPQQLSANLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRSYEALRREHDAQIVHIAMEAGLRISPEQWSSLLYGDLAHKSHMQSIIDKLQSPESFAKSVQELTIVLQRTGDPANLNRLRPHLELLANIDPNPDAVSPTWEQLENAMVAVKTVVHGLVDFIQNYS 4z3c C 1.57 BS01 dna A 0 K53 R54 H81 I83 K88 L92 K1 R2 H29 I31 K36 L40 1.14.11.80 0003677,0008270 remove_due_to_license_issue O43151 29276034 1 ~ 12 KRKRCGTCEPCRRLENCGACTSCTNRRTHQICKLRKCEVLKKKV 4z3c C 1.57 BS02 dna B 0 K53 T73 N77 T80 H81 Q82 K1 T21 N25 T28 H29 Q30 1.14.11.80 0003677,0008270 remove_due_to_license_issue O43151 29276034 1 ~ 12 KRKRCGTCEPCRRLENCGACTSCTNRRTHQICKLRKCEVLKKKV 4z3v A 1.6 BS01 4L6 A 1 L408 T410 G411 F413 V416 A428 M477 L528 D539 L20 T22 G23 F25 V28 A40 M89 L140 D151 D521 A523 R525 N526 D539 F559 D133 A135 R137 N138 D151 F171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4nM remove_due_to_license_issue EC50=28nM, IC50=5.6nM Q06187 26087137 705 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 4z4c A 2.303 BS01 rna B 0 P67 R68 R97 G178 R179 F294 Y311 H336 T337 Y338 L522 G524 K525 T526 Y529 K533 Q545 C546 Q548 N551 T559 N562 K566 K570 T599 H600 P601 P602 A603 R635 E637 S672 Q675 K709 R710 H753 I756 Q757 S760 R761 Y790 R792 C793 S798 Y804 P46 R47 R76 G151 R152 F261 Y269 H294 T295 Y296 L480 G482 K483 T484 Y487 K491 Q503 C504 Q506 N509 T517 N520 K524 K528 T557 H558 P559 P560 A561 R593 E595 S630 Q633 K667 R668 H711 I714 Q715 S718 R719 Y748 R750 C751 S756 Y762 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4c A 2.303 BS02 rna D 0 D358 S362 I365 K525 T556 P557 Q558 K726 F811 Y815 D316 S320 I323 K483 T514 P515 Q516 K684 F769 Y773 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 9 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4d A 1.6 BS01 rna B 0 P67 R68 V70 R97 V177 G178 R179 R277 F294 Y311 H316 H336 T337 Y338 I365 L522 G524 K525 T526 Y529 K533 Q545 C546 V547 Q548 N551 T559 N562 L563 K566 K570 H600 P601 P602 A603 R635 E637 S672 Q675 K709 R710 H753 I756 Q757 S760 R761 Y790 R792 C793 R795 S798 Y804 P46 R47 V49 R76 V150 G151 R152 R244 F261 Y269 H274 H294 T295 Y296 I323 L480 G482 K483 T484 Y487 K491 Q503 C504 V505 Q506 N509 T517 N520 L521 K524 K528 H558 P559 P560 A561 R593 E595 S630 Q633 K667 R668 H711 I714 Q715 S718 R719 Y748 R750 C751 R753 S756 Y762 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPECTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4d A 1.6 BS02 rna D 0 D358 T361 S362 K525 Q558 K726 Q757 F811 Y815 D316 T319 S320 K483 Q516 K684 Q715 F769 Y773 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 9 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPECTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4e A 1.8 BS01 rna B 0 P67 R68 R97 G178 R179 F294 L296 Y311 H336 T337 Y338 L522 G524 K525 T526 Y529 K533 Q545 C546 Q548 N551 T559 N562 L563 K566 K570 T599 H600 P601 P602 A603 R635 E637 S672 Q675 K709 R710 H753 I756 Q757 S760 R761 Y790 R792 C793 S798 Y804 P46 R47 R76 G152 R153 F260 L262 Y268 H293 T294 Y295 L479 G481 K482 T483 Y486 K490 Q502 C503 Q505 N508 T516 N519 L520 K523 K527 T556 H557 P558 P559 A560 R592 E594 S629 Q632 K666 R667 H710 I713 Q714 S717 R718 Y747 R749 C750 S755 Y761 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPRIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4e A 1.8 BS02 rna D 0 D358 T361 S362 I365 K525 Q558 K726 Q757 F811 Y815 D315 T318 S319 I322 K482 Q515 K683 Q714 F768 Y772 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 9 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPRIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4f A 2.8 BS01 rna B 0 R68 R97 G178 R179 F294 Y311 H336 T337 I365 L522 G524 T526 Y529 K533 Q545 C546 Q548 N551 T559 N562 K566 K570 H600 A603 R635 E637 S672 Q675 K709 R710 H753 Q757 S760 R761 Y790 R792 C793 R795 S798 Y804 R45 R74 G149 R150 F259 Y267 H292 T293 I321 L478 G480 T482 Y485 K489 Q501 C502 Q504 N507 T515 N518 K522 K526 H556 A559 R591 E593 S628 Q631 K665 R666 H709 Q713 S716 R717 Y746 R748 C749 R751 S754 Y760 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPECTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4f A 2.8 BS02 rna D 0 D358 T361 S362 I365 R438 K525 Q558 S561 K726 F811 Y815 D314 T317 S318 I321 R394 K481 Q514 S517 K682 F767 Y771 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 10 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPECTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4g A 2.7 BS01 rna B 0 P67 R68 R97 G178 R179 F294 Y311 H336 Y338 L522 G524 T526 Y529 K533 Q545 C546 Q548 N551 T559 N562 K566 K570 H600 P601 P602 A603 R635 E637 S672 Q675 K709 R710 H753 Q757 S760 R761 Y790 R792 S798 Y804 P46 R47 R74 G149 R150 F259 Y265 H290 Y292 L476 G478 T480 Y483 K487 Q499 C500 Q502 N505 T513 N516 K520 K524 H554 P555 P556 A557 R589 E591 S626 Q629 K663 R664 H707 Q711 S714 R715 Y744 R746 S752 Y758 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4g A 2.7 BS02 rna D 0 D358 S362 K525 Q558 K726 F811 Y815 D312 S316 K479 Q512 K680 F765 Y769 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 9 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4h A 2.504 BS01 rna B 0 P67 R68 R97 G178 R179 F294 Y311 H336 Y338 L522 G524 T526 Y529 K533 Q545 C546 Q548 N551 T559 N562 K566 K570 T599 H600 P601 P602 A603 R635 E637 S672 Q675 K709 R710 H753 Q757 S760 R761 Y790 R792 C793 R795 S798 Y804 P46 R47 R75 G150 R151 F260 Y268 H293 Y295 L479 G481 T483 Y486 K490 Q502 C503 Q505 N508 T516 N519 K523 K527 T556 H557 P558 P559 A560 R592 E594 S629 Q632 K666 R667 H710 Q714 S717 R718 Y747 R749 C750 R752 S755 Y761 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDTGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4h A 2.504 BS02 rna D 0 D358 T361 S362 K525 Q558 F811 Y815 D315 T318 S319 K482 Q515 F768 Y772 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 8 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGRKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIKRKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDTGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4i A 2.801 BS01 rna B 0 P67 R68 R97 G178 R179 Y311 H336 T337 Y338 I365 L522 G524 T526 Y529 K533 Q545 C546 Q548 N551 T559 N562 K566 T599 H600 P601 P602 A603 R635 E637 S672 Q675 K709 R710 H753 Q757 S760 R761 Y790 R792 C793 S798 Y804 P46 R47 R74 G149 R150 Y266 H291 T292 Y293 I320 L477 G479 T481 Y484 K488 Q500 C501 Q503 N506 T514 N517 K521 T554 H555 P556 P557 A558 R590 E592 S627 Q630 K664 R665 H708 Q712 S715 R716 Y745 R747 C748 S753 Y759 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIRKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDTGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z4i A 2.801 BS02 rna D 0 D358 T361 S362 K525 Q558 K726 Q757 F811 Y815 D313 T316 S317 K480 Q513 K681 Q712 F766 Y770 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 26359634 1 ~ 8 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGKPVFDGRKNLYTAMPLPIGRDKVELEVTLPIFKVSIKWVSCVSLQALHDALSGRLPSVPFETIQALDVVMRHLPSMRYTPVGRSFFTASEGCSNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEIRKYRVCNVTRRPASHQTFPLCTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDTGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLVDKEGRDHQALAKAVQVHQDTLRTMYFA 4z6h A 1.8 BS01 4L2 A 1 G43 F44 F45 F47 V49 I53 N100 Y106 G22 F23 F24 F26 V28 I32 N79 Y85 ? Kd=612nM remove_due_to_license_issue Q9H8M2 25864491 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 4z6i A 1.95 BS01 4L3 A 1 G43 F44 F45 F47 P48 V49 N100 Y106 G22 F23 F24 F26 P27 V28 N79 Y85 ? remove_due_to_license_issue Kd=493nM Q9H8M2 25864491 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 4z7h A 2.9 BS01 4L5 A 1 L577 K599 I642 C645 H692 L695 D711 L16 K38 I81 C84 H131 L134 D150 D688 K690 N693 D711 T734 D127 K129 N132 D150 T168 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue EC50=143nM, IC50=1180nM O75460 25968568 1001 SVVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPECFSFADREVQLLRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCKKLAVGRHSFSPGTEGWIAPEMLSNPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDKGGSVRDLLRAMRNKKHHYRELPAEVRETLGSLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFH 4z7k A 3.0 BS01 rna C 0 K22 R24 G25 Y26 H38 N39 H40 F45 V46 Y47 K48 S88 L124 N125 A126 N128 S129 E130 R146 G150 N151 L153 S154 K157 I163 K181 Q183 M185 V186 R206 S209 K22 R24 G25 Y26 H38 N39 H40 F45 V46 Y47 K48 S88 L124 N125 A126 N128 S129 E130 R146 G150 N151 L153 S154 K157 I163 K181 Q183 M185 V186 R206 S209 ? 0042802 remove_due_to_license_issue A4FXZ3 26996962 7 ~ 31 MDLEYMHISYPNILLNMRDGSKLRGYFAKKYIDEEIVHNHRDNAFVYKYPQIQFKIIDRSPLIIGIGSLGINFLESKRIFFEKELIISNDTNDITEVNVHKDMDHFGTTDKILKYQFKTPWMALNAKNSEIYKNSDEIDREEFLKRVLIGNILSMSKSLGYTIEEKLKVKINLKEVPVKFKNQNMVGFRGEFYINFDIPQYLGIGRNVSRGFGTVVKV 4z7k B 3.0 BS01 rna C 0 N125 N128 R146 G150 N151 L153 S154 K157 T162 I163 K166 L167 K181 N182 R206 N207 N102 N105 R123 G127 N128 L130 S131 K134 T139 I140 K143 L144 K158 N159 R183 N184 ? 0042802 remove_due_to_license_issue A4FXZ3 26996962 7 ~ 31 MDLEYMHISYPNILLNMRDGSKLRGYFAKKYIDYKYPQIQFKIIDRSPLIIGIGSLGINFLESKRIFFEKETEVNVHKDMDHFGTTDKILKYQFKTPWMALNAKNSEIYKNSDEIDREEFLKRVLIGNILSMSKSLGYTIEEKLKVKINLKEVPVKFKNQNMVGFRGEFYINFDIPQYLGIGRNVSRGFGTVVKV 4z7l A 3.503 BS01 rna C 0 R24 H38 N39 F45 V46 Y47 K127 N128 I149 G150 N151 L153 S154 K157 T162 I163 K166 L167 K181 Q183 G205 R206 N207 S209 R24 H38 N39 F45 V46 Y47 K127 N128 I149 G150 N151 L153 S154 K157 T162 I163 K166 L167 K181 Q183 G205 R206 N207 S209 ? 0042802 remove_due_to_license_issue A4FXZ3 26996962 16 ~ 29 MDLEYMHISYPNILLNMRDGSKLRGYFAKKYIDEEIVHNHRDNAFVYKYPQIQFKIIDRSPLIIGIGSLGINFLESKRIFFEKELIISNDTNDITEVNVHKDMDHFGTTDKILKYQFKTPWMALNAKNSEIYKNSDEIDREEFLKRVLIGNILSMSKSLGYTIEEKLKVKINLKEVPVKFKNQNMVGFRGEFYINFDIPQYLGIGRNVSRGFGTVVKV 4z7l D 3.503 BS01 rna F 0 R24 N39 F45 V46 Y47 P50 N125 K127 N128 R146 I149 G150 N151 L153 S154 S156 K157 Y161 T162 I163 L167 F180 K181 Q183 G205 R206 N207 S209 R210 R24 N39 F45 V46 Y47 P50 N125 K127 N128 R146 I149 G150 N151 L153 S154 S156 K157 Y161 T162 I163 L167 F180 K181 Q183 G205 R206 N207 S209 R210 ? 0042802 remove_due_to_license_issue A4FXZ3 26996962 16 ~ 29 MDLEYMHISYPNILLNMRDGSKLRGYFAKKYIDEEIVHNHRDNAFVYKYPQIQFKIIDRSPLIIGIGSLGINFLESKRIFFEKELIISNDTNDITEVNVHKDMDHFGTTDKILKYQFKTPWMALNAKNSEIYKNSDEIDREEFLKRVLIGNILSMSKSLGYTIEEKLKVKINLKEVPVKFKNQNMVGFRGEFYINFDIPQYLGIGRNVSRGFGTVVKV 4z7l G 3.503 BS01 rna I 0 R24 N39 F45 V46 Y47 N125 N128 R146 I149 G150 N151 L153 S154 K157 I163 K166 L167 K181 R206 N207 V208 S209 R24 N39 F45 V46 Y47 N125 N128 R146 I149 G150 N151 L153 S154 K157 I163 K166 L167 K181 R206 N207 V208 S209 ? 0042802 remove_due_to_license_issue A4FXZ3 26996962 16 ~ 29 MDLEYMHISYPNILLNMRDGSKLRGYFAKKYIDEEIVHNHRDNAFVYKYPQIQFKIIDRSPLIIGIGSLGINFLESKRIFFEKELIISNDTNDITEVNVHKDMDHFGTTDKILKYQFKTPWMALNAKNSEIYKNSDEIDREEFLKRVLIGNILSMSKSLGYTIEEKLKVKINLKEVPVKFKNQNMVGFRGEFYINFDIPQYLGIGRNVSRGFGTVVKV 4z83 E 1.8 BS02 4L7 E 1 G50 T51 G52 G55 R56 V57 A70 M120 E121 Y122 E170 M173 T183 D184 G37 T38 G39 G42 R43 V44 A57 M107 E108 Y109 E157 M160 T170 D171 N171 D184 N158 D171 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 26578105 401 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4z83 E 1.8 BS03 4L7 E 2 V15 F18 F100 L152 E155 Y306 V2 F5 F87 L139 E142 Y293 N171 D184 N158 D171 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 26578105 402 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4z84 A 1.554 BS02 NVX A 1 G50 T51 G52 G55 R56 V57 A70 K72 M120 E121 E170 M173 T183 D184 G37 T38 G39 G42 R43 V44 A57 K59 M107 E108 E157 M160 T170 D171 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 26578105 401 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 4z8d A 2.0 BS01 4LB A 1 R36 M207 G209 V212 F213 A246 R249 F304 R36 M207 G209 V212 F213 A246 R249 F304 2.3.1.180 0004315,0005737,0005829,0006631,0006633,0016746,0033818,0044281 ic50=6uM remove_due_to_license_issue P0A6R0 27626097 401 MYTKIIGTGSYLPEQVRTNADLEKMVDTSDEWIVTRTGIRERHIAAPNETVSTMGFEAATRAIEMAGIEKDQIGLIVVATTSATHAFPSAACQIQSMLGIKGCPAFDVAAACAGFTYALSVADQYVKSGAVKYALVVGSDVLARTCDPTDRGTIIIFGDGAGAAVLAASEEPGIISTHLHADGSYGELLTLPNADRVNPENSIHLTMAGNEVFKVAVTELAHIVDETLAANNLDRSQLDWLVPHQANLRIISATAKKLGMSMDNVVVTLDRHGNTSAASVPCALDEAVRDGRIKPGQLVLLEAFGGGFTWGSALVRF 4z93 A 1.27 BS01 4LD A 1 W374 P375 F376 L385 C429 N433 V439 W26 P27 F28 L37 C81 N85 V91 ? Kd=44.6nM remove_due_to_license_issue Kd=47nM, Ki=12nM, IC50=37nM O60885 26080064 501 KVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMPDE 4z9l A 2.1 BS02 880 A 1 I70 V78 A91 I92 K93 I124 L144 M146 M149 A151 Q155 S193 N194 L206 I26 V34 A47 I48 K49 I80 L100 M102 M105 A107 Q111 S149 N150 L162 D189 K191 N194 D207 T226 D145 K147 N150 D163 T172 2.7.11.24 0004672,0004707,0005524,0006468 ic50=1.6nM remove_due_to_license_issue IC50=1.6nM P53779 12954329 502 DNQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLSFMMVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFDSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPHTIEEWKELIYKEVMN 4za0 A 2.31 BS02 PAH A 1 G38 A39 S40 Q166 E167 D245 E293 D318 K343 R372 S373 K394 G38 A39 S40 Q166 E167 D245 E293 D318 K343 R372 S373 K394 S40 H158 E167 E210 D245 E293 D318 K343 H371 K394 S40 H158 E167 E210 D245 E293 D318 K343 H371 K394 4.2.1.11 0000015,0000287,0001917,0004634,0005515,0005615,0005737,0005829,0005886,0006094,0006096,0016020,0016829,0043025,0043204,0046872,0061621,0070062 remove_due_to_license_issue IC50=62.3nM P09104 27723749 503 MSIEKIWAREILDSRGNPTVEVDLYTAKGLFRAAVPSGASTGIYEALELRDGDKQRYLGKGVLKAVDHINSTIAPALISSGLSVVEQEKLDNLMLELDGTENKSKFGANAILGVSLAVCKAGAAERELPLYRHIAQLAGNSDLILPVPAFNVINGGSHAGNKLAMQEFMILPVGAESFRDAMRLGAEVYHTLKGVIKDKYGKDATNVGDEGGFAPNILENSEALELVKEAIDKAGYTEKIVIGMDVAASEFYRDGKYDLDFKSPTDPSRYITGDQLGALYQDFVRDYPVVSIEDPFDQDDWAAWSKFTANVGIQIVGDDLTVTNPKRIERAVEEKACNCLLLKVNQIGSVTEAIQACKLAQENGWGVMVSHRSGETEDTFIADLVVGLCTGQIKTGAPCRSERLAKYNQLMRIEEELGDEARFAGHNFRNPSVL 4zae A 1.86 BS01 4M1 A 1 Y99 R143 F174 S190 C191 Q192 W215 G216 C220 Y86 R132 F162 S180 C181 Q182 W205 G206 C209 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 Ki=3.6nM remove_due_to_license_issue Ki=3.6nM, IC50=3.64nM P00740 25978966 301 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGASALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKL 4zam A 1.42 BS01 MA4 A 1 I221 V224 P226 A248 V261 A280 A284 E288 I196 V199 P201 A222 V234 A253 A257 E261 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 26340563 301 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 4zb6 A 1.801 BS01 GDS A 1 H13 N18 H45 R58 V59 E74 S75 G116 P117 W176 H10 N15 H42 R55 V56 E71 S72 G113 P114 W173 G16 G13 ? Kd=0.53uM remove_due_to_license_issue A0A0R4I980 26348000 300 HGKQFTLYTHNSGPNGWKVAIVLEELGLSYEPVFLDLMKGEHKAPEYLKINPNGRVPALIDHKNNNYTVWESNAVTQYLVDKYDNDRKISVAPGTNEYYTQLQWLYFQASGQGPYYGQAAWFSVYHPEKIPSAIERYRNEIKRVLGVLESTLSKQEWLVGNKATVADFSFLTWNDIAANLLLENFRFEEEFPATAKWNKKLLERPAIAKVWEEKAKAAA 4zb6 A 1.801 BS02 GDS B 1 S113 R139 S110 R136 G16 G13 ? Kd=0.53uM remove_due_to_license_issue A0A0R4I980 26348000 300 HGKQFTLYTHNSGPNGWKVAIVLEELGLSYEPVFLDLMKGEHKAPEYLKINPNGRVPALIDHKNNNYTVWESNAVTQYLVDKYDNDRKISVAPGTNEYYTQLQWLYFQASGQGPYYGQAAWFSVYHPEKIPSAIERYRNEIKRVLGVLESTLSKQEWLVGNKATVADFSFLTWNDIAANLLLENFRFEEEFPATAKWNKKLLERPAIAKVWEEKAKAAA 4zb6 B 1.801 BS01 GDS A 1 S113 R139 S110 R136 G16 G13 ? Kd=0.53uM remove_due_to_license_issue A0A0R4I980 26348000 300 HGKQFTLYTHNSGPNGWKVAIVLEELGLSYEPVFLDLMKGEHKAPEYLKINPNGRVPALIDHKNNNYTVWESNAVTQYLVDKYDNDRKISVAPGTNEYYTQLQWLYFQASGQGPYYGQAAWFSVYHPEKIPSAIERYRNEIKRVLGVLESTLSKQEWLVGNKATVADFSFLTWNDIAANLLLENFRFEEEFPATAKWNKKLLERPAIAKVWEEKAKAA 4zb6 B 1.801 BS02 GDS B 1 H13 N18 H45 R58 V59 E74 S75 G116 P117 W176 H10 N15 H42 R55 V56 E71 S72 G113 P114 W173 G16 G13 ? Kd=0.53uM remove_due_to_license_issue A0A0R4I980 26348000 300 HGKQFTLYTHNSGPNGWKVAIVLEELGLSYEPVFLDLMKGEHKAPEYLKINPNGRVPALIDHKNNNYTVWESNAVTQYLVDKYDNDRKISVAPGTNEYYTQLQWLYFQASGQGPYYGQAAWFSVYHPEKIPSAIERYRNEIKRVLGVLESTLSKQEWLVGNKATVADFSFLTWNDIAANLLLENFRFEEEFPATAKWNKKLLERPAIAKVWEEKAKAA 4zb8 A 2.0 BS01 GDS A 1 G15 P16 N17 F39 H44 R57 I58 E73 S74 G115 P116 W175 G15 P16 N17 F39 H44 R57 I58 E73 S74 G115 P116 W175 G15 G15 ? Kd=0.94uM remove_due_to_license_issue A0A0R4I981 26348000 300 MSHGKQFTLYTHKGGPNGWKVTIVLEELGLTYESIFLDFQKGEHKAPEYLKVNPNGRIPALIDHKNNDYTVWESNAIIQYLVDKYDKDRKVSVAPGTNEYYTQLQWLYFQASGQGPYYGQAAWFSVYHPEKVPSAIERYRNEIKRVLGVLESVLSKQEFLVDGKATVADFSFLPWNEGAAKFLLEGSQFEEEFPATAKWHKKLLERPAIAKVWEERAKVS 4zba A 1.501 BS01 GDS A 1 S16 H18 Q45 R58 T59 E74 S75 Y128 S15 H17 Q44 R57 T58 E73 S74 Y127 ? Kd=3.09uM remove_due_to_license_issue A0A0R4I985 26348000 300 ASHDKQFSLFLHKASAHGWKVAFVLEELSLSYEIVLVDVAKNEQKSPEFMKLNPNGRTPALIDHGNSDFVIWESNAMVQYVADKYDTERKISMAPGTDDFYIQLQWQYFQGTGQGPYFGQLVWFTLYHEEKIPSAVTRYKEEALRVFSVLERVLSNQEWLVGGKMTIADISFVSWNDMIVHFLDNFDFEKEFPATAAWHYKMLKRPTIKRPWDERRKLMSRQ 4zba A 1.501 BS02 GDS B 1 T113 Y118 R139 T112 Y117 R138 ? Kd=3.09uM remove_due_to_license_issue A0A0R4I985 26348000 300 ASHDKQFSLFLHKASAHGWKVAFVLEELSLSYEIVLVDVAKNEQKSPEFMKLNPNGRTPALIDHGNSDFVIWESNAMVQYVADKYDTERKISMAPGTDDFYIQLQWQYFQGTGQGPYFGQLVWFTLYHEEKIPSAVTRYKEEALRVFSVLERVLSNQEWLVGGKMTIADISFVSWNDMIVHFLDNFDFEKEFPATAAWHYKMLKRPTIKRPWDERRKLMSRQ 4zba B 1.501 BS01 GDS A 1 T113 Y118 T111 Y116 ? Kd=3.09uM remove_due_to_license_issue A0A0R4I985 26348000 300 SHDKQFSLFLHKASAHGWKVAFVLEELSLSYEIVLVDVAKNEQKSPEFMKLNPNGRTPALIDHGNSDFVIWESNAMVQYVADKYDTERKISMAPGTDDFYIQLQWQYFQGTGQGPYFGQLVWFTLYHEEKIPSAVTRYKEEALRVFSVLERVLSNQEWLVGGKMTIADISFVSWNDMIVHFLDNFDFEKEFPATAAWHYKMLKRPTIKRPWDERRKLMSRQ 4zba B 1.501 BS02 GDS B 1 H13 S16 H18 Q45 R58 T59 E74 S75 Q121 Y128 H11 S14 H16 Q43 R56 T57 E72 S73 Q119 Y126 ? Kd=3.09uM remove_due_to_license_issue A0A0R4I985 26348000 300 SHDKQFSLFLHKASAHGWKVAFVLEELSLSYEIVLVDVAKNEQKSPEFMKLNPNGRTPALIDHGNSDFVIWESNAMVQYVADKYDTERKISMAPGTDDFYIQLQWQYFQGTGQGPYFGQLVWFTLYHEEKIPSAVTRYKEEALRVFSVLERVLSNQEWLVGGKMTIADISFVSWNDMIVHFLDNFDFEKEFPATAAWHYKMLKRPTIKRPWDERRKLMSRQ 4zbf A 2.2 BS01 4M7 A 1 F228 M231 M250 V253 F254 R263 T266 L267 F270 G271 I294 F58 M61 M80 V83 F84 R93 T96 L97 F100 G101 I124 ? 0042981 Ki=0.074uM remove_due_to_license_issue Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVED 4zbi A 2.5 BS01 4M6 A 1 M250 V253 F254 R263 T266 L267 F270 G271 I294 M80 V83 F84 R93 T96 L97 F100 G101 I124 ? 0042981 Ki=0.31uM remove_due_to_license_issue Ki=310nM Q07820 25844895 400 GDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 4zbn A 2.447 BS01 dna D 0 E11 F12 V18 S19 V20 W21 Y52 F54 R59 R69 E1 F2 V8 S9 V10 W11 Y40 F42 R47 R52 ? 0005102 remove_due_to_license_issue P01138 26027732 1 ~ 28 EFSVCDSVSVWVGDKTTATDIKGKEVMVLGEVNISVFKQYFFETKCRDSGCRGIDSKHWNSYCTTTHTFVKALTMDGKQAAWRFIRIDTACVCVLSR 4zbn A 2.447 BS02 dna E 0 I31 K32 F86 F101 I21 K22 F69 F84 ? 0005102 remove_due_to_license_issue P01138 26027732 1 ~ 28 EFSVCDSVSVWVGDKTTATDIKGKEVMVLGEVNISVFKQYFFETKCRDSGCRGIDSKHWNSYCTTTHTFVKALTMDGKQAAWRFIRIDTACVCVLSR 4zbn B 2.447 BS01 dna D 0 I31 K32 W76 F86 F101 R103 I28 K29 W65 F75 F86 R88 ? 0005102 remove_due_to_license_issue P01138 26027732 1 ~ 28 HPIFHRGEFSVCDSVSVWVGDKTTATDIKGKEVMVLGEVNSVFKQYFFETKCRDSGCRGIDSKHWNSYCTTTHTFVKALTMAAWRFIRIDTACVCVLSR 4zbn B 2.447 BS02 dna E 0 F7 F12 S19 V20 W21 Y52 F54 R59 R69 F4 F9 S16 V17 W18 Y46 F48 R53 R58 ? 0005102 remove_due_to_license_issue P01138 26027732 1 ~ 28 HPIFHRGEFSVCDSVSVWVGDKTTATDIKGKEVMVLGEVNSVFKQYFFETKCRDSGCRGIDSKHWNSYCTTTHTFVKALTMAAWRFIRIDTACVCVLSR 4zcs A 2.45 BS01 CDC A 1 D623 G624 V625 G632 Q636 T654 K663 W692 H709 D710 Y714 Y741 R755 T756 D8 G9 V10 G17 Q21 T39 K48 W77 H94 D95 Y99 Y108 R122 T123 F662 G664 F47 G49 2.7.7.15 0003824,0004105,0006657,0009058 remove_due_to_license_issue Q8IEE9 30046154 801 KNVVIYADGVYDMLHLGHMKQLEQAKKLFENTTLIVGVTSDNETKLFKGQVVQTLEERTETLKHIRWVDEIISPCPWVVTPEFLEKYKIDYVAHDDIPYANNQKEDIYAWLKRAGKFKATQRTEGVSTTDLIVRILKNYED 4zcw A 1.992 BS01 4NG A 1 G38 S40 Q166 E167 D245 D318 K343 H371 R372 S373 K394 G37 S39 Q165 E166 D244 D317 K342 H370 R371 S372 K393 S40 H158 E167 E210 D245 E293 D318 K343 H371 K394 S39 H157 E166 E209 D244 E292 D317 K342 H370 K393 4.2.1.11 0000015,0000287,0001917,0004634,0005515,0005615,0005737,0005829,0005886,0006094,0006096,0016020,0016829,0043025,0043204,0046872,0061621,0070062 ic50=42.5nM remove_due_to_license_issue IC50=42.5nM P09104 27723749 501 SIEKIWAREILDSRGNPTVEVDLYTAKGLFRAAVPSGASTGIYEALELRDGDKQRYLGKGVLKAVDHINSTIAPALISSGLSVVEQEKLDNLMLELDGTENKSKFGANAILGVSLAVCKAGAAERELPLYRHIAQLAGNSDLILPVPAFNVINGGSHAGNKLAMQEFMILPVGAESFRDAMRLGAEVYHTLKGVIKDKYGKDATNVGDEGGFAPNILENSEALELVKEAIDKAGYTEKIVIGMDVAASEFYRDGKYDLDFKSPTDPSRYITGDQLGALYQDFVRDYPVVSIEDPFDQDDWAAWSKFTANVGIQIVGDDLTVTNPKRIERAVEEKACNCLLLKVNQIGSVTEAIQACKLAQENGWGVMVSHRSGETEDTFIADLVVGLCTGQIKTGAPCRSERLAKYNQLMRIEEELGDEARFAGHNFRNPSVL 4ze6 A 1.17 BS01 011 A 1 D35 Y79 F116 D219 G221 D35 Y79 F116 D219 G221 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Kd=3.3mM remove_due_to_license_issue P11838 27139825 416 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 4zec A 2.15 BS01 C84 A 1 S53 N54 Y145 W178 Y375 Y376 F407 W418 S419 N420 G421 E434 R444 E510 S22 N23 Y114 W147 Y344 Y345 F376 W387 S388 N389 G390 E403 R413 E479 ? 0015833,0030288,0042597,0043190,0055085,1904680 remove_due_to_license_issue Q52012 26244338 601 RRALRLGVNGLPNSLEPVNAISNVGPRIVNQIFDTLIARDFFAKGAPGNAIDLVPALAESWERIDEKSVRFKLRQKVMFHDGVELTADDVAYTFSSERLWGPEAIKKIPLGKSYSLDFDEPVVEDKYTVTLRTKTPSYLIETFVASWMSRIVPKEYYKKLGAVDFGNKPVGTGPYKFVEFVAGDRVVLEANDAYWGPKPTASKITYQIVAEPATRVAGLISGEYDIITTLTPDDIQLINSYPDLETRGTLIENFHMFTFNMNQEVFKDKKLRRALALAVNRPIMVEALWKKQASIPAGFNFPNYGETFDPKRKAMEYNVEEAKRLVKESGYDGTPITYHTMGNYYANAMPALMMMIEMWKQIGVNVVMKTYAPGSFPPDNQTWMRNWSNGQWMTDAYATIVPEFGPNGQVQKRWGWKAPAEFNELCQKVTVLPNGKERFDAYNRMRDIFEEEAPAVILYQPYDVYAARKDVHWKPVSFEMMEFRNNLSFG 4zed A 1.75 BS01 AGW A 1 L42 N44 S53 N54 W178 M372 Y375 Y376 Y402 F407 W418 S419 N420 G421 E434 E510 L11 N13 S22 N23 W147 M341 Y344 Y345 Y371 F376 W387 S388 N389 G390 E403 E479 ? 0015833,0030288,0042597,0043190,0055085,1904680 remove_due_to_license_issue Q52012 26244338 601 RRALRLGVNGLPNSLEPVNAISNVGPRIVNQIFDTLIARDFFAKGAPGNAIDLVPALAESWERIDEKSVRFKLRQKVMFHDGVELTADDVAYTFSSERLWGPEAIKKIPLGKSYSLDFDEPVVEDKYTVTLRTKTPSYLIETFVASWMSRIVPKEYYKKLGAVDFGNKPVGTGPYKFVEFVAGDRVVLEANDAYWGPKPTASKITYQIVAEPATRVAGLISGEYDIITTLTPDDIQLINSYPDLETRGTLIENFHMFTFNMNQEVFKDKKLRRALALAVNRPIMVEALWKKQASIPAGFNFPNYGETFDPKRKAMEYNVEEAKRLVKESGYDGTPITYHTMGNYYANAMPALMMMIEMWKQIGVNVVMKTYAPGSFPPDNQTWMRNWSNGQWMTDAYATIVPEFGPNGQVQKRWGWKAPAEFNELCQKVTVLPNGKERFDAYNRMRDIFEEEAPAVILYQPYDVYAARKDVHWKPVSFEMMEFRNNLSFG 4zei A 2.3 BS01 LAO A 1 S53 N54 W178 Y375 Y376 W418 S419 N420 G421 E434 E510 S22 N23 W147 Y344 Y345 W387 S388 N389 G390 E403 E479 ? 0015833,0030288,0042597,0043190,0055085,1904680 Kd=1.33uM remove_due_to_license_issue Q52012 26244338 601 RRALRLGVNGLPNSLEPVNAISNVGPRIVNQIFDTLIARDFFAKGAPGNAIDLVPALAESWERIDEKSVRFKLRQKVMFHDGVELTADDVAYTFSSERLWGPEAIKKIPLGKSYSLDFDEPVVEDKYTVTLRTKTPSYLIETFVASWMSRIVPKEYYKKLGAVDFGNKPVGTGPYKFVEFVAGDRVVLEANDAYWGPKPTASKITYQIVAEPATRVAGLISGEYDIITTLTPDDIQLINSYPDLETRGTLIENFHMFTFNMNQEVFKDKKLRRALALAVNRPIMVEALWKKQASIPAGFNFPNYGETFDPKRKAMEYNVEEAKRLVKESGYDGTPITYHTMGNYYANAMPALMMMIEMWKQIGVNVVMKTYAPGSFPPDNQTWMRNWSNGQWMTDAYATIVPEFGPNGQVQKRWGWKAPAEFNELCQKVTVLPNGKERFDAYNRMRDIFEEEAPAVILYQPYDVYAARKDVHWKPVSFEMMEFRNNLSFG 4zek A 2.09 BS01 LAH A 1 S53 N54 W178 Y375 Y376 W418 S419 N420 G421 E434 E510 S22 N23 W147 Y344 Y345 W387 S388 N389 G390 E403 E479 ? 0015833,0030288,0042597,0043190,0055085,1904680 remove_due_to_license_issue Q52012 26244338 601 RRALRLGVNGLPNSLEPVNAISNVGPRIVNQIFDTLIARDFFAKGAPGNAIDLVPALAESWERIDEKSVRFKLRQKVMFHDGVELTADDVAYTFSSERLWGPEAIKKIPLGKSYSLDFDEPVVEDKYTVTLRTKTPSYLIETFVASWMSRIVPKEYYKKLGAVDFGNKPVGTGPYKFVEFVAGDRVVLEANDAYWGPKPTASKITYQIVAEPATRVAGLISGEYDIITTLTPDDIQLINSYPDLETRGTLIENFHMFTFNMNQEVFKDKKLRRALALAVNRPIMVEALWKKQASIPAGFNFPNYGETFDPKRKAMEYNVEEAKRLVKESGYDGTPITYHTMGNYYANAMPALMMMIEMWKQIGVNVVMKTYAPGSFPPDNQTWMRNWSNGQWMTDAYATIVPEFGPNGQVQKRWGWKAPAEFNELCQKVTVLPNGKERFDAYNRMRDIFEEEAPAVILYQPYDVYAARKDVHWKPVSFEMMEFRNNLSFG 4zfi A 2.0 BS01 4NJ A 1 L54 F55 G58 I61 Y67 V93 H96 I99 Y100 L37 F38 G41 I44 Y50 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 Kd=0.5uM remove_due_to_license_issue Q00987 27709883 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVNQ 4zg6 A 1.8 BS04 4NY A 1 S170 L214 L217 A218 F274 F275 Y307 D359 S107 L151 L154 A155 F211 F212 Y244 D296 3.1.4.39 0003676,0005044,0006955,0016787,0030247,0046872 ic50=0.011uM remove_due_to_license_issue Q13822 26371182 910 GSCKGRCFELCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFSNNAKYDPKAIIAALTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPFFQGDHGFDNKVNSMQTVFVGYGSTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPEEVTRPNYPGIMYLQSDFDLGTEERHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQAEVSSCVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 4zg7 A 1.75 BS04 4O0 A 1 L79 S82 F211 L214 Y215 K249 F250 H252 W255 W261 F275 S277 V278 L25 S28 F157 L160 Y161 K195 F196 H198 W201 W207 F221 S223 V224 3.1.4.39 0003676,0004528,0004622,0004630,0005509,0005576,0005615,0005886,0006644,0006935,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030334,0034638,0046872,0047391,0048870,0050731,2000394 ic50=0.002uM remove_due_to_license_issue Q13822 26371182 908 ISGSCKGRCFELQEAGPPDCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFSNNAKYDPKAIIAALTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPLDCFFQGDHGFDNKVNSMQTVFVGYGPTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPEEVTRPNYPGIMYLQSDFDLGCTCDDERHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQAEVSSVPDHLTSCVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 4zg9 A 2.95 BS04 4O2 A 1 S170 F211 L214 Y215 F274 F275 W276 R285 Y307 S109 F150 L153 Y154 F208 F209 W210 R219 Y241 3.1.4.39 0003676,0005044,0006955,0016787,0030247,0046872 remove_due_to_license_issue IC50=<500nM Q13822 26371182 908 SCKGRCFELQPDCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFSNNAKYDPKAIIANLTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPCFFQGDHGFDNKVNSMQTVFVGYGSTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPEEVTRPNYPGIMYLQSDFDLGRHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQPDHLTSCVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 4zg9 A 2.95 BS05 4O2 A 2 F242 W254 W255 R440 F181 W188 W189 R374 3.1.4.39 0003676,0005044,0006955,0016787,0030247,0046872 remove_due_to_license_issue IC50=<500nM Q13822 26371182 909 SCKGRCFELQPDCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFSNNAKYDPKAIIANLTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPCFFQGDHGFDNKVNSMQTVFVGYGSTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPEEVTRPNYPGIMYLQSDFDLGRHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQPDHLTSCVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 4zga A 2.6 BS05 4O3 A 1 F211 L214 Y215 W255 F274 F275 W276 Y307 F144 L147 Y148 W188 F207 F208 W209 Y240 3.1.4.39 0003676,0005044,0006955,0016787,0030247,0046872 remove_due_to_license_issue IC50=<500nM Q13822 26371182 910 GSCKGRCFELCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGNEENACHCEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFDPKAIIANLTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPFFQGDHGFDNKVNSMQTVFVGYGSTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPEEVTRPNYPGIMYLQSDFDLGTEERHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQACVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 4zgk A 2.0 BS01 4NX A 1 L54 F55 G58 H96 I99 Y100 L38 F39 G42 H80 I83 Y84 2.3.2.27 0005634,0043066,0051726 Kd=3.1uM remove_due_to_license_issue Q00987 27709883 201 MQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4zh2 C 4.204 BS01 4OB C 1 P552 Y555 G640 E641 S642 P550 Y553 G638 E639 S640 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 26190576 2001 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4zh2 D 4.204 BS01 4OB C 1 P750 F773 I774 P743 F766 I767 2.7.7.6 0000287,0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0008270,0009408,0016020,0016779,0031564,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0046872,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8T7 26190576 2001 LKAQTKTEEFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRRAAG 4zh3 C 4.082 BS01 4OD D 1 P552 Y555 R637 S642 P550 Y553 R635 S640 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 26190576 1504 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4zh3 D 4.082 BS04 4OD D 1 K749 P750 L770 F773 I774 K727 P728 L748 F751 I752 2.7.7.6 0000287,0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0008270,0009408,0016020,0016779,0031564,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0046872,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8T7 26190576 1504 LKAQTKTEEFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRRAAG 4zh4 C 3.993 BS01 4OE C 1 P552 Y555 G640 S642 P550 Y553 G638 S640 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 26190576 2001 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 4zh4 D 3.993 BS01 4OE C 1 P750 I755 F773 P728 I733 F751 2.7.7.6 0000287,0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0008270,0009408,0016020,0016779,0031564,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0046872,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8T7 26190576 2001 LKAQTKTEEFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRRAAG 4zij A 1.78 BS01 SFQ A 1 H32 Q35 F36 P163 T168 M171 F174 H32 Q35 F36 P163 T168 M171 F174 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=565uM remove_due_to_license_issue P0AEG4 27778134 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 4zim A 2.65 BS01 4OK A 1 Q853 L855 G856 K857 V863 A880 E930 Y931 L932 G935 L983 D994 Q12 L14 G15 K16 V22 A39 E86 Y87 L88 G91 L139 D150 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=2.4nM O60674 25987372 1201 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 4zip A 1.11 BS01 G64 B 1 R8 D25 A28 D30 V82 R8 D25 A28 D30 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 26096678 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4zip B 1.11 BS01 G64 B 1 D25 G27 A28 D29 I47 G48 I50 D25 G27 A28 D29 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.21nM remove_due_to_license_issue P03366 26096678 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4zj8 A 2.751 BS01 SUV A 1 A102 S103 P123 Q126 V130 Q179 F219 I314 N318 H344 Y348 A77 S78 P98 Q101 V105 Q154 F194 I444 N448 H474 Y478 ? 0004930,0007186,0007631,0016020,0016499 remove_due_to_license_issue O43613,Q9V2J8 26950369 2001 DYEDEFLRYLWRDYLYPKQYEWVLIAAYVAVFVVALVGNTLVCLAVWRNHHMRTVTNYFIVNLSLADVLVTAICLPASLLVDITESWLFGHALCKVIPYLQAVSVSVAVLTLSFIALDRWYAICHPLLFKSTARRARGSILGIWAVSLAIMVPQAAVMECSSVLPELANRTRLFSVCDERWADDLYPKIYHSCFFIVTYLAPLGLMAMAYFQIFRKLWGRQGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKQMRARRKTAKMLMVVLLVFALCYLPISVLNILKRVFGMFRQASDREAVYACFTFSHWLVYANSAANPIIYNFLSGKFREQFKAAF 4zjc A 2.832 BS01 4OT A 1 S103 P123 Q126 V130 Q179 F219 I314 N318 H344 Y348 S78 P98 Q101 V105 Q154 F194 I444 N448 H474 Y478 ? 0004930,0007186,0007631,0016020,0016499 remove_due_to_license_issue O43613,Q9V2J8 26950369 2001 DYEDEFLRYLWRDYLYPKQYEWVLIAAYVAVFVVALVGNTLVCLAVWRNHHMRTVTNYFIVNLSLADVLVTAICLPASLLVDITESWLFGHALCKVIPYLQAVSVSVAVLTLSFIALDRWYAICHPLLFKSTARRARGSILGIWAVSLAIMVPQAAVMECSSVLPELANRTRLFSVCDERWADDLYPKIYHSCFFIVTYLAPLGLMAMAYFQIFRKLWGRQGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKQMRARRKTAKMLMVVLLVFALCYLPISVLNILKRVFGMFRQASDREAVYACFTFSHWLVYANSAANPIIYNFLSGKFREQFKAAF 4zji A 1.99 BS01 4OQ A 1 E315 V318 M319 N322 I327 V328 F379 N383 H387 L405 T406 A412 E57 V60 M61 N64 I69 V70 F121 N125 H129 L147 T148 A154 D389 K391 D393 N394 D407 P416 T427 D131 K133 D135 N136 D149 P158 T163 2.7.11.1 0004672,0005524,0006468 Kd=340nM remove_due_to_license_issue Kd=340nM, IC50=323nM Q13153 26191365 601 LEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQMNLKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 4zjj A 2.2 BS01 4OR A 1 M301 I312 E315 M319 N322 I327 V328 F379 N383 H387 L405 T406 M53 I60 E63 M67 N70 I75 V76 F127 N131 H135 L153 T154 D389 K391 D393 N394 D407 T427 D137 K139 D141 N142 D155 T168 2.7.11.1 0004672,0005524,0006468 Kd=9.9nM remove_due_to_license_issue IC50=18nM, Kd=9.9nM Q13153 26191365 601 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQMNLQKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKE 4zjr A 2.702 BS01 4P3 A 1 W317 C320 H323 L324 M365 F378 E379 F388 I397 I400 F401 W53 C56 H59 L60 M101 F114 E115 F124 I133 I136 F137 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=93nM, IC50=11nM P51449 26048806 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVE 4zjw A 2.5 BS01 4P1 A 1 Q286 H323 M365 F378 E379 F388 I400 V480 Q19 H56 M98 F111 E112 F121 I133 V213 ? 0003677,0004879,0005634,0006355 ic50=0.1uM remove_due_to_license_issue IC50=100nM, EC50=200nM P51449 26048806 501 TEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIF 4zk5 A 2.89 BS02 4P4 A 1 V31 Y36 V39 K41 A52 K54 M105 F107 C108 G109 G111 L160 V170 D171 V15 Y20 V23 K25 A36 K38 M89 F91 C92 G93 G95 L144 V154 D155 D153 K155 Q157 N158 D171 T191 D137 K139 Q141 N142 D155 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=3.7nM O95819 26288693 403 SLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEDEEEEIKLEINMLKKYSHHRNIATYYGAFIKKSPPGHDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGVSANTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRTRK 4zki B 3.401 BS01 ADP B 1 N514 K517 Y518 D542 G546 I547 R561 V562 G571 G572 T573 G574 L575 G576 L577 S601 F603 N118 K121 Y122 D146 G150 I151 R165 V166 G170 G171 T172 G173 L174 G175 L176 S200 F202 2.7.13.3 0000155,0000160,0000166,0004721,0005886,0007165,0016020,0016036,0016301,0016310,0016772 remove_due_to_license_issue A0A0M3KKX3 28994408 701 QFVSNVSHELRTPLTSLRSYIEALSDGAWKDPEVAPGFLKVTQEETDRMIRMINELLSRVDMELVNINEMFNYVLDRFDMILKKDKYYTIKREFTKRDLWVEIDTDKFTQVLDNIMNNAIKYSPDGGVVTCRLLETHNQVIISISDQGLGIPRADLGHVFDRFFRVDKQGGTGLGLAISKEVVQMLGGRIWVDSVEGKGSTFYISLPYE 4zl4 A 2.37 BS01 4PK A 1 A60 D80 G82 Y139 C140 E141 L179 F180 Q183 D313 G315 S316 T317 A17 D37 G39 Y96 C97 E98 L136 F137 Q140 D238 G240 S241 T242 3.4.23.- 0004190,0006508 Kd=13.8nM remove_due_to_license_issue A5K302 26214367 501 KDLLYKYKLYGDIDEYAYYFLDIDIGTPEQRISLILDTGSSSLSFPCAGCKNCGVHMENPFNLNNSKTSSILYCENEECPFKLNCVKGKCEYMQSYCEGSQISGFYFSDVVSVVSYNNERVTFRKLMGCHMHEESLFLYQQATGVLGMSLSKPQGIPTFVNLLFDNAPQLKQVFTICISENGGELIAGGYDPAYIVRAEKVVWENVTRKYYYYIKVRGLDMFGTNMMSSSKGLEMLVDSGSTFTHIPEDLYNKLNYFFDILCIQDMNNAYDVNKRLKMTNESFNNPLVQFDDFRKSLKSIIAKENMCVKIVDGVQCWKYLEGLPDLFVTLSNNYKMKWQPHSYLYKKESFWCKGIEKQVNNKPILGLTFFKNRQVIFDIQKNRIGFVDANCPSHP 4zla A 1.9 BS05 BES A 1 K258 D263 D281 D340 E342 T367 L368 T369 G370 A461 K247 D252 D270 D329 E331 T356 L357 T358 G359 A450 K270 R344 K259 R333 3.4.11.1,3.4.11.10 0004177,0005737,0006508,0008235,0019538,0030145,0046872,0070006 ic50=49.9nM remove_due_to_license_issue O25294 26616008 505 MLKIKLEKTTFENAKAECSLVFIINKDFSHAWVKNKELLETFKYEGEGVFLDQENKILYAGVKEDDVHLLRESACLAVRTLKKLAFKSVKVGVYTCGAHNALLENLKALFLGLKLGLYEYDTFKSNKKESVLKEAIVALELHKSLEKSAKEALKYAEIMTESLNIVKDLVNTPPMIGTPVYMAEVAQKVAKENHLEIHVHDEKFLEEKKMNAFLAVNKASLSVNPPRLIHLVYKPKKAKKKIALVGKGLTYDCGGLSLKPADYMVTMKADKGGGSAVIGLLNALAKLGVEAEVHGIIGATENMIGPAAYKPDDILISKEGKSIEVRNTDAEGRLVLADCLSYAQDLNPDVIVDFATLTGACVVGLGEFTSAIMGHNEELKNLFETSGLESGELLAKLPFNRHLKKLIESKIADVCNISSSRYGGAITAGLFLNEFIRDEFKDKWLHIDIAGPAYVEKEWDVNSFGASGAGVRACTAFVEELLKKA 4zla B 1.9 BS05 BES B 1 K258 D263 D281 D340 E342 T367 L368 T369 G370 A461 K244 D249 D267 D326 E328 T353 L354 T355 G356 A447 K270 R344 K256 R330 3.4.11.1,3.4.11.10 0004177,0005737,0006508,0008235,0019538,0030145,0046872,0070006 ic50=49.9nM remove_due_to_license_issue O25294 26616008 505 MLKIKLEKTTFENAKAECSLVFIINKDFSHAWVKNKELLETFKYEGEGVFLDQENKILYAGVKEDDVHLLRESACLAVRTLKKLAFKSVKVGVYTCGAALLENLKALFLGLKLGLYEYDTFKSNKKESVLKEAIVALELHKLEKSAKEALKYAEIMTESLNIVKDLVNTPPMIGTPVYMAEVAQKVAKENHLEIHVHDEKFLEEKKMNAFLAVNKASLSVNPPRLIHLVYKPKKAKKKIALVGKGLTYDCGGLSLKPADYMVTMKADKGGGSAVIGLLNALAKLGVEAEVHGIIGATENMIGPAAYKPDDILISKEGKSIEVRNTDAEGRLVLADCLSYAQDLNPDVIVDFATLTGACVVGLGEFTSAIMGHNEELKNLFETSGLESGELLAKLPFNRHLKKLIESKIADVCNISSSRYGGAITAGLFLNEFIRDEFKDKWLHIDIAGPAYVEKEWDVNSFGASGAGVRACTAFVEELLKKA 4zla E 1.9 BS05 BES E 1 K258 D263 M278 D281 D340 E342 T367 L368 T369 G370 K246 D251 M266 D269 D328 E330 T355 L356 T357 G358 K270 R344 K258 R332 3.4.11.1,3.4.11.10 0004177,0005737,0006508,0008235,0019538,0030145,0046872,0070006 ic50=49.9nM remove_due_to_license_issue O25294 26616008 505 MLKIKLEKTTFENAKAECSLVFIINKDFSHAWVKNKELLETFKYEGEGVFLDQENKILYAGVKEDDVHLLRESACLAVRTLKKLAFKSVKVGVYTCGAALLENLKALFLGLKLGLYEYDTFKSNKKESVLKEAIVALELHKPSLEKSAKEALKYAEIMTESLNIVKDLVNTPPMIGTPVYMAEVAQKVAKENHLEIHVHDEKFLEEKKMNAFLAVNKASLSVNPPRLIHLVYKPKKAKKKIALVGKGLTYDCGGLSLKPADYMVTMKADKGGGSAVIGLLNALAKLGVEAEVHGIIGATENMIGPAAYKPDDILISKEGKSIEVRNTDAEGRLVLADCLSYAQDLNPDVIVDFATLTGACVVGLGEFTSAIMGHNEELKNLFETSGLESGELLAKLPFNRHLKKLIESKIADVCNISSSRYGGAITAGLFLNEFIRDEFKDKWLHIDIAGPAYVEKEWDVNSFGASGAGVRACTAFVEELLKKA 4zlo A 2.5 BS01 4PV A 1 E315 V318 M319 N322 I327 N383 V385 H387 L405 T406 E59 V62 M63 N66 I71 N127 V129 H131 L149 T150 D389 K391 D393 N394 D407 T427 D133 K135 D137 N138 D151 T162 2.7.11.1 0004672,0005524,0006468 ic50=12uM remove_due_to_license_issue IC50=12000nM Q13153 26191365 601 DEEILEKLRSIVSVGDPKKKYTRFEKIGQSGTVYTAMDVATGQEVAIKQMNKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATKN 4zls A 1.53 BS01 G61 B 1 D25 G27 G48 G49 I50 D25 G27 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 26107245 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4zls B 1.53 BS01 G61 B 1 L23 D25 G27 A28 D30 P81 V82 L23 D25 G27 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.82nM remove_due_to_license_issue P03366 26107245 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 4zly A 1.65 BS01 4RU A 1 L408 A428 Y476 M477 L528 L20 A40 Y88 M89 L140 D521 A523 R525 N526 D539 F559 D133 A135 R137 N138 D151 F171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3.5uM remove_due_to_license_issue IC50=3500nM Q06187 26087137 705 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4zlz A 2.0 BS01 4RV A 1 L408 T410 A428 M477 L528 D539 L20 T22 A40 M89 L140 D151 D521 A523 R525 N526 D539 F559 D133 A135 R137 N138 D151 F171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=100nM remove_due_to_license_issue IC50=100000nM, EC50=28600nM Q06187 26087137 705 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 4zme A 1.98 BS02 ADN A 1 E588 G589 V643 K645 E713 L716 F720 E38 G39 V93 K95 E160 L163 F167 2.7.11.7 0004674,0005524,0006468 Kd=50uM remove_due_to_license_issue P42527 26260792 1002 GISSETGEMGILWEFDPIINKWIRLSMKLKVERKPFAEGALREAYHTVSLGVGTDENYPLGTTTKLFPPIEMISPISKNNEAMTQLKNGTKFVLKLYKKQQASRELYFEDVKMQMVCRDWGNKFNQKKPPKKIEFLMSWVVELIDRSPSSNGQPILCSIEPLLVGEFKKNNSNYGAVLTNRSTPQAFSHFTYELSNKQMIVVDIQGVDDLYTDPQIHTPDGKGFGLGNLGKAGINKFITTHKCNAVCALLDLDVKLGGVLSG 4zmf A 2.39 BS01 AMP A 1 A587 R592 K645 E713 L716 F720 A36 R41 K92 E156 L159 F163 2.7.11.7 0004674,0005524,0006468 Kd=110uM remove_due_to_license_issue P42527 26260792 901 ISSETGEMGILWEFDPIINKWIRLSMKLKVERKPFAEGALREAYHTVSLGVGTDENYPLGTKLFPPIEMISPISKNNEAMTQLKNGTKFVLKLYKKEASRELYFEDVKMQMVCRDWGNKFNQKKPPKKIEFLMSWVVELIDRSPSSNGQPILCSIEPLLVGEFKKNNSNYGAVLTNRSTPQAFSHFTYELSNKQMIVVDIQGVDDLYTDPQIHTPDGKGFGLGNLGKAGINKFITTHKCNAVCALLDLDVK 4zo5 B 2.5 BS02 4Q0 B 1 I682 Y683 F686 M703 E711 G715 F719 I246 Y247 F250 M267 E275 G279 F283 3.1.4.17 0004114,0007165,0008081 Ki=0.15nM remove_due_to_license_issue Ki=0.15nM Q9Y233 26077491 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 4zom A 2.27 BS01 4Q3 A 1 W317 C320 H323 M365 F378 E379 F388 L391 C393 I397 I400 F401 H479 W53 C56 H59 M101 F114 E115 F124 L127 C129 I133 I136 F137 H215 ? 0003677,0004879,0005634,0006355 ic50=3nM remove_due_to_license_issue EC50=10.0nM, IC50=4.9nM P51449 26048789 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQ 4zow A 2.45 BS01 CLM A 1 Y30 N33 D34 L119 A150 Y21 N24 D25 L110 A141 ? 0005886,0015385,0015386,0016020,0022857,0030641,0035725,0046677,0055085,0071805,1902600,1990961 Kd=75uM remove_due_to_license_issue P0AEY8 26238402 500 RLGRQALLFPLCLVLYEFSTYIGNDMIQPGMLAVVEQYQAGIDWVPTSMTAYLAGGMFLQWLLGPLSDRIGRRPVMLAGVVWFIVTCLAILLAQNIEQFTLLRFLQGISLCFIGAVGYAAIRESFEEAVCIKITALMANVALIAPLLGPLVGAAWIHVLPWEGMFVLFAALAAISFFGLQRAMPETATRIGEKLSLKELGRDYKLVLKNGRFVAGALALGFVSLPLLAWIAQSPIIIITGEQLSSYEYGLLQVPIFGALIAGNLLLARLTSRRTVRSLIIMGGWPIMIGLLVAAAATVISSHAYLWMTAGLSIYAFGIGLANAGLVRLTLFASDMSKGTVSAAMGMLQMLIFTVGIEISKHAWLNGGNGLFNLFNLVNGILWLSLMVIFLK 4zpe A 1.7 BS01 4QA A 1 L30 Y71 T72 Q73 G74 F108 I110 W115 Y198 G230 L34 Y75 T76 Q77 G78 F112 I114 W119 Y189 G221 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D219 T222 3.4.23.46 0004190,0006508,0016020 ic50=0.45uM remove_due_to_license_issue P56817 26195137 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVESQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACDEFRTAAVEGPFVTLDMEDCGYN 4zpf A 1.8 BS01 4QD A 1 Q12 G13 L30 D32 Y71 T72 Q73 F108 I110 W115 G230 Q16 G17 L34 D36 Y75 T76 Q77 F112 I114 W119 G223 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=0.18uM remove_due_to_license_issue P56817 26195137 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHDEFRTAAVEGPFVTLDMEDCGYN 4zpg A 2.0 BS01 4QF A 1 L30 D32 Y71 Q73 G74 F108 I110 W115 Y198 G230 L34 D36 Y75 Q77 G78 F112 I114 W119 Y190 G222 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 ic50=0.055uM remove_due_to_license_issue P56817 26195137 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGAWAGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACDEFRTAAVEGPFVTLDMEDCGYN 4zph A 2.8 BS01 PRL A 1 R266 V305 R121 V129 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P53762 26245371 501 ERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSRRSFICRMRCPHFVVVHCTGYIKAFCLVAIGRLQVPTEFISRHNIEGIFTFVDHRCVATVGYQPQELLGKNIVEFCHPEDQQLLRDSFQQVVKLKGQVLSVMFRFRSKTREWLWMRTSSFTFQNPYSDEIEYIICTNTNV 4zpk A 3.6 BS01 dna C 0 R91 H94 E98 R99 R102 D127 K128 R5 H8 E12 R13 R16 D41 K42 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P53762 26245371 1 ~ 21 ERLARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSRRSFICRMRCGTPHFVVVHCTGYIKFCLVAIGRLQVTEFISRHNIEGIFTFVDHRCVATVGYQPQELLGKNIVEFCHPEDQQLLRDSFQQVVKLKGQVLSVMFRFRSKTREWLWMRTSSFTFQNPYSDEIEYIICTNTNV 4zpk A 3.6 BS02 dna D 0 H94 E98 R101 H8 E12 R15 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P53762 26245371 1 ~ 21 ERLARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSRRSFICRMRCGTPHFVVVHCTGYIKFCLVAIGRLQVTEFISRHNIEGIFTFVDHRCVATVGYQPQELLGKNIVEFCHPEDQQLLRDSFQQVVKLKGQVLSVMFRFRSKTREWLWMRTSSFTFQNPYSDEIEYIICTNTNV 4zpk B 3.6 BS01 dna C 0 K18 R26 N184 K186 K11 R19 N164 K166 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P97481 26245371 1 ~ 21 KRSSSELRKEKSRDAARCRRSKETEVFYELAHELPLPHSVSSHLDKASIMRLAISFLRTHKLLSSVCSENESEAEADQQMDNLYLKALEGFIAVVTQDGDMIFLSENISKFMGLTQVELTGHSIFDFTHPCDHEEIRENLTLSTERDFFMRMKCTVTNRGRTVNLKSATWKVLHCTGQVRVYNLSCLIIMCEPIQHPSHMDIPLDSKTFLSRHSMDMKFTYCDDRILELIGYHPEELLGRSAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGGYVWLETQGTVIYNLQPQCIMCVNYVLSEIKNDVVFSMDQTE 4zpk B 3.6 BS02 dna D 0 K16 S19 R20 R24 R27 K53 K9 S12 R13 R17 R20 K46 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P97481 26245371 1 ~ 21 KRSSSELRKEKSRDAARCRRSKETEVFYELAHELPLPHSVSSHLDKASIMRLAISFLRTHKLLSSVCSENESEAEADQQMDNLYLKALEGFIAVVTQDGDMIFLSENISKFMGLTQVELTGHSIFDFTHPCDHEEIRENLTLSTERDFFMRMKCTVTNRGRTVNLKSATWKVLHCTGQVRVYNLSCLIIMCEPIQHPSHMDIPLDSKTFLSRHSMDMKFTYCDDRILELIGYHPEELLGRSAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGGYVWLETQGTVIYNLQPQCIMCVNYVLSEIKNDVVFSMDQTE 4zq9 A 2.6 BS01 dna D 0 K101 M103 V104 R107 F108 R138 K93 M95 V96 R99 F100 R130 3.6.4.12 remove_due_to_license_issue P03132 26370092 1 ~ 21 PGFYEIVIKVPSDISDSFVNWVAEKEWELPPDSDMDLNLIEQAPLTVAEKLQRDFLTEWRRVSKAPEALFFVQFEKGESYFHMHVLVETTGVKSMVLGRFLSQIREKLIQRIYRGIEPTLPNWFAVTKTRNGAGGGNKVVDESYIPNFLLPKTQPELQWAWTNMEQYLSACLNLTERKRLVAQHL 4zq9 A 2.6 BS02 dna E 0 S102 M103 G106 K136 R138 G142 G143 G144 N145 S94 M95 G98 K128 R130 G134 G135 G136 N137 3.6.4.12 remove_due_to_license_issue P03132 26370092 22 ~ 42 PGFYEIVIKVPSDISDSFVNWVAEKEWELPPDSDMDLNLIEQAPLTVAEKLQRDFLTEWRRVSKAPEALFFVQFEKGESYFHMHVLVETTGVKSMVLGRFLSQIREKLIQRIYRGIEPTLPNWFAVTKTRNGAGGGNKVVDESYIPNFLLPKTQPELQWAWTNMEQYLSACLNLTERKRLVAQHL 4zq9 B 2.6 BS01 dna D 0 V104 R107 R138 V99 R102 R133 3.6.4.12 remove_due_to_license_issue P03132 26370092 1 ~ 21 PGFYEIVIKVPSDLDGISDSFVNWVAEKEWELPPDSDMDLNLIEQAPLTVAEKLQRDFLTEWRRVSKAPEALFFVQFEKGESYFHMHVLVETTGVKSMVLGRFLSQIREKLIQRIYRGIEPTLPNWFAVTKTRNGAGGGNKVVDESYIPNFLLPKTQPELQWAWTNMEQYLSACLNLTERKRLVAQHLT 4zq9 B 2.6 BS02 dna E 0 S102 M103 G106 K136 R138 G142 G143 G144 N145 S97 M98 G101 K131 R133 G137 G138 G139 N140 3.6.4.12 remove_due_to_license_issue P03132 26370092 22 ~ 42 PGFYEIVIKVPSDLDGISDSFVNWVAEKEWELPPDSDMDLNLIEQAPLTVAEKLQRDFLTEWRRVSKAPEALFFVQFEKGESYFHMHVLVETTGVKSMVLGRFLSQIREKLIQRIYRGIEPTLPNWFAVTKTRNGAGGGNKVVDESYIPNFLLPKTQPELQWAWTNMEQYLSACLNLTERKRLVAQHLT 4zq9 C 2.6 BS01 dna D 0 K101 M103 V104 R107 F108 Q111 R138 K92 M94 V95 R98 F99 Q102 R129 3.6.4.12 remove_due_to_license_issue P03132 26370092 1 ~ 21 PGFYEIVIKVPSDSDSFVNWVAEKEWELPPDSDMDLNLIEQAPLTVAEKLQRDFLTEWRRVSKAPEALFFVQFEKGESYFHMHVLVETTGVKSMVLGRFLSQIREKLIQRIYRGIEPTLPNWFAVTKTRNGAGGGNKVVDESYIPNFLLPKTQPELQWAWTNMEQYLSACLNLTERKRLVAQHLTHV 4zq9 C 2.6 BS02 dna E 0 S102 M103 G106 K136 R138 G142 G143 G144 N145 S93 M94 G97 K127 R129 G133 G134 G135 N136 3.6.4.12 remove_due_to_license_issue P03132 26370092 22 ~ 42 PGFYEIVIKVPSDSDSFVNWVAEKEWELPPDSDMDLNLIEQAPLTVAEKLQRDFLTEWRRVSKAPEALFFVQFEKGESYFHMHVLVETTGVKSMVLGRFLSQIREKLIQRIYRGIEPTLPNWFAVTKTRNGAGGGNKVVDESYIPNFLLPKTQPELQWAWTNMEQYLSACLNLTERKRLVAQHLTHV 4zqt A 1.981 BS01 4QP A 1 E319 V459 G460 A461 M462 E463 H496 E497 E519 Y575 Y580 E124 V264 G265 A266 M267 E268 H301 E302 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 remove_due_to_license_issue O96935 26406322 1101 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zs0 A 3.0 BS01 4QV A 1 L139 V147 A160 Y212 A213 G216 L263 D274 L13 V21 A34 Y86 A87 G90 L137 D148 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T161 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=2300nM O14965 27391133 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4zs2 A 2.16 BS02 FLU A 1 I85 P93 R96 L109 V228 S229 H231 I58 P66 R69 L82 V169 S170 H172 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 ic50=3.23uM remove_due_to_license_issue Q9C0B1 26457839 602 GSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKTEAEIAAACETFLKLNDYLQIETIQALEELAAKEKDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4zs3 A 2.45 BS02 A4F A 1 P93 R96 Y108 L109 V228 S229 H231 P66 R69 Y81 L82 V169 S170 H172 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 ic50=6.55uM remove_due_to_license_issue Q9C0B1 26457839 602 GSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKTEAEIAAACETFLKLNDYLQIETIQALEELAAKEKDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 4zsa A 2.0 BS01 4UT A 1 F489 A512 K514 E531 V561 Y563 A564 S565 G567 L630 F25 A48 K50 E67 V97 Y99 A100 S101 G103 L154 D623 A625 R627 N628 D641 D147 A149 R151 N152 D165 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=15nM remove_due_to_license_issue P11362 26080733 801 LPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 4zsf A 1.8 BS01 dna B 0 S78 N81 S82 K85 H89 K114 K203 S78 N81 S82 K85 H89 K114 K203 ? 0004519,0046872 remove_due_to_license_issue Q6UQ65 26240380 1 ~ 14 MNFFEYCISTYAKIFEETMNAVGDERVSQKKAIRDTMISAMREFPNVEAAEIWKAVYSAHMDRKSGIADPDIIQKVISAENSWKKSSGHAFEEMIKLLGNSSLEEYGMRILLQKDLNMMIENQEIANEPRDINWLKEQISSNVFDLYITVRNNDKEYVFGCIQSKTSIRDRVTRDREPSMKAMEAFFWSVAICLDGDFLKMPKFIAMVNGGTSNYRLNGWHGMYVFWDKPTIDRIYPIDINLELFVQHAREAAEDWLHRRQWFNYEWKAGQK 4zsg A 1.79 BS01 4QX A 1 Y66 I86 N95 R98 T99 E102 L103 I117 Y20 I40 N49 R52 T53 E56 L57 I71 D182 K184 S186 N187 D200 T224 D136 K138 S140 N141 D154 T178 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue Q13164 27139631 406 VTFDVGDEYEIIETIGNGAYGVVSSARRRLTGQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSPAEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARRE 4zsh A 1.8 BS02 4XW A 1 I268 A271 A272 Q275 F313 R316 L326 A327 C432 I23 A26 A27 Q30 F68 R71 L81 A82 C187 ? 0003677,0003707,0005634,0006355,0008270 Kd=90nM remove_due_to_license_issue P19793 26030625 501 DMPVERILEAELAVEPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 4zsj A 2.48 BS01 4R0 A 1 Y66 R98 T99 E102 L137 Y17 R49 T50 E53 L88 D182 K184 S186 N187 D200 T224 D133 K135 S137 N138 D151 T175 2.7.11.24 0004672,0004707,0005524,0006468 ic50=2.3uM remove_due_to_license_issue Q13164 27139631 405 DVGDEYEIIETIGNGAYGVVSSARRRLTGQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSPAEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARRE 4zsl A 2.25 BS01 4QZ A 1 Y66 K84 I86 N95 R98 T99 E102 I117 Y14 K32 I34 N43 R46 T47 E50 I65 D182 K184 S186 N187 D200 T224 D130 K132 S134 N135 D148 T172 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue Q13164 27139631 401 DEYEIIETIGNGAYGVVSSARRRLTGQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSPAEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARRE 4zsm A 1.96 BS01 4RW A 1 D32 Y71 D228 D36 Y75 D232 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=4000000nM P56817 26001341 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4zsp A 1.91 BS01 4RZ A 1 S10 G11 Q12 G13 D32 G34 Y71 W115 D228 G230 S15 G16 Q17 G18 D37 G39 Y76 W120 D233 G235 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 ic50=1.83uM remove_due_to_license_issue P56817 26001341 401 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4zsq A 2.3 BS01 4RX A 1 S10 G11 Q12 G13 D32 G34 Y71 W115 D228 G230 S14 G15 Q16 G17 D36 G38 Y75 W119 D232 G234 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=2.25uM remove_due_to_license_issue P56817 26001341 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4zsr A 1.65 BS01 4RY A 1 S10 G11 Q12 G13 D32 G34 W115 D228 G230 S15 G16 Q17 G18 D37 G39 W120 D233 G235 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 ic50=36.1uM remove_due_to_license_issue P56817 26001341 401 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 4zt8 A 1.98 BS01 CYT A 1 Y70 G109 I155 R163 Y70 G109 I155 R163 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 29124196 304 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 4ztl A 2.39 BS01 4S1 A 1 M192 V200 A211 Y262 Y264 M265 A315 L318 D329 M28 V36 A47 Y93 Y95 M96 A146 L149 D160 D311 K313 A315 N316 D329 T351 D142 K144 A146 N147 D160 T175 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=1.2uM remove_due_to_license_issue IC50=1193000nM Q9NWZ3 26288698 501 FHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4ztm A 2.66 BS01 4S2 A 1 M192 V200 A211 K213 V246 Y262 Y264 M265 P266 G268 D272 A315 L318 S328 M31 V39 A50 K52 V80 Y96 Y98 M99 P100 G102 D106 A149 L152 S162 D311 K313 A315 N316 D329 T351 D145 K147 A149 N150 D163 T182 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=25nM Q9NWZ3 26288698 501 DTRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4ztn A 2.23 BS01 4S3 A 1 M192 V200 A211 K213 Y262 Y264 M265 G268 D272 L318 M30 V38 A49 K51 Y96 Y98 M99 G102 D106 L152 D311 K313 A315 N316 D329 T351 D145 K147 A149 N150 D163 T181 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=19nM remove_due_to_license_issue IC50=19nM Q9NWZ3 26288698 501 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 4ztq A 2.8 BS01 4RM A 1 L139 G142 V147 K162 Q185 L210 E211 Y212 A213 L263 A273 D274 L13 G16 V21 K36 Q59 L84 E85 Y86 A87 L137 A147 D148 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T155 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=480nM O14965 27391133 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVGTLDYLPPEMIEGEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4ztr A 2.85 BS01 4RJ A 1 R137 L139 G140 G142 V147 A160 K162 L194 R195 L196 Y212 A213 G216 R220 L263 A273 F275 R11 L13 G14 G16 V21 A34 K36 L68 R69 L70 Y86 A87 G90 R94 L137 A147 F149 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T153 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue EC50=6000nM, IC50=2.0nM, Kd=5.0nM O14965 27391133 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4zts A 2.9 BS01 4RK A 1 R137 L139 G140 V147 Q185 L196 L210 A213 G216 L263 A273 F275 R11 L13 G14 V21 Q59 L70 L84 A87 G90 L137 A147 F149 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T153 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue IC50=25nM O14965 27391133 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 4zud A 2.8 BS01 OLM A 1 Y35 F77 W84 V108 S109 R167 F182 I288 Y129 F171 W178 V202 S203 R254 F269 I360 ? 0004930,0004945,0005506,0007186,0009055,0016020,0019229,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P30556 26420482 1201 DLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLILNSSDCPKAGRHNYIFVMIPTLYSIIFVVGIFGNSLVVIVIYFYMKLKTVASVFLLNLALADLCFLLTLPLWAVYTAMEYRWPFGNYLCKIASASVSFNLYASVFLLTCLSIDRYLAIVHPTMLVAKVTCIIIWLLAGLASLPAIIHRNVFFIENTNITVCAFHYESTLPIGLGLTKNILGFLFPFLIILTSYTLIWKALNDDIFKIIMAIVLFFFFSWIPHQIFTFLDVLIQLGIIRDCRIADIVDTAMPITICIAYFNNCLNPLFYGF 4zum A 1.42 BS02 FKS A 1 P156 H158 H159 G167 Y168 D195 H197 F225 E320 G321 Y323 P156 H158 H159 G167 Y168 D195 H197 F225 E320 G321 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 remove_due_to_license_issue Q48935 26200446 404 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zum B 1.42 BS02 FKS B 1 P156 H158 H159 G167 Y168 D195 H197 F225 E320 G321 Y323 P156 H158 H159 G167 Y168 D195 H197 F225 E320 G321 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 remove_due_to_license_issue Q48935 26200446 404 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zun A 1.4 BS01 SS9 A 1 H159 Y168 D195 F225 Y323 H159 Y168 D195 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=26uM remove_due_to_license_issue IC50=26000nM Q48935 26200446 401 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zun B 1.4 BS03 SS9 B 1 H159 Y168 D195 F225 Y323 H159 Y168 D195 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=26uM remove_due_to_license_issue IC50=26000nM Q48935 26200446 405 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zuo A 1.33 BS02 XS6 A 1 Y19 H158 H159 Y168 D195 H197 F225 Y323 Y19 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.39uM remove_due_to_license_issue IC50=390nM Q48935 26200446 404 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zuo B 1.33 BS02 XS6 B 1 Y19 H158 H159 Y168 D195 H197 F225 I291 Y323 Y19 H158 H159 Y168 D195 H197 F225 I291 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.39uM remove_due_to_license_issue IC50=390nM Q48935 26200446 404 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zup A 1.421 BS02 5XA A 1 E117 H158 H159 Y168 D195 H197 F225 Y323 E117 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.17uM remove_due_to_license_issue Q48935 26200446 405 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zup B 1.421 BS02 5XA B 1 E117 H158 H159 Y168 D195 H197 F225 Y323 E117 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.17uM remove_due_to_license_issue Q48935 26200446 405 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zuq A 1.22 BS01 6XA A 1 H158 H159 Y168 D195 H197 F225 Y323 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.13uM remove_due_to_license_issue Q48935 26200446 403 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zuq B 1.22 BS01 6XA B 1 E117 H158 H159 Y168 D195 H197 F225 Y323 E117 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.13uM remove_due_to_license_issue Q48935 26200446 403 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zur A 1.13 BS02 7XA A 1 H158 H159 Y168 D195 H197 F225 Y323 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.068uM remove_due_to_license_issue Q48935 26200446 404 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zur B 1.13 BS02 7XA B 1 H158 H159 Y168 D195 H197 F225 Y323 H158 H159 Y168 D195 H197 F225 Y323 3.5.1.-,3.5.1.48,3.5.1.62 0004407,0016787,0040029,0046872,0047609,0047611 ic50=0.068uM remove_due_to_license_issue Q48935 26200446 404 MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVLKVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAISPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQRLLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAGAGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPDYITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG 4zv1 A 1.52 BS01 ARG A 1 E17 F20 F58 A75 G76 M77 T78 R83 Q123 S126 T127 D167 E11 F14 F52 A69 G70 M71 T72 R77 Q117 S120 T121 D161 0015276,0016020,0030288,0071705 Kd=5.73uM remove_due_to_license_issue 26853627 301 HMRGTLRVGTEATFPPFGFKDENGKLVGFDIDLAKAIAKKLGVKVEFKPMDFDGIIPALQSGKIDVVIAGMTITEERKKQVDFSDPYFEAGQAIVVKKGNDSIKSLEDLKGKKVGVQLGSTSEQHVKKVAKDAGVKVKKFDNFSEAFQELKSGRVDAVVTDNAVALAYVKQNPNAGVKIVGETFSGEPYGIAVRKGNSELLEKINKALEEMKKDGTYDKIYEKWFG 4zv2 A 1.43 BS01 GLN A 1 E17 F20 F58 G76 M77 T78 R83 S126 T127 D167 E11 F14 F52 G70 M71 T72 R77 S120 T121 D159 0015276,0016020,0030288,0071705 Kd=1170uM remove_due_to_license_issue 26853627 301 HMRGTLRVGTEATFPPFGFKDENGKLVGFDIDLAKAIAKKLGVKVEFKPMDFDGIIPALQSGKIDVVIAGMTITEERKKQVDFSDPYFEAGQAIVVKKGNDSIKSLEDLKGKKVGVQLGSTSEQHVKKVAAGVKVKKFDNFSEAFQELKSGRVDAVVTDNAVALAYVKQNPNAGVKIVGETFSGEPYGIAVRKGNSELLEKINKALEEMKKDGTYDKIYEKWFGE 4zvi A 2.2 BS01 4S4 A 1 N46 E50 D73 R76 P79 V120 N31 E35 D58 R61 P64 V86 5.6.2.2 0003677,0003918,0005524,0006265 Kd=0.47uM remove_due_to_license_issue P0AES7 26126187 401 LDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLVGVSVVNALSQKLELVIQRGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYEGGIKAFVEYLNKNKTPIHPNIFYFSTEKDGIGVEVALQWNDGFQENIYCFTNNIPQRDGGTHLAGFRAAMTRTLNAYMDKEGYSKKAKVSATGDDAREGLIAVVSVKVPDPKFSSQTKDKLVSSEVKSAVEQQMNELLAEYLLENPTDAKIVVGKIIDAARAREAARRAREMT 4zw3 A 1.8 BS01 4S9 A 1 E319 V459 G460 A461 H496 E497 H500 E519 Y575 Y580 E124 V264 G265 A266 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=0.027uM remove_due_to_license_issue O96935 26807544 1101 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zw5 A 1.8 BS02 4SA A 1 Q317 E319 V459 G460 A461 H496 E497 H500 E519 Y575 Y580 M1034 Q122 E124 V264 G265 A266 H301 E302 H305 E324 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=37uM remove_due_to_license_issue O96935 26807544 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zw6 A 1.9 BS01 4SY A 1 E319 V459 G460 A461 R489 H496 E497 H500 E519 Y575 Y580 M1034 E124 V264 G265 A266 R294 H301 E302 H305 E324 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=1.9uM remove_due_to_license_issue O96935 26807544 1101 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zw7 A 1.95 BS02 4SZ A 1 T305 Q317 E319 A320 V459 G460 A461 H496 E497 H500 E519 E572 Y575 Y580 M1034 T109 Q121 E123 A124 V263 G264 A265 H300 E301 H304 E323 E376 Y379 Y384 M838 E463 H496 E497 H500 E519 E572 Y580 E267 H300 E301 H304 E323 E376 Y384 3.4.11.- 0006508,0008237,0008270 Ki=19uM remove_due_to_license_issue O96935 26807544 1102 KIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zw8 A 2.0 BS02 4T2 A 1 L304 T305 Q317 E319 A320 N458 V459 G460 A461 H496 E497 H500 E519 Y575 Y580 M1034 L109 T110 Q122 E124 A125 N263 V264 G265 A266 H301 E302 H305 E324 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=1.1uM remove_due_to_license_issue O96935 26807544 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zwx A 1.696 BS02 5KZ A 1 W5 H94 H119 V121 G132 L198 T199 P201 P202 W2 H91 H116 V118 G128 L194 T195 P197 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2nM remove_due_to_license_issue P00918 26203869 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4zwy A 1.5 BS02 4SN A 1 W5 F20 H94 H119 F131 L198 T199 P201 P202 W2 F17 H91 H116 F127 L194 T195 P197 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10nM remove_due_to_license_issue P00918 26203869 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4zwz A 1.62 BS02 510 A 1 H64 L91 Q92 H94 V121 L198 T199 H61 L88 Q89 H91 V118 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 26203869 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4zx0 A 1.6 BS02 5L2 A 1 W5 N62 H64 H94 V121 F131 L198 T199 T200 W2 N59 H61 H91 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 26203869 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4zx1 A 1.501 BS02 5L3 A 1 H64 Q67 Q92 H94 H119 L198 T199 P202 H61 Q64 Q89 H91 H116 L194 T195 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 26203869 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKQPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4zx3 A 2.0 BS02 4TK A 1 V459 G460 A461 E463 H496 E497 H500 E519 Y575 Y580 V264 G265 A266 E268 H301 E302 H305 E324 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=0.065uM remove_due_to_license_issue O96935 26807544 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zx4 A 1.9 BS01 4TL A 1 T305 Q317 E319 A320 V459 G460 A461 R489 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 R294 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=0.078uM remove_due_to_license_issue O96935 26807544 1101 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zx5 A 1.95 BS02 4TM A 1 E319 V459 G460 A461 R489 H496 E497 H500 E519 E572 Y575 Y580 E124 V264 G265 A266 R294 H301 E302 H305 E324 E377 Y380 Y385 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=0.64uM remove_due_to_license_issue O96935 26807544 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zx6 A 2.05 BS02 4U6 A 1 V459 G460 A461 E463 H496 E497 H500 E519 E572 Y575 Y580 M1034 V263 G264 A265 E267 H300 E301 H304 E323 E376 Y379 Y384 M838 E463 H496 E497 H500 E519 E572 Y580 E267 H300 E301 H304 E323 E376 Y384 3.4.11.- 0006508,0008237,0008270 Ki=5.4uM remove_due_to_license_issue O96935 26807544 1102 KIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 4zx8 A 2.7 BS01 4TY A 1 K374 D379 F398 N457 D459 E461 L487 T488 G489 K290 D295 F314 N373 D375 E377 L403 T404 G405 K386 R463 K302 R379 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26807544 1001 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zx8 F 2.7 BS01 4TY F 1 D379 D459 E461 L487 T488 G489 D289 D369 E371 L397 T398 G399 K386 R463 K296 R373 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26807544 1001 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zx9 A 2.6 BS01 4TK A 1 D379 D459 E461 L487 T488 G489 S554 D295 D375 E377 L403 T404 G405 S470 K386 R463 K302 R379 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26807544 1001 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zx9 F 2.6 BS01 4TK F 1 D379 D459 E461 L487 G489 D287 D367 E369 L395 G397 K386 R463 K294 R371 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26807544 1001 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKNGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zxx H 2.6 BS01 4T0 H 1 L41 H57 K60A D189 S190 K192 S195 S214 W215 G216 G219 L25 H41 K45 D186 S187 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 remove_due_to_license_issue Ki=8.0nM P08709 26151189 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4zxy H 2.06 BS01 4T1 H 1 H57 K60A G97 D189 S190 K192 S195 S214 W215 G216 G219 H41 K45 G85 D182 S183 K185 S188 S207 W208 G209 G211 3.4.21.21 0004252,0006508 Ki=400nM remove_due_to_license_issue Ki=400nM P08709 26151189 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 4zy0 A 2.2 BS01 4TM A 1 K374 D379 D459 E461 L487 T488 G489 L492 A577 K290 D295 D375 E377 L403 T404 G405 L408 A493 K386 R463 K302 R379 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.0091uM remove_due_to_license_issue A0A024V0B1 26807544 1001 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zy0 F 2.2 BS01 4TM F 1 K374 D379 D459 E461 L487 T488 G489 L492 A577 K281 D286 D366 E368 L394 T395 G396 L399 A484 K386 R463 K293 R370 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.0091uM remove_due_to_license_issue A0A024V0B1 26807544 1001 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKNGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zy1 A 2.5 BS01 4U5 A 1 K374 D379 K386 F398 D459 E461 L487 T488 G489 L492 A577 K290 D295 K302 F314 D375 E377 L403 T404 G405 L408 A492 K386 R463 K302 R379 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.0072uM remove_due_to_license_issue A0A024V0B1 26807544 1001 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zy1 F 2.5 BS01 4U5 F 1 K374 D379 K386 D459 E461 L487 T488 G489 L492 A577 K282 D287 K294 D367 E369 L395 T396 G397 L400 A485 K386 R463 K294 R371 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.0072uM remove_due_to_license_issue A0A024V0B1 26807544 1001 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zy2 A 2.1 BS04 4TL A 1 K374 D379 M392 D459 E461 L487 T488 G489 L492 A577 F583 K290 D295 M308 D375 E377 L403 T404 G405 L408 A493 F499 K386 R463 K302 R379 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.06uM remove_due_to_license_issue A0A0L7M119 26807544 1008 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zy2 F 2.1 BS04 4TL F 1 K374 D379 M392 D459 E461 L487 T488 G489 L492 A577 F583 K283 D288 M301 D368 E370 L396 T397 G398 L401 A486 F492 K386 R463 K295 R372 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=0.06uM remove_due_to_license_issue A0A0L7M119 26807544 1009 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zy4 A 2.6 BS01 4T3 A 1 A297 E345 Y346 L347 A348 G350 L396 A49 E92 Y93 L94 A95 G97 L143 N389 K391 D393 N394 D407 P416 T427 N136 K138 D140 N141 D154 P163 T174 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=22nM Q13153 26030457 601 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT 4zy5 A 2.35 BS01 4T5 A 1 V284 A297 L347 D393 L396 V33 A46 L88 D134 L137 N389 K391 D393 N394 D407 P416 T427 N130 K132 D134 N135 D148 P157 T168 2.7.11.1 0004672,0005524,0006468 Ki=26nM remove_due_to_license_issue Q13153 26030457 601 EEILEKLRSIVSVGDPKKKYTRFKIGQGASGTVYTAMDVATGQEVAIKQQPKKELIINEILVMRENKNPNIVNYLDSYLELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 4zy6 A 2.15 BS01 4T6 A 1 A297 E345 Y346 L347 D393 N394 L396 A47 E87 Y88 L89 D135 N136 L138 N389 K391 D393 N394 D407 P416 T427 N131 K133 D135 N136 D149 P158 T169 2.7.11.1 0004672,0005524,0006468 Ki=5nM remove_due_to_license_issue Q13153 26030457 601 EEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQPKKELIINEILVMRENKNPNIVNYLDSYLVELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 4zyc A 1.95 BS01 4SS A 1 K51 L54 F55 G58 F86 V93 H96 K27 L30 F31 G34 F62 V69 H72 2.3.2.27 0005634,0043066,0051726 ic50=0.38uM remove_due_to_license_issue Q00987 26141769 201 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLV 4zyc A 1.95 BS02 4SS A 2 E95 R97 K98 T101 E71 R73 K74 T77 2.3.2.27 0005634,0043066,0051726 ic50=0.38uM remove_due_to_license_issue Q00987 26141769 202 ETLVRPKPELLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLV 4zyf A 1.8 BS01 4T4 A 1 L54 F55 G58 I61 M62 Y67 Q72 F86 V93 Y100 L37 F38 G41 I44 M45 Y50 Q55 F69 V76 Y83 2.3.2.27 0005634,0043066,0051726 Kd=2.3nM remove_due_to_license_issue IC50=0.8nM, Ki=1.3nM, Kd=2.3nM Q00987 26181851 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4zyi A 1.67 BS01 4TH A 1 Q24 L54 F55 G58 M62 Y67 Q72 F86 H96 I99 Q5 L34 F35 G38 M42 Y47 Q52 F66 H76 I79 2.3.2.27 0005634,0043066,0051726 ic50=0.008uM remove_due_to_license_issue Q00987 26181851 201 PASEQETLVRPKPLLLKLLKSVGQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 4zyq A 2.6 BS01 4U6 A 1 K374 D379 G390 M392 F398 D459 E461 L487 T488 G489 L492 K288 D293 G304 M306 F312 D373 E375 L401 T402 G403 L406 K386 R463 K300 R377 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26807544 1001 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zyq F 2.6 BS01 4U6 F 1 K374 D379 G390 S391 M392 F398 D459 E461 L487 G489 L492 A577 K282 D287 G298 S299 M300 F306 D367 E369 L395 G397 L400 A485 K386 R463 K294 R371 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26807544 1001 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 4zyr A 3.312 BS01 9PG A 1 M23 R144 C148 W151 E269 H322 M18 R139 C143 W146 E248 H301 ? 0005351,0005515,0005886,0008643,0015293,0015528,0015767,0016020,0022857,0030395,0034219,0055085,1902600 remove_due_to_license_issue P02920 26157133 501 NTNFWMFGLFFFFYFFIMGAYFPFFPIWLHDINHISKSDTWIIFAAISLFSLLFQPLFGLLSDKLGLRKYLLWIITGMLVMFAPFFIFIFGPLLQYNILVGSIVGGIYLGFCFNAGAPAVEAFIEKVSRRSNFEFGRARMFGCVGWALCASIVGIMFTINNQFVFWLGSGCALILAVLLFFAKTDAFSLKLALELFRQPKLWFLSLYVIGVSCTYDVFDQQFANFFTSFFATGEQGTRVFWYVTTMGELLNASIMFFAPLIINRIGGKNALLLAGTIMSVRIIGSSFATSALEVVILKTLHMFEVPFLLVGCFKYITSQFEVRFSATIYLVCFCFFKQLAMIFMSVLAGNMYESIGFQGAYLVLGLVALGFTLISVFTLSGPGPLSL 4zyt A 1.702 BS02 3Y9 A 1 K844 H865 F895 M896 R897 I898 L899 V946 A947 V950 K37 H58 F88 M89 R90 I91 L92 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=17nM remove_due_to_license_issue IC50=6.8nM P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zyu A 1.95 BS02 3YA A 1 L892 F895 M896 R897 I898 L899 N913 V946 A947 V950 L85 F88 M89 R90 I91 L92 N106 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=1067nM remove_due_to_license_issue P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zyv A 2.053 BS02 G71 A 1 K844 F895 M896 R897 I898 L899 V946 A947 V950 K37 F88 M89 R90 I91 L92 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=22nM remove_due_to_license_issue P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWVK 4zyw A 2.05 BS02 G94 A 1 F895 M896 R897 I898 L899 S925 V946 A947 V950 F88 M89 R90 I91 L92 S118 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=68nM remove_due_to_license_issue P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zyx A 1.65 BS02 3YB A 1 R871 L892 F895 M896 R897 I898 L899 G924 V946 A947 E948 V950 R64 L85 F88 M89 R90 I91 L92 G117 V139 A140 E141 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=7nM remove_due_to_license_issue IC50=0.600000nM P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zyy A 1.85 BS02 3YC A 1 R871 L892 F895 M896 R897 I898 L899 G924 V946 A947 E948 V950 R64 L85 F88 M89 R90 I91 L92 G117 V139 A140 E141 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=9nM remove_due_to_license_issue IC50=2.03nM P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zyz A 1.6 BS02 3YD A 1 R871 L892 F895 M896 R897 I898 L899 V946 A947 E948 V950 R64 L85 F88 M89 R90 I91 L92 V139 A140 E141 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=67nM remove_due_to_license_issue IC50=2.9nM P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zz0 A 1.65 BS02 3YE A 1 F895 M896 R897 I898 L899 V946 A947 E948 V950 F88 M89 R90 I91 L92 V139 A140 E141 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=99nM remove_due_to_license_issue IC50=5.5nM P22102 27439469 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zz1 A 1.351 BS02 3YF A 1 R871 F895 M896 R897 I898 L899 G924 S925 V946 A947 V950 R64 F88 M89 R90 I91 L92 G117 S118 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=13nM remove_due_to_license_issue IC50=2.4nM, Ki=13nM P22102 26317331 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zz2 A 1.451 BS02 3YG A 1 R871 F895 M896 R897 I898 L899 G924 S925 V946 A947 V950 R64 F88 M89 R90 I91 L92 G117 S118 V139 A140 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=9.1nM remove_due_to_license_issue Ki=9.1nM, IC50=2.6nM P22102 26317331 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zz3 A 2.504 BS01 4DW A 1 L892 F895 M896 R897 I898 L899 N913 V946 A947 E948 V950 L85 F88 M89 R90 I91 L92 N106 V139 A140 E141 V143 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=1000nM remove_due_to_license_issue P22102 26317331 1101 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVQKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 4zzx A 1.65 BS01 FSU A 1 H428 G429 G454 Y462 F463 S470 Y473 H198 G199 G224 Y232 F233 S240 Y243 S470 Y473 E558 S240 Y243 E326 2.4.2.-,2.4.2.30 0003950 Kd=0.125uM remove_due_to_license_issue Kd=125nM Q9UGN5 26222319 1584 ESQLDLRVQELIKLICNVQAMEEMMMEMKYNTKKAPLGKLTVAQIKAGYQSLKKIEDCIRAGQHGRALMEACNEFYTRIPHDFGLRTPPLIRTQKELSEKIQLLEALGDIEIAIKLVKTELQSPEHPLDQHYRNLHCALRPLDHESYEFKVISQYLQSTHAPTHSDYTMTLLDLFEVEKDGEKEAFREDLHNRMLLWHGSRMSNWVGILSHGLRIAPPEAPITGYMFGKGIYFADMSSKSANYCFASRLKNTGLLLLSEVALGQCNELLEANPKAEGLLQGKHSTKGLGKMAPSSAHFVTLNGSTVPLGPASDTGILNGYTLNYNEYIVYNPNQVRMRYLLKVQFNFLQLW 4zzy A 2.2 BS01 D7N A 1 S328 I331 Q332 H428 G429 G454 Y455 Y462 F463 A464 K469 S470 Y473 S98 I101 Q102 H198 G199 G224 Y225 Y232 F233 A234 K239 S240 Y243 S470 Y473 E558 S240 Y243 E326 2.4.2.-,2.4.2.30 0003950 Kd=1.389uM remove_due_to_license_issue Kd=1389nM Q9UGN5 26222319 1584 ESQLDLRVQELIKLICNVQAMEEMMMEMKYNTKKAPLGKLTVAQIKAGYQSLKKIEDCIRAGQHGRALMEACNEFYTRIPHDFGLRTPPLIRTQKELSEKIQLLEALGDIEIAIKLVKTELQSPEHPLDQHYRNLHCALRPLDHESYEFKVISQYLQSTHAPTHSDYTMTLLDLFEVEKDGEKEAFREDLHNRMLLWHGSRMSNWVGILSHGLRIAPPEAPITGYMFGKGIYFADMSSKSANYCFASRLKNTGLLLLSEVALGQCNELLEANPKAEGLLQGKHSTKGLGKMAPSSAHFVTLNGSTVPLGPASDTGILNGYTLNYNEYIVYNPNQVRMRYLLKVQFNFLQLW 4zzz A 1.9 BS01 FSU A 1 H862 G863 Y896 F897 S904 Y907 H198 G199 Y232 F233 S240 Y243 S904 Y907 E988 S240 Y243 E324 2.4.2.-,2.4.2.30 0003950 Kd=0.087uM remove_due_to_license_issue Kd=87nM, IC50=5300nM P09874 26222319 2019 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSDKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKTSLW 5a00 A 2.75 BS01 D7N A 1 Q759 V762 H862 G863 Y889 Y896 F897 A898 K903 S904 Y907 Q93 V96 H192 G193 Y219 Y226 F227 A228 K233 S234 Y237 S904 Y907 E988 S234 Y237 E318 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Kd=8.6nM, IC50=40nM P09874 26222319 2012 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 5a09 A 1.81 BS02 JJD A 1 H57 Y94 L99 D102 V190 C191 F192 S195 A213 S214 F215 V216 H41 Y80 L85 D88 V168 C169 F170 S173 A187 S188 F189 V190 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G167 C169 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=3.5nM remove_due_to_license_issue IC50=3.5nM P08246 26083237 1244 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a0a E 1.78 BS02 JJS E 1 H57 Y94 L99 D102 V190 C191 F192 D194 S195 A213 S214 F215 V216 H41 Y80 L85 D88 V166 C167 F168 D170 S171 A185 S186 F187 V188 F192 G193 D194 S195 G196 F168 G169 D170 S171 G172 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 Ki=15nM remove_due_to_license_issue IC50=15nM, Ki=15nM P08246 26083237 1244 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a0b A 2.23 BS02 JJX A 1 H57 Y94 L99 D102 V190 C191 F192 S195 A213 S214 F215 V216 H41 Y80 L85 D88 V165 C166 F167 S170 A184 S185 F186 V187 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G164 C166 F167 G168 D169 S170 G171 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=5nM remove_due_to_license_issue P08246 26083237 1001 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a0c A 2.1 BS02 JJV A 1 H57 Y98 L103 D106 V197 C198 F199 S202 A220 S221 F222 V223 H41 Y80 L85 D88 V168 C169 F170 S173 A187 S188 F189 V190 H57 D106 G196 C198 F199 G200 D201 S202 G203 H41 D88 G167 C169 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=0.54nM remove_due_to_license_issue IC50=<0.300000nM P08246 26083237 1001 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a14 A 2.0 BS01 LQ5 A 1 A31 E51 L54 F80 F82 L83 L124 H125 L143 A144 D145 F146 F152 A31 E49 L52 F78 F80 L81 L122 H123 L141 A142 D143 F144 F150 D127 K129 Q131 N132 D145 T165 D125 K127 Q129 N130 D143 T153 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue Kd=53nM, IC50=>1.0e+4nM P24941 26158339 1297 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 5a14 A 2.0 BS02 LQ5 A 2 F213 K237 S239 P241 K242 W243 F201 K225 S227 P229 K230 W231 D127 K129 Q131 N132 D145 T165 D125 K127 Q129 N130 D143 T153 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue Kd=53nM, IC50=>1.0e+4nM P24941 26158339 1298 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 5a2s A 2.65 BS01 OTF A 1 P676 E677 R681 H802 H803 F812 D840 H842 F871 G974 P24 E25 R29 H150 H151 F160 D188 H190 F219 G322 3.5.1.98 remove_due_to_license_issue Kd=20nM P56524 26819662 1 TTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPANRQKLDSKKLLGSLASVFVRLPCGGVGVDSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELDPLPEKVLQQRPNANAVRSMEKVMEIHSKYWRCLQ 5a3n A 2.0 BS05 LQT A 1 Y425 W486 Y488 F496 H499 E501 K517 W519 H587 V600 N601 Y128 W189 Y191 F199 H202 E204 K220 W222 H290 V303 N304 G481 Y488 H499 E501 H587 A599 G184 Y191 H202 E204 H290 A302 1.14.11.67 ic50=19nM remove_due_to_license_issue IC50=19nM Q9UGL1 28262558 1759 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKRDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGKIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAE 5a3o A 1.6 BS03 MMA A 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 27308201 201 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 5a3o B 1.6 BS03 MMA B 1 N21 S22 S23 D96 D99 D101 D104 N21 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 27308201 201 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 5a3o B 1.6 BS04 DH6 B 1 D96 G97 T98 D96 G97 T98 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 27308201 202 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 5a3q A 3.05 BS02 DL5 A 1 V185 S186 K205 M361 T441 F487 M494 K515 R560 V185 S186 K205 M361 T441 F487 M494 K515 R560 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 27050689 1002 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 5a3r A 3.05 BS01 DL5 A 1 R174 E439 T441 E442 F487 K492 K515 G516 R560 C561 L562 R174 E439 T441 E442 F487 K492 K515 G516 R560 C561 L562 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 27050689 1000 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 5a3s A 3.3 BS02 128 A 1 V185 V187 K205 M361 T441 F487 K515 R560 V185 V187 K205 M361 T441 F487 K515 R560 D351 D703 D707 D351 D703 D707 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 27050689 1002 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGHFNDPVHGGSWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 5a3t A 1.9 BS02 MMK A 1 Y425 W486 Y488 F496 H499 E501 K517 W519 H587 V600 N601 Y128 W187 Y189 F197 H200 E202 K218 W220 H288 V301 N302 G481 Y488 H499 E501 H587 A599 G182 Y189 H200 E202 H288 A300 1.14.11.67 Ki=0.001uM remove_due_to_license_issue Q9UGL1 27214403 1756 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKRDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAE 5a3u A 3.3 BS02 R8J A 1 Y303 H313 D315 R322 R383 W389 Y99 H109 D111 R118 R179 W185 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue Q9GZT9 26147748 1421 QTKPLPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYLTGEKGVRVELNKPSD 5a3u C 3.3 BS02 R8J C 1 Y303 H313 D315 R383 W389 Y97 H107 D109 R177 W183 1.14.11.29 0005506,0016705,0031418 remove_due_to_license_issue Q9GZT9 26147748 1407 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYLT 5a3w A 2.0 BS03 PD2 A 1 Y425 Y488 F496 H499 E501 K517 W519 H587 Y129 Y190 F198 H201 E203 K219 W221 H289 G481 Y488 H499 E501 H587 A599 G183 Y190 H201 E203 H289 A301 1.14.11.67 Ki=0.39uM remove_due_to_license_issue IC50=3000nM Q9UGL1 27214403 1757 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKARDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAE 5a3x A 2.26 BS01 QIV A 1 F170 A186 K188 F238 L241 L294 D307 F37 A53 K55 F105 L108 L161 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 ic50=0.8uM remove_due_to_license_issue Q13627 27736065 1482 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 5a46 A 2.63 BS01 38O A 1 L484 V561 E562 Y563 A564 G567 L630 L21 V98 E99 Y100 A101 G104 L157 D623 A625 R627 N628 D641 D150 A152 R154 N155 D168 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 26203596 1769 ELPEDPRWELPRDRLVLGKPLGEGCFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 5a4c A 2.09 BS01 XOJ A 1 L484 G485 A512 K514 E531 M535 I545 V561 Y563 A564 L630 D641 F642 L21 G22 A47 K49 E66 M70 I80 V96 Y98 A99 L165 D176 F177 D623 A625 R627 N628 D641 D158 A160 R162 N163 D176 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=5.7nM remove_due_to_license_issue P11362 26203596 1774 ELPEDPRWELPRDRLVLGKPLGEFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 5a4e A 2.68 BS01 7QQ A 1 F238 L294 D307 F105 L161 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Q13627 27736065 1482 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 5a4l A 2.73 BS01 ZC3 A 1 A186 K188 F238 L294 D307 A53 K55 F105 L161 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Q13627 27736065 1481 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 5a4q A 2.37 BS01 Y3L A 1 I165 A186 F238 M240 L241 L294 I32 A53 F105 M107 L108 L161 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 ic50=2.9uM remove_due_to_license_issue Q13627 27736065 1482 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 5a4t A 2.15 BS01 AJG A 1 I165 A186 L241 I32 A53 L108 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 ic50=1.3uM remove_due_to_license_issue Q13627 27736065 1482 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 5a54 A 2.63 BS01 5PW A 1 I165 F238 L241 L294 V306 I32 F105 L108 L161 V173 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Q13627 27736065 1482 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 5a5d A 1.74 BS02 5LC A 1 Q98 R118 R205 T226 H227 R249 L253 Y288 Q77 R97 R184 T205 H206 R228 L232 Y267 ? 0006826,0030288,0030313,0046872,1901678 Kd<10nM remove_due_to_license_issue Q0P8Q4 28383577 500 AMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5a5o A 2.04 BS01 J5I A 1 V1008 V1018 N1064 I1074 V30 V40 N86 I96 3.6.1.- remove_due_to_license_issue IC50=<1000000nM Q6PL18 26155854 2112 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a5p A 2.03 BS01 JTF A 1 V1008 V1013 V1018 Y1063 N1064 D1071 I1074 V30 V35 V40 Y85 N86 D93 I96 3.6.1.- ic50=0.1mM remove_due_to_license_issue IC50=100000nM Q6PL18 26155854 2111 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a5q A 1.97 BS01 6XC A 1 V1008 E1017 N1064 D1071 I1074 V30 E39 N86 D93 I96 3.6.1.- Kd=21uM remove_due_to_license_issue IC50=15849nM, Kd=21000nM Q6PL18 26155854 2111 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a5r A 2.01 BS01 NP8 A 1 V1013 E1017 V1018 N1064 D1071 I1074 V35 E39 V40 N86 D93 I96 3.6.1.- ic50=1.3uM remove_due_to_license_issue IC50=3981nM Q6PL18 26155854 2111 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a5s A 1.36 BS01 NP8 A 1 W81 P82 L92 N140 I146 W40 P41 L51 N99 I105 ? ic50=1.3uM remove_due_to_license_issue IC50=15849nM O60885 26155854 1170 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHKFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5a5v A 2.04 BS02 PXJ A 1 V97 Q98 R118 R205 T226 H227 R249 L253 Y288 V76 Q77 R97 R184 T205 H206 R228 L232 Y266 ? 0006826,0030288,0030313,0046872,1901678 Kd=33nM remove_due_to_license_issue Q0P8Q4 28383577 500 AMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5a5z A 2.6 BS03 WJZ A 1 D124 H189 N220 H250 D88 H153 N184 H214 H120 H122 D124 H189 C208 K211 N220 H250 H84 H86 D88 H153 C172 K175 N184 H214 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue C7C422 25815530 304 QQMETGDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLRLE 5a69 A 2.2 BS01 OGN A 1 R94 D222 E223 W266 W306 Y308 Y309 W339 W373 D375 R88 D216 E217 W255 W267 Y269 Y270 W298 W332 D334 ? 0004553,0004563,0005975,0015929,0016231,0016787 Ki=1.1nM remove_due_to_license_issue A0A0H2US73 26491009 1627 RFTGLSLKQTQAIEVLKHISLPVEVAVTQSDQASISIEGEEGHYQLTYRKPHQLYRALSLLVTVLADKVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNRLLMCQHLERVLDIADKYGFHCQMWSDMFDRVTLVYWDYYQDSEEKYNRNFRNHHKIDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLPGNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFYADKDFAATTANQWHTIATASTIYTT 5a6a A 2.69 BS01 NGT A 1 R94 D222 E223 W266 W306 Y308 W339 W373 D375 R89 D217 E218 W261 W301 Y303 W334 W368 D370 3.2.1.52 0004553,0004563,0005975,0015929,0016231,0016787 remove_due_to_license_issue A0A0H2US73 26491009 1628 TGLSLKQTQAIEVLKGHISLPDVEVAVTQSDQASISIEGEGHYQLTYRKPHQLYRALSLLVTVLAEADKVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNGVVDRSLLMCQHLERVLDIADKYGFHCQMWSDMFFKLMSADGQYDRDVEIPEETRVYLDRLKDRVTLVYWDYYQDSEEKYNRNFRNHHKISHDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLPGNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFYAKDFAATTANQWHTIATASTIYTT 5a6a B 2.69 BS01 NGT B 1 R94 W266 W306 Y308 W339 W373 D375 R92 W264 W285 Y287 W318 W352 D354 3.2.1.52 0004553,0004563,0005975,0015929,0016231,0016787 remove_due_to_license_issue A0A0H2US73 26491009 1627 VRFTGLSLKQTQAIEVLKGHISLPDVEVAVTQSDQASISIEGEEGHYQLTYRKPHQLYRALSLLVTVLAEADVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNGVVDRSLLMCQHLERVLDIADKYGFHCQMWSDMFTRVYLDRLKDRVTLVYWDYYQDSEEKYNRNFRNHHKISHDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFAATTANQWHTIATASTIYTT 5a6b A 1.77 BS01 OAN A 1 R94 W266 W306 Y308 Y309 W339 W373 D375 R95 W267 W292 Y294 Y295 W325 W359 D361 ? 0004553,0004563,0005975,0015929,0016231,0016787 Ki=7.9nM remove_due_to_license_issue A0A0H2US73 26491009 1627 SMVRFTGLSLKQTQAIEVLKGHISLPDVEVAVTQSDQASISIEGEEGHYQLTYRKPHQLYRALSLLVTVLAEADKVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNGVVDRSLLMCQHLERVLDIADKYGFHCQMWSDMFFPEETRVYLDRLKDRVTLVYWDYYQDSEEKYNRNFRNHHKISHDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLPGNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFYADKDFAATTANQWHTIATASTIYTT 5a6b B 1.77 BS01 OAN B 1 R94 W266 W306 Y308 Y309 W339 W373 D375 R98 W270 W297 Y299 Y300 W330 W364 D366 ? 0004553,0004563,0005975,0015929,0016231,0016787 Ki=7.9nM remove_due_to_license_issue A0A0H2US73 26491009 1627 SMASMVRFTGLSLKQTQAIEVLKGHISLPDVEVAVTQSDQASISIEGEEGHYQLTYRKPHQLYRALSLLVTVLAEADKVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNGVVDRSLLMCQHLERVLDIADKYGFHCQMWSDMFFKLPEETRVYLDRLKDRVTLVYWDYYQDSEEKYNRNFRNHHKISHDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLPGNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFYADKDFAATTANQWHTIATASTIYTT 5a6h A 1.57 BS02 OE2 A 1 H94 H96 F131 L198 T199 T200 P201 P202 H93 H95 F129 L196 T197 T198 P199 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=88nM remove_due_to_license_issue Ki=88nM P00918 27172398 1264 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5a6h A 1.57 BS03 OE2 A 2 H4 W5 D19 H3 W4 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=88nM remove_due_to_license_issue Ki=88nM P00918 27172398 1265 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5a6h A 1.57 BS04 OE2 A 3 H3 W5 F20 P201 P202 H2 W4 F19 P199 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=88nM remove_due_to_license_issue Ki=88nM P00918 27172398 1266 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5a6i A 1.86 BS01 TCW A 1 K15 L17 A108 S117 T118 K6 L8 A99 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=56nM remove_due_to_license_issue Kd=56nM P02766 26902880 1124 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVIT 5a6k A 2.1 BS01 NSG A 1 R94 D222 E223 W266 W306 Y308 W339 W373 D375 R94 D222 E223 W266 W306 Y308 W339 W373 D375 3.2.1.52 0004553,0004563,0005975,0015929,0016231,0016787 Ki=1130nM remove_due_to_license_issue A0A0H2US73 26491009 1627 MVRFTGLSLKQTQAIEVLKGHISLPDVEVAVTQSDQASISIEGEEGHYQLTYRKPHQLYRALSLLVTVLAEADKVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNGVVDRSLLMCQHLERVLDIADKYGFHCQMWSDMFFKLMSADGQYDRDVEIPEETRVYLDRLKDRVTLVYWDYYQDSEEKYNRNFRNHHKISHDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLPGNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFYADKDFAATTANQWHTIATASTIYTT 5a6k B 2.1 BS01 NSG B 1 R94 D222 E223 W266 W306 Y308 W339 W373 D375 R93 D221 E222 W265 W305 Y307 W338 W372 D374 3.2.1.52 0004553,0004563,0005975,0015929,0016231,0016787 Ki=1130nM remove_due_to_license_issue A0A0H2US73 26491009 1627 VRFTGLSLKQTQAIEVLKGHISLPDVEVAVTQSDQASISIEGEEGHYQLTYRKPHQLYRALSLLVTVLAEADKVEIEEQAAYEDLAYMVDCSRNAVLNVASAKQMIEILALMGYSTFELYMEDTYQIEGQPYFGYFRGAYSAEELQEIEAYAQQFDVTFVPCIQTLAHLSAFVKWGVKEVQELRDVEDILLIGEEKVYDLIDGMFATLSKLKTRKVNIGMDEAHLVGLGRYLILNGVVDRSLLMCQHLERVLDIADKYGFHCQMWSDMFFKLMSADGQYDRDVEIPEETRVYLDRLKDRVTLVYWDYYQDSEEKYNRNFRNHHKISHDLAFAGGAWKWIGFTPHNHFSRLVAIEANKACRANQIKEVIVTGWGDNGGETAQFSILPSLQIWAELSYRNDLDGLSAHFKTNTGLTVEDFMQIDLANLLPDLPGNLSGINPNRYVFYQDILCPILDQHMTPEQDKPHFAQAAETLANIKEKAGNYAYLFETQAQLNAILSSKVDVGRRIRQAYQADDKESLQQIARQELPELRSQIEDFHALFSHQWLKENKVFGLDTVDIRMGGLLQRIKRAESRIEVYLAGQLDRIDELEVEILPFTDFYADKDFAATTANQWHTIATASTIYTT 5a6n A 1.7 BS01 U7E A 1 K42 D161 K35 D154 D139 K141 E143 N144 D161 T180 D132 K134 E136 N137 D154 T173 2.7.11.1 0004672,0005524,0006468 ic50=52uM remove_due_to_license_issue O43293 26486226 300 MVEDHYEMGEELGSGQFAIVRKCRQKGTGKEYAAKFIKKRRLSSSRRGVSREEIEREVNILREIRHPNIITLHDIFENKTDVVLILELVSGGELFDFLAEKESLTEDEATQFLKQILDGVHYLHSKRIAHFDLKPENIMLLDKNVPNPRIKLIDFGIAHKIEAGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGETKQETLTNISAVNYDFDEEYFSNTSELAKDFIRRLLVKDPKRRMTIAQSLEHSWIKAI 5a6x A 1.55 BS03 MFU A 1 S22 A23 D96 D99 D101 D104 S22 A23 D96 D99 D101 D104 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 30155149 201 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5a6x B 1.55 BS03 MFU B 1 S22 A23 D96 D99 D101 D104 S22 A23 D96 D99 D101 D104 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 30155149 201 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5a72 A 2.6 BS01 dna C 0 D23 C25 Q29 R43 F49 Q50 S51 R73 M77 T139 D140 G141 R144 T145 D18 C20 Q24 R38 F44 Q45 S46 R68 M72 T134 D135 G136 R139 T140 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 501 ~ 524 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLNLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVV 5a72 A 2.6 BS02 dna D 0 R33 D35 Y36 L37 Q41 R71 R73 N74 G84 K120 K142 K143 R28 D30 Y31 L32 Q36 R66 R68 N69 G79 K115 K137 K138 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 601 ~ 624 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLNLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVV 5a72 B 2.6 BS01 dna C 0 R33 D35 Y36 L37 Q41 R71 R73 N74 G84 K142 R28 D30 Y31 L32 Q36 R66 R68 N69 G79 K137 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 501 ~ 524 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLNLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVVS 5a72 B 2.6 BS02 dna D 0 A22 D23 C25 Q29 R43 F49 Q50 S51 R73 M77 T139 D140 G141 R144 T145 I146 A17 D18 C20 Q24 R38 F44 Q45 S46 R68 M72 T134 D135 G136 R139 T140 I141 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 601 ~ 624 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLNLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVVS 5a77 A 2.5 BS01 dna C 0 D23 Q50 S51 M77 D18 Q45 S46 M72 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 501 ~ 514 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLQLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVV 5a77 A 2.5 BS02 dna D 0 D35 Y36 Q41 T69 R71 R73 N74 G84 K120 D30 Y31 Q36 T64 R66 R68 N69 G79 K115 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 601 ~ 614 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLQLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVV 5a77 A 2.5 BS03 dna E 0 A22 D23 G24 Q29 R33 R43 F49 R73 K102 T139 D140 G141 K143 R144 T145 I146 A17 D18 G19 Q24 R28 R38 F44 R68 K97 T134 D135 G136 K138 R139 T140 I141 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 515 ~ 524 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLQLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVV 5a77 B 2.5 BS01 dna C 0 R33 D35 Y36 L37 Q41 R71 R73 N74 D75 G84 K120 R28 D30 Y31 L32 Q36 R66 R68 N69 D70 G79 K115 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 501 ~ 514 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLQLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVVS 5a77 B 2.5 BS02 dna D 0 D23 Q50 S51 M77 D18 Q45 S46 M72 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 601 ~ 614 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLQLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVVS 5a77 B 2.5 BS03 dna F 0 A22 G24 C25 N27 R33 R43 F49 R73 K102 T139 G141 K143 R144 I146 A17 G19 C20 N22 R28 R38 F44 R68 K97 T134 G136 K138 R139 I141 A22 D23 A17 D18 3.1.-.- 0004519,0006314,0009507 remove_due_to_license_issue P56347 26363068 615 ~ 624 NFHDQLKFAWLAGFVDADGCINAQIVSREDYLLKYQVRVSLTVFQSTTQHFILLDIQKILGCGTVRKRNDGMSEFCVVGGTSLQTTLEKLLPYLQLKRAQAKLVLQIIKKLPNTKDPSVLMEAALLADKVGLLTDGKKRTILAENVRECLKKLGHVVS 5a7b A 1.4 BS02 KMN A 1 L145 V147 D148 T150 P151 C220 E221 P222 P223 L50 V52 D53 T55 P56 C125 E126 P127 P128 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=271uM remove_due_to_license_issue P04637 26378745 1001 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5a7c A 1.9 BS01 5D4 A 1 W332 F334 V338 N391 W28 F30 V34 N87 ? ic50=0.00018M remove_due_to_license_issue Q15059 26941288 500 MGKLSEHLRYCDSILREMLSKKHAAYAWPFYKPVDAEALELHDYHDIIKHPMDLSTVKRKMDGREYPDAQGFAADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMP 5a7i A 2.89 BS01 B6K A 1 M258 H565 H566 H567 H568 H569 H570 M1 H308 H309 H310 H311 H312 H313 3.1.3.36 0016791,0046856,0052745 remove_due_to_license_issue P32019 26854536 1572 MYTYIQNFRFFAGTYNVNGQSPKECLRLWLSNGIQAPDVYCVGFQELDLSKEAFFFHDTPKEEEWFKAVSEGLHPDAKYAKVKLIRLVGIMLLLYVKQEHAAYISEVEAETVGTGIMGRMGNKGGVAIRFQFHNTSICVVNSHLAAHIEEYERRNQDYKDICSRMQFCQPDPSLPPLTISNHDVILWLGDLNYRIEELDVEKVKKLIEEKDFQMLYAYDQLKIQVAAKTVFEGFTEGELTFQPTYKYDTGSDDWDTSEKCRAPAWCDRILWKGKNITQLSYQSHMALKTSDHKPVSSVFDIGVRVVAHHHHHH 5a7j A 2.9 BS01 K2Y A 1 M258 H565 H566 M1 H308 H309 3.1.3.36 0016791,0046856,0052745 remove_due_to_license_issue IC50=6300nM P32019 26854536 1568 MYTYIQNFRFFAGTYNVNGQSPKECLRLWLSNGIQAPDVYCVGFQELDLSKEAFFFHDTPKEEEWFKAVSEGLHPDAKYAKVKLIRLVGIMLLLYVKQEHAAYISEVEAETVGTGIMGRMGNKGGVAIRFQFHNTSICVVNSHLAAHIEEYERRNQDYKDICSRMQFCQPDPSLPPLTISNHDVILWLGDLNYRIEELDVEKVKKLIEEKDFQMLYAYDQLKIQVAAKTVFEGFTEGELTFQPTYKYDTGSDDWDTSEKCRAPAWCDRILWKGKNITQLSYQSHMALKTSDHKPVSSVFDIGVRVVAHH 5a7y A 2.5 BS01 SAH A 1 L158 D159 P160 I179 G180 I209 I225 L159 D160 P161 I180 G181 I189 I205 2.1.1.218 0005737,0008033,0008168,0008175,0030488,0032259,0160106 remove_due_to_license_issue Q4J894 26673726 1291 HMTLAKVFSQKLRELGISSIYIGHERPSLQSLAIKMLLKNYGLVEERREGMLITQDHGIKLISGKGTETSRYTFRKGGKKVSIHLPEYPKMVIDLGLFEFLNEEEKEKTLLQVDLCLSVIRKFLWDGNLTVVGKADYVLGRANIVQSLSLSDEDNPVILDPYGDVVATDQILRDHNVFVIGGSFPRVKIQLRGSIIGVPDEINKILEIILRVKELDQSLEEAIISLQSKSDKISRLLHDVQLYGMEVLEEEARWLRADDKVIEIVRSRLG 5a81 A 2.03 BS01 78J A 1 N1064 G1070 D1071 I1074 N86 G92 D93 I96 3.6.1.- Kd=2.9uM remove_due_to_license_issue IC50=2512nM, Kd=2300nM Q6PL18 26230603 2111 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a82 A 1.86 BS01 YEJ A 1 V1008 V1013 N1064 G1070 D1071 I1074 R1077 V30 V35 N86 G92 D93 I96 R99 3.6.1.- ic50=2.51uM remove_due_to_license_issue Kd=1100nM, IC50=2512nM Q6PL18 26230603 2112 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a83 A 2.09 BS01 YD3 A 1 V1008 V1013 D1014 E1017 V1018 N1064 G1070 D1071 I1074 R1077 V30 V35 D36 E39 V40 N86 G92 D93 I96 R99 3.6.1.- ic50=0.158uM remove_due_to_license_issue IC50=158nM, Kd=60nM Q6PL18 26230603 1112 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5a8x A 2.23 BS02 IUY A 1 H57 Y94 L99 D102 V190 C191 F192 S195 A213 S214 F215 V216 H41 Y80 L85 D88 V165 C166 F167 S170 A184 S185 F186 V187 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G164 C166 F167 G168 D169 S170 G171 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=6.5nM remove_due_to_license_issue P08246 26333652 1001 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a8y A 1.9 BS02 VBM A 1 H57 Y94 L99 D102 V190 C191 F192 S195 A213 S214 F215 V216 R217 H41 Y80 L85 D88 V166 C167 F168 S171 A185 S186 F187 V188 R189 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G165 C167 F168 G169 D170 S171 G172 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=0.17nM remove_due_to_license_issue P08246 26333652 1001 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a8z A 2.0 BS03 IUL A 1 H57 Y94 L99 D102 V190 C191 F192 S195 A213 S214 F215 V216 H41 Y80 L85 D88 V165 C166 F167 S170 A184 S185 F186 V187 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G164 C166 F167 G168 D169 S170 G171 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=28nM remove_due_to_license_issue IC50=28nM P08246 26333652 1001 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5a9u A 1.6 BS01 5P8 A 1 L1122 G1123 A1148 L1196 M1199 G1202 N1254 L1256 G1269 D1270 Y1401 L30 G31 A45 L93 M96 G99 N151 L153 G166 D167 Y292 D1249 A1251 R1253 N1254 D1270 D146 A148 R150 N151 D167 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.08nM remove_due_to_license_issue Q9UM73 26698910 2402 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVPLQVAVKTLPEVYSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5aa8 A 1.86 BS01 5P8 A 1 L1122 G1123 A1148 L1196 F1198 M1199 G1202 N1254 L1256 G1269 D1270 Y1401 L30 G31 A45 L93 F95 M96 G99 N151 L153 G166 D167 Y292 D1249 A1251 R1253 N1254 D1270 L1291 D146 A148 R150 N151 D167 L182 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=8.6nM remove_due_to_license_issue Q9UM73 26698910 2402 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVPLQVAVKTLPEVYSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLEFMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5aa9 A 1.93 BS01 5P8 A 1 L1122 A1148 L1196 F1198 M1199 G1202 N1254 L1256 G1269 D1270 Y1401 L30 A48 L96 F98 M99 G102 N154 L156 G169 D170 Y295 D1249 A1251 R1253 N1254 D1270 L1291 D149 A151 R153 N154 D170 L185 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=6.4nM remove_due_to_license_issue Q9UM73 26698910 2402 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLEFMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5aaa A 1.73 BS01 VGH A 1 L1122 A1148 M1199 A1200 G1202 N1254 L1256 G1269 I1399 E1400 L30 A48 M99 A100 G102 N154 L156 G169 I293 E294 D1249 A1251 R1253 N1254 D1270 L1291 D149 A151 R153 N154 D170 L185 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.38nM remove_due_to_license_issue IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 26698910 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLEFMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 5aab A 2.2 BS01 VGH A 1 L1122 A1148 M1199 A1200 G1202 N1254 L1256 G1269 Y1401 L30 A46 M97 A98 G100 N152 L154 G167 Y293 D1249 A1251 R1253 N1254 D1270 L1291 D147 A149 R151 N152 D168 L183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=0.88nM remove_due_to_license_issue IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 26698910 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGGEVYEGQVPLQVAVKTLPEVYSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLEFMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5aac A 1.7 BS01 VGH A 1 A1148 M1199 A1200 G1202 N1254 L1256 G1269 D1270 Y1401 A45 M96 A97 G99 N151 L153 G166 D167 Y292 D1249 A1251 R1253 N1254 D1270 D146 A148 R150 N151 D167 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=1.3nM remove_due_to_license_issue IC50=20nM, Ki=8.2nM, EC50=22840nM, Kd=3.3nM Q9UM73 26698910 9000 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVPLQVAVKTLPEVYSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5aad A 3.1 BS01 5GX A 1 L139 G140 K141 G142 V147 A160 L194 Y212 A213 P214 G216 L263 L13 G14 K15 G16 V21 A34 L68 Y86 A87 P88 G90 L137 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 26296477 1389 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHATLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 5aae A 3.11 BS01 7HD A 1 L139 G140 G145 V147 K162 A213 G216 L263 L14 G15 G20 V22 K37 A88 G91 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 26296477 1389 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 5aaf A 2.78 BS01 NL4 A 1 R137 L139 G140 V147 Y212 A213 G216 T217 R220 L263 R12 L14 G15 V22 Y87 A88 G91 T92 R95 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 26296477 1001 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 5aag A 2.85 BS01 6F2 A 1 L139 G140 A160 Y212 A213 G216 L263 L13 G14 A34 Y86 A87 G90 L137 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 26296477 1389 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 5aan A 1.6 BS04 XOC A 1 W30 Y52 F85 W103 L182 W28 Y50 F83 W101 L180 ? 0005509,0005515,0005737,0007268,0007269,0007528,0008021,0008048,0009966,0016192,0046872,0046928 Kd=71uM remove_due_to_license_issue Kd=71000nM Q9VWX8 28119500 1189 KKNSKLKQDTIDRLTTDTYFTEKEIRQWHKGFLKDCPNGLLTEQGFIKIYKQFFPDGDPSKFASLVFRVFDENNDGAIEFEEFIRALSITSRGNLDEKLHWAFRLYDVDNDGYITREEMYNIVDAIYQMVGQQPQTEDENTPQKRVDKIFDQMDKNHDDRLTLEEFREGSKADPRMVQALSLG 5ab9 A 1.36 BS02 92O A 1 L145 V147 T150 C220 P222 P223 T230 L50 V52 T55 C125 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=470uM remove_due_to_license_issue P04637 26636255 1292 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5ab9 A 1.36 BS03 92O A 2 T150 P151 P152 P153 C220 T55 P56 P57 P58 C125 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=470uM remove_due_to_license_issue P04637 26636255 1293 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5aba A 1.62 BS02 UL7 A 1 L145 V147 D148 T150 C220 E221 P222 P223 T230 L50 V52 D53 T55 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=1040uM remove_due_to_license_issue P04637 26636255 1291 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5abe A 2.0 BS01 XQO A 1 Y137 K166 D242 D243 Y282 W337 V342 D344 Y345 Y135 K164 D240 D241 Y280 W335 V340 D342 Y343 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=890uM remove_due_to_license_issue Q89ZI2 26545827 1716 VSLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISNIKNLPLQVKANRVLISPKWAAGNSVEIELDAIYPGENIQINFLEISTDGKEWKTVDLKLSAGLQKAPVKFVRFTNLRQFVLTIEK 5abf A 2.1 BS01 XRJ A 1 G135 Y137 K166 D242 D243 Y282 W286 T310 W337 D344 Y345 G132 Y134 K163 D239 D240 Y279 W283 T307 W334 D341 Y342 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=14uM remove_due_to_license_issue Q89ZI2 26545827 1717 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISNNLPLQVKANRVLISVEIELDAIYPGENIQIGRLEISTDGKEWKTVDLKSAGLQKAPVKFVRFVLTIEK 5abg A 2.0 BS01 V0N A 1 G135 D242 D243 Y282 V314 W337 N339 D344 G132 D239 D240 Y279 V311 W334 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=9nM remove_due_to_license_issue Q89ZI2 26545827 1717 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISIKNLPLQVKANRVLISPVEIELDAIYPGENIQINEISTDGKEWKLSAGLQKAPVKFVRFLRQFVLTIEK 5abh A 1.95 BS01 YWN A 1 G135 Y137 D242 D243 Y282 W286 W337 N339 D344 G132 Y134 D239 D240 Y279 W283 W334 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 Ki=1.7nM remove_due_to_license_issue Q89ZI2 26545827 1717 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISNVKNLPLQVKANRVLISPANEVEIELDAIYPGENIQINFGKDAPGRLEISTDGKEWKTVDLSAGLQKAPVKFVRFTFVLTIEK 5abp A 1.8 BS01 GLA A 1 K10 E14 W16 D89 D90 R151 M204 N232 K9 E13 W15 D88 D89 R150 M203 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.23uM remove_due_to_license_issue P02924 2818726 307 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMMAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 5abw A 1.6 BS02 WQQ A 1 H57 L99 C191 F192 S195 A213 S214 F215 V216 R217 H41 L85 C166 F167 S170 A184 S185 F186 V187 R188 H57 D102 G189 C191 F192 G193 D194 S195 G196 H41 D88 G164 C166 F167 G168 D169 S170 G171 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 ic50=17nM remove_due_to_license_issue IC50=17nM P08246 26358162 1001 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 5acb C 2.7 BS01 5I1 C 1 I733 V741 A754 K756 F813 M816 D819 L866 Q1037 C1039 I18 V26 A39 K41 F98 M101 D104 L151 Q322 C324 D859 K861 S863 N864 D877 S889 T898 D144 K146 S148 N149 D162 S174 T183 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue Q9NYV4 27571479 2000 ESDWGKRCVDKFDIIGIIGEGTYGQVYKAKDKDTGELVALKKVRLDNEKEGFPITAIREIKILRQLIHRSVVNMKEIVTDKQDALDFKKDKGAFYLVFEYMDHDLMGLLESGLVHFSEDHIKSFMKQLMEGLEYCHKKNFLHRDIKCSNILLNNSGQIKLADFGLARLYNSEESRPYTNKVITLWYRPPELLLGEERYTPAIDVWSCGCILGELFTKKPIFQANLELAQLELISRLCGSPCPAVWPDVIKLPYFNTMKPKKQYRRRLREEFSFIPSAALDLLDHMLTLDPSKRCTAEQTLQSDFLKDVELSKMAPPDLPHWQDCH 5acw A 1.8 BS03 RHU A 1 W87 H118 D120 H196 C221 H263 W57 H86 D88 H149 C168 H210 H116 H118 D120 H196 C221 Y224 N233 H263 H84 H86 D88 H149 C168 Y171 N180 H210 3.5.2.6 Kd=145uM remove_due_to_license_issue Q9K2N0 26477515 1298 GEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5acw A 1.8 BS04 RHU A 2 A135 Y137 H170 A102 Y104 H123 H116 H118 D120 H196 C221 Y224 N233 H263 H84 H86 D88 H149 C168 Y171 N180 H210 3.5.2.6 Kd=145uM remove_due_to_license_issue Q9K2N0 26477515 1299 GEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5acx A 1.8 BS03 WL3 A 1 F61 Y67 W87 H118 D119 D120 H196 C221 R228 N233 H263 F32 Y37 W57 H86 D87 D88 H149 C168 R175 N180 H210 H116 H118 D120 H196 C221 Y224 N233 H263 H84 H86 D88 H149 C168 Y171 N180 H210 3.5.2.6 Kd=9uM remove_due_to_license_issue Q9K2N0 26477515 1298 GEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5acx B 1.8 BS03 WL3 B 1 Y67 W87 D119 D120 H196 C221 R228 N233 H263 Y37 W57 D87 D88 H149 C168 R175 N180 H210 H116 H118 D120 H196 C221 Y224 N233 H263 H84 H86 D88 H149 C168 Y171 N180 H210 3.5.2.6 Kd=9uM remove_due_to_license_issue Q9K2N0 26477515 1298 GEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5acy A 2.01 BS01 9S3 A 1 W81 P82 L92 Y139 I146 W40 P41 L51 Y98 I105 ? Kd=6.4nM remove_due_to_license_issue IC50=398nM O60885 26392221 1172 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ad1 A 1.32 BS02 8LC A 1 Q98 R118 K121 R205 T226 H227 R249 L253 Y288 Q78 R98 K101 R185 T206 H207 R229 L233 Y268 ? 0006826,0030288,0030313,0046872,1901678 Kd=58nM remove_due_to_license_issue Q0P8Q4 28383577 500 PAMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5adq A 2.1 BS02 A95 A 1 H1031 P1034 F1035 I1039 F1044 D1045 H1048 G1053 Y1060 Y1071 H80 P83 F84 I88 F93 D94 H97 G102 Y109 Y120 2.4.2.-,2.4.2.30 0003950 ic50=2.01uM remove_due_to_license_issue IC50=1995nM Q9H2K2 26706174 2117 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 5adr A 2.1 BS01 QS5 A 1 H1031 P1034 F1035 A1038 F1044 D1045 H1048 G1053 Y1060 Y1071 I1075 H80 P83 F84 A87 F93 D94 H97 G102 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=2.3uM remove_due_to_license_issue IC50=2291nM Q9H2K2 26706174 2115 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 5ads A 1.8 BS02 QNS A 1 H1031 P1034 F1035 I1039 F1044 D1045 H1048 I1051 G1053 I1059 Y1060 Y1071 I1075 H80 P83 F84 I88 F93 D94 H97 I100 G102 I108 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=2.15uM remove_due_to_license_issue IC50=2150nM Q9H2K2 26706174 2117 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 5adt A 2.15 BS02 1TC A 1 H1031 P1034 F1044 D1045 H1048 I1051 Y1060 Y1071 I1075 H80 P83 F93 D94 H97 I100 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=2.23uM remove_due_to_license_issue IC50=2230nM Q9H2K2 26706174 2116 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 5aeh A 1.85 BS01 8IR A 1 S1033 F1035 A1038 G1043 D1045 H1048 Y1060 Y1071 I1075 S82 F84 A87 G92 D94 H97 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=0.037uM remove_due_to_license_issue IC50=37nM Q9H2K2 26706174 1170 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSKMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5ael A 2.6 BS01 QAF A 1 Y99 D103 D107 R112 A169 Q172 K212 D255 K269 Y89 D93 D97 R102 A159 Q162 K202 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 remove_due_to_license_issue Q86C09 26392508 1368 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5ael B 2.6 BS01 QAF B 1 Y99 D103 D107 R112 A169 Q172 K212 D255 K269 Y89 D93 D97 R102 A159 Q162 K202 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 2.5.1.10 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 remove_due_to_license_issue Q86C09 26392508 1368 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5aen A 1.864 BS01 DP8 A 1 Q136 A137 Y267 W311 F314 P374 A377 Y378 Q134 A135 Y265 W309 F312 P372 A375 Y376 E271 H295 E296 H299 E318 D375 Y383 E269 H293 E294 H297 E316 D373 Y381 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=0.06uM remove_due_to_license_issue Kd=270nM, IC50=60nM, Ki=160nM P09960 25625859 611 IVDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 5aep A 1.95 BS01 QUP A 1 L855 G856 K857 G861 S862 V863 A880 M929 Y931 L932 N981 L983 D994 L16 G17 K18 G22 S23 V24 A41 M87 Y89 L90 N139 L141 D152 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S174 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.068uM remove_due_to_license_issue IC50=68nM O60674 25882525 2000 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 5aes A 2.751 BS02 5B0 A 1 D25 D27 S58 N59 N60 Y146 H178 D26 D28 S59 N60 N61 Y147 H179 3.1.3.16,3.1.3.74 0000287,0004721,0004722,0005515,0005737,0005829,0005856,0005886,0005911,0006338,0006357,0006470,0007088,0015629,0016311,0016787,0016791,0017018,0030027,0030496,0030836,0031072,0031247,0031258,0032154,0032361,0032465,0032587,0033192,0033883,0042803,0042995,0046872,0070938,0071318,0098794,0098978,0099159,0140791,0180004,0180005,0180006,0180007,0180008,1990439 remove_due_to_license_issue IC50=1300000nM P60487 25783190 306 GMARCERLRGAALRDVLGQAQGVLFDCDGVLWNGERIVPGAPELLQRLARAGKNTLFVSNNSRRARPELALRFARLGFAGLRAEQLFSSALCAARLLRQRLPGPPDASGAVFVLGGEGLRAELRAAGLRLAGDPGEDPRVRAVLVGYDEQFSFSRLTEACAHLRDPDCLLVATDRDPWHPLSDGSRTPGTGSLAAAVETASGRQALVVGKPSPYMFQCITEDFSVDPARTLMVGDRLETDILFGHRCGMTTVLTLTGVSSLEEAQAYLTAGQRDLVPHYYVESIADLMEGL 5aes B 2.751 BS02 5B0 B 1 D25 D27 S58 N59 N60 Y146 H178 D25 D27 S58 N59 N60 Y146 H178 3.1.3.16,3.1.3.74 0000287,0004721,0004722,0005515,0005737,0005829,0005856,0005886,0005911,0006338,0006357,0006470,0007088,0015629,0016311,0016787,0016791,0017018,0030027,0030496,0030836,0031072,0031247,0031258,0032154,0032361,0032465,0032587,0033192,0033883,0042803,0042995,0046872,0070938,0071318,0098794,0098978,0099159,0140791,0180004,0180005,0180006,0180007,0180008,1990439 remove_due_to_license_issue IC50=1300000nM P60487 25783190 306 MARCERLRGAALRDVLGQAQGVLFDCDGVLWNGERIVPGAPELLQRLARAGKNTLFVSNNSRRARPELALRFARLGFAGLRAEQLFSSALCAARLLRQRLPGPPDASGAVFVLGGEGLRAELRAAGLRLAGDPGEDPRVRAVLVGYDEQFSFSRLTEACAHLRDPDCLLVATDRDPWHPLSDGSRTPGTGSLAAAVETASGRQALVVGKPSPYMFQCITEDFSVDPARTLMVGDRLETDILFGHRCGMTTVLTLTGVSSLEEAQAYLTAGQRDLVPHYYVESIADLMEGLE 5afj A 2.2 BS01 42R A 1 L6 L10 L63 L6 L10 L63 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=42uM remove_due_to_license_issue P36544,P58154 25918415 1205 EFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afj A 2.2 BS02 42R A 2 Y91 K141 Y91 K141 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=42uM remove_due_to_license_issue P36544,P58154 25918415 1206 EFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afj B 2.2 BS01 42R A 2 L36 Q37 I165 L37 Q38 I166 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=42uM remove_due_to_license_issue P36544,P58154 25918415 1206 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afj B 2.2 BS03 42R B 1 L6 E9 L10 L63 L7 E10 L11 L64 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=42uM remove_due_to_license_issue P36544,P58154 25918415 1205 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afj B 2.2 BS04 42R B 2 Y91 N92 K141 Y184 Y92 N93 K142 Y185 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=42uM remove_due_to_license_issue P36544,P58154 25918415 1206 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afk A 2.381 BS02 5VU A 1 L6 Y7 L10 V11 L63 V76 S77 V78 S82 L7 Y8 L11 V12 L64 V77 S78 V79 S83 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=132uM remove_due_to_license_issue P36544,P58154 25918415 1207 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afk A 2.381 BS04 5VU E 1 Q3 Q75 V76 S77 L104 Q4 Q76 V77 S78 L105 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=132uM remove_due_to_license_issue P36544,P58154 25918415 1207 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afk B 2.381 BS03 5VU B 1 Q3 L6 Y7 V11 V76 S77 V78 S82 Q4 L7 Y8 V12 V77 S78 V79 S83 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=132uM remove_due_to_license_issue P36544,P58154 25918415 1207 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afl E 2.385 BS03 FHV E 1 Q3 Y7 L10 Y14 V76 V78 S82 Q4 Y8 L11 Y15 V77 V79 S83 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=398uM remove_due_to_license_issue P36544,P58154 25918415 1207 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afm A 2.85 BS02 9Z0 A 1 F31 L54 L88 A90 P97 I119 Q121 F142 F32 L55 L89 A91 P98 I120 Q122 F143 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue P36544,P58154 25918415 1207 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afm B 2.85 BS03 9Z0 B 1 F52 L54 L88 A90 P97 I119 Q121 F142 F53 L55 L89 A91 P98 I120 Q122 F143 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue P36544,P58154 25918415 1208 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKGRS 5afn A 2.149 BS02 OJD A 1 M56 V85 L88 A90 P97 Q121 M57 V86 L89 A91 P98 Q122 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=34uM remove_due_to_license_issue P36544,P58154 25918415 1215 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5afn B 2.149 BS03 OJD B 1 M56 P86 L88 A90 P97 Q121 F142 M57 P87 L89 A91 P98 Q122 F143 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 ic50=34uM remove_due_to_license_issue P36544,P58154 25918415 1217 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVFWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWVPDLAAYNAISKPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKGRS 5afv A 2.25 BS01 JH5 A 1 D306 Q308 Y333 Y354 W423 Y440 D203 Q205 Y230 Y251 W320 Y337 2.7.1.32,2.7.1.82 Kd=2.6uM remove_due_to_license_issue P35790 27490389 1463 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5afx A 2.39 BS04 PVZ A 1 Y99 D103 M106 R112 D165 A169 Q172 K212 Y216 D255 K269 Y89 D93 M96 R102 D155 A159 Q162 K202 Y206 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=1.2uM remove_due_to_license_issue Q86C09 26392508 1371 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5afx A 2.39 BS05 PVZ B 1 N131 L134 N121 L124 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=1.2uM remove_due_to_license_issue Q86C09 26392508 1371 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5afx B 2.39 BS01 PVZ A 1 N131 L134 N121 L124 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=1.2uM remove_due_to_license_issue Q86C09 26392508 1371 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5afx B 2.39 BS04 PVZ B 1 Y99 D103 R112 T168 A169 Q172 K212 Y216 D255 K269 Y89 D93 R102 T158 A159 Q162 K202 Y206 D245 K259 K47 H98 D103 D107 R112 D175 K212 F251 D255 D256 K47 H88 D93 D97 R102 D165 K202 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016740,0016765,0045337,0046872 ic50=1.2uM remove_due_to_license_issue Q86C09 26392508 1371 MPMQMFMQVYDEIQMFLLEELELKFDMDPNRVRYLRKMMDTTCLGGKYNRGLTVIDVAESLLSDGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5agi A 1.47 BS01 ANZ A 1 T316 L317 R318 V403 L404 K407 V412 D418 S419 K483 T38 L39 R40 V125 L126 K129 V134 D140 S141 K205 0000166,0002161,0004823,0005524,0006418,0006429 remove_due_to_license_issue 26172575 600 GYVGIKIRLTDVAPQAQELFKKESLDVKENKVYLVAATLRPETMYGQTCCFVSPKIDYGVFDAGNGDYFITTERAFKNMSFQNLTPKRGYYKPLFTINGKTLIGSRIDAPYAVNKNLRVLPMETVLATKGTGVVTCVPSDSPDDFVTTRDLANKPEYYGIEKDWVQTDIVPIVHTEKYGDKCAEFLVNDLKIQSPKDSVQLANAKELAYKEGFYNGTMLIGKYKGDKVEDAAPKVKQDLIDEGLAFVYNEPE 5agj A 2.0 BS01 ANZ A 1 A315 T316 L317 R318 L404 K407 V412 D418 S419 K483 Y487 A37 T38 L39 R40 L126 K129 V134 D140 S141 K205 Y209 0000166,0002161,0004823,0005524,0006418,0006429 remove_due_to_license_issue 26172575 1817 GYVGIKIRLTDVAPQAQELFKKESLDVKENKVYLVAATLRPETMYGQTCCFVSPKIDYGVFDAGNGDYFITTERAFKNMSFQNLTPKRGYYKPLFTINGKTLIGSRIDAPYAVNKNLRVLPMETVLATKGTGVVTCVPSDSPDDFVTTRDLANKPEYYGIEKDWVQTDIVPIVHTEKYGDKCAEFLVNDLKIQSPKDSVQLANAKELAYKEGFYNGTMLIGKYKGDKVEDAKPKVKQDLIDEGLAFVYDE 5agr A 1.3 BS01 A52 A 1 F335 T336 T337 R338 V431 L432 Y435 I440 M441 D447 R449 D450 F16 T17 T18 R19 V108 L109 Y112 I117 M118 D124 R126 D127 6.1.1.4 0000166,0002161,0004823,0005524,0006418,0006429 remove_due_to_license_issue P9WFV1 27503647 1514 GAVALFSARAVDIEVFTTRPDTLFGATYLVLAPEHDLVDELVAASWPAGVNPLWTYGGGTPGEAIAAYRRAIAAKSDLERQKTGVFLGSYAINPANGEPVPIFIADYVLAGYGTGAIMAVPGHDQRDWDFARAFGLPIVEVIAGGNISESAYTGDGILVNSDYLNGMSVPAAKRAIVDRLESAGRGRARI 5ags A 1.47 BS01 38Y A 1 F335 T336 T337 R338 T341 V431 L432 Y435 I440 M441 V443 H446 D447 R449 D450 F16 T17 T18 R19 T22 V110 L111 Y114 I119 M120 V122 H125 D126 R128 D129 6.1.1.4 0000166,0002161,0004823,0005524,0006418,0006429 remove_due_to_license_issue P9WFV1 27503647 1514 GAVALFSARAVDIEVFTTRPDTLFGATYLVLAPEHDLVDELVAASWPAGVNPLWTYGGGTPGEAIAAYRRAIAAKSDLERQEEKTGVFLGSYAINPANGEPVPIFIADYVLAGYGTGAIMAVPGHDQRDWDFARAFGLPIVEVIAGGNISESAYTGDGILVNSDYLNGMSVPAAKRAIVDRLESAGRGRARI 5agt A 1.45 BS01 A2H A 1 F335 T336 T337 R338 V431 L432 Y435 I440 M441 V443 H446 D447 R449 D450 F16 T17 T18 R19 V108 L109 Y112 I117 M118 V120 H123 D124 R126 D127 6.1.1.4 0000166,0002161,0004823,0005524,0006418,0006429 remove_due_to_license_issue P9WFV1 27503647 1514 GAVALFSARAVDIEVFTTRPDTLFGATYLVLAPEHDLVDELVAASWPAGVNPLWTYGGGTPGEAIAAYRRAIAAKSDLERQKTGVFLGSYAINPANGEPVPIFIADYVLAGYGTGAIMAVPGHDQRDWDFARAFGLPIVEVIAGGNISESAYTGDGILVNSDYLNGMSVPAAKRAIVDRLESAGRGRARI 5ahj H 2.8 BS01 7IM H 1 T1 T21 G47 A49 T1 T21 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 26050527 1223 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 5ahj H 2.8 BS02 7IM N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 26050527 1198 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICD 5ahj I 2.8 BS01 7IM H 1 D124 L125 D124 L125 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 26050527 1223 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 5ahj Z 2.8 BS01 7IM Y 1 H108 P127 H108 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 26050527 1215 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 5ahu B 2.69 BS01 G76 B 1 Y99 D103 R112 A169 Q172 K212 T213 D255 K269 Y26 D30 R39 A96 Q99 K139 T140 D182 K196 H98 D103 D107 R112 D175 K212 F251 D255 D256 H25 D30 D34 R39 D102 K139 F178 D182 D183 ? 0004659,0008299,0016765 remove_due_to_license_issue Q86C09 26392508 1368 DGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5ahu D 2.69 BS01 G76 D 1 Y99 D103 D107 R112 A169 Q172 K212 D255 K269 Y26 D30 D34 R39 A96 Q99 K139 D182 K196 H98 D103 D107 R112 D175 K212 F251 D255 D256 H25 D30 D34 R39 D102 K139 F178 D182 D183 ? 0004659,0008299,0016765 remove_due_to_license_issue Q86C09 26392508 1368 DGARRKRVLHDACVCGWMIEFLQAHYLVEDDIMDNSVTRRGKPCWYRHPDVTVQCAINDGLLLKSWTHMMAMHFFADRPFLQDLLCRFNRVDYTTAVGQLYDVTSMFDSNKLDPDVSQPTTTDFAEFTLSNYKRIVKYKTAYYTYLLPLVMGLIVSEALPTVDMGVTEELAMLMGEYFQVQDDVMDCFTPPERLGKVGTDIQDAKCSWLAVTFLAKASSAQVAEFKANYGSGDSEKVATVRRLYEEADLQGDYVAYEAAVAEQVKELIEKLRLCSPGFAASVETLWGKTYKRQK 5ahw A 2.15 BS01 CMP A 1 G10 T11 D12 S16 S17 A40 P95 V113 G114 V116 V129 T146 G9 T10 D11 S15 S16 A39 P73 V91 G92 V94 V107 T124 ? 0000166 Kd=0.000000064M remove_due_to_license_issue A0QYW6 25802331 1148 SAYQTVVVGTDGSDSSLRAVDRAGQIAAASNAKLIIATAYFPAPIYAILREANDRAKAAGATDIEERPVVGAPVDALVELADEVKADLLVVGNVGLSTIAGRLLGSVPANVARRSKTDVLIVHTS 5ai0 A 1.75 BS01 JF6 A 1 M339 Y343 A365 M469 N472 W473 M338 Y342 A364 M468 N471 W472 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=206.4uM remove_due_to_license_issue IC50=206400nM P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ai1 A 2.103 BS01 EQU A 1 Y16 N40 F86 M90 D103 Y15 N39 F83 M87 D96 Y16 N40 D100 D103 Y15 N39 D93 D96 5.3.3.1 0004769,0008202,0016853 Kd=0.34uM remove_due_to_license_issue P07445 25947291 1128 NLPTAQEVQGLMARYIELVDVGDIEAIVQMFADDATVENPFGQPPIHGREQIAAFFRQGLGGVRACLTGPVRASHNGCGAMPFRVEMVPCALDVIDVMRFDEHGRIQTMQAFWSEVNLSV 5ai4 A 1.93 BS01 4VY A 1 D335 W336 M339 Y383 Q384 Y466 M469 D334 W335 M338 Y382 Q383 Y465 M468 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=331.7uM remove_due_to_license_issue P34913 25931264 1555 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ai4 A 1.93 BS02 4VY A 2 F267 D335 Y383 M419 Y466 H524 W525 F266 D334 Y382 M418 Y465 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=331.7uM remove_due_to_license_issue P34913 25931264 1556 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ai5 A 2.28 BS01 BSU A 1 F267 D335 W336 Y383 Q384 Y466 F266 D334 W335 Y382 Q383 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.093uM remove_due_to_license_issue IC50=390nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ai6 A 2.3 BS01 4XH A 1 F267 L408 M419 V498 H524 W525 F266 L407 M418 V497 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=40.19uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDA 5ai8 A 1.85 BS01 K2T A 1 M419 H524 W525 M411 H516 W517 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F259 H326 D327 W328 N351 N370 Y375 Y458 D488 H516 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=125.6uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ai9 A 1.8 BS01 K78 A 1 D335 W336 M339 Y383 Q384 M419 Y466 D496 V498 L499 H524 D334 W335 M338 Y382 Q383 M418 Y465 D495 V497 L498 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.244uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aia A 2.26 BS01 KWB A 1 M419 F497 V498 H524 W525 M418 F496 V497 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=6.268uM remove_due_to_license_issue P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aib A 1.95 BS01 KJU A 1 M419 V498 H524 M418 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=160uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 5aic A 1.89 BS01 TGX A 1 M419 D496 V498 H524 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=49.6uM remove_due_to_license_issue IC50=49600nM P34913 25931264 1550 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aip A 2.3 BS01 4HP B 1 S9 N11 S9 N11 ? 0003677,0003700,0006355,0006950,0045892 remove_due_to_license_issue Q7DD70 27105075 1146 MPTQSKHASINIGLIQAREALMTQFRPILNQANITDQQWRIIRLLAENGTLDFQDLANQACILRPSLTGILTRLEKAGLVVRLKPSNDQRRVFLKLTAEGEKLYEEIGEEVDERYDAIEEVLGREKMLLLKDLLAELAKIE 5aip B 2.3 BS01 4HP B 1 M22 F25 L29 D36 W39 R43 Y115 M14 F17 L21 D28 W31 R35 Y102 ? 0003677,0003700,0006355,0006950,0045892 Kd=1.5mM remove_due_to_license_issue Q7DD70 27105075 1146 SINIGLIQAREALMTQFRPILNQANITDQQWRIIRLLAENGTLDFQDLANQACILRPSLTGILTRLEKAGLVVRLKPRVFLKLTAEGEKLYEEIGEEVDERYDAIEEVLGREKMLLLKDLLAELAKIEDALN 5ais A 1.85 BS01 CWC A 1 M11 G13 R14 M99 W104 Y152 M10 G12 R13 M98 W103 Y151 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.57uM remove_due_to_license_issue Kd=570nM, IC50=820nM O60760 25978964 1200 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 5aiv A 2.04 BS01 M1W A 1 G13 R14 D96 M99 W104 Y152 G12 R13 D95 M98 W103 Y151 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.65uM remove_due_to_license_issue IC50=170nM, Kd=650nM O60760 25978964 1200 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTENTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 5aix B 2.1 BS02 KRX B 1 F9 M11 G13 R14 Q36 M99 W104 Y152 F8 M10 G12 R13 Q35 M98 W103 Y151 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.012uM remove_due_to_license_issue IC50=60nM, EC50=130nM, Kd=44nM O60760 25978964 1201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTENTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 5ajc C 1.7 BS01 SIA F 1 W76 G80 W81 W76 G80 W81 ? 0030246,0046872 remove_due_to_license_issue A0A0S4TLR1 27198630 3 SSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 5ajc C 1.7 BS02 FUC F 1 R17 E28 G39 A40 W76 W81 R17 E28 G39 A40 W76 W81 ? 0030246,0046872 remove_due_to_license_issue A0A0S4TLR1 27198630 4 SSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 5ajc C 1.7 BS04 FUC C 1 R62 E73 A85 R62 E73 A85 ? 0030246,0046872 remove_due_to_license_issue A0A0S4TLR1 27198630 111 SSVQTAATSWGTVPSIRVYTANNGKITERCWDGKGWYTGAFNEPGDNVSVTSWLVGSAIHIRVYASTGTTTTEWCWDGNGWTKGAYTAT 5ajv B 3.01 BS01 8R2 B 1 R45 Y49 I50 V214 V217 G218 L238 M239 I241 R35 Y39 I40 V204 V207 G208 L228 M229 I231 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 remove_due_to_license_issue IC50=>30000nM Q16875 25849762 1449 LELTQSRVQKIWVPVDHLPRSNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERS 5ajw A 2.5 BS03 S6L A 1 R45 G46 Y49 I50 V159 N163 V214 V217 G218 F221 L238 M239 I241 V243 R39 G40 Y43 I44 V153 N157 V208 V211 G212 F215 L232 M233 I235 V237 R252 H253 N259 S302 E322 H387 R246 H247 N253 S296 E316 H381 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=0.104uM remove_due_to_license_issue IC50=104nM Q16875 25849762 1449 PLELTQSRVQKIWVPVDHRPSLPRSNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERS 5ajx A 2.58 BS03 FD9 A 1 R45 G46 Y49 I50 V214 V217 G218 F221 L238 M239 I241 V243 R42 G43 Y46 I47 V211 V214 G215 F218 L235 M236 I238 V240 R252 H253 N259 S302 E322 H387 R249 H250 N256 S299 E319 H384 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 remove_due_to_license_issue IC50=>30000nM Q16875 25849762 1448 PLELTQSRVQKIWVPVDHRPSLPRSCGPNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRER 5ajy A 2.37 BS03 87T A 1 R45 I50 S152 V159 V217 G218 L238 M239 I241 V243 R40 I45 S147 V154 V212 G213 L233 M234 I236 V238 R252 H253 N259 S302 E322 H387 R247 H248 N254 S297 E317 H382 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=0.496uM remove_due_to_license_issue Q16875 25849762 1448 PLELTQSRVQKIWVPVDHRPSLPRSCNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRER 5ajz A 2.35 BS03 MJP A 1 R45 G46 Y49 I50 V159 N163 V217 G218 L238 I241 V243 R40 G41 Y44 I45 V154 N158 V212 G213 L233 I236 V238 R252 H253 N259 S302 E322 H387 R247 H248 N254 S297 E317 H382 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=2.01uM remove_due_to_license_issue IC50=2010nM Q16875 25849762 1449 LELTQSRVQKIWVPVDHRPSLPRSCGNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERS 5ak0 A 2.03 BS03 8V1 A 1 R45 Y49 I50 S152 S162 I164 V217 G218 F221 L238 M239 I241 R42 Y46 I47 S149 S159 I161 V214 G215 F218 L235 M236 I238 R252 H253 N259 S302 E322 H387 R249 H250 N256 S299 E319 H384 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=0.021uM remove_due_to_license_issue IC50=21nM Q16875 25849762 1450 PLELTQSRVQKIWVPVDHRPSLPRSCGPNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERS 5ak2 A 2.19 BS01 85Z A 1 T347 A350 D351 E353 L387 M388 L391 F404 M421 I424 H524 P535 T35 A38 D39 E41 L75 M76 L79 F92 M109 I112 H205 P211 ? ic50=0.0039uM remove_due_to_license_issue IC50=3.9nM P03372 25790336 1553 GSHMALSLTADQMVSALLDAEPPILYSESMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMVPSYDLLLEMLDAHRLHAP 5ak3 A 2.28 BS01 XM0 A 1 M310 Y343 N472 A476 M309 Y342 N471 A475 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=8.49uM remove_due_to_license_issue P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak4 A 1.79 BS01 GVG A 1 L408 M419 H524 W525 L407 M418 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=59.2uM remove_due_to_license_issue P34913 25931264 1550 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak4 A 1.79 BS02 GVG A 2 D335 W336 M339 F381 Q384 Y466 D334 W335 M338 F380 Q383 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=59.2uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak4 A 1.79 BS03 GVG A 3 W336 Y343 P371 M469 N472 W473 W335 Y342 P370 M468 N471 W472 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=59.2uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak5 A 2.22 BS01 V2Z A 1 M419 V498 H524 M418 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.086uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak6 A 2.15 BS01 YPN A 1 D335 W336 Y383 Q384 Y466 D329 W330 Y377 Q378 Y460 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y460 D490 H518 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=326.4uM remove_due_to_license_issue P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak6 A 2.15 BS02 YPN A 2 M419 V498 H524 W525 M413 V492 H518 W519 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y460 D490 H518 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=326.4uM remove_due_to_license_issue P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ak9 A 2.601 BS01 dna B 0 D21 T41 A42 K43 T76 R124 T150 H152 D154 H156 R157 N164 S166 L167 D17 T37 A38 K39 T72 R120 T146 H148 D150 H152 R153 N160 S162 L163 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 14 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 A 2.601 BS02 dna C 0 G20 D21 G22 Y25 Y29 K30 R33 R37 R77 G16 D17 G18 Y21 Y25 K26 R29 R33 R73 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 15 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 A 2.601 BS03 dna D 0 N32 R33 S34 E35 Y36 R37 S67 K68 Q70 D75 R81 S83 S84 K85 E117 G118 D119 M120 R126 W128 K130 D155 H158 N28 R29 S30 E31 Y32 R33 S63 K64 Q66 D71 R77 S79 S80 K81 E113 G114 D115 M116 R122 W124 K126 D151 H154 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 E 2.601 BS01 dna C 0 R104 H175 S180 H181 R100 H171 S176 H177 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 15 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 E 2.601 BS02 dna D 0 S179 H181 L182 N183 S175 H177 L178 N179 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 E 2.601 BS03 dna F 0 D21 T41 K43 T76 R77 R124 H152 D154 R157 S166 L167 D17 T37 K39 T72 R73 R120 H148 D150 R153 S162 L163 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 14 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 E 2.601 BS04 dna G 0 G20 D21 G22 Y25 Y29 K30 R33 R37 R77 G16 D17 G18 Y21 Y25 K26 R29 R33 R73 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 15 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 E 2.601 BS05 dna H 0 N32 R33 S34 E35 Y36 R37 S67 K68 Q70 R81 S83 S84 K85 E117 G118 D119 R126 W128 K130 D155 H158 N28 R29 S30 E31 Y32 R33 S63 K64 Q66 R77 S79 S80 K81 E113 G114 D115 R122 W124 K126 D151 H154 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLPP 5ak9 J 2.601 BS01 dna K 0 D21 T41 A42 K43 T76 R77 R124 H152 D154 R157 N164 S166 L167 D17 T37 A38 K39 T72 R73 R120 H148 D150 R153 N160 S162 L163 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 14 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLP 5ak9 J 2.601 BS02 dna L 0 G20 D21 G22 Y25 Y29 K30 R33 R77 G16 D17 G18 Y21 Y25 K26 R29 R73 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 15 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLP 5ak9 J 2.601 BS03 dna N 0 N32 R33 S34 E35 Y36 R37 S67 K68 D75 R81 S83 S84 K85 E117 D119 M120 R126 W128 N129 K130 D155 H158 N28 R29 S30 E31 Y32 R33 S63 K64 D71 R77 S79 S80 K81 E113 D115 M116 R122 W124 N125 K126 D151 H154 3.1.-.- 0004519,0006314,0016539 remove_due_to_license_issue P21505 26045557 1 ~ 25 ENVSGISAYLLGLIIGDGGLYKLKYKGNRSEYRVVITAKSENLIKQHIAPLMQFLIDELNVKSKIQIVKGDTRYELRVSSKKLYYYFANMLERIRLFNMREQIAFIKGLYVAEGDMTLKRLRIWNKNKALLEIVSRWLNNLGVRNTIHLDDHRHGVYVLNISLRDRIKFVHTILSSHLNPLP 5ake A 2.26 BS01 6N0 A 1 F267 D335 W336 Y383 L408 Y466 V498 L499 W525 F266 D334 W335 Y382 L407 Y465 V497 L498 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.015uM remove_due_to_license_issue IC50=20nM P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5akg A 2.51 BS01 6N6 A 1 M310 W336 Q384 M469 N472 M309 W335 Q383 M468 N471 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue IC50=34810nM P34913 25931264 1550 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5akh A 2.1 BS01 6NM A 1 F267 Y383 L408 M419 D496 V498 H524 F266 Y382 L407 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.256uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aki A 1.81 BS01 6NF A 1 F267 D335 Y383 Q384 L408 M419 Y466 F263 D331 Y379 Q380 L404 M415 Y462 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F263 H330 D331 W332 N355 N374 Y379 Y462 D492 H520 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.754uM remove_due_to_license_issue P34913 25931264 1558 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 5akj A 2.03 BS01 6N4 A 1 D335 W336 Y383 Y466 W525 D334 W335 Y382 Y465 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50<1.37uM remove_due_to_license_issue IC50=1370nM P34913 25931264 1555 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5akk A 1.9 BS01 1P8 A 1 M310 M339 Y343 N472 A476 M306 M335 Y339 N466 A470 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F263 H330 D331 W332 N355 N374 Y379 Y460 D490 H518 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=99.3uM remove_due_to_license_issue P34913 25931264 1550 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5akk A 1.9 BS02 1P8 A 2 P371 M469 N472 P367 M463 N466 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F263 H330 D331 W332 N355 N374 Y379 Y460 D490 H518 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=99.3uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5akl A 2.0 BS01 6N8 A 1 F267 D335 W336 Y383 L408 M419 Y466 V498 H524 F254 D322 W323 Y370 L395 M406 Y453 V485 H511 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F254 H321 D322 W323 N346 N365 Y370 Y453 D483 H511 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50<0.086uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aku A 1.8 BS01 29F A 1 H1031 G1032 F1035 Y1050 Y1060 F1061 A1062 S1068 Y1071 H80 G81 F84 Y99 Y109 F110 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=150nM remove_due_to_license_issue IC50=8.7nM, EC50=1500nM Q9H2K2 26183543 2164 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5akw A 2.07 BS02 NKI A 1 H1031 G1032 S1033 Y1050 Y1060 F1061 A1062 S1068 Y1071 H80 G81 S82 Y99 Y109 F110 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=410nM remove_due_to_license_issue IC50=410nM Q9H2K2 26183543 2163 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5akz A 2.18 BS01 6NX A 1 D335 W336 Y383 Q384 Y466 D334 W335 Y382 Q383 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=5.49uM remove_due_to_license_issue P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5al1 A 1.75 BS02 GN5 A 1 H1031 G1032 Y1050 Y1060 F1061 A1062 S1068 Y1071 H80 G81 Y99 Y109 F110 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=53000nM remove_due_to_license_issue IC50=53000nM Q9H2K2 26183543 2167 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5al2 A 1.9 BS01 O53 A 1 H1031 G1032 Y1050 Y1060 F1061 A1062 S1068 Y1071 H80 G81 Y99 Y109 F110 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=360nM remove_due_to_license_issue IC50=355nM Q9H2K2 26183543 2164 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5al3 A 1.75 BS02 TGW A 1 H1031 G1032 F1035 H1048 Y1050 Y1060 F1061 A1062 S1068 Y1071 H80 G81 F84 H97 Y99 Y109 F110 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=11000nM remove_due_to_license_issue IC50=11000nM Q9H2K2 26183543 3168 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5al4 A 1.9 BS02 WLH A 1 H1031 G1032 S1033 Y1050 Y1060 S1068 Y1071 H80 G81 S82 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=300nM remove_due_to_license_issue IC50=300nM Q9H2K2 26183543 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5al5 A 2.05 BS02 JL9 A 1 H1031 G1032 S1033 F1035 Y1050 Y1060 A1062 K1067 S1068 Y1071 I1075 H80 G81 S82 F84 Y99 Y109 A111 K116 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=71nM remove_due_to_license_issue IC50=71nM Q9H2K2 26183543 2165 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5alb H 2.16 BS01 TIQ L 1 H35 I52 T56 S58 Y99 W100B P100H D100J H34 I51 T56 S58 Y102 W105 P111 D113 remove_due_to_license_issue 25788700 1210 VQLQESGAEVKKPGSSVRVSCKASGGTFDSYSIHWVRQAPGQGLEWMGGIIPAFGTLSSAQDFQARVTISADKSTSTAYMELSGLRSEDTAVYYCARGSFDYYFWSASHPPNDALAIWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKRVEP 5alb L 2.16 BS01 TIQ L 1 G89 T90 W91 Y93 A95A F98 G88 T89 W90 Y92 A95 F99 remove_due_to_license_issue 25788700 1210 VVTQPPSVSAAPGQKVTISCSGSNSDIGNNYVSWYQQLPGTAPKLLIYDNNKRPSGIPDRFSGSKSGTSATLAITGLQAGDEADYYCGTWLYDRAVGLFGGGTKVTVLGQPKAAPSVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADSSPVKAGVETTTPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAP 5alc H 1.7 BS01 TIQ L 1 H35 W47 I52 L57 Y99 D100J L100L H34 W46 I51 L57 Y102 D105 L107 remove_due_to_license_issue 25788700 1210 VQLQESGAEVKKPGSSVRVSCKASGGTFDSYSIHWVRQAPGQGLEWMGGIIPAFGTLSSAQDFQARVTISADKSTSTAYMELSGLRSEDTAVYYCARGSHLYPNDALAIWGQGTLVTVSSASTKGPSVFPLAPSSKSTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKRVEP 5alc L 1.7 BS01 TIQ L 1 G89 T90 W91 S95A F98 G88 T89 W90 S95 F99 remove_due_to_license_issue 25788700 1210 VVTQPPSVSAAPGQKVTISCSGSNSDIGNNYVSWYQQLPGTAPKLLIYDNNKRPSGIPDRFSGSKSGTSATLAITGLQAGDEADYYCGTWDISLSAGLFGGGTKVTVLGQPKAAPSVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADSSPVKAGVETTTPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAP 5ald A 2.26 BS01 FCW A 1 Y383 M419 D496 V498 H524 Y382 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=1.08uM remove_due_to_license_issue IC50=1080nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ale A 1.95 BS01 ONR A 1 Y383 L408 M419 V498 H524 W525 Y382 L407 M418 V497 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=1.132uM remove_due_to_license_issue IC50=1130nM P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alf A 2.32 BS01 OE1 A 1 F267 D335 W336 M339 F381 Y383 Q384 Y466 H524 A546 R547 F266 D334 W335 M338 F380 Y382 Q383 Y465 H523 A545 R546 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.204uM remove_due_to_license_issue P34913 25931264 1548 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alg A 2.4 BS01 R4N A 1 F267 D335 W336 F381 Y383 F387 L408 M419 L428 Y466 V498 L499 H524 F266 D334 W335 F380 Y382 F386 L407 M418 L427 Y465 V497 L498 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.03uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alh A 1.9 BS01 4UA A 1 D335 W336 T360 I375 F381 Y383 Q384 Y466 V498 M503 H524 W525 D334 W335 T359 I374 F380 Y382 Q383 Y465 V497 M502 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50<0.086uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5ali A 1.85 BS01 Q3B A 1 F267 D335 W336 M339 Y343 I363 F381 Y383 Q384 L408 M419 Y466 F266 D334 W335 M338 Y342 I362 F380 Y382 Q383 L407 M418 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50<0.086uM remove_due_to_license_issue P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alj A 2.1 BS01 T5J A 1 F267 D335 W336 F381 Q384 Y466 M469 F253 D321 W322 F361 Q364 Y442 M445 F267 H334 D335 W336 N359 Y383 Y466 D496 H524 F253 H320 D321 W322 N345 Y363 Y442 D472 H500 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=2.737uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLEVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alk A 2.33 BS01 WMR A 1 F267 Y383 F387 L408 M419 D496 V498 L499 H524 W525 F266 Y382 F386 L407 M418 D495 V497 L498 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.252uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5all A 2.2 BS01 II6 A 1 D335 Y383 Y466 H524 D334 Y382 Y465 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=2.678uM remove_due_to_license_issue IC50=2680nM P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alm A 2.0 BS01 7GM A 1 D335 W336 Y383 Q384 Y466 H524 D334 W335 Y382 Q383 Y465 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.294uM remove_due_to_license_issue IC50=290nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aln A 2.0 BS01 5ZM A 1 F267 L408 M419 D496 F497 V498 H524 F266 L407 M418 D495 F496 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.267uM remove_due_to_license_issue P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alo A 2.0 BS01 A0J A 1 W336 A365 I375 F381 M469 N472 W335 A364 I374 F380 M468 N471 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.738uM remove_due_to_license_issue IC50=740nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alp A 2.06 BS01 QYD A 1 F267 D335 W336 Y383 Q384 L408 M419 Y466 W525 F266 D334 W335 Y382 Q383 L407 M418 Y465 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50<0.086uM remove_due_to_license_issue P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alr A 2.6 BS01 8TM A 1 F267 D335 W336 Y383 Q384 F387 L408 Y466 H524 F266 D334 W335 Y378 Q379 F382 L403 Y461 H519 F267 H334 D335 W336 N359 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 Y378 Y461 D491 H519 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESKAFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5als A 2.57 BS01 5DQ A 1 F267 D335 W336 M339 Y383 Q384 Y466 V498 M503 F266 D334 W335 M338 Y377 Q378 Y460 V492 M497 F267 H334 D335 W336 N359 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 Y377 Y460 D490 H518 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alt A 2.15 BS01 9XZ A 1 D335 W336 M339 I375 Q384 M469 D334 W335 M338 I374 Q383 M468 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=13.1uM remove_due_to_license_issue IC50=13100nM P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alu A 1.87 BS01 HD2 A 1 D11 F20 F41 T51 N124 D10 F19 F40 T50 N123 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.022uM remove_due_to_license_issue P34913 25931264 1548 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alu A 1.87 BS02 HD2 A 2 I363 N366 F381 Q384 M503 I362 N365 F380 Q383 M502 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.022uM remove_due_to_license_issue P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alu A 1.87 BS03 HD2 A 3 D335 W336 Y383 Q384 Y466 V498 L499 H524 D334 W335 Y382 Q383 Y465 V497 L498 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.022uM remove_due_to_license_issue P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alv A 1.8 BS01 6TZ A 1 D335 W336 M339 T360 Y383 Q384 Y466 D329 W330 M333 T354 Y377 Q378 Y456 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y456 D486 H514 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=43.48uM remove_due_to_license_issue P34913 25931264 1550 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alw A 2.2 BS01 JQN A 1 F267 Y383 F387 L408 M419 L428 V498 H524 W525 F266 Y382 F386 L407 M418 L427 V497 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=7.05uM remove_due_to_license_issue IC50=7050nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alx A 2.23 BS01 DUL A 1 F267 S407 L408 R410 S415 L417 M419 V498 H524 W525 F266 S406 L407 R409 S414 L416 M418 V497 H523 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=3.277uM remove_due_to_license_issue IC50=3280nM P34913 25931264 1550 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5aly A 1.9 BS01 B7H A 1 F267 F387 L408 M419 D496 V498 H524 F266 F386 L407 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.1845uM remove_due_to_license_issue IC50=180nM P34913 25931264 1555 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5alz A 2.3 BS01 XQ9 A 1 F267 D335 W336 M339 Y383 Q384 M419 Y466 W525 F266 D334 W335 M338 Y382 Q383 M418 Y465 W524 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.006uM remove_due_to_license_issue IC50=3.9nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am0 A 1.88 BS01 LWS A 1 F267 M419 D496 V498 H524 F266 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=1.32uM remove_due_to_license_issue IC50=1320nM P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am1 A 2.15 BS01 I5T A 1 F267 D335 W336 M339 Y383 Y466 L499 M503 H524 F266 D334 W335 M338 Y382 Y465 L498 M502 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.003uM remove_due_to_license_issue IC50=3.0nM P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am2 A 1.7 BS01 KUF A 1 F267 Y383 F387 L408 L428 F261 Y377 F381 L402 L418 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y456 D486 H514 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=9.685uM remove_due_to_license_issue P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am2 A 1.7 BS02 KUF A 2 D496 F497 V498 H524 W525 D486 F487 V488 H514 W515 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y456 D486 H514 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=9.685uM remove_due_to_license_issue P34913 25931264 1553 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am2 A 1.7 BS03 KUF A 3 W336 M339 Y343 M469 N472 W330 M333 Y337 M459 N462 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y456 D486 H514 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=9.685uM remove_due_to_license_issue P34913 25931264 1554 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am2 A 1.7 BS04 KUF A 4 I363 S374 I357 S368 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F261 H328 D329 W330 N353 N372 Y377 Y456 D486 H514 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=9.685uM remove_due_to_license_issue P34913 25931264 1555 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am3 A 2.2 BS01 AUB A 1 F267 D335 W336 Y383 Q384 S415 M419 Y466 F266 D334 W335 Y382 Q383 S414 M418 Y465 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.005uM remove_due_to_license_issue IC50=1.5nM, Ki=1.5nM P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am4 A 1.87 BS01 MVJ A 1 F267 Y383 F387 L408 M419 D496 V498 H524 F266 Y382 F386 L407 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.113uM remove_due_to_license_issue P34913 25931264 1555 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am5 A 2.26 BS01 6NZ A 1 F267 S415 M419 D496 V498 H524 F266 S414 M418 D495 V497 H523 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=1.82uM remove_due_to_license_issue IC50=1820nM P34913 25931264 1551 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am5 A 2.26 BS02 6NZ A 2 W336 Y343 I363 N472 W335 Y342 I362 N471 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=1.82uM remove_due_to_license_issue IC50=1820nM P34913 25931264 1552 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5am6 A 1.96 BS01 38O A 1 V561 E562 Y563 A564 S565 G567 L630 V102 E103 Y104 A105 S106 G108 L160 D623 A625 R627 N628 D641 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=185nM remove_due_to_license_issue P11362 26097890 1766 VAGVSEYELPEDPRWELPRDRLVLGKPLGEGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 5am7 A 1.957 BS01 38O A 1 V492 A512 I545 M561 E562 Y563 A564 S565 K566 G567 L630 V32 A52 I85 M101 E102 Y103 A104 S105 K106 G107 L160 D623 A625 R627 N628 D641 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Kd=64.5nM remove_due_to_license_issue P11362 26097890 1000 AGVSEYELPEDPRWELPRDRLVLGKPLGEGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIMEYASKGNLREYLQARRPPGPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQ 5amd A 1.5 BS02 45I A 1 Q92 H94 H119 V121 F131 L198 T199 T200 Q89 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.8nM remove_due_to_license_issue P00918 25813715 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5amg A 1.55 BS02 IW7 A 1 Q92 H94 H119 V121 F131 L198 T199 T200 Q89 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=6nM remove_due_to_license_issue P00918 25813715 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5aml A 1.36 BS02 51J A 1 Q92 H94 H119 V121 F131 L198 T199 T200 Q89 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.7nM remove_due_to_license_issue P00918 25813715 266 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5amn A 2.57 BS01 DTQ A 1 L730 V738 A756 K758 E775 V804 A807 G810 L881 D892 L29 V37 A55 K57 E74 V103 A106 G109 L160 D171 D874 A876 R878 N879 D892 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=380nM P07949 26874741 2018 GPLSLSVDAFKIDPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVERALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMV 5anq B 2.0 BS01 5YQ B 1 Y132 G170 F185 H188 E190 D191 K206 W208 K241 H276 Y123 G161 F176 H179 E181 D182 K197 W199 K232 H267 G170 Y177 H188 E190 H276 S288 G161 Y168 H179 E181 H267 S279 1.14.11.66,1.14.11.69 ic50=3.98uM remove_due_to_license_issue O75164 26971619 1354 PSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEF 5ans A 1.6 BS01 RX8 A 1 L9 K23 N33 F72 M81 W117 D119 D120 L8 K22 N32 F71 M80 W116 D118 D119 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=2.056uM remove_due_to_license_issue P36639 26878898 1157 GASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5ant A 2.0 BS01 RJE A 1 L9 F27 N33 G34 G36 F72 M81 V83 W117 D119 D120 L8 F26 N32 G33 G35 F71 M80 V82 W116 D118 D119 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=0.44uM remove_due_to_license_issue P36639 26878898 1157 GASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5anu A 1.8 BS01 58T A 1 T8 L9 F27 N33 G34 F72 M81 V83 W117 D119 D120 T6 L7 F25 N31 G32 F70 M79 V81 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=0.0004uM remove_due_to_license_issue IC50=0.500000nM P36639 26878898 1158 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5anv A 1.16 BS01 RGJ A 1 Y7 L9 N33 G34 G37 F72 F74 M81 W117 D119 D120 F124 F139 Y5 L7 N31 G32 G35 F70 F72 M79 W114 D116 D117 F121 F136 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=0.0005uM remove_due_to_license_issue P36639 26878898 1157 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5anw A 1.37 BS01 9CQ A 1 T8 N33 G36 G37 F72 F74 M81 W117 D119 D120 F139 T6 N31 G34 G35 F70 F72 M79 W115 D117 D118 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=0.003uM remove_due_to_license_issue IC50=9.0nM P36639 26878898 1157 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5aoi B 1.78 BS02 RZH B 1 V147 T150 P151 C220 P222 P223 V53 T56 P57 C126 P128 P129 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=940uM remove_due_to_license_issue P04637 26636255 1292 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5aoj A 1.47 BS01 Y0V A 1 L145 V147 T150 P151 C220 E221 P223 T230 L50 V52 T55 P56 C125 E126 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=21uM remove_due_to_license_issue Kd=21000nM P04637 26636255 1291 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5aok A 1.35 BS02 GOH A 1 L145 V147 T150 P151 C220 E221 P223 T230 L50 V52 T55 P56 C125 E126 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 26636255 1292 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5aol A 1.5 BS01 UFV A 1 L145 V147 C220 E221 T230 L50 V52 C125 E126 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=4800uM remove_due_to_license_issue P04637 26636255 1293 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 5aom A 1.74 BS01 FY8 A 1 L145 V147 T150 P151 E221 P222 P223 T230 L50 V52 T55 P56 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=1270uM remove_due_to_license_issue P04637 26636255 1291 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5aom A 1.74 BS02 FY8 A 2 P153 C220 E221 P222 P58 C125 E126 P127 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=1270uM remove_due_to_license_issue P04637 26636255 1292 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5ap0 A 2.15 BS01 AU5 A 1 I531 V539 M602 C604 G605 N606 I607 D608 S611 L654 Q794 I17 V25 M88 C90 G91 N92 I93 D94 S97 L140 Q255 D647 K649 N652 D664 T686 D133 K135 N138 D150 T159 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=35nM P33981 26202014 1795 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQVGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ap1 A 2.05 BS01 O38 A 1 I531 V539 Q541 A551 M602 C604 N606 I607 D608 S611 L654 I663 P673 I17 V25 Q27 A37 M88 C90 N92 I93 D94 S97 L140 I149 P159 D647 K649 N652 D664 T686 D133 K135 N138 D150 T170 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 26202014 1796 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTTSVVKDVGTVNYMPPEAIKDMSSKSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 5ap2 A 2.8 BS01 PWU A 1 I531 A551 K553 I586 M602 C604 G605 N606 I607 L654 I663 P673 I16 A36 K38 I71 M87 C89 G90 N91 I92 L139 I148 P158 D647 K649 N652 D664 T686 D132 K134 N137 D149 T161 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 26202014 1795 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMSPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ap3 A 2.7 BS01 AU5 A 1 I531 V539 M602 C604 G605 N606 I607 L654 I16 V24 M87 C89 G90 N91 I92 L139 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=35nM P33981 26202014 1799 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNGWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANSQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ap4 A 2.85 BS01 O38 A 1 I531 Q541 I586 M602 C604 N606 I607 D608 L654 I663 M671 P673 I17 Q27 I72 M88 C90 N92 I93 D94 L140 I149 M156 P158 D647 K649 N652 D664 T686 D133 K135 N138 D150 T163 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 26202014 1795 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNGWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANMQPDQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ap5 A 2.8 BS01 7RO A 1 I531 A551 K553 I586 M602 C604 G605 N606 L654 I663 I17 A37 K39 I72 M88 C90 G91 N92 L140 I149 D647 K649 N652 D664 T686 D133 K135 N138 D150 T156 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=6.0nM P33981 26202014 1795 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNGWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIAGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ap6 A 2.1 BS01 PWU A 1 I531 A551 K553 I586 M602 G605 N606 I607 D608 S611 L654 I663 M671 P673 I16 A36 K38 I71 M87 G90 N91 I92 D93 S96 L139 I148 M156 P158 D647 K649 N652 D664 T686 D132 K134 N137 D149 T165 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 26202014 1795 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEWGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDDSQVGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ap7 A 2.45 BS01 SVE A 1 I531 V539 A551 K553 M602 W604 G605 N606 D608 L654 I663 I23 V31 A43 K45 M94 W96 G97 N98 D100 L146 I155 D647 K649 N652 D664 T686 D139 K141 N144 D156 T168 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=182nM P33981 26202014 1795 GTENLYFQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEWGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5aph A 1.54 BS02 VYI A 1 W317 C320 A321 H323 L324 M358 M365 F378 I400 W60 C63 A64 H66 L67 M101 M108 F121 I143 ? 0003677,0004879,0005634,0006355 ic50=0.06uM remove_due_to_license_issue IC50=60nM P51449 26553345 1510 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5apj A 2.08 BS02 76E A 1 W317 C320 H323 L324 V361 V376 F378 F388 C393 I397 I400 W60 C63 H66 L67 V104 V119 F121 F131 C136 I140 I143 ? 0003677,0004879,0005634,0006355 ic50=0.04uM remove_due_to_license_issue P51449 26553345 1508 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5aqf A 1.88 BS01 ADN A 1 G202 G230 E268 K271 R272 S275 G339 R342 G203 G231 E269 K272 R273 S276 G340 R343 D10 K71 E175 D199 D11 K72 E176 D200 3.6.4.10 0005524,0140662 remove_due_to_license_issue Kd=110000nM P11142 27708405 1382 SMSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqg A 2.24 BS01 ZJB A 1 G202 E268 K271 R272 S275 G339 S340 R342 G202 E268 K271 R272 S275 G339 S340 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqh A 2.0 BS01 ZVO A 1 R272 S275 G339 R342 R272 S275 G339 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqj E 1.96 BS01 Q88 E 1 R272 S275 G339 R342 R273 S276 G340 R343 D10 K71 E175 D199 D11 K72 E176 D200 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1383 SMSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqk A 2.09 BS01 GDP A 1 T14 G201 G202 G230 E268 K271 R272 S275 G338 G339 R342 T11 G198 G199 G227 E265 K268 R269 S272 G335 G336 R339 D10 K71 E175 D199 D7 K68 E172 D196 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 GPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqn A 2.45 BS01 JG8 A 1 R272 G339 R342 R272 G339 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqo A 2.12 BS01 CWS A 1 R272 S275 G339 R342 R272 S275 G339 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1384 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqp C 2.08 BS01 1LQ C 1 R272 S275 G339 R342 R272 S275 G339 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqq E 2.72 BS01 BBW E 1 K271 R272 S275 G339 R342 I343 K271 R272 S275 G339 R342 I343 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqr A 1.91 BS01 N8Y A 1 R272 S275 G339 R342 R272 S275 G339 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1383 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqt A 1.9 BS01 5P7 A 1 G230 E268 K271 R272 S275 G339 R342 G230 E268 K271 R272 S275 G339 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1381 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAIL 5aqu A 1.92 BS01 UX0 A 1 G230 E268 K271 R272 S275 G339 S340 R342 G230 E268 K271 R272 S275 G339 S340 R342 D10 K71 E175 D199 D10 K71 E175 D199 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1388 MSKGPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqv A 1.75 BS01 KC7 A 1 G230 E268 K271 R272 S275 G339 R342 D366 G227 E265 K268 R269 S272 G336 R339 D363 D10 K71 E175 D199 D7 K68 E172 D196 3.6.4.10 0005524,0140662 remove_due_to_license_issue P11142 27708405 1382 GPAVGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVAMNPTNTVFDAKRLIGRRFDDAVVQSDMKHWPFMVVNDAGRPKVQVEYKGETKSFYPEEVSSMVLTKMKEIAEAYLGKTVTNAVVTVPAYFNDSQRQATKDAGTIAGLNVLRIINEPTAAAIAYGLDKKVGAERNVLIFDLGGGTFDVSILTIEDGIFEVKSTAGDTHLGGEDFDNRMVNHFIAEFKRKHKKDISENKRAVRRLRTACERAKRTLSSSTQASIEIDSLYEGIDFYTSITRARFEELNADLFRGTLDPVEKALRDAKLDKSQIHDIVLVGGSTRIPKIQKLLQDFFNGKELNKSINPDEAVAYGAAVQAAILS 5aqz A 1.65 BS01 SGV A 1 E268 K271 R272 S275 G339 R342 E270 K273 R274 S277 G341 R344 D10 K71 E175 D199 D12 K73 E177 D201 3.6.3.51 0005524,0140662 Kd=3.3uM remove_due_to_license_issue P0DMV8 27119979 1389 GSMAKAAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILIKSTRAAA 5ar0 A 1.9 BS01 GB8 A 1 Y15 G202 G230 E268 K271 R272 S275 G339 R342 Y13 G198 G226 E264 K267 R268 S271 G335 R338 D10 K71 E175 D199 D8 K67 E171 D195 3.6.3.51 0005524,0140662 Kd=720nM remove_due_to_license_issue Ki=1.29e+3nM, IC50=2900nM P0DMV8 27119979 1384 KAAAIGIDLGTTYSCVGVFQKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILIKS 5ar4 A 2.7 BS01 SB2 A 1 R26 V32 A45 K47 L79 I93 T95 Y97 M98 Q150 L153 D164 R22 V28 A41 K43 L70 I84 T86 Y88 M89 Q141 L144 D155 D146 K148 Q150 N151 D164 T189 D137 K139 Q141 N142 D155 T159 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43353 26455654 1311 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLHLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLTIIYMPPENYEASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5ar5 A 2.66 BS01 IQ7 A 1 L24 V32 A45 K47 L79 T95 Y97 M98 G101 L153 D164 L21 V29 A42 K44 L72 T88 Y90 M91 G94 L146 D157 D146 K148 Q150 N151 D164 T189 D139 K141 Q143 N144 D157 T169 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=12nM O43353 26455654 1312 EAICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLHLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRMEGGTIIYMPPENYEPSIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5ar7 A 2.71 BS01 SR8 A 1 A45 K47 E66 L70 L79 T95 Y97 M98 H144 L153 I162 A163 D164 F165 R171 A40 K42 E56 L60 L69 T85 Y87 M88 H134 L143 I152 A153 D154 F155 R161 D146 K148 Q150 N151 D164 T189 D136 K138 Q140 N141 D154 T163 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=320nM O43353 26455654 1311 ICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLHLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRMTIIYMPPENYEASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5ar8 A 2.79 BS01 XYW A 1 L24 S25 V32 A45 K47 L70 L79 I81 T95 Y97 M98 G101 E105 L153 A163 D164 F165 L16 S17 V24 A37 K39 L48 L57 I59 T69 Y71 M72 G75 E79 L127 A137 D138 F139 D146 K148 Q150 N151 D164 T189 D120 K122 Q124 N125 D138 T141 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=6.3nM O43353 26455654 1311 ALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLLREAEILHKARFSYILPILGICNLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGTIIYMPPENYASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5arf A 1.92 BS01 I9H A 1 E104 T105 L108 G183 F184 T185 S196 Y217 Y240 Y258 E99 T100 L103 G178 F179 T180 S191 Y212 Y235 Y253 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 Kd=540nM remove_due_to_license_issue Q9NRG4 27075367 1001 LGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLGFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEI 5arg A 1.99 BS04 H41 A 1 E104 T105 L108 N182 G183 F184 T185 S196 A203 Y217 T238 Y240 Y258 E99 T100 L103 N177 G178 F179 T180 S191 A198 Y212 T233 Y235 Y253 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 ic50=27nM remove_due_to_license_issue Q9NRG4 27075367 1432 LGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLGFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIE 5aut A 1.7 BS01 2AN A 1 L19 V27 A40 K42 L93 V96 M146 I160 D161 L18 V26 A39 K41 L92 V95 M143 I157 D158 D139 K141 E143 N144 D161 T180 D136 K138 E140 N141 D158 T177 2.7.11.1 0004672,0005524,0006468 Kd=6.7uM remove_due_to_license_issue P53355 26322379 301 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5auu A 1.7 BS01 LU2 A 1 A40 K42 E64 L68 I77 L93 E94 L95 V96 I160 D161 F162 A39 K41 E63 L67 I76 L92 E93 L94 V95 I157 D158 F159 D139 K141 E143 N144 D161 T180 D136 K138 E140 N141 D158 T177 2.7.11.1 0004672,0005524,0006468 ic50=21uM remove_due_to_license_issue IC50=21000nM P53355 26322379 400 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5auv A 1.5 BS01 AGI A 1 G20 S21 V27 A40 E94 L95 I160 D161 G19 S20 V26 A39 E93 L94 I158 D159 D139 K141 E143 N144 D161 T180 D137 K139 E141 N142 D159 T178 2.7.11.1 0004672,0005524,0006468 ic50=31uM remove_due_to_license_issue IC50=31000nM P53355 26322379 400 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKSLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5auw A 1.5 BS01 QUE A 1 L19 A40 K42 E64 I77 L93 E94 L95 V96 I160 D161 F162 L18 A39 K41 E63 I76 L92 E93 L94 V95 I157 D158 F159 D139 K141 E143 N144 D161 T180 D136 K138 E140 N141 D158 T177 2.7.11.1 0004672,0005524,0006468 ic50=8.9uM remove_due_to_license_issue IC50=8900nM P53355 26322379 400 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5aux A 1.5 BS01 KMP A 1 L19 G20 S21 V27 A40 K42 E94 L95 V96 I160 D161 L18 G19 S20 V26 A39 K41 E93 L94 V95 I158 D159 D139 K141 E143 N144 D161 T180 D137 K139 E141 N142 D159 T178 2.7.11.1 0004672,0005524,0006468 ic50=10uM remove_due_to_license_issue IC50=10000nM P53355 26322379 400 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKSLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5auy A 2.0 BS01 MRI A 1 A40 K42 E64 L93 E94 L95 V96 M146 I160 D161 F162 A39 K41 E63 L92 E93 L94 V95 M144 I158 D159 F160 D139 K141 E143 N144 D161 T180 D137 K139 E141 N142 D159 T178 2.7.11.1 0004672,0005524,0006468 ic50=1.6uM remove_due_to_license_issue IC50=1600nM P53355 26322379 300 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKSLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5auz A 1.6 BS01 GEN A 1 V27 A40 K42 E94 L95 V96 I160 D161 V26 A39 K41 E93 L94 V95 I157 D158 D139 K141 E143 N144 D161 T180 D136 K138 E140 N141 D158 T177 2.7.11.1 0004672,0005524,0006468 ic50=98uM remove_due_to_license_issue IC50=98000nM P53355 26322379 400 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5av0 A 1.85 BS01 47X A 1 V27 A40 E94 L95 E100 I160 V26 A39 E93 L94 E99 I158 D139 K141 E143 N144 D161 T180 D137 K139 E141 N142 D159 T178 2.7.11.1 0004672,0005524,0006468 ic50=280uM remove_due_to_license_issue IC50=280000nM P53355 26322379 300 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKSLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP 5ave A 1.8 BS01 SER A 1 W141 W147 R152 W154 Y170 D172 S173 F199 D201 W85 W91 R96 W98 Y114 D116 S117 F143 D145 ? Kd=3.6uM remove_due_to_license_issue A0A0H3AES3 26878914 501 SVRDEIRSMVSDSVDEIVDGVSKTTAEVINGRKSIAQYATSLIESNPEPDNVRTIISQPLIKNTFLLVGFGLEKDGSNINNDPSWNPGPTWDPRVRPWYKDAKNAGKLVITAPYADSASGEILVSVATPVKDSATGQFLGSIFYDVSLAELAELVNEVKLFDAGYVFIVSEDGTTIAHPKKEFNGKPMSEFLGESKINVDTHQVIINGKPYAVSFSDVEGEDWYVGVVIDEEIAYAALDELRRSTLIHHHHH 5avf A 1.95 BS01 TAU A 1 W147 R152 W154 Y170 D172 S173 F199 D201 W95 R100 W102 Y118 D120 S121 F147 D149 ? Kd=3.2uM remove_due_to_license_issue Q9KL26 26878914 501 GPLGSVRDEIRSMVSDSVDEIVDGVSKTTAEVINGRKSIAQYATSLIESNPEPDNVRTIISQPLIKNTFLLVGFGLEKDGSNINNDPSWNPGPTWDPRVRPWYKDAKNAGKLVITAPYADSASGEILVSVATPVKDSATGQFLGSIFYDVSLAELAELVNEVKLFDAGYVFIVSEDGTTIAHPKKEFNGKPMSEFLGESKINVDTHQVIINGKPYAVSFSDVEGEDWYVGVVIDEEIAYAALDE 5avi A 2.7 BS02 4KM A 1 F257 L260 A261 S264 M298 E301 T302 R305 F315 F335 F39 L42 A43 S46 M80 E83 T84 R87 F97 F117 ? 0003677,0004879,0006629 remove_due_to_license_issue EC50=310nM Q13133 26238323 501 PQLSPEQLGMIEKLVAAQQRVTPWPPHSREARQQRFAHFTELAIVSVQEIVDFAKQLPGFLQLSREDQIALLKTSAIEVMLLETSRRYNPGSESITFLKDFSYNREDFAKAGLQVEFINPIFEFSRAMNELQLNDAEFALLIAISIFSADRPNVQDQLQVERLQHTYVEALHAYVSIHHPHDRLMFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVH 5awj A 2.2 BS02 YSL A 1 Y143 S233 R270 S271 S274 W282 C284 H393 Y21 S53 R90 S91 S94 W102 C104 H213 ? 0003677,0004879,0006355 ic50=0.21nM remove_due_to_license_issue P13053 26515040 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5ax3 A 2.984 BS02 5ID A 1 I22 E24 A43 D97 L98 M99 D102 K105 L147 I22 E24 A41 D95 L96 M97 D100 K103 L145 D140 K142 S144 N145 D158 T181 D138 K140 S142 N143 D156 T170 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue Ki=530nM, IC50=1200nM P28482 26733474 401 GPEMVRGQVFDVGPRYTNLSYIGEYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVAFLTEYVTRWYRAPEIMLGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5ax9 A 2.4 BS01 4KT A 1 V31 V39 A52 M105 F107 C108 G111 D115 L160 V170 D171 V20 V28 A41 M94 F96 C97 G100 D104 L149 V159 D160 D153 K155 Q157 N158 D171 T191 D142 K144 Q146 N147 D160 T166 2.7.11.1 0004672,0005524,0006468 ic50=8nM remove_due_to_license_issue IC50=8.0nM Q9UKE5 27562646 401 EIDLSALRDPAGIFELVELVGNGTYGQVYKGRHVKTGQLAAIKVMDVTGDEEEEIKQEINMLKKYSHHRNIATYYGAFIKKNPPGMDDQLWLVMEFCGAGSVTDLIKNTKGNTLKEEWIAYICREILRGLSHLHQHKVIHRDIKGQNVLLTENAEVKLVDFGVSGTPYWMAPEVIACDENPDATYDFKSDLWSLGITAIEMAEGAPPLCDMHPMRALFLIPRNPAPRLKSKKWSKKFQSFIESCLVKNHSQRPATEQLMKHPFIRDQPNERQVRIQLKDHID 5axp A 1.95 BS02 4LK A 1 H515 L625 A626 I682 Y683 F686 Q716 F719 H71 L181 A182 I238 Y239 F242 Q272 F275 3.1.4.17 0004114,0007165,0008081 ic50=0.94nM remove_due_to_license_issue IC50=0.940000nM Q9Y233 26494583 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 5axq A 1.77 BS02 4LP A 1 L625 A626 I682 Y683 F686 M703 Q716 F719 L181 A182 I238 Y239 F242 M259 Q272 F275 3.1.4.17 0004114,0007165,0008081 ic50=0.08nM remove_due_to_license_issue IC50=0.080000nM Q9Y233 26494583 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 5ayf A 2.005 BS02 C7H A 1 Y245 N263 G264 T266 Y305 Y335 X340 X341 Y130 N148 G149 T151 Y190 Y220 X223 X224 Y245 H293 H297 Y305 Y335 Y130 H178 H182 Y190 Y220 2.1.1.364 0005694,0006355,0016279,0140945 Ki=15uM remove_due_to_license_issue IC50=20000nM, Ki=15000nM Q8WTS6 27088648 402 HGVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDERTALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCISTNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITHQEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPNCIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGAAAAGGPEWYQVELKAFQATQQK 5ayt A 1.4 BS01 L6Y A 1 K15 L17 A108 L110 V121 K6 L8 A99 L101 V112 ? Ki=0.17uM remove_due_to_license_issue P02766 26639444 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5ayt B 1.4 BS01 L6Y B 1 K15 A108 L110 V121 K6 A99 L101 V112 ? Ki=0.17uM remove_due_to_license_issue P02766 26639444 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5ayy A 3.09 BS01 NTM A 1 T137 R138 H160 R161 M169 K171 S268 T137 R138 H160 R161 M169 K171 S268 R102 K139 K171 E201 D222 R102 K139 K171 E201 D222 2.4.2.19 0004514,0005515,0005737,0005829,0009435,0016757,0016763,0019363,0019674,0034213,0042802,0070062,1902494 remove_due_to_license_issue Q15274 26805589 401 MDAEGLALLLPPVTLAALVDSWLREDCPGLNYAALVSGAGPSQAALWAKSPGVLAGQPFFDAIFTQLNCQVSWFLPEGSKLVPVARVAEVRGPAHCLLLGERVALNTLARCSGIASAAAAAVEAARGAGWTGHVAGTRKTTPGFRLVEKYGLLVGGAASHRYDLGGLVMVKDNHVVAAGGVEKAVRAARQAADFALKVEVECSSLQEAVQAAEAGADLVLLDNFKPEELHPTATVLKAQFPSVAVEASGGITLDNLPQFCGPHIDVISMGMLTQAAPALDFSLKLFAKE 5ayy G 3.09 BS01 NTM G 1 T137 R138 H160 R161 M169 K171 S268 T137 R138 H160 R161 M169 K171 S268 R102 K139 K171 E201 D222 R102 K139 K171 E201 D222 2.4.2.19 0004514,0005515,0005737,0005829,0009435,0016757,0016763,0019363,0019674,0034213,0042802,0070062,1902494 remove_due_to_license_issue Q15274 26805589 401 MDAEGLALLLPPVTLAALVDSWLREDCPGLNYAALVSGAGPSQAALWAKSPGVLAGQPFFDAIFTQLNCQVSWFLPEGSKLVPVARVAEVRGPAHCLLLGERVALNTLARCSGIASAAAAAVEAARGAGWTGHVAGTRKTTPGFRLVEKYGLLVGGAASHRYDLGGLVMVKDNHVVAAGGVEKAVRAARQAADFALKVEVECSSLQEAVQAAEAGADLVLLDNFKPEELHPTATVLKAQFPSVAVEASGGITLDNLPQFCGPHIDVISMGMLTQAAPALDFSLKLFAKE 5ayy I 3.09 BS01 NTM I 1 T137 R138 H160 R161 M169 K171 S268 T137 R138 H160 R161 M169 K171 S268 R102 K139 K171 E201 D222 R102 K139 K171 E201 D222 2.4.2.19 0004514,0005515,0005737,0005829,0009435,0016757,0016763,0019363,0019674,0034213,0042802,0070062,1902494 remove_due_to_license_issue Q15274 26805589 401 MDAEGLALLLPPVTLAALVDSWLREDCPGLNYAALVSGAGPSQAALWAKSPGVLAGQPFFDAIFTQLNCQVSWFLPEGSKLVPVARVAEVRGPAHCLLLGERVALNTLARCSGIASAAAAAVEAARGAGWTGHVAGTRKTTPGFRLVEKYGLLVGGAASHRYDLGGLVMVKDNHVVAAGGVEKAVRAARQAADFALKVEVECSSLQEAVQAAEAGADLVLLDNFKPEELHPTATVLKAQFPSVAVEASGGITLDNLPQFCGPHIDVISMGMLTQAAPALDFSLKLFAKE 5b0x A 2.3 BS01 HCK A 1 V66 K68 I95 F113 V116 N117 N118 I174 D175 V65 K67 I94 F112 V115 N116 N117 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.02uM remove_due_to_license_issue IC50=20nM P68400 26850376 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 5b1s A 1.58 BS02 BSX A 1 W19 Q64 Y73 T169 T170 D171 Q201 Y237 W19 Q64 Y73 T169 T170 D171 Q201 Y237 2.5.1.16 0003824,0004766,0005829,0006596,0008295,0016740 ic50=124uM remove_due_to_license_issue Q4DA73 28751689 502 MPGSELISGGWFREENDQWPGQAMSLRVEKVLYDAPTKFQHLTIFESDPKGPWGTVMALDGCIQVTDYDEFVYHEVLGHTSLCSHPKPERVLIIGGGDGGVLREVLRHGTVEHCDLVDIDGEVMEQSKQHFPQISRSLADPRATVRVGDGLAFVRQTPDNTYDVVIIDTTDPAGPASKLFGEAFYKDVLRILKPDGICCNQGESIWLDLELIEKMSRFIRETGFASVQYALMHVPTYPCGSIGTLVCSKKAGVDVTKPLRPVEDMPFAKDLKYYDSEMHKASFALPRFARHINN 5b25 A 1.9 BS02 4QJ A 1 I371 H373 L388 F392 L409 S420 Q421 G423 F424 F427 I223 H225 L240 F244 L261 S272 Q273 G275 F276 F279 3.1.4.17 0004114,0007165,0008081 Ki=0.058nM remove_due_to_license_issue IC50=0.058000nM Q01064 26789933 603 TYSTAVLNCLKNLDLWCFDVFSLNQAADDHALRTIVFELLTRHNLISRFKIPTVFLMSFLDALETGYGKYKNPYHNQIHAADVTQTVHCFLLRTGMVHCLSEIELLAIIFAAAIHDYEHTGTTNSFHIQTKSECAIVYNDRSVLENHHISSVFRLMQDDEMNIFINLTKDEFVELRALVIEMVLATDMSCHFQQVKTMKTALQQLERIDKPKALSLLLHAADISHPTKQWLVHSRWTKALMEEFFRQGDKEAELGLPFSPLCDRTSTLVAQSQIGFIDFIVEPTFSVLTDVAEKSVQPLAGDPNPDVVSFRSTWVKRIQENKQKWKERAASGITN 5b4k A 2.9 BS02 6DT A 1 I682 Y683 F686 M703 E711 G715 Q716 F719 I238 Y239 F242 M259 E267 G271 Q272 F275 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Q9Y233 27301679 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 5b4l A 2.4 BS02 6DW A 1 H515 L665 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 H71 L221 I238 Y239 F242 P258 M259 E267 V268 G271 Q272 F275 3.1.4.17 0004114,0007165,0008081 ic50=0.76nM remove_due_to_license_issue IC50=0.760000nM Q9Y233 27301679 1003 EWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 5b5b A 2.0 BS02 AKX A 1 Y143 L223 L226 V230 S233 R270 S271 S274 W282 C284 V296 A299 H393 Q396 Y30 L52 L55 V59 S62 R99 S100 S103 W111 C113 V125 A128 H222 Q225 ? 0003677,0004879,0006355 ic50=0.43nM remove_due_to_license_issue P13053 27294600 501 SPLKDSLRPKLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5b5f A 1.2 BS01 6F3 A 1 S27 Y43 S45 G48 N49 A50 W79 S88 W108 L110 D128 S12 Y28 S30 G33 N34 A35 W64 S73 W93 L95 D113 ? 0009374 Kd=5.6uM remove_due_to_license_issue P22629 27905160 200 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKP 5b5f C 1.2 BS01 6F3 C 1 S27 Y43 W79 A86 S88 W92 W108 D128 S12 Y28 W64 A71 S73 W77 W93 D113 ? 0009374 Kd=5.6uM remove_due_to_license_issue P22629 27905160 200 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKP 5b5g C 1.5 BS02 6FX C 1 S27 Y43 W79 S88 W92 W108 D128 S12 Y28 W64 S73 W77 W93 D113 ? 0009374 Kd=5.6uM remove_due_to_license_issue P22629 27905160 202 GITGTWYNQLGSTFIVTAGADGALTGTYESAVGNAESRYVLTGRYDSAPATDGSGTALGWTVAWKNNYRNAHSATTWSGQYVGGAEARINTQWLLTSGTTEANAWKSTLVGHDTFTKVKP 5b5o A 1.2 BS05 WMM A 1 L218 H222 H232 L239 F241 P242 I243 Y244 L115 H119 H129 L136 F138 P139 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=1900nM remove_due_to_license_issue P45452 27966948 307 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGFMLPDDDVQGIQSLYGPGDEDP 5b5p A 1.6 BS06 WNN A 1 L218 H222 E223 H226 H232 L239 F241 P242 I243 Y244 T245 T247 F252 P255 L115 H119 E120 H123 H129 L136 F138 P139 I140 Y141 T142 T144 F147 P150 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.2nM remove_due_to_license_issue IC50=0.200000nM P45452 27966948 306 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGHFMLPDDDVQGIQSLYGPGDED 5bml A 2.95 BS01 4TW A 1 R84 G85 F87 G88 E89 V90 A103 K105 F120 Y155 M156 A215 D216 F368 R79 G80 F82 G83 E84 V85 A98 K100 F115 Y150 M151 A210 D211 F361 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=10.0nM Q13464 26039570 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEETFPIPKAFVGNQLPFVGFTYYSNRRY 5bms A 2.903 BS01 4T6 A 1 I327 G328 V335 A348 F397 L398 G401 D444 L447 I29 G30 V37 A50 F99 L100 G103 D146 L149 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96013 26030457 601 GSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 5bnj A 2.64 BS01 4TV A 1 V27 Y32 A50 K52 F97 A100 H106 L158 D173 R356 V29 Y34 A52 K54 F99 A102 H108 L156 D171 R337 D151 K153 N156 D173 N181 T196 D149 K151 N154 D171 N179 T183 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=7.2nM P49336 26502155 501 DKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKANQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEE 5bnm A 1.7 BS01 4VK A 1 W32 R36 C112 G209 V212 A246 N247 I250 N274 W32 R36 C112 G209 V212 A246 N247 I250 N274 2.3.1.180 0004315,0005737,0005829,0006631,0006633,0016746,0033818,0044281 ic50=15uM remove_due_to_license_issue P0A6R0 27626097 402 MYTKIIGTGSYLPEQVRTNADLEKMVDTSDEWIVTRTGIRERHIAAPNETVSTMGFEAATRAIEMAGIEKDQIGLIVVATTSATHAFPSAACQIQSMLGIKGCPAFDVAAACAGFTYALSVADQYVKSGAVKYALVVGSDVLARTCDPTDRGTIIIFGDGAGAAVLAASEEPGIISTHLHADGSYGELLTLPNADRVNPENSIHLTMAGNEVFKVAVTELAHIVDETLAANNLDRSQLDWLVPHQANLRIISATAKKLGMSMDNVVVTLDRHGNTSAASVPCALDEAVRDGRIKPGQLVLLEAFGGGFTWGSALVRF 5bnr A 1.89 BS01 4VL A 1 C112 I156 M207 G209 V212 F213 H244 A246 I250 N274 F304 C112 I156 M199 G201 V204 F205 H236 A238 I242 N266 F296 2.3.1.180 0004315,0005737,0005829,0006631,0006633,0016746,0033818,0044281 ic50=0.53uM remove_due_to_license_issue P0A6R0 27626097 401 MYTKIIGTGSYLPEQVRTNADLEKMVDTSDEWIVTRTGIRERHIAAPNETVSTMGFEAATRAIEMAGIEKDQIGLIVVATTSATHAFPSAACQIQSMLGIKGCPAFDVAAACAGFTYALSVADQYVKSGAVKYALVVGSDVLARTCDPTDRGTIIIFGDGAGAAVLAASEEPGIISTHLHADGSYGELLTLPNAIHLTMAGNEVFKVAVTELAHIVDETLAANNLDRSQLDWLVPHQANLRIISATAKKLGMSMDNVVVTLDRHGNTSAASVPCALDEAVRDGRIKPGQLVLLEAFGGGFTWGSALVRF 5bns A 2.2 BS01 4VM A 1 T28 W32 C112 R151 M207 G209 V212 A216 H244 A246 I250 N274 T28 W32 C112 R151 M207 G209 V212 A216 H244 A246 I250 N274 2.3.1.180 0004315,0005737,0005829,0006631,0006633,0016746,0033818,0044281 ic50=0.095uM remove_due_to_license_issue P0A6R0 27626097 401 MYTKIIGTGSYLPEQVRTNADLEKMVDTSDEWIVTRTGIRERHIAAPNETVSTMGFEAATRAIEMAGIEKDQIGLIVVATTSATHAFPSAACQIQSMLGIKGCPAFDVAAACAGFTYALSVADQYVKSGAVKYALVVGSDVLARTCDPTDRGTIIIFGDGAGAAVLAASEEPGIISTHLHADGSYGELLTLPNADRVNPENSIHLTMAGNEVFKVAVTELAHIVDETLAANNLDRSQLDWLVPHQANLRIISATAKKLGMSMDNVVVTLDRHGNTSAASVPCALDEAVRDGRIKPGQLVLLEAFGGGFTWGSALVRF 5bns B 2.2 BS01 4VM B 1 T28 W32 R36 C112 R151 I155 L189 M207 V212 H244 A246 I250 N274 F304 T28 W32 R36 C112 R151 I155 L189 M207 V212 H244 A246 I250 N274 F304 2.3.1.180 0004315,0005737,0005829,0006631,0006633,0016746,0033818,0044281 ic50=0.095uM remove_due_to_license_issue P0A6R0 27626097 401 MYTKIIGTGSYLPEQVRTNADLEKMVDTSDEWIVTRTGIRERHIAAPNETVSTMGFEAATRAIEMAGIEKDQIGLIVVATTSATHAFPSAACQIQSMLGIKGCPAFDVAAACAGFTYALSVADQYVKSGAVKYALVVGSDVLARTCDPTDRGTIIIFGDGAGAAVLAASEEPGIISTHLHADGSYGELLTLPNADRVNPENSIHLTMAGNEVFKVAVTELAHIVDETLAANNLDRSQLDWLVPHQANLRIISATAKKLGMSMDNVVVTLDRHGNTSAASVPCALDEAVRDGRIKPGQLVLLEAFGGGFTWGSALVRF 5boj A 1.75 BS01 4TX A 1 K15 A108 A109 K6 A99 A100 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=100nM remove_due_to_license_issue Kd=100nM, IC50=180000nM P02766 26214366 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5boj B 1.75 BS01 4TX B 1 K15 A108 A109 L110 K6 A99 A100 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=100nM remove_due_to_license_issue Kd=100nM, IC50=180000nM P02766 26214366 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5bot A 1.85 BS01 4UM A 1 H222 A238 L239 F241 P242 T245 T247 H119 A135 L136 F138 P139 T142 T144 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=39uM remove_due_to_license_issue IC50=39000nM P45452 22017539 301 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGFMLPDDDVQGIQSLYGPGDED 5boy A 2.03 BS06 4UE A 1 H222 A238 L239 F241 P242 I243 T245 T247 F252 H119 A135 L136 F138 P139 I140 T142 T144 F146 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=2.5uM remove_due_to_license_issue IC50=2500nM P45452 22017539 306 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGFMLPDDDVQGIQSLYGPGDED 5bpa A 1.79 BS06 4UF A 1 L185 L218 H222 L239 F241 I243 Y244 Y246 T247 K249 F252 L82 L115 H119 L136 F138 I140 Y141 Y143 T144 K146 F149 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=0.001uM remove_due_to_license_issue IC50=1nM P45452 22017539 306 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPGDED 5bpe A 2.7 BS01 E22 A 1 H40 E71 N126 L127 S128 T142 A144 G145 C147 H161 I162 G163 G164 H40 E71 N126 L127 S128 T142 A144 G145 C147 H161 I162 G163 G164 H40 E71 G145 C147 H40 E71 G145 C147 ? 0004197,0006508,0008234,0039618,0043657 remove_due_to_license_issue A0A0X1KHD2 26571192 201 GPAFEFAVAMMKRNSSTVKTEYGEFTMLGIYDRWAVLPRHSKPGPTILMNDQEVGVLDAKELVDKDGTNLELTLLKLNRNEKFRDIRGFLAKEEVEVNEAVLAINTSKFPNMYIPVGQVTEYGFLNLSGKPTKRMLMYNFPTKAGQCGGVLMSTGKVLGIHIGGNGRQGFSAALLKHYFN 5bpp A 2.03 BS02 A4Z A 1 Q136 Y267 G269 M270 H295 E296 H299 E318 Y378 Y383 Q133 Y264 G266 M267 H292 E293 H296 E315 Y375 Y380 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=15.86uM remove_due_to_license_issue P09960 27126280 706 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKVD 5bq0 A 1.57 BS01 4US A 1 L408 T410 V416 A428 Y476 M477 A478 N479 G480 C481 L528 L20 T22 V28 A40 Y88 M89 A90 N91 G92 C93 L140 D521 A523 R525 N526 D539 F559 D133 A135 R137 N138 D151 F165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=15nM remove_due_to_license_issue IC50=15nM Q06187 26320619 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 5bqg A 1.436 BS01 4UJ A 1 P124 S127 T131 P120 S123 T127 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=17.4uM remove_due_to_license_issue O14684 26653180 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5bqh A 1.601 BS01 4UK A 1 A123 P124 S127 V128 A119 P120 S123 V124 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50<3nM remove_due_to_license_issue O14684 26653180 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5bqi A 1.88 BS01 4UL A 1 A123 P124 S127 V128 A119 P120 S123 V124 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=0.9nM remove_due_to_license_issue O14684 26653180 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5bqs A 1.9 BS01 4VN A 1 R37 C112 F157 M212 V217 H249 A251 R254 N279 F311 R36 C111 F156 M211 V216 H248 A250 R253 N278 F310 2.3.1.180 0004315,0005737,0006633,0016746,0033818 ic50=2.3uM remove_due_to_license_issue C1CIR8 27626097 402 AFAKISQVAHYVPEQVVTNHDLAQIMDTNDEWISSRTGIRQRHISRTESTSDLATEVAKKLMAKAGITGKELDFIILATITPDSMMPSTAARVQANIGANKAFAFDLTAACSGFVFALSTAEKFIASGRFQKGLVIGSETLSKAVDWSDRSTAVLFGDGAGGVLLEASEQEHFLAESLNSDGSRSECLTYGHSGLHSPFSDQESADSFLKMDGRTVFDFAIRDVAKSIKQTIDESPIEVTDLDYLLLHQANDRILDKMARKIGVDRAKLPANMMEYGNTSAASIPILLSECVEQGLIPLDGSQTVLLSGFGGGLTWGTLILTI 5bqs B 1.9 BS01 4VN B 1 R37 C112 L189 M212 G214 V217 H249 A251 N279 F311 R36 C111 L188 M211 G213 V216 H248 A250 N278 F310 2.3.1.180 0004315,0005737,0006633,0016746,0033818 ic50=2.3uM remove_due_to_license_issue C1CIR8 27626097 402 AFAKISQVAHYVPEQVVTNHDLAQIMDTNDEWISSRTGIRQRHISRTESTSDLATEVAKKLMAKAGITGKELDFIILATITPDSMMPSTAARVQANIGANKAFAFDLTAACSGFVFALSTAEKFIASGRFQKGLVIGSETLSKAVDWSDRSTAVLFGDGAGGVLLEASEQEHFLAESLNSDGSRSECLTYGHSGLHSPFSDQESADSFLKMDGRTVFDFAIRDVAKSIKQTIDESPIEVTDLDYLLLHQANDRILDKMARKIGVDRAKLPANMMEYGNTSAASIPILLSECVEQGLIPLDGSQTVLLSGFGGGLTWGTLILTI 5brn A 2.3 BS02 4X2 A 1 I135 D137 T138 G139 T141 K165 F186 V187 I113 D115 T116 G117 T119 K143 F164 V165 E133 D134 D137 F186 R199 E111 D112 D115 F164 R177 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.5uM remove_due_to_license_issue P00492 26368337 302 SPGVVISDDEPGYDLDLFAIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVAVISETGKAKYK 5bry A 1.34 BS01 4UY B 1 D25 G27 A28 D30 G48 P81 V82 I84 D25 G27 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 26306007 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5bry B 1.34 BS01 4UY B 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.0015nM remove_due_to_license_issue P03366 26306007 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5bs4 A 1.29 BS01 4UX A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.0099nM remove_due_to_license_issue P03366 26306007 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5bs4 B 1.29 BS01 4UX A 1 D25 A28 D30 P81 V82 I84 D25 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 26306007 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5bsk A 2.61 BS01 4X7 A 1 I135 D137 T138 G139 T141 K165 F186 V187 I110 D112 T113 G114 T116 K140 F161 V162 E133 D134 D137 F186 R199 E108 D109 D112 F161 R174 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 remove_due_to_license_issue Ki=600nM P00492 26368337 301 SPGVVISDDGYDLDLFAIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVAVISETGKAKYKA 5btx A 2.1 BS01 CMP A 1 S59 Y61 Y69 N79 H106 T108 S59 Y61 Y69 N79 H106 T108 Kd=280uM remove_due_to_license_issue 26294765 201 MVTKIIWVSNNGKPNLKIEFVSEEEKSNFFKEVKKKASELGLNFPLVQGSGNSLLIEASNYPINPCGCYISPGGKLAINFGKVELSHFILPKVGVKTEHAEIFKDHNTIFFHKHKLPGVNSELTFIPTGTPV 5bue A 2.4 BS01 4V8 A 1 I29 G35 V37 A50 K52 Q103 D104 M106 E107 T108 K112 L154 C164 D165 I21 G27 V29 A42 K44 Q95 D96 M98 E99 T100 K104 L146 C156 D157 D147 K149 S151 N152 D165 T188 D139 K141 S143 N144 D157 T165 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.003uM remove_due_to_license_issue P28482 26144345 401 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVATRWYRAPEIMLNTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5bui A 2.12 BS01 4V9 A 1 I29 Y34 A50 Q103 M106 E107 T108 K112 L154 C164 D165 I21 Y26 A42 Q95 M98 E99 T100 K104 L146 C156 D157 D147 K149 S151 N152 D165 T188 D139 K141 S143 N144 D157 T170 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.089uM remove_due_to_license_issue P28482 26144345 402 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDTRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5buj A 1.85 BS01 4VB A 1 I29 Y34 A50 K52 Q103 M106 E107 T108 K112 L154 C164 D165 I23 Y28 A44 K46 Q97 M100 E101 T102 K106 L148 C158 D159 D147 K149 S151 N152 D165 T188 D141 K143 S145 N146 D159 T167 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.005uM remove_due_to_license_issue P28482 26144345 401 AGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVATRWYRAPEIMLNTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5bv3 A 2.25 BS01 M7G A 1 W161 E171 D194 M195 K196 H259 S263 H270 W147 E157 D178 M179 K180 H243 S247 H254 3.6.1.59 0000288,0000290,0000340,0000932,0000956,0005515,0005634,0005737,0005739,0006970,0006979,0007584,0009267,0009408,0016787,0016818,0031086,0042802,0042803,0044692,0046982,0048471,0050072,0090342,0106095,0110156,0140932 Kd=68nM remove_due_to_license_issue Q06151 26258763 401 MFASLIKRFQFVSVLDSNPQTKVMSLLGTIDNKDAIITAEKTHFLFDETDGRSTPVLYNCENEYSCINGIQELKEITSNDIYYWGLSVIKQDMESNPTAKLNLIWPATPIHIKKYEQQNFHLVRETPEMYKRIVQPYIEEMCGRLKWVNNILYEGAESERVVYKDFSEKDDGFLILPDMKWDGMNLDSLYLVAIVYRTDIKTIRDLRYSDRQWLINLNNKIRSIVPGCYNYAVHPDELRILVHYQPSYYHFNIHIVNIKHPGLGNSIAAGKAILLEDIIEMLNYLGPEGYMNKTITYAIGENHDLWKRGLEEELTKQLERDGIPKIPKI 5bvd A 1.9 BS01 4VF A 1 E31 G32 Y34 G35 V37 A50 K52 I54 M106 E107 T108 K112 L154 D165 E25 G26 Y28 G29 V31 A44 K46 I48 M100 E101 T102 K106 L148 D159 D147 K149 S151 N152 D165 T188 D141 K143 S145 N146 D159 T166 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.16nM remove_due_to_license_issue IC50=0.160000nM P28482 26259804 401 AGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVTRWYRAPEIMLNTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5bve A 2.0 BS01 4VG A 1 G32 Y34 G35 V37 A50 K52 M106 T108 K112 L154 C164 D165 G26 Y28 G29 V31 A44 K46 M100 T102 K106 L148 C158 D159 D147 K149 S151 N152 D165 T188 D141 K143 S145 N146 D159 T166 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.01nM remove_due_to_license_issue IC50=0.010000nM P28482 26259804 401 AGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVTRWYRAPEIMLNTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5bvf A 1.9 BS01 4VJ A 1 I29 G32 Y34 G35 V37 A50 K52 M106 T108 D109 K112 L154 C164 D165 I23 G26 Y28 G29 V31 A44 K46 M100 T102 D103 K106 L148 C158 D159 D147 K149 S151 N152 D165 D141 K143 S145 N146 D159 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.19nM remove_due_to_license_issue IC50=52nM P28482 26259804 401 AGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVRWYRAPEIMTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5bvk A 2.29 BS01 4VC A 1 E672 M676 L679 I685 T701 F762 A783 D784 F785 E53 M57 L60 I66 T82 F129 A150 D151 F152 D766 R770 N771 D784 A793 D133 R137 N138 D151 A160 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=>100000nM Q08345 26191369 1007 DFPRSRLRFKEKLGEGQFGEVHLCEVDSHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALN 5bvn A 2.21 BS01 4VD A 1 L616 V624 A653 K655 E672 M676 L679 I685 M699 T701 Y703 M704 F762 L773 A783 D784 L13 V21 A34 K36 E53 M57 L60 I66 M80 T82 Y84 M85 F129 L140 A150 D151 D766 R770 N771 D784 A793 D133 R137 N138 D151 A160 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Q08345 26191369 1002 DFPRSRLRFKEKLGEGQFGEVHLCEVDSHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALN 5bvo A 1.98 BS01 4VE A 1 A653 K655 E672 I675 M676 L679 I685 M699 T701 M704 L773 A783 D784 F785 A32 K34 E51 I54 M55 L58 I64 M78 T80 M83 L138 A148 D149 F150 D766 R770 N771 D784 A793 D131 R135 N136 D149 A158 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Q08345 26191369 1008 DFPRSRLRFKEKLGEFGEVHLCEVDSHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALN 5bvw A 1.94 BS01 1N1 A 1 A653 K655 M676 T701 Y703 M704 E705 G707 L773 F785 A34 K36 M57 T82 Y84 M85 E86 G88 L140 F152 D766 R770 N771 D784 A793 D133 R137 N138 D151 A156 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Kd=0.69nM, IC50=4.8nM Q08345 26191369 1009 DFPRSRLRFKEKLGEGQFGEVHLCEVDSHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALN 5bw4 A 2.1 BS01 SAM A 1 G38 T39 T44 D61 P62 R66 W113 L116 G34 T35 T40 D57 P58 R62 W109 L112 ? Kd=68uM remove_due_to_license_issue C7Q5P8 26609134 301 TALKVLAGKKLTDLDPDEWAKAQASAERILVDVGTGDARTAYRQAIAHPEWLVVGVDPAWQRMTETAVRAARKPAKGGAPNLVLVSSAIETVPAALHGVADEVMVLMPWGKLLRGVVLGEADVLSGLRAVAKPGAPLEISIGTSIWREPIPLEIRDLPELTPETVVSTGLTDRLAALGWQVADVRLVPHTETVLHLRAVAVDPRD 5bwb A 2.57 BS01 4VV A 1 Y70 D72 Y121 E278 W279 F330 F331 Y67 D69 Y118 E275 W276 F327 F328 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 26327369 604 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 5bwc A 2.45 BS01 HBP A 1 Y70 W84 G119 Y121 W279 F290 F330 Y334 Y67 W81 G116 Y118 W276 F287 F327 Y331 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=0.061uM remove_due_to_license_issue P04058 26327369 603 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 5byi A 1.15 BS03 4WA A 1 H94 H119 L197 T198 T199 P201 H91 H116 L194 T195 T196 P198 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=30.7nM remove_due_to_license_issue Ki=106nM P00918 26199669 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5byy A 2.79 BS01 4WG A 1 I61 L137 M140 E141 L189 I13 L89 M92 E93 L141 D182 K184 S186 N187 D200 T224 D134 K136 S138 N139 D152 T168 2.7.11.24 0004672,0004707,0005524,0006468 remove_due_to_license_issue Kd=80nM, IC50=300nM Q13164 27139631 401 FDVGDEYEIIETIGNGAYGVVSSARRRLTGQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARREG 5byz A 1.65 BS01 4WE A 1 I61 G62 Y66 K84 I115 L137 M140 D143 H145 Q146 L189 I14 G15 Y19 K37 I68 L90 M93 D96 H98 Q99 L142 D182 K184 S186 N187 D200 T224 D135 K137 S139 N140 D153 T177 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.042uM remove_due_to_license_issue Q13164 27139631 401 TFDVGDEYEIIETIGNGAYGVVSSARRRLTGQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSPAEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARREGI 5c0k A 2.2 BS02 4WK A 1 L307 T308 D309 W310 E314 Q319 W323 L59 T60 D61 W62 E66 Q71 W75 2.3.2.27 ic50=1200uM remove_due_to_license_issue P98170 26218264 404 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECL 5c1w A 1.7 BS02 4XS A 1 L665 Y683 M703 Q716 F719 L229 Y247 M267 Q280 F283 3.1.4.17 0004114,0007165,0008081 Ki=8.7uM remove_due_to_license_issue Ki=8700nM Q9Y233 26378882 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEET 5c1x A 1.86 BS01 GHX A 1 H40 E71 L127 S128 T142 K143 C147 H161 I162 G163 G164 F170 H41 E72 L128 S129 T143 K144 C148 H162 I163 G164 G165 F171 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 27185390 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5c1y A 1.97 BS01 GHY A 1 R39 H40 E71 L127 S128 T142 K143 C147 H161 I162 G163 G164 R40 H41 E72 L128 S129 T143 K144 C148 H162 I163 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 27185390 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5c20 A 2.75 BS01 GHZ A 1 R39 H40 E71 L127 S128 T142 K143 C147 H161 I162 G163 G164 R40 H41 E72 L128 S129 T143 K144 C148 H162 I163 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 27185390 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5c26 A 1.95 BS02 50H A 1 F382 V385 A400 A451 E452 G454 P455 K458 L501 F20 V23 A38 A89 E90 G92 P93 K96 L139 D494 A496 R498 N499 D512 K533 D132 A134 R136 N137 D150 K171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.17uM remove_due_to_license_issue IC50=27nM, EC50=244nM P43405 26381330 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNH 5c28 A 1.56 BS02 4XV A 1 I682 Y683 M703 Q716 F719 I246 Y247 M267 Q280 F283 3.1.4.17 0004114,0007165,0008081 Ki=2.2uM remove_due_to_license_issue Ki=2200nM Q9Y233 26378882 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEET 5c29 A 2.05 BS02 4XY A 1 H515 I682 Y683 Q716 F719 H62 I229 Y230 Q263 F266 3.1.4.17 0004114,0007165,0008081 Ki=880nM remove_due_to_license_issue Ki=880nM Q9Y233 26378882 803 LPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 5c2a A 2.0 BS02 4Y2 A 1 Y514 H515 I682 Y683 F686 M703 Q716 F719 Y78 H79 I246 Y247 F250 M267 Q280 F283 3.1.4.17 0004114,0007165,0008081 Ki=4.8nM remove_due_to_license_issue Ki=4.8nM Q9Y233 26378882 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 5c2h B 2.09 BS02 4XU B 1 H515 I682 Y683 F686 P702 M703 E711 V712 G715 Q716 F719 H79 I246 Y247 F250 P266 M267 E275 V276 G279 Q280 F283 3.1.4.17 0004114,0007165,0008081 Ki=0.0082nM remove_due_to_license_issue Ki=0.008200nM Q9Y233 26378882 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRG 5c2o A 2.35 BS03 TTP A 1 T42 Y44 G46 G47 A49 N75 Q79 T38 Y40 G42 G43 A45 N71 Q75 ? 0000166,0003824,0004132,0005737,0008270,0009972,0016787,0046872 remove_due_to_license_issue Q8DSE5 27377385 704 LSWQDYFMANAELISKRSTCNRAYVGAVLVKNNRIIATGYNGGVADTDNCDDVGHEMEDGHCIRTVHAEMNALIQCAKEGISANNTEIYVTHFPCINCTKALLQAGVKKITYNTAYRIHPFAIELMTQKEVEYVQHDVPRVKLG 5c2o B 2.35 BS03 TTP B 1 T42 Y44 G46 G47 A49 N75 Q79 T38 Y40 G42 G43 A45 N71 Q75 ? 0000166,0003824,0004132,0005737,0008270,0009972,0016787,0046872 remove_due_to_license_issue Q8DSE5 27377385 704 LSWQDYFMANAELISKRSTCNRAYVGAVLVKNNRIIATGYNGGVADTDNCDDVGHEMEDGHCIRTVHAEMNALIQCAKEGISANNTEIYVTHFPCINCTKALLQAGVKKITYNTAYRIHPFAIELMTQKEVEYVQHDVPRVKLG 5c3k A 2.02 BS02 4XF A 1 L307 T308 W310 E314 Q319 W323 L59 T60 W62 E66 Q71 W75 2.3.2.27 ic50=110uM remove_due_to_license_issue P98170 26218264 402 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c3p A 2.1 BS01 AKG A 1 R190 Y194 H214 L223 H271 V273 R286 S288 F292 R186 Y190 H210 L219 H267 V269 R282 S284 F288 R190 A211 H214 D216 H271 R186 A207 H210 D212 H267 ? 0044283,0046872,0051213 Kd=34.4uM remove_due_to_license_issue Q7RYZ9 26429971 402 MEKAAVNEDGLVIPLIDFSKFLEGDETLKLETAKAILHGFQTAGFIYLKNIPIQPDFREHVFNTSAKFFKLPKEKKLEVGWTTPEANRGYSAPGREKVTQLTDPAEIEKAPDIKESYEIGREDEPGHPNPWPAEQDDLVGFKSTMNNFFDQCKALHIEVMRAIAVGMGIDANYFDSFVDVGDNILRLLHYPAVKSEVFKINPGQVRAGEHTDYGSITLLFQDSRGGLQVKSPNGQFIDATPIENTVVVNAGDLLARWSNDTIKSTVHRVVEPPKQEDVHPPRYSIAYFCNPNHKSYIEAIPGTYAAESERKYEGINSGKYLVQRLAATY 5c42 A 3.5 BS01 29T A 1 L100 P101 V106 V108 V179 Y181 Y188 V189 G190 F227 W229 P236 Y318 L97 P98 V103 V105 V176 Y178 Y185 V186 G187 F224 W226 P233 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 26487915 601 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLPKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQ 5c4k A 3.05 BS01 GET A 1 D197 D220 E235 E238 E239 W271 Y278 D196 D219 E234 E237 E238 W270 Y277 K46 K45 ? 0000166,0016301,0046872 remove_due_to_license_issue O68183 26802312 401 RTYTFDQVEKAIEQLYPDFTINTIQISGKGNDCIAYEINRDFIFKFPKHSRGSTNLFNEVNILKRIHNKLPLPIPEVVFTGMPSETYQMSFAGFTKIKGVPLTPLLLNNLPKQSQNQAAKDLARFLSELHSINISGFKSNLVLDFREKINEDNKKIKKLLSRELKGPQMKKVDDFYRDILENEIYFKYYPCLIHNDFSSDHILFDTEKNTICGIIDFGDAAISDPDNDFISLMEDDEEYGMEFVSKILNHYKHKDIPTVLEKYRMKEKYWSFEKIIYGKEYGYMDWYEEGLNEIRS 5c4l B 2.35 BS01 SIS B 1 E235 E239 E268 W271 E235 E239 E268 W271 K46 K46 ? 0000166,0016301,0046872 Kd=2.3uM remove_due_to_license_issue O68183 26802312 401 MRTYTFDQVEKAIEQLYPDFTINTIQISGKGNDCIAYEINRDFIFKFPKHSRGSTNLFNEVNILKRIHNKLPLPIPEVVFTGMPSETYQMSFAGFTKIKGVPLTPLLLNNLPKQSQNQAAKDLARFLSELHSINISGFKSNLVLDFREKINEDNKKIKKLLSRELKGPQMKKVDDFYRDILENEIYFKYYPCLIHNDFSSDHILFDTEKNTICGIIDFGDAAISDPDNDFISLMEDDEEYGMEFVSKILNHYKHKDIPTVLEKYRMKEKYWSFEKIIYGKEYGYMDWYEEGLNEIRS 5c4o A 2.24 BS01 4F1 A 1 L324 T325 I328 Q329 L483 Q484 Q487 A496 A497 F498 L501 L505 F506 L58 T59 I62 Q63 L217 Q218 Q221 A230 A231 F232 L235 L239 F240 ? 0003677,0004879,0005634,0006355 ic50=6.1nM remove_due_to_license_issue IC50=7.8nM, EC50=16nM P51449 26640126 601 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5c4s A 2.23 BS01 4Y5 A 1 L324 T325 I328 Q329 M358 V480 L483 Q484 Q487 A496 A497 F498 L501 L505 F506 L58 T59 I62 Q63 M92 V214 L217 Q218 Q221 A230 A231 F232 L235 L239 F240 ? 0003677,0004879,0005634,0006355 ic50=3.8nM remove_due_to_license_issue IC50=3.8nM P51449 26640126 601 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5c4t A 1.77 BS01 4Y6 A 1 L324 T325 I328 Q329 M358 L483 A496 A497 F498 L501 Y502 L505 F506 L58 T59 I62 Q63 M92 L217 A230 A231 F232 L235 Y236 L239 F240 ? 0003677,0004879,0005634,0006355 ic50=21.8nM remove_due_to_license_issue P51449 26640126 601 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5c4u A 2.08 BS01 4Y7 A 1 L324 T325 I328 Q329 L483 Q484 Q487 A496 A497 F498 L501 Y502 L505 F506 L58 T59 I62 Q63 L217 Q218 Q221 A230 A231 F232 L235 Y236 L239 F240 ? 0003677,0004879,0005634,0006355 ic50=1.9nM remove_due_to_license_issue P51449 26640126 601 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5c51 A 3.426 BS01 dna P 0 R579 S764 P765 D769 A862 N864 R869 R948 R447 S551 P552 D556 A649 N651 R656 R735 2.7.7.7,3.1.11.-,4.2.99.- 0000262,0002020,0003677,0003682,0003887,0005515,0005739,0005759,0005760,0006259,0006260,0006261,0006264,0006281,0006284,0006287,0008310,0008408,0016787,0016829,0032991,0034061,0042645,0043231,0045004,0051575,0071897 remove_due_to_license_issue P54098 26124101 3 ~ 24 MLSRGLHEQIFGQGGEMPGEAAVRRSVEHLQKHGLWGQPAVPLPDVELRLPPLYGDNLDQHFRLLAQKQSLPYLEAANLLLQAQLPPKPPAWAWAEGWTRYGPEGEAVPVAIPEERALVFDVEVCLAEGTCPTLAVAISPSAWYSWCSQRLVEERYSWTSQLSPADLIPLEVQEQLVVGHNVSFDRAHIREQYLIQGSRMRFLDTMSMHMAISGLSSFQRSLWIAAKAISSWDWLDISSVNSLAEVHRLYVGGPPLEKEPRELFVKGTMKDIRENFQDLMQYCAQDVWATHEVFQQQLPLFLERCPHPVTLAGMLEMGVSYLPVNQNWERYLAEAQGTYEELQREMKKSLMDLANDACQLLSGERYKEDPWLWDLEWDLQEFKQKKAKKVKKEPATALGPCSEEEEFQQDVMARACLQKLKGTTELLPKRPQHLPGHPGWYRKLCPRLDDPAWTPGPSLLSLQMRVTPKLMALTWDGFPLHYSERHGWGYLNLAKLPTGTTLESAGVVCPYRAIESLYRKHCLEPYNDVDIPGCWFFKLPHKDGNSCNVGSPFAKDFLPKMEDGTLQAGPGGASGPRALEINKMISFWRNAHKRISSQMVVWLPRSALPRAVIRHPDYDEEGLYGAILPQVVTAGTITRRAVEPTWLTASNARPDRVGSELKAMVQAPPGYTLVGADVDSQELWIAAVLGDAHFAGMHGCTAFGWMTLQGRKSRGTDLHSKTATTVGISREHAKRFNYGRIYGAGQPFAERLLMQFNHRLTQQEAAEKAQQMYAATKGLLRKVQRETARKSQWKKWEVVAERAWKGGTESEMFNKLESIATSDIPRTPVLGCCISRALEPSAVQEEFMTSRVNWVVQSSAVDYLHLMLVAMKWLFEEFAIDGRFCISIHDEVRYLVREEDRYRAALALQITNLLTRCMFAYKLGLNDLPQSVAFFSAVDIDRCLRKEVTMDCKTPSNPTGMERRYGIPQGEALDIYQIIELTK 5c51 A 3.426 BS02 dna T 0 K498 K561 S593 M596 R597 N803 R807 T849 I850 P857 T861 R948 G952 Y955 G956 G958 F961 T1094 N1098 K385 K429 S461 M464 R465 N590 R594 T636 I637 P644 T648 R735 G739 Y742 G743 G745 F748 T849 N853 2.7.7.7,3.1.11.-,4.2.99.- 0000262,0002020,0003677,0003682,0003887,0005515,0005739,0005759,0005760,0006259,0006260,0006261,0006264,0006281,0006284,0006287,0008310,0008408,0016787,0016829,0032991,0034061,0042645,0043231,0045004,0051575,0071897 remove_due_to_license_issue P54098 26124101 2 ~ 26 MLSRGLHEQIFGQGGEMPGEAAVRRSVEHLQKHGLWGQPAVPLPDVELRLPPLYGDNLDQHFRLLAQKQSLPYLEAANLLLQAQLPPKPPAWAWAEGWTRYGPEGEAVPVAIPEERALVFDVEVCLAEGTCPTLAVAISPSAWYSWCSQRLVEERYSWTSQLSPADLIPLEVQEQLVVGHNVSFDRAHIREQYLIQGSRMRFLDTMSMHMAISGLSSFQRSLWIAAKAISSWDWLDISSVNSLAEVHRLYVGGPPLEKEPRELFVKGTMKDIRENFQDLMQYCAQDVWATHEVFQQQLPLFLERCPHPVTLAGMLEMGVSYLPVNQNWERYLAEAQGTYEELQREMKKSLMDLANDACQLLSGERYKEDPWLWDLEWDLQEFKQKKAKKVKKEPATALGPCSEEEEFQQDVMARACLQKLKGTTELLPKRPQHLPGHPGWYRKLCPRLDDPAWTPGPSLLSLQMRVTPKLMALTWDGFPLHYSERHGWGYLNLAKLPTGTTLESAGVVCPYRAIESLYRKHCLEPYNDVDIPGCWFFKLPHKDGNSCNVGSPFAKDFLPKMEDGTLQAGPGGASGPRALEINKMISFWRNAHKRISSQMVVWLPRSALPRAVIRHPDYDEEGLYGAILPQVVTAGTITRRAVEPTWLTASNARPDRVGSELKAMVQAPPGYTLVGADVDSQELWIAAVLGDAHFAGMHGCTAFGWMTLQGRKSRGTDLHSKTATTVGISREHAKRFNYGRIYGAGQPFAERLLMQFNHRLTQQEAAEKAQQMYAATKGLLRKVQRETARKSQWKKWEVVAERAWKGGTESEMFNKLESIATSDIPRTPVLGCCISRALEPSAVQEEFMTSRVNWVVQSSAVDYLHLMLVAMKWLFEEFAIDGRFCISIHDEVRYLVREEDRYRAALALQITNLLTRCMFAYKLGLNDLPQSVAFFSAVDIDRCLRKEVTMDCKTPSNPTGMERRYGIPQGEALDIYQIIELTK 5c53 A 3.567 BS01 dna T 0 S305 S306 R309 K498 K561 S593 Q595 M596 R597 N803 K806 R807 T849 I850 P857 I948 G952 Y955 G958 F961 K1050 E1091 M1093 T1094 N1098 S216 S217 R220 K385 K429 S461 Q463 M464 R465 N590 K593 R594 T636 I637 P644 I735 G739 Y742 G745 F748 K805 E846 M848 T849 N853 2.7.7.7,3.1.11.-,4.2.99.- 0000262,0002020,0003677,0003682,0003887,0005515,0005739,0005759,0005760,0006259,0006260,0006261,0006264,0006281,0006284,0006287,0008310,0008408,0016787,0016829,0032991,0034061,0042645,0043231,0045004,0051575,0071897 remove_due_to_license_issue P54098 26124101 1 ~ 26 MLSRGLHEQIFGQGGEMPGEAAVRRSVEHLQKHGLWGQPAVPLPDVELRLPPLYGDNLDQHFRLLAQKQSLPYLEAANLLLQAQLPPKPPAWAWAEGWTRYGPEGEAVPVAIPEERALVFDVEVCLAEGTCPTLAVAISPSAWYSWCSQRLVEERYSWTSQLSPADLIPLEVQEQLVVGHNVSFDRAHIREQYLIQGSRMRFLDTMSMHMAISGLSSFQRSLWIAAKAISSWDWLDISSVNSLAEVHRLYVGGPPLEKEPRELFVKGTMKDIRENFQDLMQYCAQDVWATHEVFQQQLPLFLERCPHPVTLAGMLEMGVSYLPVNQNWERYLAEAQGTYEELQREMKKSLMDLANDACQLLSGERYKEDPWLWDLEWDLQEFKQKKAKKVKKEPATALGPCSEEEEFQQDVMARACLQKLKGTTELLPKRPQHLPGHPGWYRKLCPRLDDPAWTPGPSLLSLQMRVTPKLMALTWDGFPLHYSERHGWGYLNLAKLPTGTTLESAGVVCPYRAIESLYRKHCLEPYNDVDIPGCWFFKLPHKDGNSCNVGSPFAKDFLPKMEDGTLQAGPGGASGPRALEINKMISFWRNAHKRISSQMVVWLPRSALPRAVIRHPDYDEEGLYGAILPQVVTAGTITRRAVEPTWLTASNARPDRVGSELKAMVQAPPGYTLVGADVDSQELWIAAVLGDAHFAGMHGCTAFGWMTLQGRKSRGTDLHSKTATTVGISREHAKIFNYGRIYGAGQPFAERLLMQFNHRLTQQEAAEKAQQMYAATKGLLRKVQRETARKSQWKKWEVVAERAWKGGTESEMFNKLESIATSDIPRTPVLGCCISRALEPSAVQEEFMTSRVNWVVQSSAVDYLHLMLVAMKWLFEEFAIDGRFCISIHDEVRYLVREEDRYRAALALQITNLLTRCMFAYKLGLNDLPQSVAFFSAVDIDRCLRKEVTMDCKTPSNPTGMERRYGIPQGEALDIYQIIELTK 5c53 A 3.567 BS02 dna P 0 R579 S764 P765 D769 N803 L860 A862 R869 R447 S551 P552 D556 N590 L647 A649 R656 2.7.7.7,3.1.11.-,4.2.99.- 0000262,0002020,0003677,0003682,0003887,0005515,0005739,0005759,0005760,0006259,0006260,0006261,0006264,0006281,0006284,0006287,0008310,0008408,0016787,0016829,0032991,0034061,0042645,0043231,0045004,0051575,0071897 remove_due_to_license_issue P54098 26124101 3 ~ 23 MLSRGLHEQIFGQGGEMPGEAAVRRSVEHLQKHGLWGQPAVPLPDVELRLPPLYGDNLDQHFRLLAQKQSLPYLEAANLLLQAQLPPKPPAWAWAEGWTRYGPEGEAVPVAIPEERALVFDVEVCLAEGTCPTLAVAISPSAWYSWCSQRLVEERYSWTSQLSPADLIPLEVQEQLVVGHNVSFDRAHIREQYLIQGSRMRFLDTMSMHMAISGLSSFQRSLWIAAKAISSWDWLDISSVNSLAEVHRLYVGGPPLEKEPRELFVKGTMKDIRENFQDLMQYCAQDVWATHEVFQQQLPLFLERCPHPVTLAGMLEMGVSYLPVNQNWERYLAEAQGTYEELQREMKKSLMDLANDACQLLSGERYKEDPWLWDLEWDLQEFKQKKAKKVKKEPATALGPCSEEEEFQQDVMARACLQKLKGTTELLPKRPQHLPGHPGWYRKLCPRLDDPAWTPGPSLLSLQMRVTPKLMALTWDGFPLHYSERHGWGYLNLAKLPTGTTLESAGVVCPYRAIESLYRKHCLEPYNDVDIPGCWFFKLPHKDGNSCNVGSPFAKDFLPKMEDGTLQAGPGGASGPRALEINKMISFWRNAHKRISSQMVVWLPRSALPRAVIRHPDYDEEGLYGAILPQVVTAGTITRRAVEPTWLTASNARPDRVGSELKAMVQAPPGYTLVGADVDSQELWIAAVLGDAHFAGMHGCTAFGWMTLQGRKSRGTDLHSKTATTVGISREHAKIFNYGRIYGAGQPFAERLLMQFNHRLTQQEAAEKAQQMYAATKGLLRKVQRETARKSQWKKWEVVAERAWKGGTESEMFNKLESIATSDIPRTPVLGCCISRALEPSAVQEEFMTSRVNWVVQSSAVDYLHLMLVAMKWLFEEFAIDGRFCISIHDEVRYLVREEDRYRAALALQITNLLTRCMFAYKLGLNDLPQSVAFFSAVDIDRCLRKEVTMDCKTPSNPTGMERRYGIPQGEALDIYQIIELTK 5c5h A 2.401 BS02 4YB A 1 S188 L223 L244 G246 G247 A248 A249 Y269 G270 L271 T272 S276 T277 D336 I347 K437 S189 L224 L245 G247 G248 A249 A250 Y270 G271 L272 T273 S277 T278 D337 I348 K430 T142 S162 H186 G270 E273 F356 G361 T144 S163 H187 G271 E274 F357 G362 6.2.1.26 0005524,0008756,0009234,0016874,0016877,0032991,0042802 Kd=394nM remove_due_to_license_issue P37353 26394156 502 SHMIFSDWPWRHWRQVRGETIALRLNDEQLNWRELCARVDELASGFAVQGVVEGSGVMLRAWNTPQTLLAWLALLQCGARVLPVNPQLPQPLLEELLPNLTLQFALVPDGENTFPALTSLHIQLVEGAHAATWQPTRLCSMTLTSSTGLPKAAVHTYQAHLASAQGVLSLIPFGDHDDWLLSLPLFHVSGQGIMWKWLYAGARMTVRDKQPLEQMLAGCTHASLVPTQLWRLLVNRSSVSLKAVLLGGAAIPVELTEQAREQGIRCFCGYGLTEFASTVCAKEADGLADVGSPLPGREVKIVNNEVWLRAASMAEGYWRNGQLVSLVNDEGWYATRDRGEMHNGKLTIVGRLDNLFFSGGEGIQPEEVERVIAAHPAVLQVFIVPVADKFGHRPVAVMEYDHESVDLSEWVKDKLARFQQPVRWLTLPPKISRQALKEWVQRQ 5c5t A 1.598 BS01 AKG A 1 Y129 Y135 H138 M158 T172 H207 G209 K217 I219 Y83 Y89 H92 M112 T126 H161 G163 K171 I173 ? 0005506,0016705,0031418 Kd=681uM remove_due_to_license_issue Q84406 26368022 301 GVCDGKYYEKIDGFLSDIECDVLINAAIKKGLIPKSRNSEQTWFMPGEHEVIDKIQKKTREFLNSKKHCIDKYNFEDVQVARYKPGQYYYHHYDGDDCDDACPKDQRLATLMVYLKAPEEGGGGETDFPTLKTKIKPKKGTSIFFWVADPVTRKLYKETLHAGLPVKSGEKIIANQWIRAV 5c6o A 3.0 BS01 4YH A 1 M33 Y36 N37 F60 M63 M67 F150 F154 Q252 M31 Y34 N35 F58 M61 M65 F148 F152 Q250 ? 0005886,0015297,0016020,0042908,0042910,0046677,0055085 remove_due_to_license_issue Q9KAX3 26246409 501 QKQQSERLGTEAIPKLLRSLSIPAMIGMFVMALYNVVDTIFISYAVGIEGVAGVTIAFPIMMIMMSMAGALGIGGASVISRRLGERRGEEANQVFGNILTVILVLSVIGFISAFTLLGPALQLFGATSVTQGYATDYLFPILLGSIFFFFAFAANNIIRSEGNATFAMVTMIVPAVLNILLDVLFIFGLNMGVLGASIATVIAQASVTGLVLRYFLTGKSTLSLHWSDLRMKGSVIKEVCLVGLPAFVQQSSASLMMIAINSMLLRFGSDFYVGVFGLVQRIMMFVMMPMMGIMQAMQPIVGYNYGAKQYSRLRETVMLGFKVATIFSIGIFALLMLFPEALLRVFTADREVIQAGVSAMHILFCVTFLIGAQIVAGGLYQSLGKPKQALILSLSRQIIFLIPLVLILPHIFGLSGVWWAFPIADVLSFILTVVLLYRDRNVFFLK 5c6p A 3.0 BS01 4YH A 1 A57 S61 Q284 S288 D356 P357 A53 S57 Q280 S284 D352 P353 ? 0005886,0006811,0015297,0016020,0042908,0042910,0055085 remove_due_to_license_issue Q5F9J8 26246409 601 LDRFSFSVFLKEIRLLTALALPMLLAQVAQVGIGFVDTVMAGGAGKEDLAAVALGSSAFATVYITFMGIMAALNPMIAQLYGAGKTGEAGETGRQGIWFGLILGIFGMILMWAAITPFRNWLTLSDYVEGTMAQYMLFTSLAMPAAMVHRALHAYASSLNRPRLIMLVSFAAFVLNVPLNYIFVYGKFGMPALGGAGCGVATMAVFWFSALALWIYIAKEKFFRPFGLTAKFGKPDWAVFKQIWKIGAPIGLSYFLEASAFSFIVFLIAPFGEDYVAAQQVGISLSGILYMIPQSVGSAGTVRIGFSLGRREFSRARYISGVSLVSGWVLAVITVLSLVLFRSPLASMYNDDPAVLSIASTVLLFAGLFQPADFTQCIASYALRGYKVTKVPMFIHAAAFWGCGLLPGYLLAYRFDMGIYGFWTALIASLTIAAVALVWCLEKYSMELVKSHKAVSSGL 5c7a A 2.36 BS02 4YE A 1 G306 T308 D309 W310 E314 Q319 W323 Y324 G58 T60 D61 W62 E66 Q71 W75 Y76 2.3.2.27 remove_due_to_license_issue P98170 26218264 402 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c7b A 2.68 BS02 4YD A 1 G306 L307 T308 D309 W310 E314 Q319 W323 G58 L59 T60 D61 W62 E66 Q71 W75 2.3.2.27 remove_due_to_license_issue P98170 26218264 402 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c7c A 2.32 BS02 4YC A 1 K297 G306 T308 D309 W310 E314 Q319 W323 K50 G59 T61 D62 W63 E67 Q72 W76 2.3.2.27 ic50=5.5uM remove_due_to_license_issue P98170 26218264 402 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c7d A 2.25 BS02 4YF A 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 Y324 K49 G58 L59 T60 D61 W62 E66 Q71 W75 Y76 2.3.2.27 ic50=7.7uM remove_due_to_license_issue P98170 26218264 402 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c7n A 1.75 BS01 BMF A 1 V657 P658 V662 Y707 N708 F714 V30 P31 V35 Y80 N81 F87 ? Kd=0.27uM remove_due_to_license_issue IC50=141nM P55201 27167503 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5c83 A 2.33 BS02 4YN A 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 K50 G59 L60 T61 D62 W63 E67 Q72 W76 2.3.2.27 ic50=0.16uM remove_due_to_license_issue P98170 26218264 402 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c84 A 2.36 BS02 4YL A 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 K50 G59 L60 T61 D62 W63 E67 Q72 W76 2.3.2.27 ic50=0.64uM remove_due_to_license_issue P98170 26218264 402 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5c85 A 1.7 BS01 4YO A 1 I652 V657 P658 F714 I25 V30 P31 F87 ? Kd=105uM remove_due_to_license_issue Kd=105000nM P55201 27167503 802 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5c87 A 1.55 BS01 4YS A 1 F653 V657 Y665 C704 Y707 N708 F714 F26 V30 Y38 C77 Y80 N81 F87 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 802 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5c8k A 3.0 BS01 4YV A 1 L718 G719 V726 A743 K745 M766 C775 M790 Q791 L792 M793 L844 T854 D855 L22 G23 V30 A47 K49 M68 C77 M92 Q93 L94 M95 L146 T156 D157 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26455919 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLI 5c8m A 2.9 BS01 4YW A 1 L718 F723 A743 K745 C775 M790 Q791 M793 L844 T854 L22 F27 A47 K49 C77 M92 Q93 M95 L146 T156 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26455919 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLIP 5c8n A 2.401 BS01 4YX A 1 L718 F723 A743 K745 M766 C775 M790 Q791 M793 L844 T854 D855 L23 F28 A48 K50 M68 C77 M92 Q93 M95 L146 T156 D157 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 Ki=28nM remove_due_to_license_issue P00533 26455919 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYDMDDVVDADEYLIP 5c91 A 2.44 BS01 4YU A 1 Y605 L607 C627 N628 Y87 L89 C109 N110 R549 E580 E591 D653 H865 C867 R31 E62 E73 D135 H347 C349 2.3.2.26 0004842 remove_due_to_license_issue P46934 26371805 901 SRDYKRKYEFFRRKLKKQNDIPNKFEMKLRRATVLEDSYRRIMGVKRADFLKARLWIEFDGEKGLDYGGVAREWFFLISKEMFNPYYGLFEYSATDNYTLQINPNSGLCNEDHLSYFKFIGRVAGMAVYHGKLLDGFFIRPFYKMMLHKPITLHDMESVDSEYYNSLRWILENDPTELDLRFIIDEELFGQTHQHELKNGGSEIVVTNKNKKEYIYLVIQWRFVNRIQKQMAAFKEGFFELIPQDLIKIFDENELELLMCGLGDVDVNDWREHTKYKNGYSANHQVIQWFWKAVLMMDSEKRIRLLQFVTGTSRVPMNGFAELYGSNGPQSFTVEQWGTPEKLPRAHTCFNRLDLPPYESFEELWDKLQMAIENT 5cal A 2.7 BS01 4Z8 A 1 L718 F723 A743 M790 Q791 M793 N842 L844 T854 D855 L22 F27 A47 M92 Q93 M95 N144 L146 T156 D157 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=390nM P00533 26455919 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLI 5can A 2.8 BS01 4ZB A 1 L718 A743 C775 M790 Q791 L792 M793 L844 T854 D855 L23 A48 C78 M93 Q94 L95 M96 L147 T157 D158 D837 A839 R841 N842 D855 D140 A142 R144 N145 D158 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=681nM P00533 26455919 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYDMDDVVDADEYLIP 5cao A 2.6 BS01 4ZG A 1 L718 F723 A743 K745 C775 M790 Q791 M793 L844 T854 D855 L22 F27 A47 K49 C76 M91 Q92 M94 L145 T155 D156 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=1820nM P00533 26455919 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYREEDMDDVVDADEYLIP 5cap A 2.4 BS01 4ZH A 1 L718 A743 K745 C775 M790 Q791 M793 L844 T854 D855 L22 A47 K49 C79 M94 Q95 M97 L148 T158 D159 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 Ki=52nM remove_due_to_license_issue Ki=2100nM P00533 26455919 1103 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRADMDDVVDADEYLIP 5caq A 2.5 BS01 4ZJ A 1 L718 A743 K745 M766 C775 M790 Q791 M793 L844 T854 L22 A47 K49 M68 C77 M92 Q93 M95 L146 T156 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 Ki=2.7nM remove_due_to_license_issue IC50=>10000nM, Ki=1080nM P00533 26455919 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLI 5cas A 2.1 BS01 4ZQ A 1 L718 G719 V726 A743 K745 E762 M766 C775 M790 Q791 M793 L844 T854 L23 G24 V31 A48 K50 E63 M67 C76 M91 Q92 M94 L145 T155 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 Ki=1.4nM remove_due_to_license_issue P00533 26455919 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYMDDVVDADEYLIP 5cau A 2.25 BS01 4ZR A 1 L718 G719 V726 A743 K745 M766 C775 M790 Q791 M793 L844 T854 L23 G24 V31 A48 K50 M67 C76 M91 Q92 M94 L145 T155 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 Ki=1.6nM remove_due_to_license_issue P00533 26455919 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYMDDVVDADEYLI 5cav A 2.73 BS01 4ZQ A 1 L718 V726 A743 K745 C775 T790 Q791 L792 M793 G796 L844 T854 D855 L22 V30 A47 K49 C79 T94 Q95 L96 M97 G100 L148 T158 D159 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26455919 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDEEDMDDVVDADEYLIPQ 5cbm A 2.3 BS04 4ZN A 1 K374 D379 K386 M396 F398 D399 D459 E461 T486 T488 G489 A577 K290 D295 K302 M312 F314 D315 D375 E377 T402 T404 G405 A493 K386 R463 K302 R379 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 remove_due_to_license_issue A0A024V0B1 26406322 704 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 5cbr A 1.996 BS01 4ZK A 1 Y58 P86 T88 R93 L135 S139 T140 T171 Y187 L189 E190 M193 Y217 Y58 P86 T88 R93 L135 S139 T140 T171 Y187 L189 E190 M193 Y217 ? 0015276,0016020 Kd=1.8uM remove_due_to_license_issue Ki=1740nM, IC50=3700nM P19491 26653877 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 5cbs A 1.801 BS01 E42 A 1 Y58 L87 T88 R93 I108 S139 E190 D213 K215 Y58 L87 T88 R93 I108 S139 E190 D213 K215 ? 0015276,0016020 Kd=3.9uM remove_due_to_license_issue Ki=24000nM, IC50=6300nM P19491 26653877 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECGS 5cbs C 1.801 BS01 E42 C 1 Y58 L87 T88 R93 L106 I108 S139 E190 D213 K215 Y60 L89 T90 R95 L108 I110 S141 E192 D215 K217 ? 0015276,0016020 Kd=3.9uM remove_due_to_license_issue Ki=24000nM, IC50=6300nM P19491 26653877 301 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 5cbx A 2.0 BS01 dna C 0 C431 H432 Y433 K446 C13 H14 Y15 K28 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 KICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEA 5cbx A 2.0 BS02 dna D 0 S440 R447 R470 K471 R477 S22 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 KICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEA 5cbx B 2.0 BS01 dna C 0 S440 R447 R470 K471 R477 S24 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEA 5cbx B 2.0 BS02 dna D 0 C431 H432 Y433 K446 C15 H16 Y17 K30 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEA 5cbx E 2.0 BS01 dna G 0 C431 H432 Y433 K446 C15 H16 Y17 K30 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLE 5cbx E 2.0 BS02 dna H 0 S440 R447 R470 K471 R477 S24 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLE 5cbx F 2.0 BS01 dna G 0 S440 R447 R470 K471 R477 S24 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEA 5cbx F 2.0 BS02 dna H 0 C431 H432 Y433 K442 K446 C15 H16 Y17 K26 K30 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEA 5cby A 1.997 BS01 dna C 0 C431 H432 Y433 K442 K446 C15 H16 Y17 K26 K30 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEARK 5cby A 1.997 BS02 dna D 0 S440 F444 R447 R470 K471 R477 S24 F28 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKICLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLEARK 5cby B 1.997 BS01 dna C 0 S440 R447 R470 K471 R477 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PKICLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLE 5cby B 1.997 BS02 dna D 0 C431 H432 Y433 K446 C14 H15 Y16 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PKICLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRFRKCLQAGMNLE 5cbz A 2.2 BS01 dna C 0 C431 H432 Y433 K442 K446 C14 H15 Y16 K25 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 SKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLGA 5cbz A 2.2 BS02 dna D 0 G439 S440 R447 Y455 R470 K471 R477 G22 S23 R30 Y38 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 SKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLGA 5cbz B 2.2 BS01 dna C 0 G439 S440 R447 R470 K471 R477 G22 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 SKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLGAR 5cbz B 2.2 BS02 dna D 0 C431 H432 Y433 K442 C14 H15 Y16 K25 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 SKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLGAR 5cbz E 2.2 BS01 dna G 0 C431 H432 Y433 K442 K446 C16 H17 Y18 K27 K31 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPSKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLGAR 5cbz E 2.2 BS02 dna H 0 S440 R447 Y455 R470 K471 R477 S25 R32 Y40 R55 K56 R62 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPSKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLGAR 5cbz F 2.2 BS01 dna G 0 S440 R447 R470 K471 R477 S24 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PSKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLG 5cbz F 2.2 BS02 dna H 0 C431 H432 Y433 K442 C15 H16 Y17 K26 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PSKVCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMNLG 5cc0 A 2.405 BS01 dna C 0 C431 H432 Y433 K442 K446 C14 H15 Y16 K25 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 26715749 1 ~ 16 QKVCLICGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMTLGA 5cc0 A 2.405 BS02 dna D 0 G439 S440 F444 R447 R470 K471 R477 G22 S23 F27 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 26715749 1 ~ 16 QKVCLICGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMTLGA 5cc0 B 2.405 BS01 dna C 0 S440 R447 R470 K471 R477 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 26715749 1 ~ 16 QKVCLICGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMTLG 5cc0 B 2.405 BS02 dna D 0 G430 C431 H432 Y433 K446 G13 C14 H15 Y16 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P06401 26715749 1 ~ 16 QKVCLICGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRLRKCLQAGMTLG 5cc1 A 2.302 BS01 dna C 0 C431 H432 Y433 K442 K446 C15 H16 Y17 K26 K30 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 5cc1 A 2.302 BS02 dna D 0 S440 R447 R470 K471 R477 S24 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 5cc1 B 2.302 BS01 dna C 0 S440 R447 R470 R477 S23 R30 R53 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5cc1 B 2.302 BS02 dna D 0 C431 H432 Y433 K446 C14 H15 Y16 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5cc1 W 2.302 BS01 dna Y 0 S440 F444 R447 R470 K471 R477 S24 F28 R31 R54 K55 R61 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 5cc1 W 2.302 BS02 dna Z 0 C431 H432 Y433 K442 K446 C15 H16 Y17 K26 K30 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PPKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEAR 5cc1 X 2.302 BS01 dna Y 0 C431 H432 Y433 K446 C14 H15 Y16 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5cc1 X 2.302 BS02 dna Z 0 S440 R447 R470 R477 S23 R30 R53 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 26715749 1 ~ 18 PKLCLVCGDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5cc2 A 2.501 BS01 CKA A 1 E12 F15 Y58 A85 L86 T87 R92 A138 W193 D194 Y222 E10 F13 Y56 A83 L84 T85 R90 A136 W191 D192 Y220 ? 0015276,0016020 Kd=80uM remove_due_to_license_issue Q63226 26661043 301 VVLRVVTVLEEPFVMVSENVLGKPKKYQGFSIDVLDALSNYLGFNYEIYVAPDHKYGSPQEDGTWNGLVGELVFKRADIGISALTITPDRENVVDFTTRYMDYSVGVLLRRGTSIQSLQDLSKQTDIPYGTVLDSAVYQHVRMKGLNPFERDSMYSQMWRMINRSNGSENNVLESQAGIQKVKYGNYAFVWDAAVLEYVAINDPDCSFYTVGNTVADRGYGIALQHGSPYRDVFSQRILELQQSGDMDILKHKWWP 5cc2 A 2.501 BS02 CKA A 2 V107 H142 V143 Y157 M160 V217 V105 H140 V141 Y155 M158 V215 ? 0015276,0016020 Kd=80uM remove_due_to_license_issue Q63226 26661043 302 VVLRVVTVLEEPFVMVSENVLGKPKKYQGFSIDVLDALSNYLGFNYEIYVAPDHKYGSPQEDGTWNGLVGELVFKRADIGISALTITPDRENVVDFTTRYMDYSVGVLLRRGTSIQSLQDLSKQTDIPYGTVLDSAVYQHVRMKGLNPFERDSMYSQMWRMINRSNGSENNVLESQAGIQKVKYGNYAFVWDAAVLEYVAINDPDCSFYTVGNTVADRGYGIALQHGSPYRDVFSQRILELQQSGDMDILKHKWWP 5cc2 A 2.501 BS03 CKA A 3 V174 A179 Q182 K183 V172 A177 Q180 K181 ? 0015276,0016020 Kd=80uM remove_due_to_license_issue Q63226 26661043 303 VVLRVVTVLEEPFVMVSENVLGKPKKYQGFSIDVLDALSNYLGFNYEIYVAPDHKYGSPQEDGTWNGLVGELVFKRADIGISALTITPDRENVVDFTTRYMDYSVGVLLRRGTSIQSLQDLSKQTDIPYGTVLDSAVYQHVRMKGLNPFERDSMYSQMWRMINRSNGSENNVLESQAGIQKVKYGNYAFVWDAAVLEYVAINDPDCSFYTVGNTVADRGYGIALQHGSPYRDVFSQRILELQQSGDMDILKHKWWP 5ccl A 1.5 BS05 4ZW A 1 N181 S182 F183 T184 E192 S202 Y239 Y257 N179 S180 F181 T182 E190 S200 Y237 Y255 2.1.1.354 0000978,0000993,0001162,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0008168,0014904,0032259,0042054,0045184,0045944,0046872,0071549,0140939,0140954,0140999 remove_due_to_license_issue IC50=>10000nM Q9H7B4 26985287 505 PLKVEKFATANRGNGLRAVTPLRPGELLFRSDPLAYTVCKGSRGVVCDRCLLGKEKLMRCSQCRVAKYCSAKCQKKAWPDHKRECKCLKSCKPRYPPDSVRLLGRVVFKLMDGAPSESEKLYSFYDLESNINKLTEDKKEGLRQLVMTFQHFMREEIQDASQLPPAFDLFEAFAKVICNSFTICNAEMQEVGVGLYPSISLLNHSCDPNCSIVFNGPHLLLRAVRDIEVGEELTICYLDMLMTSEERRKQLRDQYCFECDCFRCQTQDKDADMLTGDEQVWKEVQESLKKIEELKAHWKWEQVLAMCQAIISSNSERLPDINIYQLKVLDCAMDACINLGLLEEALFYGTRTMEPYRIFFPGSHPVRGVQVMKVGKLQLHQGMFPQAMKNLRLAFDIMRVTHGREHSLIEDLILLLEECDANIRA 5ccl A 1.5 BS06 4ZW A 2 R19 V21 V231 G232 R17 V19 V229 G230 2.1.1.354 0000978,0000993,0001162,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0008168,0014904,0032259,0042054,0045184,0045944,0046872,0071549,0140939,0140954,0140999 remove_due_to_license_issue IC50=>10000nM Q9H7B4 26985287 506 PLKVEKFATANRGNGLRAVTPLRPGELLFRSDPLAYTVCKGSRGVVCDRCLLGKEKLMRCSQCRVAKYCSAKCQKKAWPDHKRECKCLKSCKPRYPPDSVRLLGRVVFKLMDGAPSESEKLYSFYDLESNINKLTEDKKEGLRQLVMTFQHFMREEIQDASQLPPAFDLFEAFAKVICNSFTICNAEMQEVGVGLYPSISLLNHSCDPNCSIVFNGPHLLLRAVRDIEVGEELTICYLDMLMTSEERRKQLRDQYCFECDCFRCQTQDKDADMLTGDEQVWKEVQESLKKIEELKAHWKWEQVLAMCQAIISSNSERLPDINIYQLKVLDCAMDACINLGLLEEALFYGTRTMEPYRIFFPGSHPVRGVQVMKVGKLQLHQGMFPQAMKNLRLAFDIMRVTHGREHSLIEDLILLLEECDANIRA 5ccm A 2.3 BS05 4ZX A 1 N181 S182 F183 T184 C186 M190 E192 S202 C238 Y239 L240 D241 Y257 K329 D332 V368 N179 S180 F181 T182 C184 M188 E190 S200 C236 Y237 L238 D239 Y255 K327 D330 V366 2.1.1.354 0000978,0000993,0001162,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0008168,0014904,0032259,0042054,0045184,0045944,0046872,0071549,0140939,0140954,0140999 ic50=4nM remove_due_to_license_issue Ki=4.7nM, IC50=4.0nM Q9H7B4 26985287 505 PLKVEKFATANRGNGLRAVTPLRPGELLFRSDPLAYTVCKGSRGVVCDRCLLGKEKLMRCSQCRVAKYCSAKCQKKAWPDHKRECKCLKSCKPRYPPDSVRLLGRVVFKLMDGAPSESEKLYSFYDLESNINKLTEDKKEGLRQLVMTFQHFMREEIQDASQLPPAFDLFEAFAKVICNSFTICNAEMQEVGVGLYPSISLLNHSCDPNCSIVFNGPHLLLRAVRDIEVGEELTICYLDMLMTSEERRKQLRDQYCFECDCFRCQTQDKDADMLTGDEQVWKEVQESLKKIEELKAHWKWEQVLAMCQAIISSNSERLPDINIYQLKVLDCAMDACINLGLLEEALFYGTRTMEPYRIFFPGSHPVRGVQVMKVGKLQLHQGMFPQAMKNLRLAFDIMRVTHGREHSLIEDLILLLEECDANI 5ceh A 3.14 BS03 50P A 1 Y409 A411 Y472 F480 H483 K501 H571 N575 Y221 A223 Y284 F292 H295 K313 H383 N387 G465 Y472 H483 E485 H571 A583 G277 Y284 H295 E297 H383 A395 1.14.11.67 0003677 remove_due_to_license_issue IC50=10.0nM, EC50=5200nM P29375 27214401 904 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRVRLDFLDQLAKFWELQGSTLKIPVVERKILDLYALSKIVASKGGFEMVTKEKKWSKVGSRLGYLPGKGTGSLLKSHYERILYPYELFQSGVSLMGVQMYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINVDISGMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCTADWLPIGRQCVNHYRRLRRHCVFSHEELIFKMAADPECLDVGLAAMVCKELTLMTEEETRLRESVVQMGVLMSEEEVFELVPDDERQCSACRTTCFLSALTCSCNPERLVCLYHPTDLCPCPMQKKCLRYRYPLEDLPSLLYGVKVRAQSYDTWVSVMLEDAEDRKYPENDLFRKLR 5cei A 2.24 BS01 50R A 1 V27 Y32 V35 A50 K52 I79 Y99 A100 D103 A155 L158 D173 R356 V28 Y33 V36 A51 K53 I80 Y100 A101 D104 A151 L154 D169 R339 D151 K153 N156 D173 N181 T196 D147 K149 N152 D169 N177 T183 2.7.11.22,2.7.11.23 0004672,0005524,0006468 ic50=5.3nM remove_due_to_license_issue P49336 26985305 508 KMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKAQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLKPTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQESNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEE 5ceo A 2.28 BS01 50D A 1 G132 G134 V139 A150 F192 C193 G196 L243 G16 G18 V23 A34 F76 C77 G80 L127 D236 K238 P240 N241 D254 T273 D120 K122 P124 N125 D138 T144 2.7.11.25 0004672,0005524,0006468 Ki<0.0005uM remove_due_to_license_issue Ki=<0.500000nM, IC50=30nM Q12852 26431428 501 LWEVPFEEILDLQWVGSGAQGAVFLGRFHGEEVAVKKVRDLKETDIKHLRKLKHPNIITFKGVCTQAPCYCILMEFCAQGQLYEVLRAGRPVTPSLLVDWSMGIAGGMNYLHLHKIIHRDLKSPNMLITYDDVVKISDFGFAGTVAWMAPEVIRNEPVSEKVDIWSFGVVLWELLTGEIPYKDVDSSAIIWGVGSNSLHLPVPSSCPDGFKILLRQCWNSKPRNRPSFRQILLHLDIASADVLSTPQETYFKSQAEWREEVKLHFEKIK 5cep A 1.99 BS01 50E A 1 G132 Q136 V139 A150 M190 F192 C193 G196 Q197 L243 G16 Q20 V23 A34 M74 F76 C77 G80 Q81 L127 D236 K238 P240 N241 D254 T273 D120 K122 P124 N125 D138 T144 2.7.11.25 0004672,0005524,0006468 Ki=0.145uM remove_due_to_license_issue Ki=145nM Q12852 26431428 501 LWEVPFEEILDLQWVGSGAQGAVFLGRFHGEEVAVKKVRDLKETDIKHLRKLKHPNIITFKGVCTQAPCYCILMEFCAQGQLYEVLRAGRPVTPSLLVDWSMGIAGGMNYLHLHKIIHRDLKSPNMLITYDDVVKISDFGFAGTVAWMAPEVIRNEPVSEKVDIWSFGVVLWELLTGEIPYKDVDSSAIIWGVGSNSLHLPVPSSCPDGFKILLRQCWNSKPRNRPSFRQILLHLDIASADVLSTPQETYFKSQAEWREEVKLHFEKIK 5ceq A 1.911 BS01 50F A 1 G132 G134 V139 A150 M190 F192 C193 G196 Q197 L243 G16 G18 V23 A34 M74 F76 C77 G80 Q81 L127 D236 K238 P240 N241 D254 T273 D120 K122 P124 N125 D138 T144 2.7.11.25 0004672,0005524,0006468 Ki=0.042uM remove_due_to_license_issue Ki=42nM, IC50=536nM Q12852 26431428 4000 LWEVPFEEILDLQWVGSGAQGAVFLGRFHGEEVAVKKVRDLKETDIKHLRKLKHPNIITFKGVCTQAPCYCILMEFCAQGQLYEVLRAGRPVTPSLLVDWSMGIAGGMNYLHLHKIIHRDLKSPNMLITYDDVVKISDFGFAGTVAWMAPEVIRNEPVSEKVDIWSFGVVLWELLTGEIPYKDVDSSAIIWGVGSNSLHLPVPSSCPDGFKILLRQCWNSKPRNRPSFRQILLHLDIASADVLSTPQETYFKSQAEWREEVKLHFEKIK 5cf4 A 2.38 BS01 50Y A 1 L855 G856 G858 V863 A880 M929 Y931 L932 P933 G935 S936 L983 G993 D994 L13 G14 G16 V21 A38 M83 Y85 L86 P87 G89 S90 L137 G147 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=40nM remove_due_to_license_issue IC50=1300nM O60674 26288682 4000 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 5cf5 A 2.45 BS01 50W A 1 L855 G856 V863 A880 M929 Y931 L932 G935 R980 N981 L983 D994 L14 G15 V22 A39 M85 Y87 L88 G91 R136 N137 L139 D150 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=2.5nM remove_due_to_license_issue IC50=2.5nM O60674 26288682 4000 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAGH 5cf6 A 2.5 BS01 50O A 1 L855 G856 V863 A880 M929 Y931 L932 G935 S936 D939 N981 L983 G993 D994 L14 G15 V22 A39 M85 Y87 L88 G91 S92 D95 N137 L139 G149 D150 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=8.2nM remove_due_to_license_issue IC50=8.2nM O60674 26288682 4000 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 5cf8 A 1.8 BS01 50V A 1 L855 G856 V863 A880 M929 Y931 L932 G935 R980 N981 L983 D994 L14 G15 V22 A39 M83 Y85 L86 G89 R134 N135 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1.1nM remove_due_to_license_issue IC50=80nM, Kd=0.480000nM O60674 26288683 4000 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAGH 5cfb A 3.04 BS01 SY9 A 1 F159 Y202 F207 F151 Y194 F199 ? 0004888,0005216,0005230,0005886,0006811,0016020,0016594,0022824,0034220 remove_due_to_license_issue O75311 26416729 501 SPSDFLDKLMGRTSGYDARIRPNFKGPPVNVTCNIFINSFGSIAETTMDYRVNIFLRQKWNDPRLAYSEYPDDSLDLDPSMLDSIWKPDLFFANEKGANFHEVTTDNKLLRIFKNGNVLYSIRLTLTLSCPMDLKNFPMDVQTCIMQLESFGYTMNDLIFEWQDEAPVQVAEGLTLPQFLLKEEKDLRYCTKHYNTGKFTCIEVRFHLERQMGYYLIQMYIPSLLIVILSWVSFWINMDAAPARVALGITTVLTMTTQSSGSRASLPKVSYVKAIDIWMAVCLLFVFSALLEYAAVNFVSRAGTKVFIDRAKKIDTISRACFPLAFLIFNIFYWVIYKI 5cfb A 3.04 BS02 SY9 E 1 F44 F63 R65 L117 L127 F36 F55 R57 L109 L119 ? 0004888,0005216,0005230,0005886,0006811,0016020,0016594,0022824,0034220 remove_due_to_license_issue O75311 26416729 501 SPSDFLDKLMGRTSGYDARIRPNFKGPPVNVTCNIFINSFGSIAETTMDYRVNIFLRQKWNDPRLAYSEYPDDSLDLDPSMLDSIWKPDLFFANEKGANFHEVTTDNKLLRIFKNGNVLYSIRLTLTLSCPMDLKNFPMDVQTCIMQLESFGYTMNDLIFEWQDEAPVQVAEGLTLPQFLLKEEKDLRYCTKHYNTGKFTCIEVRFHLERQMGYYLIQMYIPSLLIVILSWVSFWINMDAAPARVALGITTVLTMTTQSSGSRASLPKVSYVKAIDIWMAVCLLFVFSALLEYAAVNFVSRAGTKVFIDRAKKIDTISRACFPLAFLIFNIFYWVIYKI 5cfb B 3.04 BS01 SY9 A 1 F63 L117 F55 L109 ? 0004888,0005216,0005230,0005886,0006811,0016020,0016594,0022824,0034220 remove_due_to_license_issue O75311 26416729 501 SPSDFLDKLMGRTSGYDARIRPNFKGPPVNVTCNIFINSFGSIAETTMDYRVNIFLRQKWNDPRLAYSEYPDDSLDLDPSMLDSIWKPDLFFANEKGANFHEVTTDNKLLRIFKNGNVLYSIRLTLTLSCPMDLKNFPMDVQTCIMQLESFGYTMNDLIFEWQDEAPVQVAEGLTLPQFLLKEEKDLRYCTKHYNTGKFTCIEVRFHLERQMGYYLIQMYIPSLLIVILSWVSFWINMDAAPARVALGITTVLTMTTQSSGSRASLPKVSYVKAIDIWMAVCLLFVFSALLEYAAVNFVSRAGTKVFIDRAKKIDTISRACFPLAFLIFNIFYWVIYKI 5cfb B 3.04 BS02 SY9 B 1 F159 Y202 F207 F151 Y194 F199 ? 0004888,0005216,0005230,0005886,0006811,0016020,0016594,0022824,0034220 remove_due_to_license_issue O75311 26416729 501 SPSDFLDKLMGRTSGYDARIRPNFKGPPVNVTCNIFINSFGSIAETTMDYRVNIFLRQKWNDPRLAYSEYPDDSLDLDPSMLDSIWKPDLFFANEKGANFHEVTTDNKLLRIFKNGNVLYSIRLTLTLSCPMDLKNFPMDVQTCIMQLESFGYTMNDLIFEWQDEAPVQVAEGLTLPQFLLKEEKDLRYCTKHYNTGKFTCIEVRFHLERQMGYYLIQMYIPSLLIVILSWVSFWINMDAAPARVALGITTVLTMTTQSSGSRASLPKVSYVKAIDIWMAVCLLFVFSALLEYAAVNFVSRAGTKVFIDRAKKIDTISRACFPLAFLIFNIFYWVIYKI 5cgc A 3.101 BS01 51D A 1 I625 I651 P655 L744 W785 F788 V806 S809 A810 I58 I84 P88 L321 W362 F365 V383 S386 A387 E1011 D1020 E121 D130 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P41594 26225459 4006 SPVQYLRWGDPAPIAAVVFACLGLLATLFVTVVFIIYRDTPVVKSSSRELCYIILAGICLGYLCTFCLIAKPKQIYCYLQRIGIGLSPAMSYSALVTKTYRAARILAMSKKNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKISACAQLVIAFILICIQLGIIVALFIMEPPDIMVYLICNTTNLGVVAPLGYNGLLILACTFYAFKTRNVPANFNEAKYIAFTMYTTCIIWLAFVPIYFGSNYKIITMCFSVSLSATVALGCMFVPKVYIILAKPERN 5cgd A 2.603 BS01 51E A 1 G624 I625 I651 S654 P655 S658 Y659 L744 W785 F788 V806 S809 G57 I58 I84 S87 P88 S91 Y92 L321 W362 F365 V383 S386 E1011 D1020 E121 D130 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P41594 26225459 4005 SPVQYLRWGDPAPIAAVVFACLGLLATLFVTVVFIIYRDTPVVKSSSRELCYIILAGICLGYLCTFCLIAKPKQIYCYLQRIGIGLSPAMSYSALVTKTYRAARILAMSKKNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKISACAQLVIAFILICIQLGIIVALFIMEPPDIMVYLICNTTNLGVVAPLGYNGLLILACTFYAFKTRNVPANFNEAKYIAFTMYTTCIIWLAFVPIYFGSNYKIITMCFSVSLSATVALGCMFVPKVYIILAKPER 5cgj A 3.36 BS01 51M A 1 Y334 S363 G364 R415 R483 Y525 A556 S602 G603 Y11 S40 G41 R92 R160 Y202 A233 S279 G280 ? remove_due_to_license_issue Kd=6000nM Q9Z2X8 26459563 705 VGRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 5cgv A 2.17 BS03 0N8 A 1 Y24 I38 H41 E80 D108 E119 K134 K137 Y24 I38 H41 E61 D89 E100 K115 K118 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 26976575 303 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERA 5chk A 2.2 BS01 55R A 1 S16 Y33 T35 W70 S73 T77 W97 N118 S14 Y31 T33 W68 S71 T75 W95 N116 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 202 KCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYTTAVTATSNEIKESPLHGTENTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 5ci7 A 1.74 BS01 51W A 1 I22 A44 M92 Y94 C95 G98 L145 I20 A42 M90 Y92 C93 G96 L143 D138 K140 Q142 N143 D165 S184 D136 K138 Q140 N141 D163 S182 2.7.11.1 0004672,0004674,0005524,0006468,0010506 ic50=120nM remove_due_to_license_issue IC50=120nM O75385 26275681 401 PGRGGTETVGKFEFSRKDLIGHGAFAVVFKGRHRAAHDLEVAVKCINKKNLAKSQTLLGKEIKILKELKHENIVALYDFQEMANSVYLVMEYCNGGDLADYLHAMRTLSEDTIRLFLQQIAGAMRLLHSKGIIHRDLKPQNILLSNPAGRRANPNSIRVKIADFGFARYLQSNMMAATLCGSPMYMAPEVIMSQHYDGKADLWSIGTIVYQCLTGKAPFQASSPQDLRLFYEKNKTLVPTIPRETSAPLRQLLLALLQRNHKDRMDFDEFFHHPFLD 5cj6 A 2.07 BS02 51Y A 1 L704 N705 L707 Q711 M745 M749 F764 T877 M895 L34 N35 L37 Q41 M75 M79 F94 T203 M221 ? Ki=2.03nM remove_due_to_license_issue Ki=2.0nM, EC50=0.499000nM P10275 26683992 1001 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT 5cjf A 1.83 BS02 520 A 1 H94 H119 S132 L198 T199 T200 H89 H115 S128 L196 T197 T198 H64 H94 H96 E106 H119 T199 H64 H89 H91 E102 H115 T197 4.2.1.1 0004089,0008270 Ki=0.26nM remove_due_to_license_issue Ki=0.260000nM Q9ULX7 26497049 302 HWTYEGPHGQDHWPASYPECGNNAQSPIDIQTDSVTFDPDLPALQPHGYDQPGTEPLDLHNNGHTVQLSLPSTLYLGGLPRKYVAAQLHLHWGQKGSPGGSEHQINSEATFAELHIVHYDSDSYDSLSEAAERPQGLAVLGILIEVGETKNIAYEHILSHLHEVRHKDQKTSVPPFNLRELLPKQLGQYFRYNGSLTTPPCYQSVLWTVFYRRSQISMEQLEKLQGTLFSTEEEPSKLLVQNYRALQPLNQRMVFASFIQAGSSYTT 5ckr A 2.95 BS01 57M A 1 T75 N190 D193 G194 L195 D196 F262 M263 G264 S268 V302 Q305 R320 A321 P322 H325 T45 N160 D163 G164 L165 D166 F232 M233 G234 S238 V272 Q275 R290 A291 P292 H295 2.7.8.13 0005886,0008360,0008963,0009252,0016020,0016740,0016780,0042802,0044038,0046872,0051301,0051992,0071555 remove_due_to_license_issue O66465 27088606 401 KYITFRSFTAVLIAFFLTLVLSPSFINRLRKIQRLFGGVKKYTPTMGGIVILIVVTLSTLLLMRWDIKYTWVVLLSFLSFGTIGFWDDYVKLKNKKGISIKTKFLLQVLSASLISVLIYYWADIDTILYFPFFKELYVDLGVLYLPFAVFVIVGSANAVNLTDGLDGLAIGPAMTTATALGVVAYAVGHSKIAQYLNIPYVPYAGELTVFCFALVGAGLGFLWFNSFPAQMFMGDVGSLSIGASLATVALLTKSEFIFAVAAGVFVFETISVILQIIYFRWTGGKRLFKRAPFHHHLELNGLPEPKIVVRMWIISILLAIIAISMLKLR 5cks B 2.1181 BS03 52L B 1 R92 Y94 K97 P98 R99 T100 K186 H268 D326 R87 Y89 K92 P93 R94 T95 K181 H263 D321 2.5.1.54 0003849,0005737,0005829,0008652,0009058,0009073,0009423,0016740,0042802 Kd=3.1uM remove_due_to_license_issue P0AB91 27933795 402 DDLRIKEIKELLPPVALLEKFPATENAANTVAHARKAIHKILKGNDDRLLVVIGPCSIHDPVAAKEYATRLLALREELKDELEIVMRVYFEKPRTTVGWKGLINDPHMDNSFQINDGLRIARKLLLDINDSGLPAAGEFLDMITPQYLADLMSWGAIGARTTESQVHRELASGLSCPVGFKNGTDGTIKVAIDAINAAGAPHCFLSVTKWGHSAIVNTSGNGDCHIILRGGKEPNYSAKHVAEVKEGLNKAGLPAQVMIDFSHANSSKQFKKQMDVCADVCQQIAGGEKAIIGVMVESHLVEGNQSLESGEPLAYGKSITDACIGWEDTDALLRQLANAVKARRG 5clm A 2.61 BS01 52K A 1 G11 Q12 G13 L30 D32 Y71 F108 I118 D228 G230 T232 G13 Q14 G15 L32 D34 Y73 F110 I120 D222 G224 T226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D222 T225 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=240nM P56817 26378740 401 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVADDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5cls A 1.75 BS02 52T A 1 F219 H231 L328 N329 H331 I338 H339 H382 A414 Y444 F110 H122 L219 N220 H222 I229 H230 H273 A305 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 remove_due_to_license_issue P50579 26686773 506 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 5cnj A 2.65 BS01 52Q A 1 R57 R61 S143 Y144 S145 A166 S167 T168 Y216 R271 S272 E273 K377 R36 R40 S100 Y101 S102 A123 S124 T125 Y173 R228 S229 E230 K334 ? 0004930,0007186,0016020 remove_due_to_license_issue Q14416 26313429 602 AKKVLTLEGDLVLGGLFPVHQKGGPAEDCGPVNEHRGIQRLEAMLFALDRINRDPHLLPGVRLGAHILDSCSKDTHALEQALDFVRASLPTAITGVIGGSYSDVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFFQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFELEARARNISVATSEKVGRAMSRAAFEGVVRALLQKPSARVAVLFTRSEDARELLAASQRLNASFTWVASDGWGALESVVAGSEGAAEGAITIELASYPISDFASYFQSLDPWNNSRNPWFREFWEQRFRCSFRQRDCAAHSLRAVPFEQESKIMFVVNAVYAMAHALHNMHRALCPNTTRLCDAMRPVNGRRLYKDFVLNVKFDAPFRPADTHNEVRFDRFGDGIGRYNIFTYLRAGSGRYRYQKVGYWAEGLTLDTSLIPWA 5cnm A 2.84 BS01 52Q A 1 R64 R68 Y150 S151 A172 S173 T174 K389 R35 R39 Y101 S102 A123 S124 T125 K334 ? 0004930,0007186,0016020 remove_due_to_license_issue Q14832 26313429 601 RREIKIEGDLVLGGLFPINEKGTGTEECGRINEDRGIQRLEAMLFAIDEINKDDYLLPGVKLGVHILDTCSRDTYALEQSLEFVRASLIPLLIAGVIGGSYSSVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFYQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFEQEARLRNISIATAEKVGIRKSYDSVIRELLQKPNARVVVLFMRSDDSRELIAAASRANASFTWVASDGWGAQESIIKGSEHVAYGAITLELASQPVRQFDRYFQSLNPYNNHRNPWFRDFWEQKFQCSLQNHRRVCDKHLAIDSSNYEQESKIMFVVNAVYAMAHALHKMQRTLCPNTTKLCDAMKILDGKKLYKDYLLKINFTAPFNPNKDADSIVKFDTFGDGMGRYNVFNFQSYLKVGHWAETLSLDVN 5cp5 A 1.79 BS01 EB0 A 1 W81 P82 F83 L92 L94 N140 D145 I146 M149 W42 P43 F44 L53 L55 N101 D106 I107 M110 ? Kd=1.234uM remove_due_to_license_issue IC50=1530nM, Kd=1234nM O60885 26731490 201 PRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5cp9 B 1.9 BS01 6O5 B 1 F162 E183 W188 F190 R197 Y198 F126 E147 W152 F154 R161 Y162 ? remove_due_to_license_issue P14210 30090230 301 NTIHEFKKSAKTTLIKIDPALKIKTKKVNTADQCANRCTRNKGLPFTCKAFVFDKARKQCLWFPFNSMSSGVKKEFGHEFDLYENKDYIRNCIIGKGRSYKGTVSITKSGIKCQPWSSMIPHEHSFLPSSYRGKDLQENYCRNPRGEEGGPWCFTSNPEVRYEVCDIPQCSEV 5cpr B 2.22 BS03 539 B 1 G229 S251 V252 W264 A268 A269 F281 A289 Y307 G127 S149 V150 W162 A166 A167 F179 A187 Y205 2.1.1.361,2.1.1.362 0042799 Kd=27.8nM remove_due_to_license_issue IC50=25nM Q4FZB7 28114273 403 MSAKELCENDDLATSLVLDPYLGFQTHKMNRQEELKEVIERFKKDEHLEKAFKCLTSGEWARHYFLNKNKMQEKLFKEHVFIYLRMFATDSGFEILPCNRYSSEQNGAKIVATKEWKRNDKIELLVGCIAELSEIEENMLLRHGENDFSVMYSTRKNCAQLWLGPAAFINHDCRPNCKFVSTGRDTACVKALRDIEPGEEISCYYGDGFFGENNEFCECYTCERRGTGAFKS 5cqj A 2.15 BS01 53Q A 1 A47 A92 E96 A35 A64 E68 D26 H43 L137 D14 H31 L109 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 ic50=15.4uM remove_due_to_license_issue P60472 26283394 301 LPAHGCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRE 5cqt A 1.6 BS01 EB3 A 1 W81 P82 F83 L92 L94 N140 I146 M149 W46 P47 F48 L57 L59 N105 I111 M114 ? Kd=0.124uM remove_due_to_license_issue Kd=124nM, IC50=130nM O60885 26731490 201 HHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5cqu A 2.35 BS01 JRJ A 1 L45 G48 V53 V66 F113 M163 I174 D175 L44 G47 V52 V65 F112 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5cr2 A 2.9 BS01 dna D 0 W14 S23 E24 Q25 H28 R29 P30 T52 T53 Q54 K56 R69 W13 S22 E23 Q24 H27 R28 P29 T51 T52 Q53 K55 R68 3.1.27.- 0003677,0003723,0004519,0004521,0005515,0006355,0006402,0006417,0009372,0016075,0030308,0032991,0040008,0042803,0043068,0044010,0044877,0051607,0110001,0140677 remove_due_to_license_issue P0AE70 27026704 1 ~ 7 VSRYVPDMGDLIWVDFDPTKGSEQAGHRPAVVLSPFMYNNKTGMCLCVPCTTQSKGYPFEVVLSGQERDGVALADQVKSIAWRARGATKKGTVAPEELQLIKAKINVLIGH 5cr2 B 2.9 BS01 dna E 0 W14 R29 P30 T52 T53 E68 R69 K91 W11 R26 P27 T49 T50 E65 R66 K88 3.1.27.- 0003677,0003723,0004519,0004521,0005515,0006355,0006402,0006417,0009372,0016075,0030308,0032991,0040008,0042803,0043068,0044010,0044877,0051607,0110001,0140677 remove_due_to_license_issue P0AE70 27026704 1 ~ 3 RYVPDMGDLIWVDFDPTKGSEQAGHRPAVVLSPFMYNNKTGMCLCVPCTTQSKGYPFEVVLSGQERDGVALADQVKSIAWRARGATKKGTVAPEELQLIKAKINVLIG 5cr2 C 2.9 BS01 dna F 0 H28 R29 P30 C51 T52 H26 R27 P28 C49 T50 3.1.27.- 0003677,0003723,0004519,0004521,0005515,0006355,0006402,0006417,0009372,0016075,0030308,0032991,0040008,0042803,0043068,0044010,0044877,0051607,0110001,0140677 remove_due_to_license_issue P0AE70 27026704 1 ~ 3 SRYVPDMGDLIWVDFDPTKGSEQAGHRPAVVLSPFMYNNKTGMCLCVPCTTQSKGYPFEVVLSGQERDGVALADQVKSIAWRARGATKKGTVAPEELQLIKAKINVLIGH 5cr7 A 2.9 BS01 5WO A 1 V59 I466 V34 I432 2.7.1.77,3.1.3.5,3.1.3.99 0000255,0005515,0005524,0005737,0005829,0006204,0008253,0009117,0016740,0016787,0042802,0046037,0046040,0046054,0046085,0046872,0050146,0050483,0050484,0050689,0061630,0070936,0106411 remove_due_to_license_issue P49902 26599519 601 KYRREAYHRVFVNRSLAMEKIKCFGFDMDYTLAVYKSPEYESLGFELTVERLVSIGYPQELLSFAYDSTFPTRGLVFDTLYGNLLKVDAYGNLLVCAHGFNFIRGPETREQYPNKFIQRDDTERFYILNTLFNLPETYLLACLVDFFTNCPRYTSCETGFKDGDLFMSYRSMFQDVRDAVDWVHYKGSLKEKTVENLEKYVVKDGKLPLLLSRMKEVGKVFLATNSDYKYTDKIMTYLFDFPHGPKPGSSHRPWQSYFDLILVDARKPLFFGEGTVLRQVDTKTGKLKIGTQHGIVYSGGSSDTICDLLGAKGKDILYIGDHIFGDKKRQGWRTFLVIPELAQELHVWTDKSSLFEELQSLDIFLAELYKHLDSSSNERPDISSIQRRIKKVTHDMDMCYGMMGSLFRSGSRQTLFASQVMRYADLYAASFINLLYYPFSYLFRAAHVLMPHESTVEHT 5cs3 B 2.5 BS01 EP1 B 1 F162 E183 W188 R197 Y198 V200 F126 E147 W152 R161 Y162 V164 ? remove_due_to_license_issue P14210 30090230 301 NTIHEFKKSAKTTLIKIDPALKIKTKKVNTADQCANRCTRNKGLPFTCKAFVFDKARKQCLWFPFNSMSSGVKKEFGHEFDLYENKDYIRNCIIGKGRSYKGTVSITKSGIKCQPWSSMIPHEHSFLPSSYRGKDLQENYCRNPRGEEGGPWCFTSNPEVRYEVCDIPQCSEV 5cs5 B 1.9 BS01 PIN B 1 F162 E183 G185 W188 F190 R197 Y198 F126 E147 G149 W152 F154 R161 Y162 ? remove_due_to_license_issue P14210 30090230 301 NTIHEFKKSAKTTLIKIDPALKIKTKKVNTADQCANRCTRNKGLPFTCKAFVFDKARKQCLWFPFNSMSSGVKKEFGHEFDLYENKDYIRNCIIGKGRSYKGTVSITKSGIKCQPWSSMIPHEHSFLPSSYRGKDLQENYCRNPRGEEGGPWCFTSNPEVRYEVCDIPQCSEV 5cs6 A 1.88 BS01 K82 A 1 Y255 I258 D259 L265 Y254 I257 D258 L264 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=630uM remove_due_to_license_issue IC50=3000000nM P68400 28451126 404 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5cs6 A 1.88 BS02 K82 A 2 F121 P159 V162 I164 M225 F120 P158 V161 I163 M224 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=630uM remove_due_to_license_issue IC50=3000000nM P68400 28451126 405 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5cs6 A 1.88 BS03 K82 A 3 W24 H183 Q186 W23 H182 Q185 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=630uM remove_due_to_license_issue IC50=3000000nM P68400 28451126 406 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5cs6 A 1.88 BS04 K82 A 4 P295 E296 P294 E295 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=630uM remove_due_to_license_issue IC50=3000000nM P68400 28451126 407 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5csd A 1.45 BS01 ACD A 1 F25 L47 I83 N109 A117 L120 S121 V124 S140 I147 F24 L46 I82 N108 A116 L119 S120 V123 S139 I146 ? Kd=0.000000064M remove_due_to_license_issue A0A093VKV7 28111099 201 TKVKRDISAFQKVIQDISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQILLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAFAGTGP 5csd A 1.45 BS02 ACD A 2 V76 L79 V124 S136 L139 S140 I143 V75 L78 V123 S135 L138 S139 I142 ? Kd=0.000000064M remove_due_to_license_issue A0A093VKV7 28111099 202 TKVKRDISAFQKVIQDISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQILLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAFAGTGP 5csh A 1.59 BS01 54E A 1 F121 P159 V162 I164 M225 F118 P156 V159 I161 M222 D156 K158 N161 D175 P184 S194 D153 K155 N158 D172 P181 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=270uM remove_due_to_license_issue IC50=500000nM P68400 28451126 401 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5csh A 1.59 BS02 54E A 2 Y39 I69 D103 T108 A110 Y36 I66 D100 T105 A107 D156 K158 N161 D175 P184 S194 D153 K155 N158 D172 P181 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=270uM remove_due_to_license_issue IC50=500000nM P68400 28451126 402 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5cso A 1.78 BS01 CTN A 1 Y70 I71 E85 G109 N110 Y111 I155 R163 Y70 I71 E85 G109 N110 Y111 I155 R163 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 29124196 804 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 5csp A 1.5 BS01 54G A 1 V53 K68 F113 I174 D175 V51 K66 F111 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Kd=58uM remove_due_to_license_issue Kd=58000nM P68400 28451126 401 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5cst A 1.78 BS01 CDP A 1 Y70 I71 E85 G109 N110 Y111 E112 I155 R163 Y70 I71 E85 G109 N110 Y111 E112 I155 R163 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 29124196 304 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 5csw A 2.66 BS01 P06 A 1 S465 V471 K483 L505 L514 F516 T529 W531 C532 F583 D594 S17 V23 K35 L57 L66 F68 T81 W83 C84 F135 D146 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S149 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.000000nM, EC50=529nM P15056 26916115 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAREL 5csx A 2.51 BS01 54J A 1 I463 V471 A481 K483 L505 L514 F516 I527 T529 W531 C532 G593 D594 F595 K601 I16 V24 A34 K36 L58 L67 F69 I80 T82 W84 C85 G146 D147 F148 K154 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S159 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.400000nM, Kd=0.330000nM P15056 26916115 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATVKSRSGSILWMAPEVIRMQDPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 5ct7 A 3.17 BS01 55J A 1 I463 V471 A481 K483 E501 L505 L514 I527 T529 W531 C532 F583 G593 D594 F595 I15 V23 A33 K35 E53 L57 L66 I79 T81 W83 C84 F135 G145 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=1200nM, IC50=40nM P15056 26396681 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLAGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 5ctb A 2.4 BS01 57J A 1 V1923 R1954 F1956 S1957 G1958 L2025 E2026 G2029 V444 R475 F477 S478 G479 L546 E547 G550 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFA 5ctb B 2.4 BS01 57J B 1 V1923 R1954 F1956 L2025 E2026 G2029 E2032 V444 R475 F477 L546 E547 G550 E553 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 5ctb B 2.4 BS02 57J C 1 A1761 L1762 K1764 A282 L283 K285 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 5ctc A 2.7 BS01 57K A 1 R1954 L2025 E2026 G2029 R475 L546 E547 G550 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHEASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLES 5ctc B 2.7 BS01 57K B 1 R1954 L2025 E2026 G2029 E2032 R474 L545 E546 G549 E552 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 RPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGL 5cte B 2.34 BS01 57L B 1 R1954 G1955 S1957 G1958 L2025 E2026 G2029 E2032 R475 G476 S478 G479 L546 E547 G550 E553 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFAQDLAKKIRSDHDNAIDGLSEVTDDKEKLLKTLKL 5cte B 2.34 BS02 57L C 1 T1757 A1761 L1762 T278 A282 L283 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 LRPIATPYPVKEWLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGLKLESFAQDLAKKIRSDHDNAIDGLSEVTDDKEKLLKTLKL 5cte C 2.34 BS01 57L B 1 A1761 L1762 A270 L271 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 WLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKSLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGNAIDGLSEVIKMLSTDDKEKLLKTLK 5cte C 2.34 BS02 57L C 1 R1954 G1955 F1956 S1957 G1958 L2025 E2026 G2029 E2032 R463 G464 F465 S466 G467 L534 E535 G538 E541 6.3.4.14,6.4.1.2 0003989,0016874 remove_due_to_license_issue Q00955 26411795 2301 WLQPKRYKAHLMGTTYVYDFPELFRQASSSQWKNFSADVKLTDDFFISNELIEDENGELTEVEREPGANAIGMVAFKITVKTPEYPRGRQFVVVANDITFKIGSFGPQEDEFFNKVTEYARKRGIPRIYLAANSGARIGMAEEIVPLFQVAWNDAANPDKGFQYLYLTSEGMETLKKFDKENSVLTERTVINGEERFVIKTIIGSEDGLGVECLRGSGLIAGATSRAYHDIFTITLVTCRSVGIGAYLVRLGQRAIQVEGQPIILTGASALNKVLGREVYTSNLQLGGTQIMYNNGVSHLTAVDDLAGVEKIVEWMSYVPAKRNMPVPILETKDTWDRPVDFTPTNDETYDVRWMIEGRETESGFEYGLFDKGSFFETLSGWAKGVVVGRARLGGIPLGVIGVETRTVENLIPADPANPNSAETLIQQAGQVWFPNSAFKTAQAINDFNNGEQLPMMILANWRGFSGGQRDMFNEVLKYGSFIVDALVDYKQPIIIYIPPTGELRGGSWVVVDPTINADQMEMYADVNARAGVLEPEGTVEIKFRREKLLDTMNRLDDKYRELRSQLSNKSLAPEVHQQISKQLADRERELLPIYGQISLQFADLHDRSSRMVAKGVISKELEWTEARRFFFWRLRRRLNEEYLIKRLSHQVASRLEKIARIRSWYPASVDHEDDRQVATWIEENYKTLDDKLKGNAIDGLSEVIKMLSTDDKEKLLKTLK 5cu2 A 1.705 BS04 54G A 1 V53 V66 K68 F113 M163 I174 D175 V52 V65 K67 F112 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Kd=58000nM P68400 28495381 404 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5cu4 A 1.56 BS01 54S A 1 V66 K68 F113 N118 L124 Y125 P159 H160 V162 I164 I174 D175 M221 M225 V64 K66 F111 N116 L122 Y123 P157 H158 V160 I162 I172 D173 M219 M223 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Kd=0.32uM remove_due_to_license_issue Kd=320nM, IC50=670nM P68400 28451126 404 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5cuh A 1.83 BS06 LTQ A 1 L187 L188 L222 H226 E227 H230 H236 L243 M247 Y248 L82 L83 L117 H121 E122 H125 H131 L138 M142 Y143 H226 E227 H230 H236 H121 E122 H125 H131 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=24000nM P14780 26871660 306 GFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5cuq A 1.696 BS01 NSC A 1 G81 G109 H110 D131 V132 F133 G76 G104 H105 D126 V127 F128 3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 ic50=7.7uM remove_due_to_license_issue C0LMU0 26726314 301 GETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 5cuu A 2.96 BS01 4GA A 1 K237 D323 K369 K205 D291 K337 3.6.1.1 0000287,0004427,0005737,0006796,0016787,0046872 remove_due_to_license_issue Q4JH30 903 NSYIGTGLDTSLENVKPLPEACKRNVTEFDLVAYGKDEFTLSMEKRVMARMFSAFDVTQLGYLEERKIEHMCKYLGRVMNEDDVKQMKSEINAIDGHITFEKFWAWWCSHPEVPAKKDFFSMVSVDFAVPYHQQQLLTRETGELYTPSYRVLYYFRDMETGKELQVSPWHDIPLYVRDLVRTKPASLPMNRYNFICEIPKWTRAKFEIATGEPFNPIKQDIKNGVPRFYKHGDMMWNYGALPQTWESTDVVFEGGYVGDNDPIDAIEIGMTQFKVGQVGAVKVLGILGMIDDGQMDWKVICISHNDPICRFLKDIHDVPKFLPGCLDAIHEWFRVYKICQGGVENKFVFNGEFKDKSFAMKVIDESHYMWGNLRKINK 5cw8 A 2.6 BS01 55X A 1 E71 F72 N107 Y118 S161 W164 L168 E60 F61 N89 Y100 S143 W146 L150 ? 0000976,0003677,0003700,0006355,0042803 remove_due_to_license_issue P96856 26858250 201 EAQRERRKRILDATMAIASKGGYEAVQMRAVADRADVAVGTLYRYFPSKVHLLVSALGREFSRIDAAGATPFQRLNFMVGKLNRAMQRNPLLTEAMTRAYVFADASAASEVDQVEKLIDSMFARAMANGEPTEDQYHIARVISDVWLSNLLAWLTRRASATDVSKRLDLAVRLLIG 5cw8 B 2.6 BS01 55X B 1 T111 I136 S161 W164 T97 I122 S147 W150 ? 0000976,0003677,0003700,0006355,0042803 remove_due_to_license_issue P96856 26858250 201 SEAQRERRKRILDATMAIASKGGYEAVQMRAVADRADVAVGTLYRYFPSKVHLLVSALGREFSRIDAKAVAGATPFQRLNFMVGKLNRAMQRNPLLTEAMTRAYVFADASAASEVDQVEKLIDSMFARAMANGEPTEDQYHIARVISDVWLSNLLAWLTRRASATDVSKRLDLAVRLLIGD 5cwa A 2.1 BS01 0GA A 1 Y439 I458 A472 G473 K492 Y433 I452 A466 G467 K486 Q254 E307 A323 E351 H388 T415 Y439 R459 G475 E488 K492 Q248 E301 A317 E345 H382 T409 Y433 R453 G469 E482 K486 4.1.3.27 0000162,0004049,0009058,0016829,0046872 ic50=17uM remove_due_to_license_issue P9WFX2 26527146 604 ADLAATTSREDFRLLAAEHRVVPVTRKVLADSETPLSAYRKLAANRPGTFLLESAENGRSWSRWSFIGAGAPTALTVREGQAVWLGAVPKDAPTGGDPLRALQVTLELLATADPGLPPLSGGMVGFFAYDMVRRLERLPERAVDDLCLPDMLLLLATDVAAVDHHEGTITLIANAVNWNGTDERVDWAYDDAVARLDVMTAALGQPLPSTVATFSRPEPRHRAQRTVEEYGAIVEYLVDQIAAGEAFQVVPSQRFEMDTDVDPIDVYRILRVTNPSPYMYLLQVPNSDGAVDFSIVGSSPEALVTVHEGWATTHPIAGTRWRGRTDDEDVLLEKELLADDKERAEHLMLVDLGRNDLGRVCTPGTVRVEDYSHIERYSHVMHLVSTVTGKLGEGRTALDAVTACFPAGTLSGAPKVRAMELIEEVEKTRRGLYGGVVGYLDFAGNADFAIAIRTALMRNGTAYVQAGGGVVADSNGSYEYNEARNKARAVLNAIAAAETLAAPGA 5cxa A 1.3 BS06 55L A 1 G178 G179 L181 T215 H218 E219 H222 H228 K233 V235 P238 T239 Y240 F248 G74 G75 L77 T111 H114 E115 H118 H124 K129 V131 P134 T135 Y136 F144 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27996256 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYAYVDINTFRLSADDIRGIQSLYG 5cxh A 1.9 BS01 55M A 1 L377 G378 V385 A400 K402 A451 G454 P455 K458 L501 S511 D512 L15 G16 V23 A38 K40 A89 G92 P93 K96 L139 S149 D150 D494 A496 R498 N499 D512 K533 D132 A134 R136 N137 D150 K171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5nM remove_due_to_license_issue IC50=132nM P43405 26320624 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHHH 5cxi A 2.0 BS01 5TW A 1 L68 E71 F72 A103 M104 L110 Y118 S161 W164 L55 E58 F59 A89 M90 L96 Y104 S147 W150 ? 0000976,0003677,0003700,0006355,0042803 Kd=280nM remove_due_to_license_issue P96856 26858250 201 QRERRKRILDATMAIASKGGYEAVQMRAVADRADVAVGTLYRYFPSKVHLLVSALGREFSRIDAKTDRSAAGATPFQRLNFMVGKLNRAMQRNPLLTEAMTRAYVFADASAASEVDQVEKLIDSMFARAMANGEPTEDQYHIARVISDVWLSNLLAWLTRRASATDVSKRLDLAVRLLIG 5cxi B 2.0 BS01 5TW B 1 F72 A103 M104 R158 S161 W164 F62 A86 M87 R141 S144 W147 ? 0000976,0003677,0003700,0006355,0042803 Kd=280nM remove_due_to_license_issue P96856 26858250 201 SEAQRERRKRILDATMAIASKGGYEAVQMRAVADRADVAVGTLYRYFPSKVHLLVSALGREFSRIDAKGATPFQRLNFMVGKLNRAMQRNPLLTEAMTRAYVFADASAASEVDQVEKLIDSMFARAMANGEPTEDQYHIARVISDVWLSNLLAWLTRRASATDVSKRLDLAVRLLIGD 5cxz A 1.7 BS01 55U A 1 L377 A400 M450 A451 G454 P455 L501 D512 L15 A38 M83 A84 G87 P88 L134 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=552nM remove_due_to_license_issue IC50=34nM P43405 26320624 703 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHH 5cy3 A 1.76 BS01 55Y A 1 L377 V385 A400 K402 M448 A451 G454 L501 S511 D512 L18 V26 A41 K43 M87 A90 G93 L140 S150 D151 D494 A496 R498 N499 D512 K533 D133 A135 R137 N138 D151 K172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=16nM remove_due_to_license_issue IC50=16nM P43405 26320624 701 PKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEG 5cy9 A 1.55 BS01 E0A A 1 F83 V87 L92 N140 I146 M149 F47 V51 L56 N104 I110 M113 ? Kd=0.218uM remove_due_to_license_issue Kd=218nM, IC50=730nM O60885 26731490 202 HLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5cyi A 2.0 BS01 55S A 1 I10 A31 V64 F80 L83 H84 Q85 D86 K89 L134 I11 A32 V65 F81 L84 H85 Q86 D87 K90 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=160nM, Kd=720nM P24941 26320860 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5cyv A 1.52 BS01 WCA B 1 L23 V37 R38 S41 M62 H117 L20 V34 R35 S38 M59 H109 ? 0003700,0006355,0006950,0046872 remove_due_to_license_issue Q0S6D0 26400178 201 SQALSDDIGFLLSRVGGMVLGAVNKALVPTGLRVRSYSVLVLACEQAEGVNQRGVAATMGLDPSQIVGLVDELEERGLVVRTLRNKLIAATEEGRRLRDDAKARVDAAHGRYFEGIPDTVVNQMRDTLQSIAFPTFVE 5cyv A 1.52 BS02 WCA B 2 F13 S16 R17 G20 G24 N27 K28 V31 R36 F10 S13 R14 G17 G21 N24 K25 V28 R33 ? 0003700,0006355,0006950,0046872 remove_due_to_license_issue Q0S6D0 26400178 202 SQALSDDIGFLLSRVGGMVLGAVNKALVPTGLRVRSYSVLVLACEQAEGVNQRGVAATMGLDPSQIVGLVDELEERGLVVRTLRNKLIAATEEGRRLRDDAKARVDAAHGRYFEGIPDTVVNQMRDTLQSIAFPTFVE 5cyv B 1.52 BS01 WCA B 1 D10 G12 F13 S16 G20 D7 G9 F10 S13 G17 ? 0003700,0006355,0006950,0046872 Kd=11uM remove_due_to_license_issue Q0S6D0 26400178 201 SQALSDDIGFLLSRVGGMVLGAVNKALVPTGLRVRSYSVLVLACEQAEGVNQRGVAATMGLDPSQIVGLVDELEERGLVVRTLDPSDRRNKLIAATEEGRRLRDDAKARVDAAHGRYFEGIPDTVVNQMRDTLQSIAFPTFVE 5cyv B 1.52 BS02 WCA B 2 L23 V37 R38 M62 H117 L20 V34 R35 M59 H114 ? 0003700,0006355,0006950,0046872 Kd=11uM remove_due_to_license_issue Q0S6D0 26400178 202 SQALSDDIGFLLSRVGGMVLGAVNKALVPTGLRVRSYSVLVLACEQAEGVNQRGVAATMGLDPSQIVGLVDELEERGLVVRTLDPSDRRNKLIAATEEGRRLRDDAKARVDAAHGRYFEGIPDTVVNQMRDTLQSIAFPTFVE 5czb A 1.96 BS01 55W A 1 L419 M423 H475 S476 Y477 I482 L489 P495 P496 L497 W528 L417 M421 H473 S474 Y475 I480 L487 P493 P494 L495 W526 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 ic50=0.0257uM remove_due_to_license_issue O92972 27520942 601 SSMSYTWTGALITPCAAEESKLPINPLSNSLLRHHNMVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSIEEACKLTPPHSAKSKFGYGAKDVRNLSSRAVNHIRSVWEDLLEDTETPIDTTIMAKSEVFCVQPGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPKQRVEFLVNTWKSKKCPMGFSYDTRCFDSTVTESDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKATAACRAAKLQDCTMLVNGDDLVVICESAGTQEDAAALRAFTEAMTRYSAPPGDPPQPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPINSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIERLHGLSAFTLHSYSPGEINRVASCLRKLGVPPLRTWRHRARSVRAKLLSQGGRAATCGRYLFNWAVRTKLKLTPIPDLSGWFVAGYSGGDIYH 5czm A 1.303 BS06 R47 A 1 H172 G179 I180 L181 A182 H183 T215 H218 E219 H222 H228 K233 A234 V235 F237 T239 Y240 V243 F248 H68 G75 I76 L77 A78 H79 T111 H114 E115 H118 H124 K129 A130 V131 F133 T135 Y136 V139 F144 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=0.260000nM P39900 27996256 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYAYVDINTFRLSADDIRGIQSLYG 5d0c A 1.49 BS01 E0B A 1 W81 P82 F83 L92 L94 N140 M149 W44 P45 F46 L55 L57 N103 M112 ? Kd=2.34uM remove_due_to_license_issue Kd=2340nM, IC50=3180nM O60885 26731490 206 LVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5d0r A 2.24 BS01 B1T A 1 F45 K95 A97 A100 L101 L102 V167 V172 R176 F336 M337 F338 F39 K89 A91 A94 L95 L96 V161 V166 R170 F330 M331 F332 4.6.1.1 0009190,0035556 Kd=0.43uM remove_due_to_license_issue Q96PN6 26961873 501 EFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFGEKVPDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 5d10 A 2.7 BS01 563 A 1 A293 E339 Y340 M341 G344 L393 A32 E74 Y75 M76 G79 L128 D386 R388 A390 N391 D404 D121 R123 A125 N126 D139 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 26275028 601 DAWEIPRESLRLEVKLGQEVWMGTWNGTTRVAIKTLKPGTMSPEAAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 5d11 A 2.3 BS01 56G A 1 L273 G274 A293 E339 Y340 M341 S342 G344 C345 L393 L16 G17 A36 E76 Y77 M78 S79 G81 C82 L130 D386 R388 A390 N391 D404 F424 D123 R125 A127 N128 D141 F145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 26275028 602 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 5d12 A 3.0 BS01 G97 A 1 L273 G274 A293 M338 Y340 M341 S342 G344 L393 L17 G18 A37 M77 Y79 M80 S81 G83 L132 D386 R388 A390 N391 D404 F424 D125 R127 A129 N130 D143 F151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 26275028 601 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 5d1j A 1.8 BS01 56H A 1 I10 A31 F80 L83 Q85 D86 L134 D145 I10 A29 F64 L67 Q69 D70 L118 D129 D127 K129 Q131 N132 D145 T165 D111 K113 Q115 N116 D129 T132 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=48nM remove_due_to_license_issue IC50=48nM, Kd=69nM, Ki=38nM P24941 15027863 4000 MENFQKVEKIGEYGVVYKARNKLTGEVVALKKIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5d1n A 2.713 BS01 SAH A 1 G38 T39 G40 D61 P62 I93 L110 M111 W113 K115 L116 S200 G30 T31 G32 D53 P54 I85 L102 M103 W105 K107 L108 S192 ? remove_due_to_license_issue C7Q5P8 26609134 301 VLAGKKLTDLDPDEWAKAQASAERILVDVGTGDARTAYRQAIAHPEWLVVGVDPAWQRMTETAVRAARKPAKGGAPNLVLVSSAIETVPAALHGVADEVMVLMPWGKLLRGVVLGEADVLSGLRAVAKPGAPLEISIGTSIWREPIPLEIRDLPELTPETVVSTGLTDRLAALGWQVADVRLVPHTDLDTISSSWARRLGSGATETVLHLRAVAVDPRDPVG 5d1r A 2.0 BS02 56S A 1 V139 C189 F190 V127 C177 F178 ? 0000976,0003677,0003700,0005737,0006355 remove_due_to_license_issue P9WMC9 26396194 305 AREQIEAKIVELGRRQLLDHGAAGLSLRAIARNLGMVSSAVYRYVSSRDELLTLLLVDAYSDLADTVDRARDDTVADSWSDDVIAIARAVRGWAVTNPARWALLYGSPVPGYHAPPDRTAGVATRVVGAFFDAIAAGIATGDIRLTDDVAPQPMSSDFEKIRQEFGFPGDDRVVTKCFLLWAGVVGAISLEVFGQYGADMLTDPGVVFDAQTRLLVAVLAEHHHHHH 5d1r B 2.0 BS01 56S A 1 A210 M212 A197 M199 ? 0000976,0003677,0003700,0005737,0006355 remove_due_to_license_issue P9WMC9 26396194 305 REQIEAKIVELGRRQLLDHGAAGLSLRAIARNLGMVSSAVYRYVSSRDELLTLLLVDAYSDLADTVDRARDDTVADSWSDDVIAIARAVRGWAVTNPARWALLYGSPVPGYHAPPDRTAGVATRVVGAFFDAIAAGIATGDIRLTDDVAPQPMSSDFEKIRQEFGFPGDDRVVTKCFLLWAGVVGAISLEVFGQYGADMLTDPGVVFDAQTRLLVAVLAEHHHHHH 5d1s A 2.1 BS01 56Q A 1 S655 K656 G657 V675 L677 H686 E687 H690 Y728 E735 E739 S386 K387 G388 V406 L408 H417 E418 H421 Y459 E466 E470 H686 E687 H690 Y728 E735 H417 E418 H421 Y459 E466 3.4.24.83 0008237 ic50=9.6uM remove_due_to_license_issue IC50=37000nM P15917 26492514 801 LSRYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDIRDSLSEEEKELLNRINPLSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 5d1t A 2.2 BS02 56R A 1 D328 S655 K656 G657 L677 H686 E687 H690 Y728 E739 D62 S367 K368 G369 L389 H398 E399 H402 Y440 E451 H686 E687 H690 Y728 E735 H398 E399 H402 Y440 E447 3.4.24.83 0008237 ic50=1.7uM remove_due_to_license_issue P15917 26492514 802 RYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDILSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 5d1u A 2.8503 BS01 56P A 1 S655 K656 G657 L677 H686 E687 H690 Y728 E735 E739 S367 K368 G369 L389 H398 E399 H402 Y440 E447 E451 H686 E687 H690 Y728 E735 H398 E399 H402 Y440 E447 3.4.24.83 0008237 remove_due_to_license_issue P15917 26492514 801 RYEKWEKIKQHYQHWSDSLSEEGRGLLKKLQIPIEPKKDDIIHSLSQEEKELLKRIQIDSSDFLSTEEKEFLKKLQIDILSEKEKEFLKKLKLDIQPYDINQRLQDTGGLIDSPSINLDVRKQYKRDIQNIDALLHQSIGSTLYNKIYLYENMNINNLTATLGADLVDSTDNTKINRGIFNEFKKNFKYSISSNYMIVDINERPALDNERLKWRIQLSPDTRAGYLENGKLILQRNIGLEIKDVQIIKQSEKEYIRIDAKVVPKSKIDTKIQEAQLNINQEWNKALGLPKYTKLITFNVHNRYASNIVESAYLILNEWKNNIQSDLIKKVTNYLVDGNGRFVFTDITLPNIAEQYTHQDEIYEQVHSKGLYVPESRSILLHGPSKGVELRNDSEGFIHEFGHAVDDYAGYLLDKNQSDLVTNSKKFIDIFKEEGSNLTSYGRTNEAEFFAEAFRLMHSTDHAERLKVQKNAPKTFQFINDQIKFIINS 5d1w A 3.59 BS01 PLM A 1 V86 G104 F105 C176 V74 G92 F93 C164 ? 0000976,0003677,0003700,0005737,0006355 remove_due_to_license_issue O05892 26396194 301 RIPYAEASRALLRDSVLDAMRDLLLTRDWSAITLSDVARAAGISRQTIYNEFGSRQGLAQGYALRLADRLVDNVHASLDANVGNFYEAFLQGFRSFFAESAADPLVISLLTGVAKPDLLQLITTDSAPIITRASARLAPAFTDTWVATTDNDANVLSRAIVRLCLSYVSMPPEADHDVAADLARLITPFAERHGV 5d21 A 1.9 BS02 56N A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 remove_due_to_license_issue Q05097 26416170 902 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 5d24 A 1.65 BS01 L26 A 1 W81 P82 F83 Q84 Q85 V87 K91 L92 Y139 N140 I146 W39 P40 F41 Q42 Q43 V45 K49 L50 Y97 N98 I104 ? Kd=5.8uM remove_due_to_license_issue Kd=5800nM O60885 26731611 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d25 A 1.7 BS01 56M A 1 W81 P82 Q85 V87 K91 L92 N140 I146 W39 P40 Q43 V45 K49 L50 N98 I104 ? Kd=0.46uM remove_due_to_license_issue Kd=460nM O60885 26731611 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5d26 A 1.82 BS01 L28 A 1 W81 P82 Q85 V87 K91 L92 N140 I146 W40 P41 Q44 V46 K50 L51 N99 I105 ? Kd=0.81uM remove_due_to_license_issue Kd=810nM O60885 26731611 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d29 A 1.8 BS04 5Q1 A 1 Y234 H377 D387 E424 E425 D453 N519 R534 G548 Y552 H553 Y700 Y179 H322 D332 E369 E370 D398 N464 R479 G487 Y491 H492 Y636 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=97nM remove_due_to_license_issue IC50=97nM Q04609 27074627 818 HNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 5d2a A 2.134 BS04 ZDC E 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 29896342 101 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 5d2a B 2.134 BS03 ZDC D 1 S22 S23 D96 D99 D101 D104 S22 S23 D96 D99 D101 D104 ? 0030246,0044010,0046872 remove_due_to_license_issue Q9HYN5 29896342 101 ATQGVFTLPANTRFGVTAFANSSGTQTVNVLVNNETAATFSGQSTNNAVIGTQVLNSGSSGKVQVQVSVNGRPSDLVSAQVILTNELNFALVGSEDGTDNDYNDAVVVINWPLG 5d2r A 1.9 BS04 56W A 1 Q46 E49 R86 N93 R94 H126 H128 G130 W148 M203 T208 A220 E222 K225 Q28 E31 R68 N75 R76 H108 H110 G112 W130 M185 T190 A202 E204 K207 ? 0046872 Ki=1.5uM remove_due_to_license_issue B5ZAD9 26735022 523 SMEMIEKAPTDLEDRDKAPHLLLLAGIQGDEPGGFNATNLFLMHYSVLKGLVEVVPVLNKPSMLRNHRGLYGDMNRKFAALDKKDPEYPTIQEIKSLIAKPNIDAVLHLHDGGGYYRPVYVDAMLNPKRWGNCFIIDQDEVKGAKFPNLLAFANNTIESINAHLLHPIEEYHLKNTRTAQGDTEMQKALTFYAINQKKSAFANEASKELPLASRVFYHLQAIEGLLNQLNIPFKRDFELNPSSVHALINDKSLWAKISSLPKIPLFNLRPRLNHFPLPHNTKIPQIPIESNAYIVGLVKNKQEVFLKYGNKLMTRLSPFYIEFDPSLEEVKMQIDNKDQMVKIGSVVEVKESFYIHAMDNIRANVIGFSVSNENKPNEAGYTIRFKDFQKRFSLDKQERIYRIEFYKNNAFSGMILVKFV 5d39 A 3.2 BS01 dna N 0 R370 S378 V379 V414 H415 N417 R208 S216 V217 V252 H253 N255 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCERKGTESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 A 3.2 BS02 dna M 0 K288 H415 K138 H253 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFLPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCERKGTESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 B 3.2 BS01 dna E 0 K288 H415 K136 H248 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCEGTESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 B 3.2 BS02 dna F 0 R370 S378 V379 V414 N417 R205 S211 V212 V247 N250 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCEGTESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 C 3.2 BS01 dna N 0 K284 K288 H415 K135 K139 H250 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCETESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 C 3.2 BS02 dna M 0 R370 V379 V414 H415 N417 Q418 R208 V214 V249 H250 N252 Q253 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCETESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 D 3.2 BS01 dna E 0 R370 S378 V379 V414 H415 Q418 R209 S214 V215 V250 H251 Q254 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALQEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCETESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d39 D 3.2 BS02 dna F 0 K284 K288 H415 K136 K140 H251 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P42226 27803324 1 ~ 21 QEELKFKTGLRRLQHRVGEIHLLREALQEALAMLLQETTGELEAAKALVLKRIQIWKRQQQLAGNGAPFEESLAPLQERCESLVDIYSQLQQEVGAAGGELEPKTRASLTGRLDEVLRTLVTSCFLVEKQPPQVLKTQTKFQAGVRFLLGLRFPAKPPLVRADMVTEKQARELESTGEIINNTVPLENSIPGNCCSALFKNLLLKKIKRCETESVTEEKCAVLFSASFTLGPGKLPIQLQALSLPLVVIVHGNQDNNAKATILWDNAFSEMDRVPFVVAERVPWEKMCETLNLKFMAEVGTNRGLLPEHFLFLAQKIFNDNSLSMEAFQHRSVSWSQFNKEILLGRGFTFWQWFDGVLDLTKRCLRSYWSDRLIIGFISKQYVTSLLLNEPDGTFLLRFSDSEIGGITIAHVIRGQDGSPQIENIQPFSAKDLSIRSLGDRIRDLAQLKNLYPKKPKDEAFRSHYKPEQMGKDGRGYVPATIKMTVE 5d3c A 1.314 BS06 56O A 1 G178 G179 I180 L181 A182 T215 H218 E219 H222 H228 K233 V235 P238 T239 Y240 F248 G74 G75 I76 L77 A78 T111 H114 E115 H118 H124 K129 V131 P134 T135 Y136 F144 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27996256 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYAYVDINTFRLSADDIRGIQSLYG 5d3g A 2.3 BS01 dna E 0 W24 F61 L74 D76 R78 E89 I94 Q151 G152 K154 P157 Y183 M184 D185 M230 G231 Q258 K259 G262 K263 W266 S280 R284 G285 K353 R358 G359 H361 R448 T473 Q475 K476 Y501 W24 F61 L74 D76 R78 E89 I94 Q151 G152 K154 P157 Y183 M184 D185 M230 G231 Q258 K259 G262 K263 W266 S280 R284 G285 K353 R358 G359 H361 R448 T473 Q475 K476 Y501 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 26296781 -2 ~ 33 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVS 5d3g C 2.3 BS01 dna F 0 W24 L74 R78 N81 E89 I94 Q151 G152 K154 P157 Y183 M184 D185 M230 G231 Q258 K259 G262 K263 W266 S280 R284 G285 T286 K353 H361 R448 T473 Q475 K476 Y501 W24 L74 R78 N81 E89 I94 Q151 G152 K154 P157 Y183 M184 D185 M230 G231 Q258 K259 G262 K263 W266 S280 R284 G285 T286 K353 H361 R448 T473 Q475 K476 Y501 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 26296781 -2 ~ 33 PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVS 5d3h A 1.7 BS01 57G A 1 W81 P82 Q85 V87 K91 L92 N140 I146 W39 P40 Q43 V45 K49 L50 N98 I104 ? Kd=7.9uM remove_due_to_license_issue Kd=7900nM O60885 26731611 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5d3j A 1.7 BS01 L33 A 1 W81 P82 V87 K91 L92 N140 W39 P40 V45 K49 L50 N98 ? Kd=5.7uM remove_due_to_license_issue Kd=5700nM O60885 26731611 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d3l A 1.5 BS01 57F A 1 W81 P82 F83 V87 L92 Y97 Y139 N140 I146 W40 P41 F42 V46 L51 Y56 Y98 N99 I105 ? Kd=0.88uM remove_due_to_license_issue Kd=880nM O60885 26731611 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d3n A 2.15 BS01 L40 A 1 W81 P82 V87 K91 L92 Y139 N140 I146 W39 P40 V45 K49 L50 Y97 N98 I104 ? Kd=9.2uM remove_due_to_license_issue Kd=9200nM O60885 26731611 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d3p A 1.95 BS01 57E A 1 W81 P82 V87 K91 L92 Y97 Y139 N140 I146 W40 P41 V46 K50 L51 Y56 Y98 N99 I105 ? Kd=7.4uM remove_due_to_license_issue O60885 26731611 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d3s A 1.75 BS01 579 A 1 W81 P82 Q85 V87 L92 Y139 N140 I146 W39 P40 Q43 V45 L50 Y97 N98 I104 ? Kd=1.3uM remove_due_to_license_issue Kd=1300nM O60885 26731611 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5d3t A 1.93 BS01 56Y A 1 P82 V87 K91 L92 Y139 N140 I146 P41 V46 K50 L51 Y98 N99 I105 ? Kd=12uM remove_due_to_license_issue Kd=12000nM O60885 26731611 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5d3x A 1.69 BS01 4IP A 1 K280 S282 N285 R289 Y300 R328 K368 K39 S41 N44 R48 Y59 R73 K113 ? Kd=440nM remove_due_to_license_issue Q8TCU6 27150042 501 GEFEKLEALEQLQSHIEGWEGSNLTDICTQLLLQGTLLKISAGNIQERAFFLFDNLLVYCKRKSINGSLYIFRGRINTEVMEVENVEDGTADYHSNGYTVTNGWKIHNTAKNKWFVCMAKTAEEKQKWLDAIIREREQRESLKLGMERDAY 5d45 A 1.65 BS01 57P A 1 F16 M40 S53 D76 R126 Y128 F20 M44 S57 D80 R130 Y132 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.12uM remove_due_to_license_issue Ki=120nM P15090 27096055 201 GSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5d47 A 1.7 BS01 L19 A 1 F16 M20 A33 M40 S53 S55 K58 D76 R126 Y128 F20 M24 A37 M44 S57 S59 K62 D80 R130 Y132 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.1uM remove_due_to_license_issue Ki=100nM P15090 27096055 201 GSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5d48 A 1.81 BS01 L96 A 1 F16 M40 I51 S53 S55 F57 K58 T60 D76 R126 Y128 F21 M45 I56 S58 S60 F62 K63 T65 D81 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.03uM remove_due_to_license_issue Ki=30nM P15090 27096055 201 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5d4a A 1.7 BS01 57Q A 1 F16 Y19 P38 F57 D76 R78 R126 Y128 F21 Y24 P43 F62 D81 R83 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 remove_due_to_license_issue Ki=>1400nM P15090 27096055 201 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5d4r A 2.07 BS01 dna T 0 P3 K4 Y5 S40 H42 T43 Q61 G62 G63 P17 K18 Y19 S54 H56 T57 Q75 G76 G77 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 1 ~ 21 HLEVLFQGPLGSEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4r A 2.07 BS02 dna U 0 L-4 T29 E30 R41 R45 Q61 G62 G64 L10 T43 E44 R55 R59 Q75 G76 G78 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 22 ~ 42 HLEVLFQGPLGSEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4r B 2.07 BS01 dna T 0 T29 E30 R41 R45 Q61 G62 G64 T32 E33 R44 R48 Q64 G65 G67 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 1 ~ 21 SEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4r B 2.07 BS02 dna U 0 P3 K4 Y5 S40 H42 T43 Q61 G62 G63 P6 K7 Y8 S43 H45 T46 Q64 G65 G66 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 22 ~ 42 SEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4s A 1.972 BS01 dna T 0 P3 K4 Y5 S40 H42 T43 Q61 G62 P5 K6 Y7 S42 H44 T45 Q63 G64 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 1 ~ 21 EFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4s A 1.972 BS02 dna U 0 T29 E30 R45 S59 Q61 G62 G64 T31 E32 R47 S61 Q63 G64 G66 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 1 ~ 21 EFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4s B 1.972 BS01 dna T 0 T29 E30 R41 R45 Q61 G62 G64 T44 E45 R56 R60 Q76 G77 G79 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 1 ~ 21 HHHLEVLFQGPLSEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d4s B 1.972 BS02 dna U 0 P3 K4 Y5 S40 H42 T43 Q61 G62 P18 K19 Y20 S55 H57 T58 Q76 G77 ? 0003700,0006355 remove_due_to_license_issue P96711 26511320 1 ~ 21 HHHLEVLFQGPLSEFMLPKYAQVKEEISSWINQGKILPDQKIPTENELMQQFGVSRHTIRKAIGDLVSQGLLYSVQGGGTFVA 5d6e A 1.49 BS01 94A A 1 F219 H231 N327 L328 N329 H331 I338 E364 A414 Y444 F111 H123 N219 L220 N221 H223 I230 E256 A306 Y336 D251 D262 H331 H339 E364 E459 D143 D154 H223 H231 E256 E351 3.4.11.18 0006508,0070006 remove_due_to_license_issue P50579 26686773 501 PKVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 5d6f A 1.55 BS01 57R A 1 H231 N327 L328 N329 I338 E364 A414 Y444 H122 N218 L219 N220 I229 E255 A305 Y335 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E255 E350 3.4.11.18 0006508,0070006 remove_due_to_license_issue P50579 26686773 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 5d6j A 2.25 BS01 ATP A 1 T187 S188 G189 S190 T191 R192 S314 E315 P316 S342 G344 L345 A346 D469 I480 R483 T187 S188 G189 S190 T191 R192 S314 E315 P316 S342 G344 L345 A346 D469 I480 R483 N207 H231 A346 N207 H231 A346 6.2.1.20 0005524,0005886,0006631,0006633,0008610,0008922,0016874,0070566 Kd=36uM remove_due_to_license_issue A0R618 26628098 702 MPFHNPFIKDGQIKFPDGSSIVAHVERWAKVRGDKLAYRFLDFSTERDGVPRDLTWAQFSARNRAVAARLQQVTQPGDRVAILCPQNLDYLVAFFGALYAGRIAVPLFDPSEPGHVGRLHAVLDNCHPSAILTTTEAAEGVRKFFRTRPANQRPRVIAVDAVPDDVASTWVNPDEPDETTIAYLQYTSGSTRIPTGVQITHLNLATNVVQVIEALEGEEGDRGLSWLPFFHDMGLITALLAPMIGHYFTFMTPAAFVRRPERWIRELARKEGDTGGTISVAPNFAFDHAAARGVPKPGSPPLDLSNVKAVLNGSEPISAATVRRFNEAFGPFGFPPKAIKPSYGLAEATLFVSTTPSAEEPKIITVDRDQLNSGRIVEVDADSPKAVAQASAGKVGIAEWAVIVDAESATELPDGQVGEIWISGQNMGTGYWGKPEESVATFQNILKSRTNPSHAEGATDDATWVRTGDYGAFYDGDLYITGRVKDLVIIDGRNHYPQDLEYSAQEASKAIRTGYVAAFSVPANQLPDEVFENAHSGIKRDPDDTSEQLVIVAERAPGAHKLDIGPITDDIRAAIAVRHGVTVRDVLLTAAGAIPRTSSGKIGRRACRAAYLDGSLRAGKVANDFPDATD 5d6p A 2.05 BS01 57U A 1 I51 S55 E58 V79 D81 R84 G85 P87 I102 I36 S40 E43 V64 D66 R69 G70 P72 I87 5.6.2.2 0003677,0003918,0005524,0006265 ic50=2.5uM remove_due_to_license_issue IC50=2500nM P0A0K8 26460684 301 AGQIQVLEGLEAVRKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYE 5d6q B 1.5 BS01 57V B 1 N54 D81 R84 I86 P87 I102 R144 N35 D62 R65 I67 P68 I80 R99 5.6.2.2 0003677,0003918,0005524,0006265 ic50=5.8uM remove_due_to_license_issue IC50=5800nM P0A0K8 26460684 303 QVLEGLEAVRKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQGRPAVEVILTSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYEG 5d75 A 1.83 BS01 FK5 A 1 Y135 D146 L162 K170 V171 I172 W175 Y198 Q203 A206 Y27 D38 L54 K62 V63 I64 W67 Y90 Q95 A98 Y135 F145 D146 I172 Y198 F216 Y27 F37 D38 I64 Y90 F108 5.2.1.8 0003755 Ki=200nM remove_due_to_license_issue Q00688 26749369 301 PKYTKSVLKKGDKTNFPKKGDVVHCWYTGTLQDGTVFDTNIQTSAKKKKNAKPLSFKVGVGKVIRGWDEALLTMSKGEKARLEIEPEWAYGKKGQPDAKIPPNAKLTFEVELVDIDLEHH 5d7a A 2.9 BS01 58C A 1 V31 V39 A52 M105 E106 C108 G111 D115 Q157 L160 V170 V21 V29 A42 M95 E96 C98 G101 D105 Q147 L150 V160 D153 K155 Q157 N158 D171 T191 D143 K145 Q147 N148 D161 T170 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9UKE5 27562646 401 DEIDLSALRDPAGIFELVELVGNGTYGQVYKGRHVKTGQLAAIKVMDVTGDEEEEIKQEINMLKKYSHHRNIATYYGAFIKKNPPGMDDQLWLVMEFCGAGSVTDLIKNTKGNTLKEEWIAYICREILRGLSHLHQHKVIHRDIKGQNVLLTENAEVKLVDFGVNTFIGTPYWMAPEVIACDENPDATYDFKSDLWSLGITAIEMAEGAPPLCDMHPMRALFLIPRNPAPRLKSKKWSKKFQSFIESCLVKNHSQRPATEQLMKHPFIRDQPNERQVRIQLKDHIDRTK 5d7c A 1.55 BS01 57W A 1 S55 E58 V79 D81 R84 G85 I86 P87 I102 R144 T173 I175 S40 E43 V64 D66 R69 G70 I71 P72 I87 R106 T135 I137 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.14uM remove_due_to_license_issue IC50=140nM P0A0K8 26460684 303 AGQIQVLEGLEAVRKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYE 5d7r A 1.55 BS02 57Y A 1 I51 N54 S55 E58 V79 D81 R84 G85 I86 P87 R144 T173 I175 I37 N40 S41 E44 V65 D67 R70 G71 I72 P73 R107 T136 I138 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.013uM remove_due_to_license_issue P0A0K8 26487916 306 GAGQIQVLEGLEAVRKRPGMYIGSTSERGLHHLVWEIVDNSIDEALAGYANQIEVVIEKDNWIKVTDNGRGIPVDIQEKMGRPAVEVILTSSVVNALSQDLEVYVHRNETIYHQAYKKGVPQFDLKEVGTTDKTGTVIRFKADGEIFTETTVYNYETLQQRIRELAFLNKGIQITLRDERDEENVREDSYHYE 5d7x A 1.35 BS01 XZ8 A 1 I652 F653 V657 P658 F714 I28 F29 V33 P34 F90 ? Kd=15uM remove_due_to_license_issue Kd=15000nM P55201 26982797 802 SMEMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5d9k A 2.55 BS01 584 A 1 G75 F79 V82 A98 V131 D148 F149 L150 L200 D211 F212 G14 F18 V21 A37 V70 D87 F88 L89 L139 D150 F151 D193 K195 E197 N198 D211 T231 D132 K134 E136 N137 D150 T158 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=4.0nM P51812 26270416 401 KADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRTKMERDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKPATFYFDP 5d9l A 2.15 BS01 583 A 1 V82 A98 K100 L147 F149 L150 L200 D211 F212 V34 A50 K52 L99 F101 L102 L152 D163 F164 D193 K195 E197 N198 D211 T231 D145 K147 E149 N150 D163 T171 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.024uM remove_due_to_license_issue P51812 26270416 1001 EIAITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRTKMERDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKEGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKPATGRPEDTFYFDP 5d9p A 1.8 BS01 NBG C 1 H112 H113 N161 E162 H238 Y240 E280 D288 W324 H107 H108 N156 E157 H233 Y235 E275 D283 W319 ? 0000272,0004553 remove_due_to_license_issue O06842 26507654 1 ATYMEESAQSAVDNFGLGFNLGNTLDANGCGTGKPVATYETFWGQPETTQDMMTFLMQNGFNAVRIPVTWYEHMDAEGNVDEAWMMRVKAIVEYAMNAGLYAIVNVHHDTAAGSGAWIKADTDVYAATKEKFKKLWTQIANALADYDQHLLFEGYNEMLDGNNSWDEPQKASGYEALNNYAQDFVDAVRATGGNNATRNLIVNTYAAAKGENVLNNFMLPTDAVNNHLIVQVHSYDPWNFFNTKTTWDSECHNTLTEIFSALSKKFTTIPYIIGEYGTHGESDISVSKSSPAEKIKLAADQAADMVKLAKDHHSATFYWMSIFDGSDRIQPQWSLPTVVEAMQEAYN 5d9y A 1.971 BS01 dna B 0 R1261 R1262 S1286 S1290 M1293 Y1294 K1299 R1302 S1303 T1372 T1463 Y1902 H1904 R130 R131 S155 S159 M162 Y163 K168 R171 S172 T241 T332 Y394 H396 1.14.11.80 0070579,0141167 remove_due_to_license_issue Q6N021 26524525 1 ~ 12 SCRCVEQIIEKDEGPFYTHLGAGPNVAAIREIMEERFGQKGKAIRIERVIYTGKEGKSSQGCPIAKWVVRRSSSEEKLLCLVRERAGHTCEAAVIVILILVWEGIPLSLADKLYSELTETLRKYGTLTNRRCALNEERTCACQGLDPETCGASFSFGCSWSMYYNGCKFARSKIPRKFKLLGDDPKEEEKLESHLQNLSTLMAPTYKKLAPDAYNNQIEYEHRAPECRLGLKEGRPFSGVTACLDFCAHAHRDLHNMQNGSTLVCTLTREDNREFGGKPEDEQLHVLPLYKVSDVDEFGSVEAQEEKKRSGAIQVLSSFRRKVRMLAEPVKTCGSDEVWSDSEQSFLDPDIGGVAVAPTHGSILIECAKRELHATTPLKNPNRNHPTRISLVFYQHKSMNEPKHGLALWEAKM 5d9y A 1.971 BS02 dna C 0 M1293 Y1294 N1296 M162 Y163 N165 1.14.11.80 0070579,0141167 remove_due_to_license_issue Q6N021 26524525 1 ~ 12 SCRCVEQIIEKDEGPFYTHLGAGPNVAAIREIMEERFGQKGKAIRIERVIYTGKEGKSSQGCPIAKWVVRRSSSEEKLLCLVRERAGHTCEAAVIVILILVWEGIPLSLADKLYSELTETLRKYGTLTNRRCALNEERTCACQGLDPETCGASFSFGCSWSMYYNGCKFARSKIPRKFKLLGDDPKEEEKLESHLQNLSTLMAPTYKKLAPDAYNNQIEYEHRAPECRLGLKEGRPFSGVTACLDFCAHAHRDLHNMQNGSTLVCTLTREDNREFGGKPEDEQLHVLPLYKVSDVDEFGSVEAQEEKKRSGAIQVLSSFRRKVRMLAEPVKTCGSDEVWSDSEQSFLDPDIGGVAVAPTHGSILIECAKRELHATTPLKNPNRNHPTRISLVFYQHKSMNEPKHGLALWEAKM 5da3 A 1.7 BS01 58V A 1 R195 L197 K219 L248 M267 A268 G270 L319 D330 R12 L14 K36 L64 M83 A84 G86 L135 D146 D312 A314 R316 N317 D330 I349 D128 A130 R132 N133 D146 I165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=80nM remove_due_to_license_issue IC50=>600nM Q13882 27993680 503 MERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRDSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPTFKALRERLSSFTSHH 5db0 A 1.5 BS01 58P A 1 S155 L177 S178 H181 F238 Y276 M278 Y319 M322 Y323 W341 E363 E366 S134 L156 S157 H160 F217 Y255 M257 Y298 M301 Y302 W320 E342 E345 ? 0005634 ic50=46nM remove_due_to_license_issue O00255 26744767 610 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5db1 A 1.86 BS01 58O A 1 S155 S178 H181 F238 Y276 M278 Y319 M322 Y323 W341 E363 S134 S157 H160 F217 Y255 M257 Y298 M301 Y302 W320 E342 ? 0005634 ic50=22nM remove_due_to_license_issue O00255 26744767 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5db2 A 1.54 BS01 58R A 1 S155 S178 H181 F238 Y276 M278 M322 Y323 W341 E363 E366 K588 S134 S157 H160 F217 Y255 M257 M301 Y302 W320 E342 E345 K466 ? 0005634 ic50=25nM remove_due_to_license_issue O00255 26744767 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5db3 A 1.71 BS01 58Q A 1 S155 L177 S178 H181 F238 Y276 M278 Y319 M322 Y323 W341 E363 E366 S134 L156 S157 H160 F217 Y255 M257 Y298 M301 Y302 W320 E342 E345 ? 0005634 ic50=12nM remove_due_to_license_issue O00255 26744767 610 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5dbm A 1.86 BS01 58N A 1 L1109 P1110 V1115 L1120 Y1125 N1168 L27 P28 V33 L38 Y43 N86 2.3.1.-,2.3.1.48 Kd=0.35uM remove_due_to_license_issue IC50=456nM Q92793 27056325 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5dcz A 2.23 BS02 59B A 1 H1031 G1032 S1033 R1047 H1048 A1049 Y1050 Y1060 S1068 Y1071 E1138 H80 G81 S82 R96 H97 A98 Y99 Y109 S117 Y120 E180 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFAHSPPGHHSVTGRPNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5dd9 A 1.62 BS01 59K A 1 S155 L177 S178 H181 F238 C241 Y276 M278 N282 Y319 M322 Y323 K588 S134 L156 S157 H160 F217 C220 Y255 M257 N261 Y298 M301 Y302 K466 ? 0005634 ic50=779nM remove_due_to_license_issue IC50=779nM O00255 26288158 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5dda A 1.83 BS01 59M A 1 S155 L177 S178 H181 F238 C241 Y276 M278 N282 Y319 Y323 S134 L156 S157 H160 F217 C220 Y255 M257 N261 Y298 Y302 ? 0005634 ic50=1653nM remove_due_to_license_issue IC50=1653nM O00255 26288158 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQM 5ddb A 1.54 BS01 59Q A 1 S155 L177 S178 H181 C241 Y276 M278 N282 Y319 M322 Y323 S133 L155 S156 H159 C219 Y254 M256 N260 Y297 M300 Y301 ? 0005634 ic50=82nM remove_due_to_license_issue IC50=82nM O00255 26288158 601 LKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQ 5ddc A 1.62 BS01 59V A 1 S155 L177 S178 H181 F238 C241 Y276 M278 N282 Y319 M322 Y323 S133 L155 S156 H159 F216 C219 Y254 M256 N260 Y297 M300 Y301 ? 0005634 ic50=92nM remove_due_to_license_issue IC50=92nM O00255 26288158 601 LKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5ddd A 2.14 BS01 59X A 1 S178 C241 Y276 M278 N282 Y319 M322 Y323 S157 C220 Y255 M257 N261 Y298 M301 Y302 ? 0005634 ic50=260nM remove_due_to_license_issue IC50=260nM O00255 26288158 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5dde A 1.78 BS01 5A0 A 1 S155 H181 F238 C241 Y276 M278 N282 Y319 M322 Y323 S134 H160 F217 C220 Y255 M257 N261 Y298 M301 Y302 ? 0005634 ic50=65nM remove_due_to_license_issue IC50=65nM O00255 26288158 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5dde A 1.78 BS02 5A0 A 2 S155 L177 F238 C241 Y276 M278 N282 Y319 M322 Y323 S134 L156 F217 C220 Y255 M257 N261 Y298 M301 Y302 ? 0005634 ic50=65nM remove_due_to_license_issue IC50=65nM O00255 26288158 602 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 5ddf A 1.66 BS01 5A1 A 1 S155 S178 E179 D180 H181 Y276 M278 N282 Y319 M322 Y323 Q586 S134 S157 E158 D159 H160 Y255 M257 N261 Y298 M301 Y302 Q464 ? 0005634 ic50=674nM remove_due_to_license_issue IC50=674nM O00255 26288158 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQ 5deu A 1.801 BS01 dna B 0 R1261 R1262 S1286 S1290 Y1294 K1299 S1303 T1372 D1384 H1386 N1387 Y1902 H1904 R130 R131 S155 S159 Y163 K168 S172 T241 D253 H255 N256 Y394 H396 1.14.11.80 0070579,0141167 remove_due_to_license_issue Q6N021 26524525 1 ~ 12 SCRCVEQIIEKDEGPFYTHLGAGPNVAAIREIMEERFGQKGKAIRIERVIYTGKEGKSSQGCPIAKWVVRRSSSEEKLLCLVRERAGHTCEAAVIVILILVWEGIPLSLADKLYSELTETLRKYGTLTNRRCALNEERTCACQGLDPETCGASFSFGCSWSMYYNGCKFARSKIPRKFKLLGDDPKEEEKLESHLQNLSTLMAPTYKKLAPDAYNNQIEYEHRAPECRLGLKEGRPFSGVTACLDFCAHAHRDLHNMQNGSTLVCTLTREDNREFGGKPEDEQLHVLPLYKVSDVDEFGSVEAQEEKKRSGAIQVLSSFRRKVRMLAEPVKTCGSDEVWSDSEQSFLDPDIGGVAVAPTHGSILIECAKRELHATTPLKNPNRNHPTRISLVFYQHKSMNEPKHGLALWEAKM 5deu A 1.801 BS02 dna C 0 W1291 M1293 Y1294 N1296 K1905 W160 M162 Y163 N165 K397 1.14.11.80 0070579,0141167 remove_due_to_license_issue Q6N021 26524525 2 ~ 12 SCRCVEQIIEKDEGPFYTHLGAGPNVAAIREIMEERFGQKGKAIRIERVIYTGKEGKSSQGCPIAKWVVRRSSSEEKLLCLVRERAGHTCEAAVIVILILVWEGIPLSLADKLYSELTETLRKYGTLTNRRCALNEERTCACQGLDPETCGASFSFGCSWSMYYNGCKFARSKIPRKFKLLGDDPKEEEKLESHLQNLSTLMAPTYKKLAPDAYNNQIEYEHRAPECRLGLKEGRPFSGVTACLDFCAHAHRDLHNMQNGSTLVCTLTREDNREFGGKPEDEQLHVLPLYKVSDVDEFGSVEAQEEKKRSGAIQVLSSFRRKVRMLAEPVKTCGSDEVWSDSEQSFLDPDIGGVAVAPTHGSILIECAKRELHATTPLKNPNRNHPTRISLVFYQHKSMNEPKHGLALWEAKM 5dex B 2.4 BS01 5E0 B 1 H88 T116 R121 T134 G135 G172 S173 T174 Y214 D215 H82 T110 R115 T128 G129 G166 S167 T168 Y208 D209 ? 0015276,0016020 Ki=22.6nM remove_due_to_license_issue Q00959 28760974 301 DNHLSIVTLEEAPFVIVEDIDPTETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGICH 5dey A 2.1 BS01 59T A 1 A297 K299 E315 V342 M344 Y346 L347 D393 L396 A48 K50 E66 V93 M95 Y97 L98 D144 L147 N389 K391 D393 N394 D407 P416 T427 N140 K142 D144 N145 D158 P167 T178 2.7.11.1 0004672,0005524,0006468 Ki=3.7nM remove_due_to_license_issue Ki=3.7nM, IC50=69nM Q13153 26713112 601 DEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATKNN 5dfp A 2.2 BS01 59U A 1 A297 R299 E315 V342 M344 Y346 L347 G350 D354 L396 A49 R51 E67 V94 M96 Y98 L99 G102 D106 L148 D389 K391 D393 N394 D407 P416 T427 D141 K143 D145 N146 D159 P168 T179 2.7.11.1 0004672,0005524,0006468 Ki=22nM remove_due_to_license_issue Ki=22nM, IC50=222nM Q13153 26713112 601 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT 5dg6 A 2.35 BS01 V66 A 1 H30 E54 I109 Q110 T134 P136 C139 H157 A158 A159 A160 H31 E55 I110 Q111 T126 P128 C131 H149 A150 A151 A152 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 26823007 203 HAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 5dgj A 1.0 BS01 V64 A 1 H30 E54 I109 Q110 C139 A158 A159 A160 H32 E56 I111 Q112 C137 A156 A157 A158 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 26823007 201 HHAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGMDLGDCGAPYVHKRGNDWVVCGVHAAATNTVVCAVQA 5dgm F 2.86 BS01 59Z F 1 Y10 K57 N59 R60 F206 F239 L344 I348 Y3 K50 N52 R53 F199 F232 L337 I341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 26457482 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5dgu A 1.22 BS01 5B7 A 1 D25 A28 D30 G48 P81 V82 D25 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.0045nM remove_due_to_license_issue P04585 26462551 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5dgu B 1.22 BS01 5B7 A 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 26462551 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5dgw A 1.62 BS01 5B5 A 1 D25 A28 D30 P81 V82 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.009nM remove_due_to_license_issue P04585 26462551 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5dgw B 1.62 BS01 5B5 A 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 26462551 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5dgz A 2.502 BS01 L20 A 1 L44 G45 F49 A65 K67 E171 N172 L174 I185 D186 L12 G13 F17 A33 K35 E139 N140 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=14nM remove_due_to_license_issue P11309 26459208 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5dh3 A 2.468 BS01 5BS A 1 L33 V41 E100 Y101 C102 G103 G105 D109 L153 L15 V23 E82 Y83 C84 G85 G87 D91 L135 D146 K148 G150 N151 D164 D173 T184 D128 K130 G132 N133 D146 D155 T166 2.7.11.1 0004672,0005524,0006468 ic50=38.1nM remove_due_to_license_issue Q13188 27535619 401 LTKQPEEVFDVLEKLGEGSYGSVFKAIHKESGQVVAIKQVPVESDLQEIIKEISIMQQCDSPYVVKYYGSYFKNTDLWIVMEYCGAGSVSDIIRLRNKTLIEDEIATILKSTLKGLEYLHFMRKIHRDIKAGNILLNTEGHAKLADFGVAGQLTDTMAKRNTVIGTPFWMAPEVIQEIGYNCVADIWSLGITSIEMAEGKPPYADIHPMRAIFMIPTNPPPTFRKPELWSDDFTDFVKKCLVKNPEQRATATQLLQHPFIKNAKPVSILRDLITEAMEIKAKRHEEQQR 5dh4 A 2.2 BS02 5AV A 1 Y514 H515 V668 I682 F686 Q716 F719 Y64 H65 V218 I232 F236 Q266 F269 3.1.4.17 0004114,0007165,0008081 Ki=58nM remove_due_to_license_issue Ki=58nM Q9Y233 26602277 803 QFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIR 5dh5 A 2.0 BS02 5AY A 1 Y514 H515 V668 I682 Y683 F686 M703 G715 Q716 F719 Y67 H68 V221 I235 Y236 F239 M256 G268 Q269 F272 3.1.4.17 0004114,0007165,0008081 Ki=0.23nM remove_due_to_license_issue Ki=0.32nM Q9Y233 26602277 803 GLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETWISSPSV 5dhg A 3.0 BS01 DGV A 1 W116 D130 Y131 M134 C200 I219 S223 Q280 V283 W70 D84 Y85 M88 C150 I169 S173 Q230 V233 ? 0001626,0004930,0004985,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41146 26526853 1201 PLGLKVTIVGLYLAVCVGGLLGNCLVMYVILRHTKMKTATNIYIFNLALADTLVLLTLPFQGTDILLGFWPFGNALCKTVIAIDYYNMFTSTFTLTAMSVDRYVAICHPIVRTSSKAQAVNVAIWALASVVGVPVAIMGSAQVEDEEIECLVEIPTPQDYWGPVFAICIFLFSFIVPVLVISVCYSLMIRRLRGVRLLSGSREKDRNLRRITRLVLVVVAVFVGCWTPVQVFVLAQGLGVQPSSETAVAILRFCTALGYVNSCLNPILYAFLDENFKACFR 5dhh A 3.004 BS01 DGW A 1 Q107 D110 D130 Y131 C200 V279 Q280 V283 Q63 D66 D86 Y87 C150 V229 Q230 V233 ? 0001626,0004930,0004985,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41146 26526853 1206 FLPLGLKVTIVGLYLAVCVGGLLGNCLVMYVILRHTKMKTATNIYIFNLALADTLVLLTLPFQGTDILLGFWPFGNALCKTVIAIDYYNMFTSTFTLTAMSVDRYVAICHPRTSSKAQAVNVAIWALASVVGVPVAIMGSAQVEDEEIECLVEIPTPQDYWGPVFAICIFLFSFIVPVLVISVCYSLMIRRLRGVRLLSGSREKDRNLRRITRLVLVVVAVFVGCWTPVQVFVLAQGLGVQPSSETAVAILRFCTALGYVNSCLNPILYAFLDENFKACFRK 5dhj A 2.457 BS01 5E5 A 1 F49 A65 K67 R122 L174 I185 D186 F17 A33 K35 R90 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=0.2uM remove_due_to_license_issue P11309 26459208 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5dhp A 2.27 BS01 5AQ A 1 N122 E123 Y163 S166 H223 N121 E122 Y162 S165 H222 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=140uM remove_due_to_license_issue Q8Y8D7 27783975 303 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhp A 2.27 BS02 5AQ C 1 G131 P132 D150 G130 P131 D149 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=140uM remove_due_to_license_issue Q8Y8D7 27783975 301 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhq A 2.29 BS01 5AK A 1 N122 E123 Y163 S166 H223 N121 E122 Y162 S165 H222 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=2uM remove_due_to_license_issue Q8Y8D7 27783975 302 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhq A 2.29 BS02 5AK C 1 G131 P132 R148 G149 D150 G130 P131 R147 G148 D149 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=2uM remove_due_to_license_issue Q8Y8D7 27783975 301 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhr A 2.31 BS01 5AJ A 1 N122 E123 Y163 S166 H223 N121 E122 Y162 S165 H222 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=23uM remove_due_to_license_issue Q8Y8D7 27783975 302 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhr A 2.31 BS02 5AJ C 1 G131 P132 R148 G149 D150 G130 P131 R147 G148 D149 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=23uM remove_due_to_license_issue Q8Y8D7 27783975 302 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhs A 2.62 BS01 5AG A 1 N122 E123 Y163 S166 H223 N121 E122 Y162 S165 H222 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 27783975 303 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhs A 2.62 BS02 5AG C 1 G131 P132 R148 G149 D150 A185 G130 P131 R147 G148 D149 A184 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 27783975 301 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dht A 2.59 BS01 5A9 A 1 N122 E123 A162 Y163 S166 N121 E122 A161 Y162 S165 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 27783975 303 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dht A 2.59 BS02 5A9 C 1 P132 G149 D150 A185 P131 G148 D149 A184 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 remove_due_to_license_issue Q8Y8D7 27783975 301 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhu A 2.33 BS01 5A8 A 1 E123 Y163 S166 H223 E122 Y162 S165 H222 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=0.5uM remove_due_to_license_issue Q8Y8D7 27783975 302 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhu A 2.33 BS02 5A8 C 1 G131 P132 R148 G149 D150 A185 G130 P131 R147 G148 D149 A184 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=0.5uM remove_due_to_license_issue Q8Y8D7 27783975 301 MKYMITSKGDEKSDLLRLNMIAGFGEYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVKLLAKGEYQKVSYPLLKTTVKYGIKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIED 5dhu C 2.33 BS01 5A8 A 1 G131 P132 R148 G149 D150 A185 G122 P123 R139 G140 D141 A176 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=0.5uM remove_due_to_license_issue Q8Y8D7 27783975 302 MKYMITSKGDEKSDLLRLNMIAGFGYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVEYQKVSYPLLKTTVKYGKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIE 5dhu C 2.33 BS02 5A8 C 1 E123 A162 Y163 S166 D222 H223 E114 A153 Y154 S157 D213 H214 2.7.1.23 0003951,0005524,0005737,0006741,0016301,0019674,0046872,0051287 Ki=0.5uM remove_due_to_license_issue Q8Y8D7 27783975 301 MKYMITSKGDEKSDLLRLNMIAGFGYDMEYDDVEPEIVISIGGDGTFLSAFHQYEERLDEIAFIGIHTGHLGFYADWRPAEADKLVEYQKVSYPLLKTTVKYGKKEATYLALNESTVKSSGGPFVVDVVINDIHFERFRGDGLCMSTPSGTTAYNKSLGGALMHPSIEAMQLTEMASINNRVYRTIGSPLVFPKHHVVSLQPVNDKDFQISVDHLSILHRDVQEIRYEVSAKKIHFARFRSFPFWRRVHDSFIE 5di1 A 2.9 BS01 5DF A 1 V31 Y36 V39 A52 K54 M105 C108 G111 D115 L160 V170 D171 V19 Y24 V27 A40 K42 M93 C96 G99 D103 L148 V158 D159 D153 K155 Q157 N158 D171 T191 D141 K143 Q145 N146 D159 T167 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=20nM O95819 26617966 4000 IDLSSLRDPAGIFELVEVVGNGTYGQVYKGRHVKTGQLAAIKVMDVTEDEEEEIKLEINMLKKYSHHRNIATYYGAFIKKSPPGHDDQLWLVMEFCGAGSITDLVKNTKGNTLKEDWIAYISREILRGLAHLHIHHVIHRDIKGQNVLLTENAEVKLVDFGNTFIGTPYWMAPEVIACDENPDATYDYRSDLWSCGITAIEMAEGAPPLCDMHPMRALFLIPRNPPPRLKSKKWSKKFFSFIEGCLVKNYMQRPSTEQLLKHPFIRDQPNERQVRIQLKDHIDRT 5dia A 1.964 BS01 5E6 A 1 L44 F49 A65 K67 L120 V126 D128 L174 I185 D186 L12 F17 A33 K35 L88 V94 D96 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue Ki=0.397nM P11309 26459208 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5diq F 2.1 BS01 5B9 F 1 K57 N59 R60 F206 F239 K347 I348 K50 N52 R53 F199 F232 K340 I341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 26381451 403 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRR 5dit A 2.25 BS01 5B8 A 1 Y57 G59 K60 F77 Q85 V86 I87 W90 Y113 I122 F130 Y45 G47 K48 F65 Q73 V74 I75 W78 Y101 I110 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=0.7uM remove_due_to_license_issue Ki=700nM Q13451 26419422 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 5diu A 1.3 BS01 5BG A 1 Y57 D68 F77 G84 Q85 V86 I87 W90 Y113 L128 Y45 D56 F65 G72 Q73 V74 I75 W78 Y101 L116 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=0.043uM remove_due_to_license_issue Ki=43nM Q13451 26954324 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 5div A 1.65 BS01 5BH A 1 Y57 D68 F77 Q85 V86 W90 Y113 K121 F130 Y45 D56 F65 Q73 V74 W78 Y101 K109 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=0.14uM remove_due_to_license_issue Ki=140nM Q13451 26954324 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKG 5dj5 A 2.4 BS01 GR2 A 1 F28 S97 V98 F136 V144 Y159 C191 F195 S220 H247 F26 S95 V96 F134 V142 Y157 C189 F193 S218 H245 S97 S95 3.1.-.- ic50=2.5uM remove_due_to_license_issue Q10QA5 26470846 800 GAKLLQILNVRVVGSGERVVVLSHGFGTDQSAWSRVLPYLTRDHRVVLYDLVCAGSVNPDHFDFRRYDNLDAYVDDLLAILDALRIPRCAFVGHSVSAMIGILASIRRPDLFAKLVLIGASPRFLNDSDYHGGFELEEIQQVFDAMGANYSAWATGYAPLAVGADVPAAVQEFSRTLFNMRPDISLHVCQTVFKTDLRGVLGMVRAPCVVVQTTRDVSVPASVAAYLKAHLGGRTTVEFLQTEGHLPHLSAPSLLAQVLRRALARY 5djp F 2.4 BS01 5BJ F 1 K57 N59 R60 F206 F239 L344 K347 K50 N52 R53 F199 F232 L337 K340 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 26381451 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5djr F 2.4 BS01 5BK F 1 Y10 K57 N59 T63 S205 F206 F239 L344 Y2 K49 N51 T55 S197 F198 F231 L336 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 26381451 403 VYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5djv F 2.3 BS01 5BL F 1 Y10 K57 N59 R60 F206 F239 Q242 L344 K347 I348 Y3 K50 N52 R53 F199 F232 Q235 L337 K340 I341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 26381451 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5dk4 A 1.9 BS02 5BX A 1 F5 S6 G7 Q9 H43 Y125 M129 D132 I133 V141 V143 Q147 F6 S7 G8 Q10 H44 Y126 M130 D133 I134 V142 V144 Q148 K111 K192 K195 K112 K193 K196 6.1.1.2 0000166,0004812,0004830,0005524,0005737,0005829,0006412,0006418,0006436 Ki=2nM remove_due_to_license_issue P00953 26555258 404 GMKTIFSGIQPSGVITIGNYIGALRQFVELQHEYNCYFCIVDQHAITVWQDPHELRQNIRRLAALYLAVGIDPTQATLFIQSEVPAHAQAAWMLQCIVYIGELERMTQFKEKSAGKEAVSAGLLTYPPLMAADILLYNTDIVPVGEDQKQHIELTRDLAERFNKRYGELFTIPEARIPKVGARIMSLVDPTKKMSKSDPNPKAYITLLDDAKTIEKKIKSAVTDSEGTIRYDKEAKPGISNLLNIYSTLSGQSIEELERQYEGKGYGVFKADLAQVVIETLRPIQERYHHWMESEELDRVLDEGAEKANRVASEMVRKMEQAMGLGRR 5dkr A 1.742 BS03 5CZ A 1 H42 F43 H43 F44 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 Kd=6uM remove_due_to_license_issue P02638 26727270 103 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFF 5dkr B 1.742 BS01 5CZ A 1 M0 V8 D12 M1 V9 D13 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 remove_due_to_license_issue P02638 26727270 103 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 5dl1 A 3.0 BS01 5C2 A 1 S98 I122 H123 Q124 P125 L126 L150 T169 S93 I117 H118 Q119 P120 L121 L145 T164 G69 S98 M99 H123 D172 G64 S93 M94 H118 D167 3.4.21.92 0004176,0004252,0005737,0006508,0006515,0008236,0009368,0051117 remove_due_to_license_issue Q2G036 26566002 201 LIPTVIETTERAYDIYSRLLKDRIIMLGSQIDDNVANSIVSQLLFLQAQDSEKDIYLYINSPGGSVTAGFAIYDTIQHIKPDVQTICIGMAASMGSFLLAAGAKGKRFALPNAEVMIHQPLGGAQGQATEIEIAANHILKTREKLNRILSERTGQSIEKIQKDTDRDNFLTAEEAKEYGLIDEVMVPE 5dl1 B 3.0 BS01 5C2 B 1 V71 S98 H123 Q124 P125 L126 Q132 R147 L150 L154 T169 V66 S93 H118 Q119 P120 L121 Q127 R142 L145 L149 T164 G69 S98 M99 H123 D172 G64 S93 M94 H118 D167 3.4.21.92 0004176,0004252,0005737,0006508,0006515,0008236,0009368,0051117 remove_due_to_license_issue Q2G036 26566002 201 LIPTVIETTERAYDIYSRLLKDRIIMLGSQIDDNVANSIVSQLLFLQAQDSEKDIYLYINSPGGSVTAGFAIYDTIQHIKPDVQTICIGMAASMGSFLLAAGAKGKRFALPNAEVMIHQPLGGAQGQATEIEIAANHILKTREKLNRILSERTGQSIEKIQKDTDRDNFLTAEEAKEYGLIDEVMVPE 5dl1 N 3.0 BS01 5C2 N 1 V71 S98 Q124 L126 Q132 H142 I143 T146 R147 L150 N151 L154 T169 V66 S93 Q119 L121 Q127 H137 I138 T141 R142 L145 N146 L149 T164 G69 S98 M99 H123 D172 G64 S93 M94 H118 D167 3.4.21.92 0004176,0004252,0005737,0006508,0006515,0008236,0009368,0051117 remove_due_to_license_issue Q2G036 26566002 201 LIPTVIETTERAYDIYSRLLKDRIIMLGSQIDDNVANSIVSQLLFLQAQDSEKDIYLYINSPGGSVTAGFAIYDTIQHIKPDVQTICIGMAASMGSFLLAAGAKGKRFALPNAEVMIHQPLGGAQGQATEIEIAANHILKTREKLNRILSERTGQSIEKIQKDTDRDNFLTAEEAKEYGLIDEVMVPE 5dls A 2.15 BS01 5CV A 1 G18 G21 A36 K38 E85 Y86 C87 G90 L137 D148 G13 G16 A31 K33 E72 Y73 C74 G77 L124 D135 D130 K132 E134 N135 D148 T170 D117 K119 E121 N122 D135 T157 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=4.4nM remove_due_to_license_issue O14757 26437226 301 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5dlv A 2.0 BS05 5D5 A 1 S81 Y82 K248 F249 H251 W254 W260 S26 Y27 K193 F194 H196 W199 W205 3.1.4.39 0001953,0003676,0004528,0004622,0004630,0005044,0005509,0005576,0005615,0006644,0006935,0006955,0008270,0008284,0009395,0010634,0016020,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0044849,0046872,0047391,0048714,0050731,0051894,0060326,0071276,0071392,1900026,1903165,2000394 ic50=10.4uM remove_due_to_license_issue Q64610 27075612 930 GSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIKVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDASFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLRLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRAKSINNSKYDPKTIIAALTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDIHLLVDRRWHVARKPLDVCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPDEVSRPNYPGIMYLQSEFDLGCTCDHTKGSTKERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWAYFQRVLVKKYASERNGVNVISGPIFDYNYDGLRDTEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCASSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5dlx A 1.9 BS01 5D2 A 1 F79 N140 D145 I146 L148 M149 F38 N99 D104 I105 L107 M108 ? Kd=2uM remove_due_to_license_issue O60885 27219844 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5dlz A 1.7 BS01 5D1 A 1 P82 K91 L92 N93 N140 I146 P41 K50 L51 N52 N99 I105 ? Kd=1.8uM remove_due_to_license_issue O60885 27219844 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5dno A 1.8 BS01 rna B 0 N336 R338 Y352 Y392 Y406 K436 T437 Y466 S470 C473 N477 R486 D487 R488 N12 R14 Y28 Y68 Y82 K112 T113 Y142 S146 C149 N153 R162 D163 R164 ? 0003723 remove_due_to_license_issue O74958 26673708 1 ~ 7 MSEHRERISMINPRVVLDENGISHRSRYFIMLCDNETAIAHAKKTSIWAVKKDSSKRISDAYKKASVYFIFVAQQTYNALGYAQVVSDLNSTELPFWSDSSHAGGVRIKWIKTCNLFSAEISEIVSHMDHGSEARDGMEMMYDEGSRLCTLINYAIMKRIGRDR 5dnu A 1.2 BS01 KKN A 1 F26 F124 L142 F157 I193 F194 A219 H246 F24 F122 L140 F155 I191 F192 A217 H244 F26 S95 L96 R216 G245 F24 S93 L94 R214 G243 ? Kd=77.6uM remove_due_to_license_issue A0A0M3PN85 27507097 301 RVEAARNVHIVGSGDTTVVLGHGFGTDQSVWKHLVPYLVDSYRVLLYDNMGAGSTNPEYFHFERYSTLQGYAHDLLVILHEFNIRSCIFVGHSLSAMTGAIASIIRPDLFQKIVMLSASPRFLNTADYLGGFEPADVEQLAGAIEANYKSWVSGFAPMVVGGDMDSVAVQEFSRTLFNMRPDIARSVFRTIFTSDLRDYLGRVTVPCHIIQSSRDMAVPVSVAGYIHNRVGGRSVVEVMNTEGHLPQLSAPEVAIPVLLRHIKNDID 5do4 H 1.859 BS01 rna A 0 H87 P88 R89 R98 R123 E169 R170 P171 D183 N184 R245 L246 K248 W249 H87 P88 R89 R98 R123 E167 R168 P169 D181 N182 R243 L244 K246 W247 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 27566147 1 ~ 25 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 5do4 L 1.859 BS01 rna A 0 G35 R36 G31 R32 3.4.21.5 0004252,0005576,0006508,0007596 remove_due_to_license_issue P00734 27566147 1 ~ 25 GEADCGLRPLFEKKSLEDKTERELLESYIDGR 5doh A 1.05 BS02 5DU A 1 Y7 H64 A65 Q92 H94 H96 H119 V121 F131 L198 T199 T200 Y5 H62 A63 Q90 H92 H94 H117 V119 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=32nM remove_due_to_license_issue P00918 28001003 304 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5doh B 1.05 BS02 5DU B 1 Y7 H64 A65 Q92 H94 H96 H119 V121 F131 L198 T199 T200 Y5 H62 A63 Q90 H92 H94 H117 V119 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=32nM remove_due_to_license_issue P00918 28001003 304 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5dp4 A 2.21 BS01 5E8 A 1 R39 H40 L127 S128 T142 K143 A144 C147 I162 G163 G164 R40 H41 L128 S129 T143 K144 A145 C148 I163 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dp5 A 2.03 BS01 5E9 A 1 R39 H40 E71 L127 S128 K130 T142 K143 A144 C147 H161 G163 G164 R40 H41 E72 L128 S129 K131 T143 K144 A145 C148 H162 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dp6 A 3.01 BS01 5EB A 1 H40 L127 S128 T142 K143 G145 C147 I162 G164 H38 L125 S126 T140 K141 G143 C145 I160 G162 H40 E71 G145 C147 H38 E69 G143 C145 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 SLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dp7 A 2.08 BS01 5EC A 1 R39 H40 L127 S128 T142 K143 A144 C147 G163 G164 R40 H41 L128 S129 T143 K144 A145 C148 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dp8 A 2.4 BS01 5ED A 1 H40 E71 N126 L127 S128 T142 K143 A144 G145 C147 I162 G163 G164 H41 E72 N127 L128 S129 T143 K144 A145 G146 C148 I163 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dp9 A 1.9 BS01 5EX A 1 H40 E71 L125 N126 L127 S128 T142 K143 A144 C147 H161 I162 G163 G164 H41 E72 L126 N127 L128 S129 T143 K144 A145 C148 H162 I163 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dpa A 2.06 BS01 5F2 A 1 R39 H40 E71 L127 S128 T142 K143 A144 G145 C147 H161 I162 G163 G164 R40 H41 E72 L128 S129 T143 K144 A145 G146 C148 H162 I163 G164 G165 H40 E71 G145 C147 H41 E72 G146 C148 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue A9XG43 26987809 201 MGPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNILDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFA 5dpx A 1.85 BS03 L3B A 1 H107 D109 F145 I149 H181 Y212 H246 H85 D87 F123 I127 H159 Y190 H224 H105 H107 D109 H110 H181 Y212 H246 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P52700 28505394 403 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 5dq8 A 2.305 BS01 FLF A 1 F233 S345 V347 K357 M379 C380 L383 I408 F12 S92 V94 K104 M126 C127 L130 I155 ? Kd=73uM remove_due_to_license_issue Q15562 26592798 501 GLGTARLQLVEFSAFVEPQRHLFVHISQLESVDVRQIYDKFPEKKGGLRELYDRGPPHAFFLVKFWADLNWGFYGVSSQYESLEHMTLTCSSKVCSFGKQVVEKVETERAQLEDGRFVYRLLRSPMCEYLVNFLHKLRQLPERYMMNSVLENFTILQVVTNRDTQELLLCTAYVFEVSTSERGAQHHIYRLVR 5dqc A 2.4651 BS01 5E7 A 1 G11 Q12 G13 L30 D32 G34 S35 Y71 T72 Q73 F108 I118 Y198 D228 G230 T232 N233 R235 G14 Q15 G16 L33 D35 G37 S38 Y74 T75 Q76 F111 I121 Y191 D221 G223 T225 N226 R228 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 Ki=45.6nM remove_due_to_license_issue P56817 27347366 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5dqe A 2.183 BS01 5E4 A 1 F233 V329 S345 V347 K357 M379 C380 L383 I408 Y426 F12 V76 S92 V94 K104 M126 C127 L130 I155 Y173 ? remove_due_to_license_issue Q15562 26592798 501 GLGTARLQLVEFSAFVEPQRHLFVHISQLESVDVRQIYDKFPEKKGGLRELYDRGPPHAFFLVKFWADLNWGFYGVSSQYESLEHMTLTCSSKVCSFGKQVVEKVETERAQLEDGRFVYRLLRSPMCEYLVNFLHKLRQLPERYMMNSVLENFTILQVVTNRDTQELLLCTAYVFEVSTSERGAQHHIYRLVR 5dqf A 2.15 BS02 CZE A 1 R208 A212 K350 E353 R205 A209 K347 E350 ? 0003677,0005504,0005576,0005615,0005737,0008289,0009267,0015643,0019825,0030170,0032991,0046872,0051902,0072732,1903981 Kd=253uM remove_due_to_license_issue P35747 26896718 613 KSEIAHRFNDLGEKHFKGLVLVAFSQYLQQCPFEDHVKLVNEVTEFAKKCAADESAENCDKSLHTLFGDKLCTVATLRATYGELADCCEKQEPERNECFLTHKDDHPNLPKLKPEPDAQCAAFQEDPDKFLGKYLYEVARRHPYFYGPELLFHAEEYKADFTECCPADDKLACLIPKLDALKERILLSSAKERLKCSSFQNFGERAVKAWSVARLSQKFPKADFAEVSKIVTDLTKVHKECCHGDLLECADDRADLAKYICEHQDSISGKLKACCDKPLLQKSHCIAEVKEDDLPSDLPALAADFAEDKEICKHYKDAKDVFLGTFLYEYSRRHPDYSVSLLLRIAKTYEATLEKCCAEADPPACYRTVFDQFTPLVEEPKSLVKKNCDLFEEVGEYDFQNALIVRYTKKAPQVSTPTLVEIGRTLGKVGSRCCKLPESERLPCSENHLALALNRLCVLHEKTPVSEKITKCCTDSLAERRPCFSALELDEGYVPKEFKAETFTFHADICTLPEDEKQIKKQSALAELVKHKPKATKEQLKTVLGNFSAFVAKCCGAEDKEACFAEEGPKLVASSQLALA 5drc A 2.18 BS03 5ER A 1 R339 E434 G459 L461 D462 M515 W541 M631 D633 R330 E423 G448 L450 D451 M504 W530 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R330 E423 D451 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 27738104 805 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAAVRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 5dri A 2.8 BS02 5EQ A 1 R339 E434 G459 L461 D462 M515 W541 M631 D633 R325 E419 G444 L446 D447 M500 W526 M616 D618 D271 E273 R339 E434 D462 D633 D267 E269 R325 E419 D447 D618 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 27738104 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDVGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 5dro A 2.01 BS02 ZH2 A 1 H58 E73 H74 T179 F180 A181 G198 H226 D230 H253 H57 E72 H73 T178 F179 A180 G197 H225 D229 H252 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue O67648 26912110 402 GLEKTVKEKLSFEGVGIHTGEYSKLIIHPEKEGTGIRFFKNGVYIPARHEFVVHTNHSTDLGFKGQRIKTVEHILSVLHLLEITNVTIEVIGNEIPILDGSGWEFYEAIRKNILNQNREIDYFVVEEPIIVEDEGRLIKAEPSDTLEVTYEGEFKNFLGRQKFTFVEGNEEEIVLARTFAFDWEIEHIKKVGLGKGGSLKNTLVLGKDKVYNPEGLRYENEPVRHKVFDLIGDLYLLGSPVKGKFYSFRGGHSLNVKLVKELAKKQK 5drq A 1.63 BS03 5EM A 1 E77 T190 F191 I197 R201 G209 S210 H237 D241 H264 E77 T190 F191 I197 R201 G209 S210 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue P47205 26912110 303 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISY 5drr A 1.59 BS03 5EN A 1 E77 T190 F191 I197 G209 S210 H237 D241 H264 E77 T190 F191 I197 G209 S210 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 remove_due_to_license_issue P47205 26912110 303 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRGRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISY 5drs A 1.1 BS02 5EF A 1 N62 N67 Q92 H94 H119 V121 F131 L198 T199 T200 N59 N64 Q89 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.1nM remove_due_to_license_issue P00918 28001003 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5drt A 2.69 BS01 5EG A 1 F131 P133 Y136 D161 G163 S164 G165 Q168 V169 F239 V240 N241 S268 S269 F115 P117 Y120 D145 G147 S148 G149 Q152 V153 F223 V224 N225 S252 S253 2.1.1.360 0031151,0051726 remove_due_to_license_issue IC50=4400nM Q8TEK3 27563395 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEKLFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSWTGKPVSYYLHTIDRTILENYFSSLKNP 5dry A 2.41 BS01 5EK A 1 F131 P133 Y136 S140 L143 M147 D161 G163 S164 Q168 V169 V240 N241 S268 S269 F121 P123 Y126 S130 L133 M137 D151 G153 S154 Q158 V159 V230 N231 S258 S259 2.1.1.360 0031151,0051726 ic50=20nM remove_due_to_license_issue IC50=20nM Q8TEK3 27563395 402 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKNP 5ds9 A 2.561 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5ds9 A 2.561 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5ds9 B 2.561 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5ds9 B 2.561 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5dsx A 2.41 BS01 5EW A 1 F131 S140 D161 S164 V169 V240 N241 F243 S268 S269 F118 S127 D148 S151 V156 V227 N228 F230 S255 S256 2.1.1.360 0031151,0051726 ic50=10nM remove_due_to_license_issue IC50=10.0nM Q8TEK3 27563395 1002 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTNTRPSTGLLRHILQQVYNHSVTDPEKLEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKNP 5dt2 A 2.3 BS01 5EV A 1 F131 S140 L143 V144 M147 D161 S164 V169 F239 V240 N241 F243 S268 S269 F114 S123 L126 V127 M130 D144 S147 V152 F222 V223 N224 F226 S251 S252 2.1.1.360 0031151,0051726 ic50=150nM remove_due_to_license_issue IC50=150nM Q8TEK3 27563395 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKN 5dtd A 2.642 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5dtd A 2.642 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5dtd B 2.642 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5dtd B 2.642 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5dtj A 2.71 BS01 5G8 A 1 Y124 Y341 Y127 Y338 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G124 G125 G157 S206 A207 G245 F294 F296 E331 H444 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 26350723 601 DPMEGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLL 5dtj A 2.71 BS02 5G8 A 2 Y72 Y124 S203 E285 W286 F295 F297 F338 N406 Y75 Y127 S206 E282 W283 F292 F294 F335 N403 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G124 G125 G157 S206 A207 G245 F294 F296 E331 H444 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 26350723 602 DPMEGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLL 5dtk A 1.6 BS01 5F3 A 1 S70 I102 T104 W105 Y117 V120 T209 G210 Y211 R250 S48 I80 T82 W83 Y95 V98 T187 G188 Y189 R228 S70 K73 S118 Y123 W157 Y211 S48 K51 S96 Y101 W135 Y189 3.5.2.6 0008658,0008800,0017001 Kd=50uM remove_due_to_license_issue Kd=50000nM, IC50=18000nM Q6XEC0 27165692 306 KEWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dtm A 2.2 BS01 5F4 A 1 F131 S140 L143 V144 F239 N241 F243 S268 S269 S311 Y312 F120 S129 L132 V133 F228 N230 F232 S257 S258 S298 Y299 2.1.1.360 0031151,0051726 Kd~50uM remove_due_to_license_issue Kd=50000nM, IC50=320000nM Q8TEK3 27563394 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSWTGKPVSYYLHTIDRTILENYFSSLKNP 5dtq A 2.61 BS01 5F6 A 1 F131 S140 L143 V144 F239 N241 F243 S268 S269 Y312 F121 S130 L133 V134 F229 N231 F233 S258 S259 Y300 2.1.1.360 0031151,0051726 remove_due_to_license_issue IC50=139000nM Q8TEK3 27563394 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSWTGKPVSYYLHTIDRTILENYFSSLKNP 5dtr A 2.34 BS01 5F7 A 1 F131 L143 F239 N241 V267 S268 S269 V310 Y312 F120 L132 F228 N230 V256 S257 S258 V297 Y299 2.1.1.360 0031151,0051726 ic50=39uM remove_due_to_license_issue IC50=39000nM Q8TEK3 27563394 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSWTGKPVSYYLHTIDRTILENYFSSLKNP 5dts C 1.94016 BS01 5F8 C 1 S70 S118 T209 R250 S46 S94 T185 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0008658,0008800,0017001 Kd=280uM remove_due_to_license_issue IC50=240000nM, Kd=280000nM Q6XEC0 27165692 301 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dtt C 2.10001 BS01 5F5 C 1 S70 I102 T209 G210 Y211 L247 R250 S47 I79 T186 G187 Y188 L224 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0008658,0008800,0017001 Kd=310uM remove_due_to_license_issue Kd=310000nM, IC50=250000nM Q6XEC0 27165692 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dtw A 2.439 BS01 5F9 A 1 E19 R20 R21 A23 A58 A60 D61 L62 H79 D83 G99 A100 Y126 W133 E20 R21 R22 A24 A59 A61 D62 L63 H80 D84 G100 A101 Y127 W134 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 Kd=3.5uM remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5dtw A 2.439 BS02 5F9 D 1 R17 R20 R18 R21 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 Kd=3.5uM remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5du4 A 1.702 BS01 5FF A 1 L75 I76 H79 D83 Q103 D131 W133 L76 I77 H80 D84 Q104 D132 W134 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 Kd=5.6uM remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5du6 A 2.61 BS01 G59 A 1 L75 D83 D131 W133 A208 K213 F216 L74 D82 D130 W132 A207 K212 F215 A60 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 P71 I75 A99 Q102 P121 T122 L127 L129 D130 P209 W219 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5du6 C 2.61 BS01 G59 C 1 L75 I76 H79 D83 Q107 D131 W133 A208 F216 L76 I77 H80 D84 Q108 D132 W134 A209 F217 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5du8 A 2.23 BS01 5FK A 1 L75 I76 H79 Q103 D131 W133 F216 L66 I67 H70 Q94 D122 W124 F207 A60 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 P63 I67 A91 Q94 P113 T114 L119 L121 D122 P201 W211 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 Kd=1.9uM remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5du8 C 2.23 BS01 5FK C 1 L75 I76 H79 D83 Q103 D131 W133 A208 F216 L76 I77 H80 D84 Q104 D132 W134 A209 F217 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 Kd=1.9uM remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5duc A 2.704 BS01 G51 A 1 L75 H79 D83 Q103 D131 W133 F216 L76 H80 D84 Q104 D132 W134 F217 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5duc C 2.704 BS01 G51 C 1 L75 I76 H79 D83 Q103 D131 W133 I205 K213 F216 L76 I77 H80 D84 Q104 D132 W134 I206 K214 F217 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A61 D66 P73 I77 A101 Q104 P123 T124 L129 L131 D132 P211 W221 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 remove_due_to_license_issue P9WNP1 27571973 301 HMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5duf A 1.5 BS01 G7A A 1 L75 I76 H79 D83 Q103 D131 W133 L77 I78 H81 D85 Q105 D133 W135 A60 D65 P72 I76 A100 Q103 P122 T123 L128 L130 D131 P210 W220 A62 D67 P74 I78 A102 Q105 P124 T125 L130 L132 D133 P212 W222 4.2.1.17 0003824,0004300,0005886,0006631,0006635,0009274,0016829,0016836 ic50=1.8uM remove_due_to_license_issue P9WNP1 27571973 301 SHMIGITQAEAVLTIELQRPERRNALNSQLVEELTQAIRKAGDGSARAIVLTGQGTAFCAGADLSGDAFAADYPDRLIELHKAMDASPMPVVGAINGPAIGAGLQLAMQCDLRVVAPDAFFQFPTSKYGLALDNWSIRRLSSLVGHGRARAMLLSAEKLTAEIALHTGMANRIGTLADAQAWAAEIARLAPLAIQHAKRVLNDDGAIEEAWPAHKELFDKAWGSQDVIEAQVARMEKRPPKFQGA 5dus A 1.432 BS01 APR A 1 D20 A21 A36 N38 G44 G46 I47 L124 S126 G128 I129 F130 N154 D21 A22 A37 N39 G45 G47 I48 L125 S127 G129 I130 F131 N155 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 Kd=2.95uM remove_due_to_license_issue K9N638 26740631 201 MPLSNFEHKVITECVTIVLGDAIQVAKCYGESVLVNAANTHLKHGGGIAGAINAASKGAVQKESDEYILAKGPLQVGDSVLLQGHSLAKNILHVVGPDARAKQDVSLLSKCYKAMNAYPLVVTPLVSAGIFGVKPAVSFDYLIREAKTRVLVVVNSQDVYKSLTI 5dv2 A 2.07 BS01 C5P A 1 H360 P365 D410 N412 N480 F485 H530 H177 P182 D215 N217 N274 F279 H324 3.1.13.4 0003824,0004535 ic50=1250uM remove_due_to_license_issue Q96LI5 27013054 601 LPPRPWITLKERDSASFTVMCYNVLCDKYATRQLYGYCPSWALNWEYRKKGIMEEIVNCDADIISLQEVETEQYFTLFLPALKERGYDGFFSPKSRAKIMSEQERKHVDGCAIFFKTEKFTLVQKHTVEFNQVAMANSDGSEAMLNRVMTKDNIGVAVVLEVHKELFKQLLIVANAHMHWDPEYSDVKLIQTMMFVSEVKNILEKASIPLVLCADLNSLPDSGVVEYLSNGGVADNHKDFKELRYNECLMNFSRITHGFQLKSAYENNLMPYTNYTFDFKGVIDYIFYSKTHMNVLGVLGPLDPQWLVENNITGCPHPHIPSDHFSLLTQLELHP 5dv4 A 1.8 BS01 NMY A 1 L206 E240 H360 M361 W363 P365 K371 D410 N412 L414 F484 I488 L35 E69 H178 M179 W181 P183 K189 D221 N223 L225 F288 I292 3.1.13.4 0003824,0004535 ic50=3370uM remove_due_to_license_issue Q96LI5 27013054 601 LPPRPWITLKERDQSASFTVMCYNVLCDKYATRQLYGYCPSWALNWEYRKKGIMEEIVNCDADIISLQEVETEQYFTLFLPALKERGYDGFFSPKSRAKIMSEQERKHVDGCAIFFKTEKFTLVQKHTVEFNQVAMANSDGSEAMLNRVMTKDNIGVAVVLEVHKELFKQLLIVANAHMHWDPEYSDVKLIQTMMFVSEVKNILEKASSRPNSIPLVLCADLNSLPDSGVVEYLSNGGVADNHKDFKELRYNECLMNFSCEGRITHGFQLKSAYENNLMPYTNYTFDFKGVIDYIFYSKTHMNVLGVLGPLDPQWLVENNITGCPHPHIPSDHFSLLTQLELHP 5dv7 C 3.5 BS01 rna A 0 Q411 S550 F555 K573 Q9 S97 F102 K120 ? 0003725 remove_due_to_license_issue Q9Z1X4 26712564 1 ~ 18 MNALMRLNQLKPGLQYKLISQTGPVHAPIFTMSVEVDGSNFEASGPSKKTAKLHVAVKVLQDMGLPILTKHGKNPVMELNEKRRGLKYELISETGGSHDKRFVMEVEVDGQKFQGAGSNKKVAKAYAALAALEKLFP 5dv7 C 3.5 BS02 rna B 0 N404 L406 M407 N527 V529 M530 N533 G549 S550 N2 L4 M5 N74 V76 M77 N80 G96 S97 ? 0003725 remove_due_to_license_issue Q9Z1X4 26712564 1 ~ 18 MNALMRLNQLKPGLQYKLISQTGPVHAPIFTMSVEVDGSNFEASGPSKKTAKLHVAVKVLQDMGLPILTKHGKNPVMELNEKRRGLKYELISETGGSHDKRFVMEVEVDGQKFQGAGSNKKVAKAYAALAALEKLFP 5dva A 2.50004 BS01 5FL A 1 S118 Y211 R250 S95 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0008658,0008800,0017001 Kd=280uM remove_due_to_license_issue Kd=280000nM, IC50=250000nM Q6XEC0 27165692 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5dw1 A 1.55 BS01 5GD A 1 W370 P371 F372 V376 L383 N429 H433 W26 P27 F28 V32 L39 N85 H89 ? ic50=0.08uM remove_due_to_license_issue P25440 27282480 500 KLSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 5dw2 A 1.12 BS01 5GD A 1 P82 F83 V87 L92 N140 D144 I146 P41 F42 V46 L51 N99 D103 I105 ? Kd=1.44uM remove_due_to_license_issue IC50=20nM O60885 27282480 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5dwa A 1.5 BS01 dna C 0 Y72 V89 R90 K140 S170 R174 K200 H206 Y72 V89 R90 K140 S170 R174 K200 H206 3.1.21.4 0004519,0009036,0009307 remove_due_to_license_issue Q9KHV6 28039325 -2 ~ 8 MRLDLDFGRGLVAHVMLDNVSEEQYQQISDYFVPLVNKPKLKSRDAIGQAFVMATEVCPDANPSDLWHHVLYRIYIREKIGTDPSQSWVRTSGEAFEVALVERYNPVLARHGIRLTALFKGQKGLALTRMGVADRVGSRKVDVMIEKQGGGRSPDAEGFGVVGGIHAKVSLAERVSDDIPASRIMMGEGLLSVLSTLDVKSFPPPHGDLVNRGELGTPDRPSDKRNYIEGHGDFSACFSYNLRTSPSNATTPSGRHIYVSGFSGQDDEFTDYLVAQLA 5dwa A 1.5 BS02 dna D 0 K42 R44 T82 D83 Q86 S87 V89 R90 K120 E173 F202 D223 K224 K42 R44 T82 D83 Q86 S87 V89 R90 K120 E173 F202 D223 K224 3.1.21.4 0004519,0009036,0009307 remove_due_to_license_issue Q9KHV6 28039325 -2 ~ 8 MRLDLDFGRGLVAHVMLDNVSEEQYQQISDYFVPLVNKPKLKSRDAIGQAFVMATEVCPDANPSDLWHHVLYRIYIREKIGTDPSQSWVRTSGEAFEVALVERYNPVLARHGIRLTALFKGQKGLALTRMGVADRVGSRKVDVMIEKQGGGRSPDAEGFGVVGGIHAKVSLAERVSDDIPASRIMMGEGLLSVLSTLDVKSFPPPHGDLVNRGELGTPDRPSDKRNYIEGHGDFSACFSYNLRTSPSNATTPSGRHIYVSGFSGQDDEFTDYLVAQLA 5dwa B 1.5 BS01 dna C 0 K42 T82 D83 Q86 S87 V89 R90 F202 K42 T82 D83 Q86 S87 V89 R90 F202 3.1.21.4 0004519,0009036,0009307 remove_due_to_license_issue Q9KHV6 28039325 -2 ~ 8 MRLDLDFGRGLVAHVMLDNVSEEQYQQISDYFVPLVNKPKLKSRDAIGQAFVMATEVCPDANPSDLWHHVLYRIYIREKIGTDPSQSWVRTSGEAFEVALVERYNPVLARHGIRLTALFKGQKGLALTRMGVADRVGSRKVDVMIEKQGGGRSPDAEGFGVVGGIHAKVSLAERVSDDIPASRIMMGEGLLSVLSTLDVKSFPPPHGDLVNRGELGTPDRPSDKRNYIEGHGDFSACFSYNLRTSPSNATTPSGRHIYVSGFSGQDDEFTDYLVAQLA 5dwa B 1.5 BS02 dna D 0 Y72 V89 R90 G93 R139 V169 S170 K200 Y72 V89 R90 G93 R139 V169 S170 K200 3.1.21.4 0004519,0009036,0009307 remove_due_to_license_issue Q9KHV6 28039325 -2 ~ 8 MRLDLDFGRGLVAHVMLDNVSEEQYQQISDYFVPLVNKPKLKSRDAIGQAFVMATEVCPDANPSDLWHHVLYRIYIREKIGTDPSQSWVRTSGEAFEVALVERYNPVLARHGIRLTALFKGQKGLALTRMGVADRVGSRKVDVMIEKQGGGRSPDAEGFGVVGGIHAKVSLAERVSDDIPASRIMMGEGLLSVLSTLDVKSFPPPHGDLVNRGELGTPDRPSDKRNYIEGHGDFSACFSYNLRTSPSNATTPSGRHIYVSGFSGQDDEFTDYLVAQLA 5dwr A 2.0 BS01 5H7 A 1 L44 G45 F49 A65 K67 I104 R122 V126 D128 E171 L174 I185 D186 L12 G13 F17 A33 K35 I72 R90 V94 D96 E139 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki<0.001uM remove_due_to_license_issue IC50=6.0nM, Ki=0.006000nM P11309 26505898 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 5dx4 A 2.3 BS01 E0C A 1 W81 F83 L92 L94 N140 M149 W40 F42 L51 L53 N99 M108 ? Kd=0.137uM remove_due_to_license_issue IC50=410nM, Kd=137nM O60885 26731490 201 GSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5dxh A 3.0 BS01 5H2 A 1 M772 I800 Y836 I848 V851 S854 M922 I932 M725 I753 Y789 I801 V804 S807 M870 I880 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue Ki=1.000000nM P42336 26741947 1101 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSLRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKALQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHRVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAKMDWIFHTI 5dxt A 2.25 BS01 5H5 A 1 S774 W780 I800 Y836 I848 V851 S854 Q859 M922 F930 I932 D933 S621 W627 I647 Y683 I695 V698 S701 Q706 M759 F767 I769 D770 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 Ki=0.2nM remove_due_to_license_issue Ki=0.350nM P42336 26741947 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVDKQKYTLKINHDCVPEQVIAEAIRKKTRSMGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRTSTKSLWVINSALRIKILCATYVNVNIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREAGFSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHRERVPFVLTQDFLIVISKGAECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGW 5dxu A 2.64 BS01 5H5 A 1 M752 W760 I825 V828 D832 M900 F908 D911 M666 W674 I736 V739 D743 M799 F807 D810 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue Ki=6.94nM O00329 26741947 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPLPNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKAVEQPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEKDCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHEEEQLQLREILERYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLNDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKV 5dy5 A 1.95 BS02 5GR A 1 I93 F96 R97 F119 F131 A135 L138 Y139 P140 F143 D170 H187 F190 I232 V233 F234 F235 I41 F44 R45 F67 F79 A83 L86 Y87 P88 F91 D118 H135 F138 I180 V181 F182 F183 P94 D95 F96 R97 N168 D170 H187 P42 D43 F44 R45 N116 D118 H135 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=0.163uM remove_due_to_license_issue IC50=160nM Q8IXJ6 26748890 402 GHMERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPSTGLYDNLEKYHLPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGQSGMIMGLGGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5dy7 A 1.69 BS01 5GT A 1 V657 P658 E661 V662 F714 V31 P32 E35 V36 F88 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5dya A 1.65 BS01 5GV A 1 I652 F653 E661 C704 F714 I25 F26 E34 C77 F87 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 802 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5dyo A 2.36 BS01 FLU A 1 H35 R99 H34 R98 remove_due_to_license_issue 26756394 301 VQLQQSGPELVKPGASVKMSCKASGYTFSTSVIHWVKQKPGQGLEWIGYIFPYNYGTQYNEEFRGKATLTSDKSSNTAYMELSSLTSEDSAVYYCASRSGPWGQGTTLTVSSAKTTAPSVYPLAPVSSVTLGCLVKGYFPEPVTLTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVTSSTWPSQSITCNVAHPASSTKVDKKIEP 5dyo B 2.36 BS01 FLU A 1 Y37 N39 W94 G96 Q101 Y37 N39 W94 G96 Q101 remove_due_to_license_issue 26756394 301 DVVMTQTPLTLSITIGQPVSISCKSSQSLFASDGRTYLNWLLQRPGQSPERLIYLVSNLDSGVLDRFTGSGSGTDFTLKISRVEAEDLGVYYCWQGTHFPQTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 5dyo B 2.36 BS02 FLU H 1 S32 D33 S32 D33 remove_due_to_license_issue 26756394 901 DVVMTQTPLTLSITIGQPVSISCKSSQSLFASDGRTYLNWLLQRPGQSPERLIYLVSNLDSGVLDRFTGSGSGTDFTLKISRVEAEDLGVYYCWQGTHFPQTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNE 5dyt A 2.55 BS03 5HB A 1 G116 G117 Q119 S198 W231 S287 F329 F398 H438 G114 G115 Q117 S196 W229 S285 F327 F396 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0004104 remove_due_to_license_issue P06276 28000737 616 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5dyw A 2.5 BS03 5HF A 1 N68 G116 G117 Q119 T120 S198 W231 S287 F329 F398 W430 N66 G114 G115 Q117 T118 S196 W229 S285 F327 F396 W428 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0004104 ic50=4.9nM remove_due_to_license_issue IC50=4.9nM P06276 28000737 601 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5dyy A 2.65 BS02 5HH A 1 G116 G117 Q119 L286 S287 Y332 G114 G115 Q117 L284 S285 Y330 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0004104 remove_due_to_license_issue P06276 28000737 605 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5e08 H 2.38 BS01 rna N 0 Y53 Y55 Y56 R99 Y100 Y101 S102 S103 G104 Y107 Y108 R109 S111 G113 D115 Y52 Y54 Y55 R98 Y99 Y100 S101 S102 G103 Y106 Y107 R108 S110 G112 D114 remove_due_to_license_issue 27593161 1 ~ 12 EVQLVESGGGLVQPGGSLRLSCAASGFSISSSYIHWVRQAPGKGLEWVAYIYPYYGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARYYSSGGSYYRYSRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTH 5e08 L 2.38 BS01 rna N 0 Y50 S51 S54 Y56 Y50 S51 S54 Y56 remove_due_to_license_issue 27593161 1 ~ 12 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSYSYPYTFGQGTKVEIKRTVAAPSVFIFPPSDSQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 5e0g A 1.2 BS01 5LG A 1 H30 I109 Q110 G133 T134 I135 P136 C139 A158 A159 A160 H32 I111 Q112 G133 T134 I135 P136 C139 A158 A159 A160 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 27235842 202 HHAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 5e0h A 1.95 BS01 5LH A 1 H30 I109 Q110 T134 I135 P136 C139 H157 A158 A159 A160 H31 I110 Q111 T127 I128 P129 C132 H150 A151 A152 A153 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 27235842 201 HAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 5e0j A 1.2 BS01 5LJ A 1 H30 E54 M107 I109 Q110 R112 L132 C139 A158 A159 A160 V168 H31 E55 M108 I110 Q111 R113 L133 C140 A159 A160 A161 V169 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 27235842 204 HAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGMDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 5e13 A 1.34 BS01 5J9 A 1 M0 K1 W7 R68 N70 A110 V128 H129 M1 K2 W8 R69 N71 A111 V129 H130 H15 K38 H16 K39 4.6.1.18 0003676 Ki=57.8uM remove_due_to_license_issue P10153 26551065 201 MKPPQFTWAQWFETQHINMTSQQCTNAMQVINNYQRRCKNQNTFLLTTFANVVNVCGNPNMTCPSNKTRKNCHHSGSQVPLIHCNLTTPSPQNISNCRYAQTPANMFYIVACDNRDQRRDPPQYPVVPVHLDRII 5e1e A 2.3 BS01 5JG A 1 L881 A906 M956 F958 L959 P960 G962 E966 R1007 N1008 L1010 L17 A42 M83 F85 L86 P87 G89 E93 R134 N135 L137 D1003 A1005 R1007 N1008 D1021 D1040 D130 A132 R134 N135 D148 D167 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.022uM remove_due_to_license_issue IC50=39nM P23458 26614408 1202 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKNHIADLKKEIEILRNLYHENIVKYKGICTNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 5e1s A 2.264 BS01 5JA A 1 L1002 G1003 V1010 A1028 M1079 H1081 G1082 M1139 L20 G21 V28 A46 M97 H99 G100 M157 N1132 R1136 N1137 D1150 N150 R154 N155 D168 2.7.10.1 0004672,0004714,0005524,0006468,0007169,0016020 Kd=12nM remove_due_to_license_issue P06213 26438154 1301 VYVPDEWEVSREKITLLRELGQGSFGMVYEGNARDIIKGEAETRVAVKTVNESASLRERIEFLNEASVMKGFTCHHVVRLLGVVSKGQPTLVVMELMAHGDLKSYLRSLRPEAENNPGRPPPTLQEMIQMAAEIADGMAYLNAKKFVHRNLAARNCMVAHDFTVKIGDFGMLPVRWMAPESLKDGVFTTSSDMWSFGVVLWEITSLAEQPYQGLSNEQVLKFVMDGGYLDQPDNCPERVTDLMRMCWQFNPKMRPTFLEIVNLLKDDLHPSFPEVSFFHSEENK 5e28 A 1.3 BS02 BC5 A 1 H94 H96 F131 L198 T199 T200 H91 H93 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=12.3nM remove_due_to_license_issue Ki=12nM P00918 26741028 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5e2k A 1.4 BS02 BX4 A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=9.3nM remove_due_to_license_issue Ki=9.3nM P00918 26741028 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5e2k A 1.4 BS03 BX4 A 2 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=9.3nM remove_due_to_license_issue Ki=9.3nM P00918 26741028 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5e2l A 2.5 BS02 DPN A 1 F91 R171 A174 N175 F91 R171 A174 N175 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=93uM remove_due_to_license_issue O53512 27128682 507 MNWTVDIPIDQLPSLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e2l B 2.5 BS01 DPN A 1 V55 Y173 V51 Y169 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=93uM remove_due_to_license_issue O53512 27128682 507 MNWTVDIPIDLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e2l B 2.5 BS03 DPN B 1 F91 R171 A174 N175 F87 R167 A170 N171 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=93uM remove_due_to_license_issue O53512 27128682 509 MNWTVDIPIDLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e2m A 1.41 BS02 V14 A 1 H64 H67 H94 H96 H119 L198 T199 H200 P201 H60 H63 H90 H92 H115 L194 T195 H196 P197 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=59nM remove_due_to_license_issue Kd=1100nM P00915 28001003 302 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 5e2n A 1.53 BS02 V14 A 1 W7 S64 H66 S67 N69 Q94 H96 H98 V123 F133 L200 T201 V202 W2 S59 H61 S62 N64 Q89 H91 H93 V118 F128 L195 T196 V197 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=0.29nM remove_due_to_license_issue Kd=42nM Q8N1Q1 28001003 307 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 5e2o A 2.08 BS01 5JM A 1 L41 C42 H57 Y143 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 L28 C29 H44 Y134 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=2nM remove_due_to_license_issue Ki=2.0nM P03951 26704266 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5e2p A 2.11 BS01 7P0 A 1 R39 H40 L41 H57 Y143 I151 D189 A190 C191 K192 G193 S195 T213 S214 W215 G218 C219 G226 V227 Y228 R26 H27 L28 H44 Y134 I141 D182 A183 C184 K185 G186 S188 T206 S207 W208 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=1.6nM remove_due_to_license_issue Ki=1.6nM P03951 26704266 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5e2r A 1.6 BS02 520 A 1 H94 H119 F131 V135 L198 T199 T200 H95 H120 F131 V135 L198 T199 T200 H64 H94 H96 E106 H119 T199 H65 H95 H97 E107 H120 T199 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=86.2nM remove_due_to_license_issue Ki=86nM P00918 26497049 302 GMSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5e2s A 1.5 BS02 5CX A 1 Q92 H94 H119 V121 F131 L198 T199 T200 Q90 H92 H117 V119 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.98nM remove_due_to_license_issue Ki=0.980000nM P00918 26741028 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5e3d A 1.71 BS01 5JL A 1 V657 N708 F714 V30 N81 F87 ? Kd=95uM remove_due_to_license_issue P55201 27167503 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5e3g A 1.65 BS01 5JQ A 1 V657 Y707 N708 F714 V30 Y80 N81 F87 ? remove_due_to_license_issue Kd=>50000nM P55201 27167503 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5e3h A 2.7 BS01 rna B 0 K379 Q380 H381 Q507 Q511 N720 H830 F853 I875 V886 K888 W908 K139 Q140 H141 Q258 Q262 N456 H562 F585 I605 V616 K618 W628 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 21947008 1 ~ 12 FKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLEFGTQKYEQWIVTVQKACMVFDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGTGMTLPAQKCILDAFKDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARCSHDWGIHVKYKTFEIPVIKIESFTLYSKWKDFHFEKIPFDPAE 5e3h A 2.7 BS02 rna C 0 N298 I300 S325 G326 T347 Q349 E510 K635 T636 R637 G663 R664 T697 S698 V699 F853 S906 N58 I60 S85 G86 T107 Q109 E261 K379 T380 R381 G407 R408 T433 S434 V435 F585 S626 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 21947008 3 ~ 14 FKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLEFGTQKYEQWIVTVQKACMVFDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGTGMTLPAQKCILDAFKDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARCSHDWGIHVKYKTFEIPVIKIESFTLYSKWKDFHFEKIPFDPAE 5e3l A 2.66 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3l A 2.66 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3l B 2.66 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3l B 2.66 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3o A 2.78 BS01 dna C 0 N84 T87 K90 N77 T80 K83 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3o A 2.78 BS02 dna D 0 N73 Q74 T75 R85 R89 N66 Q67 T68 R78 R82 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 SDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3o B 2.78 BS01 dna C 0 N73 Q74 T75 R85 R89 N73 Q74 T75 R85 R89 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e3o B 2.78 BS02 dna D 0 N84 T87 K90 N84 T87 K90 ? 0000786,0000976,0001046,0001216,0001217,0003677,0003700,0005515,0005737,0005829,0006351,0006355,0009295,0009314,0031421,0032359,0032993,0042803,0043565,0044374,0045892,0045893,0045911,0051276 remove_due_to_license_issue P0A6R3 26959646 1 ~ 27 MFEQRVNSDVLTVSTVNSQDQVTQKPLRDSVKQALKNYFAQLNGQDVNDLYELVLAEVEQPLLDMVMQYTRGNQTRAALMMGINRGTLRKKLKKYGMN 5e5g A 1.95 BS02 DTR A 1 F91 R171 N175 F87 R167 N171 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=700uM remove_due_to_license_issue O53512 27128682 503 MNWTVDIPIDLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e5g A 1.95 BS03 DTR A 2 K123 A192 N237 T240 K119 A188 N233 T236 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=700uM remove_due_to_license_issue O53512 27128682 504 MNWTVDIPIDLPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e5g B 1.95 BS01 DTR A 1 W3 V55 Y173 A174 W3 V49 Y167 A168 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=700uM remove_due_to_license_issue O53512 27128682 503 MNWTVDIPIPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e5g B 1.95 BS03 DTR B 1 F91 R171 A174 N175 F85 R165 A168 N169 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=700uM remove_due_to_license_issue O53512 27128682 506 MNWTVDIPIPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e5g B 1.95 BS04 DTR B 2 L107 K123 A192 L194 N237 L101 K117 A186 L188 N231 2.5.1.54 0003849,0005515,0005829,0005886,0008652,0009073,0009274,0009423,0016740,0030145,0046872,0051260 Kd=700uM remove_due_to_license_issue O53512 27128682 507 MNWTVDIPIPPLPTDLRTRLDAALAKPAAQQPTWPADQALAMRTVLESVPPVTVPSEIVRLQEQLAQVAKGEAFLLQGGDCAETFMDNTEPHIRGNVRALLQMAVVLTYGASMPVVKVARIAGQYAKPRSADIDALGLRSYRGDMINGFAPDAAAREHDPSRLVRAYANASAAMNLVRALTSSGLASLHLVHDWNREFVRTSPAGARYEALATEIDRGLRFMSACGVADRNLQTAEIYASHEALVLDYERAMLRLSDGDDGEPQLFDLSAHTVWIGERTRQIDGAHIAFAQVIANPVGVKLGPNMTPELAVEYVERLDPHNKPGRLTLVSRMGNHKVRDLLPPIVEKVQATGHQVIWQCDPMHGNTHESSTGFKTRHFDRIVDEVQGFFEVHRALGTHPGGIHVEITGENVTECLGGAQDISETDLAGRYETACDPRLNTQQSLELAFLVAEMLRD 5e5o A 2.36 BS01 dna B 0 E20 M24 R26 R28 T46 V47 D48 R79 N139 S191 I192 K193 Q197 F225 R231 T240 N241 F242 H281 L282 E14 M18 R20 R22 T40 V41 D42 R73 N133 S185 I186 K187 Q191 F219 R225 T234 N235 F236 H275 L276 G178 D179 G172 D173 ? 0004519 remove_due_to_license_issue F7WD42 26705195 1 ~ 25 KLNPWAVVGFIDAEGSFMVRVRKNSKYKTGWLVVAIFSVTVDKKDLFLLESLKTFFGGLGSIKKSGNSTFSYRIESSEQLTKIILPFFDKYSLITEKLGDYLLFKKVLELMGTKEHLTQRGLEKIVSLKASINKGLSEELQAAFPQCVPTPRPEINNKNIPDPFWLAGFVSGDGSFKSILKKSESIKVGFQSILVFQITQHARDVKLMESLISYLGCGFIEKDSRGPWLYYTVTNFSDIQGKIIPFFHQYKIIGSKYGDYMDWCKIALIMQNKNHLTPEGLNEIRALKGGMNKG 5e5o A 2.36 BS02 dna C 0 K32 Y33 K34 K69 S71 E81 S82 S83 H122 D179 S181 K183 L186 K187 T205 H207 W234 N298 K26 Y27 K28 K63 S65 E75 S76 S77 H116 D173 S175 K177 L180 K181 T199 H201 W228 N292 G178 D179 G172 D173 ? 0004519 remove_due_to_license_issue F7WD42 26705195 1 ~ 25 KLNPWAVVGFIDAEGSFMVRVRKNSKYKTGWLVVAIFSVTVDKKDLFLLESLKTFFGGLGSIKKSGNSTFSYRIESSEQLTKIILPFFDKYSLITEKLGDYLLFKKVLELMGTKEHLTQRGLEKIVSLKASINKGLSEELQAAFPQCVPTPRPEINNKNIPDPFWLAGFVSGDGSFKSILKKSESIKVGFQSILVFQITQHARDVKLMESLISYLGCGFIEKDSRGPWLYYTVTNFSDIQGKIIPFFHQYKIIGSKYGDYMDWCKIALIMQNKNHLTPEGLNEIRALKGGMNKG 5e69 A 1.85 BS01 dna C 0 C431 H432 Y433 K442 K446 C14 H15 Y16 K25 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 18 ~ 33 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e69 A 1.85 BS02 dna D 0 S440 F444 R447 R470 K471 R477 S23 F27 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 34 ~ 49 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e69 B 1.85 BS01 dna C 0 S440 R447 R470 K471 R477 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 18 ~ 33 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e6a A 2.197 BS01 dna C 0 C431 H432 Y433 K442 K446 C14 H15 Y16 K25 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 1 ~ 16 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e6a A 2.197 BS02 dna D 0 S440 F444 R447 R470 K471 R477 S23 F27 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 1 ~ 16 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e6a B 2.197 BS01 dna C 0 S440 R447 R470 K471 R477 S23 R30 R53 K54 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 1 ~ 16 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e6c A 2.2 BS01 dna C 0 C431 H432 Y433 K442 K446 R491 C14 H15 Y16 K25 K29 R74 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 1 ~ 16 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKK 5e6c A 2.2 BS02 dna D 0 G439 S440 R447 R470 R477 G22 S23 R30 R53 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 1 ~ 16 PKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKK 5e6c B 2.2 BS01 dna C 0 S440 R470 S22 R52 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 29626214 1 ~ 16 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5e73 A 1.71 BS01 UO1 A 1 W1887 P1888 V1893 V1898 I1950 W32 P33 V38 V43 I95 ? Kd=23uM remove_due_to_license_issue Kd=23000nM Q9UIF8 26982797 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5e74 A 1.783 BS01 5KH A 1 W1887 P1888 V1893 N1894 V1898 W32 P33 V38 N39 V43 ? Kd=39uM remove_due_to_license_issue Kd=39000nM, IC50=27000nM Q9UIF8 26982797 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5e7n A 1.21 BS01 5KR A 1 I33 R41 R43 S55 M57 I83 N85 L87 I95 I36 R44 R46 S58 M60 I86 N88 L90 I98 ? 0003677,0005634,0006260 Kd=30uM remove_due_to_license_issue P27694 26748787 201 GSHMVGQLSRGAIAAIMQKGDTNIKPILQVINIRPITTGNSPPRYRLLMSDGLNTLSSFMLATQLNPLVEEEQLSSNCVCQIHRFIVNTLKDGRRVVILMELEVLKSAEAVGVKIGNPVPYNE 5e7r A 2.11 BS01 5KW A 1 V42 A61 M104 Y106 A107 G110 L163 C174 D175 F176 V14 A30 M58 Y60 A61 G64 L117 C128 D129 F130 D156 K158 P160 N161 I173 D175 D110 K112 P114 N115 I127 D129 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 28011204 601 HMIDYKEIEVEEVVGRGVVCKAKWRAKDVAIKQILSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5e80 B 2.6 BS01 5KP B 1 M20 L54 R61 A111 I129 T131 L147 Y149 M19 L53 R60 A110 I128 T130 L146 Y148 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 remove_due_to_license_issue O43924 27094677 201 SAKDERAREILRGFKLNWMNLRDAATGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAAPESQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5e88 A 1.6 BS01 5KT A 1 R144 A146 H158 R162 W181 E184 R186 R31 A33 H45 R49 W68 E71 R73 ? 0030246 Kd=0.065uM remove_due_to_license_issue P17931 27356186 302 LIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5e89 A 1.5 BS01 TD2 A 1 R144 A146 H158 R162 E165 W181 E184 R186 R31 A33 H45 R49 E52 W68 E71 R73 ? 0030246 Kd=0.014uM remove_due_to_license_issue P17931 27356186 302 LIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5e8a A 1.5 BS01 5KS A 1 R144 A146 H158 N160 R162 W181 E184 R186 S237 G238 R31 A33 H45 N47 R49 W68 E71 R73 S124 G125 ? 0030246 Kd=0.034uM remove_due_to_license_issue P17931 27356186 302 LIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5e8i A 3.45 BS01 dna B 0 Y332 R337 R340 Y341 Y343 K350 R355 Y356 Y54 R59 R62 Y63 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 2 ~ 11 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i A 3.45 BS02 dna C 0 Q282 L283 W321 K325 K327 M330 K334 Y341 Y342 Q4 L5 W43 K47 K49 M52 K56 Y63 Y64 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 14 ~ 23 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i D 3.45 BS01 dna C 0 S294 T301 E303 S16 T23 E25 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 14 ~ 23 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i D 3.45 BS02 dna E 0 Y332 R337 R340 Y343 K350 R355 Y356 Y54 R59 R62 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 2 ~ 11 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i D 3.45 BS03 dna F 0 Q282 W321 K325 K327 M330 K334 R337 Y341 Y342 Q4 W43 K47 K49 M52 K56 R59 Y63 Y64 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 14 ~ 23 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i G 3.45 BS01 dna H 0 Y332 R337 R340 Y343 K350 R355 Y356 Y54 R59 R62 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 2 ~ 11 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i G 3.45 BS02 dna I 0 Q282 W321 K325 K327 N329 M330 K334 Y341 Y342 Q4 W43 K47 K49 N51 M52 K56 Y63 Y64 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 14 ~ 23 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i J 3.45 BS01 dna K 0 Y332 R337 R340 Y343 K350 R355 Y356 Y54 R59 R62 Y65 K72 R77 Y78 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 2 ~ 11 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8i J 3.45 BS02 dna L 0 Q282 W321 K325 K327 M330 K334 Y341 Y342 K345 Q4 W43 K47 K49 M52 K56 Y63 Y64 K67 ? 0003700,0006355,0006357,0043565 remove_due_to_license_issue Q01543 26618620 14 ~ 23 GQIQLWQFLLELLSDSANASCITWEGTNGEFKMTDPDEVARRWGERKSKPNMNYDKLSRALRYYYDKNIMTKVHGKRYAYKFDFHGIAQALQP 5e8r A 2.55 BS02 5L6 A 1 Y51 V56 E59 M60 E155 M157 Y159 H163 E164 H317 Y10 V15 E18 M19 E114 M116 Y118 H122 E123 H274 D63 E155 E164 H317 D22 E114 E123 H274 2.1.1.319 0000122,0003682,0005515,0005634,0005654,0005730,0006281,0006284,0006325,0006338,0006355,0008168,0008469,0010821,0016274,0018216,0032259,0035241,0035242,0035642,0036211,0042054,0042393,0044020,0045652,0045892,0062122,0070611,0070612,0090398,0140592,0140759,0140903,0140938,0140984,1901796,1990259,2000059 remove_due_to_license_issue IC50=4.0nM, Ki=0.8nM, Kd=6nM Q96LA8 26598975 1002 ERDQLYYECYSDVSVHEEMIADRVRTDAYRLGILRNWAALRGKTVLDVGAGTGILSIFCAQAGARRVYAVEASAIWQQAREVVRFNGLEDRVHVLPGPVETVELPEQVDAIVSEWMGYGLLHESMLSSVLHARTKWLKEGGLLLPASAELFIVPISDQMLEWRLGFWSQVKQHYGVDMSCLEGFATRCLMGHSEIVVQGLSGEDVLARPQRFAQLELSRAGLEQELEAGVGGRFRCSCYGSAPMHGFAIWFQVTFPGGEKPLVLSTSPFHPATHWKQALLYLNEPVQVEQDTDVSGEITLLPSRDNPRRLRVLLRYKVGDQEEKTKDFAMED 5e8w A 1.86 BS01 STU A 1 I211 K213 V219 A230 L260 Y282 H283 G286 K337 L340 D351 I13 K15 V21 A32 L62 Y84 H85 G88 K139 L142 D153 D333 K335 N338 D351 T375 D135 K137 N140 D153 T177 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue P36897 27139629 601 MTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEGI 5e8z A 1.51 BS01 5L4 A 1 I211 G214 A230 K232 L260 Y282 H283 G286 L340 D351 I15 G18 A34 K36 L64 Y86 H87 G90 L144 D155 D333 K335 N338 D351 T375 D137 K139 N142 D155 T179 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue P36897 27139629 601 GHMTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQE 5e90 A 2.05 BS01 5L4 A 1 V211 G214 A230 K232 L260 F282 H283 G286 N287 L340 D351 V15 G18 A34 K36 L64 F86 H87 G90 N91 L144 D155 D333 K335 K337 N338 D351 D366 T375 D137 K139 K141 N142 D155 D170 T179 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue P36897 27139629 601 GHMTIARDIVLQESVGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIFQTVMLRHENILGFIAADNKDNGTWTQLWLVTDFHEHGNLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCICDFGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQE 5e91 A 2.42 BS01 5L4 A 1 V250 V258 A275 K277 L305 F327 H328 G331 N332 L386 C396 D397 V11 V19 A29 K31 L59 F81 H82 G85 N86 L140 C150 D151 D379 K381 N384 D397 D411 T421 D133 K135 N138 D151 D165 T175 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue P37173 27139629 601 ELLPIELDTLVGKGRFAEVYKAKLKETVAVKIFPYEEYASWKTEKDIFSDINLKHENILQFLTAEERKTELGKQYWLITAFHAKGNLQEYLTRHVISWEDLRKLGSSLARGIAHLHSDHTPCGRPKMPIVHRDLKSSNILVKNDLTCCLCDFGLSLRLDPTLSVDDLANSGQVGTARYMAPEVLASAMNLENVESFKQTDVYSMALVLWEMTSRCNAVGEVKDYEPPFGSKVREHPCVASMADNVLADAGRPEIPSFWLNHQGIQMVCETLTECWDHDPEARLTAQCVAERFSELEH 5ea3 F 2.75 BS01 5NK F 1 F140 D486 F488 F66 D399 F401 ? 0019064 remove_due_to_license_issue P03420 26641933 608 NITEEFYQSTCSAVSKGYLSALRTGWYTSVITIELSNIKKVKLIKQELDKYKNAVTELQLLMFLGFLLGVGSAIASGVAVCKVLHLEGEVNKIKSALLSTNKAVVSLSNGVSVLTFKVLDLKNYIDKQLLETVIEFQQKNNRLLEITREFSVNAGVTTPVSTYMLTNSELLSLINDMPITNDQKKLMSNNVQIVRQQSYSIMCIIKEEVLAYVVQLPLYGVIDTPCWKLHTSPLCTTNTKEGSNICLTRTDRGWYCDNAGSVSFFPQAETCKVQSNRVFCDTMNSLTLPSEVNLCNVDIFNPKYDCKIMTSKTDVSSSVITSLGAIVSCYGKTKCTASNKNRGIIKTFSNGCDYVSNKGVDTVSVGNTLYYVNKQEGKSLYVKGEPIINFYDPLVFPSDEFDASISQVNEKINQSLAFI 5ea4 F 2.3 BS01 5NM F 1 F137 F140 T397 D486 F488 F74 F77 T334 D423 F425 ? 0019064 Kd=7.8nM remove_due_to_license_issue P03420 26641933 607 QNITEEFYQSTCSAVSKGYLSALRTGWYTSVITIELSNIKGTDAKVKLIKQELDKYKNAVTELQLLMQSTPATFLGFLLGVGSAIASGVAVCKVLHLEGEVNKIKSALLSTNKAVVSLSNGVSVLTFKVLDLKNYIDKQLLPILNKQSCSISNIETVIEFQQKNNRLLEITREFSVNAGVTTPVSTYMLTNSELLSLINDMPITNDQKKLMSNNVQIVRQQSYSIMCIIKEEVLAYVVQLPLYGVIDTPCWKLHTSPLCTTNTKEGSNICLTRTDRGWYCDNAGSVSFFPQAETCKVQSNRVFCDTMNSLTLPSEVNLCNVDIFNPKYDCKIMTSKTDVSSSVITSLGAIVSCYGKTKCTASNKNRGIIKTFSNGCDYVSNKGVDTVSVGNTLYYVNKQEGKSLYVKGEPIINFYDPLVFPSDEFDASISQVNEKINQSLAFI 5ea5 F 3.05 BS01 TM3 F 1 F140 D486 E487 F488 F74 D406 E407 F408 ? 0019064 remove_due_to_license_issue P03420 26641933 602 NITEEFYQSTCSAVSKGYLSALRTGWYTSVITIELSNIDAKVKLIKQELDKYKNAVTELQLLMQSTPATNFLGFLLGVGSAIASGVAVCKVLHLEGEVNKIKSALLSTNKAVVSLSNGVSVLTFKVLDLKNYIDKQLLTVIEFQQKNNRLLEITREFSVNAGVTTPVSTYMLTNSELLSLINDMPITNDQKKLMSNNVQIVRQQSYSIMCIIKEEVLAYVVQLPLYGVIDTPCWKLHTSPLCTTNTKEGSNICLTRTDRGWYCDNAGSVSFFPQAETCKVQSNRVFCDTMNSLTLPSEVNLCNVDIFNPKYDCKIMTSKTDVSSSVITSLGAIVSCYGKTKCTASNKNRGIIKTFSNGCDYVSNKGVDTVSVGNTLYYVNKQEGKSLYVKGEPIINFYDPLVFPSDEFDASISQVNEKINQSLAFI 5ea6 F 2.75 BS01 5NP F 1 F137 M396 F488 F65 M312 F404 ? 0019064 remove_due_to_license_issue P03420 26641933 606 NITEEFYQSTCSAVSKGYLSALRTGWYTSVITIELSNIKAKVKLIKQELDKYKNAVTELQLLMQFLGFLLGVGSAIASGVAVCKVLHLEGEVNKIKSALLSTNKAVVSLSNGVSVLTFKVLDLKNYIDKQLLIETVIEFQQKNNRLLEITREFSVNAGVTTPVSTYMLTNSELLSLINDMPITNDQKKLMSNNVQIVRQQSYSIMCIIKEEVLAYVVQLPLYGVIDTPCWKLHTSPLCTTNTKEGSNICLTRTDRGWYCDNAGSVSFFPQAETCKVQSNRVFCDTMNSLTLPSEVNLCNVDIFNPKYDCKIMTSKTDVSSSVITSLGAIVSCYGKTKCTASNKNRGIIKTFSNGCDYVSNKGVDTVSVGNTLYYVNKQEGKSLYVKGEPIINFYDPLVFPSDEFDASISQVNEKINQSLAFI 5eak A 2.8 BS01 24R A 1 I59 G60 K61 V67 K82 M129 Y131 A132 G135 E179 L182 D193 I13 G14 K15 V21 K36 M83 Y85 A86 G89 E133 L136 D147 D175 K177 E179 N180 D193 S212 D129 K131 E133 N134 D147 S155 2.7.11.1,2.7.11.26 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q7KZI7 27491711 1000 QPHIGNYRLLKTIGKGNFAKVKLARHILTGKEVAVKIIDKTQLNSSSLQKLFREVRIMKVLNHPNIVKLFEVIETEKTLYLVMEYASGGEVFDYLVAHGRMKEKEARAKFRQIVSAVQYCHQKFIVHRDLKAENLLLDADMNIKIADFGFSFCGSPPYAAPELFQGKKYDGPEVDVWSLGVILYTLVSGSLPFDGQNLKELRERVLRGKYRIPFYMSTDCENLLKKFLILNPSKRGTLEQIMKDRWMNVGHEDDELKPYVEPLPDYKDPRRTELMVSMGYTREEIQDSLVGQRYNEVMATYLLLG 5eb3 A 2.4 BS01 UEG A 1 L166 I169 V176 P178 L181 L129 I132 V139 P141 L144 ? Kd=35.2mM remove_due_to_license_issue Q9I4L4 27113583 202 RTSIEQRSNAVSQVLLGIFSYVRWPKEPAVLQLCVVGPTEYADGLLRGMVQANGRRVHAERRAVDNPDLGTLCNVIYLGVVDERERQQVFRSLAGHPVLSISERGTECSVGSMFCLNVGGPRITFEANLDSIARSGVRVHPSVLKLARRQATP 5ece A 2.2 BS01 5N2 A 1 H1184 G1185 F1188 F1197 H1201 I1212 Y1213 S1221 Y1224 H81 G82 F85 F94 H98 I104 Y105 S113 Y116 2.4.2.-,2.4.2.30 0003950 ic50=9nM remove_due_to_license_issue IC50=9.0nM O95271 26546219 1402 AGTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKPEAP 5ech A 2.14 BS01 JAA A 1 T121 F125 F220 V222 H328 D329 G331 W336 G537 T115 F119 F214 V216 H322 D323 G325 W330 G531 6.3.2.52 0005515,0005524,0005737,0009864,0010046,0010224,0016597,0016874,0016881,0018117,0019899,0045087,0070728,0071365,0080123,2000030 remove_due_to_license_issue Q9SKE2 28223489 601 TFDMNRVIDEFDEMTRNAHQVQKQTLKEILLKNQSAIYLQNCGLNGNATDPEEAFKSMVPLVTDVELEPYIKRMVDGDTSPILTGHPVPAISLSSGTSQGRPKFIPFTDELMENTLQLFRTAFAFRNRDFPIDDNGKALQFIFSSKQYISTGGVPVGTATTNVYRNPNFKAGMKSITSPSCSPDEVIFSPDVHQALYCHLLSGILFRDQVQYVFAVFAHGLVHAFRTFEQVWEEIVTDIKDGVLSNRITVPSVRTAMSKLLTPNPELAETIRTKCMSLSNWYGLIPALFPNAKYVYGIMTGSMEPYVPKLRHYAGDLPLVSHDYGSSEGWIAANVTPRLSPEEATFAVIPNLGYFEFLPVSETGEGEEKPVGLTQVKIGEEYEVVITNYAGLYRYRLGDVVKVIGFYNNTPQLKFICRRNLILSINIDKNTERDLQLSVESAAKRLSEEKIEVIDFSSYIDVSTDPGHYAIFWEISGETNEDVLQDCCNCLDRAFIDAGYVSSRKCKTIGALELRVVAKGTFRKIQEHFLGLGSSAGQFKMPRCVKPSNAKVLQILCENVVSSYFSTAF 5eci A 1.56 BS01 JAA A 1 T121 F125 F220 V222 H328 G331 T115 F119 F214 V216 H322 G325 6.3.2.52 0005515,0005524,0005737,0009864,0010046,0010224,0016597,0016874,0016881,0018117,0019899,0045087,0070728,0071365,0080123,2000030 remove_due_to_license_issue Q9SKE2 28223489 601 TFDMNRVIDEFDEMTRNAHQVQKQTLKEILLKNQSAIYLQNCGLNGNATDPEEAFKSMVPLVTDVELEPYIKRMVDGDTSPILTGHPVPAISLSSGTSQGRPKFIPFTDELMENTLQLFRTAFAFRNRDFPIDDNGKALQFIFSSKQYISTGGVPVGTATTNVYRNPNFKAGMKSITSPSCSPDEVIFSPDVHQALYCHLLSGILFRDQVQYVFAVFAHGLVHAFRTFEQVWEEIVTDIKDGVLSNRITVPSVRTAMSKLLTPNPELAETIRTKCMSLSNWYGLIPALFPNAKYVYGIMTGSMEPYVPKLRHYAGDLPLVSHDYGSSEGWIAANVTPRLSPEEATFAVIPNLGYFEFLPVSETGEGEEKPVGLTQVKIGEEYEVVITNYAGLYRYRLGDVVKVIGFYNNTPQLKFICRRNLILSINIDKNTERDLQLSVESAAKRLSEEKIEVIDFSSYIDVSTDPGHYAIFWEISGETNEDVLQDCCNCLDRAFIDAGYVSSRKCKTIGALELRVVAKGTFRKIQEHFLGLGSSAGQFKMPRCVKPSNAKVLQILCENVVSSYFSTAF 5ect A 1.3 BS01 DUP A 1 N77 T81 I82 D83 Y86 K91 N86 T90 I91 D92 Y95 K100 A25 R64 G66 L73 D83 A34 R73 G75 L82 D92 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046080,0046081,0046872 Kd=5.2uM remove_due_to_license_issue P9WNS5 27740761 201 SGLVPRGSHMSTTLAIVRLDPGLPLPSRAHDGDAGVDLYSAEDVELAPGRRALVRTGVAVAVPFGMVGLVHPRSGLATRVGLSIVNSPGTIDAGYRGEIKVALINLDPAAPIVVHRGDRIAQLLVQRVELVELVEVSSFDEATSRG 5ecv A 2.085 BS02 5M2 A 1 R339 E434 G459 L461 D462 M515 W541 M631 D633 R328 E423 G448 L450 D451 M504 W530 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R328 E423 D451 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 27738104 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDVNGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 5edb A 1.18 BS01 5M8 A 1 F17 M21 A34 A37 A76 D77 R127 F19 M23 A36 A39 A78 D79 R129 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.1uM remove_due_to_license_issue Ki=105nM P15090 26878596 201 SHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5edc A 1.29 BS01 5M7 A 1 F16 M20 A33 A36 S53 S55 F57 A75 D76 C117 F18 M22 A35 A38 S55 S57 F59 A77 D78 C119 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.022uM remove_due_to_license_issue Ki=22nM P15090 26878596 201 AMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5edd A 1.97 BS01 DUP A 1 N77 T81 I82 D83 Y86 K91 N88 T92 I93 D94 Y97 K102 A25 R64 G66 L73 D83 A36 R75 G77 L84 D94 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046080,0046081,0046872 Kd=5.7uM remove_due_to_license_issue P9WNS5 27740761 202 HSSGLVPRGSHMSTTLAIVRLDPGLPLPSRAHDGDAGVDLYSAEDVELAPGRRALVRTGVAVAVPFGMVGLVHPRSGLATRVGLSIVNSPGTIDAGYRGEIKVALINLDPAAPIVVHRGDRIAQLLVQRVELVELVEVSSFDEA 5edi A 2.2 BS02 5M9 A 1 L675 V678 I692 Y693 F696 P712 M713 E721 V722 G725 Q726 F729 L218 V221 I235 Y236 F239 P255 M256 E264 V265 G268 Q269 F272 3.1.4.17 0004114,0007165,0008081 ic50=0.3nM remove_due_to_license_issue IC50=0.28nM Q9Y233 26878596 803 GLMQFTLPVRLCREIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 5edl A 1.95 BS01 VIB A 1 Y23 Y42 Y46 W49 E77 V88 Q95 D131 S135 Y21 Y40 Y44 W47 E75 V86 Q93 D129 S133 ? 0005886 Kd=4.5nM remove_due_to_license_issue O34738 27447050 201 SWKVKEIVIMSVISIVFAVVYLLFTHFGNVLAGMFGPIAYEPIYGIWFIVSVIAAYMIRKPGAALVSEIIAALVECLLGNPSGPMVIVIGIVQGLGAEAVFLATRWKAYSLPVLMLAGMGSSVASFIYDLFVSGYAAYSPGYLLIMLVIRLISGALLAGLLGKAVSDSLAYTGVLNGMALGKELKKKRKRASEHASL 5edn A 3.2 BS01 dna C 0 R220 Y223 R258 I262 N266 K270 R4 Y7 R42 I46 N50 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLA 5edn A 3.2 BS02 dna F 0 R220 P222 K243 Q265 R268 R4 P6 K27 Q49 R52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLA 5edn A 3.2 BS03 dna I 0 K225 G226 K9 G10 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLA 5edn B 3.2 BS01 dna D 0 K218 R220 P222 Y223 R258 Q259 I262 N266 K270 K2 R4 P6 Y7 R42 Q43 I46 N50 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn B 3.2 BS02 dna E 0 R220 P222 F240 K243 R246 Q265 R268 R4 P6 F24 K27 R30 Q49 R52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn B 3.2 BS03 dna L 0 K225 G226 K9 G10 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn G 3.2 BS01 dna F 0 K225 G226 K8 G9 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 KKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn G 3.2 BS02 dna H 0 R220 Y223 R258 N266 K270 R3 Y6 R41 N49 K53 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 KKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn G 3.2 BS03 dna I 0 R220 P222 F240 K243 Q265 R268 K272 R3 P5 F23 K26 Q48 R51 K55 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 KKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn J 3.2 BS01 dna K 0 R217 K218 R220 I221 Y223 R258 W263 N266 K270 R1 K2 R4 I5 Y7 R42 W47 N50 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edn J 3.2 BS02 dna L 0 K218 K219 R220 F240 K243 R246 Q265 R268 K2 K3 R4 F24 K27 R30 Q49 R52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 19 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5edq A 2.8 BS01 5N3 A 1 V726 A743 K745 E762 L788 M790 M793 L844 V30 A47 K49 E66 L92 M94 M97 L148 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=1.5nM P00533 26639762 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFDMDDVVDADEYLI 5edr A 2.6 BS01 5N4 A 1 L718 V726 A743 K745 E762 L788 M790 M793 L844 L22 V30 A47 K49 E64 L90 M92 M95 L146 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=34nM P00533 26639762 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLI 5eds A 2.8 BS01 5MT A 1 M804 P810 W812 I831 Y867 E880 K890 M953 I963 M554 P560 W562 I581 Y617 E630 K640 M700 I710 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 26652588 1204 SQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEVSLWDCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCKVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISSFNADKLTSATNPDKENSMSISILLDPIALPKHEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 5edu B 2.79 BS03 TSN B 1 H500 P501 H610 H611 F620 D649 H651 F680 Y782 H390 P391 H500 H501 F510 D539 H541 F570 Y672 3.5.1.-,3.5.1.98 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q9UBN7 27454933 2501 EEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAAASRTGLVYDQNMMNHCNLWDSHHPEVPQRILRIMCRLEELGLAGRCLTLTPRPATEAELLTCHSAEYVGHLRATEKMKTRELHRESSNFDSIYICPSTFACAQLATGAACRLVEAVLSGEVLNGAAVVRPPGHHAEQDAACGFCFFNSVAVAARHAQTISGHALRILIVDWDVHHGNGTQHMFEDDPSVLYVSLHRYDHGTFFPMGDEGASSQIGRAAGTGFTVNVAWNGPRMGDADYLAAWHRLVLPIAYEFNPELVLVSAGFDAARGDPLGGCQVSPEGYAHLTHLLMGLASGRIILILEGGYNLTSISESMAACTRSLLGDPPPLLTRPPLSGALASITETIQVHRRYWRSLR 5ee7 A 2.5 BS01 5MV A 1 F345 R346 K349 S350 T353 L399 N404 K405 F348 R349 K352 S353 T356 L397 N402 K403 E1009 D1018 E117 D126 3.2.1.17 0003796,0004888,0004930,0007166,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 Kd=0.62nM remove_due_to_license_issue P00720,P47871 27111510 1201 YSSFQVMYTVGYSLSLAALLLALAILGGLSKLHCTANAIHANLFLSFVLKASAVLFIDGLLRTVSTWLSDGAVAACRVAAVFMQYGIVANYCWLLVEGLYLHNLLGLNIFEMLRIDEGLRLKIYKDYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYPERSFFSLYLGIGWGAPALFVVPWAVVKCLFENVQCWTNMGFWWILRFPVFLAILINFFIFVRIVQLLVAKLRARQMHHTDYAFRLAKSTLTLIPLLGVHFVVFAFVTDEHRSAKLFFDLALSSFQGLLVAVLYCFLNKEVQSELRRRWHRA 5ee8 A 1.54 BS01 ZXM A 1 M69 S70 S130 N132 E166 T167 N170 T235 A237 R243 M44 S45 S105 N107 E141 T142 N145 T210 A212 R218 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue P0AD64 26729491 301 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 5eea A 2.195 BS01 dna E 0 K225 G226 K9 G10 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAKV 5eea A 2.195 BS02 dna C 0 R217 K218 R220 I221 Y223 I262 N266 K270 R1 K2 R4 I5 Y7 I46 N50 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAKV 5eea A 2.195 BS03 dna F 0 R220 K243 R246 Q265 R268 K272 R4 K27 R30 Q49 R52 K56 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAKV 5eea B 2.195 BS01 dna D 0 R220 I221 P222 Y223 Q259 I262 N266 K270 K273 R4 I5 P6 Y7 Q43 I46 N50 K54 K57 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5eea B 2.195 BS02 dna E 0 R220 P222 F240 K243 R246 Q265 R268 K272 R4 P6 F24 K27 R30 Q49 R52 K56 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5eea B 2.195 BS03 dna F 0 K225 G226 K9 G10 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5eea G 2.195 BS01 dna H 0 R217 K218 R220 I221 Y223 Q259 I262 N266 K270 R1 K2 R4 I5 Y7 Q43 I46 N50 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAKVK 5eea G 2.195 BS02 dna I 0 R220 P222 K243 R246 Q265 R268 R4 P6 K27 R30 Q49 R52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAKVK 5eea J 2.195 BS01 dna K 0 K218 R220 I221 P222 Y223 I262 N266 K270 K2 R4 I5 P6 Y7 I46 N50 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5eea J 2.195 BS02 dna L 0 R220 K243 R246 Q265 R268 R4 K27 R30 Q49 R52 ? 0000981,0003677,0006355 remove_due_to_license_issue Q92826 29638214 1 ~ 18 RKKRIPYSKGQLRELEREYAANKFITKDKRRKISAATSLSERQITIWFQNRRVKEKKVLAK 5eec A 1.87 BS01 ZXM A 1 C69 S70 W105 S130 N132 E166 N170 T235 T237 C238 G239 C44 S45 W80 S105 N107 E141 N145 T210 T212 C213 G214 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 26729491 301 LTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 5eef A 2.151 BS02 TSN A 1 S150 H192 H193 F202 D230 H232 W261 K330 Y363 S87 H129 H130 F139 D167 H169 W198 K267 Y300 ? remove_due_to_license_issue F8W4B7 27454933 2002 SATGTGLVYVDAFTRFHSHPECPARVSTVMEMLETEGLLGRCVQVEARAVTEDELLLVHTKEYVELMKSTQNMTEEELKTLAEKYDSVYLHPGFFSSACLSVGSVLQLVDKVMTSQLRNGFSINRPPGHHAQADKMNGFCMFNNLAIAARYAQKRHRVQRVLIVDWDVHHGQGIQYIFEEDPSVLYFSVHRYEDGSFWPHLKESDSSSVGSGAGQGYNINLPWNKVGMESGDYITAFQQLLLPVAYEFQPQLVLVAAGFDAVIGDPKGGMQVSPECFSILTHMLKGVAQGRLVLALEGGYNLQSTAEGVCASMRSLLGDPCPHLPSSGAPCESALKSISKTISDLYPFWKSLQT 5eei A 1.32 BS02 SHH A 1 P464 H573 H574 F583 D612 H614 F643 Y745 P23 H132 H133 F142 D171 H173 F202 Y304 3.5.1.98 remove_due_to_license_issue F8W4B7 27454933 2004 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 5eek A 1.59 BS02 TSN A 1 P464 H573 H574 F583 D612 H614 F643 L712 Y745 P24 H133 H134 F143 D172 H174 F203 L272 Y305 3.5.1.98 remove_due_to_license_issue F8W4B7 27454933 2004 SPITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLLTPLKTSATVSINNVLRAHAPFWSSLR 5een B 1.861 BS02 5OG B 1 P464 S531 H573 H574 F583 D612 H614 F643 L712 Y745 P23 S90 H132 H133 F142 D171 H173 F202 L271 Y304 3.5.1.98 remove_due_to_license_issue F8W4B7 27454933 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLPLKTSATVSINNVLRAHAPFWSSLR 5ef7 A 1.9 BS02 5OJ A 1 S531 H574 G582 F583 H614 F643 D705 L712 Y745 S91 H134 G142 F143 H174 F203 D265 L272 Y305 3.5.1.98 Ki=1nM remove_due_to_license_issue F8W4B7 27454933 804 SPITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 5ef8 A 2.6 BS02 LBH A 1 D460 H463 P464 S531 H573 H574 F583 D612 H614 F643 Y745 D19 H22 P23 S90 H132 H133 F142 D171 H173 F202 Y304 3.5.1.98 remove_due_to_license_issue F8W4B7 27454933 2004 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 5efa A 1.9 BS01 MGT A 1 R326 K341 W359 E363 F365 K378 F406 Y434 R8 K23 W41 E45 F47 K60 F88 Y116 ? Kd=14.7uM remove_due_to_license_issue Q9QLL6 26559973 501 MKIRQRQRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSQMRMEKLLINSAKKEDMKDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSNDLFDQWGYEESPKASELHGINELMNASDYTLKGVVVTKNVDHHH 5efb D 2.543 BS02 5OK D 1 H463 S531 H573 H574 F583 D612 H614 F643 L712 Y745 H22 S90 H132 H133 F142 D171 H173 F202 L271 Y304 3.5.1.98 remove_due_to_license_issue F8W4B7 27454933 2004 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLLTPLKTSATVSINNVLRAHAPFWSSLR 5efc A 1.9 BS01 GTP A 1 Q325 F327 R334 W359 E363 F406 Y434 Q2 F4 R11 W36 E40 F83 Y111 ? Kd=14.1uM remove_due_to_license_issue Q9QLL6 26559973 501 RQRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSQMRMEKLLINSAKKEDMKDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSNDLFDQWGYEESPKASELHGINELMNASDYTLKGVVVTKNVD 5efh D 2.162 BS02 FKS D 1 P571 H573 H574 G582 F583 D612 H614 F643 G743 Y745 P129 H131 H132 G140 F141 D170 H172 F201 G301 Y303 3.5.1.98 Ki=0.8uM remove_due_to_license_issue F8W4B7 27454933 2004 ITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 5eg4 A 1.32 BS02 5N7 A 1 H57 S96 N97 L99 D189 S190 C191 V213 S214 W215 G216 S217 G219 C220 H40 S78 N79 L81 D171 S172 C173 V191 S192 W193 G194 S195 G196 C197 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=21nM remove_due_to_license_issue P00760 27280436 504 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5ega A 2.15 BS03 GK0 A 1 E26 K34 H41 E80 D108 E119 K134 E26 K34 H41 E61 D89 E100 K115 3.1.-.- 0003723,0039694 ic50=8.7uM remove_due_to_license_issue C3W5S0 27510745 303 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 5egb A 1.977 BS01 dna C 0 H733 R736 H737 T740 R754 F756 R757 H761 R764 H765 R782 R785 N789 H793 R810 F812 N814 H817 R820 H821 H18 R21 H22 T25 R39 F41 R42 H46 R49 H50 R67 R70 N74 H78 R95 F97 N99 H102 R105 H106 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 EKPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5egb A 1.977 BS02 dna D 0 Y719 K731 S732 H733 K759 S760 H761 L763 R764 R767 Y775 D786 K787 S788 K815 S816 L819 R823 Y4 K16 S17 H18 K44 S45 H46 L48 R49 R52 Y60 D71 K72 S73 K100 S101 L104 R108 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 EKPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5egm A 1.841 BS01 5NY A 1 H57 Y99 H147 F174 C191 Q192 S195 W215 G216 E217 H41 Y86 H135 F162 C181 Q182 S185 W205 G206 E207 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 Ki=2.4nM remove_due_to_license_issue IC50=2.38nM P00740 26318999 303 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGASALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKLT 5egs A 2.15 BS02 5NR A 1 C50 Y51 V56 M60 E155 M157 Y159 E164 H317 C12 Y13 V18 M22 E117 M119 Y121 E126 H277 D63 E155 E164 H317 D25 E117 E126 H277 2.1.1.319 0000122,0003682,0005515,0005634,0005654,0005730,0006281,0006284,0006325,0006338,0006355,0008168,0008469,0010821,0016274,0018216,0032259,0035241,0035242,0035642,0036211,0042054,0042393,0044020,0045652,0045892,0062122,0070611,0070612,0090398,0140592,0140759,0140903,0140938,0140984,1901796,1990259,2000059 Kd=0.97uM remove_due_to_license_issue Kd=970nM, IC50=21000nM Q96LA8 26824386 402 TKRERDQLYYECYSDVSVHEEMIADRVRTDAYRLGILRNWAALRGKTVLDVGAGTGILSIFCAQAGARRVYAVEASAIWQQAREVVRFNGLEDRVHVLPGPVETVELPEQVDAIVSEWMGYGLLHESMLSSVLHARTKWLKEGGLLLPASAELFIVPISDQMLEWRLGFWSQVKQHYGVDMSCLEGFATRCLMGHSEIVVQGLSGEDVLARPQRFAQLELSRAGLEQELEAGVGGRFRCSCYGSAPMHGFAIWFQVTFPGGEKPLVLSTSPFHPATHWKQALLYLNEPVQVEQDTDVSGEITLLPSRDNPRRLRVLLRYKVGDQEEKTKDFAMED 5egs A 2.15 BS03 5NR A 2 L162 S168 L267 L343 L344 P345 L124 S130 L229 L303 L304 P305 D63 E155 E164 H317 D25 E117 E126 H277 2.1.1.319 0000122,0003682,0005515,0005634,0005654,0005730,0006281,0006284,0006325,0006338,0006355,0008168,0008469,0010821,0016274,0018216,0032259,0035241,0035242,0035642,0036211,0042054,0042393,0044020,0045652,0045892,0062122,0070611,0070612,0090398,0140592,0140759,0140903,0140938,0140984,1901796,1990259,2000059 Kd=0.97uM remove_due_to_license_issue Kd=970nM, IC50=21000nM Q96LA8 26824386 403 TKRERDQLYYECYSDVSVHEEMIADRVRTDAYRLGILRNWAALRGKTVLDVGAGTGILSIFCAQAGARRVYAVEASAIWQQAREVVRFNGLEDRVHVLPGPVETVELPEQVDAIVSEWMGYGLLHESMLSSVLHARTKWLKEGGLLLPASAELFIVPISDQMLEWRLGFWSQVKQHYGVDMSCLEGFATRCLMGHSEIVVQGLSGEDVLARPQRFAQLELSRAGLEQELEAGVGGRFRCSCYGSAPMHGFAIWFQVTFPGGEKPLVLSTSPFHPATHWKQALLYLNEPVQVEQDTDVSGEITLLPSRDNPRRLRVLLRYKVGDQEEKTKDFAMED 5egu A 2.21 BS01 5NQ A 1 P82 F83 Q85 V87 D88 L92 L94 N140 P36 F37 Q39 V41 D42 L46 L48 N94 ? Kd=1.4uM remove_due_to_license_issue IC50=5000nM, Kd=1400nM O60885 26735842 201 NPPPPETSNPNRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5eh0 A 2.18 BS01 5NW A 1 I531 G605 N606 I607 D608 S611 L654 M671 I16 G90 N91 I92 D93 S96 L139 M156 S646 D647 K649 P650 N652 D664 D674 T686 S131 D132 K134 P135 N137 D149 D159 T161 2.7.12.1 0004672,0005524,0006468 Ki=0.0005uM remove_due_to_license_issue IC50=140nM, Ki=0.440000nM P33981 27055065 801 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5eh2 E 2.05 BS01 dna A 0 R726 H733 R736 T740 F756 H761 R764 H765 T768 R782 R785 N789 H793 R810 F812 N814 H817 R820 H821 R10 H17 R20 T24 F40 H45 R48 H49 T52 R66 R69 N73 H77 R94 F96 N98 H101 R104 H105 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 KPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5eh2 E 2.05 BS02 dna B 0 Y719 K731 S732 K759 S760 Y775 K787 S788 K815 S816 L819 R823 Y3 K15 S16 K43 S44 Y59 K71 S72 K99 S100 L103 R107 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 KPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5eh2 F 2.05 BS01 dna C 0 R726 F728 R736 H737 F756 H761 R764 H765 T768 R782 R785 N789 H793 T796 R810 N814 H817 R820 H821 R9 F11 R19 H20 F39 H44 R47 H48 T51 R65 R68 N72 H76 T79 R93 N97 H100 R103 H104 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 PYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5eh2 F 2.05 BS02 dna D 0 S760 H761 Y775 D786 K787 S788 K815 S816 L819 R823 S43 H44 Y58 D69 K70 S71 K98 S99 L102 R106 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 PYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5eh5 A 1.207 BS02 XCZ A 1 H94 H96 H119 L197 T198 H90 H92 H115 L193 T194 H64 H94 H96 E106 H119 T198 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.35uM remove_due_to_license_issue P00918 26882437 303 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5eh7 A 1.425 BS02 5O5 A 1 Q92 H94 H119 F130 L197 T198 T199 W208 Q88 H90 H115 F126 L193 T194 T195 W204 H64 H94 H96 E106 H119 T198 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=330uM remove_due_to_license_issue P00918 26882437 303 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5eh8 A 1.381 BS02 5O6 A 1 F130 L197 T199 P201 F128 L195 T197 P199 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=791uM remove_due_to_license_issue P00918 26882437 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ehe A 1.5 BS02 WWO A 1 Q92 H94 H119 V121 F131 L198 T199 T200 P201 P202 Q89 H91 H116 V118 F127 L194 T195 T196 P197 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=6.1nM P00918 28001003 306 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ehg A 2.02 BS02 5O0 A 1 G107 G109 E111 E112 G101 G103 E105 E106 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P27915 27750202 302 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 5ehi A 1.303 BS02 5O3 A 1 W64 R68 M70 M233 L237 W58 R62 M64 M227 L231 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P27915 27750202 4002 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 5ehn A 2.6 BS01 5NZ A 1 Y72 D74 W86 G121 Y124 E202 W286 S293 Y337 Y341 W439 H447 Y72 D74 W86 G121 Y124 E202 W281 S288 Y332 Y336 W434 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Kd=0.033000nM P21836 26731630 1502 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 5ehp A 1.85 BS01 5OA A 1 R111 F113 H114 T219 E249 T253 L254 Q257 P491 K492 Q495 R107 F109 H110 T202 E226 T230 L231 Q234 P460 K461 Q464 D425 C459 R465 T466 Q506 D394 C428 R434 T435 Q475 3.1.3.48 0004725,0006470,0016311 ic50=12uM remove_due_to_license_issue Q06124 27347692 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHQLKEKNGDVIELKYPLNCADPTSERWFHGHLSGEAEKLLTEKGKHGSFLVRESSHPGDFVLSVRTGSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVELGTVLQLKQPLNTTRINAAEIESRVRELSKLAKQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGPNEPVSDYINANIIMPEFKPKKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 5ehq A 2.5 BS01 5O2 A 1 Y72 D74 W86 G121 Y124 E202 W286 Y337 Y341 W439 H447 Y72 D74 W86 G121 Y124 E202 W281 Y332 Y336 W434 H442 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Ki=33pM remove_due_to_license_issue P21836 26731630 1504 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 5ehr A 1.7 BS01 5OD A 1 E110 R111 F113 T219 E249 E250 T253 L254 Q257 P491 K492 Q495 E96 R97 F99 T192 E216 E217 T220 L221 Q224 P451 K452 Q455 D425 C459 R465 T466 Q506 D385 C419 R425 T426 Q466 3.1.3.48 0004725,0006470,0016311 Kd=73nM remove_due_to_license_issue IC50=70.0nM Q06124 27362227 601 RRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESGDFVLSVRTGDSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLAKQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPNEPVSDYINANIIMPEFKPKKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 5ehv A 1.208 BS01 5ON A 1 H94 H96 L197 T198 T199 P201 H92 H94 L195 T196 T197 P199 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=826uM remove_due_to_license_issue P00918 26882437 301 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ehw A 1.392 BS01 5OO A 1 H94 H96 F130 L197 T199 P201 H92 H94 F128 L195 T197 P199 H64 H94 H96 E106 H119 T198 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1005uM remove_due_to_license_issue P00918 26882437 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ehy A 2.26 BS01 5O4 A 1 I531 V539 A551 I586 M602 E603 G605 L654 I17 V25 A37 I72 M88 E89 G91 L140 D647 K649 N652 D664 T686 D133 K135 N138 D150 T159 2.7.12.1 0004672,0005524,0006468 ic50=0.81uM remove_due_to_license_issue P33981 27055065 908 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQVGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ei2 A 2.67 BS01 5O7 A 1 I531 M602 C604 G605 N606 I607 D608 L654 I16 M87 C89 G90 N91 I92 D93 L139 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=4840nM P33981 27055065 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ei3 A 1.71 BS02 5O8 A 1 W56 M101 W102 E103 R112 W166 A204 W30 M75 W76 E77 R86 W140 A178 ? 0000082,0000339,0000340,0000932,0001662,0003723,0003743,0005515,0005634,0005737,0005829,0006406,0006412,0006413,0006417,0010494,0010507,0016281,0016442,0016604,0016607,0017148,0019827,0019899,0030182,0031370,0033391,0036464,0045665,0045931,0048471,0051028,0051168,0070062,0071549,0098794,0098808,0098978,0099578,0140297 Kd=56.5uM remove_due_to_license_issue P06730 27592390 301 EVANPEHYIKHPLQNRWALWFFKNDKSKTWQANLRLISKFDTVEDFWALYNHIQLSSNLMPGCDYSLFKDGIEPMWEDEKNKRGGRWLITLNKQQRRSDLDRFWLETLLCLIGESFDDYSDDVCGAVVNVRAKGDKIAIWTTECENREAVTHIGRVYKERLGLPPKIVIGYQSHADTATKSGSTTKNRFVV 5ei4 A 1.05 BS01 5NV A 1 W81 P82 Q85 V87 D88 L92 N140 W40 P41 Q44 V46 D47 L51 N99 ? ic50=26.4uM remove_due_to_license_issue O60885 26735842 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ei6 A 2.01 BS01 5OQ A 1 I531 M602 G605 N606 I607 D608 L654 I663 P673 I16 M87 G90 N91 I92 D93 L139 I148 P158 D647 K649 N652 D664 T686 D132 K134 N137 D149 T166 2.7.12.1 0004672,0005524,0006468 ic50=0.099uM remove_due_to_license_issue IC50=74nM P33981 27055065 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDKDSQVGTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5ei8 A 2.17 BS01 5OE A 1 I531 A551 M602 C604 G605 N606 I607 D608 S611 L654 P673 I16 A36 M87 C89 G90 N91 I92 D93 S96 L139 P158 D647 K649 N652 D664 T686 D132 K134 N137 D149 T162 2.7.12.1 0004672,0005524,0006468 ic50=0.008uM remove_due_to_license_issue IC50=8nM P33981 27055065 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDVGTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 5ei9 E 1.921 BS01 dna A 0 R726 R736 H737 T740 R754 F756 H761 R764 H765 T768 R782 R785 N789 H793 T796 R810 F812 N814 H817 R820 H821 T824 R11 R21 H22 T25 R39 F41 H46 R49 H50 T53 R67 R70 N74 H78 T81 R95 F97 N99 H102 R105 H106 T109 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 EKPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5ei9 E 1.921 BS02 dna B 0 R736 S760 H761 Y775 D786 K787 S788 K815 S816 L819 R823 R21 S45 H46 Y60 D71 K72 S73 K100 S101 L104 R108 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 22 ~ 42 EKPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5ei9 F 1.921 BS01 dna C 0 R726 F728 H733 R736 H737 T740 K745 F756 R757 H761 R764 H765 T768 R782 F784 R785 N789 H793 T796 R810 F812 N814 H817 R820 H821 R10 F12 H17 R20 H21 T24 K29 F40 R41 H45 R48 H49 T52 R66 F68 R69 N73 H77 T80 R94 F96 N98 H101 R104 H105 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 1 ~ 21 KPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5ei9 F 1.921 BS02 dna D 0 S732 S760 H761 Y775 D786 K787 S788 K815 S816 L819 R823 S16 S44 H45 Y59 D70 K71 S72 K99 S100 L103 R107 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 remove_due_to_license_issue Q9NQV7 26833727 22 ~ 42 KPYVCRECGRGFSNKSHLLRHQRTHTGEKPYVCRECGRGFRDKSHLLRHQRTHTGEKPYVCRECGRGFRDKSNLLSHQRTHTGEKPYVCRECGRGFSNKSHLLRHQRTHT 5eie A 2.1 BS01 TZ2 A 1 W86 G121 Y124 E202 F297 Y337 W439 H447 Y449 W86 G121 Y124 E202 F292 Y332 W434 H442 Y444 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F292 F294 E329 H442 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Ki=23000pM remove_due_to_license_issue P21836 26731630 605 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSAT 5eif A 1.5 BS02 4M0 A 1 G107 S128 G129 G101 S122 G123 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P27915 27750202 302 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 5eij A 1.99 BS02 5OT A 1 H94 H96 H119 F131 L198 T199 T200 P202 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=1025nM P00918 26810836 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5eim A 1.54 BS01 rna C 0 N336 R338 R349 Y352 Y392 Y406 K436 T437 Y466 S470 C473 N477 M481 I484 R486 N7 R9 R20 Y23 Y63 Y77 K107 T108 Y137 S141 C144 N148 M152 I155 R157 ? 0003723 remove_due_to_license_issue O74958 28735863 1 ~ 8 ERISMINPRVVLDENGISHRSRYFIMLCDNETAIAHAKKTSIWAVKKDSSKRISDAYKKASVYFIFVAQQTYNALGYAQVVSDLNSTELPFWSDSSHAGGVRIKWIKTCNLFSAEISEIVSHMDHGSEARDGMEMMYDEGSRLCTLINYAIMKRIGR 5eim B 1.54 BS01 rna C 0 N414 R431 N88 R105 ? 0003723 remove_due_to_license_issue O74958 28735863 1 ~ 8 EKGERISMINPRVVLDENGISHRSRYFIMLCDNETAIAHAKKTSIWAVKKDSSKRISDAYKKASVYFIFVAQQTYNALGYAQVVSDLNSTELPFWSDSSHAGGVRIKWIKTCNLFSAEISEIVSHMDHGSEARDGMEMMYDEGSRLCTLINYAIMKRIGRD 5eim B 1.54 BS02 rna D 0 N336 R338 Y352 Y392 Y406 K436 T437 Y466 C473 N477 R483 N10 R12 Y26 Y66 Y80 K110 T111 Y140 C147 N151 R157 ? 0003723 remove_due_to_license_issue O74958 28735863 1 ~ 8 EKGERISMINPRVVLDENGISHRSRYFIMLCDNETAIAHAKKTSIWAVKKDSSKRISDAYKKASVYFIFVAQQTYNALGYAQVVSDLNSTELPFWSDSSHAGGVRIKWIKTCNLFSAEISEIVSHMDHGSEARDGMEMMYDEGSRLCTLINYAIMKRIGRD 5eis A 1.6 BS01 5OU A 1 P82 F83 V87 N140 I146 P41 F42 V46 N99 I105 ? Kd=1.8uM remove_due_to_license_issue IC50=1900nM, Kd=1800nM O60885 26735842 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5eiw A 1.611 BS02 X0V A 1 G107 P108 E112 G101 P102 E106 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue Q6YMS4 27750202 302 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 5eje A 1.9 BS01 AP5 A 1 P9 G10 G12 K13 G14 T15 T31 G32 L35 R36 K57 V59 V64 G85 R88 Q92 R119 R123 Y133 H134 F137 R156 R167 V202 P9 G10 G12 K13 G14 T15 T31 G32 L35 R36 K57 V59 V64 G85 R88 Q92 R119 R123 Y133 H134 F137 R156 R167 V202 K13 R88 R123 R156 R167 K13 R88 R123 R156 R167 2.7.4.3 0000287,0004017,0004550,0005515,0005524,0005737,0005829,0006139,0006172,0009123,0009132,0009165,0015951,0016208,0016301,0016776,0019205,0044209,0046083,0046940,0050145 remove_due_to_license_issue P69441 28559350 301 MRIILLGAPGAGKGTQAQFIMEKYGIPQISTGDMLRAAVKSGSELGKQAKDIMDACKLVTDELVIALVKERIAQEDCRNGFLLDGFPRTIPQADAMKEAGINVDYVLEFDVPDELIVDRIVGRRVHAPSGRVYHVKFNPPKVEGKDDVTGEELTTRKDDQEECVRKRLVEYHQMTAPLIGYYSKEAEAGNTKYAKVDGTKPVAEVRADLEKILG 5ejl A 2.3 BS01 C2E A 1 R106 R107 R108 R111 D138 I139 S140 G142 G143 C144 A145 K182 S203 C204 Q205 R113 R114 R115 R118 D145 I146 S147 G149 G150 C151 A152 K189 S210 C211 Q212 ? 0000166 Kd=0.24uM remove_due_to_license_issue G3FT00 27650952 301 SSGLVPRGSHMTEGTIKTSKYEIIAIFREELRKRTEIEIFFNNTSIITQLTRVDFAEFHIQTHRKIPSGHKIRFLLHSDSGKIEFNAALTKHDNDKGIRYAFSLPECLQVVQRRRDPRFRLRHEHDFYCRGRHKNGENYLFDIKDISDGGCALMTKTPNLKFLSHNALLKNAVLMLAEYGEITIDLVVKNVIVITLDNANEESESYYQISCQFKFRHLDDQRRIEKILLDLILEA 5ejl A 2.3 BS02 C2E A 2 L65 H67 G71 K72 Q105 R106 R107 R111 N183 I185 L75 H77 G81 K82 Q112 R113 R114 R118 N190 I192 ? 0000166 Kd=0.24uM remove_due_to_license_issue G3FT00 27650952 302 SSGLVPRGSHMTEGTIKTSKYEIIAIFREELRKRTEIEIFFNNTSIITQLTRVDFAEFHIQTHRKIPSGHKIRFLLHSDSGKIEFNAALTKHDNDKGIRYAFSLPECLQVVQRRRDPRFRLRHEHDFYCRGRHKNGENYLFDIKDISDGGCALMTKTPNLKFLSHNALLKNAVLMLAEYGEITIDLVVKNVIVITLDNANEESESYYQISCQFKFRHLDDQRRIEKILLDLILEA 5ejv A 2.58 BS02 444 A 1 W317 C320 A321 L324 M365 I397 I400 H479 W55 C58 A59 L62 M103 I135 I138 H217 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=60nM, EC50=54nM, Ki=51nM P51449 27080181 601 PYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5ejw A 2.6 BS01 5PZ A 1 F11 W32 W35 F23 W44 W47 ? 0035102 remove_due_to_license_issue Q8VDS3 27326334 101 HHSSGLVPRGSHMELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEERDRASG 5ek0 A 3.53 BS01 5P2 A 1 E1534 Y1537 W1538 N1540 V1541 G1581 M1582 D1586 E1589 F1598 R1602 A1604 R1605 R1608 E47 Y50 W51 N53 V54 G94 M95 D99 E102 F111 R115 A117 R118 R121 ? 0005216,0005261,0005886,0006811,0016020,0055085 remove_due_to_license_issue A8EVM5,Q15858 26680203 1808 PRGSHMYLRITNIVESSFFTKFIIYLIVLNMVTMMVEKEGQSQHMTEVLYWINVVFIILFTIEIILRIYVHRISFFKDPWSLFDFVVVIISIVGMFLADLIETYFVSPTLFRVIRLARIGRILRLVTAVPQMRKIVSALISVIPGMLSVIALMTLFFYIFAIMATQLFGERFPEWFGTLGESFYTLFQVMTLESWSMGIVRPLMEVYPYAWVFFIPFIFVVTFVMINLVVAIIVDAMAILNQKEEQHIID 5ek9 A 2.08 BS01 5P4 A 1 W370 P371 L381 N429 V435 W23 P24 L34 N82 V88 ? remove_due_to_license_issue Kd=47nM, IC50=2020nM, EC50=480nM P25440 29170024 501 EQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMP 5ekh A 1.34 BS02 5RD A 1 H94 H96 H119 L198 T199 T200 H91 H93 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.11uM remove_due_to_license_issue P00918 26692420 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ekj A 1.129 BS02 TG4 A 1 H94 H119 L198 T199 T200 P202 H92 H117 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1uM remove_due_to_license_issue P00918 26692420 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ekm A 1.33 BS02 TG5 A 1 Q92 H94 H96 H119 F131 T199 T200 Q89 H91 H93 H116 F127 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.48uM remove_due_to_license_issue P00918 26692420 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ekn A 2.594 BS01 N58 A 1 V39 A52 E72 M107 P108 F109 M110 D168 F169 V38 A51 E71 M106 P107 F108 M109 D167 F168 D150 K152 N155 D168 T185 D149 K151 N154 D167 T170 2.7.11.24 0000165,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005737,0005829,0006468,0006970,0007254,0018105,0032755,0033554,0034644,0035556,0050729,0051403,0070301,0071347,0072709,0072740,0106310,1903936 remove_due_to_license_issue O15264 27369736 401 SLIRKKGFYKQDVNKTAWELPKTYVSPTHVGSGAYGSVCSAIDKRSGEKVAIKKLSRPFQSEIFAKRAYRELLLLKHMQHENVIGLLDVFTPASSLRNFYDFYLVMPFMQTDLQKIMGMEFSEEKIQYLVYQMLKGLKYIHSAGVVHRDLKPGNLAVNEDCELKILDFVTRWYRAPEVILSWMHYNQTVDIWSVGCIMAEMLTGKTLFKGKDYLDQLTQILKVTGVPGTEFVQKLNDKAAKSYIQSLPQTPRKDFTQLFPRASPQAADLLEKMLELDVDKRLTAAQALTHPFFEPFRDPEEETEAQQPFDDSLEHEKLTVDEWKQHIYKEIVNFSP 5eko A 2.0 BS01 N17 A 1 A52 R68 E72 M107 M110 L167 D168 F169 L171 A51 R67 E71 M106 M109 L166 D167 F168 L170 D150 K152 N155 D168 T185 D149 K151 N154 D167 T175 2.7.11.24 0000165,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005737,0005829,0006468,0006970,0007254,0018105,0032755,0033554,0034644,0035556,0050729,0051403,0070301,0071347,0072709,0072740,0106310,1903936 ic50=15785nM remove_due_to_license_issue IC50=15785nM O15264 27369736 401 SLIRKKGFYKQDVNKTAWELPKTYVSPTHVGSGAYGSVCSAIDKRSGEKVAIKKLSRPFQSEIFAKRAYRELLLLKHMQHENVIGLLDVFTPASSLRNFYDFYLVMPFMQTDLQKIMGMEFSEEKIQYLVYQMLKGLKYIHSAGVVHRDLKPGNLAVNEDCELKILDFGLGYVVTRWYRAPEVILSWMHYNQTVDIWSVGCIMAEMLTGKTLFKGKDYLDQLTQILKVTGVPGTEFVQKLNDKAAKSYIQSLPQTPRKDFTQLFPRASPQAADLLEKMLELDVDKRLTAAQALTHPFFEPFRDPEEETEAQQPFDDSLEHEKLTVDEWKQHIYKEIVNFSP 5ekx A 1.76 BS02 2CQ A 1 G107 P108 E112 G101 P102 E106 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 remove_due_to_license_issue P27915 27750202 302 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTR 5el2 A 1.75 BS01 KBR A 1 L76 H77 M89 G92 K93 L96 W114 L76 H77 M89 G92 K93 L96 W114 0005549 remove_due_to_license_issue 27535661 202 DTTPRRDAEYPPPELLEALKPLHDICLGKTGVTEEAIKKFSDEEIHEDEKLKCYMNCLFHEAKVVDDNGDVHLEKLHDSLPSSMHDIAMHMGKRCLYPEGETLCDKAFWLHKCWKQSDPKHYFLV 5el2 A 1.75 BS02 KBR A 2 A62 L80 F123 L124 V125 A62 L80 F123 L124 V125 0005549 remove_due_to_license_issue 27535661 203 DTTPRRDAEYPPPELLEALKPLHDICLGKTGVTEEAIKKFSDEEIHEDEKLKCYMNCLFHEAKVVDDNGDVHLEKLHDSLPSSMHDIAMHMGKRCLYPEGETLCDKAFWLHKCWKQSDPKHYFLV 5el2 B 1.75 BS01 KBR B 1 L76 H77 A88 M89 G92 L96 W114 L76 H77 A88 M89 G92 L96 W114 0005549 remove_due_to_license_issue 27535661 201 DTTPRRDAEYPPPELLEALKPLHDICLGKTGVTEEAIKKFSDEEIHEDEKLKCYMNCLFHEAKVVDDNGDVHLEKLHDSLPSSMHDIAMHMGKRCLYPEGETLCDKAFWLHKCWKQSDPKHYFLV 5el2 B 1.75 BS02 KBR B 2 L19 L58 F59 A62 F123 V125 L19 L58 F59 A62 F123 V125 0005549 remove_due_to_license_issue 27535661 202 DTTPRRDAEYPPPELLEALKPLHDICLGKTGVTEEAIKKFSDEEIHEDEKLKCYMNCLFHEAKVVDDNGDVHLEKLHDSLPSSMHDIAMHMGKRCLYPEGETLCDKAFWLHKCWKQSDPKHYFLV 5el9 A 1.1 BS01 5DL A 1 R99 R121 S199 K201 R91 R113 S191 K193 4.2.1.19 0000105,0004424 Ki=23nM remove_due_to_license_issue O23346 27717128 303 SARIGEVKRETKETNVSVKINLDGHGVSDSSTGIPFLDHMLDQLASHGLFDVHVRATGDTHIDDHHTNEDVALAIGTALLKALGERKGINRFGDFTAPLDEALIHVSLDLSGRPYLGYNLEIPTQRVGTYDTQLVEHFFQSLVNTSGMTLHIRQLAGKNSHHIIEATFKAFARALRQATESDPRRGGTIPSSKGVLSRS 5eld A 1.4 BS01 FUC F 1 N44 A46 N44 A46 ? 0005576 remove_due_to_license_issue D6R7L2 27082955 3 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5eld A 1.4 BS02 FUC F 2 T47 F48 P93 H94 T47 F48 P93 H94 ? 0005576 remove_due_to_license_issue D6R7L2 27082955 5 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5eld A 1.4 BS03 GAL A 1 E51 Q56 H57 W88 N90 K91 E51 Q56 H57 W88 N90 K91 ? 0005576 remove_due_to_license_issue D6R7L2 27082955 202 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5eld E 1.4 BS01 FUC I 1 N44 A46 N44 A46 ? 0005576 remove_due_to_license_issue D6R7L2 27082955 3 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5eld E 1.4 BS02 FUC I 2 T47 F48 H94 T47 F48 H94 ? 0005576 remove_due_to_license_issue D6R7L2 27082955 5 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5eld E 1.4 BS03 GAL E 1 E51 Q56 W88 N90 K91 E51 Q56 W88 N90 K91 ? 0005576 remove_due_to_license_issue D6R7L2 27082955 202 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5ele D 1.6 BS01 GAL K 1 Y18 H94 Y18 H94 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 2 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5ele D 1.6 BS02 FUC K 1 N44 A46 N44 A46 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 3 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5ele D 1.6 BS03 FUC K 2 I47 P93 H94 I47 P93 H94 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 5 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elf A 1.55 BS01 GLC K 1 G45 I47 G45 I47 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 1 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elf A 1.55 BS02 GAL K 1 Y18 H94 Y18 H94 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 2 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elf A 1.55 BS03 FUC K 1 I47 F48 H94 I47 F48 H94 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 5 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elf E 1.55 BS01 GLC M 1 G45 I47 G45 I47 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 1 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elf E 1.55 BS02 GAL M 1 Y18 H94 Y18 H94 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 2 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elf E 1.55 BS03 FUC M 1 A46 I47 F48 P93 H94 A46 I47 F48 P93 H94 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 27082955 5 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5elv A 1.92 BS01 5PX A 1 P105 S108 S217 K218 G219 P105 S108 S217 K218 G219 ? 0015276,0016020 Kd=0.16uM remove_due_to_license_issue P19491 27276258 312 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 5elv A 1.92 BS03 5PX B 1 P105 F106 M107 S108 P105 F106 M107 S108 ? 0015276,0016020 Kd=0.16uM remove_due_to_license_issue P19491 27276258 312 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 5elv B 1.92 BS01 5PX A 1 P105 F106 M107 S108 P105 F106 M107 S108 ? 0015276,0016020 Kd=0.16uM remove_due_to_license_issue P19491 27276258 312 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 5elv B 1.92 BS02 5PX B 1 P105 S108 S217 K218 G219 P105 S108 S217 K218 G219 ? 0015276,0016020 Kd=0.16uM remove_due_to_license_issue P19491 27276258 312 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITYVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLSEQGLLDKLKNKWWYDKGECGS 5elw A 1.4 BS01 5LD A 1 R99 R121 S199 K201 R91 R113 S191 K193 4.2.1.19 0000105,0004424 Ki=15nM remove_due_to_license_issue O23346 27717128 303 SARIGEVKRETKETNVSVKINLDGHGVSDSSTGIPFLDHMLDQLASHGLFDVHVRATGDTHIDDHHTNEDVALAIGTALLKALGERKGINRFGDFTAPLDEALIHVSLDLSGRPYLGYNLEIPTQRVGTYDTQLVEHFFQSLVNTSGMTLHIRQLAGKNSHHIIEATFKAFARALRQATESDPRRGGTIPSSKGVLSRS 5ely A 1.81 BS04 5PU A 1 Y234 H377 D387 E424 E425 D453 R534 G548 Y552 H553 Y176 H319 D329 E366 E367 D395 R476 G486 Y490 H491 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=44nM remove_due_to_license_issue IC50=44nM Q04609 27074627 817 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 5elz A 1.8 BS02 3V9 A 1 E70 G100 R113 G116 I117 E69 G99 R112 G115 I116 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 remove_due_to_license_issue Q2FWC7 27759386 303 KVGIDAGGTLIKIVQEQDNQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLEKHHHHHH 5em3 A 1.4 BS01 5Q0 A 1 I652 V657 Y707 N708 F714 I28 V33 Y83 N84 F90 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 801 SMEMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5em3 A 1.4 BS02 5Q0 A 2 I652 V657 F714 I28 V33 F90 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 802 SMEMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5em5 A 2.65 BS01 5Q2 A 1 L718 V726 A743 K745 L788 M790 Q791 M793 G796 L844 L22 V30 A47 K49 L88 M90 Q91 M93 G96 L144 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=37nM P00533 26819674 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKETSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLIP 5em6 A 2.78 BS01 5Q3 A 1 L718 A743 K745 E762 M790 Q791 M793 G796 L844 T854 D855 L22 A47 K49 E63 M91 Q92 M94 G97 L145 T155 D156 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=850nM P00533 26819674 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYEEDMDDVVDADEYLIP 5em7 A 2.81 BS01 5Q4 A 1 L718 A743 M790 M793 G796 L844 T854 L23 A48 M92 M95 G98 L146 T156 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=1090nM P00533 26819674 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKEATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYDMDDVVDADEYLIP 5em8 A 2.8 BS01 5Q4 A 1 L718 A743 M793 P794 F795 G796 L844 T854 D855 L23 A48 M95 P96 F97 G98 L146 T156 D157 D837 A839 R841 N842 D855 G874 D139 A141 R143 N144 D157 G174 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=1090nM P00533 26819674 1101 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKEATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPDMDDVVDADEYLI 5emj A 2.273 BS02 5QJ A 1 F300 Y304 L312 L319 F327 E435 E444 S578 W579 F288 Y292 L300 L307 F315 E423 E432 S566 W567 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 ic50=33nM remove_due_to_license_issue IC50=<100nM O14744 26985292 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 5emk A 2.52 BS02 5QH A 1 F300 Y304 Q309 S310 P311 L312 L319 F327 E435 E444 V503 S578 W579 F288 Y292 Q297 S298 P299 L300 L307 F315 E423 E432 V491 S566 W567 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 remove_due_to_license_issue IC50=<100nM O14744 26985292 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 5eml A 2.39 BS02 5QK A 1 Y304 Q309 L312 L319 F327 E435 E444 V503 S578 W579 F580 Y292 Q297 L300 L307 F315 E423 E432 V491 S566 W567 F568 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 ic50=23nM remove_due_to_license_issue IC50=<100nM O14744 26985292 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 5emm A 2.37 BS02 5QL A 1 F300 Q309 L319 F327 E435 E444 F577 S578 W579 F580 F288 Q297 L307 F315 E423 E432 F565 S566 W567 F568 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 remove_due_to_license_issue IC50=<100nM O14744 26985292 702 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 5en1 A 2.58 BS01 rna B 0 K22 F24 D49 V51 M53 F64 F66 A96 V97 R99 H108 K11 F13 D38 V40 M42 F53 F55 A85 V86 R88 H97 ? 0003676,0003723 remove_due_to_license_issue P22626 1 ~ 7 RKKREKEQFRKLFIGGLSFETTEESLRNYYEQWGKLTDCVVMRDPASKRSRGFGFVTFSSMAEVDAAMAARPHSIDGRVVEPKRAVAREESGKPGAHVTVKKLFVGGIKEDTEEHHLRDYFEEYGKIDTIEIITDRQSGKKRGFGFVTFDDHDPVDKIVLQKYHTINGHNAEVRKALSRQEMQE 5en3 A 1.25 BS01 7LU A 1 S117 T118 T119 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=620nM remove_due_to_license_issue P02766 27050398 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5en3 B 1.25 BS01 7LU B 1 K15 L17 S117 T118 T119 K6 L8 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=620nM remove_due_to_license_issue P02766 27050398 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5enb A 1.73 BS01 5Q5 A 1 Y1350 Y1353 N1391 S1392 Y1395 Y38 Y41 N79 S80 Y83 ? remove_due_to_license_issue Q8WWQ0 29910922 1501 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRN 5enc A 1.59 BS01 5QD A 1 V1345 Y1350 V33 Y38 ? remove_due_to_license_issue Q8WWQ0 29910922 1503 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRNT 5ene A 1.49 BS01 5Q8 A 1 F1341 V1345 Y1350 T1396 F29 V33 Y38 T84 ? remove_due_to_license_issue Q8WWQ0 29910922 1501 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRN 5enf A 1.37 BS01 5Q7 A 1 V1345 Y1350 T1396 I1403 V33 Y38 T84 I91 ? remove_due_to_license_issue Q8WWQ0 29910922 1503 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRN 5eng A 1.3 BS01 5QN A 1 L1109 P1110 Q1113 V1115 L1120 N1168 V1174 L27 P28 Q31 V33 L38 N86 V92 2.3.1.-,2.3.1.48 remove_due_to_license_issue Q92793 30258543 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5enh A 1.95 BS01 5QB A 1 P1340 F1341 V1345 Y1350 Y1395 P28 F29 V33 Y38 Y83 ? remove_due_to_license_issue Q8WWQ0 29910922 1501 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRN 5eni A 1.69 BS01 5QA A 1 P1340 V1345 Y1350 Y1353 Y1395 P28 V33 Y38 Y41 Y83 ? remove_due_to_license_issue Q8WWQ0 29910922 1501 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRN 5enj A 1.63 BS01 5Q9 A 1 P1340 F1341 V1345 Y1350 P28 F29 V33 Y38 ? remove_due_to_license_issue Q8WWQ0 29910922 1501 SMSYDIQAWKKQCEELLNLIFQCEDSEPFRQPVDLLEYPDYRDIIDTPMDFATVRETLEAGNYESPMELCKDVRLIFSNSKAYTPSKRSRIYSMSLRLSAFFEEHISSVLSDYKSALRFHKRN 5enk A 2.11 BS01 5QV A 1 G59 G61 L78 D80 Y119 T120 F156 D276 G278 G13 G15 L32 D34 Y73 T74 F110 D218 G220 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=8nM remove_due_to_license_issue IC50=8.0nM P56817 26985314 503 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5enm A 1.98 BS01 5QU A 1 G59 G61 D80 Y119 F156 W163 D276 G278 G13 G15 D34 Y73 F110 W117 D218 G220 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=70nM remove_due_to_license_issue P56817 26985314 503 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5eob A 1.75 BS01 5QQ A 1 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 A54 Y105 M106 D110 R154 M157 A167 D168 Y176 D1204 A1206 R1208 N1209 D1222 A1243 D150 A152 R154 N155 D168 A186 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.24nM remove_due_to_license_issue IC50=0.850000nM P08581 27061987 1401 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 5eol A 2.2 BS01 5QO A 1 F49 A65 K67 I104 L174 I185 D186 F17 A33 K35 I72 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.3nM remove_due_to_license_issue IC50=0.300000nM P11309 27096050 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5eom A 2.55 BS01 CTP A 1 R23 K24 I27 I31 R62 Y63 L66 V68 K248 S252 K255 R23 K24 I27 I31 R61 Y62 L65 V67 K238 S242 K245 2.7.7.- 0001654,0005515,0005524,0005525,0005634,0008283,0008284,0009653,0016779,0043010,0046872 remove_due_to_license_issue Q13394 27271801 403 DIAAQAKLVYHLNKYYNEKCQARKAAIAKTIREVCKVVSDVLKEVEVQEPRFISSLNEMNRYEGLEVISPTEFEVVLYLNQMGVFNFVDDGSLPGCAVLKLSDGRKRSMSLWVEFITASGYLSARKIRSRFQTLVAQAVDKCSYRDVVKMVADTSEVKLRIRDRYVVQITPAFKCTGIWPRSAAHWPLPHIPWPGPNRVAEVKAEGFNLLSKECHESDAWVLQFAEAENRLQMGGCRKKCLSILKTLRDRHLELPGQPLNNYHMKTLVSYECEKHPRESDWDESCLGDRLNGILLQLISCLQCRRCPHYFLPNLDLFQGKPHSALENAAKQTWRLAREILTNPKSLEKL 5eou B 2.4 BS01 ATP B 1 S18 S19 T20 K23 G201 A202 T203 M204 K247 K248 G296 S299 S9 S10 T11 K14 G189 A190 T191 M192 K235 K236 G284 S287 ? 0005524,0005737,0043107,0043683,0044096,0046872,0051301 Kd=4.37uM remove_due_to_license_issue G3XD28,G3XD30 27022027 401 NTLLGIDISSTSVKLLELSRSGGRYKVEAYAVEPLPPNAVVEKNIVELEGVGQALSRVLVKAKTNLKSAVVAVAGSAVITKTIEMEAGLSEDELENQLKIEADQYIPYPLEEVAIDFEVQGLSRNPERVDVLLAACRKENVEVREAALALAGLTAKVVDVEAYALERSYALLSSQLDTDQLTVAVVDIGATMTTLSVLHNGRTIYTREQLFGGRQLTEEIQRRYGLSVEEAGLAKKQGGLPDDYDSEVLRPFKDAVVQQVSRSLQFFFAAGQFNDVDYIVLAGGTASIQDLDRLIQQKIGTPTLVANPFADMALNGKVNAGALASDAPALMIACGLALRSFDSMARINLLPW 5ep7 A 1.198 BS01 5QR A 1 P1110 V1115 L1120 N1168 P32 V37 L42 N90 2.3.1.-,2.3.1.48 remove_due_to_license_issue Kd=4000nM Q92793 30258543 1201 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5epn A 2.3 BS02 5R2 A 1 Q1041 F1043 H1057 V1078 D1081 K1136 G1137 S1139 F1154 R1155 A1156 A1157 Q59 F61 H75 V96 D99 K154 G155 S157 F172 R173 A174 A175 H1057 D1081 G1137 S1139 H75 D99 G155 S157 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 Kd=2.2nM remove_due_to_license_issue C1KIK8 26682473 1203 MASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVDFIPVESLETTM 5epr A 1.65 BS01 5QY A 1 V657 V662 F714 V30 V35 F87 ? Kd=91uM remove_due_to_license_issue Kd=91000nM P55201 27167503 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5eps A 1.47 BS01 5QX A 1 V657 P658 E661 V662 Y707 N708 F714 V31 P32 E35 V36 Y81 N82 F88 ? Kd=38uM remove_due_to_license_issue Kd=38000nM P55201 27167503 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5epy A 2.3 BS02 5R2 A 1 Q1041 F1043 Y1056 H1057 V1078 D1081 I1132 K1136 G1137 A1139 F1154 R1155 T1156 A1157 Q60 F62 Y75 H76 V97 D100 I151 K155 G156 A158 F173 R174 T175 A176 H1057 D1081 G1137 A1139 H76 D100 G156 A158 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 remove_due_to_license_issue C1KIK8 26682473 1203 HMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTM 5eq1 A 1.55 BS01 BEA A 1 P658 F714 P31 F87 ? Kd=21uM remove_due_to_license_issue P55201 27167503 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5eqe A 2.4 BS01 5R8 A 1 D306 Y354 W420 F435 Y440 D202 Y250 W316 F331 Y336 2.7.1.32,2.7.1.82 Kd=132uM remove_due_to_license_issue Kd=132000nM, IC50=87000nM P35790 26700752 501 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAIMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5eqp A 2.35 BS01 5R9 A 1 D306 Y333 Y354 W420 F435 D201 Y228 Y249 W315 F330 2.7.1.32,2.7.1.82 Kd=4uM remove_due_to_license_issue Kd=4000nM, IC50=3900nM P35790 26700752 501 QPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5eqq A 1.65 BS02 5RS A 1 F1043 H1057 V1078 D1081 L1135 K1136 G1137 A1139 F1154 R1155 A1156 A1157 F54 H68 V89 D92 L146 K147 G148 A150 F165 R166 A167 A168 H1057 D1081 G1137 A1139 H68 D92 G148 A150 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 Kd=6.7nM remove_due_to_license_issue C1KIK8 26682473 1203 GSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSAGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTM 5eqy A 2.5 BS01 5RA A 1 D306 Y333 Y354 F361 W420 E434 F435 D201 Y228 Y249 F256 W315 E329 F330 2.7.1.32,2.7.1.82 Kd=10nM remove_due_to_license_issue IC50=66nM, Kd=10.0nM P35790 26700752 501 QPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5er1 E 2.0 BS01 0HT E 1 D32 G34 S74 Y75 G76 D77 L128 F189 D215 G217 D35 G37 S78 Y79 G80 D81 L133 F194 D219 G221 3.4.23.22 0004190,0006508 Ki=960nM remove_due_to_license_issue P11838 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 5er2 E 1.8 BS01 0EK E 1 D30 D32 G34 Y75 G76 D77 D114 L128 F189 I213 D215 G217 T218 T219 I297 I301 D33 D35 G37 Y79 G80 D81 D119 L133 F194 I217 D219 G221 T222 T223 I300 I304 3.4.23.22 0004190,0006508 Ki=0.27uM remove_due_to_license_issue P11838 2676515 327 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 5er4 X 1.813 BS03 5RL X 1 C84 H85 F88 C85 H86 F89 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 remove_due_to_license_issue P02638 27303795 103 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 5er5 A 1.26 BS03 ET A 1 F88 E89 F89 E90 ? 0005509,0005515,0005576,0005615,0005634,0005737,0006417,0007155,0007409,0007611,0008270,0008284,0016310,0019210,0042803,0043123,0044548,0045917,0046872,0048143,0048156,0048306,0050786,0071638,0097490,1990845 remove_due_to_license_issue P02638 27303795 103 MSELEKAVVALIDVFHQYSGREGDKHKLKKSELKELINNELSHFLEEIKEQEVVDKVMETLDSDGDGECDFQEFMAFVAMITTACHEFFE 5erg B 2.202 BS01 SAM B 1 Q92 V94 G118 G120 S121 S123 F124 E139 F140 R144 R167 D168 V169 D203 L204 P205 Q84 V86 G110 G112 S113 S115 F116 E131 F132 R136 R159 D160 V161 D195 L196 P197 2.1.1.220 0005515,0005634,0008033,0008168,0030488,0031515,0032259,0160107 Kd=44.33uM remove_due_to_license_issue P46959 27582183 401 NCFSGYKDLIKEGDLTLIWVSRDNIKPVRMHSEEVFNTRYGSFPHKDIIGKPYGSQIAIRTFAFVHVLQPTPELWTLSLPHRTQIVYTPDSSYIMQRLNCSPHSRVIEAGTGSGSFSHAFARSVGHLFSFEFHHIRYEQALEEFKEHGLIDDNVTITHRDVCQGGFLIKKGDTTSYEFGNNETAASLNANVVFLDLPAPWDAIPHLDSVISVDEKVGLCCFSPCIEQVDKTLDVLEKYGWTDVEMVEIQGRQYESRRQMVRSLNDALERLRDIKRHKIKEGDSNYKWKEVTKMEAEIKSHTSYLTFAFKVVNRSRDDEKVNEIL 5es1 A 2.8 BS01 5RC A 1 G65 V70 A83 K85 M132 Y134 A135 G138 E182 D196 G15 V20 A33 K35 M82 Y84 A85 G88 E132 D146 D178 K180 E182 N183 D196 S215 D128 K130 E132 N133 D146 S152 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q96L34 26841763 4000 PHVGNYRLLRTIGKGNFAKVKLARHILTGREVAIKIIDKTQLNPSSLQKLFREVRIMKGLNHPNIVKLFEVIETEKTLYLVMEYASAGEVFDYLVSHGRMKEKEARAKFRQIVSAVHYCHQKNIVHRDLKAENLLLDAEANIKIADFGFSNSPPYAAPELFQGKKYDGPEVDIWSLGVILYTLVSGSLPFDGHNLKELRERVLRGKYRVPFYMSTDCESILRRFLVLNPAKRCTLEQIMKDKWINIGYEGEELKPYTEPEEDFGDTKRIEVMVGMGYTREEIKESLTSQKYNEVTATYLLLGRK 5est E 2.09 BS01 0P2 E 1 H57 W172 C191 Q192 S195 S214 F215 V216 H45 W164 C184 Q185 S188 S207 F208 V209 3.4.21.36 0004252,0005515,0005576,0005615,0006508,0008236,0046872 remove_due_to_license_issue P00772 2611205 1 VVGGTEAQRNSWPSQISLQYRSGSSWAHTCGGTLIRQNWVMTAAHCVDRELTFRVVVGEHNLNQNNGTEQYVGVQKIVVHPYWNTDDVAAGYDIALLRLAQSVTLNSYVQLGVLPRAGTILANNSPCYITGWGLTRTNGQLAQTLQQAYLPTVDYAICSSSSYWGSTVKNSMVCAGGDGVRSGCQGDSGGPLHCLVNGQYAVHGVTSFVSRLGCNVTRKPTVFTRVSAYISWINNVIASN 5etb A 1.33 BS01 5RO A 1 F653 V657 F714 F26 V30 F87 ? Kd=29uM remove_due_to_license_issue Kd=29000nM P55201 27167503 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5eth A 2.803 BS01 5RT A 1 C320 H323 L324 A327 M365 V376 F378 F388 I400 F401 V480 C52 H55 L56 A59 M97 V108 F110 F120 I132 F133 V212 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=56nM P51449 27080181 501 EIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIF 5etj A 2.3 BS01 IM5 A 1 Y88 A116 G118 F200 E201 M219 N243 H257 Y90 A118 G120 F202 E203 M221 N245 H259 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S35 H66 H88 Y90 E91 A118 M221 S222 N245 V247 H259 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 Kd=66pM remove_due_to_license_issue Ki=7nM P00491 26927977 301 TLMENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHDEVAAAGKQAAQKLEQFVSILMASIPLPD 5etj B 2.3 BS01 IM5 B 1 Y88 A116 A117 G118 F200 E201 M219 N243 H257 V260 Y89 A117 A118 G119 F201 E202 M220 N244 H258 V261 S33 H64 H86 Y88 E89 A116 M219 S220 N243 V245 H257 S34 H65 H87 Y89 E90 A117 M220 S221 N244 V246 H258 2.4.2.1 0000255,0001882,0002060,0003824,0004731,0005515,0005576,0005737,0005829,0006139,0006148,0006149,0006157,0006166,0006204,0006738,0006955,0009116,0009165,0009410,0016757,0016763,0032743,0034418,0034774,0042102,0042301,0042802,0043101,0046059,0046638,0047975,0070062,1904813 Kd=66pM remove_due_to_license_issue Ki=7nM P00491 26927977 301 LMENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVMMQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFPAMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSLITNKVIMDYESLEKANHDEVAAAGKQAAQKLEQFVSILMASIPLPD 5etk A 1.09 BS02 5RU A 1 T42 P43 L45 G46 Y53 N55 W89 R121 F123 T43 P44 L46 G47 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=1.5uM remove_due_to_license_issue P26281 27094768 202 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5etl A 1.82 BS05 5RV A 1 T42 P43 L45 Y53 N55 R121 F123 T45 P46 L48 Y56 N58 R118 F120 R82 R92 D95 D97 R85 R89 D92 D94 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=23uM remove_due_to_license_issue P26281 27094768 206 SAMTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5etm A 1.46 BS01 5RW A 1 T42 P43 P44 L45 Y53 N55 W89 R121 F123 T43 P44 P45 L46 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=3.9uM remove_due_to_license_issue P26281 27094768 201 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5etn A 1.4 BS06 5RX A 1 T42 P43 P44 L45 Y53 N55 W89 R121 F123 T43 P44 P45 L46 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=4.3uM remove_due_to_license_issue P26281 27094768 206 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5eto A 1.07 BS01 5RY A 1 T42 P43 L45 G46 Y53 N55 W89 R121 F123 T43 P44 L46 G47 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=2.7uM remove_due_to_license_issue Kd=2700nM P26281 27094768 201 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5etp A 1.05 BS06 5RZ A 1 T42 P43 L45 Y53 N55 W89 R121 F123 T44 P45 L47 Y55 N57 W91 R123 F125 R82 R92 D95 D97 R84 R94 D97 D99 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0046654,0046656 Kd=0.7uM remove_due_to_license_issue Kd=700nM P26281 27094768 209 AMTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5etq A 1.96 BS04 YH2 A 1 T43 A44 P45 V46 Q51 F54 N56 G90 P91 R92 F123 T43 A44 P45 V46 Q51 F54 N56 G90 P91 R92 F123 R83 R92 D95 D97 R83 R92 D95 D97 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=0.33uM remove_due_to_license_issue Q2G0Q5 27094768 204 MIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 5etr B 1.32 BS02 5RW B 1 T43 A44 V46 Y48 Q51 F54 N56 G90 R92 F123 T43 A44 V46 Y48 Q51 F54 N56 G90 R92 F123 R83 R92 D95 D97 R83 R92 D95 D97 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=0.3uM remove_due_to_license_issue Q2G0Q5 27094768 202 MIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 5ets B 1.95 BS02 5RX B 1 T43 A44 P45 V46 Y48 Q51 F54 N56 G90 P91 R92 F123 T43 A44 P45 V46 Y48 Q51 F54 N56 G90 P91 R92 F123 R83 R92 D95 D97 R83 R92 D95 D97 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=1.24uM remove_due_to_license_issue Q2G0Q5 27094768 202 MIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 5ett B 1.55 BS02 5RY B 1 T43 A44 P45 V46 Y48 Q51 F54 N56 W89 G90 P91 R92 F123 T43 A44 P45 V46 Y48 Q51 F54 N56 W89 G90 P91 R92 F123 R83 R92 D95 D97 R83 R92 D95 D97 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=0.59uM remove_due_to_license_issue Q2G0Q5 27094768 202 MIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 5etv A 1.72 BS02 5RZ A 1 T43 A44 P45 V46 G47 F54 N56 R121 F123 T44 A45 P46 V47 G48 F55 N57 R122 F124 R83 R92 D95 D97 R84 R93 D96 D98 2.7.6.3 0003848,0005524,0009396,0016301,0046654,0046656,0046872 Kd=0.57uM remove_due_to_license_issue Q2G0Q5 27094768 202 HMIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 5etx A 2.35 BS02 5RS A 1 Q1041 F1043 H1057 L1135 K1136 G1137 S1139 F1154 R1155 T1156 A1157 Q48 F50 H64 L142 K143 G144 S146 F161 R162 T163 A164 H1057 D1081 G1137 S1139 H64 D88 G144 S146 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 remove_due_to_license_issue C1KIK8 26682473 1202 GSVVIVGRINLAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTMR 5etx A 2.35 BS03 5RS C 1 D1079 R1155 D86 R162 H1057 D1081 G1137 S1139 H64 D88 G144 S146 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 remove_due_to_license_issue C1KIK8 26682473 1202 GSVVIVGRINLAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRTAVSTRGVAKAVDFIPVESLETTMR 5ety A 2.9 BS02 K56 A 1 H1184 S1186 F1188 A1191 I1192 D1198 H1201 I1212 Y1213 Y1224 I1228 H80 S82 F84 A87 I88 D94 H97 I108 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue IC50=31nM O95271 27196752 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTIKMAHAPPGHHSVIGRPSLAYAEYVIYRGEQAYPEYLITYQIMKPE 5eu1 A 1.6 BS01 5SW A 1 F44 F45 V49 I53 A54 N100 Y106 F23 F24 V28 I32 A33 N79 Y85 ? Kd=15.4nM remove_due_to_license_issue Kd=0.794328nM, IC50=19nM Q9H8M2 26914985 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5eud A 2.24 BS01 5S6 A 1 H201 F249 X311 F500 H147 F195 X257 F446 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 ic50=0.15uM remove_due_to_license_issue Q67PY4 27013389 602 SQIKPYRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEVH 5eud A 2.24 BS02 5S6 A 2 L128 P130 W340 I344 Y345 A346 L74 P76 W286 I290 Y291 A292 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 ic50=0.15uM remove_due_to_license_issue Q67PY4 27013389 603 SQIKPYRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEVH 5eud B 2.24 BS01 5S6 A 1 L128 P130 I344 Y345 A346 L70 P72 I286 Y287 A288 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 remove_due_to_license_issue Q67PY4 27013389 602 PYRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEV 5eud B 2.24 BS02 5S6 A 2 H201 F249 X311 F500 H143 F191 X253 F442 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 remove_due_to_license_issue Q67PY4 27013389 603 PYRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEV 5eue A 2.83 BS01 5S5 A 1 P130 I344 Y345 A346 P74 I288 Y289 A290 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 remove_due_to_license_issue Q67PY4 27013389 601 IKPYRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEV 5eue A 2.83 BS02 5S5 B 1 F249 F500 F193 F444 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 remove_due_to_license_issue Q67PY4 27013389 602 IKPYRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEV 5eue B 2.83 BS01 5S5 A 1 N432 V496 F500 N373 V437 F441 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 remove_due_to_license_issue Q67PY4 27013389 601 YRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEVH 5eue B 2.83 BS02 5S5 B 1 L128 P130 I344 Y345 A346 L69 P71 I285 Y286 A287 ? 0004058,0008117,0016020,0016829,0016830,0019752,0030149,0030170,0042802 remove_due_to_license_issue Q67PY4 27013389 602 YRDRFPSHARLPRAGLPRAEILAEIAAMGAAESPAWRDGYASGAVYHGDEHHIAFLNEVYALQSQSNPLHPDLWPSTAKFEAEVVAMTAHMLGGDAAGGTVCGTVTSGGTESLLLAMKTYRDWARATKGITAPEAVVPVSAHAAFDKAAQYFGIKLVRTPLDADYRADVAAMREAITPNTVVVAGSAPGFPHGVVDPIPEIAALAAEHGIGCHVDACLGGFILPWAERLGYPVPPFDFRLEGVTSVSADTHKYGYGAKGTSVILYRRPDLLHYQYFIAADWPGGIYASPTFAGSRPGALSATAWAAMLSLGEEGYLDATRRILQAADRLKAGVRAIPSLKILGDPLWVIAVASDELNIYQVMEEMAGRGWRLNGLHRPPAFHVALTLRHTEPGVVDRFLADLQDAVAQVRAHPEKATGMAPVYGMAAAAPPELVRQVSTGFIDLLYEVH 5ev8 A 2.3 BS03 3R9 A 1 D81 H139 C158 K161 N167 H197 D79 H137 C156 K159 N165 H195 H77 H79 D81 H139 C158 K161 N167 H197 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P52699 27303030 303 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESK 5ev8 A 2.3 BS04 3R9 A 2 G110 V112 G108 V110 H77 H79 D81 H139 C158 K161 N167 H197 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue P52699 27303030 304 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESK 5eva A 1.45 BS01 5S9 A 1 P658 E661 Y707 N708 F714 P32 E35 Y81 N82 F88 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5evb A 1.841 BS03 3R9 A 1 H118 D120 F156 I162 H196 P227 H85 D87 F123 I127 H159 P188 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=10uM remove_due_to_license_issue P52700 27303030 403 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 5evd A 1.8 BS01 VC2 A 1 H118 D120 F156 I162 H196 P227 H86 D88 F124 I128 H160 P189 H116 H118 D120 H121 H196 Y229 H263 H84 H86 D88 H89 H160 Y191 H225 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=10uM remove_due_to_license_issue P52700 27303030 401 AEVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 5evk A 1.627 BS01 3C7 A 1 W39 D120 H196 S225 W16 D87 H159 S186 H116 H118 D120 H121 H196 Y229 H263 H83 H85 D87 H88 H159 Y190 H224 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=12uM remove_due_to_license_issue P52700 27303030 401 EVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLTALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRRTGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAGHTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCDVLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAG 5evz A 1.85 BS02 ADP A 1 T38 Y39 G226 G227 G255 E293 K296 R297 S300 G363 G364 R367 T13 Y14 G201 G202 G230 E268 K271 R272 S275 G338 G339 R342 D34 K96 E201 D224 D9 K71 E176 D199 3.6.4.10 0005524,0140662 Kd=0.000000064M remove_due_to_license_issue P11021 27144892 503 DVGTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQLTSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDIGGGQTKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLSG 5ew0 A 1.3 BS02 3C7 A 1 H109 D111 F146 T147 H186 N213 H247 H69 D71 F106 T107 H146 N173 H207 N107 H109 D111 H186 C205 K208 N213 H247 N67 H69 D71 H146 C165 K168 N173 H207 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=0.26uM remove_due_to_license_issue Q9RMI1 27303030 302 NLTLTHFKGPLYIVEDKEYVQENSMVYIGTDGITIIGATWTPETAETLYKEIRKVSPLPINEVINTNYHTDRAGGNAYWKTLGAKIVATQMTYDLQKSQWGSIVNFTRQGNNKYPNLEKSLPDTVFPGDFNLQNGSIRAMYLGEAHTKDGIFVYFPAERVLYGNCILKENLGNMSFANRTEYPKTLEKLKGLIEQGELKVDSIIAGHDTPIHDVGLIDHYLTLLEKAP 5ew3 A 2.5 BS01 5T2 A 1 A866 K868 E885 V916 C919 H1026 L1035 I1044 C1045 D1046 F1047 A46 K48 E65 V96 C99 H150 L159 I168 C169 D170 F171 D1028 A1030 R1032 N1033 D1046 D152 A154 R156 N157 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=0.0012uM remove_due_to_license_issue IC50=23nM P35968 26629594 1201 PYDASKWEFPRDRLKLGKPLGRGAFGQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVIVEFCKFGNLSTYLRSKRNEFVPYKVKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANA 5ew9 A 2.181 BS01 5VC A 1 L139 V147 A160 A213 G216 L263 A273 W277 L13 V21 A34 A87 G90 L137 A147 W151 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T161 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Ki<0.01nM remove_due_to_license_issue IC50=0.064000nM O14965 26732741 1000 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 5ewa A 2.3 BS03 9BZ A 1 W28 D81 H139 K161 H197 W26 D79 H137 K159 H195 H77 H79 D81 H139 C158 K161 N167 H197 H75 H77 D79 H137 C156 K159 N165 H195 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=15uM remove_due_to_license_issue P52699 27303030 303 SLPDLKIEKLDEGVYVHTSFEEVNGWGVVPKHGLVVLVNAEAYLIDTPFTAKDTEKLVTWFVERGYKIKGSISSHFHSDSTGGIEWLNSRSIPTYASELTNELLKKDGKVQATNSFSGVNYWLVKNKIEVFYPGPGHTPDNVVVWLPERKILFGGCFIKPYGLGNLGDANIEAWPKSAKLLKSKYGKAKLVVPSHSEVGDASLLKLTLEQAVKGLNESK 5ewd A 1.58 BS01 5SH A 1 V662 N708 F714 V36 N82 F88 ? remove_due_to_license_issue Kd=>200000nM P55201 27167503 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5ewh A 1.63 BS01 5SG A 1 I652 N708 F714 I26 N82 F88 ? Kd=170uM remove_due_to_license_issue Kd=170000nM P55201 27167503 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5ewj A 2.77 BS01 QEL B 1 Y109 S132 L135 Y82 S105 L108 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 26912815 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGGET 5ewj B 2.77 BS01 QEL B 1 Q110 I111 F114 F176 E236 Q70 I71 F74 F136 E196 ? remove_due_to_license_issue Ki=10.0nM, Kd=7.6nM, IC50=110nM Q13224 26912815 503 PPSIGIAVILVGTSDEVAIKDLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPAEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPR 5ewk A 1.6 BS01 P34 A 1 R77 S78 K94 N110 S117 T118 L124 W128 Q158 E160 R42 S43 K59 N75 S82 T83 L89 W93 Q123 E125 2.4.2.31 Kd=14uM remove_due_to_license_issue C9Z6T8 27002155 301 KAAAPACPRFDDPVHAAADPRVDVERITPDPVWRTTCGTLYRSDSRGPAVVFEQGFLPKDVIDGQYDIESYVLVNQPSPYVSTTYDHDLYKTWYKSGYNYYIDAPGGVDVNKTIGDRHKWADQVEVAFPGGIRTEFVIGVCPVDKKTRTEKMSECVGNPHYEPWH 5ewm A 2.76 BS01 5SM B 1 Y109 I133 Y82 I106 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 26912815 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGGET 5ewm B 2.76 BS01 5SM B 1 P78 Q110 I111 F114 M134 A135 P177 P41 Q73 I74 F77 M97 A98 P140 ? remove_due_to_license_issue IC50=12nM Q13224 26912815 503 PPSIGIAVILVGTSDEVAIKDFHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPAEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPR 5ewy A 1.4 BS01 5TQ A 1 R77 S78 K94 S117 W128 Q158 E160 R42 S43 K59 S82 W93 Q123 E125 2.4.2.31 Kd=50uM remove_due_to_license_issue C9Z6T8 27002155 301 KAAAPACPRFDDPVHAAADPRVDVERITPDPVWRTTCGTLYRSDSRGPAVVFEQGFLPKDVIDGQYDIESYVLVNQPSPYVSTTYDHDLYKTWYKSGYNYYIDAPGGVDVNKTIGDRHKWADQVEVAFPGGIRTEFVIGVCPVDKKTRTEKMSECVGNPHYEPWH 5exh C 1.3 BS01 dna A 0 K53 R54 H81 R87 K88 L92 K2 R3 H30 R36 K37 L41 1.14.11.80 0003677,0008270 remove_due_to_license_issue Q8BG87 26774490 1 ~ 12 KKRKRCGTCDPCRRLENCGSCTSCTNRRTHQICKLRKCEVLKKKA 5exh C 1.3 BS02 dna B 0 K53 T73 R79 T80 H81 Q82 K2 T22 R28 T29 H30 Q31 1.14.11.80 0003677,0008270 remove_due_to_license_issue Q8BG87 26774490 1 ~ 12 KKRKRCGTCDPCRRLENCGSCTSCTNRRTHQICKLRKCEVLKKKA 5exl A 2.3 BS01 5SS A 1 R39 H40 L41 C42 H57 Y143 I151 D189 A190 C191 K192 G193 S195 T213 W215 G218 R26 H27 L28 C29 H44 Y134 I141 D182 A183 C184 K185 G186 S188 T206 W208 G211 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=3.7nM remove_due_to_license_issue Ki=3.7nM P03951 27073051 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5exm A 2.09 BS01 5ST A 1 R39 H40 L41 C42 H57 I151 D189 A190 C191 K192 G193 S195 T213 W215 R26 H27 L28 C29 H44 I141 D182 A183 C184 K185 G186 S188 T206 W208 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=6.3nM remove_due_to_license_issue Ki=6.3nM P03951 27073051 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5exn A 1.49 BS01 5SU A 1 R39 H40 L41 C42 H57 I151 D189 A190 C191 K192 G193 S195 W215 G216 G218 C219 G226 V227 Y228 R26 H27 L28 C29 H44 I141 D182 A183 C184 K185 G186 S188 W208 G209 G211 C212 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=23nM remove_due_to_license_issue Ki=23nM P03951 27073051 302 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVNYTDSQRPISLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQA 5exw A 1.9 BS01 7DT A 1 G36 T37 T38 Y39 G226 G227 G228 T229 G255 E293 K296 R297 S300 G363 G364 R367 G10 T11 T12 Y13 G200 G201 G202 T203 G229 E267 K270 R271 S274 G337 G338 R341 D34 K96 E201 D224 D8 K70 E175 D198 3.6.4.10 0005524,0140662 Kd=0.000000064M remove_due_to_license_issue P11021 27144892 501 VGTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQLTSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDIGGGQTKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLSG 5exx A 3.311 BS01 C2E A 1 R144 E330 S333 R334 H337 R7 E193 S196 R197 H200 ? 0005524,0006355,0008134,0016887,0043565 remove_due_to_license_issue G3XCV0 26712005 502 REPNLFRSLVGTSRAIQQVRQMMQQVADTDASVLILGESGTGKEVVARNLHYHSKRREGPFVPVNCGAIPAELLESELFGHEKGAFTGAITSRAGRFELANGGTLFLDEIGDMPLPMQVKLLRVLQERTFERVGSNKTQNVDVRIIAATHKNLEKMIEDGTFREDLYYRLNVFPIEMAPLRERVEDIALLLNELISRMEHEKRGSIRFNSAAIMSLCRHDWPGNVRELANLVERLAIMHPYGVIGVGELPKKFRHV 5exx A 3.311 BS02 C2E A 2 L142 F143 R144 R185 N186 Y189 R334 L5 F6 R7 R48 N49 Y52 R197 ? 0005524,0006355,0008134,0016887,0043565 remove_due_to_license_issue G3XCV0 26712005 503 REPNLFRSLVGTSRAIQQVRQMMQQVADTDASVLILGESGTGKEVVARNLHYHSKRREGPFVPVNCGAIPAELLESELFGHEKGAFTGAITSRAGRFELANGGTLFLDEIGDMPLPMQVKLLRVLQERTFERVGSNKTQNVDVRIIAATHKNLEKMIEDGTFREDLYYRLNVFPIEMAPLRERVEDIALLLNELISRMEHEKRGSIRFNSAAIMSLCRHDWPGNVRELANLVERLAIMHPYGVIGVGELPKKFRHV 5ey0 A 1.6 BS02 GTP A 1 V22 F24 S43 R44 R45 K47 L49 E157 K158 V22 F24 S43 R44 R45 K47 L49 E157 K158 ? 0003677,0003700,0005525,0005737,0006355,0045892 Kd=2.26mM remove_due_to_license_issue A7X1N2 27596595 302 MSLLSKTRELNTLLQKHKGIAVDFKDVAQTISSVTVTNVFIVSRRGKILGSSLNELLKSQRIIQMLEERHIPSEYTERLMEVKQTESNIDIDNVLTVFPPENRELFIDSRTTIFPILGGGERLGTLVLGRVHDDFNENDLVLGEYAATVIGMEILREKHSEVEKEARDKAAITMAINSLSYSEKEAIEHIFEELGGTEGLLIASKVADRVGITRSVIVNALRKLESAGVIESRSKGTFIKVKKEKFLDELEK 5ey4 A 1.86 BS01 DTP A 1 R60 R297 S300 G364 S365 R367 N389 R35 R268 S271 G335 S336 R338 N360 D34 K96 E201 D224 D9 K71 E172 D195 3.6.4.10 0005524,0140662 Kd=0.00075M remove_due_to_license_issue P11021 27144892 501 DVGTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQLTSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDITKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLSG 5ey8 A 3.5 BS01 5SV A 1 H231 D232 T237 S314 E315 P316 S342 Y343 G344 L350 D469 I480 H218 D219 T224 S301 E302 P303 S329 Y330 G331 L337 D456 I467 N207 H231 A346 N194 H218 A333 6.2.1.20 0005524,0005886,0006631,0006633,0008610,0008922,0016874,0070566 remove_due_to_license_issue A0R618 26900152 701 GQIKFPDGSSIVAHVERWAKVRGDKLAYRFLDFSTERDGVPRDLTWAQFSARNRAVAARLQQVTQPGDRVAILCPQNLDYLVAFFGALYAGRIAVPLFDPSEPGHVGRLHAVLDNCHPSAILTTTEAAEGVRKFFRTRPANQRPRVIAVDAVPDDVASTWVNPDEPDETTIAYLQYTSRIPTGVQITHLNLATNVVQVIEALEGEEGDRGLSWLPFFHDMGLITALLAPMIGHYFTFMTPAAFVRRPERWIRELARKEGDTGGTISVAPNFAFDHAAARGVPKPGSPPLDLSNVKAVLNGSEPISAATVRRFNEAFGPFGFPPKAIKPSYGLAEATLFVSTTPSAEEPKIITVDRDQLNSGRIVEVDADSPKAVAQASAGKVGIAEWAVIVDAESATELPDGQVGEIWISGQNMGTGYWGKPEESVATFQNILKSRTNPSHAEGATDDATWVRTGDYGAFYDGDLYITGRVKDLVIIDGRNHYPQDLEYSAQEASKAIRTGYVAAFSVPANQLPDEVFENAHSGIKRDPDDTSEQLVIVAERAPDIGPITDDIRAAIAVRHGVTVRDVLLTAAGAIPRTSSGKIGRRACRAAYLDGSL 5ey9 A 2.5 BS01 5SV A 1 H230 D231 M232 S278 L310 S313 E314 P315 S341 Y342 G343 L344 L349 D468 I479 R482 K600 H219 D220 M221 S267 L299 S302 E303 P304 S330 Y331 G332 L333 L338 D457 I468 R471 K589 6.2.1.20 0005524,0005886,0006631,0006633,0008610,0008922,0016874,0070566 Kd=3.87uM remove_due_to_license_issue B2HMK0 26900152 701 YHNPFIVNGKIRFPENTNLVRHVEKWARVRGDKLAYRFLDFSTERDGVERDILWSEFSARNRAVGARLQQVTQPGDRIAILCPQNLDYLISFFGALYSGRIAVPLFDPAEHVGRLHAVLDDCTPSTILTTTDSAEGVRKFIRSRSAKERPRVIAVDAVPTEVASTWQQPNELTTAYLQYTVPSGVQITHLNLPTNVLQVLNALEGQEGDRGVSWLPFFHDMGLITVLLASVLGHSFTFMTPAAFVRRPGRWIRELARKPGETGGTFSAAPNFAFEHAAMRGVPRDDEPPLDLSNVKGILNGSEPVSPASMRKFFKAFEPYGLRETAVKPSYGLAEATLFVSTTPMDEVPTVIHVDRDELNKQRFVEVAADAPNAVAQVSAGKVGVDEWAVIVDTETASELPDGQIGEIWLHGNNLGIGYWGKEEESAQTFRNILKSRVPESHAEGAPDDGLWVRTGDYGTYFKGHLYIAGRIKDLVIIDGRNHYPQDLEYTAQESTKALRVGYVAAFSVPANQLPQKVFDDPHAGLSFDPEDTSEQLVIVGERAAGTHKLEYQPIADDIRAAIAVGHGVTVRDVLLVSAGTIPRTSSGKIGRRACRTAYIDGSLRSTVFA 5eyc A 1.8 BS01 5SZ A 1 I1084 V1092 A1108 Y1159 M1160 D1164 R1208 N1209 M1211 A1221 D1222 Y1230 I32 V40 A51 Y102 M103 D107 R151 N152 M154 A164 D165 Y173 D1204 A1206 R1208 N1209 D1222 A1243 D147 A149 R151 N152 D165 A186 2.7.10.1 0004672,0004713,0005524,0006468 ic50=3nM remove_due_to_license_issue IC50=3nM P08581 26812066 1401 IDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 5eyd A 1.85 BS01 5T1 A 1 I1084 V1092 A1108 Y1159 M1160 D1164 R1208 N1209 M1211 A1221 D1222 Y1230 I33 V41 A51 Y100 M101 D105 R149 N150 M152 A162 D163 Y171 D1204 A1206 R1208 N1209 D1222 A1243 D145 A147 R149 N150 D163 A184 2.7.10.1 0004672,0004713,0005524,0006468 ic50=1nM remove_due_to_license_issue IC50=1nM P08581 26812066 1401 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEH 5eyk A 1.93 BS02 5U5 A 1 L99 G100 K122 E141 Q145 L154 M156 L170 F172 A173 P174 G176 E177 L223 L12 G13 K35 E54 Q58 L67 M69 L83 F85 A86 P87 G89 E90 L136 D216 K218 E220 N221 D234 T252 D129 K131 E133 N134 D147 T161 2.7.11.1 0004672,0005524,0006468 ic50=3nM remove_due_to_license_issue Q6DE08 27496137 401 FTIDDFDIVRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHARRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY 5eym A 2.7 BS01 5U5 A 1 L74 A95 K97 I141 M143 H145 M146 G149 Q153 L197 L34 A52 K54 I98 M100 H102 M103 G106 Q110 L151 D190 K192 S194 N195 D208 D217 T226 D144 K146 S148 N149 D162 D171 T174 2.7.12.2 0000165,0000187,0004672,0004674,0004708,0004712,0004713,0005078,0005515,0005524,0005634,0005737,0005739,0005769,0005770,0005783,0005794,0005813,0005829,0005856,0005886,0005925,0006338,0006468,0006935,0007165,0007254,0007507,0008285,0008545,0010628,0014044,0016020,0021697,0030182,0030216,0030295,0030878,0032872,0035401,0035987,0038133,0042552,0043410,0043539,0044342,0045893,0048009,0048538,0048679,0048870,0050772,0060020,0060324,0060425,0060440,0060502,0060674,0060711,0070371,0070374,0071902,0090170,0090398,0097110,0106310,0140801,1903226,2000641 remove_due_to_license_issue IC50=25nM Q02750 27496137 401 ELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMTRSYMSPERLVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL 5eyo A 2.39 BS01 dna B 0 R25 H28 N29 R33 R36 S59 R60 R6 H9 N10 R14 R17 S40 R41 ? 0046983 remove_due_to_license_issue P61244 27903915 4 ~ 19 HMADKRAHHNALERKRRDHIKDSFHSLRDSVPSLQGEKASRAQILDKATEYIQYMRRKNHTHQQDIDDLKRQNALLEQQVRALEKAR 5eyo C 2.39 BS01 dna D 0 R25 H28 N29 R33 R36 R60 R6 H9 N10 R14 R17 R41 ? 0046983 remove_due_to_license_issue P61244 27903915 4 ~ 19 HMADKRAHHNALERKRRDHIKDSFHSLRDSVPSLQGEKASRAQILDKATEYIQYMRRKNHTHQQDIDDLKRQNALLEQQVRALEKARS 5eyr A 1.57 BS01 5T0 A 1 L87 M102 W103 G106 F110 W145 Y148 N176 N179 W207 L66 M81 W82 G85 F89 W124 Y127 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=5uM remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ezg A 1.84 BS01 5T4 A 1 L87 F110 W138 Y148 N176 N179 W207 L66 F89 W117 Y127 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=12uM remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ezg A 1.84 BS02 5T4 A 2 L76 V80 F114 T121 G124 L137 W138 E180 F184 F187 L55 V59 F93 T100 G103 L116 W117 E159 F163 F166 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=12uM remove_due_to_license_issue P9WMC1 26806381 302 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ezh A 1.7 BS01 841 A 1 L76 V80 F114 G124 R128 L137 W138 E180 F184 F187 L55 V59 F93 G103 R107 L116 W117 E159 F163 F166 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=24uM remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ezh A 1.7 BS02 841 A 2 L87 W103 G106 F110 W138 Y148 N176 N179 W207 L66 W82 G85 F89 W117 Y127 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=24uM remove_due_to_license_issue P9WMC1 26806381 302 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ezx A 1.9 BS01 5T5 A 1 Q73 G74 L91 D93 S96 V130 Y132 R189 D289 G291 T292 Q17 G18 L35 D37 S40 V74 Y76 R133 D222 G224 T225 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=87nM remove_due_to_license_issue P56817 26878596 501 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5ezz A 2.1 BS01 5T6 A 1 Q73 G74 D93 S96 N98 W137 F169 I171 I179 D289 G291 Q17 G18 D37 S40 N42 W81 F113 I115 I123 D222 G224 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=145nM remove_due_to_license_issue P56817 26878596 501 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5f00 A 1.95 BS01 5T8 A 1 G74 L91 D93 Y132 I179 D289 G291 T293 G18 L35 D37 Y76 I123 D221 G223 T225 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=250nM remove_due_to_license_issue IC50=250nM P56817 26878596 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5f01 A 1.52 BS01 5T7 A 1 G74 L91 D93 Y132 D289 G291 T292 T293 G18 L35 D37 Y76 D227 G229 T230 T231 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D227 T230 3.4.23.46 0004190,0006508,0016020 ic50=420nM remove_due_to_license_issue P56817 26878596 504 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVASIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5f02 A 1.43 BS01 5T9 A 1 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A214 G23 C25 E63 G67 G68 L69 M70 A135 M161 D162 H163 A213 Q19 C25 H163 N187 Q19 C25 H163 N186 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 26878596 302 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTSDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 5f04 A 1.84 BS01 5TB A 1 F110 F114 T121 Q125 M142 Y148 T149 N176 N179 E180 L183 F184 W207 F87 F91 T98 Q102 M119 Y125 T126 N153 N156 E157 L160 F161 W184 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 remove_due_to_license_issue P9WMC1 26806381 301 DRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f08 A 1.92 BS01 5TG A 1 L87 W103 I107 F110 W145 Y148 N176 N179 W207 L66 W82 I86 F89 W124 Y127 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=3uM remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f0c A 1.87 BS01 5TE A 1 F110 F114 W145 Y148 T149 N176 N179 E180 L183 W207 F89 F93 W124 Y127 T128 N155 N158 E159 L162 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f0f A 1.76 BS01 5TD A 1 L87 M102 W103 F110 W145 Y148 N176 N179 W207 L66 M81 W82 F89 W124 Y127 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=1uM remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f0h A 1.99 BS01 5TC A 1 L76 V80 L87 M102 F110 W138 M142 W145 Y148 N176 N179 F184 W207 L55 V59 L66 M81 F89 W117 M121 W124 Y127 N155 N158 F163 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=33uM remove_due_to_license_issue P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f1c A 2.9 BS02 ATP A 1 D188 N311 R313 K327 D159 N282 R284 K298 ? 0001614,0004931,0005524,0005886,0007165,0015267,0016020,0033198,0034220,0035590,0046872,0060079,0070588,0098655,0098794 remove_due_to_license_issue G3MM57 26804916 409 LNRLIQLLILGYIIGYVIIYQKGYQQFSTFNAATTTKVKGVVSTKNLSDDAFYPFLSDKTVYKRVWDIADIVVPPEESNQFFVTTNLIITPSQEIKTCPEDPSIKEAHCKSENDTTSCTAGKSIMIGNGVMTGRCVQAAKPQETLHVCEISGWCPVEQDYGPLKDGTPLLSDVQNFTVLIKNYIEFSLFHVRRSNLHDIENSTYLKYCRYHPEKDPHCPVFRIGDMVDAAGEDFDDVAAKGGVIQVLISWDCNLDYDVKYCIPNYSFLRLDDPKTVLAKGWNFRYPKYYNEKERSLVKAYGITFVILVQGRAGKLSPIPIAINIGSGLGLMVVATVLCDLVVL 5f1c A 2.9 BS03 ATP C 1 K66 K68 T206 V207 L208 K37 K39 T177 V178 L179 ? 0001614,0004931,0005524,0005886,0007165,0015267,0016020,0033198,0034220,0035590,0046872,0060079,0070588,0098655,0098794 remove_due_to_license_issue G3MM57 26804916 401 LNRLIQLLILGYIIGYVIIYQKGYQQFSTFNAATTTKVKGVVSTKNLSDDAFYPFLSDKTVYKRVWDIADIVVPPEESNQFFVTTNLIITPSQEIKTCPEDPSIKEAHCKSENDTTSCTAGKSIMIGNGVMTGRCVQAAKPQETLHVCEISGWCPVEQDYGPLKDGTPLLSDVQNFTVLIKNYIEFSLFHVRRSNLHDIENSTYLKYCRYHPEKDPHCPVFRIGDMVDAAGEDFDDVAAKGGVIQVLISWDCNLDYDVKYCIPNYSFLRLDDPKTVLAKGWNFRYPKYYNEKERSLVKAYGITFVILVQGRAGKLSPIPIAINIGSGLGLMVVATVLCDLVVL 5f1c B 2.9 BS01 ATP A 1 K66 K68 T206 L208 K48 K50 T188 L190 ? 0001614,0004931,0005524,0005886,0007165,0015267,0016020,0033198,0034220,0035590,0046872,0060079,0070588,0098655,0098794 remove_due_to_license_issue G3MM57 26804916 409 GSREFDQKIGVLNRLIQLLILGYIIGYVIIYQKGYQQFSTFNAATTTKVKGVVSTKNLSDDAFYPFLSDKTVYKRVWDIADIVVPPEESNQFFVTTNLIITPSQEIKTCPEDPSIKEAHCKSENDTTSCTAGKSIMIGNGVMTGRCVQAAKPQETLHVCEISGWCPVEQDYGPLKDGTPLLSDVQNFTVLIKNYIEFSLFHVRRSNLHDIENSTYLKYCRYHPEKDPHCPVFRIGDMVDAAGEDFDDVAAKGGVIQVLISWDCNLDYDVKYCIPNYSFLRLDDPKTVLAKGWNFRYPKYYNEKERSLVKAYGITFVILVQGRAGKLSPIPIAINIGSGLGLMVVATVLCDLVVLN 5f1c B 2.9 BS04 ATP B 1 D188 N311 R313 K327 D170 N293 R295 K309 ? 0001614,0004931,0005524,0005886,0007165,0015267,0016020,0033198,0034220,0035590,0046872,0060079,0070588,0098655,0098794 remove_due_to_license_issue G3MM57 26804916 407 GSREFDQKIGVLNRLIQLLILGYIIGYVIIYQKGYQQFSTFNAATTTKVKGVVSTKNLSDDAFYPFLSDKTVYKRVWDIADIVVPPEESNQFFVTTNLIITPSQEIKTCPEDPSIKEAHCKSENDTTSCTAGKSIMIGNGVMTGRCVQAAKPQETLHVCEISGWCPVEQDYGPLKDGTPLLSDVQNFTVLIKNYIEFSLFHVRRSNLHDIENSTYLKYCRYHPEKDPHCPVFRIGDMVDAAGEDFDDVAAKGGVIQVLISWDCNLDYDVKYCIPNYSFLRLDDPKTVLAKGWNFRYPKYYNEKERSLVKAYGITFVILVQGRAGKLSPIPIAINIGSGLGLMVVATVLCDLVVLN 5f1h A 1.82 BS01 5U6 A 1 F44 F45 F47 V49 I53 A54 N100 Y106 F23 F24 F26 V28 I32 A33 N79 Y85 ? Kd=14.1nM remove_due_to_license_issue Kd=47nM, IC50=75nM Q9H8M2 26914985 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5f1j A 1.631 BS01 5TO A 1 F110 W145 N176 N179 W207 F89 W124 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=12uM remove_due_to_license_issue Kd=1.2e+4nM P9WMC1 26806381 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGEN 5f1j A 1.631 BS02 5TO A 2 F114 G124 R128 W138 E180 F184 F93 G103 R107 W117 E159 F163 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=12uM remove_due_to_license_issue Kd=1.2e+4nM P9WMC1 26806381 302 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGEN 5f1l A 2.3 BS01 5U2 A 1 H42 F44 F45 F47 V49 I53 Y99 N100 Y106 H21 F23 F24 F26 V28 I32 Y78 N79 Y85 ? ic50=21nM remove_due_to_license_issue IC50=21nM Q9H8M2 26914985 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5f1r A 2.25 BS01 42O A 1 Y62 F67 K122 Y126 I149 W224 C229 Y61 F66 K121 Y125 I148 W216 C221 ? 0003677,0003700,0005829,0006355 Kd=1uM remove_due_to_license_issue IC50=4500nM P22262 26991105 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 5f1r A 2.25 BS02 42O B 1 F131 F134 F130 F133 ? 0003677,0003700,0005829,0006355 Kd=1uM remove_due_to_license_issue IC50=4500nM P22262 26991105 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 5f1r B 2.25 BS01 42O B 1 Q61 K130 F131 S142 Q60 K129 F130 S141 ? 0003677,0003700,0005829,0006355 Kd=1uM remove_due_to_license_issue IC50=4500nM P22262 26991105 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 5f1u A 2.35 BS01 3VN A 1 S51 A52 L54 H59 N84 E88 S50 A51 L53 H58 N83 E87 T47 Y111 Y137 R142 K166 I207 T46 Y110 Y136 R141 K165 I206 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0044281 ic50=400nM remove_due_to_license_issue Q9PPB4 26836694 301 DKNIIIGAMTALITPFKNGKVDEQSYARLIKRQIENGIDAVVPVGTTGESATLTHEEHRTCIEIAVETCKGTKVKVLAGAGSNATHEAVGLAKFAKEHGADGILSVAPFYNKPTQQGLYEHYKAIAQSVDIPVLLYNVPGRTGCEISTDTIIKLFRDCENIYGVKEASGNIDKCVDLLAHEPRMMLISGEDAINYPILSNGGKGVISVTSNLLPDMISALTHFALDENYKEAKKINDELYNINKILFCESNPIPIKTAMYLAGLIESLEFRLPLCSPSKENFAKIEEVMKKYKIKGF 5f1u B 2.35 BS01 3VN A 1 S51 A52 H56 H59 N84 E88 F110 S48 A49 H53 H56 N81 E85 F107 T47 Y111 Y137 R142 K166 I207 T44 Y108 Y134 R139 K163 I204 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0044281 remove_due_to_license_issue Q9PPB4 26836694 301 NIIIGAMTALITPFKNGKVDEQSYARLIKRQIENGIDAVVPVGTTGESATLTHEEHRTCIEIAVETCKGTKVKVLAGAGSNATHEAVGLAKFAKEHGADGILSVAPFYNKPTQQGLYEHYKAIAQSVDIPVLLYNVPGRTGCEISTDTIIKLFRDCENIYGVKEASGNIDKCVDLLAHEPRMMLISGEDAINYPILSNGGKGVISVTSNLLPDMISALTHFALDENYKEAKKINDELYNINKILFCESNPIPIKTAMYLAGLIESLEFRLPLCSPSKENFAKIEEVMKKYKIKGF 5f1v A 2.2 BS01 3VN A 1 K71 T73 K74 K76 G100 D102 K69 T71 K72 K74 G98 D100 T47 Y111 Y137 R142 K166 I207 T45 Y109 Y135 R140 K164 I205 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0044281 Ki~200nM remove_due_to_license_issue Q9PPB4 26836694 301 KNIIIGAMTALITPFKNGKVDEQSYARLIKRQIENGIDAVVPVGTTGESATLTHEEHRTCIEIAVETCKGTKVKVLAGAGSNATHEAVGLAKFAKEHGADGILSVAPYYNKPTQQGLYEHYKAIAQSVDIPVLLYNVPGRTGCEISTDTIIKLFRDCENIYGVKEASGNIDKCVDLLAHEPRMMLISGEDAINYPILSNGGKGVISVTSNLLPDMISALTHFALDENYKEAKKINDELYNINKILFCESNPIPIKTAMYLAGLIESLEFRLPLCSPSKENFAKIEEVMKKYKIKGF 5f1v A 2.2 BS02 3VN A 2 S51 A52 H56 H59 N84 E88 Y110 S49 A50 H54 H57 N82 E86 Y108 T47 Y111 Y137 R142 K166 I207 T45 Y109 Y135 R140 K164 I205 4.3.3.7 0005737,0005829,0008840,0009085,0009089,0016829,0019877,0044281 Ki~200nM remove_due_to_license_issue Q9PPB4 26836694 304 KNIIIGAMTALITPFKNGKVDEQSYARLIKRQIENGIDAVVPVGTTGESATLTHEEHRTCIEIAVETCKGTKVKVLAGAGSNATHEAVGLAKFAKEHGADGILSVAPYYNKPTQQGLYEHYKAIAQSVDIPVLLYNVPGRTGCEISTDTIIKLFRDCENIYGVKEASGNIDKCVDLLAHEPRMMLISGEDAINYPILSNGGKGVISVTSNLLPDMISALTHFALDENYKEAKKINDELYNINKILFCESNPIPIKTAMYLAGLIESLEFRLPLCSPSKENFAKIEEVMKKYKIKGF 5f1x A 1.9 BS01 ATP A 1 G36 T37 T38 Y39 G226 G227 G228 T229 G255 E293 K296 R297 S300 G363 G364 R367 G11 T12 T13 Y14 G199 G200 G201 T202 G228 E266 K269 R270 S273 G336 G337 R340 D34 K96 E201 D224 D9 K69 E174 D197 3.6.4.10 0005524,0140662 Kd=0.000000064M remove_due_to_license_issue P11021 27144892 501 DVGTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDIGGGQTKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLSG 5f1z A 2.65 BS01 5U3 A 1 L903 V911 A928 Y980 V981 P982 G984 L1030 L18 V26 A43 Y84 V85 P86 G88 L134 N1023 A1025 R1027 N1028 D1041 P1064 N127 A129 R131 N132 D145 P168 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue P29597 26701356 1200 ASDPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKSGWKQEIDILRTLYHEHIIKYKGCCEDKSLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHSQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPCEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYH 5f20 A 2.91 BS01 5U4 A 1 L903 G904 E905 G906 I960 Y980 V981 G984 L1030 L16 G17 E18 G19 I64 Y80 V81 G84 L130 N1023 A1025 R1027 N1028 D1041 P1064 N123 A125 R127 N128 D141 P164 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=30nM P29597 26701356 1200 DPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKGWKQEIDILRTLYHEHIIKYKGCCEDSLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHSQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGQGQMTVLRLTELLERGERLPRPDKCPCEVYHLMKNCWETEASFRPTFENLIPILKTVHEKY 5f25 A 1.68 BS01 5TU A 1 F44 F45 V49 I53 Y99 N100 Y106 F23 F24 V28 I32 Y78 N79 Y85 ? Kd=9.1uM remove_due_to_license_issue Kd=9100nM, IC50=9338nM Q9H8M2 26914985 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5f27 A 1.684 BS01 5TT A 1 F110 T121 M142 W145 I146 N176 E180 L183 F83 T94 M115 W118 I119 N149 E153 L156 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 remove_due_to_license_issue P9WMC1 26806381 301 DRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f27 A 1.684 BS02 5TT A 2 G106 F110 Y148 W207 G79 F83 Y121 W180 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 remove_due_to_license_issue P9WMC1 26806381 302 DRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5f29 A 1.821 BS01 2BA A 1 L160 R161 F165 I170 F171 H184 G185 L18 R19 F23 I28 F29 H42 G43 ? 0006813,0008324 remove_due_to_license_issue Q2FZQ4 26171638 301 TSLYEIQMLNYKYENIQLRNFPFGGDIIFVRIIRNNESIVPHGDTQLRYGDRLIVTGAKEYVDELKQELE 5f29 B 1.821 BS01 2BA A 1 R161 F165 I170 F171 P183 H184 G185 R19 F23 I28 F29 P41 H42 G43 ? 0006813,0008324 remove_due_to_license_issue Q2FZQ4 26171638 301 TSLYEIQMLNYKYENIQLRNFPFGGDIIFVRIIRNNESIVPHGDTQLRYGDRLIVTGAKEYVDELKQELEF 5f2f A 1.665 BS01 5U7 A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 ? 0007155,0009289 remove_due_to_license_issue P08191 26812660 201 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 5f2k A 1.6 BS01 SAH A 1 M19 Y24 G64 A66 N70 D98 V99 S133 F134 Y135 S150 W151 M9 Y14 G54 A56 N60 D88 V89 S123 F124 Y125 S140 W141 ? 0008168,0032259 remove_due_to_license_issue B2HHT4 26526103 400 SVVVRPAPMESATYSQSSRLQAAGLSPAITLFEKAAQTVPLPDAPQPVVIADYGVATGHNSLKPMMAAINALRRRIREDRAIMVAHTDVPDNDFTALFRTLADDPDSYLHHDSASFASAVGRSFYTQILPSNTVSLGWSSWAIQWLSRIPAGAPELTDHVQVAYSKDERARAAYAHQAATDWQDFLAFRGRELCPGGRLVVLTMALDEHGHFGYRPMNDALVAALNDQVRDGLLRPEELRRMAIPVVARAEKDLRAPFAPRGWFEGLTIEQLDVFNAEDRFWAAFQSDGDAESFGAQWAGFARAALFPTLAAALDCGTGDPRATAFIEQLEASVADRLASQPEPMRIPLASLVLAKRA 5f2p A 1.8 BS01 5TY A 1 F44 F45 V49 I53 N100 Y106 F23 F24 V28 I32 N79 Y85 ? Kd=37.5uM remove_due_to_license_issue Kd=37500nM, IC50=48900nM Q9H8M2 26914985 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5f2r A 2.15 BS01 ACP A 1 G36 T37 T38 Y39 G226 G227 T229 G255 E293 K296 R297 S300 G363 G364 R367 G10 T11 T12 Y13 G200 G201 T203 G229 E267 K270 R271 S274 G337 G338 R341 D34 K96 E201 D224 D8 K70 E175 D198 3.6.4.10 0005524,0140662 Kd=0.000052M remove_due_to_license_issue P11021 27144892 501 VGTVVGIDLGTTYSCVGVFKNGRVEIIANDQGNRITPSYVAFTPEGERLIGDAAKNQLTSNPENTVFDAKRLIGRTWNDPSVQQDIKFLPFKVVEKKTKPYIQVDIGGGQTKTFAPEEISAMVLTKMKETAEAYLGKKVTHAVVTVPAYFNDAQRQATKDAGTIAGLNVMRIINEPTAAAIAYGLDKREGEKNILVFDLGGGTFDVSLLTIDNGVFEVVATNGDTHLGGEDFDQRVMEHFIKLYKKKTGKDVRKDNRAVQKLRREVEKAKRALSSQHQARIEIESFYEGEDFSETLTRAKFEELNMDLFRSTMKPVQKVLEDSDLKKSDIDEIVLVGGSTRIPKIQQLVKEFFNGKEPSRGINPDEAVAYGAAVQAGVLSG 5f2s A 2.08 BS03 5TZ A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 H276 Y124 Y169 F177 H180 E182 K198 W200 K233 H268 G170 Y177 H188 E190 H276 S288 G162 Y169 H180 E182 H268 S280 1.14.11.66,1.14.11.69 ic50=0.2uM remove_due_to_license_issue IC50=200nM O75164 26741168 403 NPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f2u A 1.85 BS02 FAR C 1 M20 Q78 M19 Q77 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 remove_due_to_license_issue O43924 27063844 701 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAAPESQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5f2w A 2.6 BS03 5UP A 1 Y132 F185 H188 E190 K206 W208 K241 H276 Y124 F177 H180 E182 K198 W200 K233 H268 G170 Y177 H188 E190 H276 S288 G162 Y169 H180 E182 H268 S280 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=104200nM O75164 26741168 403 NPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f32 A 2.05 BS03 5V7 A 1 Y132 Y177 F185 H188 E190 K206 W208 H276 Y122 Y167 F175 H178 E180 K196 W198 H266 G170 Y177 H188 E190 H276 S288 G160 Y167 H178 E180 H266 S278 1.14.11.66,1.14.11.69 ic50=11.5uM remove_due_to_license_issue IC50=11500nM O75164 26741168 403 SARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f37 A 2.22 BS03 N5J A 1 Y132 Y177 F185 H188 K206 W208 K241 H276 Y128 Y173 F181 H184 K202 W204 K237 H272 G170 Y177 H188 E190 H276 S288 G166 Y173 H184 E186 H272 S284 1.14.11.66,1.14.11.69 ic50=1.7uM remove_due_to_license_issue IC50=1700nM O75164 26741168 403 SETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f39 A 2.65 BS03 5UB A 1 Y132 Y177 F185 H188 E190 K206 W208 H276 Y124 Y169 F177 H180 E182 K198 W200 H268 G170 Y177 H188 E190 H276 S288 G162 Y169 H180 E182 H268 S280 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=8000nM O75164 26741168 403 NPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f3c A 2.06 BS03 5U8 A 1 Y132 D135 E169 G170 Y177 F185 H188 E190 K206 W208 K241 H276 Y123 D126 E160 G161 Y168 F176 H179 E181 K197 W199 K232 H267 G170 Y177 H188 E190 H276 S288 G161 Y168 H179 E181 H267 S279 1.14.11.66,1.14.11.69 ic50=0.9uM remove_due_to_license_issue IC50=900nM O75164 26741168 403 PSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f3e A 2.16 BS03 5UO A 1 Y132 D135 Y175 Y177 F185 H188 E190 K206 W208 K241 Y127 D130 Y160 Y162 F170 H173 E175 K191 W193 K226 Y177 H188 E190 H276 S288 Y162 H173 E175 H261 S273 1.14.11.66,1.14.11.69 ic50=0.138uM remove_due_to_license_issue IC50=138nM O75164 26741168 403 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f3g A 2.5 BS03 5UL A 1 Y132 D135 G170 Y177 F185 H188 E190 K206 W208 H276 Y125 D128 G158 Y165 F173 H176 E178 K194 W196 H264 G170 Y177 H188 E190 H276 S288 G158 Y165 H176 E178 H264 S276 1.14.11.66,1.14.11.69 ic50=0.126uM remove_due_to_license_issue IC50=126nM O75164 26741168 403 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 5f3i A 2.24 BS03 5UJ A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 H276 Y127 Y165 F173 H176 E178 K194 W196 K229 H264 G170 Y177 H188 E190 H276 S288 G158 Y165 H176 E178 H264 S276 1.14.11.66,1.14.11.69 ic50=0.08uM remove_due_to_license_issue IC50=80nM O75164 26741168 403 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 5f3t A 2.05 BS03 5UH A 1 L511 C709 H711 R729 Y766 T794 S796 H798 A799 W803 L213 C411 H413 R431 Y468 T496 S498 H500 A501 W505 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 Kd=210uM remove_due_to_license_issue Q6YMS4 26872970 1003 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAADSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 5f3z A 2.0 BS03 5V5 A 1 L511 C709 R729 M761 T794 S796 H798 A799 W803 L213 C411 R431 M463 T496 S498 H500 A501 W505 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 Kd=29uM remove_due_to_license_issue Q6YMS4 26872970 1003 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAADSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 5f41 A 2.0 BS03 5V6 A 1 L511 C709 H711 R729 M761 T794 S796 H798 A799 W803 L213 C411 H413 R431 M463 T496 S498 H500 A501 W505 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 Kd=67uM remove_due_to_license_issue Q6YMS4 26872970 1003 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAADSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 5f4l A 2.7 BS01 5VE A 1 S256 E370 S375 F376 F382 N425 M426 W427 G473 M475 S135 E224 S229 F230 F236 N276 M277 W278 G318 M320 ? 0019031 remove_due_to_license_issue C6G099 26985324 501 KTTLFCASDAKAYEKEVHNVWATHACVPTDPNPQEMVLANVTENFNMWKNDMVEQMHEDIISLWDESLKPCVKLTGGSAITQACPKVSFDPIPLHYCAPAGFAILKCNNKTFNGTGPCRNVSTVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNESVNIVCTRPNNIRQAHCNINESKWNNTLQKVGEELAKHFPSKTIKFEPSSGGDLEITTHSFNCRGEFFYCNTSDLFNGTYRNGTYNHTGRSSNGTITLQCKIKQIINMWQEVGRAIYAPPIEGEITCNSNITGLLLLRDDTETFRPGGGDMRDNWRSELYKYKVVEI 5f4n A 1.91 BS01 5UY A 1 L15 A36 K38 V68 L84 E85 Y86 C87 E91 E134 L137 S147 D148 L11 A32 K34 V55 L71 E72 Y73 C74 E78 E121 L124 S134 D135 D130 K132 E134 N135 D148 T170 D117 K119 E121 N122 D135 T157 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=2.2nM remove_due_to_license_issue IC50=2.00nM O14757 27167172 301 FVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 5f4n A 1.91 BS02 5UY A 2 W9 V35 Y71 F83 W5 V31 Y58 F70 D130 K132 E134 N135 D148 T170 D117 K119 E121 N122 D135 T157 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=2.2nM remove_due_to_license_issue IC50=2.00nM O14757 27167172 302 FVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 5f4p D 2.6 BS01 5VG D 1 E370 I371 S375 F376 F382 N425 M426 W427 E429 G431 G473 M475 E224 I225 S229 F230 F236 N276 M277 W278 E280 G282 G318 M320 ? 0019031 remove_due_to_license_issue C6G099 26985324 507 KTTLFCASDAKAYEKEVHNVWATHACVPTDPNPQEMVLANVTENFNMWKNDMVEQMHEDIISLWDESLKPCVKLTGGSAITQACPKVSFDPIPLHYCAPAGFAILKCNNKTFNGTGPCRNVSTVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNESVNIVCTRPNNIRQAHCNINESKWNNTLQKVGEELAKHFPSKTIKFEPSSGGDLEITTHSFNCRGEFFYCNTSDLFNGTYRNGTYNHTGRSSNGTITLQCKIKQIINMWQEVGRAIYAPPIEGEITCNSNITGLLLLRDDTETFRPGGGDMRDNWRSELYKYKVVE 5f4r A 2.8 BS01 5VF A 1 E370 S375 F376 F382 N425 M426 W427 V430 G431 G473 M475 E224 S229 F230 F236 N276 M277 W278 V281 G282 G318 M320 ? 0019031 remove_due_to_license_issue C6G099 26985324 508 KTTLFCASDAKAYEKEVHNVWATHACVPTDPNPQEMVLANVTENFNMWKNDMVEQMHEDIISLWDESLKPCVKLTGGSAITQACPKVSFDPIPLHYCAPAGFAILKCNNKTFNGTGPCRNVSTVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNESVNIVCTRPNNIRQAHCNINESKWNNTLQKVGEELAKHFPSKTIKFEPSSGGDLEITTHSFNCRGEFFYCNTSDLFNGTYRNGTYNHTGRSSNGTITLQCKIKQIINMWQEVGRAIYAPPIEGEITCNSNITGLLLLRDDTETFRPGGGDMRDNWRSELYKYKVVE 5f4u A 3.1 BS01 5VH A 1 V255 S256 S375 F376 N425 M426 W427 E429 V430 G431 G473 M475 V134 S135 S229 F230 N276 M277 W278 E280 V281 G282 G318 M320 ? 0019031 remove_due_to_license_issue C6G099 26985324 507 KTTLFCASDAKAYEKEVHNVWATHACVPTDPNPQEMVLANVTENFNMWKNDMVEQMHEDIISLWDESLKPCVKLTGGSAITQACPKVSFDPIPLHYCAPAGFAILKCNNKTFNGTGPCRNVSTVQCTHGIKPVVSTQLLLNGSLAEEEIIIRSENLTNNAKTIIVHLNESVNIVCTRPNNIRQAHCNINESKWNNTLQKVGEELAKHFPSKTIKFEPSSGGDLEITTHSFNCRGEFFYCNTSDLFNGTYRNGTYNHTGRSSNGTITLQCKIKQIINMWQEVGRAIYAPPIEGEITCNSNITGLLLLRDDTETFRPGGGDMRDNWRSELYKYKVVE 5f5h A 2.23 BS01 rna C 0 R188 R190 R219 S238 K239 T240 Q247 Y250 R251 S253 F255 K259 R11 R13 R42 S61 K62 T63 Q70 Y73 R74 S76 F78 K82 2.3.2.27 remove_due_to_license_issue Q4VGL6 27010430 2 ~ 22 QLSSNLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRTYEALRREHDSQIVQIAMEAGLRIAPDQWSSLLYGDQSHKSHMQSIIDKLQ 5f5h B 2.23 BS01 rna D 0 R190 R219 S238 K239 T240 Q247 Y250 R251 S253 F255 V257 K259 R17 R46 S65 K66 T67 Q74 Y77 R78 S80 F82 V84 K86 2.3.2.27 remove_due_to_license_issue Q4VGL6 27010430 2 ~ 22 QNPQQLSSNLWAAVRARGCQFLGPAMQEEALKLVLLALEDGSALSRKVLVLFVVQRLEPRFPQASKTSIGHVVQLLYRASCFKVTKRDEDSSLMQLKEEFRTYEALRREHDSQIVQIAMEAGLRIAPDQWSSLLYGDQSHKSHMQSIIDKLQ 5f5i A 2.63 BS02 5V1 A 1 Y132 G170 Y175 Y177 F185 H188 E190 K206 W208 S288 Y129 G167 Y172 Y174 F182 H185 E187 K203 W205 S285 G170 Y177 H188 E190 H276 S288 G167 Y174 H185 E187 H273 S285 1.14.11.66,1.14.11.69 remove_due_to_license_issue O75164 26741168 504 ESETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAE 5f5z A 1.76 BS01 5VY A 1 W81 P82 F83 V87 D88 K91 L92 L94 N140 I146 W40 P41 F42 V46 D47 K50 L51 L53 N99 I105 ? Kd=86nM remove_due_to_license_issue O60885 28336808 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5f60 A 1.35 BS01 5VZ A 1 W81 P82 F83 V87 L92 L94 N140 I146 W40 P41 F42 V46 L51 L53 N99 I105 ? Kd=43nM remove_due_to_license_issue O60885 28336808 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5f61 A 1.45 BS01 5W0 A 1 W81 P82 F83 Q85 V87 D88 K91 L92 L94 N140 I146 W40 P41 F42 Q44 V46 D47 K50 L51 L53 N99 I105 ? Kd=35nM remove_due_to_license_issue O60885 28336808 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5f62 A 1.35 BS01 5W1 A 1 W81 P82 F83 V87 L92 L94 N140 I146 W40 P41 F42 V46 L51 L53 N99 I105 ? Kd=6.8nM remove_due_to_license_issue O60885 28336808 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5f63 A 1.45 BS01 5W2 A 1 W81 P82 F83 V87 L92 L94 N140 I146 W40 P41 F42 V46 L51 L53 N99 I105 ? Kd=12nM remove_due_to_license_issue O60885 28336808 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5f6d A 1.553 BS01 5VJ A 1 E42 C43 K59 L60 E41 C42 K58 L59 C93 C92 2.3.2.- 0000122,0000795,0001221,0003723,0005515,0005524,0005634,0005635,0005643,0005654,0005737,0005829,0006511,0007059,0007084,0008134,0016605,0016740,0016925,0019787,0019789,0019899,0030335,0032446,0036211,0044388,0045892,0048471,0051168,0051301,0061656,0071535,0106068,1903755,1990234 remove_due_to_license_issue P63279 27038327 201 SGIALSRLAQERKAWRKDHPFGFVAVPTKNPDGTMNLMNWECAIPGAAGTPWAGGLFKLRMLFKDDYPSSPPKCKFEPPLFHPNVYPSGTVCLSILEEDKDWRPAITIKQILLGIQELLNEPNIQDPAQAEAYTIYCQNRVEYEKRVRAQAKKFAP 5f6u A 1.552 BS01 5VK A 1 E42 C43 K59 L60 R61 E41 C42 K58 L59 R60 C93 C92 2.3.2.- 0000122,0000795,0001221,0003723,0005515,0005524,0005634,0005635,0005643,0005654,0005737,0005829,0006511,0007059,0007084,0008134,0016605,0016740,0016925,0019787,0019789,0019899,0030335,0032446,0036211,0044388,0045892,0048471,0051168,0051301,0061656,0071535,0106068,1903755,1990234 ic50=3mM remove_due_to_license_issue P63279 27038327 201 SGIALSRLAQERKAWRKDHPFGFVAVPTKNPDGTMNLMNWECAIPGAAGTPWAGGLFKLRMLFKDDYPSSPPKCKFEPPLFHPNVYPSGTVCLSILEEDKDWRPAITIKQILLGIQELLNEPNIQDPAQAEAYTIYCQNRVEYEKRVRAQAKKFAP 5f6v A 1.492 BS01 5VL A 1 E42 C43 K59 L60 R61 E41 C42 K58 L59 R60 C93 C92 2.3.2.- 0000122,0000795,0001221,0003723,0005515,0005524,0005634,0005635,0005643,0005654,0005737,0005829,0006511,0007059,0007084,0008134,0016605,0016740,0016925,0019787,0019789,0019899,0030335,0032446,0036211,0044388,0045892,0048471,0051168,0051301,0061656,0071535,0106068,1903755,1990234 ic50=5.8mM remove_due_to_license_issue P63279 27038327 201 SGIALSRLAQERKAWRKDHPFGFVAVPTKNPDGTMNLMNWECAIPGAAGTPWAGGLFKLRMLFKDDYPSSPPKCKFEPPLFHPNVYPSGTVCLSILEEDKDWRPAITIKQILLGIQELLNEPNIQDPAQAEAYTIYCQNRVEYEKRVRAQAKKFAP 5f74 A 2.35 BS02 AMP A 1 K51 R58 K122 R129 N175 K50 R57 K119 R126 N172 ? 0004860,0004864,0005515,0005634,0005737,0005829,0006605,0019899,0019904,0042470,0042802,0042826,0045184,0045744,0048471,0050815,0051219,0051220 Kd=7.6uM remove_due_to_license_issue Q9CQV8 26984404 301 TMDKSELVQKAKLAEQAERYDDMAAAMKAVTEQGHELSNEERNLLSVAYKNVVGARRSSWRVISSIEQKTNEKKQQMGKEYREKIEAELQDICNDVLELLDKYLILNATQAESKVFYLKMKGDYFRYLSEVASGENKQTTVSNSQQAYQEAFEISKKEMQPTHPIRLGLALNFSVFYYEILNSPEKACSLAKTAFDEAIAELDTLNEESYKDSTLIMQLLRDNLTLWTS 5f8y A 1.7 BS01 X6X A 1 N27 H64 Y66 G67 G68 H81 D83 H85 N26 H63 Y65 G66 G67 H80 D82 H84 ? 0030246 Kd=57uM remove_due_to_license_issue H2FH31 27010847 201 TTFLIKHKASGKFLHPYGGSSNPANNTKLVLHSDIHERMYFQFDVVDERWGYIKHVASGKIVHPYGGQANPPNETNMVLHQDRHDRALFAMDFFNDNIMHKGGKYIHPKGGSPNPPNNTETVIHGDKHAAMEFIFVSPKNKDKRVLVYA 5f8y A 1.7 BS02 X6X A 2 E75 H108 K110 G111 G112 H125 D127 H129 E74 H107 K109 G110 G111 H124 D126 H128 ? 0030246 Kd=57uM remove_due_to_license_issue H2FH31 27010847 202 TTFLIKHKASGKFLHPYGGSSNPANNTKLVLHSDIHERMYFQFDVVDERWGYIKHVASGKIVHPYGGQANPPNETNMVLHQDRHDRALFAMDFFNDNIMHKGGKYIHPKGGSPNPPNNTETVIHGDKHAAMEFIFVSPKNKDKRVLVYA 5f8y A 1.7 BS03 X6X A 3 H16 Y18 G19 G20 H33 D35 H37 N119 H15 Y17 G18 G19 H32 D34 H36 N118 ? 0030246 Kd=57uM remove_due_to_license_issue H2FH31 27010847 203 TTFLIKHKASGKFLHPYGGSSNPANNTKLVLHSDIHERMYFQFDVVDERWGYIKHVASGKIVHPYGGQANPPNETNMVLHQDRHDRALFAMDFFNDNIMHKGGKYIHPKGGSPNPPNNTETVIHGDKHAAMEFIFVSPKNKDKRVLVYA 5f90 A 1.64 BS01 GLA C 1 H16 Y18 G19 G20 D35 H37 N119 H16 Y18 G19 G20 D35 H37 N119 ? 0030246 remove_due_to_license_issue H2FH31 27010847 3 MTTFLIKHKASGKFLHPYGGSSNPANNTKLVLHSDIHERMYFQFDVVDERWGYIKHVASGKIVHPYGGQANPPNETNMVLHQDRHDRALFAMDFFNDNIMHKGGKYIHPKGGSPNPPNNTETVIHGDKHAAMEFIFVSPKNKDKRVLVYA 5f90 A 1.64 BS02 GLA D 1 N27 H64 Y66 G67 G68 D83 H85 N27 H64 Y66 G67 G68 D83 H85 ? 0030246 remove_due_to_license_issue H2FH31 27010847 2 MTTFLIKHKASGKFLHPYGGSSNPANNTKLVLHSDIHERMYFQFDVVDERWGYIKHVASGKIVHPYGGQANPPNETNMVLHQDRHDRALFAMDFFNDNIMHKGGKYIHPKGGSPNPPNNTETVIHGDKHAAMEFIFVSPKNKDKRVLVYA 5f91 A 1.998 BS01 5WJ A 1 L303 T304 L429 R432 L291 T292 L409 R412 T186 H187 K324 E331 T174 H175 K304 E311 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 Ki=3.2uM remove_due_to_license_issue P9WN93 27325754 501 NYRIEHEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 5f91 A 1.998 BS02 5WJ C 1 A307 N394 H397 R400 L401 R432 A295 N374 H377 R380 L381 R412 T186 H187 K324 E331 T174 H175 K304 E311 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 Ki=3.2uM remove_due_to_license_issue P9WN93 27325754 501 NYRIEHEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 5f91 C 1.998 BS01 5WJ A 1 A307 H397 R400 L401 R432 A299 H379 R382 L383 R414 T186 H187 E331 T178 H179 E313 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 Ki=3.2uM remove_due_to_license_issue P9WN93 27325754 501 NYRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKA 5f91 C 1.998 BS02 5WJ C 1 L303 T304 L429 R432 L295 T296 L411 R414 T186 H187 E331 T178 H179 E313 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 Ki=3.2uM remove_due_to_license_issue P9WN93 27325754 501 NYRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKA 5f94 A 2.51 BS01 3UO A 1 A83 K85 Y134 V135 R141 L188 D200 A48 K50 Y99 V100 R106 L153 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=3.4nM P49841 26751161 401 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPH 5f95 A 2.525 BS01 3UP A 1 A83 K85 V135 L188 D200 A48 K50 V100 L153 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue P49841 26751161 401 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 5f98 A 3.28 BS01 rna B 0 N298 Q299 I300 S325 G326 T347 Q349 I350 K379 Q507 E510 R546 K635 T636 R637 T662 G663 T697 S698 H830 F853 S854 K858 K888 K909 N59 Q60 I61 S86 G87 T108 Q110 I111 K140 Q260 E263 R299 K388 T389 R390 T415 G416 T425 S426 H558 F581 S582 K586 K616 K637 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 25 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f98 C 3.28 BS01 rna D 0 N298 Q299 I300 S325 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 R546 K635 T636 R637 T662 T697 S698 N720 H830 F853 K858 I875 K888 S906 K909 N59 Q60 I61 S86 G87 T108 Q110 K140 Q141 H142 Q259 E262 Q263 R298 K387 T388 R389 T414 T423 S424 N446 H556 F579 K584 I601 K614 S632 K635 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 25 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRIDKFKYIIAQLMRDTESLAKRICKDLREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f98 E 3.28 BS01 rna F 0 N298 I300 S325 G326 T347 Q349 I350 K379 Q380 Q507 K635 T636 R637 T662 T697 S698 K750 H830 F853 S854 K858 K888 S906 W908 N57 I59 S84 G85 T106 Q108 I109 K138 Q139 Q255 K381 T382 R383 T408 T416 S417 K469 H549 F572 S573 K577 K607 S625 W627 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 25 KPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRIDKFKYIIAQLMRDTESLAKRICKREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f98 G 3.28 BS01 rna H 0 Q299 I300 G326 T347 Q349 I350 K379 Q380 Q507 Q511 K518 R546 K635 T636 R637 G663 R664 T697 S698 N720 H830 F853 S854 K858 K861 K888 K907 W908 K909 Q60 I61 G87 T108 Q110 I111 K140 Q141 Q260 Q264 K271 R299 K388 T389 R390 G416 R417 T425 S426 N448 H555 F578 S579 K583 K586 K613 K632 W633 K634 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 25 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f98 I 3.28 BS01 rna J 0 N298 Q299 I300 S325 G326 T347 Q349 I350 K379 Q380 H381 Q507 V514 R546 K635 T636 R637 T697 S698 N720 H830 F853 K858 K861 I875 K888 W908 N59 Q60 I61 S86 G87 T108 Q110 I111 K140 Q141 H142 Q263 V270 R302 K391 T392 R393 T426 S427 N449 H555 F578 K583 K586 I600 K613 W633 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 25 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLENNREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f98 K 3.28 BS01 rna L 0 N298 Q299 I300 S325 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 V514 R546 K635 T636 R637 G663 R664 T697 S698 N720 C829 H830 F853 I875 K888 S906 N58 Q59 I60 S85 G86 T107 Q109 K139 Q140 H141 Q260 E263 Q264 V267 R299 K383 T384 R385 G411 R412 T420 S421 N443 C551 H552 F575 I597 K610 S628 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 25 FKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLNREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVREIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9b B 2.25 BS01 5VN B 1 G284 C285 R288 I326 Y327 L330 I341 S342 F363 M364 G62 C63 R66 I104 Y105 L108 I119 S120 F140 M141 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 27283034 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIY 5f9e A 2.0 BS01 5VS A 1 L386 G387 F391 V394 A407 K409 T442 M458 E459 Y460 L461 N509 L511 D522 F664 L13 G14 F18 V21 A34 K36 T69 M85 E86 Y87 L88 N136 L138 D149 F291 D504 K506 D508 N509 D522 T542 D131 K133 D135 N136 D149 T169 2.7.11.13 0004672,0004674,0004697,0005524,0006468 ic50=0.46nM remove_due_to_license_issue IC50=16nM Q04759 27117263 1001 KLKIEDFELHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNEFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPPFRPKVKSPFDCSNFDKEFLNEKPRLSFADRALINSMDQNMFRNFSFMNPGMERLISHHH 5f9f A 2.601 BS01 rna B 0 N298 Q299 I300 S325 G326 T347 Q349 K379 Q380 Q507 E510 Q511 K518 R546 K635 T636 R637 T662 G663 T667 N668 T697 S698 N720 C829 H830 F853 K858 I875 V886 K888 N59 Q60 I61 S86 G87 T108 Q110 K140 Q141 Q260 E263 Q264 K271 R299 K388 T389 R390 T415 G416 T420 N421 T450 S451 N473 C580 H581 F604 K609 I626 V637 K639 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 1 ~ 24 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKTNQNTGMTLPAQKCILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9f C 2.601 BS01 rna D 0 N298 I300 S325 G326 T347 Q349 K379 Q380 Q507 E510 K518 R546 K635 T636 R637 T662 G663 R664 T667 N668 T697 S698 N720 K750 H830 F853 K858 I875 V886 K888 W908 K909 N58 I60 S85 G86 T107 Q109 K139 Q140 Q257 E260 K268 R296 K385 T386 R387 T412 G413 R414 T417 N418 T447 S448 N470 K500 H576 F599 K604 I621 V632 K634 W654 K655 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 1 ~ 24 FKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDEFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKTNQNTGMTLPAQKCILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9f E 2.601 BS01 rna F 0 N298 I300 S325 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 V514 R546 K635 T636 R637 T662 G663 T667 N668 T697 S698 V718 N720 K750 H830 F853 K858 I875 V886 K888 N57 I59 S84 G85 T106 Q108 K138 Q139 H140 Q257 E260 Q261 V264 R296 K385 T386 R387 T412 G413 T417 N418 T447 S448 V468 N470 K500 H580 F603 K608 I625 V636 K638 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 1 ~ 24 KPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKTNQNTGMTLPAQKCILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9f G 2.601 BS01 rna H 0 N298 Q299 I300 S325 G326 T347 Q349 K379 Q380 Q507 K508 E510 Q511 R546 K635 T636 R637 T662 G663 R664 T667 N668 T697 S698 K750 H830 F853 K858 I875 V886 K888 W908 K909 N59 Q60 I61 S86 G87 T108 Q110 K140 Q141 Q258 K259 E261 Q262 R297 K386 T387 R388 T413 G414 R415 T418 N419 T448 S449 K501 H577 F600 K605 I622 V633 K635 W655 K656 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 1 ~ 24 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKTNQNTGMTLPAQKCILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9f I 2.601 BS01 rna J 0 N298 I300 S325 G326 T347 Q349 I350 K379 Q380 Q507 E510 Q511 R546 K635 T636 R637 T662 G663 R664 T667 N668 T697 S698 V718 N720 K750 H830 F853 K858 I875 V886 K888 N59 I61 S86 G87 T108 Q110 I111 K140 Q141 Q261 E264 Q265 R300 K389 T390 R391 T416 G417 R418 T421 N422 T451 S452 V472 N474 K504 H582 F605 K610 I627 V638 K640 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 1 ~ 24 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLEREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKTNQNTGMTLPAQKCILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9f K 2.601 BS01 rna L 0 N298 I300 S325 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 K518 R546 K635 T636 R637 T662 G663 R664 T667 N668 T697 S698 N720 K750 H830 K851 F853 K858 I875 V886 K888 W908 N57 I59 S84 G85 T106 Q108 K138 Q139 H140 Q258 E261 Q262 K269 R297 K386 T387 R388 T413 G414 R415 T418 N419 T448 S449 N471 K501 H579 K600 F602 K607 I624 V635 K637 W657 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 1 ~ 24 KPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKTNQNTGMTLPAQKCILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 5f9h A 3.1 BS01 rna B 0 I300 G326 T347 Q349 K379 Q380 H381 Q507 K508 E510 Q511 R546 K635 T636 R637 G663 T697 S698 V718 N720 S854 K888 I60 G86 T107 Q109 K139 Q140 H141 Q259 K260 E262 Q263 R298 K386 T387 R388 G414 T423 S424 V444 N446 S578 K612 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 24 FKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDLREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9h C 3.1 BS01 rna D 0 Q299 I300 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 R546 K635 T636 R637 G663 T697 S698 V718 N720 K888 K907 Q59 I60 G86 T107 Q109 K139 Q140 H141 Q258 E261 Q262 R297 K386 T387 R388 G414 T428 S429 V449 N451 K613 K632 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 24 FKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKDREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9h E 3.1 BS01 rna F 0 I300 S325 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 R546 K635 T636 R637 G663 T697 S698 V718 N720 F853 K888 I59 S84 G85 T106 Q108 K138 Q139 H140 Q254 E257 Q258 R293 K378 T379 R380 G406 T415 S416 V436 N438 F570 K605 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 24 KPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRIDKFKYIIAQLMRDTESLAKRICREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQEPKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATVQTLYSKWKDFHFEKIPFDPAE 5f9h G 3.1 BS01 rna H 0 I300 G326 T347 Q349 K379 Q380 H381 Q507 K508 E510 Q511 R546 K635 T636 R637 T662 G663 T697 S698 N720 K888 S906 I61 G87 T108 Q110 K140 Q141 H142 Q258 K259 E261 Q262 R297 K386 T387 R388 T413 G414 T432 S433 N455 K619 S637 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 24 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRISDKFKYIIAQLMRDTESLAKRICKREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAGFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRILDAFKASGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5f9h I 3.1 BS01 rna J 0 N298 Q299 I300 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 R546 K635 T636 R637 G663 R664 T697 S698 N720 K750 F853 S854 K888 N59 Q60 I61 G87 T108 Q110 K140 Q141 H142 Q255 E258 Q259 R294 K382 T383 R384 G410 R411 T421 S422 N444 K474 F574 S575 K609 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 24 PFKPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRIDKFKYIIAQLMRDTESLAKRICKDEFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAAFDEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGRGGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAEM 5f9h K 3.1 BS01 rna L 0 I300 S325 G326 T347 Q349 K379 Q380 H381 Q507 E510 Q511 V514 R546 K635 T636 R637 G663 T697 V718 N720 S854 K888 I59 S84 G85 T106 Q108 K138 Q139 H140 Q253 E256 Q257 V260 R292 K379 T380 R381 G407 T415 V436 N438 S569 K603 3.6.4.13 0003676,0005524 remove_due_to_license_issue O95786 26733676 2 ~ 24 KPRNYQLELALPAMKGKNTIICAPTGCGKTFVSLLICEHHLKKFPQGQKGKVVFFANQIPVYEQQKSVFSKYFERHGYRVTGISGATAENVPVEQIVENNDIIILTPQILVNNLKKGTIPSLSIFTLMIFDECHNTSKQHPYNMIMFNYLDQKLGGSSGPLPQVIGLTASVGVGDAKNTDEALDYICKLCASLDASVIATVKHNLEELEQVVYKPQKFFRKVESRIDKFKYIIAQLMRDTESLAKRIREFGTQKYEQWIVTVQKACMVFQMPDKDEESRICKALFLYTSHLRKYNDALIISEHARMKDALDYLKDFFSNVRAADEIEQDLTQRFEEKLQELESVSRDPSNENPKLEDLCFILQEEYHLNPETITILFVKTRALVDALKNWIEGNPKLSFLKPGILTGDHNILIATSVADEGIDIAQCNLVILYEYVGNVIKMIQTRGRGRARGSKCFLLTSNAGVIEKEQINMYKEKMMNDSILRLQTWDEAVFREKILHIQTHEKFIRDSQKPVPDKENKKLLCRKCKALACYTADVRVIEECHYTVLGDAFKECFVSRPHPKPKQFSSFEKRAKIFCARQNCSHDWGIHVKYKTFEIPVIKIESFVVEDIATGVQTLYSKWKDFHFEKIPFDPAE 5fa7 A 1.67 BS01 5VR A 1 S70 N104 S130 N132 N170 T235 G236 S237 S44 N78 S104 N106 N144 T209 G210 S211 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9EXV5 26731698 301 TADVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTD 5fah A 1.1 BS01 5VT A 1 H41 C42 H57 F151 A190 N192 G193 S195 W215 G216 C220 H25 C26 H41 F130 A165 N167 G168 S170 W186 G187 C191 H57 D102 N192 G193 D194 S195 G196 H41 D83 N167 G168 D169 S170 G171 3.4.21.117 0001533,0002803,0004222,0004252,0005576,0005615,0006508,0008233,0008236,0008544,0016787,0022617,0030141,0051604,0097209 ic50=0.7uM remove_due_to_license_issue P49862 27775713 302 IIDGAPCARGSHPWQVALLSGNQLHCGGVLVNERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNSQARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVNSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCKFTKWINDTMKKHR 5fao A 3.01 BS01 5VW A 1 S70 N104 S130 N132 P167 N170 T216 T235 S237 S43 N77 S103 N105 P140 N143 T189 T208 S210 S70 K73 S130 E166 K234 S237 S43 K46 S103 E139 K207 S210 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9EXV5 26731698 301 ADVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTD 5fap B 2.7 BS01 602 B 1 S70 N104 S130 N132 P167 N170 T235 G236 S237 S42 N76 S102 N104 P139 N142 T207 G208 S209 S70 K73 S130 E166 K234 S237 S42 K45 S102 E138 K206 S209 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9EXV5 26731698 301 DVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTD 5faq A 1.96 BS01 5VW A 1 S70 D101 I102 S118 T209 G210 Y211 R250 S46 D77 I78 S94 T185 G186 Y187 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 remove_due_to_license_issue Q6XEC0 26731698 305 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5fas A 1.74 BS01 5VR A 1 S70 W105 S118 V120 T209 G210 Y211 T213 R214 R250 S47 W82 S95 V97 T186 G187 Y188 T190 R191 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 remove_due_to_license_issue Q6XEC0 26731698 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5fat A 2.09 BS01 602 A 1 S70 S118 V120 T209 G210 Y211 R214 R250 S48 S96 V98 T187 G188 Y189 R192 R228 S70 K73 S118 Y123 W157 Y211 S48 K51 S96 Y101 W135 Y189 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 remove_due_to_license_issue Q6XEC0 26731698 301 KEWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5fb7 A 1.5 BS01 ACD A 1 F25 L47 I83 N109 S121 S140 I147 F19 L41 I77 N103 S115 S134 I141 ? Kd=0.000000064M remove_due_to_license_issue A0A093VKV7 28111099 201 DISAFQKVIQDISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQILLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAFAGT 5fb7 A 1.5 BS02 ACD A 2 L72 V76 L79 S136 S140 L66 V70 L73 S130 S134 ? Kd=0.000000064M remove_due_to_license_issue A0A093VKV7 28111099 202 DISAFQKVIQDISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQILLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAFAGT 5fb7 C 1.5 BS01 ACD C 1 F25 L40 L47 I83 N109 Q113 A117 L120 S121 S140 F23 L38 L45 I81 N107 Q111 A115 L118 S119 S138 ? Kd=0.000000064M remove_due_to_license_issue A0A093VKV7 28111099 201 KVKRDISAFQKVIQDISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQILLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAFAGT 5fb7 C 1.5 BS02 ACD C 2 I15 V76 V124 S136 S140 I143 I13 V74 V122 S134 S138 I141 ? Kd=0.000000064M remove_due_to_license_issue A0A093VKV7 28111099 202 KVKRDISAFQKVIQDISLAVNKFNVDIERYVGGDASHLLADGNVLIKATLDGVQSLQNEPPLSSMEALALVGPVQDLSNQILLAIQNLIDKKEPLVQAGFGGKVENNLRQQEEAAQKLSELVSTKVPHELADISRQLSDGIAAGIKKGIDAFAGT 5fbe A 1.43 BS01 5W5 A 1 L41 C42 H57 C58 R151 S190 C191 K192 G193 S195 S215 R218 C220 L25 C26 H41 C42 R137 S178 C179 K180 G181 S183 S199 R202 C204 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=14uM remove_due_to_license_issue IC50=14000nM P00746 27775713 302 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 5fbi A 1.47 BS01 5WD A 1 C191 K192 S195 S217 R218 C179 K180 S183 S201 R202 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=1600uM remove_due_to_license_issue Kd=1600000nM P00746 27775713 302 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 5fbn C 1.8 BS01 5WF C 1 L408 V416 A428 K430 F442 M449 L460 I472 T474 M477 C481 N484 L528 S538 D539 F540 L542 L14 V22 A34 K36 F48 M55 L66 I78 T80 M83 C87 N90 L134 S144 D145 F146 L148 N526 D539 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.27nM remove_due_to_license_issue IC50=8.0nM, EC50=<10.00nM Q06187 26985298 701 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 5fbo A 1.894 BS01 5WH A 1 L408 V416 A428 K430 E445 M449 I472 T474 M477 G480 C481 N484 L528 D539 L542 L17 V25 A37 K39 E54 M58 I81 T83 M86 G89 C90 N93 L137 D148 L151 D521 A523 R525 N526 D539 F559 D130 A132 R134 N135 D148 F155 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.31nM remove_due_to_license_issue IC50=0.300000nM Q06187 26985298 1001 YGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 5fck A 1.86 BS01 5WC A 1 H40 L41 C42 H57 C58 R151 C191 K192 G193 S195 S215 G216 S217 R218 C220 H24 L25 C26 H41 C42 R133 C175 K176 G177 S179 S195 G196 S197 R198 C200 H57 D102 K192 G193 D194 S195 G196 H41 D85 K176 G177 D178 S179 G180 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=0.006uM remove_due_to_license_issue IC50=10nM P00746 27775713 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLDGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLAS 5fcw A 1.979 BS01 5YA A 1 Y100 D101 H142 H143 D178 H180 F208 Y306 Y87 D88 H129 H130 D165 H167 F195 Y293 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=0.3uM remove_due_to_license_issue IC50=300nM Q9BY41 27374062 401 SLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 5fcw A 1.979 BS03 5YA B 3 Y100 F152 Y87 F139 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 ic50=0.3uM remove_due_to_license_issue IC50=300nM Q9BY41 27374062 405 SLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 5fcz A 2.45 BS01 TNX A 1 R162 D313 E314 W344 W361 Y393 D395 W408 W442 E444 R155 D306 E307 W337 W354 Y386 D388 W401 W435 E437 D313 E314 D306 E307 3.2.1.52 0004553,0004563,0005975,0016020,0016231,0016798,0030203 Ki=68uM remove_due_to_license_issue O85361 27253678 601 DRKAPVRPTPLDRVIPAPASVDPGGAPYRITRGTHIRVDDSREARRVGDYLADLLRPATGYRLPVTAHGHGGIRLRLAGGPYGDEGYRLDSGPAGVTITARKAAGLFHGVQTLRQLLPPAVEKDSAQPGPWLVAGGTIEDTPRYAWRSAMLDVSRHFFGVDEVKRYIDRVARYKYNKLHLHLSDDQGWRIAIDSWPRLATYGGSTEVGGGPGGYYTKAEYKEIVRYAASRHLEVVPEIDMPGHTNAALASYAELNCDGVAPPLYTGTKVGFSSLCVDKDVTYDFVDDVIGELAALTPGRYLHIGGDEAHSTPKADFVAFMKRVQPIVAKYGKTVVGWHQLAGAEPVEGALVQYWGLDRTGDAEKAEVAEAARNGTGLILSPADRTYLDMKYTKDTPLGLSWAGYVEVQRSYDWDPAGYLPGAPADAVRGVEAPLWTETLSDPDQLDYMAFPRLPGVAELGWSPASTHDWDTYKVRLAAQAPYWEAAGIDFYRSPQVPWT 5fd2 A 2.89 BS01 5XJ A 1 V471 A481 K483 L505 L514 I527 T529 W531 C532 F583 D594 F595 V24 A34 K36 L58 L67 I80 T82 W84 C85 F136 D147 F148 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 27085672 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 5fd3 A 2.42 BS01 dna H 0 K534 L535 Y536 R574 C599 N600 C601 K602 R603 S604 Y610 E612 K13 L14 Y15 R53 C64 N65 C66 K67 R68 S69 Y75 E77 ? remove_due_to_license_issue Q6MZP7 27465258 1 ~ 12 RKPCNCTKSLCLKLYCDCFANGEFCNNCNCTNCYNNLEHENERQKAIKACLDRNPEAFKPKKGCNCKRSGCLKNYCECYEAKIMCSSICKCIGCKNFEESPERKTLMH 5fd3 A 2.42 BS02 dna I 0 C525 N526 C527 K529 S530 Y536 N609 Y610 C4 N5 C6 K8 S9 Y15 N74 Y75 ? remove_due_to_license_issue Q6MZP7 27465258 1 ~ 13 RKPCNCTKSLCLKLYCDCFANGEFCNNCNCTNCYNNLEHENERQKAIKACLDRNPEAFKPKKGCNCKRSGCLKNYCECYEAKIMCSSICKCIGCKNFEESPERKTLMH 5fd3 B 2.42 BS01 dna C 0 K534 L535 Y536 R574 C599 N600 C601 K602 R603 S604 Y610 E612 K13 L14 Y15 R53 C63 N64 C65 K66 R67 S68 Y74 E76 ? remove_due_to_license_issue Q6MZP7 27465258 1 ~ 12 RKPCNCTKSLCLKLYCDCFANGEFCNNCNCTNCYNNLEHENERQKAIKACLDRNPEAFKPKGCNCKRSGCLKNYCECYEAKIMCSSICKCIGCKNFEESPERKTLMHL 5fd3 B 2.42 BS02 dna D 0 C525 N526 C527 T528 K529 S530 Y536 K608 N609 Y610 C4 N5 C6 T7 K8 S9 Y15 K72 N73 Y74 ? remove_due_to_license_issue Q6MZP7 27465258 1 ~ 13 RKPCNCTKSLCLKLYCDCFANGEFCNNCNCTNCYNNLEHENERQKAIKACLDRNPEAFKPKGCNCKRSGCLKNYCECYEAKIMCSSICKCIGCKNFEESPERKTLMHL 5fdc A 1.75 BS02 5WN A 1 H94 H96 V121 F131 L198 T199 T200 H92 H94 V119 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=34.8nM remove_due_to_license_issue IC50=110000nM P00918 27151329 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fdd A 2.506 BS01 4P8 A 1 Y29 H46 E65 Y115 K119 Y29 H46 E65 Y115 K119 3.1.-.- 0003723,0039694 remove_due_to_license_issue IC50=63000nM P03433 27088785 201 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 5fdg A 2.1 BS03 0N8 A 1 Y29 H46 E65 L91 E104 K119 Y29 H46 E65 L91 E104 K119 3.1.-.- 0003723,0039694 remove_due_to_license_issue IC50=430nM P03433 27088785 204 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 5fdi A 1.85 BS02 5WM A 1 Q92 H94 H96 F131 L198 T199 Q90 H92 H94 F128 L195 T196 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=18.5nM remove_due_to_license_issue P00918 27151329 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fdo A 2.8 BS01 5X2 A 1 F228 M231 M250 G262 R263 T266 L267 F270 G271 F50 M53 M72 G84 R85 T88 L89 F92 G93 ? 0042981 remove_due_to_license_issue Ki=361nM, IC50=400nM Q07820 26878343 400 GDELYRQSLEIISRYLREQATGAKGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 5fdo A 2.8 BS02 5X2 B 1 N223 H224 N45 H46 ? 0042981 remove_due_to_license_issue Ki=361nM, IC50=400nM Q07820 26878343 400 GDELYRQSLEIISRYLREQATGAKGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 5fdp A 2.25 BS01 5WR A 1 V624 A653 E672 M676 L679 M699 T701 Y703 M704 F762 L773 A783 D784 V21 A37 E56 M60 L63 M83 T85 Y87 M88 F135 L146 A156 D157 D766 R770 N771 D784 D139 R143 N144 D157 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=309nM remove_due_to_license_issue IC50=21nM Q08345 27219676 1001 DFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKAAGPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNT 5fdr A 2.6 BS01 5X3 A 1 H224 A227 F228 M231 M250 V253 N260 G262 R263 T266 F270 G271 H54 A57 F58 M61 M80 V83 N90 G92 R93 T96 F100 G101 ? 0042981 remove_due_to_license_issue IC50=0.940000nM, Ki=0.360000nM Q07820 26878343 400 DDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLE 5fdr A 2.6 BS02 5X3 B 1 R222 N223 R52 N53 ? 0042981 remove_due_to_license_issue IC50=0.940000nM, Ki=0.360000nM Q07820 26878343 400 DDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLE 5fdz A 2.4 BS01 5X0 A 1 P747 E756 Y802 N803 P804 Y809 P24 E33 Y79 N80 P81 Y86 2.3.1.48,2.3.1.57 0004402 Kd=6.8uM remove_due_to_license_issue Kd=6800nM Q92831 26731131 901 DPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLI 5fe6 A 1.77 BS01 5WZ A 1 F748 Y802 N803 Y809 F26 Y80 N81 Y87 2.3.1.48,2.3.1.57 0004402 Kd=6910uM remove_due_to_license_issue Q92831 26731131 909 RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 5fe7 A 2.08 BS01 5WU A 1 P747 V752 E756 Y802 N803 Y809 P25 V30 E34 Y80 N81 Y87 2.3.1.48,2.3.1.57 0004402 Kd=488uM remove_due_to_license_issue Q92831 26731131 902 RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 5fe9 A 2.35 BS01 5WS A 1 P747 E750 K753 E756 N803 P25 E28 K31 E34 N81 2.3.1.48,2.3.1.57 0004402 Kd=20.98uM remove_due_to_license_issue Kd=20980nM Q92831 26731131 901 RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 5fgk A 2.36 BS01 5XG A 1 V27 Y32 A50 K52 I79 F97 A100 L158 D173 R356 V27 Y32 A50 K52 I79 F97 A100 L151 D166 R325 D151 K153 N156 D173 T196 D144 K146 N149 D166 T172 2.7.11.22,2.7.11.23 0004672,0005524,0006468 ic50=1.7nM remove_due_to_license_issue P49336 26796641 401 MDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRAVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFAVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEE 5fh6 A 2.3 BS01 5XM A 1 I683 F684 L687 Y696 A735 N739 I745 I31 F32 L35 Y44 A83 N87 I93 ? 0006338,0016586 remove_due_to_license_issue Q86U86 27119626 801 KYMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDL 5fh7 A 1.47 BS01 5XL A 1 I683 F684 L687 Y696 M731 A735 N739 I745 I32 F33 L36 Y45 M80 A84 N88 I94 ? 0006338,0016586 Kd=137nM remove_due_to_license_issue Q86U86 27119626 803 SKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDLEGD 5fh8 A 1.55 BS01 5XK A 1 I683 F684 R686 L687 Y696 M731 A735 N739 I745 I32 F33 R35 L36 Y45 M80 A84 N88 I94 ? 0006338,0016586 Kd=170nM remove_due_to_license_issue Q86U86 27119626 801 SKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDL 5fhm A 1.55 BS01 5XP A 1 E13 S14 Y16 Y61 P89 T91 R96 G141 S142 T143 E193 T195 M196 E10 S11 Y13 Y58 P86 T88 R93 G138 S139 T140 E190 T192 M193 ? 0015276,0016020 remove_due_to_license_issue EC50=432000nM, Ki=8150nM P19491 26862980 304 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 5fhn A 1.6 BS01 5XO A 1 S14 Y16 Y61 P89 L90 T91 R96 L138 G141 S142 T143 E193 T195 M196 Y220 W255 S10 Y12 Y57 P85 L86 T87 R92 L134 G137 S138 T139 E189 T191 M192 Y216 W251 ? 0015276,0016020 remove_due_to_license_issue P19491 26862980 305 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 5fho A 2.3 BS01 5XN A 1 E13 S14 Y16 Y61 P89 L90 T91 R96 G141 S142 T143 E193 T195 M196 E10 S11 Y13 Y58 P86 L87 T88 R93 G138 S139 T140 E190 T192 M193 ? 0015276,0016020 remove_due_to_license_issue P19491 26862980 301 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWEC 5fi2 A 2.5 BS01 5XX A 1 K319 L320 F321 L322 Y393 K184 L185 F186 L187 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 ic50=70nM remove_due_to_license_issue IC50=30nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi2 D 2.5 BS01 5XX D 1 K319 L320 F321 L322 E324 Y393 K184 L185 F186 L187 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 ic50=70nM remove_due_to_license_issue IC50=30nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi6 A 2.52 BS01 5XY A 1 R316 F317 K319 L320 F321 L322 N323 E324 Y393 R181 F182 K184 L185 F186 L187 N188 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=70nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi6 B 2.52 BS01 5XY A 1 K319 L320 F321 L322 N323 E324 Y393 K184 L185 F186 L187 N188 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=70nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi6 C 2.52 BS01 5XY C 1 K319 L320 F321 L322 N323 E324 Y393 K184 L185 F186 L187 N188 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=70nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi6 D 2.52 BS01 5XY C 1 K319 L320 F321 L322 E324 Y393 K184 L185 F186 L187 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=70nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi7 A 2.5 BS01 5XZ A 1 K319 L320 F321 L322 E324 Y393 K184 L185 F186 L187 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 ic50=40nM remove_due_to_license_issue IC50=40nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fi7 C 2.5 BS01 5XZ C 1 K319 L320 F321 L322 N323 E324 D326 Y393 K184 L185 F186 L187 N188 E189 D191 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 ic50=40nM remove_due_to_license_issue IC50=40nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5fiv A 1.9 BS01 3TL A 1 G32 A33 D34 M56 I57 G58 I59 G28 A29 D30 M52 I53 G54 I55 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 Ki=22nM remove_due_to_license_issue P16088 10651036 201 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITILNRRDFQVKNSIENGRQNMIGIGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLIQPLLGRDNMIKFNIRLVM 5fkj C 3.133 BS01 G0W C 1 Y72 D74 W86 G121 Y124 S203 W286 H287 I294 F295 Y337 F338 Y341 Y69 D71 W83 G118 Y121 S200 W283 H284 I291 F292 Y334 F335 Y338 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G118 G119 G151 S200 A201 G239 F294 F296 E331 H444 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 26929400 550 EDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCPPGGAGGNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKL 5fky A 1.8 BS01 2J4 A 1 G135 K166 D242 Y282 V314 W337 N339 D344 G129 K160 D236 Y276 V308 W331 N333 D338 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 29997861 1717 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMLPLQVKANRVLISPVEIELDAIYPGENIQINFLSAGLQKAPVKFVRFQFVLTIEK 5fl0 A 1.95 BS01 71I A 1 G135 K166 D242 C278 Y282 M308 W309 T310 W337 N339 D344 G132 K163 D239 C275 Y279 M305 W306 T307 W334 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 29997861 1718 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISKNLPLQVKANRVLISPANEVEIELDAIYPGENIQINLEISTDGKEWKTVDLLSAGLQKAPVKFVRFQFVLTIEK 5fl1 A 1.95 BS01 DV1 A 1 G135 K166 D242 C278 Y282 M308 T310 W337 N339 D344 G127 K158 D234 C270 Y274 M300 T302 W329 N331 D336 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 29997861 1716 SLQPPPQQLIVNKTIDLPAVYQLNGGEEANPHAVKVLKELLSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELECFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPYQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISNVEQIKNLPLQVKANRVLISPANEVVKWAAGNSVEIELDAIYPGENIQINFGCTWGRLEISTDGKEWKTVDLKQKESRLSAGLQKAPVKFVRFTNVSDEEQQVYLRQFVLTIEK 5fl4 A 1.82 BS02 9FK A 1 H94 H119 V130 L134 L199 T200 T201 W210 H86 H111 V122 L126 L191 T192 T193 W202 H68 H94 H96 E106 H119 T200 H60 H86 H88 E98 H111 T192 4.2.1.1 0004089,0008270 Ki=101nM remove_due_to_license_issue Ki=101nM Q16790 26522624 269 WRYGGDPPWPRVSPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 5fl5 A 2.05 BS01 82E A 1 H94 H119 V130 L199 T200 T201 W210 H86 H111 V122 L191 T192 T193 W202 H68 H94 H96 E106 H119 T200 H60 H86 H88 E98 H111 T192 4.2.1.1 0004089,0008270 Ki=6.4nM remove_due_to_license_issue Ki=6.4nM Q16790 26522624 266 WRYGGDPPWPRVSPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 5fl6 A 1.95 BS01 Y0R A 1 Q92 H94 V130 L199 T200 T201 W210 Q84 H86 V122 L191 T192 T193 W202 H68 H94 H96 E106 H119 T200 H60 H86 H88 E98 H111 T192 4.2.1.1 0004089,0008270 Ki=43.6nM remove_due_to_license_issue Ki=44nM Q16790 26522624 268 WRYGGDPPWPRVSPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 5flo A 1.66 BS02 J4K A 1 Q92 H94 H119 L198 T199 T200 W209 Q90 H92 H117 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=709uM remove_due_to_license_issue P00918 26882437 1263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5flp A 1.71 BS02 6J5 A 1 H94 F131 L198 T199 T200 H91 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=631uM remove_due_to_license_issue P00918 26882437 1264 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5flp A 1.71 BS03 6J5 A 2 F131 P202 F127 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=631uM remove_due_to_license_issue P00918 26882437 1265 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5flq A 1.7 BS02 IO2 A 1 H94 H119 V121 F131 L198 T200 P202 H92 H117 V119 F128 L195 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1080uM remove_due_to_license_issue P00918 26882437 1264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fls A 1.67 BS02 6ZX A 1 L198 T200 P202 L195 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=905uM remove_due_to_license_issue P00918 26882437 1263 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5flt A 1.67 BS02 VJJ A 1 Q92 H94 F131 L198 T200 P202 Q90 H92 F128 L195 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1280uM remove_due_to_license_issue P00918 26882437 1264 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5flv A 3.005 BS01 dna B 0 R141 V142 F144 Q180 I183 W184 N187 N1162 S1175 M1176 T1215 P1231 F1232 K1234 G1235 R2 V3 F5 Q41 I44 W45 N48 N162 S175 M176 T203 P219 F220 K222 G223 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 -1 ~ 19 PRVLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKGIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFRG 5flv A 3.005 BS02 dna C 0 Y161 Q186 R189 Y190 R1081 R1082 Y1217 T1223 K1226 F1232 F1236 Y22 Q47 R50 Y51 R81 R82 Y205 T211 K214 F220 F224 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 5 ~ 24 PRVLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKGIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFRG 5flv A 3.005 BS03 dna O 0 K1055 R1061 K55 R61 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 4 ~ 25 PRVLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKGIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFRG 5flv E 3.005 BS01 dna F 0 V142 F144 Q180 I183 W184 N187 N1162 S1175 T1215 P1231 K1234 G1235 V1 F3 Q39 I42 W43 N46 N165 S178 T205 P221 K224 G225 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 -1 ~ 19 VLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKSKRQRQIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKASTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFR 5flv E 3.005 BS02 dna G 0 Y161 Q186 R189 Y190 R1081 R1082 K1159 Y1217 T1223 I1227 N1230 F1232 F1236 Y20 Q45 R48 Y49 R84 R85 K162 Y207 T213 I217 N220 F222 F226 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 5 ~ 25 VLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKSKRQRQIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKASTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFR 5flv I 3.005 BS01 dna J 0 F144 Q180 I183 W184 N187 K191 N1162 S1175 T1215 P1231 F1232 K1234 G1235 F5 Q41 I44 W45 N48 K52 N163 S176 T204 P220 F221 K223 G224 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 -1 ~ 19 PRVLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKSKRQRVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFR 5flv I 3.005 BS02 dna K 0 R141 Y161 Q186 R189 Y190 R1081 R1082 K1159 Y1217 T1223 N1230 F1232 F1236 R2 Y22 Q47 R50 Y51 R83 R84 K160 Y206 T212 N219 F221 F225 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 4 ~ 25 PRVLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKSKRQRVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFR 5flv M 3.005 BS01 dna N 0 F144 Q180 I183 W184 N187 K191 N1162 S1175 T1215 P1231 F1232 K1234 G1235 F3 Q39 I42 W43 N46 K50 N164 S177 T207 P223 F224 K226 G227 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 -1 ~ 19 VLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKSKRQGIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADAFSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFR 5flv M 3.005 BS02 dna O 0 Y161 Q186 R189 Y190 R1081 R1082 K1159 Y1217 T1223 N1230 F1232 F1236 Y20 Q45 R48 Y49 R83 R84 K161 Y209 T215 N222 F224 F228 ? 0000978,0000981,0003677,0003700,0005634,0006355,0045893 remove_due_to_license_issue P42582,P70326 26875865 4 ~ 25 VLFSQAQVYELERRFKQQRYLSAPERDQLASVLKLTSTQVKIWFQNRRYKSKRQGIKVFLHERELWLKFHEVGTEMIITKAGRRMFPSYKVKVTGLNPKTKYILLMDIVPADDHRYKFADNKWSVTGKAEPAMPGRLYVHPDSPATGAHWMRQLVSFQKLKLTNNHLDPFGHIILNSMHKYQPRLHIVKADAFSTHVFPETAFIAVTSYQNHKITQLKIENNPFAKGFR 5fnc A 2.2 BS01 IEE A 1 A55 G97 M98 L107 F138 E223 A40 G82 M83 L92 F123 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=77uM remove_due_to_license_issue P07900 28221352 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5fnd A 2.0 BS01 IQ5 A 1 A55 K58 I96 G97 M98 L107 G108 T184 E223 A40 K43 I81 G82 M83 L92 G93 T169 E208 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=320uM remove_due_to_license_issue P07900 28221352 1225 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5fnf A 2.1 BS01 TQL A 1 N51 A55 D93 G97 M98 N36 A40 D78 G82 M83 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=700uM remove_due_to_license_issue P07900 28221352 1226 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5fng A 2.05 BS02 YIE A 1 Q92 H94 H119 L198 T199 T200 W209 Q89 H91 H116 L194 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1105uM remove_due_to_license_issue P00918 26882437 1263 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fni A 1.6 BS02 YIH A 1 Q92 H94 H119 F131 L198 T199 T200 W209 Q90 H92 H117 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=330uM remove_due_to_license_issue P00918 26882437 1265 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fnj A 1.67 BS02 YI6 A 1 Q92 H94 H96 V121 F131 T199 T200 Q90 H92 H94 V119 F128 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=5150uM remove_due_to_license_issue P00918 26882437 1267 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fnj A 1.67 BS03 YI6 A 2 D72 D130 F131 G132 D70 D127 F128 G129 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=5150uM remove_due_to_license_issue P00918 26882437 1268 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5fnq A 1.91 BS01 S0W A 1 R415 G462 R483 S508 G509 A556 R92 G139 R160 S185 G186 A233 ? remove_due_to_license_issue Q9Z2X8 27031670 1614 VGRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 5fnr A 1.89 BS01 XMS A 1 R415 G462 F478 R483 S508 G509 Y525 S555 A556 Y572 R91 G138 F154 R159 S184 G185 Y201 S231 A232 Y248 ? Kd=59uM remove_due_to_license_issue Q9Z2X8 27031670 1614 GRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 5fns A 1.79 BS01 XYY A 1 Y334 G364 R415 G462 R483 S508 G509 Y525 S555 A556 S602 G603 Y10 G40 R91 G138 R159 S184 G185 Y201 S231 A232 S278 G279 ? Kd=4uM remove_due_to_license_issue Q9Z2X8 27031670 1614 GRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 5fnt A 1.79 BS01 0PL A 1 Y334 G364 R415 G462 F478 R483 S508 G509 Y525 S555 A556 S602 G603 Y10 G40 R91 G138 F154 R159 S184 G185 Y201 S231 A232 S278 G279 ? Kd=0.67uM remove_due_to_license_issue Q9Z2X8 27031670 1615 GRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 5fnu A 1.78 BS01 L6I A 1 Y334 G364 R415 G462 F478 R483 S508 G509 Y525 S555 A556 Y572 S602 G603 Y9 G39 R90 G137 F153 R158 S183 G184 Y200 S230 A231 Y247 S277 G278 ? Kd=0.0013uM remove_due_to_license_issue Q9Z2X8 27031670 1615 RLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 5fog A 2.3 BS01 VRT A 1 T287 L288 S415 K418 V423 T424 D433 K496 T34 L35 S153 K156 V161 T162 D171 K234 6.1.1.4 0000166,0002161,0004823,0005524,0006418,0006429 Kd=213uM remove_due_to_license_issue B6AA20 27431220 1542 GPQEYTLIKLKIHLIPEFLGSIVKGREVFVVCATLRPETMYGQTNCWILPDGEYDLVLAFDQVIPYDAKTSDGVLCKIFDKYEDTMKECNTVYICSERSAYNMAYQGIVPLIHGLPRIVSLGKVYGEQLIGTPLSAPMTPYSLIFILPMFSISMEKGTGIVTSVPSDSPDDYAALRDIKTKPLLREKYSIKDEWILDPLEIIEVPGFGFMTAELLCNQYKIQSQNDSAKLKQAKEEIYKKEFYEGILIRGKYSGMKICDAKELIRESLIKDGYALIYLE 5fol A 1.77 BS01 SO8 A 1 T287 L288 T292 S415 K418 V423 T424 D433 T34 L35 T39 S148 K151 V156 T157 D166 6.1.1.4 0000166,0002161,0004823,0005524,0006418,0006429 Kd=215uM remove_due_to_license_issue B6AA20 27431220 1544 GPQEYTLIKLKIHLIPEFLGSIVKGREVFVVCATLRPETMYGQTNCWILPDGEYDLVLAFDQKIFDKYEDTMKECNTVYICSERSAYNMAYQGIVPLIHGREQGVSDKLLPRIVSLGKVYGEQLIGTPLSAPMTPYSLIFILPMFSISMEKGTGIVTSVPSDSPDDYAALRDIKTKPLLREKYSIKDEWILDPLEIIEVPGFGFMTAELLCNQYKIQSQNDSAKLKQAKEEIYKKEFYEGILIRGKYSGMKICDAKELIRESLIKDGYALIYLE 5fom A 2.1 BS01 A2H A 1 Y258 A286 T287 L288 R289 T292 I414 S415 K418 V423 T424 S430 D433 K496 Y5 A33 T34 L35 R36 T39 I147 S148 K151 V156 T157 S163 D166 K229 6.1.1.4 0000166,0002161,0004823,0005524,0006418,0006429 Kd=9.8uM remove_due_to_license_issue B6AA20 27431220 1542 GPQEYTLIKLKIHLIPEFLGSIVKGREVFVVCATLRPETMYGQTNCWILPDGEYDLVLAFDQKIFDKYEDTMKECNTVYICSERSAYNMAYQGIVPLIHGREQGVSDKLLPRIVSLGKVYGEQLIGTPLSAPMTPYSLIFILPMFSISMEKGTGIVTSVPSDSPDDYAALRDIKTKPLLREKYSIKDEWILDPLEIIEVPGFGFMTAELLCNQYKIQSQNDSAKLKQAKEEIYKKEFYEGILIRGKYSGMKICDAKELIRESLIKDGYALIYLE 5foo A 2.1 BS01 JAZ A 1 Q18 H119 E165 Y299 K337 E366 W416 S423 Y432 Q18 H119 E165 Y299 K337 E366 W416 S423 Y432 R74 H119 E165 V168 N297 Y299 E366 R74 H119 E165 V168 N297 Y299 E366 '3.2.1.21,3.2.1.86' 0004553,0005829,0005975,0008422,0016052,0016798 remove_due_to_license_issue Q99YP9 26790390 1464 MLAFPKEFWWGGATSGPQSEGRFAKQHRNLFDYWYEEEPDLFYDYVGPDTASDAYHQIESDLTLLASLGHNSYRTSIQWTRLIDDFEQATINPDGLAYYNRVIDACLANGIRPVINLHHFDLPIALYQAYGGWESKHVVDLFVAFSKVCFEQFGDRVKDWFVHNEPMVVVEGSYLMQFHYPAIVDGKKAVQVAYNLALATAKVIQAYRRGPAELSDGRIGTILNLTPAYPASQSEADMAAAHFAELWNNDLFMEAAVHGKFPEELVAVLKKDGVLWQSTPEELALIAENRVDYLGLNFYHPKRVKAPDAIPVISPSWSPEWYYDPYLMPGHRMNVDKGWEIYPEAVYDIAIKMRDHYDNIPWFLSENGVGISGEDRYRDETGQIQDDYRIQFLKEHLTYLHKGIEAGSNCFGYHVWTPIDGWSWLNAYKNRYGLVENNIHTQVRRPKASAYWFKKVATHNRLI 5fp0 A 2.35 BS01 SZC A 1 F267 D335 W336 M339 Y383 Q384 Y466 M503 H524 F266 D334 W335 M338 Y379 Q380 Y462 M499 H520 F267 H334 D335 W336 N359 N378 Y383 Y466 D496 H524 F266 H333 D334 W335 N358 N374 Y379 Y462 D492 H520 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 ic50=0.017uM remove_due_to_license_issue P34913 26845235 1549 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESNPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 5fpp A 2.4 BS01 HI6 A 1 D74 Y124 X203 W286 F297 Y337 F338 Y341 D74 Y124 X203 W279 F290 Y330 F331 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 Kd=100uM remove_due_to_license_issue P21836 27140636 1552 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSATATEAP 5fpu A 2.24 BS03 K0I A 1 Q88 T97 R98 Y425 Y488 F496 H499 E501 K517 Q65 T74 R75 Y128 Y190 F198 H201 E203 K219 G481 Y488 H499 E501 H587 A599 G183 Y190 H201 E203 H289 A301 1.14.11.67 Ki=0.14uM remove_due_to_license_issue IC50=210nM Q9UGL1 27214403 1756 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKRDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAE 5fq9 A 1.5 BS01 C6S A 1 S67 K70 S115 V117 T206 G207 F208 R250 S49 K52 S97 V99 T188 G189 F190 R232 S67 K70 S115 F120 W154 F208 S49 K52 S97 F102 W136 F190 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0042597,0046677,0071555 remove_due_to_license_issue P14489 27499424 300 MGSITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNDLARASKEYLPASTFKIPNAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLTLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLYLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKETEVYFFAFNMDIDNESKLPLRKSIPTKIMESEGII 5fqb A 1.899 BS03 OK3 A 1 F65 W90 H119 H121 A122 D123 H199 C224 N236 D239 H266 F29 W51 H78 H80 A81 D82 H141 C160 N172 D175 H202 H119 H121 D123 H199 C224 K227 N236 H266 H78 H80 D82 H141 C160 K163 N172 H202 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.3uM remove_due_to_license_issue P04190 27499424 297 KTVIKNETGTISISQLNKNVWVHTELGSFAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 5fqc A 1.449 BS03 OK3 A 1 H114 H116 D118 H179 C198 N210 H240 H83 H85 D87 H148 C167 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=0.003uM remove_due_to_license_issue Q9K2N0 27499424 600 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5fqp A 1.88 BS01 GQD A 1 L346 T347 A350 E353 F404 L525 V533 V534 L40 T41 A44 E47 F98 L219 V227 V228 ? ic50=19nM remove_due_to_license_issue IC50=1.3nM P03372 26819673 1549 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPSYDLLLEMLDAHR 5fqr A 1.88 BS01 QHG A 1 L346 T347 A350 E353 M421 L525 V534 L37 T38 A41 E44 M112 L213 V217 ? ic50=26nM remove_due_to_license_issue IC50=25nM P03372 26819673 1546 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMVPSYDLLLEMLD 5fqs A 1.94 BS01 J0W A 1 T347 A350 E353 L525 V533 V534 T38 A41 E44 L213 V221 V222 ? ic50=44nM remove_due_to_license_issue IC50=44nM P03372 26819673 1546 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPSYDLLLEMLD 5fqt A 1.99 BS01 7QN A 1 L346 T347 A350 E353 L387 M388 L391 H524 V533 V534 L37 T38 A41 E44 L78 M79 L82 H212 V221 V222 ? ic50=160nM remove_due_to_license_issue IC50=170nM P03372 26819673 1546 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPSYDLLLEMLD 5fqv A 1.74 BS01 VQI A 1 T347 L349 A350 E353 F404 L525 V533 V534 T38 L40 A41 E44 F95 L213 V221 V222 ? ic50=610nM remove_due_to_license_issue IC50=160nM P03372 26819673 1546 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPSYDLLLEMLD 5fs5 A 1.42 BS01 KGM A 1 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 D54 Q133 N135 D140 ? 0007155,0009289 Kd=206.4nM remove_due_to_license_issue P08191 28250938 1159 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNANSDDFQFVWNIYANNDVVVPT 5fsb A 1.65 BS01 6YR A 1 G8 S9 N25 Y31 W41 G7 S8 N24 Y30 W40 ? remove_due_to_license_issue B0CZL6 29398527 300 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsb A 1.65 BS02 6YR A 2 G46 A47 N63 Y69 W78 G45 A46 N62 Y68 W77 ? remove_due_to_license_issue B0CZL6 29398527 301 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsb A 1.65 BS03 6YR A 3 G83 A84 N100 Y106 W116 G82 A83 N99 Y105 W115 ? remove_due_to_license_issue B0CZL6 29398527 302 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsb A 1.65 BS04 6YR A 4 V122 N138 Y144 W156 V121 N137 Y143 W155 ? remove_due_to_license_issue B0CZL6 29398527 303 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsb A 1.65 BS05 6YR A 5 A162 N178 Y184 A161 N177 Y183 ? remove_due_to_license_issue B0CZL6 29398527 304 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsc A 1.95 BS01 G8Z A 1 G83 A84 N100 Y106 G82 A83 N99 Y105 ? remove_due_to_license_issue B0CZL6 29398527 302 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsc A 1.95 BS02 G8Z A 2 G121 V122 N138 Y144 G120 V121 N137 Y143 ? remove_due_to_license_issue B0CZL6 29398527 303 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsc A 1.95 BS03 G8Z A 3 G161 A162 N178 Y184 G160 A161 N177 Y183 ? remove_due_to_license_issue B0CZL6 29398527 304 PWKGISGSLSRISAGSVTNVWGVNAANNIYRYTGDDAKPWVQIPGALTDIGAAADGTVWGVNAAGNIYRYVWDSNHWTQIKGALKRISAGSRTNVWGVNAGGAIYRYTGDDANPWVQIPGVLSDIGAGADGTVWGVNAAGEIYRYTGDQGDPNHWVKIPGALSAISAGIKTNVWGVNSANNIYTSTGDDKNPWLGIGGSLVDIGAGTDGVVWGVNAGGGIYRWIRD 5fsl A 1.24 BS01 UAN A 1 N33 F72 W117 D119 D120 N31 F70 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=24uM remove_due_to_license_issue P36639 26999531 1157 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5fsm A 1.67 BS01 N91 A 1 L9 N33 G34 F72 W117 D119 D120 L7 N31 G32 F70 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd>40uM remove_due_to_license_issue P36639 26999531 202 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5fsn A 1.69 BS01 6Q3 A 1 F27 F72 M81 W117 D119 F139 F25 F70 M79 W115 D117 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=1.7uM remove_due_to_license_issue P36639 26999531 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5fso A 1.67 BS01 S76 A 1 L9 N33 F72 W117 D119 D120 L7 N31 F70 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=0.81uM remove_due_to_license_issue P36639 26999531 1158 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5fsx A 2.0 BS01 ADP A 1 A120 G130 V131 C208 S210 G212 V213 Y214 F248 E252 A92 G102 V103 C180 S182 G184 V185 Y186 F220 E224 ? 0000166 Ka=540M^-1 remove_due_to_license_issue C9ZP98 27064071 1262 EFVTYSGEESSPTRTRILSAALSPAERAIFDVPIEKWLSIDRSSLSGWKCAVPRPVTIEQLRPVDPSDAILRHIALYRGPVTDLQLDAIVNAANTRCLGGGGVDGAIHRVAGPLLLRECATFNGCQTGECRLTKGYQLPARYVLHTVGPVGERPDMLRKCYRSILSLALKNGLRSIGFCCVSTGVYGYPLLPATRIALGETRKFLEEHGGALDMCCFACFQEDEYKTYEKCVG 5fsy A 1.7 BS01 AR6 A 1 A120 N122 G129 G130 V131 D132 C208 S210 G212 V213 Y214 F248 Q249 E252 A91 N93 G100 G101 V102 D103 C179 S181 G183 V184 Y185 F219 Q220 E223 ? 0000166 Ka=790000M^-1 remove_due_to_license_issue C9ZP98 27064071 1262 EFVTYSGEESPTRTRILSAALSPAERAIFDVPIEKWLSIDRSSLSGWKCAVPRPVTIEQLRPVDPSDAILRHIALYRGPVTDLQLDAIVNAANTRCLGGGGVDGAIHRVAGPLLLRECATFNGCQTGECRLTKGYQLPARYVLHTVGPVGERPDMLRKCYRSILSLALKNGLRSIGFCCVSTGVYGYPLLPATRIALGETRKFLEEHGGALDMCCFACFQEDEYKTYEKCVG 5ftg A 1.45 BS01 NBR A 1 D306 Q308 Y333 Y354 E357 F361 W420 W423 E434 Y440 D202 Q204 Y229 Y250 E253 F257 W316 W319 E330 Y336 2.7.1.32,2.7.1.82 Kd=0.7uM remove_due_to_license_issue P35790 27029499 1458 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5fto A 2.22 BS01 YMX A 1 L1122 G1123 F1127 V1130 A1148 L1196 M1199 A1200 G1202 D1203 N1254 L1256 G1269 L30 G31 F35 V38 A52 L100 M103 A104 G106 D107 N158 L160 G173 D1249 A1251 R1253 N1254 D1270 R1279 D153 A155 R157 N158 D174 R183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=6.2nM remove_due_to_license_issue IC50=55nM, Ki=6.2nM Q9UM73 27003761 2402 GPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSGMSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5ftq A 1.7 BS01 U4W A 1 L1122 G1123 F1127 V1130 A1148 L1196 E1197 L1198 M1199 A1200 G1202 D1203 N1254 L1256 G1269 L30 G31 F35 V38 A49 L97 E98 L99 M100 A101 G103 D104 N155 L157 G170 D1249 A1251 R1253 N1254 D1270 R1279 D150 A152 R154 N155 D171 R180 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.01uM remove_due_to_license_issue IC50=10.0nM Q9UM73 27003761 2402 GPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRCAMLPVKWMPPEAFEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5fue A 2.199 BS02 UV4 A 1 K20 H142 G150 D186 H188 F216 H292 Y341 K19 H141 G149 D176 H178 F206 H275 Y312 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=468.2nM remove_due_to_license_issue A5H660 26937828 700 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 5ful A 1.89 BS01 SAH A 1 Y114 F115 Y118 M127 R133 G157 C158 I162 E180 A181 K207 V208 E223 M234 S237 Y8 F9 Y12 M21 R27 G51 C52 I56 E74 A75 K101 V102 E117 M128 S131 D130 E223 E232 H381 D24 E117 E126 H275 2.1.1.125 0008168,0016274,0018216,0032259,0046872 ic50=18.3uM remove_due_to_license_issue Q3UKX1 27879050 1446 DTWQDEEYFDSYGTLKLHLEMLADQPRTTKYHSVILQNKESLKDKVILDVGCGTGIISLFCAHHARPKAVYAVEASDMAQHTSQLVLQNGFADTITVFQQKVEDVVLPEKVDVLVSEWMGTCLLFEFMIESILYARDTWLKGDGIIWPTTAALHLVPCSAEKDYHSKVLFWDNAYEFNLSALKSLAIKEFFSRPKSNHILKPEDCLSEPCTILQLDMRTVQVPDLETMRGELRFDIQKAGTLHGFTAWFSVYFQSLEEGQPQQVLSTGPLHPTTHWKQTLFMMDDPVPVHTGDVVTGSVVLQRNPVWRRHMSVSLSWVVTSALDPTSQRVGEKVFPIWW 5fum A 2.5 BS01 SOF A 1 Y72 W86 Y124 Y337 F338 Y72 W86 Y124 Y330 F331 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue IC50=18000nM P21836 27598521 1543 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 5fun A 2.3 BS03 GZA A 1 R86 Y425 Y488 F496 H499 N509 K517 W519 H587 R63 Y128 Y190 F198 H201 N211 K219 W221 H289 G481 Y488 H499 E501 H587 A599 G183 Y190 H201 E203 H289 A301 1.14.11.67 Ki=0.01uM remove_due_to_license_issue IC50=26nM Q9UGL1 27214403 1756 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVARDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGKKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAE 5fut A 1.6 BS01 PQ7 A 1 D306 Y333 Y354 W420 W423 I433 F435 Y440 D204 Y231 Y252 W318 W321 I331 F333 Y338 2.7.1.32,2.7.1.82 Kd=352nM remove_due_to_license_issue P35790 27616047 1467 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5fv7 A 2.84 BS03 R3Z A 1 G2 M37 Y40 E160 D179 G1 M36 Y39 E110 D129 3.1.-.- 0003677,0003824,0004518,0016788 remove_due_to_license_issue IC50=0.011nM P39748 27526030 1341 GIQGLAKLIADVAPSAIRENDIKSYFGRKVAIDASMSIYQFLITTSHLMGMFYRTIRMMENGIKPVYVFDGKPPQLKSGEVKVTKQHNDECKHLLSLMGIPYLDAPSEAEASCAALVKAGKVYAAATEDMDCLTFGSPVLMRHLTKLPIQEFHLSRILQELGLNQEQFVDLCILLGSDYCESIRGIGPKRAVDLIQKHKSIEEIVRRLDPNKYPVPENWLHKEAHQLFLEPEVLDPESVELKWSEPNEEELIKFMCGEKQFSEERIRSGVKRLSKSRQGSTLE 5fwa A 1.8 BS01 J7C A 1 Y114 F115 Y118 G157 E180 A181 K207 E223 W224 M225 E232 M234 S237 Y8 F9 Y12 G51 E74 A75 K101 E117 W118 M119 E126 M128 S131 D130 E223 E232 H381 D24 E117 E126 H275 2.1.1.125 0008168,0016274,0018216,0032259,0046872 ic50=16.3uM remove_due_to_license_issue Q3UKX1 27879050 1446 DTWQDEEYFDSYGTLKLHLEMLADQPRTTKYHSVILQNKESLKDKVILDVGCGTGIISLFCAHHARPKAVYAVEASDMAQHTSQLVLQNGFADTITVFQQKVEDVVLPEKVDVLVSEWMGTCLLFEFMIESILYARDTWLKGDGIIWPTTAALHLVPCSAEKDYHSKVLFWDNAYEFNLSALKSLAIKEFFSRPKSNHILKPEDCLSEPCTILQLDMRTVQVPDLETMRGELRFDIQKAGTLHGFTAWFSVYFQSLEEGQPQQVLSTGPLHPTTHWKQTLFMMDDPVPVHTGDVVTGSVVLQRNPVWRRHMSVSLSWVVTSALDPTSQRVGEKVFPIWW 5fwg A 2.0 BS01 GPR A 1 Y6 X7 G11 L12 X45 N58 L59 Q71 S72 I111 S209 Y6 X7 G11 L12 X45 N58 L59 Q71 S72 I111 S209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005496,0005576,0005737,0005829,0006629,0006693,0006749,0007608,0009410,0010038,0010288,0016151,0016740,0018916,0019899,0019901,0032991,0042178,0042802,0042803,0043200,0043295,0045471,0048678,0051122,0070458,0071466,1901687 remove_due_to_license_issue P04905 9572843 218 PMILGYWNVRGLTHPIRLLLEYTDSSYEEKRYAMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGSRKITQSNAIMRYLARKHHLCGETEEERIRADIVENQVMDNRMQLIMLCYNPDFEKQKPEFLKTIPEKMKLYSEFLGKRPWFAGDKVTYVDFLAYDILDQYHIFEPKCLDAFPNLKDFLARFEGLKKISAYMKSSRYLSTPIFSKLAQWSNK 5fwg B 2.0 BS01 GPR B 1 Y6 X7 G11 L12 R42 X45 K49 N58 L59 Q71 S72 I111 Y6 X7 G11 L12 R42 X45 K49 N58 L59 Q71 S72 I111 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005496,0005576,0005737,0005829,0006629,0006693,0006749,0007608,0009410,0010038,0010288,0016151,0016740,0018916,0019899,0019901,0032991,0042178,0042802,0042803,0043200,0043295,0045471,0048678,0051122,0070458,0071466,1901687 remove_due_to_license_issue P04905 9572843 218 PMILGYWNVRGLTHPIRLLLEYTDSSYEEKRYAMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGSRKITQSNAIMRYLARKHHLCGETEEERIRADIVENQVMDNRMQLIMLCYNPDFEKQKPEFLKTIPEKMKLYSEFLGKRPWFAGDKVTYVDFLAYDILDQYHIFEPKCLDAFPNLKDFLARFEGLKKISAYMKSSRYLSTPIFSKLAQWSNK 5fwj A 2.1 BS06 MMK A 1 Y440 D443 W501 Y503 F511 H514 E516 K532 W534 H602 V615 N616 Y122 D125 W183 Y185 F193 H196 E198 K214 W216 H268 V281 N282 G496 Y503 H514 E516 H602 A614 G178 Y185 H196 E198 H268 A280 1.14.11.67 Ki=0.0061uM remove_due_to_license_issue P41229 27214403 1775 SMFLPPPECPVFEPSWAEFRDPLGYIAKIRPIAEKSGICKIRPPADWQPPFAVEVDNFRFTPRIQRLNELTREYTLQSFGEMADSFKADYFNMPVHMVPTELVEKEFWRLVNSIEEDVTVEYGADIHSKEFGSGFPVSDSKRHLTPEEEEYATSGWNLNVMPVLEQSVLCHINADISGMKVPWLYVGMVFSAFCWHIEDHWSYSINYLHWGEPKTWYGVPSLAAEHLEEVMKKLTLMNPNTLMSHGVPVVRTNQCAGEFVITFPRAYHSGFNQGYNFAEAVNFCTADWLPAGRQCIEHYRRLRRYCVFSHEELICKMAACPEKLDLNLAAAVHKEMFIMVQEERRLRKALLEKGITEAEREAFELLPDDERQCIKCKTTCFLSALACYDCPDGLVCLSHINDLCKCSSSRQYLRYRYTLDELPAMLHKLKVRAES 5fwr A 2.13 BS01 3X8 A 1 F1 I13 N46 Y48 I52 D54 Q133 N135 Y137 D140 F1 I13 N46 Y48 I52 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=17.7nM remove_due_to_license_issue P08191 28250938 182 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 5fxq A 2.3 BS01 GD5 A 1 V1013 A1031 M1079 M1082 T1083 G1085 M1142 D1153 V35 A53 M100 M103 T104 G106 M161 D172 D1135 R1139 N1140 D1153 E1162 D154 R158 N159 D172 E181 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=55nM P08069 27078757 2287 SYFSAADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 5fxr A 2.4 BS01 8LN A 1 L1005 V1013 A1031 M1079 M1082 G1085 M1156 L26 V34 A52 M99 M102 G105 M176 D1135 R1139 N1140 D1153 E1162 D155 R159 N160 D173 E182 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=38nM P08069 27078757 2284 GYFSADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSE 5fxs A 1.9 BS01 OZN A 1 L1005 V1013 A1031 M1079 M1082 G1085 M1142 M1156 L27 V35 A53 M101 M104 G107 M164 M178 D1135 R1139 N1140 D1153 E1162 D157 R161 N162 D175 E184 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P08069 27078757 2290 SYFSAADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRAIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEEPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 5fyx A 1.8 BS04 FD6 A 1 I51 F72 F85 T92 L182 I45 F66 F79 T86 L166 ? 0005509,0005515,0005737,0007268,0007269,0007528,0008021,0008048,0009966,0016192,0046872,0046928 remove_due_to_license_issue Q9VWX8 28119500 1195 KLKQDTIDRLTTDTYFTEKEIRQWHKGFLKDCPNGLLTEQGFIKIYKQFFPDGDPSKFASLVFRVFDENNDGAIEFEEFIRALSITSRGNLDEKLHWAFRLYDVDNDGYITREEMYNIVDAIYQMVTPQKRVDKIFDQMDKNHDDRLTLEEFREGSKADPRMVQALSLG 5g0q A 1.65 BS01 IF6 A 1 E45 G79 N80 D105 N172 E173 Y243 E245 E287 Y292 Q293 H327 Y334 E28 G62 N63 D88 N155 E156 Y226 E228 E270 Y275 Q276 H310 Y317 3.2.1.31 0016020,0016798 remove_due_to_license_issue C1F2K5 28581485 1476 SPVRVGLSVDASALGHTIPPDYTGLSYEQAQMANPNYFSGANTQLAGFLRTLGRQGVLRIGGNTSEYTFWNRHAKPTAADEHLAAGPDKGHHAAAREVITPEAVNNLSEFLDKTGWKLIYGLNLGKGTPENAADEAAYVMETIGADRLLAFQLGNEPDLFYRNGIRPASYDFAAYAGDWQRFFTAIRKRVPNAPFAGPDTAYNTKWLVPFADKFKHDVKFISSHYYAEGPPTDPSMTIERLMKPNPRLLGETAGLKQVEADTGLPFRLTETNSCYQGGKQGVSDTFAAALWAGDLMYQQAAAGSTGINFHGGGYGWYTPVAGTPEDGFIARPEYYGMLLFAQAGAGQLLGAKLTDNSAAPLLTAYALRGTDGRTRIALFNKNLDADVEVAISGVASPSGTVLRLEAPRADDTTDVTFGGAPVGASGSWSPLVQEYVPGQFVLHMRKASGALLEFA 5g10 A 1.71 BS02 6DK A 1 T24 D101 P141 H143 H144 G152 F153 D181 H183 F209 E310 G311 Y313 T23 D100 P140 H142 H143 G151 F152 D180 H182 F208 E309 G310 Y312 3.5.1.- 0004407,0016787,0040029,0046872 ic50=9.7nM remove_due_to_license_issue Q9HXM1 27951649 1375 TRRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGYSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGLC 5g10 B 1.71 BS01 6DK A 1 L340 F343 L339 F342 3.5.1.- 0004407,0016787,0040029,0046872 ic50=9.7nM remove_due_to_license_issue Q9HXM1 27951649 1375 TRRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGYSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGLCPAQPLQ 5g10 B 1.71 BS03 6DK B 1 T24 D101 H143 H144 G152 F153 D181 H183 F209 E310 G311 Y313 T23 D100 H142 H143 G151 F152 D180 H182 F208 E309 G310 Y312 3.5.1.- 0004407,0016787,0040029,0046872 ic50=9.7nM remove_due_to_license_issue Q9HXM1 27951649 1381 TRRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGYSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGLCPAQPLQ 5g11 A 2.48 BS01 7H1 A 1 T24 L25 D101 H143 H144 G152 F153 D181 H183 F209 L276 T22 L23 D99 H141 H142 G150 F151 D179 H181 F207 L274 3.5.1.- 0004407,0016787,0040029,0046872 ic50=62nM remove_due_to_license_issue Q9HXM1 27951649 1372 RRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGFSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGLC 5g11 B 2.48 BS01 7H1 B 1 T24 D101 H143 H144 G152 F153 D181 H183 F209 L276 T22 D99 H141 H142 G150 F151 D179 H181 F207 L274 3.5.1.- 0004407,0016787,0040029,0046872 ic50=62nM remove_due_to_license_issue Q9HXM1 27951649 1378 RRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGFSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGLCPAQPLQ 5g17 A 1.51 BS02 6DK A 1 P140 H142 H143 G151 F152 D180 H182 F208 G310 Y312 P139 H141 H142 G150 F151 D179 H181 F207 G309 Y311 3.5.1.- 0004407,0016787,0040029,0046872 Kd=0.2uM remove_due_to_license_issue Q70I53 28389333 373 AIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGIAMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g17 B 1.51 BS02 6DK B 1 P140 H142 H143 G151 F152 D180 H182 F208 G310 Y312 P140 H142 H143 G151 F152 D180 H182 F208 G310 Y312 3.5.1.- 0004407,0016787,0040029,0046872 Kd=0.2uM remove_due_to_license_issue Q70I53 28389333 373 HAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGIAMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g1a A 1.42 BS02 7H1 A 1 L21 I100 H142 H143 G151 F152 D180 H182 F208 Y312 L22 I101 H143 H144 G152 F153 D181 H183 F209 Y313 3.5.1.- 0004407,0016787,0040029,0046872 Kd=0.27uM remove_due_to_license_issue Kd=540nM Q70I53 28389333 373 HHAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEIVPLLADIR 5g1a B 1.42 BS02 7H1 B 1 L21 I100 H142 H143 G151 F152 D180 H182 F208 Y312 L23 I102 H144 H145 G153 F154 D182 H184 F210 Y314 3.5.1.- 0004407,0016787,0040029,0046872 Kd=0.27uM remove_due_to_license_issue Kd=540nM Q70I53 28389333 373 HHHAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g1c A 1.81 BS02 9RB A 1 L21 H142 H143 G151 F152 D180 H182 F208 Y312 L22 H143 H144 G152 F153 D181 H183 F209 Y313 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.14uM remove_due_to_license_issue Q70I53 27756124 373 HHAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g1c B 1.81 BS02 9RB B 1 L21 A22 H142 H143 G151 F152 D180 H182 F208 Y312 L22 A23 H143 H144 G152 F153 D181 H183 F209 Y313 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.14uM remove_due_to_license_issue Q70I53 27756124 373 HHAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g1n D 2.1 BS01 PAL D 1 S1973 T1974 R1975 T1976 R2024 H2052 R2085 T2086 R2146 M2185 S54 T55 R56 T57 R105 H133 R166 T167 R227 M266 R1975 T1976 K2003 R2024 H2052 Q2055 T2145 P2184 G2210 R56 T57 K84 R105 H133 Q136 T226 P265 G291 2.1.3.2,3.5.1.2,3.5.2.3,6.3.4.16,6.3.5.5 0004070,0006207,0006520,0016597,0016743 Kd=0.017uM remove_due_to_license_issue P27708 27265852 3226 SLVGQHILSVQQFTKDQMSHLFNVAHTLRMMVQKERSLDILKGKVMASMFYEVSTRTSSSFAAAMARLGGAVLSFSEATSSVQKGESLADSVQTMSCYADVVVLRHPQPGAVELAAKHCRRPVINAGDGVGEHPTQALLDIFTIREELGTVNGMTITMVGDLKHGRTVHSLACLLTQYRVSLRYVAPPSLRMPPTVRAFVASRGTKQEEFESIEEALPDTDVLYMTRIQKERFGSTQEYEACFGQFILTPHIMTRAKKKMVVMHPMPRVNEISVEVDSDPRAAYFRQAENGMYIRMALLATVLGRF 5g1n D 2.1 BS02 PAL F 1 S2000 K2003 S81 K84 R1975 T1976 K2003 R2024 H2052 Q2055 T2145 P2184 G2210 R56 T57 K84 R105 H133 Q136 T226 P265 G291 2.1.3.2,3.5.1.2,3.5.2.3,6.3.4.16,6.3.5.5 0004070,0006207,0006520,0016597,0016743 Kd=0.017uM remove_due_to_license_issue P27708 27265852 3226 SLVGQHILSVQQFTKDQMSHLFNVAHTLRMMVQKERSLDILKGKVMASMFYEVSTRTSSSFAAAMARLGGAVLSFSEATSSVQKGESLADSVQTMSCYADVVVLRHPQPGAVELAAKHCRRPVINAGDGVGEHPTQALLDIFTIREELGTVNGMTITMVGDLKHGRTVHSLACLLTQYRVSLRYVAPPSLRMPPTVRAFVASRGTKQEEFESIEEALPDTDVLYMTRIQKERFGSTQEYEACFGQFILTPHIMTRAKKKMVVMHPMPRVNEISVEVDSDPRAAYFRQAENGMYIRMALLATVLGRF 5g1n E 2.1 BS01 PAL D 1 S2000 K2003 S82 K85 R1975 T1976 K2003 R2024 H2052 Q2055 T2145 P2184 G2210 R57 T58 K85 R106 H134 Q137 T227 P266 G292 2.1.3.2,3.5.1.2,3.5.2.3,6.3.4.16,6.3.5.5 0004070,0006207,0006520,0016597,0016743 Kd=0.017uM remove_due_to_license_issue P27708 27265852 3226 HSLVGQHILSVQQFTKDQMSHLFNVAHTLRMMVQKERSLDILKGKVMASMFYEVSTRTSSSFAAAMARLGGAVLSFSEATSSVQKGESLADSVQTMSCYADVVVLRHPQPGAVELAAKHCRRPVINAGDGVGEHPTQALLDIFTIREELGTVNGMTITMVGDLKHGRTVHSLACLLTQYRVSLRYVAPPSLRMPPTVRAFVASRGTKQEEFESIEEALPDTDVLYMTRIQKERFGSTQEYEACFGQFILTPHIMTRAKKKMVVMHPMPRVNEISVEVDSDPRAAYFRQAENGMYIRMALLATVLGRF 5g1n E 2.1 BS02 PAL E 1 S1973 T1974 R1975 T1976 R2024 H2052 R2085 R2146 Q2148 M2185 S55 T56 R57 T58 R106 H134 R167 R228 Q230 M267 R1975 T1976 K2003 R2024 H2052 Q2055 T2145 P2184 G2210 R57 T58 K85 R106 H134 Q137 T227 P266 G292 2.1.3.2,3.5.1.2,3.5.2.3,6.3.4.16,6.3.5.5 0004070,0006207,0006520,0016597,0016743 Kd=0.017uM remove_due_to_license_issue P27708 27265852 3226 HSLVGQHILSVQQFTKDQMSHLFNVAHTLRMMVQKERSLDILKGKVMASMFYEVSTRTSSSFAAAMARLGGAVLSFSEATSSVQKGESLADSVQTMSCYADVVVLRHPQPGAVELAAKHCRRPVINAGDGVGEHPTQALLDIFTIREELGTVNGMTITMVGDLKHGRTVHSLACLLTQYRVSLRYVAPPSLRMPPTVRAFVASRGTKQEEFESIEEALPDTDVLYMTRIQKERFGSTQEYEACFGQFILTPHIMTRAKKKMVVMHPMPRVNEISVEVDSDPRAAYFRQAENGMYIRMALLATVLGRF 5g1p D 3.19 BS01 CP D 1 S1973 T1976 R2024 Q2055 M2185 S53 T56 R101 Q132 M252 R1975 T1976 R2024 H2052 Q2055 T2145 P2184 G2210 R55 T56 R101 H129 Q132 T219 P251 G277 2.1.3.2,3.5.1.2,3.5.2.3,6.3.4.16,6.3.5.5 0004070,0006207,0006520,0016597,0016743 remove_due_to_license_issue P27708 27265852 3226 LVGQHILSVQQFTKDQMSHLFNVAHTLRMMVQKERSLDILKGKVMASMFYEVSTRTSSSFAAAMARLGGAVLSFSEATSSVESLADSVQTMSCYADVVVLRHPQPGAVELAAKHCRRPVINAGDGVGEHPTQALLDIFTIREELGTVNGMTITMVGDLKHGRTVHSLACLLTQYRVSLRYVAPPSMPPTVRAFVASRGKQEEFESIEEALPDTDVLYMTRIQKEREACFGQFILTPHIMTRAKKKMVVMHPMPRVNEISVEVDSDPRAAYFRQAENGMYIRMALLATVLGRF 5g1p E 3.19 BS01 CP E 1 S1973 R1975 T1976 R2024 Q2055 M2185 S55 R57 T58 R106 Q137 M261 R1975 T1976 K2003 R2024 H2052 Q2055 T2145 P2184 G2210 R57 T58 K85 R106 H134 Q137 T225 P260 G284 2.1.3.2,3.5.1.2,3.5.2.3,6.3.4.16,6.3.5.5 0004070,0006207,0006520,0016597,0016743 remove_due_to_license_issue P27708 27265852 3226 HSLVGQHILSVQQFTKDQMSHLFNVAHTLRMMVQKERSLDILKGKVMASMFYEVSTRTSSSFAAAMARLGGAVLSFSEATSSVQKGESLADSVQTMSCYADVVVLRHPQPGAVELAAKHCRRPVINAGDGVGEHPTQALLDIFTIREELGTVNGMTITMVGDLKHGRTVHSLACLLTQYRVSLRYVAPPSMPPTVRAFVASRGTKQEEFESIEEALPDTDVLYMTRIQKERFGYEACFGQFILTPHIMTRAKKKMVVMHPMPRVNEISVESDPRAAYFRQAENGMYIRMALLATVLGRF 5g1z A 1.5 BS02 U53 A 1 V96 E97 D98 F103 F105 Y211 H213 F226 S319 Y334 N365 V71 E72 D73 F78 F80 Y186 H188 F201 S294 Y309 N340 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=4.74uM remove_due_to_license_issue A5K1A2 28626547 1001 IDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 5g22 A 2.32 BS02 YN4 A 1 E97 D98 F103 F105 Y211 H213 F226 S319 L330 Y334 L388 L410 E72 D73 F78 F80 Y186 H188 F201 S294 L305 Y309 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 Ki=0.1uM remove_due_to_license_issue A5K1A2 28626547 1001 IDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 5g2b A 1.83 BS02 LQY A 1 M785 D822 V840 Y845 N867 Q874 F877 M200 D237 V255 Y260 N282 Q289 F292 3.1.4.- 0004114,0007165,0008081 Ki=0.1uM remove_due_to_license_issue Ki=100nM Q8WQX9 29672041 1003 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLETR 5g2g A 1.599 BS01 EQU A 1 Y16 D40 F86 M90 L99 D103 K116 W120 Y15 D39 F85 M89 L98 D102 K115 W119 Y16 D40 D100 D103 Y15 D39 D99 D102 5.3.3.1 0004769,0008202,0016853 Kd=0.9uM remove_due_to_license_issue P07445 27375051 1129 NLPTAQEVQGLMARYIELVDVGDIEAIVQMYADDATVEDPFGQPPIHGREQIAAFYRQGLGGGKVRACLTGPVRASHNGCGAMPFRVEMVWNGQPCALDVIDVMRFDEHGRIQTKQAYWSEVNLSVR 5g2n A 2.68 BS01 6E2 A 1 K802 W812 I831 K833 D841 I879 E880 V882 M953 I963 D964 K558 W568 I587 K589 D597 I635 E636 V638 M703 I713 D714 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=6.4nM P48736 27310202 2001 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEEWCDRKFRVKIRGIDIPVLDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIAAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 5g3m A 1.85 BS02 9JH A 1 L5 P17 M21 G28 H46 D47 I94 L5 P17 M21 G28 H46 D47 I94 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 ic50=2.2uM remove_due_to_license_issue IC50=2200nM O15496 27774123 1134 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD 5g3n A 1.8 BS03 X28 A 1 L2 F5 H6 A17 C28 G29 V30 G31 H47 D48 L2 F5 H6 A17 C28 G29 V30 G31 H47 D48 H27 G29 G31 H47 D48 Y51 Y66 D91 H27 G29 G31 H47 D48 Y51 Y66 D91 3.1.1.4 0004623,0005509,0005543,0005576,0005615,0005739,0005741,0005783,0005789,0005886,0006629,0006644,0006954,0010744,0016042,0016787,0030141,0031640,0034374,0036335,0042742,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0048471,0050482,0050729,0050830,0070062,0070374,1902563 ic50=0.012uM remove_due_to_license_issue IC50=12nM P14555 27774123 1129 ALVNFHRMIKLTTGKEAALSYGFYGCHCGVGGRGSPKDATDRCCVTHDCCYKRLEKRGCGTKFLSYKFSNSGSRISCAKQDSCRSQLCECDKAAATCFARNKTTYNKKYQYYSNKHCRGSTPRCGHH 5g3w A 1.6 BS02 C65 A 1 L21 I100 H142 H143 F152 D180 H182 F208 D268 Y312 L21 I100 H142 H143 F152 D180 H182 F208 D268 Y312 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 27756124 376 HAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g3w B 1.6 BS02 C65 B 1 L21 I100 H142 H143 F152 D180 H182 F208 D268 Y312 L21 I100 H142 H143 F152 D180 H182 F208 D268 Y312 3.5.1.- 0004407,0016787,0040029,0046872 remove_due_to_license_issue Q70I53 27756124 377 HAIGYVWNTLYGWVDTGTGSLAAANLTARMQPISHHLAHPDTKRRFHELVCASGQIEHLTPIAAVAATDADILRAHSAAHLENMKRVSNLPTGGDTGDGITMMGNGGLEIARLSAGGAVELTRRVATGELSAGYALVNPPGHHAPHNAAMGFCIFNNTSVAAGYARAVLGMERVAILDWDVHHGNGTQDIWWNDPSVLTISLHQHLCFPPDSGYSTERGAGNGHGYNINVPLPPGSGNAAYLHAMDQVVLPALRAYRPQLIIVGSGFDASMLDPLARMMVTADGFRQMARRTIDCAADICDGRIVFVQEGGYSPHYLPFCGLAVIEELTGVRSLPDPYHEFLAGMGGNTLLDAERAAIEEIVPLLADIR 5g42 A 1.72 BS02 4TU A 1 C320 H323 V376 F377 F378 F388 C63 H66 V119 F120 F121 F131 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P51449 27432277 1510 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5g43 A 2.58 BS02 5IM A 1 C320 F388 Y502 C63 F131 Y245 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P51449 27432277 1510 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5g45 A 2.07 BS02 A7W A 1 M365 V376 F377 F378 I400 F401 M101 V112 F113 F114 I136 F137 ? 0003677,0004879,0005634,0006355 Kd=500uM remove_due_to_license_issue P51449 27432277 1509 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSG 5g46 A 1.76 BS02 6VD A 1 F403 S406 K465 L466 P467 P468 F140 S143 K202 L203 P204 P205 ? 0003677,0004879,0005634,0006355 Kd=2.5mM remove_due_to_license_issue P51449 27432277 1510 GASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5g4m B 1.38 BS02 O82 B 1 L145 W146 V147 T150 P151 C220 E221 P222 P223 D228 T230 L52 W53 V54 T57 P58 C127 E128 P129 P130 D135 T137 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=138uM remove_due_to_license_issue P04637 27267810 1294 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5g4n B 1.35 BS02 O83 B 1 L145 V147 T150 C220 E221 P222 P223 D228 T230 L52 V54 T57 C127 E128 P129 P130 D135 T137 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=101uM remove_due_to_license_issue P04637 27267810 1293 SSSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLR 5g4o A 1.48 BS02 O80 A 1 L145 V147 T150 C220 E221 P222 P223 D228 T230 L50 V52 T55 C125 E126 P127 P128 D133 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=37.2uM remove_due_to_license_issue P04637 27267810 1293 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5g53 A 3.4 BS01 NEC A 1 F168 E169 N181 W246 L249 H250 N253 M270 S277 H278 F151 E152 N164 W217 L220 H221 N224 M241 S248 H249 ? 0001609,0001973,0004930,0007186,0016020 remove_due_to_license_issue Ki=16nM, IC50=3.7nM, EC50=251nM P29274 27462812 400 SSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLENLY 5g57 A 1.73 BS02 6M5 A 1 M785 N825 A837 V840 G873 Q874 F880 M200 N240 A252 V255 G288 Q289 F295 3.1.4.- 0004114,0007165,0008081 Ki=4nM remove_due_to_license_issue IC50=4.0nM, Ki=4.0nM Q8WQX9 29672041 1931 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLETR 5g5f A 2.3 BS01 GSH A 1 S14 Y16 K41 K54 I55 E67 S68 S12 Y14 K39 K52 I53 E65 S66 2.5.1.18 0004364,0005737,0005829,0006749,0009407,0009636,0016740 Kd=5.2uM remove_due_to_license_issue A0A1P8NWC2 28104507 1222 KSDVKLLGAWPSPYVMRARITLNVKSVDYELLEETLGSKSDLLLKSNPVHKKIPVLIHNDKPICESLIIVHYIDEFWSSGPSILPSDPYDRAIARFWAAYLDEKWYPSLKGIASAQGEEAKKAAVDQVGESLALIEDTYVKLSKGKPFFGGEKIGYLDIAFGCFLGWLRVTEKTSGVKFLNEAKTPHLAKWAVRFCADPAVKDVMPETEKLAEFAKLLA 5g5v A 1.8 BS02 8Z4 A 1 M785 D822 V840 T841 Y845 M861 N867 G873 Q874 F877 M203 D240 V258 T259 Y263 M279 N285 G291 Q292 F295 3.1.4.- 0004114,0007165,0008081 Ki=200nM remove_due_to_license_issue Ki=200nM Q8WQX9 29672041 1936 VKRVTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLET 5ggj A 1.424 BS01 PNA A 1 R129 Y152 D179 E180 R207 R33 Y56 D83 E84 R111 2.4.1.- Kd=17.78mM remove_due_to_license_issue Q8WZA1 27493216 301 RVLDVEVYSSRSKVYVAVDGTTVLEDEAREQGRGIHVIVLNQATGHVMAKRVFDTYSPHEDEAMVLFLNMVAPGRVLICTVKDEGSFHLKDTAKALLRSLGSQAGPALGWRDTWAFVGRKGGPVFGEKHSKSPALSSWGDPVLLKTDVPLSSA 5ggk A 1.3 BS01 MBE A 1 R129 Y152 D179 E180 R207 R33 Y56 D83 E84 R111 2.4.1.- Kd=0.29mM remove_due_to_license_issue Q8WZA1 27493216 301 RVLDVEVYSSRSKVYVAVDGTTVLEDEAREQGRGIHVIVLNQATGHVMAKRVFDTYSPHEDEAMVLFLNMVAPGRVLICTVKDEGSFHLKDTAKALLRSLGSQAGPALGWRDTWAFVGRKGGPVFGEKHSKSPALSSWGDPVLLKTDVPLSSA 5ggl A 1.27 BS01 6ZC A 1 R129 D179 E180 R207 R35 D85 E86 R113 2.4.1.- Kd=16.52mM remove_due_to_license_issue Q8WZA1 27493216 301 PRRVLDVEVYSSRSKVYVAVDGTTVLEDEAREQGRGIHVIVLNQATGHVMAKRVFDTYSPHEDEAMVLFLNMVAPGRVLICTVKDEGSFHLKDTAKALLRSLGSQAGPALGWRDTWAFVGRKGGPVFGEKHSKSPALSSWGDPVLLKTDVPLSSA 5ggn A 1.211 BS01 LEC A 1 R129 Y152 D179 R207 R33 Y56 D83 R111 2.4.1.- Kd=0.22mM remove_due_to_license_issue Q8WZA1 27493216 301 RVLDVEVYSSRSKVYVAVDGTTVLEDEAREQGRGIHVIVLNQATGHVMAKRVFDTYSPHEDEAMVLFLNMVAPGRVLICTVKDEGSFHLKDTAKALLRSLGSQAGPALGWRDTWAFVGRKGGPVFGEKHSKSPALSSWGDPVLLKTDVPLSSA 5ggo A 1.502 BS01 LEC C 1 R129 Y152 D179 E180 R207 R33 Y56 D83 E84 R111 2.4.1.- remove_due_to_license_issue Q8WZA1 27493216 1 RVLDVEVYSSRSKVYVAVDGTTVLEDEAREQGRGIHVIVLNQATGHVMAKRVFDTYSPHEDEAMVLFLNMVAPGRVLICTVKDEGSFHLKDTAKALLRSLGSQAGPALGWRDTWAFVGRKGGPVFGEKHSKSPALSSWGDPVLLKTDVPLSSA 5ggz B 2.015 BS01 6TN B 1 N51 A55 K58 D93 I96 G97 M98 F138 T184 N36 A40 K43 D78 I81 G82 M83 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.056uM remove_due_to_license_issue P07900 27933959 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGVDISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5ggz D 2.015 BS01 6TN D 1 N51 A55 D93 I96 G97 F138 T184 N36 A40 D78 I81 G82 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=0.056uM remove_due_to_license_issue P07900 27933959 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGVDISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKK 5ghv A 2.8 BS01 X5G A 1 L377 A400 M448 M450 A451 G454 P455 R498 L501 D512 L15 A38 M82 M84 A85 G88 P89 R132 L135 D146 D494 A496 R498 N499 D512 K533 D128 A130 R132 N133 D146 K163 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=12nM P43405 27504936 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 5gic A 2.352 BS02 DLC A 1 S233 I267 R270 S271 S274 W282 V296 H393 Y397 S50 I84 R87 S88 S91 W99 V113 H210 Y214 ? 0003677,0004879,0006355 Kd=330.9nM remove_due_to_license_issue P13053 27500498 501 LSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5gid A 2.151 BS02 VDP A 1 L220 L223 S233 I267 R270 S271 S274 W282 H393 Y397 F418 L38 L41 S51 I85 R88 S89 S92 W100 H211 Y215 F236 ? 0003677,0004879,0006355 Kd=769.2nM remove_due_to_license_issue P13053 27500498 501 LSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 5gj9 A 2.1 BS02 VGL A 1 K161 L177 H180 D182 L189 H237 A251 K156 L172 H175 D177 L184 H232 A246 K161 H180 D182 H237 K156 H175 D177 H232 1.14.17.4 0005507,0005634,0005783,0005794,0005829,0005886,0006952,0009505,0009506,0009693,0009727,0009815,0010030,0016491,0031418,0046872,0071398,0071732 remove_due_to_license_issue Q41931 28604689 402 KFPVVDLSKLNGEERDQTMALINEACENWGFFEIVNHGLPHDLMDKIEKMTKDHYKTCQEQKFNDMLKSKGLDNLETEVEDVDWESTFYVRHLPQSNLNDISDVSDEYRTAMKDFGKRLENLAEDLLDLLCENLGLEKGYLKKVFHGTKGPTFGTKVSNYPPCPKPEMIKGLRAHTDAGGIILLFQDDKVSGLQLLKDGDWIDVPPLNHSIVINLGDQLEVITNGKYKSVLHRVVTQQEGNRMSVASFYNPGSDAEISPATSLVEKDSEYPSFVFDDYMKLYAGVKFQPKEPRFAAMK 5gja A 2.1 BS02 6PC A 1 K161 L177 H180 D182 I187 L189 N219 H237 A251 F253 K157 L173 H176 D178 I183 L185 N215 H233 A247 F249 K161 H180 D182 H237 K157 H176 D178 H233 1.14.17.4 0005507,0005634,0005783,0005794,0005829,0005886,0006952,0009505,0009506,0009693,0009727,0009815,0010030,0016491,0031418,0046872,0071398,0071732 remove_due_to_license_issue Q41931 28604689 402 MKFPVVDLSKLNGEERDQTMALINEACENWGFFEIVNHGLPHDLMDKIEKMTKDHYKTCQEQKFNDMLKSKGLDNLETEVEDVDWESTFYVRHLPQSNLNDISDVSDEYRTAMKDFGKRLENLAEDLLDLLCENLGLEKGYLKKVFHGTKGPTFGTKVSNYPPCPKPEMIKGLRAHTDAGGIILLFQDDKVSGLQLLKDGDWIDVPPLNHSIVINLGDQLEVITNGKYKSVLHRVVTQQEGNRMSVASFYNPGSDAEISPATSLVEKDSEYPSFVFDDYMKLYAGVKFQPKEPRFAAMK 5gjd A 2.79 BS01 6V3 A 1 V50 A61 E77 Q80 L81 M104 Y106 A107 I153 H154 L163 C174 D175 F176 V25 A36 E52 Q55 L56 M79 Y81 A82 I128 H129 L138 C149 D150 F151 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 27803473 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTACGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPGRVEPYVDFAEFYRLWSVDH 5gjf A 2.89 BS01 6V4 A 1 V42 V50 A61 E77 L81 V90 M104 Y106 A107 L163 C174 D175 V17 V25 A36 E47 L51 V60 M74 Y76 A77 L133 C144 D145 D156 K158 P160 N161 I173 D175 M186 D126 K128 P130 N131 I143 D145 M156 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 27803473 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIRKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTACDIQTHMTNNKGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPGRVEPYVDFAEFYRLWSVDHG 5gjg A 2.61 BS01 6V5 A 1 V42 A61 K63 M104 Y106 A107 G110 L163 D175 F176 V17 A36 K38 M79 Y81 A82 G85 L138 D150 F151 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 27803473 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPGRVEPYVDFAEFYRLWSVDHG 5gke A 2.4 BS01 dna C 0 K71 R72 E73 K100 L128 E132 G162 I163 K181 R182 R183 Q192 Y196 K70 R71 E72 K99 L127 E131 G161 I162 K180 R181 R182 Q191 Y195 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gke A 2.4 BS02 dna D 0 Y41 R44 N76 W77 Q78 E103 R184 R191 T218 S219 G220 Y40 R43 N75 W76 Q77 E102 R183 R190 T217 S218 G219 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gke B 2.4 BS01 dna C 0 Y41 R44 A45 N76 W77 R184 E186 L187 R191 T218 G220 Y40 R43 A44 N75 W76 R183 E185 L186 R190 T217 G219 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gke B 2.4 BS02 dna D 0 K71 R72 E73 K100 S131 E132 G162 I163 K181 R182 R183 Q192 Y196 K70 R71 E72 K99 S130 E131 G161 I162 K180 R181 R182 Q191 Y195 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkf A 2.8 BS01 dna C 0 Y41 R44 A45 N76 W77 P80 R184 E186 L187 R191 T218 S219 G220 Y40 R43 A44 N75 W76 P79 R183 E185 L186 R190 T217 S218 G219 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkf A 2.8 BS02 dna D 0 K71 R72 E73 K100 S131 E132 G162 K181 R182 R183 Q192 Y196 K70 R71 E72 K99 S130 E131 G161 K180 R181 R182 Q191 Y195 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkf B 2.8 BS01 dna C 0 K71 R72 S131 E132 G162 I163 E179 K181 R182 R183 Q192 Y196 K70 R71 S130 E131 G161 I162 E178 K180 R181 R182 Q191 Y195 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkf B 2.8 BS02 dna D 0 Y41 R44 N76 W77 P80 R191 T218 G220 Y40 R43 N75 W76 P79 R190 T217 G219 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkg A 2.6 BS01 dna C 0 Y41 R44 N76 W77 P80 E103 R184 L187 R191 T218 S219 G220 Y40 R43 N75 W76 P79 E102 R183 L186 R190 T217 S218 G219 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkg A 2.6 BS02 dna D 0 K71 R72 E73 K100 E132 G162 I163 R182 R183 Q192 Y196 K70 R71 E72 K99 E131 G161 I162 R181 R182 Q191 Y195 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkg B 2.6 BS01 dna C 0 K71 R72 E73 K100 L128 E132 G162 I163 E179 K181 R182 R183 Q192 Y196 K70 R71 E72 K99 L127 E131 G161 I162 E178 K180 R181 R182 Q191 Y195 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkg B 2.6 BS02 dna D 0 Y41 R44 N76 W77 Q78 E103 R184 E186 L187 R191 T218 S219 G220 Y40 R43 N75 W76 Q77 E102 R183 E185 L186 R190 T217 S218 G219 3.1.-.- 0000014,0003676,0003677,0004519,0005737,0006259 remove_due_to_license_issue Q5JER9 27773688 1 ~ 15 SKDKVTVITSPSTEELVSLVNSALLEEAMLTIFARCKVHYDGRAKSELGSGDRVIIVKPDGSFLIHQSKKREPVNWQPPGSRVRLELRENPVLVSIRRKPRETLEVELEEVYMVSVFRAEDYEELALTGSEAEMAELIFENPEVIEPGFKPLFREKAIGTGIVAVLGRDSDGNIVVLELKRRRAELHAVRQLKSYVEILREEYGDKVRGILVAPSLTSGAKRLLEKEGLEFRKLEPPKR 5gkr A 2.1 BS01 dna T 0 F33 Y50 Y52 S54 G55 S56 N58 H95 N97 W98 F32 Y49 Y51 S53 G54 S55 N57 H97 N99 W100 remove_due_to_license_issue 29180749 1 ~ 4 VQLQESGPGLVKSSETLSLTCTVSGGSISSYFWSWIRQPPGKGLEWIGYIYYSGSTNYNPSLKSRVTISLHTSKNQFSLKLSSVTAADTAVYYCARHRNWLFDYWGQGTLVTVSSASTKGPSVFPLAPGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYTCNVDHKPSNTKVDKTVE 5gkr B 2.1 BS01 dna T 0 Y95 Y96 Y97 Y99 remove_due_to_license_issue 29180749 1 ~ 4 QSALTQPRSVSGSPGQSVTISCTGTSSDVGGYNYVSWYQQHPGKAPKVMIYDVSKRPSGVPDRFSGSKSGNTASLTISGLQAEDEADYYCCSYAGSYTYVFGTGTKVTVLGQPKANPTVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADGSPVKAGVETTKPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAPT 5glu A 2.1 BS01 GAL C 1 H192 N194 R196 W212 E215 H192 N194 R196 W212 E215 ? 0016936,0030246 remove_due_to_license_issue A0A1L1QJZ7 27742836 2 MATETNYPVPYRSKLTEPFEPGQTLIIKGKTAEDSVRFTINLHNTSADFSGNDVPLHISVRFDEGKIVFNTFSKGEWGKEERKSNPYKKGDDIDIRIRAHDSKFSISVDQKEVKEYEHRVPLSSVTHFSVDGDILITYIHWGGKYYPVPYESGLAGDGLAPGKSLLIFATPEKKGKRFHINLLKKNGDIALHFNPRFDEKAIVRNSLISGEWGNEEREGKNPLEKGIGCDLEFRNEEYAFQIYVDGERFATYAHRLDPHDINGLQIGGDVEVTGIQMV 5gmh A 2.2 BS01 RX8 A 1 D555 L557 T586 D492 L494 T523 ? 0002224,0004888,0006955,0016020 Kd=0.49uM remove_due_to_license_issue B3Y653 27742543 901 ARWFPKTLPCDVTLDVSKNHVIVDCTDKHLTEIPGGIPTNTTNLTLTINHIPDISPASFHRLVHLVEIDFRCNCVPIRLGSKSNMCPRRLQIKPRSFSGLTYLKSLYLDGNQLLEIPQGLPPSLQLLSLEANNIFSIRKEQLTELANIEILYLGQNCYYRNPCYVSYSIEKDAFLNLTKLKVLSLKDNNVTTVPTVLPSTLTELYLYNNMIAEIQEDDFNNLNQLQILDLSGNCPRCYNAPFPCTPCKNNSPLQIPVNAFDALTELKVLRLHSNSLQHVPPRWFKNINNLQELDLSQNFLAKEIGDAKFLHFLPNLIQLDLSFNFELQVYRASMNLSQAFSSLKSLKILRIRGYVFKELKSFQLSPLHNLQNLEVLDLGTNFIKIANLSMFKQFKRLKVIDLSVNKISPVLEQLYYFRYDKYARSCSCYKYGQTLDLSKNSIFFIKSSDFQHLSFLKCLNLSGNLISQTLNGSEFQPLAELRYLDFSNNRLDLLHSTAFEELRKLEVLDISSNSHYFQSEGITHMLNFTKNLKVLQKLMMNDNDISSSTSRTMESESLRTLEFRGNHLDVLWRDGDNRYLQLFKNLLKLEELDISKNSLSFLPSGVFDGMPPNLKNLSLAKNGLKSFIWEKLRYLKNLETLDLSHNQLTTVPERLSNCSRSLKNLILKNNQIRSLTKYFLQDAFQLRYLDLSSNKIQMIQKTSFPENVLNNLKMLLLHHNRFLCTCDAVWFVWWVQHTEVTIPYLATDVTCVGPGAHKGQSVISLDLYTCEL 5gmh A 2.2 BS02 RX8 B 1 F351 V355 Y356 F408 F325 V329 Y330 F382 ? 0002224,0004888,0006955,0016020 Kd=0.49uM remove_due_to_license_issue B3Y653 27742543 901 ARWFPKTLPCDVTLDVSKNHVIVDCTDKHLTEIPGGIPTNTTNLTLTINHIPDISPASFHRLVHLVEIDFRCNCVPIRLGSKSNMCPRRLQIKPRSFSGLTYLKSLYLDGNQLLEIPQGLPPSLQLLSLEANNIFSIRKEQLTELANIEILYLGQNCYYRNPCYVSYSIEKDAFLNLTKLKVLSLKDNNVTTVPTVLPSTLTELYLYNNMIAEIQEDDFNNLNQLQILDLSGNCPRCYNAPFPCTPCKNNSPLQIPVNAFDALTELKVLRLHSNSLQHVPPRWFKNINNLQELDLSQNFLAKEIGDAKFLHFLPNLIQLDLSFNFELQVYRASMNLSQAFSSLKSLKILRIRGYVFKELKSFQLSPLHNLQNLEVLDLGTNFIKIANLSMFKQFKRLKVIDLSVNKISPVLEQLYYFRYDKYARSCSCYKYGQTLDLSKNSIFFIKSSDFQHLSFLKCLNLSGNLISQTLNGSEFQPLAELRYLDFSNNRLDLLHSTAFEELRKLEVLDISSNSHYFQSEGITHMLNFTKNLKVLQKLMMNDNDISSSTSRTMESESLRTLEFRGNHLDVLWRDGDNRYLQLFKNLLKLEELDISKNSLSFLPSGVFDGMPPNLKNLSLAKNGLKSFIWEKLRYLKNLETLDLSHNQLTTVPERLSNCSRSLKNLILKNNQIRSLTKYFLQDAFQLRYLDLSSNKIQMIQKTSFPENVLNNLKMLLLHHNRFLCTCDAVWFVWWVQHTEVTIPYLATDVTCVGPGAHKGQSVISLDLYTCEL 5gmh B 2.2 BS01 RX8 A 1 F351 Y356 F408 F325 Y330 F382 ? 0002224,0004888,0006955,0016020 Kd=0.49uM remove_due_to_license_issue B3Y653 27742543 901 ARWFPKTLPCDVTLDVSKNHVIVDCTDKHLTEIPGGIPTNTTNLTLTINHIPDISPASFHRLVHLVEIDFRCNCVPIRLGSKSNMCPRRLQIKPRSFSGLTYLKSLYLDGNQLLEIPQGLPPSLQLLSLEANNIFSIRKEQLTELANIEILYLGQNCYYRNPCYVSYSIEKDAFLNLTKLKVLSLKDNNVTTVPTVLPSTLTELYLYNNMIAEIQEDDFNNLNQLQILDLSGNCPRCYNAPFPCTPCKNNSPLQIPVNAFDALTELKVLRLHSNSLQHVPPRWFKNINNLQELDLSQNFLAKEIGDAKFLHFLPNLIQLDLSFNFELQVYRASMNLSQAFSSLKSLKILRIRGYVFKELKSFQLSPLHNLQNLEVLDLGTNFIKIANLSMFKQFKRLKVIDLSVNKISPVLEQLYYFRYDKYARSCSCYKYGQTLDLSKNSIFFIKSSDFQHLSFLKCLNLSGNLISQTLNGSEFQPLAELRYLDFSNNRLDLLHSTAFEELRKLEVLDISSNSHYFQSEGITHMLNFTKNLKVLQKLMMNDNDISSSTSRTMESESLRTLEFRGNHLDVLWRDGDNRYLQLFKNLLKLEELDISKNSLSFLPSGVFDGMPPNLKNLSLAKNGLKSFIWEKLRYLKNLETLDLSHNQLTTVPERLSNCSRSLKNLILKNNQIRSLTKYFLQDAFQLRYLDLSSNKIQMIQKTSFPENVLNNLKMLLLHHNRFLCTCDAVWFVWWVQHTEVTIPYLATDVTCVGPGAHKGQSVISLDLYTCEL 5gmh B 2.2 BS02 RX8 B 1 D555 L557 T586 D492 L494 T523 ? 0002224,0004888,0006955,0016020 Kd=0.49uM remove_due_to_license_issue B3Y653 27742543 901 ARWFPKTLPCDVTLDVSKNHVIVDCTDKHLTEIPGGIPTNTTNLTLTINHIPDISPASFHRLVHLVEIDFRCNCVPIRLGSKSNMCPRRLQIKPRSFSGLTYLKSLYLDGNQLLEIPQGLPPSLQLLSLEANNIFSIRKEQLTELANIEILYLGQNCYYRNPCYVSYSIEKDAFLNLTKLKVLSLKDNNVTTVPTVLPSTLTELYLYNNMIAEIQEDDFNNLNQLQILDLSGNCPRCYNAPFPCTPCKNNSPLQIPVNAFDALTELKVLRLHSNSLQHVPPRWFKNINNLQELDLSQNFLAKEIGDAKFLHFLPNLIQLDLSFNFELQVYRASMNLSQAFSSLKSLKILRIRGYVFKELKSFQLSPLHNLQNLEVLDLGTNFIKIANLSMFKQFKRLKVIDLSVNKISPVLEQLYYFRYDKYARSCSCYKYGQTLDLSKNSIFFIKSSDFQHLSFLKCLNLSGNLISQTLNGSEFQPLAELRYLDFSNNRLDLLHSTAFEELRKLEVLDISSNSHYFQSEGITHMLNFTKNLKVLQKLMMNDNDISSSTSRTMESESLRTLEFRGNHLDVLWRDGDNRYLQLFKNLLKLEELDISKNSLSFLPSGVFDGMPPNLKNLSLAKNGLKSFIWEKLRYLKNLETLDLSHNQLTTVPERLSNCSRSLKNLILKNNQIRSLTKYFLQDAFQLRYLDLSSNKIQMIQKTSFPENVLNNLKMLLLHHNRFLCTCDAVWFVWWVQHTEVTIPYLATDVTCVGPGAHKGQSVISLDLYTCEL 5gmm A 2.003 BS02 949 A 1 H64 H94 H96 H119 L131 L198 T199 H200 H61 H91 H93 H116 L128 L195 T196 H197 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=29.1uM remove_due_to_license_issue P00915 27475498 302 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 5gmm A 2.003 BS03 949 A 2 I60 V62 H67 Q92 K170 I57 V59 H64 Q89 K167 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=29.1uM remove_due_to_license_issue P00915 27475498 303 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 5gmm A 2.003 BS04 949 A 3 A132 S136 Y204 A129 S133 Y201 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Kd=29.1uM remove_due_to_license_issue P00915 27475498 304 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 5gmn A 1.8 BS02 949 A 1 I91 H94 H119 V121 F130 L197 T198 T199 I88 H91 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=18.8uM remove_due_to_license_issue P00918 27475498 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5gmp A 2.797 BS01 F62 A 1 L718 V726 A743 M790 Q791 L792 M793 P794 G796 C797 L844 L23 V31 A48 M95 Q96 L97 M98 P99 G101 C102 L149 D837 A839 R841 N842 D855 D142 A144 R146 N147 D160 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=386nM P00533 28033579 1101 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPRALMDEEDMDDVVDADEYLIP 5gnj A 2.7 BS01 dna C 0 H453 R461 N465 K483 H2 R10 N14 K32 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 603 ~ 616 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAGR 5gnj A 2.7 BS02 dna D 0 E457 R460 E6 R9 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 804 ~ 817 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAGR 5gnj B 2.7 BS01 dna C 0 E457 R460 E9 R12 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 603 ~ 616 EPLNHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAGR 5gnj B 2.7 BS02 dna D 0 H453 E457 R458 R461 K483 H5 E9 R10 R13 K35 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 804 ~ 817 EPLNHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAGR 5gnj E 2.7 BS01 dna H 0 H453 V454 R458 R461 K483 H2 V3 R7 R10 K31 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 603 ~ 616 NHVEAERQRREKLNQRFYALRAVVPNVKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAGR 5gnj F 2.7 BS01 dna H 0 N452 E457 R460 N1 E6 R9 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 603 ~ 616 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnj F 2.7 BS02 dna J 0 H453 R461 K483 H2 R10 K32 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 805 ~ 817 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnj G 2.7 BS01 dna K 0 H453 E457 R461 K483 H2 E6 R10 K32 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 603 ~ 616 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnj I 2.7 BS01 dna L 0 H453 E457 R458 R461 H5 E9 R10 R13 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 804 ~ 817 EPLNHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELA 5gnj M 2.7 BS01 dna O 0 H453 R458 N465 K483 H2 R7 N14 K32 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 604 ~ 616 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnj M 2.7 BS02 dna P 0 E457 R460 E6 R9 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 805 ~ 816 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnj N 2.7 BS01 dna O 0 E457 R460 E6 R9 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 604 ~ 616 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnj N 2.7 BS02 dna P 0 H453 R461 D482 K483 H2 R10 D31 K32 ? 0003700,0006355,0046983 remove_due_to_license_issue Q39204 28514654 805 ~ 816 NHVEAERQRREKLNQRFYALRAVVPNVSKMDKASLLGDAIAYINELKSKVVKTESEKLQIKNQLEEVKLELAG 5gnk A 1.796 BS01 80U A 1 L718 V726 A743 K745 M766 C775 L788 M790 M793 C797 R841 L844 T854 D855 L22 V30 A47 K49 M70 C79 L92 M94 M97 C101 R145 L148 T158 D159 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 28282122 1001 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 5goe A 1.801 BS01 GDP A 1 S85 G87 K88 S89 S90 N237 R238 D240 S284 K286 S82 G84 K85 S86 S87 N220 R221 D223 S267 K269 3.6.5.- 0003924,0005525,0005741,0008053,0016020 Kd=45.7uM remove_due_to_license_issue Q8IWA4 28114303 901 PVSPLKHFVLAKKAITAIFDQLLEFVTEGSHFVEATYKNPELDRIATEDDLVEMQGYKDKLSIIGEVLSRRHMKVAFFGRTSSGKSSVINAMLWDKVLPSGIGHITNCFLSVEGTDGDKAYLMTEGSDEKKSVKTVNQLAGCLVRVFWPKAKCALLRDDLVLVDSPGTDVTDSWIDKFCLDADVFVLVANSESTLMNTEKHFFHKVNERLSKPNIFILNNRWDASASEPEYMEDVRRQHMERCLHFLVEELKVVNALEAQNRIFFVSAKEVLSARKQKAALAEGFHARLQEFQNFEQIFEECISQSAVKTKFEQHTIRAKQILATVKNIMDSVNLAAEDKRHYSARLPKEIDQLEKIQNNSKLLRNKAVQLENELENFTKQFLP 5gof A 1.604 BS01 GTP A 1 T84 S85 G87 K88 S89 S90 N237 R238 D240 S284 K286 T81 S82 G84 K85 S86 S87 N225 R226 D228 S272 K274 3.6.5.- 0003924,0005525,0005741,0008053,0016020 Kd=90.1uM remove_due_to_license_issue Q8IWA4 28114303 901 PVSPLKHFVLAKKAITAIFDQLLEFVTEGSHFVEATYKNPELDRIATEDDLVEMQGYKDKLSIIGEVLSRRHMKVAFFGRTSSGKSSVINAMLWDKVLPSGIGHITNCFLSVEGTDGDKAYLMTEGSDEKKSVKTVNQLAHALHAGCLVRVFWPKAKCALLRDDLVLVDSPGTDELDSWIDKFCLDADVFVLVANSESTLMNTEKHFFHKVNERLSKPNIFILNNRWDASASEPEYMEDVRRQHMERCLHFLVEELKVVNALEAQNRIFFVSAKEVLSARKQKVALAEGFHARLQEFQNFEQIFEECISQSAVKTKFEQHTIRAKQILATVKNIMDSVNLAAEDKRHYSARLPKEIDQLEKIQNNSKLLRNKAVQLENELENFTKQFLPS 5gpc A 2.8 BS01 dna G 0 Q29 V30 Y45 K51 Q26 V27 Y42 K48 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KKGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLR 5gpc A 2.8 BS02 dna E 0 K8 A40 G42 T43 Y47 K5 A37 G39 T40 Y44 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KKGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLR 5gpc B 2.8 BS01 dna G 0 K8 A40 G42 T43 Y47 K4 A36 G38 T39 Y43 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLRH 5gpc B 2.8 BS02 dna E 0 Q29 V30 G42 Y45 N50 K51 Q25 V26 G38 Y41 N46 K47 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLRH 5gpc C 2.8 BS01 dna G 0 K8 A40 G42 T43 L46 Y47 K5 A37 G39 T40 L43 Y44 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KKGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLR 5gpc C 2.8 BS02 dna E 0 Q29 V30 Y45 K51 Q26 V27 Y42 K48 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KKGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLR 5gpc D 2.8 BS01 dna G 0 Q29 V30 Y45 N50 K51 Q25 V26 Y41 N46 K47 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLRH 5gpc D 2.8 BS02 dna E 0 K8 A40 G42 T43 L46 Y47 K4 A36 G38 T39 L42 Y43 ? 0003677 remove_due_to_license_issue Q9K8A4 28160603 1 ~ 21 KGPKYDQIIDAAVQVIAEHGYHQAQVSKIAKAAGVADGTIYLYFNNKEDVLISLFQEKMGRFVDKIRSQMNEATDVEEKLKILVNMHFKQLAADHKLAIVTQLELRQSNTELRLKINEVLKGYLNLLDELLMEGKEKGYFFQELDTRLARQMIFGTLDEVVTNWVMKDCKYDLTALVKPVHQLLLGGLRH 5gs9 A 2.5 BS01 ARG A 1 S111 V112 L113 L273 G274 E277 I280 V281 T300 F301 F303 D304 S107 V108 L109 L258 G259 E262 I265 V266 T285 F286 F288 D289 ? 0005515,0005737,0005829,0034198,0034618,0042802,0061700,0140299,0140311,1903577,1904262,1904263 Kd=5.5uM remove_due_to_license_issue Q8WTX7 27648300 401 MELHILEHRVRVLSVARPGLWLYTHPLIKLLFLPRRSRCKFFSLTETPEDYTLMVDEEGFKELPPSEFLQVAEATWLVLNVSSHSQAAGVTKIARSVIAPLAEHHVSVLMLSTYQTDFILVREQDLSVVIHTLAQEFDIYREVGGEPVPVTRDTQHGPSPTVHPIQSPQNRFCVLTLDPETLPAIATTLIDVLFYSHSTPKESSPEPSSITFFAFSLIEGYISIVMDAETQKKFPSDLLLTSSSGELWRMVRIGGQPLGFDECGIVAQIAGPLAAADISAYYISTFNFDHALVPEDGIGSVIEVLQRRQ 5gsa A 2.49 BS02 73K A 1 F97 Y148 N194 K211 L240 D310 Y365 R367 F20 Y71 N117 K134 L163 D229 Y284 R286 ? Kd=82.5nM remove_due_to_license_issue Kd=82nM, IC50=53.5nM O75530 28135235 501 CKYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5gso A 2.6 BS01 5GI A 1 H40 E71 K130 T142 K143 C147 H161 I162 G163 G164 H40 E71 K130 T142 K143 C147 H161 I162 G163 G164 V30 H40 E71 G145 C147 V30 H40 E71 G145 C147 ? 0004197,0006508,0008234,0019062,0030430,0039618,0046718 remove_due_to_license_issue E7E815 28461310 201 GPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNVLDAVELVDEQGVNLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKIIGIHIGGNGRQGFCAGLKRSYFAS 5gsw A 3.19 BS01 5GI A 1 H40 E71 S128 K130 T142 K143 C147 H161 I162 G163 G164 H40 E71 S128 K130 T142 K143 C147 H161 I162 G163 G164 H40 E71 G145 C147 H40 E71 G145 C147 ? 0004197,0006508,0008234,0019062,0030430,0039618,0046718 remove_due_to_license_issue E7E815 28461310 201 GPSLDFALSLLRRNVRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWIEHKLVNVLDAVELVDEQGVSLELTLITLDTNEKFRDITKFIPENISTASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKIIGIHIGGNGRQGFCAGLKRSYFAS 5gty A 3.14 BS01 816 A 1 G719 V726 A743 I744 K745 R776 L777 M790 M793 G796 C797 R841 L844 D855 G20 V27 A44 I45 K46 R73 L74 M87 M90 G93 C94 R138 L141 D152 D837 A839 R841 N842 D855 D134 A136 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 28407693 1101 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDAD 5gub A 1.78 BS01 GCD D 1 W284 S287 L389 Q405 Y409 E410 W258 S261 L363 Q379 Y383 E384 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 28432302 2 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5gut A 2.099 BS01 SAH A 1 F1148 S1149 G1153 L1154 E1171 M1172 D1193 C1194 L1250 N1580 A1581 V1582 F343 S344 G348 L349 E366 M367 D388 C389 L445 N775 A776 V777 C1229 E1269 R1313 R1315 C424 E464 R508 R510 2.1.1.37 0003682,0008168 remove_due_to_license_issue P13864 29381856 1701 MKIEENRTYYQKVSIDEEMLEVGDCVSVIPDDSSKPLYLARVTALWEDKNGQMMFHAHWFCAGTDTVLGATSDPLELFLVGECENMQLSYIHSKVKVIYKAPSENWAMEGYFFQLWYNQEYARFESPPKTQPHKFCLSCIRLAELRQKEMPKVLEQIEEVDGRVYCSSITKNGVVYRLGDSVYLPPEAFTFNIKVASPDPVNETLYPEHYRKYDAPEPYRIGRIKEIHCGKKKGKVNEADIKLRLYKFYRPENTHRSYNGSYHTDINMLYWSDEEAVVNFSDVQGRCTVEYGEDLLESIQDYSQGGPDRFYFLEAYNSKTKNFEDPPNHARSPLPKLRTLDVFSGCGGLSEGFHQAGISETLWAIEMWDPAAQAFRLNNPGTTVFTEDCNVLLKLVMAGEVTNSLGQRLPQKGDVEMLCGGPPCQGFSGMNRFNSRTYSKFKASLVVSFLSYCDYYRPRFFLLENVRNFVSYRRSMVLKLTLRCLVRMGYQCTFGVLQAGQYGVAQTRRRAIILAAAPGEKLPLFPEPLHVFAPRACQLSVVVDDKKFVSNITRLSSGPFRTITVRDTMSDLPEIQNGASNSEIPYNGEPLSWFQRQLRGSHYQPILRDHICKDMSPLVAARMRHIPLFPGSDWRDLPNIQVRLGDGVIAHKLQYTFHDVKNGYSSTGALRGVCSCAEGKACDPESRQFSTLIPWCLPHTGNRHNHWAGLYGRLEWDGFFSTTVTNPEPMGKQGRVLHPEQHRVVSVRECARSQGFPDSYRFFGNILDRHRQVGNAVPPPLAKAIGLEIKLCLL 5gv2 A 2.06 BS01 ARG A 1 V112 L113 L273 G274 E277 I280 V281 T300 F301 F303 D304 V120 L121 L253 G254 E257 I260 V261 T280 F281 F283 D284 ? 0005515,0005737,0005829,0034198,0034618,0042802,0061700,0140299,0140311,1903577,1904262,1904263 remove_due_to_license_issue Q8WTX7 28066558 401 GLVPRGSHMELHILEHRVRVLSVARPGLWLYTHPLIKLLFLPRRSRCKFFSLTETPEDYTLMVDEEGFKELPPSEFLQVAEATWLVLNVSSHSGAAVQAAGVTKIARSVIAPLAEHHVSVLMLSTYQTDFILVREQDLSVVIHTLAQEFDIYREVGGEPVPVTRDDTVHPIQSPQNRFCVLTLDPETLPAIATTLIDVLFYSHPSSITFFAFSLIEGYISIVMDAETQKKFPSDLLLTSGELWRMVRIGGQPLGFDECGIVAQIAGPLAAADISAYYISTFNFDHALVPEDGIGSVIEVLQRRQ 5gvk A 2.24 BS02 G45 A 1 L124 G128 L130 F134 V141 T183 N354 N356 T357 P367 R371 L124 G128 L130 F134 V141 T183 N354 N356 T357 P367 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=99nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvk A 2.24 BS04 G45 B 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=99nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvk B 2.24 BS02 G45 A 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=99nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvk B 2.24 BS04 G45 B 1 L124 G128 H129 L130 F134 V141 T183 K355 N356 T357 C364 P367 R371 L124 G128 H129 L130 F134 V141 T183 K355 N356 T357 C364 P367 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=99nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvl A 2.5 BS02 GI8 A 1 L124 G128 H129 L130 V141 T183 N354 K355 N356 T357 C364 P367 R371 L124 G128 H129 L130 V141 T183 N354 K355 N356 T357 C364 P367 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=42nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvl A 2.5 BS04 GI8 B 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=42nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvl B 2.5 BS02 GI8 A 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=42nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvl B 2.5 BS04 GI8 B 1 L124 G128 H129 T183 N354 K355 N356 T357 C364 P367 R371 L124 G128 H129 T183 N354 K355 N356 T357 C364 P367 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=42nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvm A 2.24 BS02 G57 A 1 L124 G128 H129 T183 K355 N356 T357 L124 G128 H129 T183 K355 N356 T357 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=186nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvm A 2.24 BS04 G57 B 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=186nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvm B 2.24 BS02 G57 A 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=186nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvm B 2.24 BS04 G57 B 1 L124 G128 H129 T183 K355 N356 T357 P367 L124 G128 H129 T183 K355 N356 T357 P367 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=186nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvn A 2.3 BS02 G6F A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=90nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvn A 2.3 BS04 G6F B 1 L124 G128 T183 N356 T357 R371 L124 G128 T183 N356 T357 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=90nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvn B 2.3 BS02 G6F A 1 L124 G128 T183 N354 N356 T357 R371 L124 G128 T183 N354 N356 T357 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=90nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvn B 2.3 BS04 G6F B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=90nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvp A 2.26 BS02 GCF A 1 L124 G128 H129 T183 K355 C364 P367 L124 G128 H129 T183 K355 C364 P367 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=165nM remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvp A 2.26 BS03 GCF A 2 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 ic50=165nM remove_due_to_license_issue A5K8L9 28537728 503 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvp B 2.26 BS02 GCF A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28537728 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gvp B 2.26 BS03 GCF A 2 L124 G128 T183 K355 C364 P367 L124 G128 T183 K355 C364 P367 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28537728 503 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5gwa A 1.59 BS01 NXL A 1 S56 W93 S120 N122 T225 G226 S227 S45 W82 S109 N111 T214 G215 S216 S56 K59 S120 E156 K224 S227 S45 K48 S109 E145 K213 S216 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue A0A0B6VPP7 28739781 301 GTDSLKNSIEKYLKDKKAKVGVAVLGIEDNFKLNVNEKHHYPMQSTYKFHLALAVLDKLDKENISVDKKLFVKKSDLQPNTWSPLKDKYPNGNLELSFSEIIKSTVSHSDNNGCDILFRFVGGTNKVHNFISKLGVKNISIKATEEEMHKAWNVQYTNWTTPDATVQLLKKFYKNEILSKNSYDFLLNTMIETTTGPKRLKGLLPDGTVVAHKTGSSDTNNKGITAATNDIGIITLPNGKHFAIAVYVSDSSEKSDVNEKIIAEICKSVWDYLVK 5gx6 A 1.81 BS01 ASG D 1 H36 L37 Y146 R204 K210 R393 H10 L11 Y120 R178 K184 R367 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 28432302 1 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5gx6 A 1.81 BS02 GCD D 1 W284 S287 L389 Q405 Y409 E410 W258 S261 L363 Q379 Y383 E384 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 28432302 2 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5gx7 A 1.991 BS01 NG6 D 1 H36 Y146 R204 K210 W284 R393 H10 Y120 R178 K184 W258 R367 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 28432302 1 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5gx7 A 1.991 BS02 GCD D 1 W284 S287 L389 Q405 Y409 E410 W258 S261 L363 Q379 Y383 E384 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 28432302 2 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5gxh A 1.8 BS01 rna B 0 N13 W14 Y15 R33 R66 R359 G380 F381 Y383 Y474 T540 N582 K641 Y660 R684 N11 W12 Y13 R31 R64 R317 G338 F339 Y341 Y432 T490 N532 K591 Y610 R634 ? remove_due_to_license_issue Q8TEQ6 27881600 2 ~ 8 QEPRTLPPSPNWYCARCSDAVPGGLFGFAARTSVFLVRVGPGAGESPGTPPFRVIGELVGHTERVSGFTFSHHPGQYNLCATSSDDGTVKIWDVETKTVVTEHALHQHTISTLHWSPRVKDLIVSGDEKGVVFCYWFNRNDSQHLFIEPRTIFCLTCSPHHEDLVAIGYKDGIVVIIDISKKGEVIHRLRGHDDEIHSIAWCPLPGEGCYLATGSKDQTIRIWSCSRGRGVMILKLPFLKRRERLWLTLHWPSNQPTQLVSSCFGGELLQWDLTQRRKYTLFSASSEGQNHSRIVFNLCPLQTEDDKQLLLSTSMDRDVKCWDIATLECSWTLPSLGGFAYSLAFSSVDIGSLAIGVGDGMIRVWNTLSIKNNYDVKNFWQGVKSKVTALCWHPTKEGCLAFGTDDGKVGLYDTYSNKPPQISSTYHKKTVYTLAWGPPVPPMSSLALYSCGGEGIVLQHNPWKLSGEAFDINKLIRDTNSIKYKLPVHTEISWKADGKIMALGNEDGSIEIFQIPNLKLICTIQQHHKLVNTISWHHEHGSQPELSYLMASGSNNAVIYVHNLKTVIESSPESPVTITEPYRTLSGHTAKITSVAWSPHHDGRLVSASYDGTAQVWDALREEPLCNFRGHQGRLLCVAWSPLDPDCIYSGADDFCVHKWLTSMQDHSRPPQ 5gzb A 2.704 BS01 dna B 0 L68 Q97 S100 R108 R111 L27 Q56 S59 R67 R70 ? 0003700,0006355 remove_due_to_license_issue Q15561 28368398 1 ~ 13 VWSPDIEQSFQEALAIYPPCGRRKIILSDEGKMYGRNELIARYIKLRTGKTRTRKQVSSHIQVLARRKAREIQAKLKDQAAKDKALQSMAA 5gzb A 2.704 BS02 dna C 0 K65 I66 M74 G76 N78 E79 R95 K96 Q103 K24 I25 M33 G35 N37 E38 R54 K55 Q62 ? 0003700,0006355 remove_due_to_license_issue Q15561 28368398 1 ~ 13 VWSPDIEQSFQEALAIYPPCGRRKIILSDEGKMYGRNELIARYIKLRTGKTRTRKQVSSHIQVLARRKAREIQAKLKDQAAKDKALQSMAA 5h08 A 2.53 BS01 7WL A 1 Y1896 Q1898 W1899 P1905 R1939 Y1943 Q1977 E1980 Q1981 F1984 Y183 Q185 W186 P192 R226 Y230 Q264 E267 Q268 F271 E1831 W1899 D1901 H1932 C1933 R1939 T1940 Q1977 E129 W186 D188 H219 C220 R226 T227 Q264 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P23471 28717188 2101 GPAIPIKHFPKHVADLHASSGFTEEFEEVQSCTVDLGITADSSNHPDNKHKNRYINIVAYDHSRVKLAQLAEKDGKLTDYINANYVDGYNRPKAYIAAQGPLKSTAEDFWRMIWEHNVEVIVMITNLVEKGRRKCDQYWPADGSEEYGNFLVTQKSVQVLAYYTVRNFTLRNTKIRVVTQYHYTQWPDMGVPEYSLPVLTFVRKAAYAKRHAVGPVVVHCSAGVGRTGTYIVLDSMLQQIQHEGTVNIFGFLKHIRSQRNYLVQTEEQYVFIHDTLVEAILS 5h09 A 1.945 BS01 OOO A 1 L273 A275 V281 A293 K295 V323 L325 T338 M341 D348 L393 D404 F405 L189 A191 V197 A209 K211 V239 L241 T254 M257 D264 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=1323nM remove_due_to_license_issue P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 5h0b A 1.651 BS01 OOQ A 1 L273 A275 V281 A293 K295 V323 L325 T338 M341 D348 L393 D404 F405 L189 A191 V197 A209 K211 V239 L241 T254 M257 D264 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=11nM remove_due_to_license_issue P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 5h0e A 2.1 BS01 OOS A 1 L273 V281 A293 K295 V323 L325 T338 M341 D348 L393 D404 F405 L189 V197 A209 K211 V239 L241 T254 M257 D264 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=210nM remove_due_to_license_issue IC50=209nM P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 5h0g A 1.8 BS01 OOU A 1 L273 V281 A293 K295 V323 T338 M341 S345 D348 A390 L393 D404 F405 L189 V197 A209 K211 V239 T254 M257 S261 D264 A306 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=111nM remove_due_to_license_issue IC50=111nM P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 5h0h A 1.72 BS01 OOV A 1 L273 A275 V281 A293 K295 V323 L325 T338 M341 D348 L393 D404 F405 L189 A191 V197 A209 K211 V239 L241 T254 M257 D264 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=686nM remove_due_to_license_issue IC50=692nM P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP 5h13 A 1.9 BS01 LQA A 1 P95 F97 N146 Y148 N194 Y365 R367 R414 P30 F32 N75 Y77 N123 Y286 R288 R335 ? ic50=11.58uM remove_due_to_license_issue O75530 28072869 503 GILENLYFQGKKCKYSFKCVNSLKEDHNQPLFGVQFNWHLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5h14 A 1.9 BS02 LQB A 1 F97 Y148 N194 L240 D310 Y365 R367 R414 F22 Y73 N119 L165 D235 Y290 R292 R339 ? ic50=8.76uM remove_due_to_license_issue O75530 28072869 502 KKCKYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5h15 A 2.27 BS02 LQD A 1 F97 Y148 E238 L240 D310 Y365 R367 R414 F20 Y71 E161 L163 D226 Y281 R283 R330 ? ic50=1.57uM remove_due_to_license_issue Ki=600nM, Kd=38000nM O75530 28072869 501 CKYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5h17 A 2.3 BS02 LQE A 1 F97 Y148 N194 D310 Y365 R367 R414 F21 Y72 N118 D227 Y282 R284 R331 ? ic50=0.89uM remove_due_to_license_issue IC50=2500nM O75530 28072869 501 KCKYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5h19 A 1.9 BS02 LQF A 1 P95 F97 Y148 N194 K211 L240 D310 Y365 R367 R414 D430 P18 F20 Y71 N117 K134 L163 D228 Y283 R285 R329 D345 ? ic50=0.32uM remove_due_to_license_issue IC50=620nM O75530 28072869 501 CKYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5h1k A 1.9 BS01 rna C 0 N13 W14 Y15 R33 R66 R284 R335 G380 F381 Y383 W422 K428 E556 K579 L580 N605 Y660 N11 W12 Y13 R31 R64 R246 R293 G338 F339 Y341 W380 K386 E508 K531 L532 N557 Y612 ? remove_due_to_license_issue Q8TEQ6 27881601 -2 ~ 10 QEPRTLPPSPNWYCARCSDAVPGGLFGFAARTSVFLVRVGPGAGESPGTPPFRVIGELVGHTERVSGFTFSHHPGQYNLCATSSDDGTVKIWDVETKTVVTEHALHQHTISTLHWSPRVKDLIVSGDEKGVVFCYWFNRNDSQHLFIEPRTIFCLTCSPHHEDLVAIGYKDGIVVIIDISKKGEVIHRLRGHDDEIHSIAWCPLPGEDCLSIGCYLATGSKDQTIRIWSCSRGRGVMILKLPFKERLWLTLHWPSNQPTQLVSSCFGGELLQWDLTQKYTLFSASSEGQNHSRIVFNLCPLQTEDDKQLLLSTSMDRDVKCWDIATLECSWTLPSLGGFAYSLAFSSVDIGSLAIGVGDGMIRVWNTLSIKNNYDVKNFWQGVKSKVTALCWHPTKEGCLAFGTDDGKVGLYDTYSNKPPQISSTYHKKTVYTLAWGPPVPPMSLPSLALYSCGGEGIVLQHNPWKLSGEAFDINKLIRDTNSIKYKLPVHTEISWKADGKIMALGNEDGSIEIFQIPNLKLICTIQQHHKLVNTISWHHEHGSQPELSYLMASGSNNAVIYVHNLKTVIESSPESPVTITEPYRTLSGHTAKITSVAWSPHHDGRLVSASYDGTAQVWDALREEPLCNFRGHRGRLLCVAWSPLDPDCIYSGADDFCVHKWLTSMQDHSRPPQ 5h1k B 1.9 BS01 rna D 0 N13 W14 Y15 R33 R66 R284 R335 R359 G380 F381 Y383 W422 K428 E556 K579 L580 N605 F705 N21 W22 Y23 R41 R74 R257 R308 R332 G353 F354 Y356 W395 K401 E523 K546 L547 N572 F672 ? remove_due_to_license_issue Q8TEQ6 27881601 -1 ~ 10 GAMGIRNSMGQEPRTLPPSPNWYCARCSDAVPGGLFGFAARTSVFLVRVGPGAGESPGTPPFRVIGELVGHTERVSGFTFSHHPGQYNLCATSSDDGTVKIWDVETKTVVTEHALHQHTISTLHWSPRVKDLIVSGDEKGVVFCYWFNRNDSQHLFIEPRTIFCLTCSPHHEDLVAIGYKDGIVVIIDISKKGEVIHRLRGHDDEIHSIAWCPLPGEDCLSIGCYLATGSKDQTIRIWSCSRGRGVMILKLPFLKERLWLTLHWPSNQPTQLVSSCFGGELLQWDLTQSWRRKYTLFSASSEGQNHSRIVFNLCPLQTEDDKQLLLSTSMDRDVKCWDIATLECSWTLPSLGGFAYSLAFSSVDIGSLAIGVGDGMIRVWNTLSIKNNYDVKNFWQGVKSKVTALCWHPTKEGCLAFGTDDGKVGLYDTYSNKPPQISSTYHKKTVYTLAWGPPVPPMSLPSLALYSCGGEGIVLQHNPWKLSGEAFDINKLIRDTNSIKYKLPVHTEISWKADGKIMALGNEDGSIEIFQIPNLKLICTIQQHHKLVNTISWHHEHGSQPELSYLMASGSNNAVIYVHNLKTVIESSPESPVTITEPYRTLSGHTAKITSVAWSPHHDGRLVSASYDGTAQVWDALREEPLCNFRGHRGRLLCVAWSPLDPDCIYSGADDFCVHKWLTSMQDHSRPPQG 5h1t A 1.951 BS03 7FF A 1 A923 F924 F979 N980 A89 F90 F145 N146 2.3.2.27 Kd=0.16mM remove_due_to_license_issue O15164 28207202 1103 NEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 5h1u B 1.901 BS01 6KT B 1 A923 F924 N980 A91 F92 N148 2.3.2.27 Kd=63uM remove_due_to_license_issue O15164 28207202 1101 DWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYDCDAPKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQEDYSMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 5h1v A 2.002 BS03 7FU A 1 A923 F924 V928 Y935 C976 N980 A88 F89 V93 Y100 C139 N143 2.3.2.27 Kd=34uM remove_due_to_license_issue O15164 28207202 1103 NEDWCAVCQNGGELLCCEKCPKVFHLSCHVPTLTNFPSGEWICTFCRDLSKPEVEYKKTEGLVKLTPIDKRKCERLLLFLYCHEMSLAFQDPVPLTVPDYYKIIKNPMDLSTIKKRLQESMYSKPEDFVADFRLIFQNCAEFNEPDSEVANAGIKLENYFEELLKNLYP 5h21 A 1.591 BS01 RMR A 1 F83 L92 Y97 Y139 N140 I146 F41 L50 Y55 Y97 N98 I104 ? remove_due_to_license_issue O60885 30108844 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5h2u A 2.24 BS01 1N1 A 1 L197 A217 I218 K219 L248 I262 T264 M267 A268 G270 L319 G329 D330 L14 A34 I35 K36 L65 I79 T81 M84 A85 G87 L135 G145 D146 D312 A314 R316 N317 D330 I349 D128 A130 R132 N133 D146 I165 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM remove_due_to_license_issue Kd=7.8nM, IC50=5.3nM Q13882 27993680 501 MERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPTFKALRERLSSFTSHHHH 5h3q A 2.1 BS01 7HF A 1 L486 G488 H489 I490 F521 K544 E560 V573 M587 F589 L641 V647 H648 G667 D668 F669 G670 L795 L3 G5 H6 I7 F38 K55 E67 V80 M94 F96 L148 V154 H155 G174 D175 F176 G177 L302 D650 A652 R654 N655 D668 S677 L689 D157 A159 R161 N162 D175 S184 L196 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=6nM remove_due_to_license_issue IC50=6.0nM P04629 28159414 1001 SGLQGHIIENPQYFSDACVHHIKRRDIVLKWELGEGAFGKVFLAECHNKMLVAVKALKEARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 5h4j A 1.8 BS01 FKM A 1 V65 G99 V100 Y105 N108 G110 V112 V42 G76 V77 Y82 N85 G87 V89 A46 R85 G87 I94 D102 A23 R62 G64 I71 D79 3.6.1.23 0000287,0004170,0006226,0046081 Ki=0.13uM remove_due_to_license_issue IC50=60nM P33316 29748212 201 MQLRFARLSEHATAPTRGSARAAGYDLYSAYDYTIPPMEKAVVKTDIQIALPSGCYGRVAPRSGLAAKHFIDVGAGVIDEDYRGNVGVVLFNFGKEKFEVKKGDRIAQLICERIFYPEIEEVQALD 5h5f A 1.7 BS01 SAM A 1 L83 D84 P85 G105 D115 R116 T117 L133 Q137 M138 A143 L101 D102 P103 G123 D133 R134 T135 L151 Q155 M156 A161 2.1.1.- 0005575,0005737,0008168,0032259,0035241 Kd=37.2uM remove_due_to_license_issue Q12314 27990635 301 SHHHHHHLEVLFQGPHMASKYIIEHMEEGFSEWVILEYSQILREVGAENLILSSLPESTTEKDIPQRLLKLGLRWTTKDLKGINEDFKDLELLKDGRVCLLDPRATIDLQPEDATKFDYFVFGGILGDHPPRDRTKELKTAYPNLLISRRLGDKQMTTDTAIRTTQLIIKDRIAFEDIKFIDYPEFRFNKNEATEMPFRYVLDKEGKPILPEGMLDLIKKDSAQ 5h5o A 2.122 BS01 PCG A 1 L71 F73 K80 F88 G89 E90 H98 R100 S101 R141 N145 E146 L49 F51 K58 F66 G67 E68 H76 R78 S79 R119 N123 E124 2.7.7.65 Kd=0.293uM remove_due_to_license_issue B0RM05 23881098 201 GLHALMTAEELAFFARFGRMREIAAGQALFERGAVGTQMFIVVTGQIDLDFGEDLMLKHLGPGEFFGELGLLIGDHARSAGASASVDSRLIELAHDDFQRLVDHDPSMVAHFLRRSIVRVVNNEQ 5h5o B 2.122 BS01 PCG B 1 L71 F73 K80 G89 E90 L91 G92 H98 R100 S101 R141 N145 E146 Q147 L47 F49 K56 G65 E66 L67 G68 H74 R76 S77 R117 N121 E122 Q123 2.7.7.65 Kd=0.293uM remove_due_to_license_issue B0RM05 23881098 201 HALMTAEELAFFARFGRMREIAAGQALFERGAVGTQMFIVVTGQIDLDFGEDLMLKHLGPGEFFGELGLLIGDHARSAGASASVDSRLIELAHDDFQRLVDHDPSMVAHFLRRSIVRVVNNEQ 5h63 A 1.92 BS01 UD1 A 1 Q64 W65 F66 Y88 H200 F203 D204 R207 D239 D241 N272 G273 N338 S340 S345 S346 W347 R348 Q25 W26 F27 Y49 H161 F164 D165 R168 D200 D202 N233 G234 N299 S301 S306 S307 W308 R309 2.4.1.- 0005576,0016757,0035821,0043657,0044177,0046872,0090729,0106362 remove_due_to_license_issue Q8ZNP4 30327479 401 SGHVSFAGIDYPLLPLNHQTPLVFQWFERNPDRFGQNEIPIINTQKNPYLNNIINAAIIEKERIIGIFVDGDFSKGQRKALGKLEQNYRNIKVIYNSDLNYSMYDKKLTTIYLENITKLEAQSASERDEVLLNGVKKSLEDVLKNNPEETLISSHNKDKGHLWFDFYRNLFLLKGSDAFLEAGKPGCHHLQPGGGCIYLDADMLLTDKLGTLYLPDGIAIHVSRKDNHVSLENGIIAVNRSEHPALIKGLEIMHSKPYGDPYNDWLSKGLRHYFDGSHIQDYDAFCDFIEFKHENIIMNTSSLTASSWR 5h6v A 2.422 BS01 7HS B 1 G82 D83 G33 D34 3.4.21.91,3.6.1.15,3.6.4.13 0004252,0044423 remove_due_to_license_issue H8XX12 28689970 201 DMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLV 5h6v B 2.422 BS01 7HS B 1 H51 D129 Y130 S135 G151 N152 G153 Y161 H35 D113 Y114 S119 G135 N136 G137 Y145 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0005524 remove_due_to_license_issue H8XX12 28689970 201 ETTDGVYRVMTRKLLGSTQVGVGVMQEGVFHTMWHVTKGAALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGLSEVQLLAVPPGERAKNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQGKRE 5h85 A 1.701 BS01 5XS A 1 P1110 Q1113 V1115 L1120 N1168 V1174 P31 Q34 V36 L41 N89 V95 2.3.1.-,2.3.1.48 remove_due_to_license_issue Kd=20000nM Q92793 30258543 1201 MRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5h8b A 2.55 BS01 5Y2 A 1 V53 V66 K68 I95 V116 N118 M163 I174 D175 V52 V65 K67 I94 V115 N117 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=<3.0nM, Kd=4.9nM P68400 26985319 417 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 5h8e A 2.15 BS01 5Y3 A 1 V53 V66 K68 I95 F113 V116 N118 N161 M163 I174 D175 V52 V65 K67 I94 F112 V115 N117 N160 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=6.33pM remove_due_to_license_issue Kd=6.3nM, IC50=<3.0nM P68400 26985319 421 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 5h8g A 2.0 BS01 5Y4 A 1 V53 V66 K68 I95 F113 V116 M163 I174 D175 V51 V64 K66 I91 F109 V112 M159 I170 D171 D156 K158 N161 D175 P184 S194 D152 K154 N157 D171 P180 S190 2.7.11.1 0004672,0004674,0005524,0006468 Kd=48.2pM remove_due_to_license_issue IC50=<3.0nM, Kd=48nM P68400 26985319 421 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5h8x A 1.3 BS05 5XT A 1 I159 L160 A161 H162 L193 V194 H197 E198 H201 L214 P217 N218 Y219 A220 R222 I80 L81 A82 H83 L114 V115 H118 E119 H122 L135 P138 N139 Y140 A141 R143 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=3.1uM remove_due_to_license_issue P22894 27556138 305 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 5h9p A 2.04 BS01 TD2 A 1 R144 I145 A146 H158 N160 R162 N174 W181 E184 R186 R32 I33 A34 H46 N48 R50 N62 W69 E72 R74 ? 0030246 Kd=0.068uM remove_due_to_license_issue P17931 27416897 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5h9q B 1.931 BS01 TD2 B 1 H33 H49 R53 N62 W69 E72 R74 H30 H46 R50 N59 W66 E69 R71 ? 0005515,0005576,0005615,0005634,0005737,0006915,0007157,0030246,0070062 Kd=38uM remove_due_to_license_issue P47929 27416897 201 PHKSSLPEGIRPGTVLRIRGLVPPNASRFHVNLLCGEEQGSDAALHFNPRLDTSEVVFNSKEQGSWGREERGPGVPFQRGQPFEVLIIASDDGFKAVVGDAQYHHFRHRLPLARVRLVEVGGDVQLDSVRIF 5h9r A 1.58 BS01 TGZ A 1 R144 I145 A146 H158 N160 R162 W181 E184 S237 R32 I33 A34 H46 N48 R50 W69 E72 S125 ? 0030246 Kd=0.84uM remove_due_to_license_issue P17931 27416897 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5h9s B 1.821 BS01 TGZ B 1 H49 R53 N62 W69 E72 R74 H47 R51 N60 W67 E70 R72 ? 0005515,0005576,0005615,0005634,0005737,0006915,0007157,0030246,0070062 Kd=87uM remove_due_to_license_issue P47929 27416897 201 VPHKSSLPEGIRPGTVLRIRGLVPPNASRFHVNLLCGEEQGSDAALHFNPRLDTSEVVFNSKEQGSWGREERGPGVPFQRGQPFEVLIIASDDGFKAVVGDAQYHHFRHRLPLARVRLVEVGGDVQLDSVRIF 5ha1 A 1.35 BS01 RNE A 1 K40 R58 I77 W106 M119 K40 R58 I77 W106 M119 ? 0002138,0005501,0005504,0005515,0005634,0005654,0005737,0005811,0005829,0006776,0008289,0015908,0016918,0019841,0055088,1904768 Kd=64.1nM remove_due_to_license_issue P09455 26900151 201 PVDFTGYWKMLVNENFEEYLRALDVNVALRKIANLLKPDKEIVQDGDHMIIRTLSTFRNYIMDFQVGKEFEEDLTGIDDRKCMTTVSWDGDKLQCVQKGEKEGRGWTQWIEGDELHLEMRVEGVVCKQVFKKVQHHHHHH 5ha9 B 4.01 BS01 TP0 B 1 E102 D109 H201 Y235 S243 Y246 E103 D110 H202 Y236 S244 Y247 S243 Y246 E327 S244 Y247 E328 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue P09874 28442756 406 MKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKVEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 5hbe A 2.38 BS01 5Y6 A 1 Y32 V35 A50 K52 F97 A100 L158 A172 D173 R356 Y33 V36 A51 K53 F98 A101 L155 A169 D170 R339 D151 K153 N156 D173 N181 T196 D148 K150 N153 D170 N178 T184 2.7.11.22,2.7.11.23 0004672,0005524,0006468 ic50=2.3nM remove_due_to_license_issue IC50=2.3nM P49336 26796641 401 KMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKANQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLKVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQSNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTE 5hbh A 2.5 BS01 5Y7 A 1 Y32 V35 A50 K52 F97 A100 D103 H106 A155 L158 D173 F176 R356 Y34 V37 A52 K54 F99 A102 D105 H108 A150 L153 D168 F171 R331 D151 K153 N156 D173 T196 D146 K148 N151 D168 T177 2.7.11.22,2.7.11.23 0004672,0005524,0006468 ic50=49.2nM remove_due_to_license_issue IC50=49nM P49336 26796641 401 DKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQEPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTE 5hbj A 3.0 BS01 5Y8 A 1 V27 Y32 V35 A50 K52 I79 A100 L158 A172 D173 R356 V29 Y34 V37 A52 K54 I81 A102 L156 A170 D171 R337 D151 K153 N156 D173 N181 T196 D149 K151 N154 D171 N177 T182 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=2.3nM P49336 26796641 401 DKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKAVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFLFNSPLVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQSNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTE 5hbn A 1.602 BS01 RPI A 1 G30 T31 E32 T81 R83 G118 V119 G26 T27 E28 T77 R79 G114 V115 ? Kd=12.9uM remove_due_to_license_issue P37571 27749819 206 RFTERAQKVLALAQEEALRLGHNNIGTEHILLGLVREGEGIAAKALQALGLGSEKIQKEVESLIGRGQEMSQTIHYTPRAKKVIELSMDEARKLGHSYVGTEHILLGLIREGEGVAARVLNNLGVSLNKARQQVLQLLGSNETGS 5hbn A 1.602 BS02 RPI A 2 T7 R9 G44 I45 T105 E106 T147 G148 T3 R5 G40 I41 T101 E102 T143 G144 ? Kd=12.9uM remove_due_to_license_issue P37571 27749819 207 RFTERAQKVLALAQEEALRLGHNNIGTEHILLGLVREGEGIAAKALQALGLGSEKIQKEVESLIGRGQEMSQTIHYTPRAKKVIELSMDEARKLGHSYVGTEHILLGLIREGEGVAARVLNNLGVSLNKARQQVLQLLGSNETGS 5hbs A 0.89 BS01 RTL A 1 K40 R58 I77 W106 Q108 M119 K40 R58 I77 W106 Q108 M119 ? 0002138,0005501,0005504,0005515,0005634,0005654,0005737,0005811,0005829,0006776,0008289,0015908,0016918,0019841,0055088,1904768 Kd=18.5nM remove_due_to_license_issue P09455 26900151 201 PVDFTGYWKMLVNENFEEYLRALDVNVALRKIANLLKPDKEIVQDGDHMIIRTLSTFRNYIMDFQVGKEFEEDLTGIDDRKCMTTVSWDGDKLQCVQKGEKEGRGWTQWIEGDELHLEMRVEGVVCKQVFKKVQHHHHH 5hcl A 1.5 BS01 5Y9 A 1 P82 F83 V87 N140 I146 P41 F42 V46 N99 I105 ? ic50=6mM remove_due_to_license_issue O60885 28176838 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5hct A 1.36 BS01 61P A 1 D33 D35 Y79 G80 D81 F116 D219 G221 T222 Y226 I300 D33 D35 Y79 G80 D81 F116 D219 G221 T222 Y226 I300 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=0.0254uM remove_due_to_license_issue P11838 27400756 406 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 5hcv A 2.5 BS01 60R A 1 L769 N770 M807 S810 L814 F829 M845 L938 F941 C942 T945 L28 N29 M66 S69 L73 F88 M104 L192 F195 C196 T199 ? Ki=2nM remove_due_to_license_issue P08235 26897089 1001 PVMVLENIEPEIVYAGYPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLSSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFH 5hcx A 2.6 BS01 60B A 1 L718 F723 V726 A743 K745 M766 C775 M790 Q791 M793 N842 L844 T854 D855 L23 F28 V31 A48 K50 M68 C77 M92 Q93 M95 N144 L146 T156 D157 D837 A839 R841 N842 D855 D139 A141 R143 N144 D157 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 27564586 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFDMDDVVDADEYLI 5hcy A 2.46 BS01 60D A 1 L718 F723 A743 K745 M766 C775 M790 Q791 M793 G796 N842 L844 T854 D855 L23 F28 A48 K50 M69 C78 M93 Q94 M96 G99 N145 L147 T157 D158 D837 A839 R841 N842 D855 D140 A142 R144 N145 D158 2.7.10.1 0004672,0004713,0005524,0006468 Ki=1.2nM remove_due_to_license_issue P00533 27564586 1102 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYDMDDVVDADEYLIP 5hd0 A 1.65 BS01 60Y A 1 Q73 G74 L91 D93 S96 V130 Y132 F169 I179 D289 G291 T292 Q16 G17 L34 D36 S39 V73 Y75 F112 I122 D232 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=4nM remove_due_to_license_issue P56817 26937601 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hdu A 1.58 BS01 60W A 1 G74 D93 S96 N98 V130 T133 Q134 W137 I171 D289 G291 T292 G17 D36 S39 N41 V73 T76 Q77 W80 I114 D232 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=1nM remove_due_to_license_issue Ki=1.000000nM, IC50=18nM P56817 26937601 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hdv A 1.71 BS01 60V A 1 L91 D93 S96 N98 I179 R189 D289 G291 L34 D36 S39 N41 I119 R129 D229 G231 D93 S96 N98 A100 D289 T292 D36 S39 N41 A43 D229 T232 3.4.23.46 0004190,0006508,0016020 Ki=15nM remove_due_to_license_issue Ki=15nM, IC50=40nM P56817 26937601 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hdx A 1.602 BS01 60U A 1 L91 D93 S96 N98 V130 Y132 W176 I179 R189 D289 G291 L34 D36 S39 N41 V73 Y75 W119 I122 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=48nM remove_due_to_license_issue Ki=48nM, IC50=361nM P56817 26937601 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hdz A 1.49 BS01 954 A 1 L91 D93 S96 V130 Y132 W176 I179 R189 D289 G291 L34 D36 S39 V73 Y75 W119 I122 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=45nM remove_due_to_license_issue IC50=36nM, Ki=45nM P56817 26937601 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5he0 A 2.56 BS01 453 A 1 I197 G198 R199 G200 G201 F202 G203 V205 A218 L235 M274 L324 S334 D335 I168 G169 R170 G171 G172 F173 G174 V176 A189 L206 M245 L295 S305 D306 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 remove_due_to_license_issue P21146 27050625 701 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 5he1 A 3.15 BS01 ZS2 A 1 G198 R199 G200 F202 G203 A218 L235 M274 A321 L324 S334 D335 G170 R171 G172 F174 G175 A190 L207 M246 A293 L296 S306 D307 D317 K319 N322 D335 K344 T353 D289 K291 N294 D307 K316 T325 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue IC50=2600nM P25098 27050625 701 SKKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 5he2 A 2.79 BS01 F0S A 1 I197 R199 G200 F202 G203 A218 L222 M274 L324 S334 D335 G337 L338 I168 R170 G171 F173 G174 A189 L193 M245 L295 S305 D306 G308 L309 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 remove_due_to_license_issue IC50=130nM P21146 27050625 701 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGSFDEEDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 5he3 A 2.74 BS02 FF1 A 1 I197 R199 G200 G201 F202 V205 A218 D272 M274 L324 S334 D335 I168 R170 G171 G172 F173 V176 A189 D243 M245 L295 S305 D306 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 remove_due_to_license_issue P21146 27050625 702 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKPRS 5he4 A 1.53 BS01 60T A 1 D93 S96 N98 V130 Y132 W137 F169 W176 I179 R189 D289 G291 D36 S39 N41 V73 Y75 W80 F112 W119 I122 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=20nM remove_due_to_license_issue P56817 26937601 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5he5 A 1.55 BS01 60S A 1 L91 D93 S96 V130 Y132 F169 W176 R189 D289 G291 L34 D36 S39 V73 Y75 F112 W119 R132 D232 G234 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=336nM remove_due_to_license_issue IC50=157nM, Ki=336nM P56817 26937601 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5he7 A 1.71 BS01 60X A 1 D93 S96 N98 V130 Y132 F169 W176 I179 R189 D289 G291 D36 S39 N41 V73 Y75 F110 W117 I120 R130 D230 G232 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D230 T233 3.4.23.46 0004190,0006508,0016020 Ki=5nM remove_due_to_license_issue IC50=14nM, Ki=4.7nM P56817 26937601 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hes A 2.14 BS01 032 A 1 G23 F27 V30 A43 I66 I80 T82 E83 Y84 A85 C150 D151 F152 G153 G18 F22 V25 A38 I61 I75 T77 E78 Y79 A80 C145 D146 F147 G148 D133 K135 R137 N138 D151 T169 D128 K130 R132 N133 D146 T158 2.7.11.25 0004672,0005524,0006468 Kd=29nM remove_due_to_license_issue IC50=23nM Q9NYL2 26999302 401 ASFVQIKFDDLQFFENCGGGSFGSVYRAKWISQDKEVAVKKLLKIEKEAEILSVLSHRNIIQFYGVILEPPNYGIVTEYASLGSLYDYINSNRSEEMDMDHIMTWATDVAKGMHYLHMEAPVKVIHRDLKSRNVVIAADGVLKICDFGASRFHNHTGTFPWMAPEVIQSLPVSETCDTYSYGVVLWEMLTREVPFKGLEGLQVAWLVVEKNERLTIPSSCPRSFAELLHQCWEADAKKRPSFKQIISILESMSNDTSLPDKCNSFLHNKAEWRCEIEATLERLKKLER 5hex A 2.734 BS01 604 A 1 S155 P157 N208 D209 I229 G231 T232 G233 N235 E260 Q291 E294 G414 S415 S136 P138 N177 D178 I198 G200 T201 G202 N204 E229 Q260 E263 G383 S384 R539 S603 K618 D657 R508 S572 K587 D626 2.7.1.1 0001666,0001678,0002931,0004340,0004396,0005515,0005524,0005536,0005737,0005739,0005741,0005813,0005829,0005975,0006002,0006006,0006096,0007595,0008637,0008865,0016020,0016301,0016529,0016773,0019318,0035795,0043231,0045766,0046324,0046835,0051156,0061621,0072655,0072656,1905091,1990830,2000378 remove_due_to_license_issue P52789 26985301 1001 DQVQKVDQYLYHMRLSDETLLEISKRFRKEMEKGLGATTHPTAAVKMLPTFVRSTPDGTEHGEFLALDLGGTNFRVLWVKVTDNGLQKVEMENQIYAIPEDISGTQLFDHIAECLANFMDKLQIKDKKLPLGFTFSFPCHQTKLDESFLVGRDVVALIRKAIQRRGDFDIDIVAVVNDTVGTMMTCGYDDHNCEIGLIVGTGSNACYMEEMRHIDMVEGDEGRMCINMEWGAFGDDGSLNDIRTEFDQEIDMGSLNPGKQLFEKMISGMYMGELVRLILVKMAKEELLFGGKLSPELLNTGRFETKDISDIEGEKDGIRKAREVLMRLGLDPTQEDCVATHRICQIVSTRSASLCAATLAAVLQRIKENKGEERLRSTIGVDGSVYKKHPHFAKRLHKTVRRLVPGCDVRFLRSEDGSGKGAAMVTAVAYRLADQHRARQKTLEHLQLSHDQLLEVKRRMKVEMERGLSKETHASAPVKMLPTYVCATPDGTEKGDFLALDLGGTNFRVLLVRVRNGKWGGVEMHNKIYAIPQEVMHGTGDELFDHIVQCIADFLEYMGMKGVSLPLGFTFSFPCQQNSLDESILLKWTKGFKASGCEGEDVVTLLKEAIHRREEFDLDVVAVVNDTVGTMMTCGFEDPHCEVGLIVGTGSNACYMEEMRNVELVEGEEGRMCVNMEWGAFGDNGCLDDFRTEFDVAVDELSLNPGKQRFEKMISGMYLGEIVRNILIDFTKRGLLFRGRISERLKTRGIFETKFLSQIESDCLALLQVRAILQHLGLESTCDDSIIVKEVCTVVARRAAQLCGAGMAAVVDRIRENRGLDALKVTVGVDGTLYKLHPHFAKVMHETVKDLAPKCDVSFLQSEDGSGKGAALITAVACRI 5hex A 2.734 BS02 604 A 2 D657 I677 G679 T680 N683 E708 D861 G862 T863 D626 I646 G648 T649 N652 E677 D830 G831 T832 R539 S603 K618 D657 R508 S572 K587 D626 2.7.1.1 0001666,0001678,0002931,0004340,0004396,0005515,0005524,0005536,0005737,0005739,0005741,0005813,0005829,0005975,0006002,0006006,0006096,0007595,0008637,0008865,0016020,0016301,0016529,0016773,0019318,0035795,0043231,0045766,0046324,0046835,0051156,0061621,0072655,0072656,1905091,1990830,2000378 remove_due_to_license_issue P52789 26985301 1002 DQVQKVDQYLYHMRLSDETLLEISKRFRKEMEKGLGATTHPTAAVKMLPTFVRSTPDGTEHGEFLALDLGGTNFRVLWVKVTDNGLQKVEMENQIYAIPEDISGTQLFDHIAECLANFMDKLQIKDKKLPLGFTFSFPCHQTKLDESFLVGRDVVALIRKAIQRRGDFDIDIVAVVNDTVGTMMTCGYDDHNCEIGLIVGTGSNACYMEEMRHIDMVEGDEGRMCINMEWGAFGDDGSLNDIRTEFDQEIDMGSLNPGKQLFEKMISGMYMGELVRLILVKMAKEELLFGGKLSPELLNTGRFETKDISDIEGEKDGIRKAREVLMRLGLDPTQEDCVATHRICQIVSTRSASLCAATLAAVLQRIKENKGEERLRSTIGVDGSVYKKHPHFAKRLHKTVRRLVPGCDVRFLRSEDGSGKGAAMVTAVAYRLADQHRARQKTLEHLQLSHDQLLEVKRRMKVEMERGLSKETHASAPVKMLPTYVCATPDGTEKGDFLALDLGGTNFRVLLVRVRNGKWGGVEMHNKIYAIPQEVMHGTGDELFDHIVQCIADFLEYMGMKGVSLPLGFTFSFPCQQNSLDESILLKWTKGFKASGCEGEDVVTLLKEAIHRREEFDLDVVAVVNDTVGTMMTCGFEDPHCEVGLIVGTGSNACYMEEMRNVELVEGEEGRMCVNMEWGAFGDNGCLDDFRTEFDVAVDELSLNPGKQRFEKMISGMYLGEIVRNILIDFTKRGLLFRGRISERLKTRGIFETKFLSQIESDCLALLQVRAILQHLGLESTCDDSIIVKEVCTVVARRAAQLCGAGMAAVVDRIRENRGLDALKVTVGVDGTLYKLHPHFAKVMHETVKDLAPKCDVSFLQSEDGSGKGAALITAVACRI 5hfj A 3.1 BS01 SAM A 1 D8 A9 D29 P30 K165 K167 F195 M196 G197 S198 T200 E216 S217 Y221 D8 A9 D29 P30 K139 K141 F165 M166 G167 S168 T170 E186 S187 Y191 D29 P30 D29 P30 2.1.1.- 0003676,0003677,0005737,0008168,0008170,0009007,0009307,0032259 remove_due_to_license_issue O24891 27259995 301 MIQIYHADAFEIIKDFYQQNLKVDAIITDPPYNFKLLEWIARYAPLVNPNGCMVIFCSYRFISYIADFLEENGFVVKDFIQWVKNNPMPRNIHRRYVQDTEFALWAVKKKAKWVFNKPKNEKYLRPLILKSPVVSGLEKTKHSLALMEKIISIHTNPNDIVLDPFMGSGTTGLACKNLERNFIGIESEKEYFQTAKKRLNL 5hfu A 2.923 BS01 603 A 1 K62 S155 P157 C158 N208 D209 G233 N235 E260 Q291 E294 K46 S139 P141 C142 N192 D193 G217 N219 E244 Q275 E278 R539 S603 K618 D657 R523 S587 K602 D641 2.7.1.1 0001666,0001678,0002931,0004340,0004396,0005515,0005524,0005536,0005737,0005739,0005741,0005813,0005829,0005975,0006002,0006006,0006096,0007595,0008637,0008865,0016020,0016301,0016529,0016773,0019318,0035795,0043231,0045766,0046324,0046835,0051156,0061621,0072655,0072656,1905091,1990830,2000378 remove_due_to_license_issue P52789 26985301 1001 DQVQKVDQYLYHMRLSDETLLEISKRFRKEMEKGLGATTHPTAAVKMLPTFVRSTPDGTEHGEFLALDLGGTNFRVLWVKVTDNGLQKVEMENQIYAIPEDIMRGSGTQLFDHIAECLANFMDKLQIKDKKLPLGFTFSFPCHQTKLDESFLVSWTKGFKSSGVEGRDVVALIRKAIQRRGDFDIDIVAVVNDTVGTMMTCGYDDHNCEIGLIVGTGSNACYMEEMRHIDMVEGDEGRMCINMEWGAFGDDGSLNDIRTEFDQEIDMGSLNPGKQLFEKMISGMYMGELVRLILVKMAKEELLFGGKLSPELLNTGRFETKDISDIEGEKDGIRKAREVLMRLGLDPTQEDCVATHRICQIVSTRSASLCAATLAAVLQRIKENKGEERLRSTIGVDGSVYKKHPHFAKRLHKTVRRLVPGCDVRFLRSEDGSGKGAAMVTAVAYRLADQHRARQKTLEHLQLSHDQLLEVKRRMKVEMERGLSKETHASAPVKMLPTYVCATPDGTEKGDFLALDLGGTNFRVLLVRVRNGKWGGVEMHNKIYAIPQEVMHGTGDELFDHIVQCIADFLEYMGMKGVSLPLGFTFSFPCQQNSLDESILLKWTKGFKASGCEGEDVVTLLKEAIHRREEFDLDVVAVVNDTVGTMMTCGFEDPHCEVGLIVGTGSNACYMEEMRNVELVEGEEGRMCVNMEWGAFGDNGCLDDFRTEFDVAVDELSLNPGKQRFEKMISGMYLGEIVRNILIDFTKRGLLFRGRISERLKTRGIFETKFLSQIESDCLALLQVRAILQHLGLESTCDDSIIVKEVCTVVARRAAQLCGAGMAAVVDRIRENRGLDALKVTVGVDGTLYKLHPHFAKVMHETVKDLAPKCDVSFLQSEDGSGKGAALITAVACRI 5hfu A 2.923 BS02 603 A 2 K621 N656 D657 I677 G681 S682 N683 E708 Q739 E742 K605 N640 D641 I661 G665 S666 N667 E692 Q723 E726 R539 S603 K618 D657 R523 S587 K602 D641 2.7.1.1 0001666,0001678,0002931,0004340,0004396,0005515,0005524,0005536,0005737,0005739,0005741,0005813,0005829,0005975,0006002,0006006,0006096,0007595,0008637,0008865,0016020,0016301,0016529,0016773,0019318,0035795,0043231,0045766,0046324,0046835,0051156,0061621,0072655,0072656,1905091,1990830,2000378 remove_due_to_license_issue P52789 26985301 1002 DQVQKVDQYLYHMRLSDETLLEISKRFRKEMEKGLGATTHPTAAVKMLPTFVRSTPDGTEHGEFLALDLGGTNFRVLWVKVTDNGLQKVEMENQIYAIPEDIMRGSGTQLFDHIAECLANFMDKLQIKDKKLPLGFTFSFPCHQTKLDESFLVSWTKGFKSSGVEGRDVVALIRKAIQRRGDFDIDIVAVVNDTVGTMMTCGYDDHNCEIGLIVGTGSNACYMEEMRHIDMVEGDEGRMCINMEWGAFGDDGSLNDIRTEFDQEIDMGSLNPGKQLFEKMISGMYMGELVRLILVKMAKEELLFGGKLSPELLNTGRFETKDISDIEGEKDGIRKAREVLMRLGLDPTQEDCVATHRICQIVSTRSASLCAATLAAVLQRIKENKGEERLRSTIGVDGSVYKKHPHFAKRLHKTVRRLVPGCDVRFLRSEDGSGKGAAMVTAVAYRLADQHRARQKTLEHLQLSHDQLLEVKRRMKVEMERGLSKETHASAPVKMLPTYVCATPDGTEKGDFLALDLGGTNFRVLLVRVRNGKWGGVEMHNKIYAIPQEVMHGTGDELFDHIVQCIADFLEYMGMKGVSLPLGFTFSFPCQQNSLDESILLKWTKGFKASGCEGEDVVTLLKEAIHRREEFDLDVVAVVNDTVGTMMTCGFEDPHCEVGLIVGTGSNACYMEEMRNVELVEGEEGRMCVNMEWGAFGDNGCLDDFRTEFDVAVDELSLNPGKQRFEKMISGMYLGEIVRNILIDFTKRGLLFRGRISERLKTRGIFETKFLSQIESDCLALLQVRAILQHLGLESTCDDSIIVKEVCTVVARRAAQLCGAGMAAVVDRIRENRGLDALKVTVGVDGTLYKLHPHFAKVMHETVKDLAPKCDVSFLQSEDGSGKGAALITAVACRI 5hg1 A 2.76 BS01 62C A 1 P605 K618 T620 K621 N656 D657 I677 G681 N683 E708 N735 K738 Q739 E742 P559 K572 T574 K575 N610 D611 I631 G635 N637 E662 N689 K692 Q693 E696 R539 S603 K618 D657 R496 S557 K572 D611 2.7.1.1 0001666,0001678,0002931,0004340,0004396,0005515,0005524,0005536,0005737,0005739,0005741,0005813,0005829,0005975,0006002,0006006,0006096,0007595,0008637,0008865,0016020,0016301,0016529,0016773,0019318,0035795,0043231,0045766,0046324,0046835,0051156,0061621,0072655,0072656,1905091,1990830,2000378 remove_due_to_license_issue P52789 26985301 1001 DQVQKVDQYLYHMRLSDETLLEISKRFRKEMEKGLGATTHPTAAVKMLPTFVRSTPDGTEHGEFLALDLGGTNFRVLWVKVTDNGLQKVEMENQIYGTQLFDHIAECLANFMDKLQIKDKKLPLGFTFSFPCHQTKLDESFLVSGRDVVALIRKAIQIDIVAVVNDTVGTMMTCGYDDHNCEIGLIVGTGSNACYMEEMRHIDMVEGDEGRMCINMEWGAFGDDGSLNDIRTEFDQEIDMGSLNPGKQLFEKMISGMYMGELVRLILVKMAKEELLFGGKLSPELLNTGRFETKDISDIEGEKDGIRKAREVLMRLGLDPTQEDCVATHRICQIVSTRSASLCAATLAAVLQRIKENKGEERLRSTIGVDGSVYKKHPHFAKRLHKTVRRLVPGCDVRFLRSEDGSGKGAAMVTAVAYRLADQHRARQKTLEHLQLSHDQLLEVKRRMKVEMERGLSKETHASAPVKMLPTYVCATPDGTEKGDFLALDLGGTNFRVLLVRVRNGGVEMHNKIYAIPQEVMHGTGDELFDHIVQCIADFLEYMGMKGVSLPLGFTFSFPCQQNSLDESILLKWTKGFKASGCEGEDVVTLLKEAIHRREEFDLDVVAVVNDTVGTMMTCGFEDPHCEVGLIVGTGSNACYMEEMRNVELVEGEEGRMCVNMEWGAFGDNGCLDDFRTEFDVAVDELSLNPGKQRFEKMISGMYLGEIVRNILIDFTKRGLLFRGRISERLKTRGIFETKFLSQIESDCLALLQVRAILQHLGLESTCDDSIIVKEVCTVVARRAAQLCGAGMAAVVDRIRENRGLDALKVTVGVDGTLYKLHPHFAKVMHETVKDLAPKCDVSFLQSEDGSGKGAALITAVACRIRE 5hg1 A 2.76 BS02 62C A 2 D209 N235 E260 K290 E294 D166 N192 E217 K247 E251 R539 S603 K618 D657 R496 S557 K572 D611 2.7.1.1 0001666,0001678,0002931,0004340,0004396,0005515,0005524,0005536,0005737,0005739,0005741,0005813,0005829,0005975,0006002,0006006,0006096,0007595,0008637,0008865,0016020,0016301,0016529,0016773,0019318,0035795,0043231,0045766,0046324,0046835,0051156,0061621,0072655,0072656,1905091,1990830,2000378 remove_due_to_license_issue P52789 26985301 1002 DQVQKVDQYLYHMRLSDETLLEISKRFRKEMEKGLGATTHPTAAVKMLPTFVRSTPDGTEHGEFLALDLGGTNFRVLWVKVTDNGLQKVEMENQIYGTQLFDHIAECLANFMDKLQIKDKKLPLGFTFSFPCHQTKLDESFLVSGRDVVALIRKAIQIDIVAVVNDTVGTMMTCGYDDHNCEIGLIVGTGSNACYMEEMRHIDMVEGDEGRMCINMEWGAFGDDGSLNDIRTEFDQEIDMGSLNPGKQLFEKMISGMYMGELVRLILVKMAKEELLFGGKLSPELLNTGRFETKDISDIEGEKDGIRKAREVLMRLGLDPTQEDCVATHRICQIVSTRSASLCAATLAAVLQRIKENKGEERLRSTIGVDGSVYKKHPHFAKRLHKTVRRLVPGCDVRFLRSEDGSGKGAAMVTAVAYRLADQHRARQKTLEHLQLSHDQLLEVKRRMKVEMERGLSKETHASAPVKMLPTYVCATPDGTEKGDFLALDLGGTNFRVLLVRVRNGGVEMHNKIYAIPQEVMHGTGDELFDHIVQCIADFLEYMGMKGVSLPLGFTFSFPCQQNSLDESILLKWTKGFKASGCEGEDVVTLLKEAIHRREEFDLDVVAVVNDTVGTMMTCGFEDPHCEVGLIVGTGSNACYMEEMRNVELVEGEEGRMCVNMEWGAFGDNGCLDDFRTEFDVAVDELSLNPGKQRFEKMISGMYLGEIVRNILIDFTKRGLLFRGRISERLKTRGIFETKFLSQIESDCLALLQVRAILQHLGLESTCDDSIIVKEVCTVVARRAAQLCGAGMAAVVDRIRENRGLDALKVTVGVDGTLYKLHPHFAKVMHETVKDLAPKCDVSFLQSEDGSGKGAALITAVACRIRE 5hg5 A 1.52 BS01 633 A 1 L718 A743 C775 Q791 M793 P794 G796 C797 R841 L844 L19 A44 C76 Q92 M94 P95 G97 C98 R142 L145 D837 A839 R841 N842 D855 G874 D138 A140 R142 N143 D156 G175 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26756222 9001 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRAL 5hg7 A 1.85 BS01 630 A 1 L718 F723 V726 A743 C775 M790 Q791 M793 P794 G796 C797 R841 L844 F856 L17 F22 V25 A42 C71 M86 Q87 M89 P90 G92 C93 R137 L140 F152 D837 A839 R841 N842 D855 G874 D133 A135 R137 N138 D151 G170 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26756222 9001 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGD 5hg8 A 1.42 BS01 634 A 1 L718 A743 C775 Q791 M793 G796 C797 R841 L844 L19 A44 C76 Q92 M94 G97 C98 R142 L145 D837 A839 R841 N842 D855 G874 D138 A140 R142 N143 D156 G175 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26756222 9001 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYR 5hg9 A 2.15 BS01 63A A 1 L718 G719 S720 F723 V726 A743 M793 G796 C797 R841 L844 L17 G18 S19 F22 V25 A42 M88 G91 C92 R136 L139 D837 A839 R841 N842 D855 G874 D132 A134 R136 N137 D150 G169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 26756222 9001 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 5hgc A 2.43 BS01 HCY A 1 P33 R246 F256 K274 I277 Q278 S281 F380 N385 P13 R226 F236 K254 I257 Q258 S261 F355 N360 ? 0004867,0005615 remove_due_to_license_issue H0ZQY2 501 SNAEAMAALKLVPNNADFAFQFFREVTQEAPNKNIFYSPVSISTAFAMLALGARSATQSQILEGLAFNLTEIQEKEIHEGFHNLIHMLNHPEGGVQLNMMNAIFVTAALALLRKFLDDAKALYQLEAFTTDFNKPTEAEKQINDYIERKTHGKITNLVKDMDPQTVMLLASFVYFKGSWEKPFEAEHTEEREFFVDAETTVKVPMMYQMGRFDFYFDEELSCTVVRLHYNGSATAFLVLPAKGKMKQLEQTLDKETIQKWSDHLFQRFMNLYFPKFSISGSYEISNTLRKMGIVDVFTNQADLSGITGSPDLKVSKVVHKASLDVDEKGTTAVEIMPISFPPTIEFSHPFLMLIFDRDTNSTLFIGKIVNPTI 5hgq A 3.283 BS02 KRS A 1 E257 H263 N264 F267 E427 I428 V429 G483 R486 E240 H246 N247 F250 E404 I405 V406 G443 R446 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 remove_due_to_license_issue 27806050 602 EYFKLRTALINERRSKGINPYPHKFHVSISLADFIAKYNSLEKDVILNDIVQSVAGRVFSKREKLIFYDLHGEGTRLQVLANARFHSGDEAFDNLHDRIKRGDIIGVNGYPARSKSGELSIIPYEIIQLTPCLHMLPHETRYRMRYLDLIMNPDVKNRFVTRSRMISFLRRYLDNLGFLEVETPMMNLIAGGATAKPFITHHNDLDMDLYLRVAPELYLKMLVVGGIDRVYEIGRVFRNEGIDQTHNPEFTSCEFYMAYADYEDLMKITEDMLARMVYYMHGTYKIQYHPNGIVENPVYEVDFTPPFRKVNIYDGLQEKLGIQFPPADTLDTDEANKFFDKLAVEAPRTTARLLDKLIGEFLEPTFISPTFLTGHPQIMSPLAKWHRSIPGLTERFELFVVTKEIVNAYTELNDPLTQRLRFDENYCTALEYGLPPTAGWGMGIDRLAMILTDSNNIKEVLFFPA 5hi7 A 2.15 BS05 62X A 1 R14 N16 Y124 N132 C180 N181 F183 S202 N205 H206 Y239 Y257 F259 R12 N14 Y122 N130 C178 N179 F181 S200 N203 H204 Y237 Y255 F257 2.1.1.354 0000978,0000993,0001162,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0008168,0014904,0032259,0042054,0045184,0045944,0046872,0071549,0140939,0140954,0140999 Ki=14nM remove_due_to_license_issue Q9H7B4 27066749 507 PLKVEKFATANRGNGLRAVTPLRPGELLFRSDPLAYTVCKGSRGVVCDRCLLGKEKLMRCSQCRVAKYCSAKCQKKAWPDHKRECKCLKSCKPRYPPDSVRLLGRVVFKLMDGAPSESEKLYSFYDLESNINKLTEDKKEGLRQLVMTFQHFMREEIQDASQLPPAFDLFEAFAKVICNSFTICNAEMQEVGVGLYPSISLLNHSCDPNCSIVFNGPHLLLRAVRDIEVGEELTICYLDMLMTSEERRKQLRDQYCFECDCFRCQTQDKDADMLTGDEQVWKEVQESLKKIEELKAHWKWEQVLAMCQAIISSNSERLPDINIYQLKVLDCAMDACINLGLLEEALFYGTRTMEPYRIFFPGSHPVRGVQVMKVGKLQLHQGMFPQAMKNLRLAFDIMRVTHGREHSLIEDLILLLEECDANIRAS 5hip A 1.992 BS03 61O A 1 H71 D73 H159 D178 L193 F195 H221 L277 S285 H72 D74 H160 D179 L194 F196 H222 L278 S286 3.1.2.32 0016787,0044550,0046872 Kd=0.9uM remove_due_to_license_issue P20581 27082157 403 HMLRLSAPGQLDDDLCLLGDVQVPVFLLRLGEASWALVEGGISRDAELVWADLCRWVADPSQVHYWLITHKHYDHCGLLPYLCPRLPNVQVLASERTCQAWKSESAVRVVERLNRQLLRAEQRLPEACAWDALPVRAVADGEWLELGPRHRLQVIEAHGHSDDHVVFYDVRRRRLFCGDALGEFDEAEGVWRPLVFDDMEAYLESLERLQRLPTLLQLIPGHGGLLRGRLAADGAESAYTECLRLCRRLLWRQSMGESLDELSEELHRAWGGQSVDFLPGELHLGSMRRMLEILSRQA 5his A 1.77 BS03 60P A 1 D178 L193 F195 H221 L277 H282 D179 L194 F196 H222 L278 H283 3.1.2.32 0016787,0044550,0046872 Kd=19.6uM remove_due_to_license_issue P20581 27082157 403 HMLRLSAPGQLDDDLCLLGDVQVPVFLLRLGEASWALVEGGISRDAELVWADLCRWVADPSQVHYWLITHKHYDHCGLLPYLCPRLPNVQVLASERTCQAWKSESAVRVVERLNRQLLRAEQRLPEACAWDALPVRAVADGEWLELGPRHRLQVIEAHGHSDDHVVFYDVRRRRLFCGDALGEFDEAEGVWRPLVFDDMEAYLESLERLQRLPTLLQLIPGHGGLLRGRLAADGAESAYTECLRLCRRLLWRQSMGESLDELSEELHRAWGGQSVDFLPGELHLGSMRRMLEILSRQA 5hj9 A 1.28 BS03 X7A A 1 H114 D137 H139 D141 S150 H154 G155 D194 D243 E288 H102 D125 H127 D129 S138 H142 G143 D182 D231 E276 H114 D137 H139 D141 H154 D243 D245 E288 H102 D125 H127 D129 H142 D231 D233 E276 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 remove_due_to_license_issue Q6TUJ5 27050264 403 KKMSIVLAPFSGGQPHSGVELGPDYLLKQGLQQDMEKLGWDTRLERVFDGKVVEARKASDNGDRIGRVKRPRLTAECTEKIYKCVRRVAEQGRFPLTIGGDHSIALGTVAGVLSVHPDAGVIWVDAHADINTMSGTVSGNLHGCPLSILLGLDRENIPECFSWVPQVLKPNKIAYIGLRAVDDEEKKILHDLNIAAFSMHHVDRYGIDKVVSMAIEAVSPKGTEPVMVSYDVDTIDPLYVPATGTPVRGGLSFREALFLCERIAECGRLVALDVVECNPLLAATESHVNDTISVGCAIARCMMGETLLYTP 5hja A 1.65 BS03 XA2 A 1 H114 D137 H139 D141 S150 H154 G155 A192 V193 D194 D243 D245 H102 D125 H127 D129 S138 H142 G143 A180 V181 D182 D231 D233 H114 D137 H139 D141 H154 D243 D245 E288 H102 D125 H127 D129 H142 D231 D233 E276 3.5.3.1 0000050,0004053,0005634,0005737,0005829,0006525,0016787,0016813,0019547,0030145,0046872 remove_due_to_license_issue Q6TUJ5 27050264 403 KKMSIVLAPFSGGQPHSGVELGPDYLLKQGLQQDMEKLGWDTRLERVFDGKVVEARKASDNGDRIGRVKRPRLTAECTEKIYKCVRRVAEQGRFPLTIGGDHSIALGTVAGVLSVHPDAGVIWVDAHADINTMSGTVSGNLHGCPLSILLGLDRENIPECFSWVPQVLKPNKIAYIGLRAVDDEEKKILHDLNIAAFSMHHVDRYGIDKVVSMAIEAVSPKGTEPVMVSYDVDTIDPLYVPATGTPVRGGLSFREALFLCERIAECGRLVALDVVECNPLLNDTISVGCAIARCMMGETLLYT 5hjq A 2.3 BS01 I3P A 1 K75 R79 K277 R281 R335 G336 T339 K21 R25 K217 R221 R275 G276 T279 ? Kd=19uM remove_due_to_license_issue Q9VIH7 27669036 401 ALRSYTEIQQLLQQGKKRDVKNILRENSWPINSPIRAQLWPMLCGQHLDGFYWEMVHQVFGTTELSEKPIMLPAFVDATHCLPYHLTSTGRAVADRIVNVLGYDCPDITYSPVLYPITSILLHFMSEEEAYICLAGLVGSKEKVFINQTKLQHEVTWKTVMQIAKKHTKSATSYFQRICPGLKLERIFMDWCWWILAGLPFQHLVRIMDCYFHEGIKVLYRVALVILNLFHKECQSNNEWSPDNIKNDIGNALIKFCKKIPVSPAKLLHAAFSIRGLSTQYISR 5hk1 A 2.5051 BS01 61W A 1 L105 F107 Y120 H154 E172 L182 Y206 L98 F100 Y113 H147 E165 L175 Y199 ? 0004985,0005515,0005634,0005635,0005637,0005640,0005783,0005789,0005811,0005829,0005886,0006869,0007399,0014069,0016020,0030426,0031410,0038003,0038023,0042995,0043523,0045202,0045211,0070161,0070207,0098794,0098839,0098978,0150052 remove_due_to_license_issue Ki=2.0nM Q99720 27042935 301 RWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRYWAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLF 5hk2 A 3.2 BS01 61V A 1 M93 L105 F107 S117 Y120 D126 H154 E172 Y206 M92 L104 F106 S116 Y119 D125 H153 E171 Y205 ? 0004985,0005515,0005634,0005635,0005637,0005640,0005783,0005789,0005811,0005829,0005886,0006869,0007399,0014069,0016020,0030426,0031410,0038003,0038023,0042995,0043523,0045202,0045211,0070161,0070207,0098794,0098839,0098978,0150052 remove_due_to_license_issue Ki=1.7nM Q99720 27042935 301 QWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRYWAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYL 5hk9 A 1.8 BS01 64O A 1 D129 F164 P165 L174 V175 H177 Y239 G270 G271 M272 D105 F140 P141 L150 V151 H153 Y215 G246 G247 M248 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? 0016787 ic50=0.29uM remove_due_to_license_issue A0A0H2ZD27 27120257 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSRGRH 5hk9 B 1.8 BS01 64O B 1 D129 F164 L174 V175 H177 H207 Y239 G270 M272 F275 H297 D105 F140 L150 V151 H153 H183 Y215 G246 M248 F251 H273 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? 0016787 ic50=0.29uM remove_due_to_license_issue A0A0H2ZD27 27120257 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSRGRHH 5hka A 2.05 BS01 64N A 1 D129 F164 L174 V175 H177 F178 Y239 G270 G271 M272 F275 H297 D105 F140 L150 V151 H153 F154 Y215 G246 G247 M248 F251 H273 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? 0016787 ic50=0.35uM remove_due_to_license_issue A0A0H2ZD27 27120257 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSRGRHH 5hka B 2.05 BS01 64N B 1 D129 F164 L174 V175 H177 H207 Y239 G270 G271 M272 F275 H297 D105 F140 L150 V151 H153 H183 Y215 G246 G247 M248 F251 H273 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? 0016787 ic50=0.35uM remove_due_to_license_issue A0A0H2ZD27 27120257 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSR 5hkb A 1.65 BS01 64L A 1 R163 F164 P165 L174 V175 G270 G271 M272 F275 R139 F140 P141 L150 V151 G246 G247 M248 F251 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? 0016787 ic50=2.6uM remove_due_to_license_issue IC50=2700nM A0A0H2ZD27 27120257 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSRGRHH 5hkb B 1.65 BS01 64L B 1 F164 L174 V175 G270 M272 F275 H297 F140 L150 V151 G246 M248 F251 H273 F63 T66 D129 I130 H177 Y239 H269 H297 F39 T42 D105 I106 H153 Y215 H245 H273 ? 0016787 ic50=2.6uM remove_due_to_license_issue IC50=2700nM A0A0H2ZD27 27120257 401 AEEFPVPNGFESAYREVDGVKLHYVKGGQGPLVMLVHGFGQTWYEWHQLMPELAKRFTVIAPDLPGLGQSEPPKTGYSGEQVAVYLHKLARQFSPDRPFDLVAHDIGIWNTYPMVVKNQADIARLVYMEAPIPDARIYRFPAFTAQGESLVWHFSFFAADDRLAETLIAGKERFFLEHFIKSHASNTEVFSERLLDLYARSYAKPHSLNASFEYYRALNESVRQNAELAKTRLQMPTMTLAGGGHGGMGTFQLEQMKAYAEDVEGHVLPGCGHWLPEECAAPMNRLVIDFLSRGRHH 5hkm A 2.1 BS01 61Y A 1 V96 A109 S160 A162 G165 L212 T222 V21 A34 S85 A87 G90 L137 T147 D205 K207 E209 N210 D223 T245 D130 K132 E134 N135 D148 T160 2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.013uM remove_due_to_license_issue IC50=13nM O15530 27217002 403 KKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 5hl9 A 2.7 BS01 AIX A 1 S510 D553 S572 T699 G700 T701 Y734 S408 D451 S470 T597 G598 T599 Y632 2.4.99.28,3.4.16.4 0008233,0008658,0008955,0009252,0009274,0046677 remove_due_to_license_issue P02919 27899450 901 LLLKLAIVFAVLIAIYGVYLDQKIRSRIDGKVWQLPAAVYGRMVNLEPDMTISKNEMVKLLEATQYRQVSKMTRPGEFTVQANSIEMIRRPFDFPDSKEGQVRARLTFDGDHLATIVNMENNRQFGFFRLDPRLITMISNGEQRLFVPRSGFPDLLVDTLLATEDRHFYTLTQQLVKNLFLSSERSYWRKANEAYMALIMDARYSKDRILELYMNEVYLGQSGDNEIRGFPLASLYYFGRPVEELSLDQQALLVGMVKGASIYNPWRNPKLALERRNLVLRLLQQQQIIDQELYDMLSARPLGVQPRGISPQPAFMQLVRQELQAKLVKDLSGVKIFTTFDSVAQDAAEKAAVEGIPALKKQRKLSDLETAIVVVDRFSGEVRAMVGGSEPQFAGYNRAMQARRSIGSLAKPATYLTALSQPKIYRLNTWIADAPIALRQPNGQVWSPQNDDRRYSESGRVMLVDALTRSMNVPTVNLGMALGLPAVTETWIKLGVPKDQLHPVPAMLLGALNLTPIEVAQAFQTIASGGNRAPLSALRSVIAEDGKVLYQSFPQAERAVPAQAAYLTLWTMQQVVQRGTGRQLGAKYPNLHLAGKTGTTNNNVDTWFAGIDGSTVTITWVGRDNNQPTKLYGASGAMSIYQRYLANQTPTPLNLVPPEDIADMGVDYDGNFVCSGGMRILPVWTSDPQSLCQQS 5hlb A 2.42 BS02 AZR A 1 S507 S510 L611 T682 T699 G700 T701 T702 N703 S441 S444 L545 T616 T633 G634 T635 T636 N637 2.4.99.28,3.4.16.4 0008233,0008658,0008955,0009252,0009274,0046677 remove_due_to_license_issue P02919 27899450 902 WLLLKLAIVFAVLIAIYGVYLDQKIRSRIDGKVWQLPAAVYGRMVNLEPDMTISKNEMVKLLEATQYRQVSKMTRPGEFTVQANSIEMIRRPFDFPDSKEGQVRARLTFDGDHLATIVNMENNRQFGFFRLDPRLITMISSPNGEQRLFVPRSGFPDLLVDTLLATEDRHFYEHDGISLYSIGRAVLANLTAGRTVQGASTLTQQLVKNLFLSSERSYWRKANEAYMALIMDARYSKDRILELYMNEVYLGQSGDNEIRGFPLASLYYFGRPVEELSLDQQALLVGMVKGASIYNPWRNPKLALERRNLVLRLLQQQQIIDQELYDMLSARPLGVQPRGGVISPQPAFMQLVRQELQAKLGDKVKDLSGVKIFTTFDSVAQDAAEKAAVEGIPALKKQRKLSDLETAIVVVDRFSGEVRAMVGGSEPQFAGYNRAMQARRSIGSLAKPATYLTALSQPKIYRLNTWIADAPIALRQPNGQVWSPQNDDRRYSESGRVMLVDALTRSMNVPTVNLGMALGLPAVTETWIKLGVPKDQLHPVPAMLLGALNLTPIEVAQAFQTIASGGNRAPLSALRSVIAEDGKVLYQSFPQAERAVPAQAAYLTLWTMQQVVQRGTGRQLGAKYPNLHLAGKTGTTNNNVDTWFAGIDGSTVTITWVGRDNNQPTKLYGASGAMSIYQRYLANQTPTPLNLVPPEDIADMGVDYDGNFVCSGGMRILPVWTSDPQSLCQQSEM 5hld A 2.31 BS01 63V A 1 S510 D553 N574 T699 T701 T702 N703 S361 D404 N425 T550 T552 T553 N554 2.4.99.28,3.4.16.4 0008233,0008658,0008955,0009252,0009274,0046677 remove_due_to_license_issue P02919 27899450 901 AIVFAVLIAIYGVYLDQKIRSRIDGKVWQLPAAVYGRMVNLEPDMTISKNEMVKLLEATQYRQVSKMTRPGEFTVQANSIEMIRRPFDFPDSKEGQVRARLTFDGDHLATIVNMENNRQFGFFRLDPRLITMISSPNGEQRLFVPRSGFPDLLVDTLLATETQQLVKNLFLSKANEAYMALIMDARYSKDRILELYMNEVYLGQSGDNEIRGFPLASLYYFGRPVEELSLDQQALLVGMVLALERRNLVLRLLYDMLSARPQPAFMQLVRQELQAKLGDKVKDLSGVKIFTTFDSVAQDAAEKAAVEGIPALKKQRKLSDLETAIVVVDRFSGEVRAMVGGSEPQFAGYNRAMQARRSIGSLAKPATYLTALSQPKIYRLNTWIADAPIALRQPNGQVWSPQNDDRRYSESGRVMLVDALTRSMNVPTVNLGMALGLPAVTETWIKLGVPKDQLHPVPAMLLGALNLTPIEVAQAFQTIASGGNRAPLSALRSVIAEDGKVLYQSFPQAERAVPAQAAYLTLWTMQQVVQRGTGRQLGAKYPNLHLAGKTGTTNNNVDTWFAGIDGSTVTITWVGRDNNQPTKLYGASGAMSIYQRYLANQTPTPLNLVPPEDIADMGVDYDGNFVCSGGMRILPVWTSDPQSLCQQSE 5hlg A 3.0 BS01 dna I 0 Y17 R21 L55 N56 S66 N67 T70 R92 Q93 Y15 R19 L53 N54 S64 N65 T68 R90 Q91 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 QEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLETKYVFEELEQTLKHLIEK 5hlg A 3.0 BS02 dna J 0 T37 S39 N67 T68 M72 R75 K91 T35 S37 N65 T66 M70 R73 K89 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 QEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLETKYVFEELEQTLKHLIEK 5hlg B 3.0 BS01 dna I 0 T37 S39 Q40 N67 T68 M72 R75 K91 R92 T37 S39 Q40 N67 T68 M72 R75 K91 R92 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 MKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLPQEFTEYDETKYVFEELEQTLKHLIE 5hlg B 3.0 BS02 dna J 0 Y17 R21 N56 S66 N67 T70 R86 R92 Y17 R21 N56 S66 N67 T70 R86 R92 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 MKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLPQEFTEYDETKYVFEELEQTLKHLIE 5hlg C 3.0 BS01 dna K 0 Y17 L55 N56 S66 N67 T70 R92 L94 Y14 L52 N53 S63 N64 T67 R89 L91 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 EQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLYDETKYVFEELEQTLKHLIE 5hlg C 3.0 BS02 dna L 0 T37 S39 Q40 N67 T68 M72 R75 D90 K91 R92 T34 S36 Q37 N64 T65 M69 R72 D87 K88 R89 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 EQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLYDETKYVFEELEQTLKHLIE 5hlg D 3.0 BS01 dna K 0 T37 S39 N67 T68 M72 R75 D90 K91 R92 T39 S41 N69 T70 M74 R77 D92 K93 R94 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 CNMKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLPQDETKYVFEELEQTLKHLI 5hlg D 3.0 BS02 dna L 0 Y17 R21 L55 N56 S66 N67 T70 R92 Q93 L94 Y19 R23 L57 N58 S68 N69 T72 R94 Q95 L96 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 CNMKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLPQDETKYVFEELEQTLKHLI 5hlg E 3.0 BS01 dna M 0 Y17 R21 L55 N56 S66 N67 T70 K74 R86 R92 L94 Y18 R22 L56 N57 S67 N68 T71 K75 R87 R93 L95 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 NMKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLDETKYVFEELEQTLKHLIE 5hlg E 3.0 BS02 dna N 0 T37 S39 Q40 N67 T68 M72 R75 D90 K91 R92 T38 S40 Q41 N68 T69 M73 R76 D91 K92 R93 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 NMKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLDETKYVFEELEQTLKHLIE 5hlg F 3.0 BS01 dna M 0 T37 S39 Q40 N67 T68 M72 R75 D90 R92 T38 S40 Q41 N68 T69 M73 R76 D91 R93 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 NMKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLYDETKYVFEELEQTLKHLIE 5hlg F 3.0 BS02 dna N 0 Y17 R21 L55 N56 S66 N67 T70 R86 R92 Q93 L94 Y18 R22 L56 N57 S67 N68 T71 R87 R93 Q94 L95 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 NMKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLYDETKYVFEELEQTLKHLIE 5hlg G 3.0 BS01 dna O 0 Y17 L55 N56 S66 N67 T70 R92 L94 Y15 L53 N54 S64 N65 T68 R90 L92 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 QEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLEYDETKYVFEELEQTLKHLIE 5hlg G 3.0 BS02 dna P 0 T37 S39 Q40 N67 T68 M72 R75 D90 K91 R92 T35 S37 Q38 N65 T66 M70 R73 D88 K89 R90 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 QEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLEYDETKYVFEELEQTLKHLIE 5hlg H 3.0 BS01 dna O 0 T37 S39 Q40 N67 T68 M72 R75 K91 R92 T37 S39 Q40 N67 T68 M72 R75 K91 R92 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 MKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLPYDETKYVFEELEQTLKHLIE 5hlg H 3.0 BS02 dna P 0 Y17 R21 L55 N56 S66 N67 T70 K74 R92 L94 Y17 R21 L55 N56 S66 N67 T70 K74 R92 L94 ? 0003677,0003700,0005737,0006355,0006950 remove_due_to_license_issue Q5HKZ1 28086264 1 ~ 24 MKQEQMRLANQLCFSAYNVSRLFAQFYEKKLKQFGITYSQYLVLLTLWEENPQTLNSIGRHLDLSSNTLTPMLKRLEQSGWVKRERQQSDKRQLIITLTDNGQQQQEAVFEAISSCLPYDETKYVFEELEQTLKHLIE 5hlm A 2.5 BS01 B9F A 1 S16 Y33 W70 S75 T77 W97 R114 S14 Y31 W61 S66 T68 W88 R105 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 201 KCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYITAVTNEIKESPLHGTQNTTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 5hlm C 2.5 BS01 B9F A 1 W110 K111 W105 K106 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 201 RKCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYITAVNEIKESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 5hlm C 2.5 BS02 B9F C 1 L14 S16 Y33 T35 W70 S73 S75 T77 W97 R114 L13 S15 Y32 T34 W65 S68 S70 T72 W92 R109 ? 0005576,0009374,0019731 remove_due_to_license_issue P02701 301 RKCSLTGKWTNDLGSNMTIGAVNSRGEFTGTYITAVNEIKESPLHGTQNTINKRTQPTFGFTVNWKFSESTTVFTGQCFIDRNGKEVLKTMWLLRSSVNDIGDDWKATRVGINIFTRL 5hln A 3.1 BS01 65C A 1 I62 G63 N64 F67 V70 A83 Y134 V135 P136 T138 Q185 L188 C199 I29 G30 N31 F34 V37 A50 Y97 V98 P99 T101 Q148 L151 C162 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue IC50=30nM, EC50=1500nM P49841 27128528 501 GSKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 5hlp A 2.45 BS01 65A A 1 A83 D133 Y134 V135 L188 C199 A48 D93 Y94 V95 L148 C159 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=0.054uM remove_due_to_license_issue P49841 27128528 501 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 5hls A 2.182 BS01 62G A 1 W81 P82 F83 L92 L94 Y139 N140 I146 M149 W40 P41 F42 L51 L53 Y98 N99 I105 M108 ? ic50=0.039uM remove_due_to_license_issue IC50=39nM O60885 26815195 201 STNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5hlw A 1.97 BS01 62E A 1 I1084 A1108 Y1159 M1160 K1161 G1163 M1211 D1222 H1230 I27 A48 Y93 M94 K95 G97 M145 D156 H164 D1204 A1206 R1208 N1209 D1222 A1243 D138 A140 R142 N143 D156 A172 2.7.10.1 0004672,0004713,0005524,0006468 ic50=23nM remove_due_to_license_issue IC50=29nM P08581 27355974 1402 ALNPELVQAVQHVVIGSSLIVHFNEVIGRHFGCVYHGTLLDGKKIHCAVKSLNRIDIGEVSQFLTEGIIMKDFSHPNVLSLLGICSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMHDKEYYSVAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNAT 5hm0 A 1.395 BS01 62V A 1 W81 P82 L92 I146 W40 P41 L51 I105 ? ic50=0.44uM remove_due_to_license_issue O60885 26815195 201 STNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5hm3 A 2.25 BS01 649 A 1 L222 D239 M240 L247 A248 F285 L318 S321 E322 P323 S349 Y350 G351 L352 A353 L357 D476 K608 L211 D228 M229 L236 A237 F274 L307 S310 E311 P312 S338 Y339 G340 L341 A342 L346 D465 K597 6.2.1.20 0005524,0005886,0006631,0006633,0008610,0008922,0009274,0016874,0070566,0071766,0071769 ic50=6.8uM remove_due_to_license_issue O53580 27547819 701 FVTGNPFIVNGKIRFTNLVRHVEKWAKVRGDKLAYRFLDFSTERDGVARDILWSDFSARNRAVGARLQQVTQPGDRVAILCPQNLDYLISFFGALYSGRIAVPLFDPAEPGHVGRLHAVLDDCAPSTILTTTDSAEGVRKFIRARSAKERPRVIAVDAVPTEVAATWQQPEANEETVAYLQYTSGSTRIPSGVQITHLNLPTNVVQVLNALEGQEGDRGVSWLPFFHDMGLITVLLASVLGHSFTFMTPAAFVRRPGRWIRELARKPGETGGTFSAAPNFAFEHAAVRGVPRDDEPPLDLSNVKGILNGSEPVSPASMRKFFEAFAPYGLKQTAVKPSYGLAEATLFVSTTPMDEVPTVIHVDRDELNNQRFVEVAADAPNAVAQVSAGKVGVSEWAVIVDADTASELPDGQIGEIWLHGNNLGTGYWGKEEESAQTFKNILKSRISESRAEGAPDDALWVRTGDYGTYFKDHLYIAGRIKDLVIIDGRNHYPQDLECTAQESTKALRVGYAAAFSVPANQLPQTVFDDSHAGLKFDPEDTSEQLVIVGERAAGTHKLDHQPIVDDIRAAIAVGHGVTVRDVLLVSAGTIPRTSSGKIGRRACRAAYLDGSLRSGVGSPTVFATS 5hmh A 1.79 BS01 62R A 1 Q24 L54 G58 I61 M62 Y67 Q72 F91 V93 H96 I99 Y100 Q6 L36 G40 I43 M44 Y49 Q54 F73 V75 H78 I81 Y82 2.3.2.27 0005634,0043066,0051726 ic50=0.007uM remove_due_to_license_issue Q00987 26985323 201 ASASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLYYLGQYIMTKRLYDEKQQHIVHCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVNQQ 5hmi A 1.74 BS01 62T A 1 Q24 L54 G58 I61 M62 Y67 Q72 F91 V93 H96 I99 Y100 Q7 L37 G41 I44 M45 Y50 Q55 F74 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 ic50=0.015uM remove_due_to_license_issue Q00987 26985323 1001 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLYYLGQYIMTKRLYDEKQQHIVHCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVNQQ 5hmk A 2.17 BS01 62Q A 1 L54 L57 G58 I61 M62 Y67 Q72 F91 V93 H96 I99 Y100 L29 L32 G33 I36 M37 Y42 Q47 F66 V68 H71 I74 Y75 2.3.2.27 0005634,0043066,0051726 ic50=0.04uM remove_due_to_license_issue Q00987 26985323 1001 TLVRPKPLLLKLLKSVGAQKDTYTMKEVLYYLGQYIMTKRLYDEKQQHIVHCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5hmk A 2.17 BS02 62Q B 1 K51 Y55 K26 Y30 2.3.2.27 0005634,0043066,0051726 ic50=0.04uM remove_due_to_license_issue Q00987 26985323 1001 TLVRPKPLLLKLLKSVGAQKDTYTMKEVLYYLGQYIMTKRLYDEKQQHIVHCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5hmy A 2.1 BS03 LNY A 1 L511 C709 R729 M761 M765 T794 S796 H798 A799 H800 Q802 W803 L213 C411 R431 M463 M467 T496 S498 H500 A501 H502 Q504 W505 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 ic50=0.5uM remove_due_to_license_issue Q6YMS4 26984786 1003 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAADSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYMPSMKRF 5hn0 A 2.05 BS03 LNN A 1 L511 C709 R729 M761 Y766 T794 S796 H798 A799 L213 C411 R431 M463 Y468 T496 S498 H500 A501 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0005524,0039694 remove_due_to_license_issue Q6YMS4 26984786 1003 NMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNAADSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGAGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 5hn7 A 2.15 BS01 04M A 1 G80 K81 R84 Q119 F122 M129 R135 R136 Q195 T199 K243 Y247 F283 G45 K46 R49 Q80 F83 M90 R96 R97 Q156 T160 K198 Y202 F236 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K46 A82 D87 D91 R96 D159 K198 F236 D240 D241 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 ic50=120uM remove_due_to_license_issue A5K4U6 27564465 401 FFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSIDVNNINVPQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTG 5hn7 A 2.15 BS02 04M E 1 N154 L157 N115 L118 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K46 A82 D87 D91 R96 D159 K198 F236 D240 D241 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 ic50=120uM remove_due_to_license_issue A5K4U6 27564465 401 FFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSIDVNNINVPQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTG 5hn7 E 2.15 BS01 04M E 1 G80 K81 R84 Q119 F122 D126 R136 T191 I192 Q195 T244 Y247 F283 G47 K48 R51 Q86 F89 D93 R103 T158 I159 Q162 T209 Y212 F246 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A88 D93 D97 R102 D165 K208 F246 D250 D251 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 ic50=120uM remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSDAHREIDVNNINPEPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTGV 5hn8 A 2.7 BS01 HXK A 1 G80 K81 R84 Q119 F122 L123 R136 Q195 T244 Y247 G47 K48 R51 Q81 F84 L85 R98 Q157 T202 Y205 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A83 D88 D92 R97 D160 K201 F239 D243 D244 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSDIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDSDIQNNKLTWPLIKTFELCPDKIIVKNYGKVIDSLYEQYKHYESYEKAQKAKILSAIELHHEGIEYVLKYLLEI 5hn8 C 2.7 BS01 HXK C 1 G80 K81 R84 F122 R136 Q195 K243 D287 G41 K42 R45 F79 R93 Q152 K198 D240 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K42 A78 D83 D87 R92 D155 K198 F236 D240 D241 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 27564465 401 FRNMYDKYRDAFLSHLNEEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYDAREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEIL 5hn9 A 2.12 BS01 04W A 1 G80 K81 R84 Q119 F122 L123 A125 M129 R135 R136 Q195 K301 G45 K46 R49 Q83 F86 L87 A89 M93 R99 R100 Q159 K258 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K46 A85 D90 D94 R99 D162 K203 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 ic50=50uM remove_due_to_license_issue A5K4U6 27564465 401 FFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKRDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTG 5hn9 A 2.12 BS02 04W B 1 N154 L157 N118 L121 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K46 A85 D90 D94 R99 D162 K203 F241 D245 D246 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 ic50=50uM remove_due_to_license_issue A5K4U6 27564465 401 FFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKRDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSEIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTG 5hn9 B 2.12 BS01 04W B 1 K81 R84 Q119 F122 L123 M129 R135 R136 Q195 Y247 F283 K301 K48 R51 Q86 F89 L90 M96 R102 R103 Q162 Y213 F245 K263 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A88 D93 D97 R102 D165 K209 F245 D249 D250 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 ic50=50uM remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKNRDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSDAREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGNLIYKKIEDISMLMGEYFQIHDDYLDIFGDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFTG 5hna A 2.693 BS01 63D A 1 K81 R84 Q119 F122 L123 M129 R135 R136 Y160 Q195 K243 F283 K48 R51 Q84 F87 L88 M94 R100 R101 Y125 Q160 K205 F243 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A86 D91 D95 R100 D163 K205 F243 D247 D248 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFT 5hna A 2.693 BS02 63D B 1 N154 L157 N119 L122 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A86 D91 D95 R100 D163 K205 F243 D247 D248 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFT 5hna B 2.693 BS01 63D A 1 N154 L157 N119 L122 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A86 D91 D95 R100 D163 K205 F243 D247 D248 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFT 5hna B 2.693 BS02 63D B 1 K81 R84 Q119 F122 L123 M129 R135 R136 Q195 K243 Q284 K48 R51 Q84 F87 L88 M94 R100 R101 Q160 K205 Q244 K81 A121 D126 D130 R135 D198 K243 F283 D287 D288 K48 A86 D91 D95 R100 D163 K205 F243 D247 D248 ? 0004161,0004337,0004659,0005737,0008299,0016020,0016740,0016765,0045337,0046872 remove_due_to_license_issue A5K4U6 27564465 401 LAFFRNMYDKYRDAFLSHLNEYSLEEEIKEHISKYYKLLFDYNCLGGKNNRGILVILIYEYVKDINSSEWEKAACLAWCIEILQAAFLVADDIMDKGEMRRNKYCWYLLKDVETKNAVNDVLLLYNSIYKLIEIYLRNESCYVDVIATFRDATLKTIIGQHLDTNIFSDKYSREIDVNNINVPEQPVIDINMINFGVYKNIVIHKTAYYSFFLPIVCGMLLAGIDNLIYKKIEDISMLMGEYFQIHDDYLDIFDSTKTGKVSDIQNNKLTWPLIKTFELCSEPDKIKIVKNYGKNNLACVKVIDSLYEQYKIRKHYESYEKAQKAKILSAINELHHEGIEYVLKYLLEILFT 5hng A 3.01 BS01 62O A 1 A109 S160 Y161 A162 G165 L212 A39 S90 Y91 A92 G95 L142 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T167 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue O15530 27217002 403 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 5ho4 A 1.85 BS01 rna B 0 Q19 K22 F24 G26 G27 D49 V51 M53 R62 G63 F64 F66 E92 A96 V97 R99 Q5 K8 F10 G12 G13 D35 V37 M39 R48 G49 F50 F52 E78 A82 V83 R85 ? 0003676,0003723 remove_due_to_license_issue P22626 29379020 1 ~ 10 REKEQFRKLFIGGLSFETTEESLRNYYEQWGKLTDCVVMRDPASKRSRGFGFVTFSSMAEVDAAMAARPHSIDGRVVEPKRAVAREESGKPGAHVTVKKLFVGGIKEDTEEHHLRDYFEEYGKIDTIEIITDRQSGKKRGFGFVTFDDHDPVDKIVLQKYHTINGHNAEVRKALSRQEM 5ho6 A 1.97 BS01 63K A 1 A1108 L1157 Y1159 M1160 K1161 H1162 G1163 D1164 M1211 D1222 A1226 A22 L58 Y60 M61 K62 H63 G64 D65 M112 D123 A127 D1204 A1206 R1208 N1209 D1222 D105 A107 R109 N110 D123 2.7.10.1 0004672,0004713,0005524,0006468 ic50=204nM remove_due_to_license_issue IC50=204nM, Kd=0.900000nM P08581 27355974 1401 VQAVQHVVIGPCVYHGTLIHCAVKSVSQFLTEGIIMKDFSHPNVLSLLGICGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATY 5ho7 A 3.0 BS01 63L A 1 L88 V143 L159 Y161 L212 T222 L18 V73 L89 Y91 L142 T152 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T167 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=17000nM O15530 27217002 701 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 5ho8 A 2.7 BS01 63E A 1 V96 A109 Y161 A162 E209 L212 T222 V26 A39 Y91 A92 E139 L142 T152 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T166 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=>10000nM O15530 27217002 701 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKL 5hoa A 2.14 BS01 63K A 1 Y1159 M1160 K1161 D1164 R1208 M1211 A1221 D1222 Y45 M46 K47 D50 R94 M97 A107 D108 D1204 A1206 R1208 N1209 D1222 D90 A92 R94 N95 D108 2.7.10.1 0004672,0004713,0005524,0006468 ic50=64nM remove_due_to_license_issue IC50=204nM, Kd=0.900000nM P08581 27355974 1401 AVQHVVVYHGTLKIHCAVKQFLTEGIIMKDFSHPNVLSLLGVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFVASKKFVHRDLAARNCMLDEKFTVKVADFGLARLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATY 5hor A 2.2 BS01 63K A 1 A1108 L1157 Y1159 M1160 K1161 G1163 D1164 R1208 M1211 A1221 D1222 A23 L63 Y65 M66 K67 G69 D70 R114 M117 A127 D128 D1204 A1206 R1208 N1209 D1222 D110 A112 R114 N115 D128 2.7.10.1 0004672,0004713,0005524,0006468 ic50=6nM remove_due_to_license_issue IC50=204nM, Kd=0.900000nM P08581 27355974 1401 QAVQHVVIGPGCVYHGTLKIHCAVKSVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMLPVKWTALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATY 5hrt A 1.997 BS01 dna B 0 R244 G245 R246 E247 H315 H452 A454 R455 P457 L458 S465 K467 F469 F470 D473 R188 G189 R190 E191 H259 H396 A398 R399 P401 L402 S409 K411 F413 F414 D417 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 remove_due_to_license_issue Q9R1E6 27043297 2001 ~ 2034 TNTSGSCKGRCFELQDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPLDVYKKPSGKCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCDSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYESEI 5hrv A 1.7 BS01 64C A 1 I683 F684 L687 Y696 M704 D705 M731 A735 I32 F33 L36 Y45 M53 D54 M80 A84 ? 0006338,0016586 remove_due_to_license_issue Q86U86 27617704 801 SKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDLEGD 5hrw A 1.8 BS01 64E A 1 I683 F684 L687 Y696 M704 A735 I745 I30 F31 L34 Y43 M51 A82 I92 ? 0006338,0016586 remove_due_to_license_issue Q86U86 27617704 801 YMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDL 5hrx A 1.73 BS01 64F A 1 I683 F684 L687 Y696 M704 A735 I30 F31 L34 Y43 M51 A82 ? 0006338,0016586 remove_due_to_license_issue Q86U86 27617704 803 YMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDL 5hsw A 3.3 BS01 rna B 0 F179 K246 C247 R248 F249 Y373 F145 K211 C212 R213 F214 Y329 ? 0003677,0004519,0004527,0005515,0030430,0042025,0046872 remove_due_to_license_issue P88925 28132029 3 ~ 28 TPADLFSEDAVLASLSFSKFLKHAKVRDWCAQAKIQPSMPALRMAYNYFLFSKVGEFIGSEDVCNFFVDRVFGGVRLLDVASVYAACSQMNAHQRHHICCLVERATSSQSLNPVWDALRDGIISSSKFHWAVKQQNKIFSPPLAFGLRCEEVVKTLLATLLHPDETNCLDYGFMQSPQNGIFGVSLDFAANVKTDTGRLQFDPNCKVYSIKCRFKYTFAKMECDPIYAAYQRLYEAPGKLALKDFFYSISKPAVEYVGLGKLPSESDYLVAYDQEWEACLHNLIRECILHNSTTESDVYVLTDPQDTRGQISIKARFKANLFVNVRHSYFYQVLLQSSIVEEYIGSPKYYIATGFFRKRGYQDPVNCTIGGDALDPHVEIPTLLIVTPVYFPRGAKHRLLHQAANFWSRSAKDTFPYIKWDFSYLSAN 5htb A 1.7 BS02 6L5 B 1 I490 E492 G493 F495 G496 V498 A509 I557 F607 G608 D611 G653 L656 T689 I20 E22 G23 F25 G26 V28 A39 I87 F137 G138 D141 G183 L186 T219 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q8TF76 27139824 101 GPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 5htc A 1.5 BS02 66M B 1 I490 E492 G493 F495 V498 A509 F607 G608 D611 G653 L656 I686 T689 I20 E22 G23 F25 V28 A39 F137 G138 D141 G183 L186 I216 T219 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q8TF76 27139824 101 GPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 5htl A 1.371 BS01 C2E A 1 R7 R9 L10 G11 D12 L29 Q32 R38 L39 G40 D41 L58 Q61 D108 R3 R5 L6 G7 D8 L25 Q28 R34 L35 G36 D37 L54 Q57 D104 ? Kd=0.5uM remove_due_to_license_issue Q9KUV7 27578558 201 KLRKRLGDLLVEEGIVSEAQLEQALNAQKNTGRRLGDTLISLGFLSETQLLNFLAQQLSLPVIDLSRAHVDIDAVPLLPEVHARRLRALVIGRSGDTLRIAMSDPADLFAQEALLNQLPDYGFEFVIAPEKQLVDGFDRYY 5htl A 1.371 BS02 C2E B 1 S63 P65 S59 P61 ? Kd=0.5uM remove_due_to_license_issue Q9KUV7 27578558 201 KLRKRLGDLLVEEGIVSEAQLEQALNAQKNTGRRLGDTLISLGFLSETQLLNFLAQQLSLPVIDLSRAHVDIDAVPLLPEVHARRLRALVIGRSGDTLRIAMSDPADLFAQEALLNQLPDYGFEFVIAPEKQLVDGFDRYY 5htl B 1.371 BS01 C2E B 1 R7 R9 L10 G11 D12 L29 Q32 R38 L39 G40 D41 L54 L58 Q61 A110 R1 R3 L4 G5 D6 L23 Q26 R32 L33 G34 D35 L48 L52 Q55 A104 ? Kd=0.5uM remove_due_to_license_issue Q9KUV7 27578558 201 RKRLGDLLVEEGIVSEAQLEQALNAQKNTGRRLGDTLISLGFLSETQLLNFLAQQLSLPVIDLSRAHVDIDAVPLLPEVHARRLRALVIGRSGDTLRIAMSDPADLFAQEALLNQLPDYGFEFVIAPEKQLVDGFDRYY 5htz A 1.95 BS01 66J A 1 S71 Q73 G74 L91 D93 Y132 Q134 F169 W176 D289 S290 G291 T292 S15 Q17 G18 L35 D37 Y76 Q78 F113 W120 D233 S234 G235 T236 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 Ki=2.4nM remove_due_to_license_issue Ki=2.387nM P56817 27933948 501 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hu0 A 1.83 BS01 66H A 1 Q73 G74 L91 D93 S96 Y132 W137 F169 I179 D289 G291 T292 Q16 G17 L34 D36 S39 Y75 W80 F112 I122 D232 G234 T235 D93 S96 N98 A100 Y132 D289 T292 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 Ki=595nM remove_due_to_license_issue P56817 27933948 502 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hu1 A 1.5 BS01 66F A 1 S71 Q73 G74 L91 D93 Y132 Q134 F169 I179 D289 G291 T292 T293 S15 Q17 G18 L35 D37 Y76 Q78 F113 I123 D233 G235 T236 T237 D93 S96 N98 A100 Y132 D289 T292 D37 S40 N42 A44 Y76 D233 T236 3.4.23.46 0004190,0006508,0016020 Ki=2.2nM remove_due_to_license_issue P56817 27933948 501 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5hu9 A 1.529 BS01 66K A 1 K271 E286 M290 I313 T315 F317 M318 G321 I360 H361 L370 A380 D381 F382 K47 E62 M66 I89 T91 F93 M94 G97 I136 H137 L146 A156 D157 F158 D363 A365 R367 N368 D381 P402 D139 A141 R143 N144 D157 P173 2.7.10.2 0004672,0004713,0005524,0006468 Kd=24.2nM remove_due_to_license_issue P00519 27322145 601 AMGSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQE 5hu9 A 1.529 BS02 66K A 2 L387 I403 A412 Y449 L163 I174 A183 Y220 D363 A365 R367 N368 D381 P402 D139 A141 R143 N144 D157 P173 2.7.10.2 0004672,0004713,0005524,0006468 Kd=24.2nM remove_due_to_license_issue P00519 27322145 602 AMGSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQE 5hv0 A 1.63 BS03 AKG A 1 Y118 H127 T159 H193 K203 I205 T207 W209 Y108 H117 T149 H183 K193 I195 T197 W199 ? 0003674,0004656,0005506,0008150,0016705,0031418,0046872,0051213 Kd=1.1uM remove_due_to_license_issue A0A4Y1WAP5 27139630 310 NQIKEQTIFDHKGNVIKTEDREIQIISKFEEPLIVVLGNVLSDEECDELIELSKSKLARSKVGSSNDIRTSSGAFLDDNELTAKIEKRISSIMNVPASHGEGLHILNYEVDQQYKAHYDYFAEHSRSAANNRISTLVMYLNDVEEGGETFFPKLNLSVHPRKGMAVYFEYFYQDQSLNELTLHGGAPVTKGEKWIATQWVRRGTYK 5hv1 A 3.103 BS02 RFP A 1 Y351 T355 P356 V368 F479 I487 Y351 T355 P356 V368 F459 I467 0005524,0016301,0016310,0016772 remove_due_to_license_issue 27001859 902 MKPYVLKFQEIRPHSEALVGGKGMNLGACSNIEGVHVPAGFCLTTEAYKRTLAENNEFTQLLQRLSSLKTSDMDAIREISETIRTLIQHTQIPSEIASYMDATLLDVGGYEMPFAVRSSATAEDLPHASFAGQHDTYLNIIGKDALLQHISMCWASLFTERAIIYRIQNQFDHRKVQLAVVIQQMISPEASGILFTADPITSNRKSLSIDASFGLGEALVSGLVSADSYTVRENTITNKIIATKKLAIYSLKEGGTETRILEKSQQTKQTLTDQQIIQLAKLGRKIEAYFGKPQDIEWCLAEGAFYIVQSRPITTLYPIPEVNEPGNRVYISVAHQQMMTDAMKPLGLSFYLMTTPATMYTAGGRLFVDITQSLSAKVSRDMMVNSLGQSDPLIKDALLTVINKKGFLPSIPDSSSVFELVRNSENSIKHLKQSIETKSGSDLFDFIVEDLEELKRVLFNPTSIDAIMAGMDASAWLNEHIYQWLGEKNVADKLSESAPNNITSQMGLELLDVADVIRPYPAVRAYLEQTKNPDFMNELATLEGGAETKKALEDYLQKYGMRCAGEIDLTKTRWIENPLTLIPLILSNIKNFDSSASMHKFAQGEKEAFHKEQEILRRLQELPDGEQKAMETKEKIDILRHFIGYREYPKYGMINRYFIYKLALLRAGEQLVKDGILQEHEDIYFLYFEELREVVRTGQVDYELINARKRDFATFEKLTPPRILTSDGEMINGEYKRENLPKDAILGLPVSSGTVEGRARVILEMEKADLEDGDILVTAYTDPSWTPAFVSIKGLVTEVGGLMTHGAVIAREYGLPAVVGVENATTIIKDGQQIRINGTEGYIEILD 5hva A 2.1 BS02 DUP C 1 N109 K112 K122 Q123 N105 K108 K118 Q119 ? 0046872,0047429 remove_due_to_license_issue Q9RS96 27739259 201 PCPPTNAERLHEFHRAIGAATPERPTPPPPELLRLRQTLLDEESAEVRAEIDHLLARQAAGEALSAGDLAPLAHELADLLYVTYGALDQLGIDADAVFAEVHRANLSKASGPRRADGKQLKPEGWRPADVRGVIERLQHA 5hva C 2.1 BS01 DUP C 1 F17 E47 E50 D82 Y85 F13 E43 E46 D78 Y81 ? 0046872,0047429 Kd=0.086uM remove_due_to_license_issue Q9RS96 27739259 201 PCPPTNAERLHEFHRAIGAATPERPTPPPPELLRLRQTLLDEESAEVRAEIDHLLARQAAGEALSAGDLAPLAHELADLLYVTYGALDQLGIDADAVFAEVHRANLSKASGKPEGWRPADVRGVIERLQHA 5hvs A 1.75 BS01 65V A 1 P1 M2 K32 P33 Y36 H62 I64 M101 V106 F113 P1 M2 K32 P33 Y36 H62 I64 M101 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.071uM remove_due_to_license_issue Ki=23.0nM P14174 27299179 203 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvs A 1.75 BS02 65V B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.071uM remove_due_to_license_issue Ki=23.0nM P14174 27299179 203 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvs C 1.75 BS01 65V A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.071uM remove_due_to_license_issue Ki=23.0nM P14174 27299179 203 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvs C 1.75 BS02 65V C 1 P1 M2 K32 P33 Y36 H62 I64 M101 V106 F113 P1 M2 K32 P33 Y36 H62 I64 M101 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.071uM remove_due_to_license_issue Ki=23.0nM P14174 27299179 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvt A 1.75 BS01 NVS A 1 P1 M2 K32 Y36 H62 S63 I64 V106 F113 P1 M2 K32 Y36 H62 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.055uM remove_due_to_license_issue P14174 27299179 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvt A 1.75 BS02 NVS C 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.055uM remove_due_to_license_issue P14174 27299179 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvt B 1.75 BS01 NVS A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.055uM remove_due_to_license_issue P14174 27299179 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvt B 1.75 BS02 NVS B 1 P1 M2 K32 Y36 H62 S63 I64 V106 F113 P1 M2 K32 Y36 H62 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.055uM remove_due_to_license_issue P14174 27299179 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5hvu A 2.8 BS01 65R A 1 F87 G88 E89 V90 A103 K105 D117 F120 M156 A215 D216 F82 G83 E84 V85 A98 K100 D112 F115 M151 A210 D211 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=13nM, IC50=7.0nM Q13464 29945794 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEETFPIPKAFVGNQLPFVGFTYYSNRRY 5hvy A 2.39 BS01 66X A 1 A50 E66 L69 I79 Y99 A100 L148 L158 A172 D173 M174 A48 E64 L67 I77 Y97 A98 L140 L150 A164 D165 M166 D151 K153 N156 D173 T196 D143 K145 N148 D165 T176 2.7.11.22,2.7.11.23 0004672,0005524,0006468 ic50=17.4nM remove_due_to_license_issue IC50=>10000nM P49336 27326333 501 DKMDYDFKVKLSSERERVEDLFEYEGCKVGGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLPVVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRKTSNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 5hwu A 2.1 BS02 DUP B 1 N109 K112 K122 Q123 K125 N102 K105 K115 Q116 K118 ? 0046872,0047429 remove_due_to_license_issue Q9RS96 27739259 201 PPTNAERLHEFHRAIGATPERPTPPPPELLRLRQTLLDAESAEVRAEIDHLLARQAAGEALSAGDLAPLAHELADLLYVTYGALDQLGIDADAVFAEVHRANLSKASGPRRADGKQLKPEGWRPADVRGVIERLQHA 5hwu B 2.1 BS01 DUP B 1 E47 H78 D82 E41 H72 D76 ? 0046872,0047429 Kd=5.35uM remove_due_to_license_issue Q9RS96 27739259 201 PPTNAERLHEFHRAIGAATPERPTPPPPELLRLRQTLLDAESAEVRAEIDHLLARQAAGEALSAGDLAPLAHELADLLYVTYGALDQLGIDADAVFAEVHRANLSKASGPLKPEGWRPADVRGVIERLQHA 5hwv A 1.65 BS01 MBN A 1 F46 F79 F128 F5 F38 F87 2.7.13.3 Kd=8.5uM remove_due_to_license_issue A5W4E3 26903514 501 ALYEFVGLLDAHGNVLEVNQVALEGGGITMEEIRGKPFWKARWWQISKKTEATQKRLVETASSGEFVRCDVEILGKSGGREVIAVDFSLLPICNEEGSIVYLLAEGRNITDKKKAEAMLALKNQ 5hx6 A 2.23 BS01 65U A 1 V31 K45 V76 L78 L90 M92 H136 D156 L157 F162 V19 K33 V64 L66 L78 M80 H124 D144 L145 F150 D138 K140 E142 N143 D156 T189 D126 K128 E130 N131 D144 T159 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.6nM, Ki=0.800000nM Q13546 26854747 301 IKMKSSDFLESAELDSGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 5hx8 A 2.2 BS01 66P A 1 L881 V889 A906 M956 E957 F958 L959 G962 R1007 L1010 G1020 L27 V35 A52 M95 E96 F97 L98 G101 R146 L149 G159 D1003 A1005 R1007 N1008 D1021 D1040 D142 A144 R146 N147 D160 D179 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM P23458 26927423 1201 IVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 5hz5 A 1.4 BS01 65X A 1 F19 L32 M35 A39 T56 A78 I107 R109 V118 C120 Y131 F18 L31 M34 A38 T55 A77 I106 R108 V117 C119 Y130 ? 0001972,0005324,0005504,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005886,0006006,0006629,0006656,0006869,0008289,0008544,0010829,0014069,0015908,0015909,0030667,0031392,0035360,0035578,0042593,0042802,0045202,0051930,0070062,0098921,0098978,0099092,0099178,0099524,0120162,1990379 Ki=0.086uM remove_due_to_license_issue Ki=86nM Q01469 27658368 203 ATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTLKTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVECVMNNVTCTRIYEKVE 5hz6 A 1.14 BS01 65Y A 1 F17 A34 A37 P39 S54 S56 K59 D77 R127 F16 A33 A36 P38 S53 S55 K58 D76 R126 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.016uM remove_due_to_license_issue P15090 27658368 201 AGAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5hz8 A 1.12 BS01 65Z A 1 M21 A34 A37 S56 F58 A76 D77 R107 L116 L118 R127 M24 A37 A40 S59 F61 A79 D80 R110 L119 L121 R130 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.016uM remove_due_to_license_issue Ki=16nM P15090 27658368 200 GSHMCDAFVGTWKLVSSENFDDYMKELGVGFATRKVAGMAKPNTIISVNGDVITLKTESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTLKRKREDDKLVLELVMKGVTCTRVYERA 5hz9 A 2.3 BS01 5M8 A 1 T54 S56 F58 A76 D77 T56 S58 F60 A78 D79 ? 0005515,0005615,0005634,0005737,0005829,0008092,0008285,0008289,0015909,0032365,0036041,0042632,0046320,0050873,0055091,0070062,0070538,0071073,0140214,2001245 Ki=0.093uM remove_due_to_license_issue Ki=93nM P05413 27658368 204 SHMVDAFLGTWKLVDSKNFDDYMKSLGVGFATRQVASMTKPTTIIEKNGDILTLKTHSTFKNTEISFKLGVEFDETTADDRKVKSIVTLDGGKLVHLQKWDGQETTLVRELIDGKLILTLTHGTAVCTRTYEKEA 5hz9 A 2.3 BS02 5M8 A 3 K22 G27 F28 R31 K24 G29 F30 R33 ? 0005515,0005615,0005634,0005737,0005829,0008092,0008285,0008289,0015909,0032365,0036041,0042632,0046320,0050873,0055091,0070062,0070538,0071073,0140214,2001245 Ki=0.093uM remove_due_to_license_issue Ki=93nM P05413 27658368 206 SHMVDAFLGTWKLVDSKNFDDYMKSLGVGFATRQVASMTKPTTIIEKNGDILTLKTHSTFKNTEISFKLGVEFDETTADDRKVKSIVTLDGGKLVHLQKWDGQETTLVRELIDGKLILTLTHGTAVCTRTYEKEA 5hzn A 2.2 BS01 66A A 1 G1003 Q1004 G1005 F1007 A1028 K1030 E1047 V1060 M1076 M1079 M1139 G1149 D1150 G24 Q25 G26 F28 A49 K51 E68 V81 M97 M100 M152 G162 D163 D1132 R1136 N1137 D1150 E1159 D145 R149 N150 D163 E172 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.061uM remove_due_to_license_issue IC50=61nM P08069 26951750 1301 AADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVNEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSEENK 5hzx A 1.9 BS01 2GE A 1 F27 N33 F72 F74 M81 W117 D119 D120 F25 N31 F70 F72 M79 W115 D117 D118 3.6.1.-,3.6.1.56 0003723,0005634,0005737,0005739,0005759,0005829,0008413,0009151,0016787,0016791,0016818,0042262,0046872,0047429 ic50=2.8nM remove_due_to_license_issue Q7ZWC3 26862114 201 TSKLLTLVLVVQPGRVLLGMKKRGFGAGKWNGFGGKVQTGETIEQAARRELLEESGLTVDTLHKIGNIKFEFIGETELMDVHIFRADNYEGEPAESDEMRPQWFDIDKIPFSQMWADDILWFPLMLQKKRFLGYFKFQGHDVIVEHKLDEVEDL 5i0b A 3.09 BS01 67U A 1 I327 A348 L398 E399 G401 A402 L447 I27 A48 L98 E99 G101 A102 L147 D440 K442 D444 S445 D458 K467 T478 D140 K142 D144 S145 D158 K167 T178 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O96013 27117431 601 HEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 5i0l A 2.45 BS01 H27 A 1 I180 A182 H183 L214 T215 H218 E219 H222 H228 V235 F237 P238 Y240 I75 A77 H78 L109 T110 H113 E114 H117 H123 V130 F132 P133 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=18nM remove_due_to_license_issue P39900 27356908 301 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i0l A 2.45 BS07 H27 B 1 P232 K233 P127 K128 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50=18nM remove_due_to_license_issue P39900 27356908 301 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i12 A 1.59 BS06 H27 A 1 L187 A189 H226 E227 H230 H236 Y245 P246 M247 Y248 L75 A77 H114 E115 H118 H124 Y133 P134 M135 Y136 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 ic50=1200nM remove_due_to_license_issue P14780 27356908 306 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5i13 A 2.151 BS03 4P9 A 1 K34 A37 W188 F191 S194 E195 K39 A42 W173 F176 S179 E180 3.1.-.- 0003723,0039694 remove_due_to_license_issue IC50=8300nM P03433 27088785 304 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 5i13 A 2.151 BS04 4P9 A 2 H41 D108 E119 K134 H46 D93 E104 K119 3.1.-.- 0003723,0039694 remove_due_to_license_issue IC50=8300nM P03433 27088785 305 GPLGSMEDFVRQCFNPMIVELAEKTMKEYGEDLKIETNKFAAICTHLEVCFMYSDASKHRFEIIEGRDRTMAWTVVNSICNTTGAEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRGLWDSFRQSER 5i1q A 1.5 BS01 67C A 1 W1526 P1527 F1528 V1532 F1536 V1537 Y1582 N1583 Y1589 W26 P27 F28 V32 F36 V37 Y82 N83 Y89 2.3.1.48,2.7.11.1 0004402,0005669,0006366,0016251,0017025 Kd=12nM remove_due_to_license_issue IC50=9900nM P21675 27219867 1701 DDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESLD 5i23 A 1.95 BS01 66V A 1 F271 D299 Y376 W410 D412 R463 W477 D480 F513 H540 F233 D261 Y338 W372 D374 R425 W439 D442 F475 H502 2.4.1.161 0003824,0004553,0005975,0016757,0030246,0033825 remove_due_to_license_issue B3PEE6 27280170 910 AVFYKEHKLRNDGLVITTNQGNIRLQFKSEAAIEVLYRADSKQLPSFALAQPESAIKAQLTETENHLQFSGGTLTARIQKRPFAISYYRDSELLLAEESGFQKINFRFYLSPGEKILGGGQRILGMDRRGQRFPLYNRAHYGYSDHSGQMYFGLPAIMSSKQYILVFDNSASGAMDIGKTESDILQLEAKSGRSAYILVAGNSYPSLIENFTQVTGRQPLPPRWALGSFASRFGYRSEAETRATVQKYKTEDFPLDTIVLDLYWFGKDIKGHMGNLDWDKENFPTPLDMMADFKQQGVKTVLITEPFVLTSSKRWDDAVKAKALAKDPQGQPKAFELYFGNGGIIDVFSKEGSRWFSSIYKDLSKQGVAGWWGDLGEPEMHPEDTQHAIGDADTVHNAYGHRWAEMLYQQQLDQFPELRPFIMMRAGFVGSQRYGMIPWTGDVSRTWGGLASQVELALQMSLLGFGYIHSDLGGFADGETLDKEMYIRWLQYGVFQPVYRPHGQDHIPSEPVFQDEETKAILRPLVKLRYRMLPYIYTAAYQNTLTGMPLMRPLFFSDEKNPALIDNKTSYFWGDSLLVTPITQAGVESVSIPAPKGVWFDFWKDTRYQTDGAPLTLPTDLHTIPVLVKAGAFMPYVPAVSTTEDYRSDSLEIHYYADASVPLAQGEIFEDDGKDPNSIKRNQFDLLTLQATHTDNQLHFQLARTGKGYRGMPERRATTLVIHNASDQYQHLDINGKTIAIAQADCASTPALACYDQERRQLQLVFTWGREALNLRLHK 5i24 A 1.85 BS01 66U A 1 F271 D299 W410 D412 R463 W477 D480 F513 H540 F233 D261 W372 D374 R425 W439 D442 F475 H502 2.4.1.161 0003824,0004553,0005975,0016757,0030246,0033825 remove_due_to_license_issue B3PEE6 27280170 907 AVFYKEHKLRNDGLVITTNQGNIRLQFKSEAAIEVLYRADSKQLPSFALAQPESAIKAQLTETENHLQFSGGTLTARIQKRPFAISYYRDSELLLAEESGFQKINFRFYLSPGEKILGGGQRILGMDRRGQRFPLYNRAHYGYSDHSGQMYFGLPAIMSSKQYILVFDNSASGAMDIGKTESDILQLEAKSGRSAYILVAGNSYPSLIENFTQVTGRQPLPPRWALGSFASRFGYRSEAETRATVQKYKTEDFPLDTIVLDLYWFGKDIKGHMGNLDWDKENFPTPLDMMADFKQQGVKTVLITEPFVLTSSKRWDDAVKAKALAKDPQGQPKAFELYFGNGGIIDVFSKEGSRWFSSIYKDLSKQGVAGWWGDLGEPEMHPEDTQHAIGDADTVHNAYGHRWAEMLYQQQLDQFPELRPFIMMRAGFVGSQRYGMIPWTGDVSRTWGGLASQVELALQMSLLGFGYIHSDLGGFADGETLDKEMYIRWLQYGVFQPVYRPHGQDHIPSEPVFQDEETKAILRPLVKLRYRMLPYIYTAAYQNTLTGMPLMRPLFFSDEKNPALIDNKTSYFWGDSLLVTPITQAGVESVSIPAPKGVWFDFWKDTRYQTDGAPLTLPTDLHTIPVLVKAGAFMPYVPAVSTTEDYRSDSLEIHYYADASVPLAQGEIFEDDGKDPNSIKRNQFDLLTLQATHTDNQLHFQLARTGKGYRGMPERRATTLVIHNASDQYQHLDINGKTIAIAQADCASTPALACYDQERRQLQLVFTWGREALNLRLHK 5i29 A 1.21 BS01 67B A 1 W1526 P1527 V1532 N1533 F1536 V1537 Y1582 N1583 Y1589 W27 P28 V33 N34 F37 V38 Y83 N84 Y90 2.3.1.48,2.7.11.1 0004402,0005669,0006366,0016251,0017025 Kd=15nM remove_due_to_license_issue IC50=3600nM P21675 27219867 1701 DDDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESLDPMT 5i2e A 1.6 BS01 67D A 1 I22 F41 D43 I44 N99 G105 Q106 S107 H112 H114 I11 F30 D32 I33 N88 G94 Q95 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=0.23uM remove_due_to_license_issue P49773 27563403 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5i2e B 1.6 BS01 67D A 1 M121 H122 W123 M106 H107 W108 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 27563403 201 DTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5i2f A 1.25 BS01 BS5 A 1 I18 D43 I44 N99 G105 Q106 S107 H112 H114 I8 D33 I34 N89 G95 Q96 S97 H102 H104 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue Kd=320nM, IC50=1000nM P49773 27563403 201 ARPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5i2r A 2.5 BS02 67A A 1 L675 I692 M713 Q726 F729 L218 I235 M256 Q269 F272 3.1.4.17 0004114,0007165,0008081 ic50=0.019uM remove_due_to_license_issue IC50=14nM Q9Y233 26878596 803 GLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 5i2z A 2.3 BS01 V24 A 1 G179 I180 L181 A182 H183 L214 T215 H218 H228 P238 T239 Y240 G73 I74 L75 A76 H77 L108 T109 H112 H122 P132 T133 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27356908 301 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i38 A 2.6 BS03 KOJ A 1 H42 H60 N205 H208 V217 V218 H38 H56 N201 H204 V213 V214 H60 H69 H56 H65 ? 0016491,0046872 remove_due_to_license_issue IC50=52000nM B2ZB02 27725765 303 YRVRKNVLHLTDTEKRDFVRTVLILKEKGIYDRYIAWHGAAGKFHTPPGSDRNAAHMSSAFLPWHREYLLRFERDLQSINPEVTLPYWEWETDAQMQDPSQSQIWSADFMGGNGNPIKDFIVDTGPFAAGRWTTIDEQGNPSGGLKRNFGATKEAPTLPTRDDVLNALKITQYDTPPWDMTSQNSFRNQLEGFINGPQLHNRVHRWVGGQMGVVPTAPNDPVFFLHHANVDRIWAVWQIIHRNQNYQPMKNGPFGQNFRDPMYPWNTTPEDVMNHRKLGYVYDIEL 5i3a A 2.2 BS03 HQE A 1 H42 H60 H204 N205 H208 V218 H39 H57 H201 N202 H205 V215 H60 H69 H57 H66 ? 0016491,0046872 Kd=9uM remove_due_to_license_issue B2ZB02 27725765 303 KYRVRKNVLHLTDTEKRDFVRTVLILKEKGIYDRYIAWHGAAGKFHTPPGSDRNAAHMSSAFLPWHREYLLRFERDLQSINPEVTLPYWEWETDAQMQDPSQSQIWSADFMGGNGNPIKDFIVDTGPFAAGRWTTIDEQGNPSGGLKRNFGATKEAPTLPTRDDVLNALKITQYDTPPWDMTSQNSFRNQLEGFINGPQLHNRVHRWVGGQMGVVPTAPNDPVFFLHHANVDRIWAVWQIIHRNQNYQPMKNGPFGQNFRDPMYPWNTTPEDVMNHRKLGYVYDIEL 5i3m A 2.17 BS01 67F A 1 I180 A182 H183 L214 T215 H218 Q219 H222 H228 F237 P238 T239 Y240 I74 A76 H77 L108 T109 H112 Q113 H116 H122 F131 P132 T133 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27356908 301 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i3v A 1.62 BS01 68M A 1 D32 G34 Y71 K75 W76 F108 D228 D34 G36 Y73 K77 W78 F110 D220 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 Kd=16nM remove_due_to_license_issue IC50=16nM P56817 26978477 404 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5i3w A 2.15 BS01 68L A 1 G11 Q12 G13 L30 D32 Y71 F108 R128 D228 G230 T232 G13 Q14 G15 L32 D34 Y73 F110 R130 D219 G221 T223 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 Kd=0.6nM remove_due_to_license_issue P56817 26978477 406 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 5i3x A 1.85 BS01 68J A 1 G13 D32 G34 V69 Y71 K75 W76 F108 Y198 D228 G230 T232 G15 D34 G36 V71 Y73 K77 W78 F110 Y190 D220 G222 T224 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 Kd=8nM remove_due_to_license_issue Kd=8.0nM, IC50=191nM P56817 26978477 401 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIP 5i3y A 2.15 BS01 68K A 1 G11 Q12 G13 D32 G34 V69 Y71 K75 W76 F108 I118 R128 Y198 D228 S229 G230 T232 G13 Q14 G15 D34 G36 V71 Y73 K77 W78 F110 I120 R130 Y191 D221 S222 G223 T225 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D221 T224 3.4.23.46 0004190,0006508,0016020 Kd=0.4nM remove_due_to_license_issue IC50=16nM, Kd=0.400000nM P56817 26978477 401 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5i40 A 1.0402 BS01 67N A 1 F44 F45 V49 I53 N100 Y106 F23 F24 V28 I32 N79 Y85 ? ic50=13.7uM remove_due_to_license_issue IC50=13700nM Q9H8M2 27219867 206 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSK 5i43 A 1.95 BS06 67M A 1 G178 G179 I180 A182 H183 L214 H218 Q219 H222 H228 P238 Y240 G72 G73 I74 A76 H77 L108 H112 Q113 H116 H122 P132 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27356908 306 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i44 A 2.621 BS01 dna U 0 T7 N8 K19 Q22 K26 R34 G38 H39 Y40 T6 N7 K18 Q21 K25 R33 G37 H38 Y39 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 A 2.621 BS02 dna W 0 S17 R23 L37 S16 R22 L36 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 B 2.621 BS01 dna U 0 T20 R23 Q27 T19 R22 Q26 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 B 2.621 BS02 dna W 0 T7 K19 Q22 K26 R34 H39 Y40 T6 K18 Q21 K25 R33 H38 Y39 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 D 2.621 BS01 dna U 0 S17 R23 S16 R22 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 D 2.621 BS02 dna R 0 I63 Q64 I62 Q63 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 D 2.621 BS03 dna W 0 T7 N8 K19 Q22 K26 R34 G38 H39 Y40 T6 N7 K18 Q21 K25 R33 G37 H38 Y39 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 E 2.621 BS01 dna U 0 T7 K19 K26 R34 H39 Y40 T6 K18 K25 R33 H38 Y39 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 E 2.621 BS02 dna W 0 S17 K19 T20 R23 Q27 S16 K18 T19 R22 Q26 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 F 2.621 BS01 dna R 0 T7 N8 K19 Q22 R34 G38 H39 Y40 T6 N7 K18 Q21 R33 G37 H38 Y39 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 F 2.621 BS02 dna P 0 S17 R23 S16 R22 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 G 2.621 BS01 dna R 0 K17 R21 I61 K17 R21 I61 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 SHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLPK 5i44 G 2.621 BS02 dna P 0 T5 K17 Q20 K24 R32 H37 Y38 T5 K17 Q20 K24 R32 H37 Y38 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 SHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLPK 5i44 H 2.621 BS01 dna T 0 N2 T3 K15 Q18 K22 G34 H35 Y36 N2 T3 K15 Q18 K22 G34 H35 Y36 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 MNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 H 2.621 BS02 dna Z 0 S13 T16 R19 S13 T16 R19 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 MNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 I 2.621 BS01 dna R 0 V12 S13 T16 R19 V12 S13 T16 R19 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 MNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 I 2.621 BS02 dna P 0 T3 K15 Q18 R30 H35 Y36 T3 K15 Q18 R30 H35 Y36 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 MNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHLP 5i44 J 2.621 BS01 dna T 0 K19 Q22 R34 H39 Y40 K18 Q21 R33 H38 Y39 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 J 2.621 BS02 dna Z 0 K19 R23 K18 R22 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 GSHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 K 2.621 BS01 dna T 0 S15 R21 S15 R21 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 SHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i44 K 2.621 BS02 dna Z 0 T5 K17 Q20 G36 H37 Y38 T5 K17 Q20 G36 H37 Y38 ? 0003677,0006355 remove_due_to_license_issue P45870 27085804 1 ~ 14 SHMNTNMVASELGVSAKTVQRWVKQLNLPAERNELGHYSFTAEDVKVLKSVKKQISEGTAIQDIHL 5i4o A 2.05 BS01 V28 A 1 G179 I180 A182 L214 T215 H218 Q219 H222 H228 V235 F237 P238 Y240 G72 I73 A75 L107 T108 H111 Q112 H115 H121 V128 F130 P131 Y133 H218 Q219 H222 H228 H111 Q112 H115 H121 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27356908 301 VWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i4v A 2.61 BS01 67S A 1 F271 T272 L274 E281 M312 F329 L330 H435 F54 T55 L57 E64 M95 F112 L113 H218 ? 0003677,0004879,0006629 remove_due_to_license_issue P55055,Q15596 26990539 501 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGADPASGSASQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVHEGSGSGSHKILHRLLQD 5i50 A 2.701 BS01 dna C 0 E16 R19 E16 R19 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 27748763 1 ~ 22 MATEENVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAETQKLISEIDLLRKQNEQLKHKLEQLRNSCA 5i50 A 2.701 BS02 dna D 0 R9 H12 N13 E16 R17 R20 K24 P44 K45 R9 H12 N13 E16 R17 R20 K24 P44 K45 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 27748763 1 ~ 22 MATEENVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAETQKLISEIDLLRKQNEQLKHKLEQLRNSCA 5i50 B 2.701 BS01 dna C 0 R9 H12 N13 E16 R17 R20 P44 K45 R13 H16 N17 E20 R21 R24 P48 K49 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 27748763 1 ~ 22 FQGAMATEENVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAETQKLISEIDLLRKQNEQLKHKLEQLRNSCA 5i50 B 2.701 BS02 dna D 0 H12 E16 R19 H16 E20 R23 ? 0003700,0006355,0046983 remove_due_to_license_issue P01106 27748763 1 ~ 22 FQGAMATEENVKRRTHNVLERQRRNELKRSFFALRDQIPELENNEKAPKVVILKKATAYILSVQAETQKLISEIDLLRKQNEQLKHKLEQLRNSCA 5i56 A 2.28 BS02 67P B 1 P140 Y143 R363 S364 G365 P135 Y138 R242 S243 G244 ? 0015276,0016020 remove_due_to_license_issue P35439 27618671 802 TRLKIVTIHQEPFVYVKPTMSDGTCKEEFTVNGDPVKKVICTGPNDTSPGSPRHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWVRYQECD 5i56 B 2.28 BS02 67P B 1 P130 F131 V132 E133 V267 M272 E276 P126 F127 V128 E129 V263 M268 E272 ? 0015276,0016020 ic50=1530nM remove_due_to_license_issue IC50=170nM Q00959 27618671 802 DDNHLSIVTLEEAPFVIVEDIDPLTETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGIC 5i58 A 2.52 BS02 67R B 1 P140 Y143 R247 G249 P112 Y115 R219 G221 ? 0015276,0016020 remove_due_to_license_issue P35439 27618671 302 STRLKIVTIHQEPFVYVKPTMSDGTCVKKVICTGPVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWV 5i58 B 2.52 BS02 67R B 1 V129 P130 F131 V132 E133 V267 M272 E276 V122 P123 F124 V125 E126 V260 M265 E269 ? 0015276,0016020 remove_due_to_license_issue Q00959 27618671 302 DNHLSIVTLEEAPFVIVEDIDPETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGIC 5i59 A 2.25 BS02 67Q B 1 P140 R247 S248 G249 P117 R224 S225 G226 ? 0015276,0016020 remove_due_to_license_issue P35439 27618671 302 TRLKIVTIHQEPFVYVKPTMSDGTCVKKVICTGPHTVPQCCYGFCIDLLIKLARTMNFTYEVHLVADGKFGTQERVNSNKKEWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKGTRITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQNVSLSILKSHENGFMEDLDKTWV 5i59 B 2.25 BS02 67Q B 1 P130 F131 V132 E133 V267 E276 L280 P121 F122 V123 E124 V258 E267 L271 ? 0015276,0016020 ic50=641nM remove_due_to_license_issue Q00959 27618671 302 DNHLSIVTLEEAPFVIVEDIETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGIC 5i5x A 1.65 BS02 68C A 1 F30 F75 K79 Y141 V170 Y173 A314 F25 F70 K74 Y136 V165 Y168 A307 K202 K195 2.6.1.42 0003824,0004084,0005515,0005654,0005739,0005759,0006549,0006550,0006551,0006573,0006629,0008483,0008652,0009081,0009082,0009083,0009098,0009099,0010817,0052654,0052655,0052656,1990830 ic50=0.2uM remove_due_to_license_issue IC50=200nM O15382 26938474 402 SSFKAADLQLEMTQKPHKKPGPLVFGKTFTDHMLMVEWNDKGWGQPRIQPFQNLTLHPASSSLHYSLQLFEGMKAFKGKDQQVRLFRPWLNMDRMLRSAMRLCLPSFDKLELLECIRRLIEVDKDWVPDAAGTSLYVRPVLIGNEPSLGVSQPTRALLFVILCPVGAYFGSVTPVSLLADPAFIRAWVGGVGNYKLGGNYGPTVLVQQEALKRGCEQVLWLYGPDHQLTEVGTMNIFVYWTHEDGVLELVTPPLNGVILPGVVRQSLLDMAQTWGEFRVVERTITMKQLLRALEEGRVREVFGSGTACQVCPVHRILYKDRNLHIPTMENGPELILRFQKELKEIQYGIRAHEWMFPV 5i5x B 1.65 BS02 68C B 1 F30 F75 K79 Y141 Y173 A314 F29 F74 K78 Y140 Y172 A313 K202 K201 2.6.1.42 0003824,0004084,0005515,0005654,0005739,0005759,0006549,0006550,0006551,0006573,0006629,0008483,0008652,0009081,0009082,0009083,0009098,0009099,0010817,0052654,0052655,0052656,1990830 ic50=0.2uM remove_due_to_license_issue IC50=200nM O15382 26938474 402 SHMASSSFKAADLQLEMTQKPHKKPGLVFGKTFTDHMLMVEWNDKGWGQPRIQPFQNLTLHPASSSLHYSLQLFEGMKAFKGKDQQVRLFRPWLNMDRMLRSAMRLCLPSFDKLELLECIRRLIEVDKDWVPDAAGTSLYVRPVLIGNEPSLGVSQPTRALLFVILCPVGAYFPGGSVTPVSLLADPAFIRAWVGGVGNYKLGGNYGPTVLVQQEALKRGCEQVLWLYGPDHQLTEVGTMNIFVYWTHEDGVLELVTPPLNGVILPGVVRQSLLDMAQTWGEFRVVERTITMKQLLRALEEGRVREVFGSGTACQVCPVHRILYKDRNLHIPTMENGPELILRFQKELKEIQYGIRAHEWMFPV 5i5z A 2.6 BS01 68U A 1 V27 Y32 A50 K52 F97 A100 H106 L158 R356 V30 Y35 A53 K55 F100 A103 H109 L156 R339 D151 K153 N156 D173 N181 T196 D149 K151 N154 D171 N179 T184 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.900000nM P49336 27326329 401 DDKMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKANLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLKTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQSNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEE 5i7u A 1.95 BS01 6AJ A 1 E205 E206 Y547 S630 Y631 V656 Y662 Y666 V711 E167 E168 Y509 S592 Y593 V618 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=1.7nM remove_due_to_license_issue IC50=1.7nM P27487 27190600 812 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5i7x A 1.1752 BS01 67B A 1 F44 F45 V49 I53 N100 Y106 F23 F24 V28 I32 N79 Y85 ? Kd=53nM remove_due_to_license_issue IC50=230nM Q9H8M2 27219867 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 5i7y A 1.4514 BS01 69G A 1 F44 F45 V49 I53 N100 Y106 F23 F24 V28 I32 N79 Y85 ? Kd=52nM remove_due_to_license_issue Q9H8M2 27219867 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 5i80 A 1.4501 BS01 67B A 1 W81 P82 V87 L92 N140 I146 W40 P41 V46 L51 N99 I105 ? Kd=62nM remove_due_to_license_issue IC50=92nM O60885 27219867 201 STNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5i83 A 1.35 BS01 68Y A 1 P1110 V1115 L1120 Y1125 N1168 R1173 V1174 P28 V33 L38 Y43 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=4.1uM remove_due_to_license_issue IC50=652nM Q92793 27190605 1202 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5i86 A 1.05 BS01 69A A 1 P1110 V1115 L1120 I1122 Y1125 N1168 R1173 V1174 P29 V34 L39 I41 Y44 N87 R92 V93 2.3.1.-,2.3.1.48 ic50=0.53uM remove_due_to_license_issue IC50=530nM Q92793 27190605 1203 KKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5i88 A 1.4 BS01 69G A 1 W81 P82 F83 V87 L92 N140 I146 W40 P41 F42 V46 L51 N99 I105 ? Kd=250nM remove_due_to_license_issue O60885 27219867 205 STNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5i89 A 1.07 BS01 69B A 1 P1110 V1115 L1120 Y1125 N1168 R1173 V1174 P28 V33 L38 Y43 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=0.033uM remove_due_to_license_issue IC50=49.0nM, EC50=3000nM Q92793 27190605 1203 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5i8b A 1.5218 BS04 69F A 1 P1110 V1115 L1120 N1168 R1173 V1174 P32 V37 L42 N90 R95 V96 2.3.1.-,2.3.1.48 0004402,0006355 ic50=0.11uM remove_due_to_license_issue EC50=>10000nM, IC50=110nM Q92793 27190605 1404 GSRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLGYCCGRKYEFSPQTLCCYGKQLCTIPRDAAYYSYQNRYHFCEKCFTLGDDPSQPQTTISKDQFEKKKNDTLDPEPFVDCKECGRKMHQICVLHYDIIWPSGFVCDNCL 5i8g A 1.41 BS04 69E A 1 L1109 P1110 Q1113 V1115 L1120 N1168 V1174 L31 P32 Q35 V37 L42 N90 V96 2.3.1.-,2.3.1.48 0004402,0006355 Kd=0.03uM remove_due_to_license_issue IC50=30nM, Kd=30nM, EC50=300nM Q92793 27190605 1404 GSRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLGYCCGRKYEFSPQTLCCYGKQLCTIPRDAAYYSYQNRYHFCEKCFTLGDDPSQPQTTISKDQFEKKKNDTLDPEPFVDCKECGRKMHQICVLHYDIIWPSGFVCDNCL 5i8p A 2.37 BS01 VQ7 A 1 F110 L121 G152 L153 L159 S273 F274 W298 F322 H351 Q352 A355 F357 L371 F57 L68 G99 L100 L106 S220 F221 W245 F269 H298 Q299 A302 F304 L318 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 Kd=0.000000064M remove_due_to_license_issue Kd=1.9nM, IC50=1.7nM Q13093 27078579 501 TKIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNI 5i94 A 2.983 BS01 69V A 1 R316 K319 L320 F321 Y393 R181 K184 L185 F186 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=30nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTADGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5i94 B 2.983 BS01 69V B 1 K319 L320 F321 L322 N323 Y393 K184 L185 F186 L187 N188 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=30nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTADGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5i94 C 2.983 BS01 69V B 1 K319 L320 F321 L322 N323 Y393 K184 L185 F186 L187 N188 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=30nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTADGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5i94 D 2.983 BS01 69V A 1 K319 L320 F321 L322 E324 Y393 K184 L185 F186 L187 E189 Y258 S285 K288 Y413 Y465 V483 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=30nM O94925 26988803 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTADGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5i9i A 2.7 BS01 5HV A 1 F110 L111 L121 G152 L153 G154 L159 S273 F274 W298 H351 Q352 F357 L369 L371 F57 L58 L68 G99 L100 G101 L106 S220 F221 W245 H298 Q299 F304 L316 L318 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 remove_due_to_license_issue IC50=0.250000nM, Ki=110nM, Kd=5.0nM Q13093 27078579 501 TKIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINT 5i9x A 1.427 BS01 DB8 A 1 I619 A644 I645 K646 E663 I690 T692 Y694 M695 G698 L746 I16 A36 I37 K38 E55 I82 T84 Y86 M87 G90 L138 D739 A741 R743 N744 D757 D766 P780 D131 A133 R135 N136 D149 D158 P168 2.7.10.1 0004672,0004713,0005524,0006468 Kd=30nM remove_due_to_license_issue Kd=18nM P29317 27768280 1001 FTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5i9y A 1.228 BS01 1N1 A 1 I619 A644 I645 K646 E663 I690 T692 Y694 M695 E696 G698 E706 L746 I20 A42 I43 K44 E61 I88 T90 Y92 M93 E94 G96 E104 L144 D739 A741 R743 N744 D757 D766 P780 D137 A139 R141 N142 D155 D164 P171 2.7.10.1 0004672,0004713,0005524,0006468 Kd=2.8nM remove_due_to_license_issue Kd=0.85nM, IC50=137nM P29317 27768280 1001 AVLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5i9z A 1.698 BS01 627 A 1 I619 A644 K646 E693 Y694 M695 G698 L746 S756 I16 A35 K37 E84 Y85 M86 G89 L137 S147 D739 A741 R743 N744 D757 P780 D130 A132 R134 N135 D148 P157 2.7.10.1 0004672,0004713,0005524,0006468 Kd=9nM remove_due_to_license_issue P29317 27768280 1001 FTTEIHPSCVTRQKVIGAGGEVYKGMLKTKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5ia0 A 1.948 BS01 A5B A 1 I619 A621 V627 A644 K646 Y694 M695 E696 G698 K702 L746 I16 A18 V24 A37 K39 Y87 M88 E89 G91 K95 L139 D739 A741 R743 N744 D757 P780 D132 A134 R136 N137 D150 P154 2.7.10.1 0004672,0004713,0005524,0006468 Kd=187nM remove_due_to_license_issue P29317 27768280 1001 FTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDP 5ia1 A 2.036 BS01 ZZL A 1 I619 V627 A644 K646 Y694 M695 G698 L746 S756 D757 I15 V23 A34 K36 Y84 M85 G88 L136 S146 D147 D739 A741 R743 N744 D757 P780 D129 A131 R133 N134 D147 P153 2.7.10.1 0004672,0004713,0005524,0006468 Kd=530nM remove_due_to_license_issue Kd=370nM P29317 27768280 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFD 5ia2 A 1.619 BS01 L66 A 1 I619 V627 A644 E663 T692 Y694 M695 G698 L746 D757 I22 V30 A43 E62 T91 Y93 M94 G97 L145 D156 D739 A741 R743 N744 D757 D766 P780 D138 A140 R142 N143 D156 D165 P179 2.7.10.1 0004672,0004713,0005524,0006468 Kd=19nM remove_due_to_license_issue IC50=2.3nM P29317 27768280 1001 NQAVLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTSGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFD 5ia3 A 1.788 BS01 P17 A 1 V627 A644 I645 K646 E663 T692 Y694 M695 G698 L746 V26 A39 I40 K41 E58 T87 Y89 M90 G93 L141 D739 A741 R743 N744 D757 P780 D134 A136 R138 N139 D152 P159 2.7.10.1 0004672,0004713,0005524,0006468 Kd=46nM remove_due_to_license_issue Kd=3.8nM P29317 27768280 1001 LKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5ia4 A 1.797 BS01 88Z A 1 I619 A644 K646 E663 M667 Y694 M695 E696 L730 L746 S756 D757 F758 I15 A36 K38 E55 M59 Y86 M87 E88 L122 L138 S148 D149 F150 D739 A741 R743 N744 D757 D766 P780 D131 A133 R135 N136 D149 D158 P172 2.7.10.1 0004672,0004713,0005524,0006468 Kd=52nM remove_due_to_license_issue P29317 27768280 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTSGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRA 5ia5 A 1.776 BS01 GV0 A 1 A644 K646 M667 Y694 M695 E696 G698 E706 L730 S756 D757 A37 K39 M60 Y87 M88 E89 G91 E99 L123 S149 D150 D739 A741 R743 N744 D757 D766 P780 D132 A134 R136 N137 D150 D159 P173 2.7.10.1 0004672,0004713,0005524,0006468 Kd=25nM remove_due_to_license_issue P29317 27768280 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKTSKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTSGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDS 5icp A 2.18 BS01 69Z A 1 V27 Y32 V35 A50 K52 F97 A100 L158 D173 R356 V27 Y32 V35 A50 K52 F97 A100 L151 D166 R337 D151 K153 N156 D173 N181 T196 D144 K146 N149 D166 N174 T181 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=70nM P49336 27490956 401 MDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLKVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQESNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEE 5icv A 1.53 BS02 1XE C 1 S100 L101 G102 V103 R108 K109 G111 G113 S114 H138 V139 F149 Y150 N152 R153 S96 L97 G98 V99 R104 K105 G107 G109 S110 H134 V135 F145 Y146 N148 R149 2.3.1.259,2.3.1.48 0004596,0016747 remove_due_to_license_issue Q9H7X0 27320834 101 VPSSALSEVSLRLLCHDDIDTVKHLCGDWFPIEYPDSWYRDITSNKKFFSLAATYRGAIVGMIVAEIKNRTKIHKEDGDILASNFSVDTQVAYILSLGVVKEFRKHGIGSLLLESLKDHISTTAQDHCKAIYLHVLTTNNTAINFYENRDFKQHHYLPYYYSIRGVLKDGFTYVLYINGG 5id6 A 2.382 BS01 rna G 0 K15 T16 R18 F19 K20 K514 Y516 K518 N706 K707 S710 K712 H714 G715 T716 N718 L719 H720 R747 H759 I765 A766 N767 K768 N769 N772 K774 T777 L779 Y781 V783 Y784 K785 D786 R788 N861 N862 F863 Y872 L875 S905 Q906 H909 K953 K960 K16 T17 R19 F20 K21 K502 Y504 K506 N694 K695 S698 K700 H702 G703 T704 N706 L707 H708 R735 H747 I753 A754 N755 K756 N757 N760 K762 T765 L767 Y769 V771 Y772 K773 D774 R776 N849 N850 F851 Y860 L863 S893 Q894 H897 K941 K948 ? 0046872 remove_due_to_license_issue A0A182DWE3 27096363 3 ~ 23 AASKLEKFTNCYSLSKTLRFKAIPVGKTQENIDNKRLLVEDEKRAEDYKGVKKLLDRYYLSFINDVLHSIKLKNLNNYISLFRKKTRTEKENKELENLEINLRKEIAKAFKGAAGYKSLFKKDIIETILPEAAKDEIALVNSFNGFTTAFTGFFDNRENMFSEEAKSTSIAFRCINENLTRYISNMDIFEKVDAIFDKHEVQEIKEKILNSDYDVEDFFEGEFFNFVLTQEGIDVYNAIIGGFVTESGEKIKGLNEYINLYNAKTKQALPKFKPLYKQVEGYTSDEEVLEVFRNTLNKNSEIFSSIKKLEKLFKNFDEYSSAGIFVKNGPAISTISKDIFGEWNLIRDKWNAEYDDIHLKKKAVVTEKYEDDRRKSFKKIGSFSLEQLQEYADADLSVVEKLKEIIIQKVDEIYKVYGSSEKLFDADFVLEKSLKKNDAVVAIMKDLLDSVKSFENYIKAFFGEGKETNRDESFYGDFVLAYDILLKVDHIYDAIRNYVTQKPYSKDKFKLYFQNPQFMGGWDKDKETDYRATILRYGSKYYLAIMDKKYAKCLQKIDKDDVNGNYEKINYKLLPGPNKMLPKVFFSKKWMAYYNPSEDIQKIYKNGTFKKGDMFNLNDCHKLIDFFKDSISRYPKWSNAYDFNFSETEKYKDIAGFYREVEEQGYKVSFESASKKEVDKLVEEGKLYMFQIYNKDFSDKSHGTPNLHTMYFKLLFDENNHGQIRLSGGAELFMRRASLKKEELVVHPANSPIANKNPDNPKKTTTLSYDVYKDKRFSEDQYELHIPIAINKCPKNIFKINTEVRVLLKHDDNPYVIGIDRGERNLLYIVVVDGKGNIVEQYSLNEIINNFNGIRIKTDYHSLLDKKEKERFEARQNWTSIENIKELKAGYISQVVHKICELVEKYDAVIALEDLNSGFKNSRVKVEKQVYQKFEKMLIDKLNYMVDKKSNPCATGGALKGYQITNKFESFKSMSTQNGFIFYIPAWLTSKIDPSTGFVNLLKTKYTSIADSKKFISSFDRIMYVPEEDLFEFALDYKNFSRTDADYIKKWKLYSYGNRIRIFAAAAWEEVCLTSAYKELFNKYGINYQQGDIRALLCEQSDKAFYSSFMALMSLMLQMRNSITGRTDVDFLISPVKNSDGIFYDSRNYEAQENAILPKNADANGAYNIARKVLWAIGQFKKAEDEKLDKVKIAISNKEWLEYAQTSVK 5idn A 2.26 BS01 6A7 A 1 V27 Y32 A50 K52 F97 A100 L158 R356 V27 Y32 A50 K52 F97 A100 L153 R329 D151 K153 N156 D173 T196 D146 K148 N151 D168 T175 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P49336 27490956 401 MDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKANLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEEE 5idp A 2.65 BS01 6A6 A 1 V27 Y32 V35 A50 F97 D98 A100 A155 L158 D173 R356 V28 Y33 V36 A51 F98 D99 A101 A151 L154 D169 R339 D151 K153 N156 D173 N181 T196 D147 K149 N152 D169 N177 T182 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=800nM P49336 27490956 401 KMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLKTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQETSNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFL 5ie1 A 2.298 BS01 6BS A 1 D32 G34 Y71 K75 W76 F108 R128 Y198 D228 D34 G36 Y73 K77 W78 F110 R130 Y189 D219 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D219 T222 3.4.23.46 0004190,0006508,0016020 Kd=140nM remove_due_to_license_issue Kd=140nM P56817 26978477 407 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5iee A 1.92 BS01 NOJ A 1 W423 D451 W562 D564 M565 R624 W637 D640 F673 H698 W314 D342 W453 D455 M456 R515 W528 D531 F564 H589 3.2.1.207 0003824,0004553,0005975,0030246 remove_due_to_license_issue Q8BHN3 27462106 1023 VDRSNFKTCDESSFCKRQRSIRPGLSPYRALLDTLQLGPDALTVHLIHEVTKVLLVLELQGLQKNMTRIRIDELEPRRPRYRVPDVLVADPPTARLSVSGRDDNSVELTVAEGPYKIILTAQPFRLDLLEDRSLLLSVNARGLMAFEHQRAPREPGAWEETFKTHSDSKPYGPTSVGLDFSLPGMEHVYGIPEHADSLRLKVTEGGEPYRLYNLDVFQYELNNPMALYGSVPVLLAHSFHRDLGIFWLNAAETWVDISSNTPQTDIRWMSESGIIDVFLMLGPSVFDVFRQYASLTGTQALPPLFSLGYHQSRWNYRDEADVLEVDQGFDDHNMPCDVIWLDIEHADGKRYFTWDPTRFPQPLNMLEHLASKRRKLVAIVDPHIKVDSGYRVHEELRNHGLYVKTRDGSDYEGWCWPGSASYPDFTNPRMRAWWSNMFSFDNYEGSAPNLYVWNDMNEPSVFNGPEVTMLKDAVHYGGWEHRDIHNIYGLYVHMATADGLIQRSGGIERPFVLSRAFFSGSQRFGAVWTGDNTAEWDHLKISIPMCLSLALVGLSFCGADVGGFFKNPEPELLVRWYQMGAYQPFFRAHAHLDTGRREPWLLASQYQDAIRDALFQRYSLLPFWYTLFYQAHKEGFPVMRPLWVQYPEDMSTFSIEDQFMLGDALLIHPVSDAGAHGVQVYLPGQEEVWYDIQSYQKHHGPQTLYLPVTLSSIPVFQRGGTIVPRWMRVRRSSDCMKDDPITLFVALSPQGTAQGELFLDDGHTFNYQTRHEFLLRRFSFSGSTLVSSSADPKGHLETPIWIERVVIMGAGKPAAVVLQTKGSPESRLSFQHDPETSVLILRKPGVSVASDWSIHLR 5ief A 2.38 BS01 NBV A 1 W423 D451 W562 D564 F571 R624 W637 D640 F673 H698 W314 D342 W453 D455 F462 R515 W528 D531 F564 H589 3.2.1.207 0003824,0004553,0005515,0005783,0005794,0005975,0006491,0015926,0016798,0017177,0030246,0033919,0042470,0043231,0090599,0106407 remove_due_to_license_issue Q8BHN3 27462106 1005 VDRSNFKTCDESSFCKRQRSIRPGLSPYRALLDTLQLGPDALTVHLIHEVTKVLLVLELQGLQKNMTRIRIDELEPRRPRYRVPDVLVADPPTARLSVSGRDDNSVELTVAEGPYKIILTAQPFRLDLLEDRSLLLSVNARGLMAFEHQRAPREPGAWEETFKTHSDSKPYGPTSVGLDFSLPGMEHVYGIPEHADSLRLKVTEGGEPYRLYNLDVFQYELNNPMALYGSVPVLLAHSFHRDLGIFWLNAAETWVDISSNTPQTDIRWMSESGIIDVFLMLGPSVFDVFRQYASLTGTQALPPLFSLGYHQSRWNYRDEADVLEVDQGFDDHNMPCDVIWLDIEHADGKRYFTWDPTRFPQPLNMLEHLASKRRKLVAIVDPHIKVDSGYRVHEELRNHGLYVKTRDGSDYEGWCWPGSASYPDFTNPRMRAWWSNMFSFDNYEGSAPNLYVWNDMNEPSVFNGPEVTMLKDAVHYGGWEHRDIHNIYGLYVHMATADGLIQRSGGIERPFVLSRAFFSGSQRFGAVWTGDNTAEWDHLKISIPMCLSLALVGLSFCGADVGGFFKNPEPELLVRWYQMGAYQPFFRAHAHLDTGRREPWLLASQYQDAIRDALFQRYSLLPFWYTLFYQAHKEGFPVMRPLWVQYPEDMSTFSIEDQFMLGDALLIHPVSDAGAHGVQVYLPGQEEVWYDIQSYQKHHGPQTLYLPVTLSSIPVFQRGGTIVPRWMRVRRSSDCMKDDPITLFVALSPQGTAQGELFLDDGHTFNYQTRHEFLLRRFSFSGSTLVSSSADPKGHLETPIWIERVVIMGAGKPAAVVLQTKGSPESRLSFQHDPETSVLILRKPGVSVASDWSIHLRA 5ieg A 1.822 BS01 6A9 A 1 F307 W423 D451 I452 W562 D564 R624 W637 D640 F673 H698 F217 W314 D342 I343 W450 D452 R512 W525 D528 F561 H586 3.2.1.207 0003824,0004553,0005515,0005783,0005794,0005975,0006491,0015926,0016798,0017177,0030246,0033919,0042470,0043231,0090599,0106407 remove_due_to_license_issue Q8BHN3 27462106 1003 VDRSNFKTCDESSFCKRQRSIRPGLSPYRALLDTLQLGPDALTVHLIHEVTKVLLVLELQGLQKNMTRIRIDELEPRRPRYRVPDVLVADPPTARLSVSGRDDNSVELTVAEGPYKIILTAQPFRLDLLEDRSLLLSVNARGLMAFEHQRAPREPGAWEETFKTHSDSKPYGPTSVGLDFSLPGMEHVYGIPEHADSLRLKVTEGGEPYRLYNLDVFQYELNNPMALYGSVPVLLAHSFHRDLGIFWLNAAETWVDISSNTPQTDIRWMSESGIIDVFLMLGPSVFDVFRQYASLTGTQALPPLFSLGYHQSRWNYRDEADVLEVDQGFDDHNMPCDVIWLDIEHADGKRYFTWDPTRFPQPLNMLEHLASKRRKLVAIVDPHIKVDSGYRVHEELRNHGLYVKTRDGSDYEGWCSASYPDFTNPRMRAWWSNMFSFDNYEGSAPNLYVWNDMNEPSVFNGPEVTMLKDAVHYGGWEHRDIHNIYGLYVHMATADGLIQRSGGIERPFVLSRAFFSGSQRFGAVWTGDNTAEWDHLKISIPMCLSLALVGLSFCGADVGGFFKNPEPELLVRWYQMGAYQPFFRAHAHLDTGRREPWLLASQYQDAIRDALFQRYSLLPFWYTLFYQAHKEGFPVMRPLWVQYPEDMSTFSIEDQFMLGDALLIHPVSDAGAHGVQVYLPGQEEVWYDIQSYQKHHGPQTLYLPVTLSSIPVFQRGGTIVPRWMRVRRSSDCMKDDPITLFVALSPQGTAQGELFLDDGHTFNYQTRHEFLLRRFSFSGSTLVSSSADPKGHLETPIWIERVVIMGAGKPAAVVLQTKGSPESRLSFQHDPETSVLILRKPGVSVASDWSIHLRAS 5ien A 2.089 BS01 VDY A 1 F15 L58 Y104 E106 L125 F14 L57 Y103 E105 L124 remove_due_to_license_issue 30566669 201 QSAKEAIEAALADFVKAYNSKDAAGVASKYMDDAAIFPLDMARVDGRQNIQKLWQGLMDMGVSEPKLTTLDVQESGDFAFESGSISLKGPGKDSKLVDIAGKYVEVWRKGQDGGWKLYRTIANLDPAEH 5ieo A 1.851 BS01 VDY A 1 F15 P39 M61 F86 L88 Y104 E106 F15 P39 M61 F86 L88 Y98 E100 remove_due_to_license_issue 30566669 206 LPTAHEAIEAALADFVKVYNSKDAAGVASKYMDDAVIFPLDMARVDGRQNIQKLWQGLMDMGVSEPKFTTLNVQESGDFAFESGSFSLKGPVDIAGIYVEVWRKGGWKLYRTIANLDP 5iep A 1.893 BS01 VDY A 1 F15 M61 F86 L88 Y104 E106 F14 M60 F85 L87 Y98 E100 remove_due_to_license_issue 30566669 201 QSAKEAIEAALADFVKVYNSKDAAGVASKYMDDAAIFPLDMAPVDGRQNIQKLWQGLMDMGVSEPKFTTLNVQKSGDFAFESGSFSLKGPLVDIAGIYVEVWRKGQDGGWKLYRTIANLDP 5ier A 2.005 BS01 3QZ A 1 L12 T43 A91 S93 F107 Y109 L11 T42 A90 S92 F106 Y108 remove_due_to_license_issue 28980354 201 QSPALIASQSLWRCTQAHDREGWLALMADDVVIETPIGKSVTNPDGSGIKGKEAVGAFFDTHIAATRLTVTCEETFPSSSPDEIAHILVAHSEFDGGFTSEVRGVFTYRVNKAGLITNLRGYWNLDMMTFG 5iez A 2.6 BS01 6AL A 1 A227 F228 M231 M250 F254 R263 T266 L267 F270 G271 A57 F58 M61 M80 F84 R93 T96 L97 F100 G101 ? 0042981 remove_due_to_license_issue Ki=23nM Q07820 27878989 400 DDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 5if4 A 2.392 BS01 6AK A 1 H224 A227 F228 M231 V249 M250 V253 F254 N260 R263 L267 F270 G271 I294 H53 A56 F57 M60 V78 M79 V82 F83 N89 R92 L96 F99 G100 I123 ? 0042981 Ki<1nM remove_due_to_license_issue Ki=<1.000000nM Q07820 27878989 400 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 5if6 A 2.501 BS01 3QZ A 1 L12 F107 Y124 L12 F107 Y124 remove_due_to_license_issue 28980354 201 TQSPALIASQSLGRCTQAKDREGWLALMADDVVIETPIGKSVTNPDGSGIKGKEAVGAFWDTHIADDRVTVTCEETFPSSSPDEIAHILVAHAEFDGGFTSEVRGVFTYRVNKAGLITNLRGYYNLDMMTFGNQ 5ifu A 2.45 BS01 GBM A 1 F262 Y266 E404 R514 G517 M521 Y746 F12 Y16 E103 R213 G216 M220 Y438 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=34uM remove_due_to_license_issue Q8I5R7 27798837 801 ILGITSKKIENFSDWYTQVIVKSELIEYYDISGCYILRPAAYYIWECVQAFFNKEIKKLNVENSYFPLFVTSETIMYSVFPKWIRSYRDLPLKLNQWNTVTREFLWQEGHTAHKNEEEAVKLVFDILDLYRRWYEEYLAVPIIKGIKSEGEKFGGANFTSTAEAFISENGRAIQAATSHYLGTNFAKMFKIEFEDENEVKQYVHQTSWGCTTRSIGIMIMTHGDDKGLVLPPNVSKYKVVIVPIFYKTTDENAIHSYCKDIEKILKNAQINCVYDDRASYSPGYKFNHWELRGIPIRIEVGPKDLQNNSCVIVRRDNNEKCNVKKESVLLETQQMLVDIHKNLFLKAKKKLDDSIVQVTSFSEVMNALNKKKMVLAPWCEDIATEEEIKKETQRLSLNLSGAMKPLCIPLDQPPMPPNMKCFWSGKPAKRWCLFGRSY 5igk A 1.7 BS01 BMF A 1 W81 F83 Q85 V87 K91 L92 N140 I146 W40 F42 Q44 V46 K50 L51 N99 I105 ? Kd=41.8nM remove_due_to_license_issue Kd=42nM, IC50=116nM O60885 27757418 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5igl A 2.1 BS01 BMF A 1 F1547 V1551 N1552 V1556 Y1601 N1602 Y1608 F36 V40 N41 V45 Y90 N91 Y97 ? 0004402,0005669,0006366,0016251,0017025 Kd=42.7nM remove_due_to_license_issue Kd=25000nM Q8IZX4 27757418 1701 LGTENLYFQSMQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKMIVNPVDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNICYQTITEYDEHLTQLEKDICTAKEAALEEAEL 5igm A 1.6 BS01 BMF A 1 F160 F161 F163 V165 I169 N216 Y222 F23 F24 F26 V28 I32 N79 Y85 ? Kd=41.7nM remove_due_to_license_issue IC50=47nM, Kd=114nM Q9H8M2 27757418 301 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5ih5 A 2.25 BS02 AUE A 1 I23 A36 K38 E52 M80 M82 L84 L85 I148 I22 A35 K37 E51 M79 M81 L83 L84 I147 D128 K130 D127 K129 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.5uM remove_due_to_license_issue IC50=5e+2nM P48730 27049670 302 ELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 5ih6 A 2.3 BS02 AUG A 1 I23 A36 M80 M82 L84 L85 L135 I148 I22 A35 M79 M81 L83 L84 L134 I147 D128 K130 D127 K129 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=2.5uM remove_due_to_license_issue IC50=2.5e+3nM P48730 27049670 305 ELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 5ih8 A 1.85 BS01 6BJ A 1 E15 I17 L27 A38 E87 Y88 C89 P90 L139 I149 E14 I16 L23 A34 E80 Y81 C82 P83 L132 I142 D132 K134 E136 N137 D150 S171 D125 K127 E129 N130 D143 S150 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.18uM remove_due_to_license_issue IC50=180nM Q14680 27187609 401 MDYDELLKYYELHETIGTAKVKLACHILTGEMVAIKIMDKNTDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARG 5ih9 A 1.79 BS01 6BF A 1 I17 L27 A38 Y88 C89 P90 E93 L139 I149 I16 L26 A37 Y83 C84 P85 E88 L134 I144 D132 K134 E136 N137 D150 S171 D127 K129 E131 N132 D145 S152 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 Kd=0.002uM remove_due_to_license_issue IC50=2.0nM Q14680 27187609 401 MDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARG 5iha A 1.96 BS01 6BE A 1 I17 L27 A38 Y88 C89 P90 L139 I149 I16 L22 A33 Y78 C79 P80 L129 I139 D132 K134 E136 N137 D150 S171 D122 K124 E126 N127 D140 S147 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.41uM remove_due_to_license_issue IC50=410nM Q14680 27187609 401 MDYDELLKYYELHETIGAKVKLACHILTGEMVAIKIMDKNTLRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARG 5ihc A 2.14 BS01 6BB A 1 I17 L27 A38 Y88 C89 P90 E93 L139 I149 I16 L23 A34 Y84 C85 P86 E89 L135 I145 D132 K134 E136 N137 D150 S171 D128 K130 E132 N133 D146 S149 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=0.013uM remove_due_to_license_issue IC50=13nM Q14680 27187609 401 MDYDELLKYYELHETIGTAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARG 5ihh A 1.35 BS01 6B5 A 1 K15 L17 L110 S117 T119 K6 L8 L101 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=390nM remove_due_to_license_issue P02766 27050398 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5ihh B 1.35 BS01 6B5 B 1 K15 L17 L110 S117 T119 K6 L8 L101 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=390nM remove_due_to_license_issue P02766 27050398 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5ii1 A 2.02 BS01 6BL A 1 I683 F684 L687 Y696 M704 A735 I745 I32 F33 L36 Y45 M53 A84 I94 ? 0006338,0016586 remove_due_to_license_issue Q86U86 27617704 801 SKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDL 5ii2 A 2.1 BS01 LU2 A 1 I683 F684 L687 P688 Y696 D705 M731 A735 I745 I32 F33 L36 P37 Y45 D54 M80 A84 I94 ? 0006338,0016586 remove_due_to_license_issue Kd=12900nM Q86U86 27617704 803 SKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAIFLRLPSRSELPDYYLTIKKPMDMEKIRSHMMANKYQDIDSMVEDFVMMFNNACTYNEPESLIYKDALVLHKVLLETRRDLEGD 5iis A 2.1 BS01 6CB A 1 L44 F49 V52 A65 K67 I104 L120 E121 V126 D128 E171 L174 I185 D186 L13 F18 V21 A34 K36 I73 L89 E90 V95 D97 E140 L143 I154 D155 D167 K169 N172 D186 L193 T204 D136 K138 N141 D155 L162 T173 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Ki<0.001uM remove_due_to_license_issue Ki=<1nM P11309 26995528 402 EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5ij7 A 2.62 BS01 6BN A 1 I109 Y111 G623 W624 Y658 Y661 C663 F665 T678 R685 F686 N688 I93 Y95 G355 W356 Y390 Y393 C395 F397 T410 R417 F418 N420 2.1.1.356 0006338,0042054,0046976 remove_due_to_license_issue G1KPH4,Q15910 27122193 9001 EKGPICWRKRVKSEYMRLRQLKRFRRADEVKSMFNSNRQKIQERTEILNQEWKQRRIQPVHIMTRECSVTSDLDFPKQVIPLKTLNAVASVPIMYSWSPLQQNFMVEDINDEIFVELVNALGQLDRRDEKPSDKIFEAISSMFPDKGTAEELKEKYKECTPNIDGPNAKSVQREQSLHSFHTLFCRRCFKYDCFLHPFHATPNTYKRWSGAEASMFRVLIGTYYDNFCAIARLIGTKTCRQVYEFRVKVYNYQPCDHPRQPCDNSCPCVIAQNFCEKFCQCSSECQNRFPGCRCKAQCNTKQCPCYLAVRECDPDLCLTCGAADHWDSKNVSCKNCSIQRGSKKHLLLAPSDVAGWGIFIKDPVQKNEFISEYCGEIISQDEADRRGKVYDKYMCSFLFNLNNDFVVDATRKGNKIRFANHSVNPNCYAKVMMVNGDHRIGIFAKRAIQTGEELFFDYRYSQADA 5ij7 E 2.62 BS01 6BN A 1 R222 D223 R156 D157 ? remove_due_to_license_issue O75530 27122193 9001 SFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5ijr A 1.52 BS01 HRG A 1 W301 T316 D320 S346 E348 Y353 G414 I415 W28 T43 D47 S73 E75 Y80 G141 I142 ? remove_due_to_license_issue O14786 29430837 501 KCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 5ikb A 2.05 BS01 KAI A 1 Y61 G88 T90 R95 I137 G140 S141 S142 E190 Y57 G84 T86 R91 I133 G136 S137 S138 E186 ? 0015276,0016020 Kd=1.9nM remove_due_to_license_issue Ki=4.7nM Q01812 27524200 301 TLVVTTILENPYLMLKGNHQDMEGNDRYEGFCVDMLKELAEILRFNYKIRLVGDGVYGVPEANGTWTGMVGELIARKADLAVAGLTITAEREKVIDFSKPFMTLGISILYRKGTPIESVDDLADQTAIEYGTIHGGSSMTFFQNSRYQTYQRMWNYMYSKQPSVFVKSTEEGIARVLNSNYAFLLESTMNEYYRQRNCNLTQIGGLLDTKGYGIGMPVGSVFRDEFDLAILQLQENNRLEILKRKWWEG 5il1 A 1.71 BS01 SAM A 1 D377 I378 D395 S511 K513 F534 R536 H538 N539 N549 Q550 D9 I10 D27 S143 K145 F166 R168 H170 N171 N181 Q182 2.1.1.348 0001510,0001734,0005634 Kd=1.5uM remove_due_to_license_issue Q86U44 27281194 601 FPPQWICCDIRYLDVSILGKFAVVMADPPWDIHMELPYGTLTDDEMRRLNIPVLQDDGFLFLWVTGRAMELGRECLNLWGYERVDEIIWVKTNQLQRIIRTGRTGHWLNHGKEHCLVGVKGNPQGFNQGLDCDVIVAEVRSTSHKPDEIYGMIERLSPGTRKIELFGRPHNVQPNWITLGNQLDGIHLLDPDVVARFKQRYP 5im3 A 2.298 BS01 DTP A 1 V34 K36 Y44 T45 K48 I98 I101 Q102 V3 K5 Y13 T14 K17 I67 I70 Q71 C373 N585 C587 E589 C602 Y904 Y905 C342 N547 C549 E551 C564 Y866 Y867 1.17.4.1 0004748,0005524,0005971,0009263,0016491 Kd~1.5uM remove_due_to_license_issue Q9I4I1 27133024 1001 LRVIKRNGTVVPYTDDKITVAITKAFLAVEGGTAAASSRIHDTVRRLTEQVTATFKRRMPSGGTIHIEEIQDQVELALMRAGEQKVARDYVIYREARAAERKNAGAASDVAQPHPSIRITRADGSLSPLDMGRLNTIISEACEGLAEVDGALIERETLKNLYDGVAEKDVNTALVMTARTLVEREPNYSYVTARLLMDTLRAEALGFLGVAESATHHEMAELYAKALPAYIEKGAEFELVDAKLKEFDLEKLGKAIDHERDQQFTYLGLQTLYDRYFIHKDGIRFELPQIFFMRVAMGLAIEEKDREARAIEFYNLLSSFDYMSSTPTLFNAGTLRPQLSSCYLTTVPDDLSGIYGAIHDNAMLSKFAGGLGNDWTPVRALGSYIKGTNGKSQGVVPFLKVVNDTAVAVNAVCAYLETWHLDIEEFLELRKNTGDDRRRTHDMNTANWIPDLFMKRVFDDGSWTLFSPSDVPDLHDLYGKAFEERYEYYEALASYGKLKLHKVVQAKDLWRKMLSMLFETGHPWLTFKDPCNLRSPQQHVGVVHSSNLCTEITLNTNKDEIAVCNLGSINLVNHIVDGKLDTAKLEKTVKTAVRMLDNVIDINYYSVPQAQNSNFKHRPVGLGIMGFQDALYLQHIPYGSDAAIAFADQSMEAISYYAIQASCDLADERGAYQTFQGSLWSQGILPIDSEKKLIEERGAKYIEVDLSETLDWAPLRERVQKGIRNSNIMAIAPTATIANITGVSQSIEPTYQNLYVKSNLSGEFTVINPYLVRDLKARGLWDPVMVNDLKYYDGSVQQIERIPQDLKDLYATAFEVETRWIVEAASRRQKWIDQAQSLNLYIAGASGKKLDVTYRMAWFRGLKTTYYLRALAAT 5im3 A 2.298 BS02 DTP A 2 A52 K55 A59 Q102 D120 Y121 Y124 A21 K24 A28 Q71 D89 Y90 Y93 C373 N585 C587 E589 C602 Y904 Y905 C342 N547 C549 E551 C564 Y866 Y867 1.17.4.1 0004748,0005524,0005971,0009263,0016491 Kd~1.5uM remove_due_to_license_issue Q9I4I1 27133024 1002 LRVIKRNGTVVPYTDDKITVAITKAFLAVEGGTAAASSRIHDTVRRLTEQVTATFKRRMPSGGTIHIEEIQDQVELALMRAGEQKVARDYVIYREARAAERKNAGAASDVAQPHPSIRITRADGSLSPLDMGRLNTIISEACEGLAEVDGALIERETLKNLYDGVAEKDVNTALVMTARTLVEREPNYSYVTARLLMDTLRAEALGFLGVAESATHHEMAELYAKALPAYIEKGAEFELVDAKLKEFDLEKLGKAIDHERDQQFTYLGLQTLYDRYFIHKDGIRFELPQIFFMRVAMGLAIEEKDREARAIEFYNLLSSFDYMSSTPTLFNAGTLRPQLSSCYLTTVPDDLSGIYGAIHDNAMLSKFAGGLGNDWTPVRALGSYIKGTNGKSQGVVPFLKVVNDTAVAVNAVCAYLETWHLDIEEFLELRKNTGDDRRRTHDMNTANWIPDLFMKRVFDDGSWTLFSPSDVPDLHDLYGKAFEERYEYYEALASYGKLKLHKVVQAKDLWRKMLSMLFETGHPWLTFKDPCNLRSPQQHVGVVHSSNLCTEITLNTNKDEIAVCNLGSINLVNHIVDGKLDTAKLEKTVKTAVRMLDNVIDINYYSVPQAQNSNFKHRPVGLGIMGFQDALYLQHIPYGSDAAIAFADQSMEAISYYAIQASCDLADERGAYQTFQGSLWSQGILPIDSEKKLIEERGAKYIEVDLSETLDWAPLRERVQKGIRNSNIMAIAPTATIANITGVSQSIEPTYQNLYVKSNLSGEFTVINPYLVRDLKARGLWDPVMVNDLKYYDGSVQQIERIPQDLKDLYATAFEVETRWIVEAASRRQKWIDQAQSLNLYIAGASGKKLDVTYRMAWFRGLKTTYYLRALAAT 5im3 A 2.298 BS03 DTP A 3 K397 A439 V440 K366 A408 V409 C373 N585 C587 E589 C602 Y904 Y905 C342 N547 C549 E551 C564 Y866 Y867 1.17.4.1 0004748,0005524,0005971,0009263,0016491 Kd~1.5uM remove_due_to_license_issue Q9I4I1 27133024 1004 LRVIKRNGTVVPYTDDKITVAITKAFLAVEGGTAAASSRIHDTVRRLTEQVTATFKRRMPSGGTIHIEEIQDQVELALMRAGEQKVARDYVIYREARAAERKNAGAASDVAQPHPSIRITRADGSLSPLDMGRLNTIISEACEGLAEVDGALIERETLKNLYDGVAEKDVNTALVMTARTLVEREPNYSYVTARLLMDTLRAEALGFLGVAESATHHEMAELYAKALPAYIEKGAEFELVDAKLKEFDLEKLGKAIDHERDQQFTYLGLQTLYDRYFIHKDGIRFELPQIFFMRVAMGLAIEEKDREARAIEFYNLLSSFDYMSSTPTLFNAGTLRPQLSSCYLTTVPDDLSGIYGAIHDNAMLSKFAGGLGNDWTPVRALGSYIKGTNGKSQGVVPFLKVVNDTAVAVNAVCAYLETWHLDIEEFLELRKNTGDDRRRTHDMNTANWIPDLFMKRVFDDGSWTLFSPSDVPDLHDLYGKAFEERYEYYEALASYGKLKLHKVVQAKDLWRKMLSMLFETGHPWLTFKDPCNLRSPQQHVGVVHSSNLCTEITLNTNKDEIAVCNLGSINLVNHIVDGKLDTAKLEKTVKTAVRMLDNVIDINYYSVPQAQNSNFKHRPVGLGIMGFQDALYLQHIPYGSDAAIAFADQSMEAISYYAIQASCDLADERGAYQTFQGSLWSQGILPIDSEKKLIEERGAKYIEVDLSETLDWAPLRERVQKGIRNSNIMAIAPTATIANITGVSQSIEPTYQNLYVKSNLSGEFTVINPYLVRDLKARGLWDPVMVNDLKYYDGSVQQIERIPQDLKDLYATAFEVETRWIVEAASRRQKWIDQAQSLNLYIAGASGKKLDVTYRMAWFRGLKTTYYLRALAAT 5im3 A 2.298 BS04 DTP A 4 D380 D381 L382 I385 R410 I416 D349 D350 L351 I354 R379 I385 C373 N585 C587 E589 C602 Y904 Y905 C342 N547 C549 E551 C564 Y866 Y867 1.17.4.1 0004748,0005524,0005971,0009263,0016491 Kd~1.5uM remove_due_to_license_issue Q9I4I1 27133024 1005 LRVIKRNGTVVPYTDDKITVAITKAFLAVEGGTAAASSRIHDTVRRLTEQVTATFKRRMPSGGTIHIEEIQDQVELALMRAGEQKVARDYVIYREARAAERKNAGAASDVAQPHPSIRITRADGSLSPLDMGRLNTIISEACEGLAEVDGALIERETLKNLYDGVAEKDVNTALVMTARTLVEREPNYSYVTARLLMDTLRAEALGFLGVAESATHHEMAELYAKALPAYIEKGAEFELVDAKLKEFDLEKLGKAIDHERDQQFTYLGLQTLYDRYFIHKDGIRFELPQIFFMRVAMGLAIEEKDREARAIEFYNLLSSFDYMSSTPTLFNAGTLRPQLSSCYLTTVPDDLSGIYGAIHDNAMLSKFAGGLGNDWTPVRALGSYIKGTNGKSQGVVPFLKVVNDTAVAVNAVCAYLETWHLDIEEFLELRKNTGDDRRRTHDMNTANWIPDLFMKRVFDDGSWTLFSPSDVPDLHDLYGKAFEERYEYYEALASYGKLKLHKVVQAKDLWRKMLSMLFETGHPWLTFKDPCNLRSPQQHVGVVHSSNLCTEITLNTNKDEIAVCNLGSINLVNHIVDGKLDTAKLEKTVKTAVRMLDNVIDINYYSVPQAQNSNFKHRPVGLGIMGFQDALYLQHIPYGSDAAIAFADQSMEAISYYAIQASCDLADERGAYQTFQGSLWSQGILPIDSEKKLIEERGAKYIEVDLSETLDWAPLRERVQKGIRNSNIMAIAPTATIANITGVSQSIEPTYQNLYVKSNLSGEFTVINPYLVRDLKARGLWDPVMVNDLKYYDGSVQQIERIPQDLKDLYATAFEVETRWIVEAASRRQKWIDQAQSLNLYIAGASGKKLDVTYRMAWFRGLKTTYYLRALAAT 5ime A 2.217 BS01 6BZ A 1 A297 K299 M301 E315 V342 M344 Y346 L347 L396 D407 A36 K38 M40 E49 V76 M78 Y80 L81 L130 D141 N389 K391 D393 N394 D407 P416 T427 N123 K125 D127 N128 D141 P150 T161 2.7.11.1 0004672,0005524,0006468 Ki=4.6nM remove_due_to_license_issue Ki=4.6nM Q13153 27167326 601 EEILEKLRSIVSVGDPKKIGQGASGTVYTAMDQEVAIKQMNLKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATKNNHG 5in9 A 2.6 BS01 6C0 A 1 N107 D149 M154 N162 K168 F199 T245 I247 N34 D76 M81 N89 K95 F121 T167 I169 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P41148 27003516 410 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTEASTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKKTVWDWELMN 5inh A 1.84 BS06 6C1 A 1 D171 T209 N230 D311 F312 H359 H474 D119 T157 N178 D259 F260 H307 H422 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 remove_due_to_license_issue Q9R1E6 28564542 914 NTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPLDVYKKPSGKCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMGCTCDGSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5ioy A 1.77 BS01 6C5 A 1 F110 W145 N176 N179 W207 F89 W124 N155 N158 W186 ? 0000976,0003677,0003700,0006355,0045892 Kd=6uM remove_due_to_license_issue A5U9I4 28314097 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ioy A 1.77 BS02 6C5 A 2 F114 R128 W138 E180 F184 F93 R107 W117 E159 F163 ? 0000976,0003677,0003700,0006355,0045892 Kd=6uM remove_due_to_license_issue A5U9I4 28314097 302 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ioy A 1.77 BS03 6C5 A 3 L87 M102 W103 Y148 V152 E156 L66 M81 W82 Y127 V131 E135 ? 0000976,0003677,0003700,0006355,0045892 Kd=6uM remove_due_to_license_issue A5U9I4 28314097 304 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ioz A 2.02 BS01 6C4 A 1 F110 W145 T149 N176 N179 E180 W207 F89 W124 T128 N155 N158 E159 W186 ? 0000976,0003677,0003700,0006355,0045892 Kd=11uM remove_due_to_license_issue A5U9I4 28314097 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ipa A 1.78 BS01 6C8 A 1 F114 R128 W138 E180 L183 F93 R107 W117 E159 L162 ? 0000976,0003677,0003700,0006355,0045892 Kd=20uM remove_due_to_license_issue A5U9I4 28314097 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ipa A 1.78 BS02 6C8 A 2 I107 F110 T149 N176 N179 E180 W207 I86 F89 T128 N155 N158 E159 W186 ? 0000976,0003677,0003700,0006355,0045892 Kd=20uM remove_due_to_license_issue A5U9I4 28314097 302 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ipa A 1.78 BS03 6C8 A 3 I107 F110 W138 M142 W145 T149 N176 N179 E180 W207 I86 F89 W117 M121 W124 T128 N155 N158 E159 W186 ? 0000976,0003677,0003700,0006355,0045892 Kd=20uM remove_due_to_license_issue A5U9I4 28314097 303 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5ipc A 1.3 BS01 6CE A 1 I18 F41 D43 I44 L53 N99 G105 Q106 S107 V108 N112 H114 I7 F30 D32 I33 L42 N88 G94 Q95 S96 V97 N101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=13uM remove_due_to_license_issue P49773 28691797 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVNLHVLGGRQMHWPPG 5ipj A 2.1 BS01 6CD A 1 F49 A65 K67 L174 I185 D186 F17 A33 K35 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Kd=1.3nM remove_due_to_license_issue IC50=0.300000nM, Kd=1.3nM P11309 27285051 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5irr A 2.04 BS02 GSP A 1 S119 G120 G122 K123 T124 T125 H141 Y145 T146 G182 K263 D265 A324 R344 S15 G16 G18 K19 T20 T21 H37 Y41 T42 G78 K151 D153 A212 R232 ? 0005525 Kd=5.4uM remove_due_to_license_issue A8IYS5 28476887 402 IWKKKYIKLIVVGDSGLGKTTLIKSLISIPGERLQVHDGSYTPTEQFRRDPESLSSTVSWRDEEDRVIWVYKIQDTPGYGDELDVFRNLKMVQDYIESQNRKWLELEQARIEDPRVDLCIFCIPPHRLRPIDLKYMFELGKHVPVVPVVTKADTMTIREANTYRTEVANRIANPMVPGIHDKINIFKFERDTLERAGVQDHATPHPPFLVIASNDISEELAAAEPPLFWPERRYPWGTAEAFNKEHSDLLAVRALLMKEALEEISKTKRARYEAWRRT 5irr A 2.04 BS03 GSP B 1 H238 R239 T266 E271 H126 R127 T154 E159 ? 0005525 Kd=5.4uM remove_due_to_license_issue A8IYS5 28476887 402 IWKKKYIKLIVVGDSGLGKTTLIKSLISIPGERLQVHDGSYTPTEQFRRDPESLSSTVSWRDEEDRVIWVYKIQDTPGYGDELDVFRNLKMVQDYIESQNRKWLELEQARIEDPRVDLCIFCIPPHRLRPIDLKYMFELGKHVPVVPVVTKADTMTIREANTYRTEVANRIANPMVPGIHDKINIFKFERDTLERAGVQDHATPHPPFLVIASNDISEELAAAEPPLFWPERRYPWGTAEAFNKEHSDLLAVRALLMKEALEEISKTKRARYEAWRRT 5isl A 1.694 BS01 MMK A 1 Y409 W470 Y472 F480 H483 E485 K501 W503 H571 V584 N585 Y136 W188 Y190 F198 H201 E203 K219 W221 H289 V302 N303 Y472 H483 E485 H571 A583 Y190 H201 E203 H289 A301 1.14.11.67 Kd=0.052uM remove_due_to_license_issue P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5ism A 2.0 BS01 6DG A 1 E205 E206 F357 Y547 S630 Y662 Y666 N710 V711 E167 E168 F319 Y509 S592 Y624 Y628 N672 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.7nM remove_due_to_license_issue IC50=0.700000nM P27487 27106708 811 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5itd A 3.02 BS01 6CY A 1 I800 K802 I848 E849 V851 Q859 M922 I932 I744 K746 I792 E793 V795 Q803 M858 I868 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue IC50=262nM P42336 27563400 1101 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRISTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTTKMDWIF 5ith A 2.31 BS01 dna B 0 F98 D101 R125 K136 Y138 F140 R167 N169 A171 F7 D10 R34 K45 Y47 F49 R76 N78 A80 ? 0003676,0003723 remove_due_to_license_issue P31483 28184449 1 ~ 3 GNHFHVFVGDLSPEITTEDIKAAFAPFGRISDARVVKDMATGKSKGYGFVSFFNKWDAENAIQQMGGQWLGGRQIRTNWA 5ito A 2.35 BS01 6DB A 1 E36 Y39 W77 A94 A95 G97 R102 Q165 T168 S169 H170 S207 E10 Y13 W51 A68 A69 G71 R76 Q139 T142 S143 H144 S181 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=68.9uM remove_due_to_license_issue P35120 27801902 304 DYKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPNTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASP 5itp A 1.85 BS01 6DB A 1 E36 Y39 Y42 W77 A94 A95 G97 R102 M117 Q165 T168 H170 S207 E9 Y12 Y15 W50 A67 A68 G70 R75 M90 Q138 T141 H143 S180 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=9.9uM remove_due_to_license_issue P35120 27801902 301 YKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPMTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASP 5iu2 A 2.7 BS01 6DA A 1 W132 L134 F149 V152 A165 K167 M207 A209 G210 G213 E217 S257 V260 V269 D270 W56 L58 F72 V75 A88 K90 M130 A132 G133 G136 E140 S180 V183 V192 D193 D253 K255 N258 D270 T290 D176 K178 N181 D193 T213 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=16nM P41279 27502541 401 LSSVRYGTVEDLLAFANHISNFYGQRPQESGILLNMVITPQNGRYQIDSDVLLIPWKLTYRNGSDFIPRGAFGKVYLAQDIKTKKRMACKLIPVDQFKPSDVEIQACFRHENIAELYGAVLWGETVHLFMEAGEGGSVLEKLESCGPMREFEIIWVTKHVLKGLDFLHSKKVIHHDIKPSNIVFMSTKAVLVDFGLSVQMTEDVYFPKDLRGTEIYMSPEVILCRGHSTKADIYSLGATLIHMQTGTPPWVKRYPRSAYPSYLYIIHKQAPPLEDIADDCSPGMRELIEASLERNPNHRPRAADLLKHEALN 5iu4 A 1.72 BS01 ZMA A 1 L85 F168 E169 M177 L249 H250 N253 M270 L87 F170 E171 M179 L332 H333 N336 M353 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 Ki=0.53nM remove_due_to_license_issue P0ABE7,P29274 27312113 2401 GAPPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 5iu6 A 2.51 BS01 7HX A 1 C91 G92 F159 V178 E179 C91 G92 F159 V178 E179 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0006974,0009116,0009164,0016020,0016757,0016763,0019686,0042278,0042802,0047975 remove_due_to_license_issue P0ABP8 29870020 301 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHIRTHEQTTAAERQTTFNDMIKIALESVLLGDK 5iu6 B 2.51 BS01 7HX B 1 G92 F159 V178 I206 G92 F159 V178 I206 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 H4 G20 R24 R43 E75 R87 S90 S203 D204 I206 R217 2.4.2.1 0003824,0004731,0005737,0005829,0006139,0006152,0006974,0009116,0009164,0016020,0016757,0016763,0019686,0042278,0042802,0047975 remove_due_to_license_issue P0ABP8 29870020 301 ATPHINAEMGDFADVVLMPGDPLRAKYIAETFLEDAREVNNVRGMLGFTGTYKGRKISVMGHGMGIPSCSIYTKELITDFGVKKIIRVGSCGAVLPHVKLRDVVIGMGACTDSKVNRIRFKDHDFAAIADFDMVRNAVDAAKALGIDARVGNLFSADLFYSPDGEMFDVMEKYGILGVEMEAAGIYGVAAEFGAKALTICTVSDHIRTHEQTTAAERQTTFNDMIKIALESVLLGDK 5iu7 A 1.9 BS01 6DY A 1 L85 F168 E169 M177 L249 H250 N253 H264 L267 M270 L89 F172 E173 M181 L334 H335 N338 H349 L352 M355 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 Ki=1.1nM remove_due_to_license_issue P0ABE7,P29274 27312113 2401 DDGAPPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRSHV 5iu8 A 2.002 BS01 6DZ A 1 L85 F168 E169 M177 L249 H250 N253 L267 M270 L87 F170 E171 M179 L331 H332 N335 L349 M352 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 Ki=18nM remove_due_to_license_issue P0ABE7,P29274 27312113 2401 GAPPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 5iua A 2.2 BS01 6DX A 1 L85 F168 E169 M177 L249 H250 N253 H264 L267 M270 I274 L87 F170 E171 M179 L331 H332 N335 H346 L349 M352 I356 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 Ki=1.5nM remove_due_to_license_issue P0ABE7,P29274 27312113 2401 GAPPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRSH 5iub A 2.1 BS01 6DV A 1 L85 F168 E169 M177 W246 L249 H250 N253 H264 A265 L267 I274 L87 F170 E171 M179 W329 L332 H333 N336 H347 A348 L350 I357 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 Ki=0.35nM remove_due_to_license_issue P0ABE7,P29274 27312113 2401 GAPPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADILVGVLAIPFAITISTGFCAACHGCLFIACFVLVLAQSSIFSLLAIAIDRYIAIAIPLRYNGLVTGTRAAGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFAAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSAAIIAGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLAHTNSVVNPFIYAYRIREFRQTFRKIIRS 5iug A 1.93 BS01 729 A 1 A1148 E1167 I1171 F1174 L1196 E1197 M1199 A1200 G1201 G1202 H1247 L1256 G1269 D1270 F1271 A45 E64 I68 F71 L93 E94 M96 A97 G98 G99 H140 L149 G162 D163 F164 D1249 A1251 R1253 N1254 D1270 D142 A144 R146 N147 D163 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=177nM remove_due_to_license_issue IC50=177nM, Kd=2.4nM Q9UM73 27031565 1501 NPNYSFAGKTSSISDLKEVPRKNITLIRGLGGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMAGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYGPL 5iuh A 2.1 BS01 34Y A 1 E1167 I1171 F1174 V1180 L1196 E1197 M1199 A1200 G1201 G1202 F1245 H1247 L1256 G1269 D1270 E64 I68 F71 V77 L93 E94 M96 A97 G98 G99 F139 H141 L150 G163 D164 D1249 A1251 R1253 N1254 D1270 D143 A145 R147 N148 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=402nM remove_due_to_license_issue IC50=402nM Q9UM73 27031565 1501 NPNYSFAGKTSSISDLKEVPRKNITLIRGLGEVYEGQVSGPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMACAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEYGPL 5iui A 1.88 BS01 45Q A 1 L1122 F1127 A1148 V1180 L1196 E1197 M1199 A1200 G1201 G1202 L1256 G1269 L34 F39 A56 V88 L104 E105 M107 A108 G109 G110 L164 G177 D1249 A1251 R1253 N1254 D1270 R1279 D157 A159 R161 N162 D178 R187 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=>10000nM Q9UM73 27031565 1501 MTDYNPNYSFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSGPSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRAGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 5iv4 A 1.79 BS01 LRI A 1 F45 K95 L102 L166 V167 V172 R176 F336 M337 F39 K89 L96 L160 V161 V166 R170 F330 M331 4.6.1.1 0009190,0035556 remove_due_to_license_issue IC50=3300nM Q96PN6 27547922 501 EFQDWPIVRIAAHLPDLIVYGHFSPERPFMDYFDGVLMFVDISGFTAMTEKFSSAMYMDRGAEQLVEILNYHISAIVEKVLIFGGDILKFAGDALLALWRVERKQLKNIITVVIKCSLEIHGLFETQEWEEGLDIRVKIGLAAGHISMLVFGDETHSHFLVIGQAVDDVRLAQNMAQMNDVILSPNCWQLCDRSMIEIESVPDQRAVKVNFLKPPPNFNFDEFFTKCTTFMHYYPSGEHKNLLRLACTLKPDPELEMSLQKYVMESILKQIDNKQLQGYLSELRPVTIVFVNLMFEDQDKAEEIGPAIQDAYMHITSVLKIFQGQINKVFMFDKGCSFLCVFGFPGEKVDELTHALECAMDIFDFCSQVHKIQTVSIGVASGIVFCGIVGHTVRHEYTVIGQKVNLAARMMMYYPGIVTCDSVTYNGSNLPAYFFKELPKKVMKGVADSGPLYQYWGRTEK 5ivc A 1.573 BS01 6E7 A 1 R73 Y409 A411 F480 H483 E485 K501 W503 H571 R62 Y135 A137 F200 H203 E205 K221 W223 H291 Y472 H483 E485 H571 A583 Y192 H203 E205 H291 A303 1.14.11.67 Kd=1.2uM remove_due_to_license_issue P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMRPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5ive A 1.783 BS01 6E8 A 1 Y409 Y472 F480 H483 K501 Y136 Y189 F197 H200 K218 Y472 H483 E485 H571 A583 Y189 H200 E202 H288 A300 1.14.11.67 Kd=0.027uM remove_due_to_license_issue IC50=9.3nM P29375 27427228 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5ivf A 1.683 BS01 6EB A 1 R73 Q75 Y409 A411 Y472 F480 H483 E485 K501 W503 H571 R62 Q64 Y135 A137 Y192 F200 H203 E205 K221 W223 H291 Y472 H483 E485 H571 A583 Y192 H203 E205 H291 A303 1.14.11.67 remove_due_to_license_issue IC50=<100nM P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMRPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5ivj A 1.569 BS01 6ED A 1 R73 Y409 A411 D412 Y472 F480 H483 K501 W503 H571 R62 Y129 A131 D132 Y180 F188 H191 K209 W211 H279 Y472 H483 E485 H571 A583 Y180 H191 E193 H279 A291 1.14.11.67 Kd=0.046uM remove_due_to_license_issue IC50=<100nM P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5ivs A 1.46 BS01 6EF B 1 D25 G27 D29 D30 V32 G48 G49 I50 D25 G27 D29 D30 V32 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q77VV3 27437081 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5ivs B 1.46 BS01 6EF B 1 R8 L23 D25 A28 D30 V32 G48 I50 P81 V82 I84 R8 L23 D25 A28 D30 V32 G48 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=6.1nM remove_due_to_license_issue Q77VV3 27437081 101 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5ivt A 1.15 BS01 6EE A 1 D25 G27 A28 D29 D30 G48 G49 I50 V82 I84 D25 G27 A28 D29 D30 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.8nM remove_due_to_license_issue G0X8E8 27437081 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5ivt A 1.15 BS02 6EE B 1 R8 D25 G27 G48 I50 V82 R8 D25 G27 G48 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.8nM remove_due_to_license_issue G0X8E8 27437081 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5ivt B 1.15 BS01 6EE A 1 R8 D25 G27 G48 I50 P81 V82 I84 R8 D25 G27 G48 I50 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.8nM remove_due_to_license_issue G0X8E8 27437081 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5ivt B 1.15 BS02 6EE B 1 R8 D25 G27 A28 D29 D30 G48 G49 I50 V82 R8 D25 G27 A28 D29 D30 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.8nM remove_due_to_license_issue G0X8E8 27437081 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5ivv A 1.848 BS01 6EN A 1 R73 Y409 A411 D412 Y472 F480 H483 K501 W503 H571 R62 Y131 A133 D134 Y184 F192 H195 K213 W215 H283 Y472 H483 E485 H571 A583 Y184 H195 E197 H283 A295 1.14.11.67 Kd=0.45uM remove_due_to_license_issue IC50=<100nM P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5ivy A 1.45 BS01 6EO A 1 Y409 Y472 F480 H483 K501 W503 H571 Y127 Y184 F192 H195 K213 W215 H283 Y472 H483 E485 H571 A583 Y184 H195 E197 H283 A295 1.14.11.67 Kd=0.36uM remove_due_to_license_issue P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5iw0 A 1.63 BS01 6EP A 1 R73 Q75 Y409 A411 Y472 F480 H483 E485 K501 W503 H571 R62 Q64 Y133 A135 Y190 F198 H201 E203 K219 W221 H289 Y472 H483 E485 H571 A583 Y190 H201 E203 H289 A301 1.14.11.67 Kd=0.06uM remove_due_to_license_issue IC50=<100nM, EC50=90nM P29375 27427228 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 5iwg A 1.66 BS03 IWX A 1 M35 R39 F114 L144 H145 H146 G154 F155 C156 D181 H183 L276 G305 G306 Y308 M24 R28 F103 L133 H134 H135 G143 F144 C145 D170 H172 L265 G294 G295 Y297 3.5.1.-,3.5.1.98 0004407 Ki=0.346uM remove_due_to_license_issue IC50=62nM Q92769 27377864 403 GKKKVCYYYDGDIGNYYYGQGHPMKPHRIRMTHNLLLNYGLYRKMEIYRPHKATAEEMTKYHSDEYIKFLRSIRPDNMSEYSKQMQRFNVGEDCPVFDGLFEFCQLSTGGSVAGAVKLNRQQTDMAVNWAGGLHHAKKSEASGFCYVNDIVLAILELLKYHQRVLYIDIDIHHGDGVEEAFYTTDRVMTVSFHKYGEYFPGTGDLRDIGAGKGKYYAVNFPMRDGIDDESYGQIFKPIISKVMEMYQPSAVVLQCGADSLSGDRLGCFNLTVKGHAKCVEVVKTFNLPLLMLGGGGYTIRNVARCWTYETAVALDCEIPNELPYNDYFEYFGPDFKLHISPSNMTNQNTPEYMEKIKQRLFENLRMLP 5ix0 A 1.72 BS04 6EZ A 1 M35 R39 F114 L144 H145 H146 G154 F155 C156 D181 H183 F210 G305 G306 Y308 M25 R29 F104 L134 H135 H136 G144 F145 C146 D171 H173 F200 G295 G296 Y298 3.5.1.-,3.5.1.98 0004407 Ki=0.519uM remove_due_to_license_issue IC50=168nM, Ki=519nM Q92769 27377864 404 GGKKKVCYYYDGDIGNYYYGQGHPMKPHRIRMTHNLLLNYGLYRKMEIYRPHKATAEEMTKYHSDEYIKFLRSIRPDNMSEYSKQMQRFNVGEDCPVFDGLFEFCQLSTGGSVAGAVKLNRQQTDMAVNWAGGLHHAKKSEASGFCYVNDIVLAILELLKYHQRVLYIDIDIHHGDGVEEAFYTTDRVMTVSFHKYGEYFPGTGDLRDIGAGKGKYYAVNFPMRDGIDDESYGQIFKPIISKVMEMYQPSAVVLQCGADSLSGDRLGCFNLTVKGHAKCVEVVKTFNLPLLMLGGGGYTIRNVARCWTYETAVALDCEIPNELPYNDYFEYFGPDFKLHISPSNMTNQNTPEYMEKIKQRLFENLRMLP 5iyy A 1.6 BS01 R40 A 1 Y297 W301 T316 D320 S346 T349 Y353 G414 I415 Y26 W30 T45 D49 S75 T78 Y82 G143 I144 ? remove_due_to_license_issue O14786 29430837 501 MFKCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 5izc A 1.92 BS02 6F4 A 1 S95 F97 C168 Y174 V206 L209 P210 S94 F96 C149 Y155 V187 L190 P191 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0000166,0016491,0047040 remove_due_to_license_issue O76290 28983525 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5izj A 1.85 BS02 6J9 A 1 F18 F100 L152 Y306 F5 F87 L139 Y293 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 27389935 414 SVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFNFDDYEEEEIRVSINEKCGKEFSEF 5izk A 3.25 BS01 GDP A 1 G19 K20 T21 A22 D149 K187 G18 K19 T20 A21 D108 K146 D17 K20 T21 H96 D16 K19 T20 H55 3.6.5.- 0000049,0001514,0003746,0003924,0005525,0005634,0005737,0006412,0016787,0035368,0043021,1990904 remove_due_to_license_issue P57772 27708257 1001 AGRRVNVNVGVLGHIDSGKTALARALSTTASTGFSCFSVPLPALLQVTLVDCPGHASLIRTIIGGAQIIDLMMLVIDVTKGMQTQSAECLVIGQIACQKLVVVLNKIDLLPEGKRQAAIDKMTKKMQKTLENTKFRGAPIIPVAAKPGGPEAPQGIPELIELLTSQISIPTRDPSGPFLMSVDHCTVMTGTILSGSISLGDSVEIPALKVVKKVKSMQMFHMPITSAMQGDRLGICVTQFDPKLLERGLVCAPESLHTVHAALISVEKIPYFRGPLQTKAKFHITVGHETVMGRLMFFSPAPDNFDQEPILDSFNFSQEYLFQEQYLSKHCPRQQWALVEFEKPVTCPRLCLVIGSRLDATCRLAFHGILLHGLEDRNYADSFLPRLKVYKLKHKHGLVERAMDDYSVIGRSLFTNIQLFVGLKVHLSTGELGIIDGKFKIHIPGLSPESKKISAERSEPSQHVVLSLTFKRYVFDTHKR 5izm A 3.4 BS02 GNP A 1 D17 G19 K20 T21 A22 T48 N146 K147 D149 L150 A185 A186 K187 D15 G17 K18 T19 A20 T31 N113 K114 D116 L117 A152 A153 K154 D17 K20 T21 T48 H96 D15 K18 T19 T31 H63 3.6.5.- 0000049,0001514,0003746,0003924,0005525,0005634,0005737,0006412,0016787,0035368,0043021,1990904 remove_due_to_license_issue P57772 27708257 1002 GRRVNVNVGVLGHIDSGKTALARALSTTAITLDLGFSCFSVPLPARLRSSPLLQVTLVDCPGHASLIRTIIGGAQIIDLMMLVIDVTKGMQTQSAECLVIGQIACQKLVVVLNKIDLLPEGKRQAAIDKMTKKMQKTLENTKFRGAPIIPVAAKPGGAPQGIPELIELLTSQISIPTRDPSGPFLMSVDHCFSIGTVMTGTILSGSISLGDSVEIPALKVVKKVKSMQMFHMPITSAMQGDRLGICVTQFDPKLLERGLVCAPESLHTVHAALISVEKIPYFRGPLQTKAKFHITVGHETVMGRLMFFSPAPDNFDQEPILDSFNFSQEYLFQEQYLSPRQQWALVEFEKPVTCPRLCLVIGSRLDADIHTNTCRLAFHGILLHGLEDRNYADSFLPRLKVYKLKHKDDYSVQLFVGLKVHLSTGELGIIDSFKIHIPGGLLSLTFKRYVFDTHKRMVQS 5izq A 3.6 BS01 83A A 1 D81 Y85 W102 W134 H135 K136 G137 W138 W140 W171 S174 Y175 D74 Y78 W95 W127 H128 K129 G130 W131 W133 W164 S167 Y168 ? remove_due_to_license_issue IC50=3.0nM P15328 27458733 300 RTELLNVCMNAKHHKEKPGPEDKLHEQCRPWRKNACCSTNTSQEAHKDVSYLYRFNWNHCGEMAPACKRHFIQDTCLYECSPNLGPWIQQVDQSWRKERVLNVPLCKEDCEQWWEDCRTSYTCKSNWHKGWNWTSGFNKCAVGAACQPFHFYFPTPTVLCNEIWTHSYKVSNYSRGSGRCIQMWFDPAQGNPNEEVARFYAAAMSGT 5j0d A 1.05 BS01 6F9 A 1 L1109 P1110 F1111 V1115 N1168 R1173 V1174 F1177 L29 P30 F31 V35 N88 R93 V94 F97 2.3.1.-,2.3.1.48 Kd=134nM remove_due_to_license_issue Kd=134nM Q92793 27673482 1201 RKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5j18 A -1.00 BS01 6FS A 1 K154 I156 R166 T167 V168 M187 K4 I6 R16 T17 V18 M37 2.7.11.1 0007165 remove_due_to_license_issue P15056 27104980 301 SPQKPIVRVFLPNKQRTVVPARCGVTVRDSLKKALMMRGLIPECCAVYRIQDGEKKPIGWDTDISWLTGEELHVEVLENVPL 5j1r A 1.92 BS01 6FG A 1 F110 W138 W145 T149 N176 N179 W207 F89 W117 W124 T128 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=22uM remove_due_to_license_issue Kd=2.2e+4nM P9WMC1 28314097 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5j1v A 2.52 BS01 6FD A 1 L167 V175 A189 K191 F241 L244 L295 L22 V30 A44 K46 F96 L99 L150 D288 K290 N293 D325 T342 D143 K145 N148 D180 T197 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=41nM P49759 27128181 501 SMHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKKS 5j1w A 2.42 BS01 6FB A 1 V175 A189 K191 F241 L244 L295 V30 A44 K46 F96 L99 L150 D288 K290 N293 D325 T342 D143 K145 N148 D180 T197 2.7.12.1 0004672,0005524,0006468 ic50=0.19uM remove_due_to_license_issue IC50=190nM P49759 27128181 506 SMHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKKS 5j1x A 2.1 BS01 AR5 A 1 Y297 W301 T316 D320 S346 T349 Y353 G414 I415 Y25 W29 T44 D48 S74 T77 Y81 G142 I143 ? remove_due_to_license_issue O14786 29430837 501 FKCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 5j20 A 1.76 BS01 6FJ A 1 N51 A55 D93 I96 G97 M98 L103 L107 F138 V150 W162 V186 N36 A40 D78 I81 G82 M83 L88 L92 F123 V135 W147 V171 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 AVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j27 A 1.7 BS01 6FF A 1 N51 A55 K58 D93 I96 G97 M98 L107 F138 V186 N36 A40 K43 D78 I81 G82 M83 L92 F123 V171 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5j2x A 1.22 BS01 6DL A 1 N51 S52 A55 K58 D93 I96 G97 M98 L107 G108 F138 N36 S37 A40 K43 D78 I81 G82 M83 L92 G93 F123 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 AVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5j32 A 1.933 BS02 IPM A 1 R136 R174 Y181 D288 R106 R144 Y151 D258 L48 Y181 K232 D264 D288 D292 L18 Y151 K202 D234 D258 D262 1.1.1.85 0000287,0003862,0005829,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 Kd=8.3uM remove_due_to_license_issue P93832 27137927 502 QMGRGSEFGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSVDS 5j32 B 1.933 BS02 IPM A 2 R136 R146 R174 Y181 D288 R101 R111 R139 Y146 D253 L48 Y181 K232 D264 D288 D292 L13 Y146 K197 D229 D253 D257 1.1.1.85 0000287,0003862,0005829,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 remove_due_to_license_issue P93832 27137927 504 SEFGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSVDSQ 5j3l A 1.66 BS01 6FR A 1 G106 F110 M142 T149 N176 N179 G85 F89 M121 T128 N155 N158 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 Kd=16uM remove_due_to_license_issue Kd=1.6e+4nM P9WMC1 28314097 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5j3s A 3.4 BS01 6FQ A 1 R231 R266 I307 C311 R120 R150 I191 C195 3.1.4.- 0003824 remove_due_to_license_issue IC50=590nM, EC50=40nM O95551 27099339 401 HMFSLITWNIDGLDLNNLSERARGVCSYLALYSPDVIFLQEVIPPYYSYLKKRSSNYEIITGHEEGYFTAIMLKKSRVKLKSQEIIPFPSTKMMRNLLCVHVNVSGNELCLMTSHLESTRGHAAERMNQLKMVLKKMQEAVIFAGDTNLRDREVTRSGGLPNNIVDVWEFLGKPKHCQYTWDTQMNSNLGITAACKLRFDRIFFRIIPRSLDLLGLEKLDCGRFPSDHWGLLCNLD 5j41 A 1.19035 BS01 3LF A 1 F8 R13 I104 Y108 F8 R13 I104 Y108 Y7 R13 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 27872191 301 PPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 5j41 A 1.19035 BS02 GSH A 1 F8 R13 W38 K44 Q51 L52 Q64 S65 F8 R13 W38 K44 Q51 L52 Q64 S65 Y7 R13 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 27872191 302 PPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 5j41 B 1.19035 BS01 3LF B 1 F8 R13 I104 Y108 F7 R12 I103 Y107 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 27872191 301 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 5j41 B 1.19035 BS02 GSH B 1 F8 R13 W38 K44 Q51 L52 Q64 S65 F7 R12 W37 K43 Q50 L51 Q63 S64 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 27872191 302 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 5j47 A 1.99 BS02 6JJ A 1 W394 D430 T435 K551 L554 R555 L558 L565 W129 D165 T170 K283 L286 R287 L290 L297 3.6.4.- 0003677,0005524,0006260 ic50=4.9uM remove_due_to_license_issue IC50=4900nM P03072 27385654 703 TKQVSWKLVTQYALDTKCEDVFLLMGMYLNFQEAPAACAACAAADQPNHFNHHEKHYYNAQIFADSKNQKSICQQAVDTVAAKQRVDSLHMTREEMLVERFNFLLDKMDLIFGAHGNAVLEQYMAGVAWIHCLLPQMDTVIYEFLKCIVLNIPKKRYWLFKGPIDSGKTTLAAALLDLCGGKSLNVNMPLERLNFELGVGIDQFMVVFEDVKGTGAESRDLPSGHGISNLDCLRDYLDGSVKVNLERNKRTQVFPPGIVTMNEYSVPRTLQARFVRQIDFRPKAYLRKSLSCSEYLLEKRILQSGMTLLLLLIWFRPVADFAAAIHERIVQWKERLDLEISMYTFSTMKANVGMGAPILD 5j4n A 2.594 BS01 AG2 A 1 I23 A96 C97 G100 N101 M104 W293 I19 A92 C93 G96 N97 M100 W289 ? 0003333,0005886,0006865,0015297,0015695,0016020,0022857,0043862,0055085,1905039,1990451 remove_due_to_license_issue P60061 27582465 501 ADAHKVGLIPVTLMVSGNIMGSGVFLLPANLASTGGIAIYGWLVTIIGALGLSMVYAKMSFLDPSPGGSYAYARRCFGPFLGYQTNVLYWLACWIGNIAMVVIGVGYLSYFFPILKDPLVLTITCVVVLWIFVLLNIVGPKMITRVQAVATVLALIPIVGIAVFGWFWFRGETYMAAWNVSGLGTFGAIQSTLNVTLWSFIGVESASVAAGVVKNPKRNVPIATIGGVLIAAVCYVLSTTAIMGMIPNAALRVSASPFGDAARMALGDTAGAIVSFCAAAGCLGSLGGWTLLAGQTAKAAADDGLFPPIFARVNKAGTPVAGLIIVGILMTIFQLSSISPNATKEFGLVSSVSVIFTLVPYLYTCAALLLLGHGHFGKARPAYLAVTTIAFLYCIWAVVGSGAKEVMWSFVTLMVITAMYALNYNRLHKNPYPLDAP 5j4v A 2.94 BS02 6JH A 1 W394 L398 D430 S431 G432 P550 K551 L554 R555 L558 L565 W129 L133 D165 S166 G167 P280 K281 L284 R285 L288 L295 3.6.4.- 0003677,0005524,0006260 remove_due_to_license_issue IC50=1400nM P03072 27385654 704 TKQVSWKLVTQYALDTKCEDVFLLMGMYLNFQEAPAACAACAAADQPNHFNHHEKHYYNAQIFADSKNQKSICQQAVDTVAAKQRVDSLHMTREEMLVERFNFLLDKMDLIFGAHGNAVLEQYMAGVAWIHCLLPQMDTVIYEFLKCIVLNIPKKRYWLFKGPIDSGKTTLAAALLDLCGGKSLNVNMPLERLNFELGVGIDQFMVVFEDVKGTGAESRDLPSGHGISNLDCLRDYLDGSVKVNLERRTQVFPPGIVTMNEYSVPRTLQARFVRQIDFRPKAYLRKSLSCSEYLLEKRILQSGMTLLLLLIWFRPVADFAAAIHERIVQWKERLDLEISMYTFSTMKANVGMGAPILD 5j4y A 2.59 BS02 6JG A 1 W394 D430 S431 T435 P550 K551 L554 R555 L558 L565 W129 D165 S166 T170 P285 K286 L289 R290 L293 L300 3.6.4.- 0003677,0005524,0006260 remove_due_to_license_issue IC50=900nM P03072 27385654 705 TKQVSWKLVTQYALDTKCEDVFLLMGMYLNFQEAPAACAACAAADQPNHFNHHEKHYYNAQIFADSKNQKSICQQAVDTVAAKQRVDSLHMTREEMLVERFNFLLDKMDLIFGAHGNAVLEQYMAGVAWIHCLLPQMDTVIYEFLKCIVLNIPKKRYWLFKGPIDSGKTTLAAALLDLCGGKSLNVNMPLERLNFELGVGIDQFMVVFEDVKGTGAESRDLPSGHGISNLDCLRDYLDGSVKVNLERKHQNKRTQVFPPGIVTMNEYSVPRTLQARFVRQIDFRPKAYLRKSLSCSEYLLEKRILQSGMTLLLLLIWFRPVADFAAAIHERIVQWKERLDLEISMYTFSTMKANVGMGAPILD 5j58 B 2.8 BS01 N56 B 1 Y250 D287 G290 V473 W474 F522 H523 Y19 D56 G59 V237 W238 F286 H287 H256 H259 S364 D367 S390 S393 K554 K557 H25 H28 S133 D136 S154 S157 K318 K321 6.1.1.10 0000166,0004812,0004825,0005524,0006418,0006431 remove_due_to_license_issue Q38C91 27788467 803 GPGSMKVEKVFFVTSPIYYVNAAPHIGHVYSTLITDVIGRYHRVKGERVFALTGTDEHGQKVAEAAKQKQVSPYDFTTAVAGEFKKCFEQMDYSIDYFIRTTNEQHKAVVKELWTKLEQKGDIYLGRYEGWYSISDESFLTPQNITDGNPCKVSLESGHVVTWVSEENYMFRLSAFRERLLEWYHANPGCIVPEFRRREVIRAVEKGLPDLSVSRARATLHNWAIPVPGNPDHCVYVWLDALTNYLTGSRLRVDESGKEVSLVDDFNELERFPADVHVIGKDILKFHAIYWPAFLLSAGLPLPKKIVAHGWWTKDRKKISKSLGNVFDPVEKAEEFGYDALKYFLLRESGFSDDGDYSDKNMIARLNGELADTLGNLVMRCTSAKINVNGEWPSPAAYTEEDESLIQLIKDLPGTADHYYLIPDIQKAIIAVFDVLRAINAYVTDMAPWKLVKTDPERLRTVLYITLEGVRVTTLLLSPILPRKSVVIFDMLGVPEVHRKGIENFEFGAVPPGTRLGPAVEGEVLFSKRST 5j59 B 2.4 BS01 N93 B 1 I248 Y250 D287 H289 G290 V473 W474 F522 H523 I17 Y19 D56 H58 G59 V239 W240 F288 H289 H256 H259 S364 D367 S390 S393 K554 K557 H25 H28 S133 D136 S156 S159 K320 K323 6.1.1.10 0000166,0004812,0004825,0005524,0006418,0006431 ic50<50nM remove_due_to_license_issue Q38C91 27788467 802 GPGSMKVEKVFFVTSPIYYVNAAPHIGHVYSTLITDVIGRYHRVKGERVFALTGTDEHGQKVAEAAKQKQVSPYDFTTAVAGEFKKCFEQMDYSIDYFIRTTNEQHKAVVKELWTKLEQKGDIYLGRYEGWYSISDESFLTPQNITDGVDNPCKVSLESGHVVTWVSEENYMFRLSAFRERLLEWYHANPGCIVPEFRRREVIRAVEKGLPDLSVSRARATLHNWAIPVPGNPDHCVYVWLDALTNYLTGSRLRVDESGKEVSLVDDFNELERFPADVHVIGKDILKFHAIYWPAFLLSAGLPLPKKIVAHGWWTKDRKKISKSLGNVFDPVEKAEEFGYDALKYFLLRESGFSDDGDYSDKNMIARLNGELADTLGNLVMRCTSAKINVNGEWPSPAAYTEEDESLIQLIKDLPGTADHYYLIPDIQKAIIAVFDVLRAINAYVTDMAPWKLVKTDPERLRTVLYITLEGVRVTTLLLSPILPRKSVVIFDMLGVPEVHRKGIENFEFGAVPPGTRLGPAVEGEVLFSKRST 5j5d A 2.4 BS01 6GT A 1 A18 T54 T55 Y143 R148 K171 G194 A15 T51 T52 Y140 R145 K168 G191 T54 Y117 Y143 R148 K171 I211 T51 Y114 Y140 R145 K168 I208 4.3.3.7 0005737,0005829,0005886,0008840,0009085,0009089,0016829,0019877,0044281 remove_due_to_license_issue P9WP25 27501775 403 VGFDVAARLGTLLTAMVTPFSGDGSLDTATAARLANHLVDQGCDGLVVSGTTGESPTTTDGEKIELLRAVLEAVGDRARVIAGAGTYDTAHSIRLAKACAAEGAHGLLVVTPYYSKPPQRGLQAHFTAVADATELPMLLYDIPGRSAVPIEPDTIRALASHPNIVGVKDAKADLHSGAQIMADTGLAYYSGDDALNLPWLAMGATGFISVIAHLAAGQLRELLSAFGSGDIATARKINIAVAPLCNAMSRLGGVTLSKAGLRLQGIDVGDPRLPQVAATPEQIDALAADMRAASVLR 5j5r A 1.6 BS01 6G1 A 1 T203 G285 E318 T190 G272 E281 1.1.1.205 0003824,0003938,0006164,0016491 Ki=130nM remove_due_to_license_issue G7CNL4 27726334 401 PVPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAGL 5j5t A 2.85 BS01 6G2 A 1 I22 V30 A43 M90 F92 C93 G96 L143 D154 I11 V19 A32 M79 F81 C82 G85 L132 D143 D136 K138 A140 N141 D154 A163 T174 D125 K127 A129 N130 D143 A152 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q8IVH8 27727493 901 SQEDFELIQRIGSGTYGDVYKARNVNTGELAAIKVIKLEPGEDFAVVQQEIIMMKDCKHPNIVAYFGSYLRRDKLWICMEFCGGGSLQDIYHVTGPLSELQIAYVSRETLQGLYYLHSKGKMHRDIKGANILLTDNGHVKLADFGVSAQITATIAAFIGTPYWMAPEVAAVERKGGYNQLCDLWAVGITAIELAELQPPMFDLHPMRALFLMTKSNFQPPKLKDKMKWSNSFHHFVKMALTKNPKKRPTAEKLLQHPFVTQHLTRSLAIELLDKVNNPSTYHDFDDDDPEPLVAVPHR 5j5x A 2.6 BS02 6J9 A 1 V15 F18 L152 E155 I303 Y306 V7 F10 L144 E147 I295 Y298 D166 K168 E170 N171 D184 T201 D158 K160 E162 N163 D176 T193 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 27389935 404 GSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 5j64 A 1.38 BS01 6G7 A 1 N51 A55 K58 D93 I96 G97 M98 L107 G108 T184 N36 A40 K43 D78 I81 G82 M83 L92 G93 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j6a A 2.045 BS01 P46 A 1 N255 R258 A259 E262 S263 D290 G294 V295 T354 N233 R236 A237 E240 S241 D268 G272 V273 T318 H247 E251 K254 N255 H225 E229 K232 N233 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=22nM remove_due_to_license_issue Q15119 28085286 501 ASLAGAPKYIEHFSKFSPSPLSMKQFLDFGSCEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTGFGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPV 5j6d A 1.9 BS02 6H5 A 1 L129 Y235 L236 R257 Y264 T265 P266 P268 H272 A309 Y312 F313 E317 S336 S337 I366 L28 Y134 L135 R156 Y163 T164 P165 P167 H171 A208 Y211 F212 E216 S235 S236 I265 H272 H277 E317 S336 H171 H176 E216 S235 1.14.16.4 0004497,0005506,0009072,0016714 ic50=6nM remove_due_to_license_issue P17752 27146606 504 METVPWFPKKISDLDHCANRVLMYGSELDADHPGFKDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFQELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTI 5j6l A 1.75 BS01 6GC A 1 N51 A55 K58 D93 I96 G97 M98 F138 V150 W162 T184 N36 A40 K43 D78 I81 G82 M83 F123 V135 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j6m A 1.64 BS01 6FJ A 1 N51 A55 K58 D93 I96 G97 M98 L103 N106 F138 V150 W162 N36 A40 K43 D78 I81 G82 M83 L88 N91 F123 V135 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKER 5j6n A 1.9 BS01 6FF A 1 N51 A55 D93 I96 G97 M98 N106 F138 W162 T184 V186 N36 A40 D78 I81 G82 M83 N91 F123 W147 T169 V171 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5j6s A 2.8 BS02 6GA A 1 D198 P333 G334 A335 H370 E371 H374 E393 Y455 Y892 D146 P281 G282 A283 H318 E319 H322 E341 Y403 Y840 E337 H370 E371 H374 E393 Q447 Y455 E285 H318 E319 H322 E341 Q395 Y403 3.4.11.- 0002250,0002474,0004175,0004177,0005515,0005615,0005737,0005783,0005788,0005789,0006508,0008217,0008237,0008270,0016020,0019885,0042277,0043171,0046872,0070006 remove_due_to_license_issue IC50=>100000nM Q6P179 28337326 1015 FPVATNGERFPWQELRLPSVVIPLHYDLFVHPNLTSLDFVASEKIEVLVSNATQFIILHSKDLEITNATLQSEEDSRYMKPGKELKVLSYPAHEQIALLVPEKLTPHLKYYVAMDFQAKLGDGFEGFYKSTYRTLGGETRILAVTDFEPTQARMAFPCFDEPLFKANFSIKIRRESRHIALSNMPKVKTIELEGGLLEDHFETTVKMSTYLVAYIVCDFHSLSGFTSSGVKVSIYASPDKRNQTHYALQASLKLLDFYEKYFDIYYPLSKLDLIAIPDFAPGAMENWGLITYRETSLLFDPKTSSASDKLWVTRVIAHELAHQWFGNLVTMEWWNDIWLNEGFAKYMELIAVNATYPELQFDDYFLNVCFEVITKDSLNSSRPISKPAETPTQIQEMFDEVSYNKGACILNMLKDFLGEEKFQKGIIQYLKKFSYRNAKNDDLWSSLSNSCLESDFTSGGVCHSDPKMTSNMLAFLGENAEVKEMMTTWTLQKGIPLLVVKQDGCSLRLQQERFLQGVFQEDPEWRALQERYLWHIPLTYSTSSSNVIHRHILKSKTDTLDLPEKTSWVKFNVDSNGYYIVHYEGHGWDQLITQLNQNHTLLRPKDRVGLIHDVFQLVGAGRLTLDKALDMTYYLQHETSSPALLEGLSYLESFYHMMDRRNISDISENLKRYLLQYFKPVIDRQSWSDKGSVWDRMLRSALLKLACDLNHAPCIQKAAELFSQWMESSGKLNIPTDVLKIVYSVGAQTTAGWNYLLEQYELSMSSAEQNKILYALSTSKHQEKLLKLIELGMEGKVIKTQNLAALLHAIARRPKGQQLAWDFVRENWTHLLKKFDLGSYDIRMIISGTTAHFSSKDKLQEVKLFFESLEAQGSHLDIFQTVLETITKNIKWLEKNLPTLRTWLMVNTRH 5j71 A 1.65 BS01 P35 A 1 N255 R258 A259 E262 D290 G294 V295 T354 N227 R230 A231 E234 D262 G266 V267 T307 H247 E251 K254 N255 H219 E223 K226 N227 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 remove_due_to_license_issue Kd=110nM, IC50=195nM Q15119 28085286 502 SLAGAPKYIEHFSKFSPSPLSMKQFLDCEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYDWC 5j74 A 2.7 BS01 6GN A 1 S35 W47 L99 Y108 K175 Y179 W234 Y241 S34 W46 L98 Y107 K152 Y156 W211 Y218 remove_due_to_license_issue 26442911 302 VQLVESEAEVKKPGSSVKVSCKASGGTFSSYAISWVRQAPGQGLEWMGGTIPIFGTADYAQEFQGRVTITTDESTSTAYMELSGLRSEDTAVYYCVLLGTTMVTGHYFDYWGQGTLVTVNFMLTQPPSASGTPGQSVTISCSGSGSNIGNNKVNWYQQLPGTAPKLLIYSNNQRPSGVPDRFSGSKSGTSASLAISGLQSEDEADYYCAAWDDGLSGYVFGTGTKLTVLAA 5j75 A 2.0 BS01 6GQ A 1 S35 W47 G50 T57 A58 D59 L99 Y179 W234 Y241 S34 W46 G49 T56 A57 D58 L98 Y158 W213 Y220 Ki=0.63nM remove_due_to_license_issue 26442911 303 VQLVESEAEVKKPGSSVKVSCKASGGTFSSYAISWVRQAPGQGLEWMGGTIPIFGTADYAQEFQGRVTITTDESTSTAYMELSGLRSEDTAVYYCVLLGTTMVTGHYFDYWGQGTLVTVSSNFMLTQPPSASGTPGQSVTISCSGSGSNIGNNKVNWYQQLPGTAPKLLIYSNNQRPSGVPDRFSGSKSGTSASLAISGLQSEDEADYYCAAWDDGLSGYVFGTGTKLTVLAA 5j75 A 2.0 BS02 6GQ B 1 F55 T57 W234 F54 T56 W213 Ki=0.63nM remove_due_to_license_issue 26442911 303 VQLVESEAEVKKPGSSVKVSCKASGGTFSSYAISWVRQAPGQGLEWMGGTIPIFGTADYAQEFQGRVTITTDESTSTAYMELSGLRSEDTAVYYCVLLGTTMVTGHYFDYWGQGTLVTVSSNFMLTQPPSASGTPGQSVTISCSGSGSNIGNNKVNWYQQLPGTAPKLLIYSNNQRPSGVPDRFSGSKSGTSASLAISGLQSEDEADYYCAAWDDGLSGYVFGTGTKLTVLAA 5j79 A 2.69 BS01 6GE A 1 S25 A45 K47 E66 L79 T95 M98 L153 D164 S24 A44 K46 E55 L68 T84 M87 L142 D153 D146 K148 Q150 N151 D164 P185 T189 D135 K137 Q139 N140 D153 P164 T168 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=20nM O43353 27109867 401 NGEAICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLRKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRMSAPEGGTIIYMPPENYEPSIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5j7b A 2.53 BS01 6GD A 1 L24 S25 A45 K47 L79 I93 T95 M98 G101 E105 L153 D164 L20 S21 A41 K43 L70 I84 T86 M89 G92 E96 L144 D155 D146 K148 Q150 N151 D164 T189 D137 K139 Q141 N142 D155 T160 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43353 27109867 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLGTIIYMPPENYESRASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5j7f A 2.0 BS01 6GG A 1 V14 L54 G58 I61 F86 V93 H96 Y100 V4 L44 G48 I51 F76 V83 H86 Y90 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=58nM Q00987 28482147 201 DGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5j7f A 2.0 BS02 6GG D 1 M62 Q72 M52 Q62 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=58nM Q00987 28482147 201 DGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5j7f D 2.0 BS01 6GG A 1 M62 Y67 Q72 M51 Y56 Q61 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=58nM Q00987 28482147 201 GAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 5j7f D 2.0 BS02 6GG D 1 V14 L54 L57 G58 I61 Y67 V93 H96 I99 Y100 V3 L43 L46 G47 I50 Y56 V82 H85 I88 Y89 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=58nM Q00987 28482147 201 GAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 5j7g A 1.85 BS01 6GG A 1 L54 L57 G58 I61 Y67 F86 V93 H96 I99 Y100 L38 L41 G42 I45 Y51 F70 V77 H80 I83 Y84 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=58nM Q00987 28482147 201 MQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 5j7g A 1.85 BS02 6GG B 1 Y67 Q72 Y51 Q56 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Ki=58nM Q00987 28482147 201 MQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 5j7p A 1.85 BS01 6H1 A 1 P1 M2 Y36 H62 S63 I64 V106 F113 P1 M2 Y36 H62 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 27156768 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5j7p A 1.85 BS02 6H1 B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 27156768 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5j7p C 1.85 BS01 6H1 A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 27156768 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5j7p C 1.85 BS02 6H1 C 1 P1 M2 K32 Y36 H62 I64 V106 F113 P1 M2 K32 Y36 H62 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue P14174 27156768 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5j7q A 2.05 BS01 6H2 A 1 P1 M2 K32 S63 I64 V106 P1 M2 K32 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=26.6uM remove_due_to_license_issue Ki=26600nM P14174 27156768 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 5j7s A 2.368 BS01 6H3 A 1 V42 V50 M104 Y106 A107 L163 C174 F176 V16 V22 M65 Y67 A68 L124 C135 F137 D156 K158 P160 N161 I173 D175 D117 K119 P121 N122 I134 D136 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 28011204 601 SLHMIDYKEIEVEEVVGRGGVVCKAKWRAKDVAIKKAFIVELRQLSRVNHPNIVKLYLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5j7w D 2.5 BS01 MTX D 1 L55 I80 W81 W84 D220 L223 G224 F227 Y260 I313 A314 L55 I80 W81 W84 D220 L223 G224 F227 Y260 I313 A314 E59 W81 Y145 C197 R217 D220 E59 W81 Y145 C197 R217 D220 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 Ki=13uM remove_due_to_license_issue Q834R3 27517810 402 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGPDMTDFGHRVLQDPAFAEQYKEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPIAV 5j82 A 2.17 BS01 6GV A 1 N51 A55 K58 D93 G97 M98 L107 F138 V150 T184 V186 N36 A40 K43 D78 G82 M83 L92 F123 V135 T169 V171 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j86 A 1.87 BS01 6GW A 1 N51 A55 D93 I96 G97 M98 L103 F138 V150 W162 T184 N36 A40 D78 I81 G82 M83 L88 F123 V135 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j87 A 1.59 BS01 N42 A 1 L408 Q412 F413 V416 A428 K430 Y476 M477 A478 G480 C481 N526 L528 D539 L542 Y551 L13 Q17 F18 V21 A33 K35 Y81 M82 A83 G85 C86 N131 L133 D144 L147 Y156 D521 A523 R525 N526 D539 F559 D126 A128 R130 N131 D144 F164 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue EC50=<30nM, Ki=8.9nM, IC50=7.0nM Q06187 28315597 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 5j8i A 2.404 BS01 6H4 A 1 V42 V50 A61 M104 Y106 A107 L163 C174 D175 V16 V22 A33 M75 Y77 A78 L134 C145 D146 D156 K158 P160 N161 I173 D175 D127 K129 P131 N132 I144 D146 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 28011204 601 SLHMIDYKEIEVEEVVGRFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGCLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5j8m A 1.9 BS01 6DL A 1 N51 A55 K58 D93 I96 G97 M98 G108 F138 T184 N36 A40 K43 D78 I81 G82 M83 G93 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5j8m B 1.9 BS01 6DL B 1 N51 A55 K58 D93 I96 G97 M98 F138 T184 N36 A40 K43 D78 I81 G82 M83 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5j8u A 1.75 BS01 6DL A 1 N51 A55 K58 D93 I96 G97 M98 G108 T184 N35 A39 K42 D77 I80 G81 M82 G92 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5j8u B 1.75 BS01 6DL B 1 N51 A55 K58 D93 I96 G97 M98 T184 N35 A39 K42 D77 I80 G81 M82 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j8x A 2.53 BS01 OK3 A 1 S44 S110 L153 R198 T214 G215 H216 D218 R248 S41 S92 L135 R180 T196 G197 H198 D200 R230 L22 G28 L45 M48 M49 T50 L19 G25 L42 M45 M46 T47 3.4.16.4,3.5.2.6 0000270,0004180,0005515,0005886,0006508,0008233,0008360,0008658,0008800,0009002,0009252,0030288,0042803,0051301,0071555 remove_due_to_license_issue P0AEB2 27499424 400 NIKTMIPGVPQIDAESYILIDYNSGKVLAEQNADVRRDPASLTKMMTSYVIGQAMKAGKFKETDLVTIGNMFLKPGMQVPVSQLIRGINLQSGNDACVAMADFAAGSQDAFVGLMNSYVNALGLKNTHFQTVHGLDADGQYSSARDMALIGQALIRDVPNEYSIYKEKEFTFNGIRQLNRNGLLWDNSLNVDGIKTGHTDKAGYNLVASATEGQMRLISAVMGGRTFKGREAESKKLLTWGFRFFETVNPLKVGKEFASEPVWFGDSDRASLGVDKDVYLTIPRGRMKDLKASYVLNSSELHAPLQKNQVVGTINFQLDGKTIEQRPLVVLQEIPEGNFF 5j8z A 1.7 BS02 FC4 A 1 H94 H119 F131 L198 T199 T200 H95 H120 F131 L198 T199 T200 H64 H94 H96 E106 H119 T199 H65 H95 H97 E107 H120 T199 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=5nM remove_due_to_license_issue P00918 27316543 303 GMSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5j9f A 2.1 BS02 83A A 1 F895 M896 R897 I898 L899 V946 A947 V950 D951 F88 M89 R90 I91 L92 V139 A140 V143 D144 N913 H915 T942 D951 N106 H108 T135 D144 2.1.2.2,6.3.3.1,6.3.4.13 0004644,0006189,0009058 Ki=59nM remove_due_to_license_issue IC50=666nM, Ki=59nM P22102 27458733 1102 ARVAVLISGTGSNLQALIDSTREPNSSAQIDIVISNKAAVAGLDKAERAGIPTRVINHKLYKNRVEFDSAIDLVLEEFSIDIVCLAGFMRILSGPFVAKWNGKMLNIHPSLLPSFKGSNAHEQALETGVTVTGCTVHFVAEDVDAGQIILQEAVPVKRGDTVATLSERVKLAEHKIFPAALQLVASGTVQLGENGKICWV 5j9l A 2.7515 BS01 6HF A 1 V42 V50 A61 M104 Y106 A107 G110 S111 P160 L163 F176 V16 V22 A31 M72 Y74 A75 G78 S79 P128 L131 F144 D156 K158 P160 N161 I173 D175 D124 K126 P128 N129 I141 D143 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 28011204 501 SLHMIDYKEIEVEEVVGRGGVVCKAWRADVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYCLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5j9x A 1.8 BS01 6GC A 1 N51 A55 K58 D93 G97 M98 L107 F138 V150 T184 N36 A40 K43 D78 G82 M83 L92 F123 V135 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29273709 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5j9y A 2.8 BS01 6HL A 1 A743 K745 M790 M793 C797 D800 A47 K49 M94 M97 C101 D104 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G175 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=60nM P00533 27496389 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDEDMDDVVDADEYLIP 5j9z A 2.5 BS01 6HJ A 1 A743 K745 M790 M793 C797 R841 L844 A48 K50 M95 M98 C102 R146 L149 D837 A839 R841 N842 D855 D142 A144 R146 N147 D160 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=35nM P00533 27496389 1101 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMMDDVVDADEYLIPQ 5ja0 F 1.9 BS02 FPP F 1 Y10 K57 N59 R60 V66 F239 V340 L344 K347 Y1 K43 N45 R46 V52 F225 V321 L325 K328 2.5.1.1,2.5.1.10 0004659,0008299,0016765 Kd=5.3uM remove_due_to_license_issue P14324 28098152 402 YAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 5jah A 2.06 BS01 6HQ A 1 G152 L153 S273 F274 W298 H351 G98 L99 S219 F220 W244 H297 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 remove_due_to_license_issue Q13093 27167608 502 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jal A 2.06 BS01 6HO A 1 L107 F110 L111 G154 Q352 F357 L371 L53 F56 L57 G100 Q298 F303 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 Kd=980uM remove_due_to_license_issue IC50=500000nM, Kd=980000nM Q13093 27167608 505 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jan A 2.12 BS01 6HP A 1 L153 E214 W298 F322 L99 E160 W244 F268 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 remove_due_to_license_issue IC50=1000000nM Q13093 27167608 504 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jao A 2.06 BS02 6HX A 1 L111 F125 F357 L371 L57 F71 F303 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 remove_due_to_license_issue IC50=100000nM Q13093 27167608 504 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jap A 2.46 BS01 6HZ A 1 L107 F110 L111 F125 G154 Q352 F357 L371 L53 F56 L57 F71 G100 Q298 F303 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=0.23uM remove_due_to_license_issue IC50=230nM Q13093 27167608 504 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jar A 2.11 BS01 6HV A 1 L107 F110 L111 F125 G154 Q352 F357 L371 L53 F56 L57 F71 G100 Q298 F303 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=2uM remove_due_to_license_issue IC50=2000nM Q13093 27167608 504 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jas A 2.06 BS01 6HW A 1 F110 L111 F125 F357 L371 F56 L57 F71 F303 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=1.7uM remove_due_to_license_issue IC50=1700nM Q13093 27167608 504 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jat A 2.04 BS01 6HR A 1 L107 F110 L111 L121 F125 Q352 F357 L371 L53 F56 L57 L67 F71 Q298 F303 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=0.23uM remove_due_to_license_issue IC50=7100nM Q13093 27167608 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jau A 1.95 BS01 6HU A 1 L107 F110 L111 F125 L153 A155 F357 L369 L371 L53 F56 L57 F71 L99 A101 F303 L315 L317 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=0.0014uM remove_due_to_license_issue IC50=18nM Q13093 27167608 504 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5jaz A 1.4 BS01 LC5 A 1 S232 S269 S270 S306 N311 K312 H341 P358 M360 S156 S193 S194 S230 N235 K236 H265 P282 M284 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.28uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jbi A 1.7 BS01 6J8 A 1 S232 S270 W296 S306 N311 K312 P358 D359 S156 S194 W220 S230 N235 K236 P282 D283 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.12uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jc1 A 1.65 BS01 6JB A 1 S232 E233 S269 S270 S306 N311 K312 H341 P358 D359 M360 S156 E157 S193 S194 S230 N235 K236 H265 P282 D283 M284 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.15uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jcb A 2.3 BS04 NV4 B 1 S178 T179 A180 V181 S178 T179 A180 V181 3.6.5.- 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0015630,0016787,0046872 remove_due_to_license_issue Q2XVP4 28035796 505 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVDS 5jcb B 2.3 BS02 NV4 B 1 C241 L248 A250 D251 K254 L255 N258 M259 V315 A316 K352 T353 C236 L243 A245 D246 K249 L250 N253 M254 V308 A309 K345 T346 ? 0000226,0000278,0003924,0005200,0005515,0005525,0005737,0005856,0005874,0007017,0046872 remove_due_to_license_issue P02554 28035796 505 REIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5jcj A 1.76 BS02 6JM A 1 S95 F97 Y174 L208 L209 W221 S94 F96 Y155 L189 L190 W202 R14 D161 Y174 K178 R13 D142 Y155 K159 ? 0000166,0016491,0047040 remove_due_to_license_issue O76290 27411733 303 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jcj D 1.76 BS02 6JM D 1 S95 F97 Y174 V206 L208 L209 W221 S94 F96 Y154 V186 L188 L189 W201 R14 D161 Y174 K178 R13 D141 Y154 K158 ? 0000166,0016491,0047040 remove_due_to_license_issue O76290 27411733 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jdc A 1.78 BS02 6JP A 1 F97 D161 M163 C168 L208 L209 P210 W221 F96 D142 M144 C149 L189 L190 P191 W202 R14 D161 Y174 K178 R13 D142 Y155 K159 ? 0000166,0016491,0047040 ic50=104.2uM remove_due_to_license_issue O76290 27411733 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jdc C 1.78 BS02 6JP C 1 F97 D161 M163 C168 L209 P210 F96 D140 M142 C147 L187 P188 R14 D161 Y174 K178 R13 D140 Y153 K157 ? 0000166,0016491,0047040 ic50=104.2uM remove_due_to_license_issue O76290 27411733 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVKTVETQVAELIGTNAIAPFLLTMSFAQRQNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLPEEKDKWRRKVPLGRRSAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jdc D 1.78 BS02 6JP D 1 F97 D161 M163 C168 P210 W221 F96 D141 M143 C148 P190 W201 R14 D161 Y174 K178 R13 D141 Y154 K158 ? 0000166,0016491,0047040 ic50=104.2uM remove_due_to_license_issue O76290 27411733 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jdi A 1.38 BS02 6JO A 1 S95 F97 Y174 L208 L209 P210 W221 S94 F96 Y155 L189 L190 P191 W202 R14 D161 Y174 K178 R13 D142 Y155 K159 ? 0000166,0016491,0047040 remove_due_to_license_issue O76290 27411733 304 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jdi D 1.38 BS02 6JO D 1 S95 F97 Y174 V206 L208 P210 W221 S94 F96 Y154 V186 L188 P190 W201 R14 D161 Y174 K178 R13 D141 Y154 K158 ? 0000166,0016491,0047040 remove_due_to_license_issue O76290 27411733 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQKTVETQVAELIGTNAIAPFLLTMSFAQRQNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5jf1 A 2.0 BS01 BB2 A 1 G70 V71 G72 Q77 L125 G128 E129 G130 C131 L132 Y167 H174 E175 H178 G69 V70 G71 Q76 L124 G127 E128 G129 C130 L131 Y166 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=64nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf2 A 2.0 BS01 SF7 A 1 G69 G70 V71 G72 Q77 E129 C131 H174 E175 H178 G68 G69 V70 G71 Q76 E128 C130 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=13nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf3 A 1.6 BS01 SF5 A 1 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=38nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf4 A 2.4 BS01 6JT A 1 V71 Q77 C131 L132 H174 E175 H178 V70 Q76 C130 L131 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=65nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf5 A 1.8 BS01 7JT A 1 G70 V71 G72 Q77 E129 C131 L132 H174 E175 H178 G69 V70 G71 Q76 E128 C130 L131 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=63nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf6 A 1.7 BS01 BB4 A 1 G72 Q77 E129 G130 C131 L132 H174 E175 H178 G71 Q76 E128 G129 C130 L131 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=62nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf7 A 2.1 BS01 6JU A 1 G72 Q77 E129 G130 C131 L132 H174 E175 H178 G71 Q76 E128 G129 C130 L131 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=909nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jf8 A 1.8 BS01 PN3 A 1 G72 Q77 E129 G130 C131 H174 E175 H178 G71 Q76 E128 G129 C130 H173 E174 H177 G72 Q77 C131 L132 H174 E175 H178 G71 Q76 C130 L131 H173 E174 H177 3.5.1.88 0006412,0016787,0042586,0043686,0046872 Ki=1428nM remove_due_to_license_issue Q8E378 27762275 301 AAIDKLVKASHLIDMNDIIREGNPTLRKVAEEVTFPLSEKEEILGEKMMQFLKHSQDPIMAEKLGLRGGVGLAAPQLDISKRIIAVLVPNVEDAQGNPPKEAYSLQEVMYNPKVVSHSVQDAALSDGEGCLSVDREVPGYVVRHARVTIEYFDKTGEKHRLKLKGYNSIVVQHEIDHIDGIMFYDRINEKNPFAVKEGLLILE 5jfp A 1.49 BS01 6KK B 1 D25 A28 D30 V82 I84 D25 A28 D30 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 27389367 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5jfp B 1.49 BS01 6KK B 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.48nM remove_due_to_license_issue P03366 27389367 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5jfr A 1.6 BS03 6KP A 1 H231 D262 H331 I338 H339 A414 Y444 H122 D153 H222 I229 H230 A302 Y332 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E252 E347 3.4.11.18 0006508,0070006 ic50=5nM remove_due_to_license_issue P50579 27136719 505 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGTRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 5jfu A 1.7 BS01 6KQ B 1 D25 A28 D30 T80 V82 I84 D25 A28 D30 T80 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 27389367 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5jfu B 1.7 BS01 6KQ B 1 D25 G27 A28 D29 G48 G49 I50 I84 D25 G27 A28 D29 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=8.5nM remove_due_to_license_issue P03366 27389367 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5jg1 A 1.16 BS01 6KR B 1 D25 A28 D30 G48 V82 I84 D25 A28 D30 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 27389367 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5jg1 B 1.16 BS01 6KR B 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.9nM remove_due_to_license_issue P03366 27389367 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5jga A 2.0 BS01 6KC A 1 V42 G43 R44 K63 M104 Y106 A107 G110 L163 C174 D175 V17 G18 R19 K38 M79 Y81 A82 G85 L138 C149 D150 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 ic50=2.3nM remove_due_to_license_issue O43318,Q15750 27448772 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTAGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5jgb A 2.8 BS01 6JV A 1 V42 V50 M104 Y106 A107 G110 L163 C174 D175 V17 V25 M79 Y81 A82 G85 L138 C149 D150 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 27448772 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5jgd A 3.101 BS01 6KD A 1 V42 M104 A107 G110 S111 N114 L163 C174 D175 V17 M79 A82 G85 S86 N89 L138 C149 D150 D156 K158 P160 N161 I173 D175 D131 K133 P135 N136 I148 D150 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 27448772 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTAGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDH 5jgi B 1.38 BS01 AAG B 1 Y297 T316 D320 S346 T349 Y353 G414 I415 Y24 T43 D47 S73 T76 Y80 G141 I142 ? remove_due_to_license_issue O14786 29430837 501 KCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 5jgq B 1.6 BS01 6JY B 1 Y297 T316 D320 S346 T349 Y353 G414 I415 Y24 T43 D47 S73 T76 Y80 G141 I142 ? remove_due_to_license_issue O14786 29430837 501 KCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 5jh0 A 2.18 BS01 dna B 0 K27 K30 K118 F123 L144 M147 K148 W154 Y169 K1 K4 K92 F97 L118 M121 K122 W128 Y143 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 KASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYPL 5jh0 A 2.18 BS02 dna C 0 K27 T32 K117 K118 I124 R131 Q143 K1 T6 K91 K92 I98 R105 Q117 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 KASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYPL 5jh0 A 2.18 BS03 dna E 0 R45 S48 Y50 F51 A71 S74 K75 W81 Q82 Y100 R19 S22 Y24 F25 A45 S48 K49 W55 Q56 Y74 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 KASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYPL 5jh0 A 2.18 BS04 dna F 0 K44 R45 T47 F51 Q55 R58 R69 P70 K18 R19 T21 F25 Q29 R32 R43 P44 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 KASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYPL 5jh0 D 2.18 BS01 dna B 0 R45 S48 Y50 F51 A71 S74 K75 W81 Q82 Y100 R21 S24 Y26 F27 A47 S50 K51 W57 Q58 Y76 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 HHKASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYP 5jh0 D 2.18 BS02 dna C 0 K44 R45 T47 F51 R69 P70 K20 R21 T23 F27 R45 P46 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 HHKASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYP 5jh0 D 2.18 BS03 dna E 0 S29 K30 K118 F123 L144 M147 W154 Q155 Y169 S5 K6 K94 F99 L120 M123 W130 Q131 Y145 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 HHKASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYP 5jh0 D 2.18 BS04 dna F 0 H0 K27 S29 R31 T32 K117 K118 I124 N128 Q143 H2 K3 S5 R7 T8 K93 K94 I100 N104 Q119 ? remove_due_to_license_issue Q02486 27899643 1 ~ 22 HHKASKRTQLRNELIKQGPKRPTSAYFLYLQDHRSQFVKENPTLRPAEISKIAGEKWQNLEADIKEKYISERKKLYSEYQKAKKEFDEKLPPKKPAGPFIKYANEVRSQVFAQHPDKSQLDLMKIIGDKWQSLDQSIKDKYIQEYKKAIQEYNARYP 5jh6 A 2.365 BS01 T92 A 1 V42 V50 A61 A107 L163 C174 V16 V23 A34 A77 L133 C144 D156 K158 P160 N161 I173 D175 D126 K128 P130 N131 I143 D145 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 28011204 601 SLHMIDYKEIEVEEVVGRGAFVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5jha A 2.51 BS01 6K7 A 1 I831 K833 D836 I879 E880 I881 V882 I963 D964 I570 K572 D575 I618 E619 I620 V621 I697 D698 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 28276440 1201 EESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHSQTIKVSPDDTPGAILQSFFTQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIRVPFVLTPDFLFVMGTTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFL 5jhb A 2.48 BS01 6K5 A 1 K833 D836 E880 I881 V882 M953 I963 D964 K574 D577 E621 I622 V623 M687 I697 D698 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 Kd=873nM remove_due_to_license_issue P48736 28276440 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRCDRKFRVKIRGIDIPVLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIAAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSASSQVISQLKQKLENLQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 5jhk A 1.8 BS01 6K8 A 1 Y297 W301 T316 D320 S346 T349 Y353 G414 I415 Y24 W28 T43 D47 S73 T76 Y80 G141 I142 ? remove_due_to_license_issue O14786 29430837 501 KCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 5ji6 A 2.15 BS03 6KN A 1 H231 D262 H331 I338 H339 A414 Y444 H122 D153 H222 I229 H230 A304 Y334 D251 D262 H331 H339 E364 E459 D142 D153 H222 H230 E254 E349 3.4.11.18 0006508,0070006 ic50=0.011uM remove_due_to_license_issue P50579 27155900 504 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY 5ji8 A 1.42 BS01 6KT A 1 F161 V165 I169 N216 Y222 F23 V27 I31 N78 Y84 ? Kd=23.4uM remove_due_to_license_issue Q9H8M2 27194508 301 TPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 5jic A 1.4 BS02 N7E A 1 E70 G100 R113 G116 I117 E66 G96 R109 G112 I113 2.7.1.33 0004594,0005524,0005737,0005829,0015937,0016301 ic50=0.13uM remove_due_to_license_issue Q2FWC7 27759386 303 KVGIDAGGTLIKIVQEQRTFKTELTKNIDQVVEWLNQQQIEKLCLTGGNAGVIAENINIPAQIFVEFDAASQGLGILLKEQGHDLADYIFANVGTGTSLHYFDGQSQRRVGGIGTGGGMIQGLGYLLSQITDYKQLTDMAQHGDRNTIDLKVRHIYKDTEPPIPGDLTAANFGHVLHHLDADFTPSNKLAAVIGVVGEVVTTMAITVAREFKTENIVYIGSSFHNNALLRKVVEDYTVLRGCKPYYVENGAFSGAIGALYLEKHHHHHH 5jid A 1.2 BS01 8PF A 1 K15 L17 A108 L110 S117 T119 K6 L8 A99 L101 S108 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 27668830 301 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5jid B 1.2 BS01 8PF B 1 K15 A108 K6 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 27668830 301 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5jim A 1.26 BS01 P8S A 1 K15 L17 A108 L110 K6 L8 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5jim B 1.26 BS01 P8S B 1 K15 A108 L110 S117 T118 T119 K6 A99 L101 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5jiq A 1.45 BS01 27M A 1 S117 T118 T119 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5jiq B 1.45 BS01 27M B 1 L17 S117 T118 L8 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5jjr A 1.99 BS04 68E A 1 L511 C709 S710 H711 R729 R737 M761 M765 T794 S796 H798 A799 H800 Q802 W803 L478 C676 S677 H678 R696 R704 M723 M727 T756 S758 H760 A761 H762 Q764 W765 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0004482,0004483,0005524,0008168,0032259,0039694 ic50=0.016uM remove_due_to_license_issue Q6YMS4 27500641 1004 ETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTRHVNAEPETPNMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTWDSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMMGSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYM 5jjs A 1.65 BS03 6L2 A 1 L511 C709 H711 R729 R737 M765 T794 W795 S796 H798 A799 H800 Q802 W803 L478 C676 H678 R696 R704 M730 T759 W760 S761 H763 A764 H765 Q767 W768 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003968,0004482,0004483,0005524,0008168,0032259,0039694 ic50=0.048uM remove_due_to_license_issue Q6YMS4 27500641 1004 GETLGEKWKKKLNQLSRKEFDLYKKSGITEVDRTEAKEGLKRGETTHHAVSRGSAKLQWFVERNMVIPEGRVIDLGCGRGGWSYYCAGLKKVTEVRGYTKGGPGHEEPVPMSTYGWNIVKLMSGKDVFYLPPEKCDTLLCDIGESSPSPTVEESRTIRVLKMVEPWLKNNQFCIKVLNPYMPTVIEHLERLQRKHGGMLVRNPLSRNSTHEMYWISNGTGNIVSSVNMVSRLLLNRFTMTHRRPTIEKDVDLGAGTRHVNAEPETPNMDVIGERIKRIKEEHNSTWHYDDENPYKTWAYHGSYEVKATGSASSMINGVVKLLTKPWDVVPMVTQMAMTDTTPFGQQRVFKEKVDTRTPRPLPGTRKVMEITAEWLWRTLGRNKRPRLCTREEFTKKVRTNWDSAKAAVEDEEFWKLVDRERELHKLGKCGSCVYNMSRAIWYMWLGVRYLEFEALGFLNEDHWFSRENSYSGVEGEGLHKLGYILRDISKIPGGAMYADDTAGWDTRITEDDLHNEEKIIQQMDPEHRQLANAIFKLTYQNKVVKVQRPTPTGTVMDIISRKDQRGSGQVGTYGLNTFTNMEAQLVRQMEGEGVLTKADLENPHLLEKKITQWLETKGVERLKRMAISGDDCVVKPIDDRFANALLALNDMGKVRKDIPQWQPSKGWHDWQQVPFCSHHFHELIMKDGRKLVVPCRPQDELIGRARISQGWSLRETACLGKAYAQMWSLMYFHRRDLRLASNAICSAVPVHWVPTSRTTWSIHAHHQWMTTEDMLTVWNRVWIEENPWMEDKTPVTTWENVPYLGKREDQWCGSLIGLTSRATWAQNIPTAIQQVRSLIGNEEFLDYMP 5jk0 A 2.1 BS01 dna E 0 K62 R65 N66 L120 S121 A123 T124 N127 S193 R199 N277 Q278 T284 A286 Y287 K305 H309 A336 K62 R65 N66 L116 S117 A119 T120 N123 S178 R184 N262 Q263 T269 A271 Y272 K290 H294 A321 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 1 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLIAFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHFDKQRLEEAASIWEEN 5jk0 A 2.1 BS02 dna F 0 K26 L30 S31 Q34 G71 T74 Y75 K126 R129 R213 S214 N215 Q285 Y289 G307 H309 K26 L30 S31 Q34 G71 T74 Y75 K122 R125 R198 S199 N200 Q270 Y274 G292 H294 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 1 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLIAFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHFDKQRLEEAASIWEEN 5jk0 B 2.1 BS01 dna G 0 K62 R65 N66 L77 L120 S121 T124 N127 S193 R199 R213 N277 L283 T284 A286 Y287 K305 H309 H335 A336 K62 R65 N66 L77 L116 S117 T120 N123 S178 R184 R198 N262 L268 T269 A271 Y272 K290 H294 H320 A321 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 1 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLITFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHFDKQRLEEAASIWE 5jk0 B 2.1 BS02 dna H 0 K26 L30 S31 L70 G71 N73 T74 Y75 K126 R129 K158 S214 N215 Q285 Y289 G307 H309 K26 L30 S31 L70 G71 N73 T74 Y75 K122 R125 K154 S199 N200 Q270 Y274 G292 H294 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 2 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLITFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHFDKQRLEEAASIWE 5jk0 C 2.1 BS01 dna E 0 K26 L30 S31 T74 Y75 R213 N215 Q285 Y289 G307 H309 K26 L30 S31 T74 Y75 R204 N206 Q276 Y280 G298 H300 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 1 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLITERLAFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKNIKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHFRLEEAASIWE 5jk0 C 2.1 BS02 dna F 0 K62 R65 N66 L77 S121 A123 T124 N127 S193 R199 N277 Q278 T284 A286 Y287 A336 T340 K62 R65 N66 L77 S121 A123 T124 N127 S184 R190 N268 Q269 T275 A277 Y278 A327 T331 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 1 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLITERLAFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKNIKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHFRLEEAASIWE 5jk0 D 2.1 BS01 dna G 0 K26 L30 S31 L70 T74 Y75 I130 R213 S214 N215 Q285 Y289 K305 G307 H309 K26 L30 S31 L70 T74 Y75 I130 R205 S206 N207 Q277 Y281 K297 G299 H301 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 1 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLITERLAFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKNISKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHRLEEAASIWEE 5jk0 D 2.1 BS02 dna H 0 K62 R65 N66 S121 A123 T124 N127 S193 R199 N277 Q278 T284 A286 Y287 H335 A336 K62 R65 N66 S121 A123 T124 N127 S185 R191 N269 Q270 T276 A278 Y279 H327 A328 ? 0003677,0005737,0006310,0007059,0009037,0015074,0051301 remove_due_to_license_issue O25386 28009253 2 ~ 30 MKHPLEELKDPTENLLLWIGRFLRYKCTSLSNSQVKDQNKVFECLNELNQACSSSQLEKVCKKARNAGLLGINTYALPLLKFHEYFSKARLITERLAFNSLKNIDEVMLAEFLSVYTGGLSLATKKNYRIALLGLFSYIDKQNQDENEKSYIYNITLKNISKLPTHLNNEELEKFLESIDKIEMSAKVRARNRLLIKIIVFTGMRSNEALQLKIKDFTLENGCYTILIKGKGDKYRAVMLKAFHIESLLKEWLIERELYPVKNDLLFCNQKGSALTQAYLYKQVERIINFAGLRREKNGAHMLRHSFATLLYQKRHDLILVQEALGHASLNTSRIYTHRLEEAASIWEE 5jk3 A 2.371 BS01 6L4 A 1 A107 L163 C174 A59 L115 C126 D156 K158 P160 N161 I173 D175 D108 K110 P112 N113 I125 D127 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue O43318,Q15750 28011204 601 SLHMIIEVEEVVGRVCKAIKQISESERKAFIVELRQLSRVNHPNIVKLYNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5jlt A 2.955 BS01 dna E 0 R98 T100 R101 A103 R104 R135 R161 R1 T3 R4 A6 R7 R38 R64 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 RATRKAREITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt A 2.955 BS02 dna F 0 R98 R101 R145 Y165 K166 R1 R4 R48 Y68 K69 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 RATRKAREITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt B 2.955 BS01 dna G 0 R135 R161 R32 R58 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 REITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt B 2.955 BS02 dna H 0 Y165 K166 Y62 K63 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 REITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt C 2.955 BS01 dna G 0 K129 R145 Y165 K166 K28 R44 Y64 K65 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 KAREITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt C 2.955 BS02 dna H 0 A103 R135 S136 K183 A185 Y191 A2 R34 S35 K82 A84 Y90 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 KAREITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt D 2.955 BS01 dna E 0 R145 R150 Y165 K166 R40 R45 Y60 K61 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 ITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlt D 2.955 BS02 dna F 0 R135 R161 A185 R30 R56 A80 ? remove_due_to_license_issue P22915 29718457 1 ~ 22 ITSDMEEDKDLMLKLLDKNGFVLKKVEIYRSNYLAILEKRTNGIRNFEINNNGNMRIFGYKMMEHHIQKFTDIGMSCKIAKNGNVYLDIKRSAENIEAVITVASEL 5jlw A 2.088 BS01 dna B 0 R5 T7 Y25 R31 Q50 R53 M54 R2 T4 Y22 R28 Q47 R50 M51 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 0 ~ 14 GRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlw A 2.088 BS02 dna C 0 R5 Q6 Y8 R43 Q44 I47 N51 R2 Q3 Y5 R40 Q41 I44 N48 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 0 ~ 14 GRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlw D 2.088 BS01 dna E 0 R5 Y25 R31 Q50 R53 M54 R2 Y22 R28 Q47 R50 M51 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 1 ~ 15 GRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlw D 2.088 BS02 dna F 0 R5 Q6 Y8 R43 Q44 I47 N51 K55 R2 Q3 Y5 R40 Q41 I44 N48 K52 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 1 ~ 15 GRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlx A 2.748 BS01 dna B 0 R5 T7 Y25 R31 K46 Q50 R53 M54 K57 R2 T4 Y22 R28 K43 Q47 R50 M51 K54 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 0 ~ 14 GRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlx A 2.748 BS02 dna C 0 R5 Q6 Y8 Q44 W48 N51 R2 Q3 Y5 Q41 W45 N48 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 0 ~ 14 GRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlx D 2.748 BS01 dna E 0 Y25 R31 Q50 R53 M54 Y23 R29 Q48 R51 M52 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 1 ~ 15 RGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jlx D 2.748 BS02 dna F 0 R5 Q6 Y8 R43 I47 W48 N51 R3 Q4 Y6 R41 I45 W46 N49 ? 0000981,0003677,0006355 remove_due_to_license_issue P02833 27271797 1 ~ 15 RGRQTYTRYQTLELEKEFHFNRYLTRRRRIEIAHALSLTERQIKIWFQNRRMKWKKEN 5jmp A 1.7 BS01 LC7 A 1 S232 E233 S269 S270 W296 S306 N311 K312 H341 P358 D359 M360 S156 E157 S193 S194 W220 S230 N235 K236 H265 P282 D283 M284 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.067uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jmw A 1.55 BS01 L50 A 1 S232 S269 S270 W296 M298 S306 N311 K312 H341 P358 D359 S156 S193 S194 W220 M222 S230 N235 K236 H265 P282 D283 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.175uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jmx A 1.44 BS03 DZ5 A 1 H118 D120 H179 C198 N210 H240 H78 D80 H139 C158 N170 H200 H116 H118 D120 H179 C198 K201 N210 H240 H76 H78 D80 H139 C158 K161 N170 H200 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue IC50=8200nM P04190 29655609 304 KTVIKNETGTISISQLNKNVWVHTELGAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 5jn8 A 1.85 BS01 AZM A 1 Q92 H94 H119 L198 T199 T200 Q95 H97 H122 L199 T200 T201 H64 H94 H96 E106 H119 T199 H70 H97 H99 E109 H122 T200 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 remove_due_to_license_issue Ki=74nM, Kd=100nM, IC50=17.5nM P22748 28975383 701 AESHWCYEVQAESSNYPCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKGTSDPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 5jn9 A 2.1 BS02 EZL A 1 H94 L198 T199 T200 W209 H97 L199 T200 T201 W210 H64 H94 H96 E106 H119 T199 H70 H97 H99 E109 H122 T200 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 remove_due_to_license_issue Ki=93nM P22748 28975383 302 AESHWCYEVQAESSNYPCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKGTSDPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 5jna A 2.0 BS02 TOR A 1 N62 S65 Q92 H94 H119 L198 T199 T200 N68 S71 Q95 H97 H122 L199 T200 T201 H64 H94 H96 E106 H119 T199 H70 H97 H99 E109 H122 T200 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 remove_due_to_license_issue Ki=4900nM P22748 28975383 302 AESHWCYEVQAESSNYPCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKGTSDPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 5jnl A 1.6 BS01 L54 A 1 S232 S269 S270 W296 S306 N311 K312 H341 P358 D359 M360 S156 S193 S194 W220 S230 N235 K236 H265 P282 D283 M284 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.27uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jnn A 2.3 BS01 6LM A 1 K64 Y124 N173 K51 Y111 N160 ? 0004864,0005515,0005634,0005737,0005886,0009738,0010427,0038023,0042802,0042803,0062049 ic50=4504nM remove_due_to_license_issue O80992 27518563 800 EQKTLEPVIKTYHQFEPDPTTCTSLITQRIHAPASVVWPLIRRFDNPERYKHFVKRCRLISGDGDVGSVREVTVISGLPASTSTERLEFVDDDHRVLSFRVVGGEHRLKNYKSVTSVNEFLNQDSGKVYTVVLESYTVDIPEGNTEEDTKMFVDTVVKLNLQKLGVAATSAPMHD 5jo0 A 1.8 BS01 L56 A 1 S232 E233 S269 S270 S306 N311 K312 P358 M360 S156 E157 S193 S194 S230 N235 K236 P282 M284 1.1.1.267 0008299,0030604,0046872,0070402 ic50=0.05uM remove_due_to_license_issue Q8IKG4 27487410 501 PINVAIFGSTGSIGTNALNIIRECNKIENVFNVKALYVNKSVNELYEQAREFLPEYLCIHDKSVYEELKELVKNIKDYKPIILCGDEGMKEICSSNSIDKIVIGIDSFQGLYSTMYAIMNNKIVALANKESIVSAGFFLKKLLNIHKNAKIIPVDSEHSAIFQCLDNNKVLKTKCLQDNFSKINNINKIFLCSSGGPFQNLTMDELKNVTSENALKHPKWKMGKKITIDSATMMNKGLEVIETHFLFDVDYNDIEVIVHKECIIHSCVEFIDKSVISQMYYPDMQIPILYSLTWPDRIKTNLKPLDLAQVSTLTFHKPSLEHFPCIKLAYQAGIKGNFYPTVLNASNEIANNLFLNNKIKYFDISSIISQVLESFNSQKVSENSEDLMKQILQIHSWAKDKATDIYNKHN 5jog A 2.46 BS02 6LT A 1 E76 V77 M78 W136 H138 H140 D151 T154 N158 E73 V74 M75 W126 H128 H130 D141 T144 N148 3.4.-.- 0008233,0008237 ic50=0.0058uM remove_due_to_license_issue IC50=5.8nM Q92905 27774986 302 SGSGMAQKTWELANNMQEAQSIDEIYKYDKKQQQEILAAKPWTKDHHYFKYCKISALALLKMVMHARSGGNLEVMGLMLGKVDGETMIIMDSFALPVNAQAAAYEYMAAYIENAKQVGRLENAIGWYHSHPGYGCWLSGIDVSTQMLNQQFQEPFVAVVIDPTRKVNLGAFRTYPKGYKPPDEGPSEYQTIPLNKIEDFGVHCKQYYALEVSYFKSSLDRK 5joh A 1.99 BS02 6M3 A 1 E76 W136 H138 H140 D151 T154 E73 W126 H128 H130 D141 T144 3.4.-.- 0008233,0008237 ic50=1.1uM remove_due_to_license_issue Q92905 27774986 302 SGSGMAQKTWELANNMQEAQSIDEIYKYDKKQQQEILAAKPWTKDHHYFKYCKISALALLKMVMHARSGGNLEVMGLMLGKVDGETMIIMDSFALPVNAQAAAYEYMAAYIENAKQVGRLENAIGWYHSHPGYGCWLSGIDVSTQMLNQQFQEPFVAVVIDPTRKVNLGAFRTYPKGYKPPDEGPSEYQTIPLNKIEDFGVHCKQYYALEVSYFKSSLDRK 5jox A 1.8 BS01 EDG A 1 D34 F51 A94 D140 E189 H253 R283 D15 F32 A75 D121 E170 H234 R264 3.2.1.55 0000272,0004553,0005975,0016798,0042597,0046556,0085030,2000899 Kd=35uM remove_due_to_license_issue A7LXT8 27466444 601 HQGYSNPVIPGFHPDPSVCKAGDDYYLVNSSFQYFPGVPLFHSKDLVHWEQIGNCLTRPSQLDLTNANSGSGIFAPTIRYNDGVFYMITTNVSGKGNFLVHTTDPRSEWSEPVWLEQGGIDPSLYFEDGKCFMVSNPDGYINLCEIDPMTGKQLSSSKRIWNGTGGRYAEGPHIYKKDGWYYLLISEGGTELGHKVTIARSRYIDGPYQGNPANPILTHANESGQSSPIQGTGHADLVEGTDGSWWMVCLAYRIMPGTHHTLGRETYLAPVRWDKDAWPVVNSNGTISLKMDVPTLPQQEMKGRPERIDFKEGKLSPEWIHLQNPEAKNYIFTKDGKLRLIATPVTLSDWKSPTFVALRQEHFDMEASAPVVLQKAGVNDEAGISVFMEFHSHYDLFVRQDKDRKRSVGLRYKLGEITHYAKEVSLPTDGEVELVVKSDINYYYFGYKVNGIYHDLGKMNTRYLSTETAGGFTGVVLGLYITSASKDSKAYADFEYFKYKGK 5jpt A 2.935 BS01 CDP A 1 G119 G121 K122 T123 T124 S155 V156 R159 F357 T384 D386 R430 G117 G119 K120 T121 T122 S153 V154 R157 F355 T382 D384 R428 3.6.4.13 0000390,0000462,0000463,0000466,0003676,0003689,0003723,0003724,0003729,0004386,0005515,0005524,0005634,0005681,0005730,0005739,0006338,0006364,0006396,0006397,0008186,0008380,0016787,0016887,0022613,0030490,0030686,0032040,0042273,0061775,0071014,0140584,0140588,0140665,0140849,1990904 remove_due_to_license_issue P53131 28180308 801 SKRRFSSEHPDPVETSIPEQAAEIAEELSKQHPLPSEEPLVHHDAGEFKGLQRHHTSAEEAQKLEDGKINPFTGREFTPKYVDILKIRRELPVHAQRDEFLKLYQNNQIMVFVGETGSGKTTQIPQFVLFDEMPHLENTQVACTQPRRVAAMSVAQRVAEEMDVKLGEEVGYSIRFENKTSNKTILKYMTDGMLLREAMEDHDLSRYSCIILDEAHERTLATDILMGLLKQVVKRRPDLKIIIMSATLDAEKFQRYFNDAPLLAVPGRTYPVELYYTPEFQRDYLDSAIRTVLQIHATEEAGDILLFLTGEDEIEDAVRKISLEGDQLVREEGCGPLSVYPLYGSLPPHQQQRIFEPAPESHNGRPGRKVVISTNIAETSLTIDGIVYVVDPGFSKQKVYNPRIRVESLLVSPISKASAQQRAGRAGRTRPGKCFRLYTEEAFQKELIEQSYPEILRSNLSSTVLELKKLGIDDLVHFDFMDPPAPETMMRALEELNYLACLDDEGNLTPLGRLASQFPLDPMLAVMLIGSFEFQCSQEILTIVAMLSVPNVFIRPTKDKKRADDAKNIFAHPDGDHITLLNVYHAFKSDEAYEYGIHKWCRDHYLNYRSLSAADNIRSQLERLMNRYNLELNTTDYESPKYFDNIRKALASGFFMQVAKKRSGGYITVKDNQDVLIHPSTVLGHDAEWVIYNEFVLTSKNYIRTVTSVRPEWLIEIAPAYYDLSNFQKGDVKLSLERIKEKVDR 5jq5 A 1.94 BS01 I74 A 1 I10 V18 A31 F80 F82 L83 Q85 N132 L134 A144 D145 I8 V16 A29 F69 F71 L72 Q74 N121 L123 A133 D134 D127 K129 Q131 N132 D145 T158 T165 D116 K118 Q120 N121 D134 T147 T154 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=2341nM remove_due_to_license_issue IC50=620nM P24941 28125165 302 NFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5jq7 A 2.69 BS01 T0R B 1 R64 V66 E100 A101 L186 R35 V37 E71 A72 L157 ? remove_due_to_license_issue EC50=63nM, Kd=16000nM Q05320 27362232 705 GRSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTEWAFWETSEELSFTVVAAAAAAA 5jq7 B 2.69 BS01 T0R B 1 L515 Y517 T519 M548 L558 L14 Y16 T18 M47 L57 ? remove_due_to_license_issue EC50=63nM, Kd=16000nM Q05320 27362232 705 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVD 5jq8 A 1.94 BS01 I73 A 1 I10 G13 V18 A31 L83 H84 Q131 N132 L134 D145 I8 G11 V16 A29 L72 H73 Q120 N121 L123 D134 D127 K129 Q131 N132 D145 T165 D116 K118 Q120 N121 D134 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=580nM P24941 28125165 301 NFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5jq9 A 2.101 BS01 6MB A 1 D96 N115 I117 D185 G189 F190 G217 K221 S222 R255 D84 N103 I105 D167 G171 F172 G199 K203 S204 R237 K221 R255 K203 R237 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue A0A2S9PLG4 27423480 301 MHLTARGLTLDLSRPQVMGILNVTPNLDQALQHAQRMLSAGATLIDIGGESTRAAEVSEQEELDRVVPVVEALAQRFDVWLSVDTSKAAVITESAHAGAHLINDIRSLQEPGALEAAAKTGLPVCLMHMQQHSPYYDDLMTDINRFFQHHIERCVAAGIAKNKLLLDPGFGFGKNLAHNYQLLAHLSELHHFELPLLVGMSRKSMVGQLLNVPPQQRVIGSVACAVIAAMQGAQIIRVHDVKETVEAMCIVEATRSA 5jqb B 2.68 BS01 IBP B 1 Y517 M548 Y16 M47 ? remove_due_to_license_issue Q05320 27362232 706 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPHDWTKNITDKIDQIIHDFVD 5jrq A 2.287 BS01 6N9 A 1 I463 V471 A481 K483 L514 T529 W531 C532 S535 F583 D594 F595 G596 I17 V25 A35 K37 L68 T83 W85 C86 S89 F137 D148 F149 G150 D576 K578 N580 N581 D594 D130 K132 N134 N135 D148 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 27571413 801 FDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATEKSRSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAR 5jrq B 2.287 BS01 6N9 B 1 I463 V471 A481 K483 L514 T529 W531 C532 S535 F583 D594 F595 G596 I17 V23 A33 K35 L66 T81 W83 C84 S87 F135 D146 F147 G148 D576 K578 N580 N581 D594 D128 K130 N132 N133 D146 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 27571413 801 FDDWEIPDGQITVGQRIGSGSTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATEILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE 5jrs A 1.97 BS01 6MV A 1 L408 G409 T410 V416 A428 Y476 M477 G480 C481 N484 L528 L14 G15 T16 V22 A34 Y82 M83 G86 C87 N90 L130 D521 A523 R525 N526 D539 F559 D123 A125 R127 N128 D141 F161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4nM remove_due_to_license_issue IC50=30nM Q06187 27531604 4000 MEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMD 5js3 E 1.16 BS06 6MG E 1 N112 A113 H142 E143 H146 Y157 E166 L202 R203 H231 N112 A113 H142 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.185uM remove_due_to_license_issue P00800 27933956 411 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5jsg A 2.5 BS01 6P9 A 1 H60 W62 W72 Y91 Y98 L100 F141 W151 Y170 D173 F251 H14 W16 W26 Y45 Y52 L54 F95 W105 Y124 D127 F184 ? 0007276 Kd=14.2uM remove_due_to_license_issue Q9Y657 28504676 301 HGSRRNIVGCRIQHGWKEGNGPVTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELNKDERVSALEVLPDRVATSRISDAHLADTMIGKAVEHMFETEDGSKDEWRGMVLARAPVMNTWFYITYEKDPVLYMYQLLDDYKEGDLRIMPDSLVGKQVEYAKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLV 5jsj A 2.348 BS01 6PD A 1 W62 W72 Y91 F94 C96 Y98 F141 W151 D173 Y177 Y179 H252 W14 W24 Y43 F46 C48 Y50 F93 W103 D125 Y129 Y131 H188 ? 0007276 Kd=4uM remove_due_to_license_issue Kd=4000nM Q9Y657 28504676 301 SRRNIVGCRIQHGWKEGNGPVTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELNKDERVSALEVLPDRVATSRISDAHLADTMIGKAVEHMFETEDGSKDEWRGMVLARAPVMNTWFYITYEKDPVLYMYQLLDDYKEGDLRIMPDSLVGKQVEYAKEDGSKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLV 5jsm A 2.19 BS01 6NB B 1 Q461 I463 V471 A481 K483 L514 F516 T529 Q530 W531 C532 S535 H539 F583 D594 F595 G596 Q17 I19 V27 A37 K39 L70 F72 T85 Q86 W87 C88 S91 H95 F139 D150 F151 G152 D576 K578 N580 N581 D594 S616 D132 K134 N136 N137 D150 S160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 27571413 801 SEFDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATEKSGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAREL 5jsm B 2.19 BS01 6NB B 1 I463 V471 A481 K483 L514 F516 T529 Q530 W531 C532 S535 H539 F583 D594 F595 G596 I20 V28 A38 K40 L71 F73 T86 Q87 W88 C89 S92 H96 F140 D151 F152 G153 D576 K578 N580 N581 D594 S616 D133 K135 N137 N138 D151 S161 2.7.11.1 0004672,0005524,0006468 ic50=260nM remove_due_to_license_issue P15056 27571413 801 GSEFDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATEKSRSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAREL 5jsq A 1.503 BS01 6MS A 1 L53 E113 I115 D117 T118 A119 T121 K145 F166 V167 D173 L49 E87 I89 D91 T92 A93 T95 K119 F140 V141 D147 E113 D114 D117 F166 R179 E87 D88 D91 F140 R153 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=21.3uM remove_due_to_license_issue Q07010 27786284 301 CKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRDIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGKEL 5jss E 1.19 BS06 6NG E 1 N112 A113 F114 H142 E143 H146 E166 L202 R203 H231 N112 A113 F114 H142 E143 H146 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.354uM remove_due_to_license_issue P00800 27933956 406 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5jt2 A 2.702 BS01 6NC A 1 V471 A481 K483 L514 T529 Q530 W531 C532 S535 F583 D594 F595 G596 V28 A38 K40 L71 T86 Q87 W88 C89 S92 F140 D151 F152 G153 D576 K578 N580 N581 D594 S616 D133 K135 N137 N138 D151 S162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 27571413 802 GSEFDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATEKSRWSILWMAPEVIPYSFQSDVYAFGIVLYELMTGQLPYSNINDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAR 5jt2 B 2.702 BS01 6NC A 1 I463 A481 K483 L514 T529 W531 C532 S535 H539 F583 D594 F595 G596 I17 A35 K37 L64 T79 W81 C82 S85 H89 F133 D144 F145 G146 D576 K578 N580 N581 D594 S616 D126 K128 N130 N131 D144 S150 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P15056 27571413 802 FDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATSILWMAPEVIRMSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAR 5jt9 E 1.26 BS06 7AF E 1 N112 A113 F114 H142 E143 H146 E166 L202 R203 H231 N112 A113 F114 H142 E143 H146 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.233uM remove_due_to_license_issue P00800 27933956 412 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5jur A 2.93 BS01 6NS A 1 F23 F25 H57 E61 F63 K76 F104 Q106 M131 F3 F5 H37 E41 F43 K56 F84 Q86 M98 ? remove_due_to_license_issue Q30NP1 28197322 4000 SSFSFGGFTFKRTSGSSIKREEEVLTGNLQTLKIRVHEGYEEFTMVGKRATAILRKATRRLVQLIVSGKDEQSIAEAIIVAMVFSQEDCMIKAVRNPMHQLLRHFQKDAKVLFQNWGIEHIDNVMGMVGVLPDMTPSTEMSMRGIRVSKM 5juz F 2.4 BS01 YL4 F 1 K57 N59 F206 F239 D243 L344 K44 N46 F192 F225 D229 L330 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=3uM remove_due_to_license_issue IC50=3000nM P14324 28208018 403 YAQEKQDFVQHFSQIVRVLTEHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv0 F 2.4 BS01 YL5 F 1 N59 F206 F239 Q242 L246 L344 K347 N52 F197 F230 Q233 L237 L335 K338 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.1uM remove_due_to_license_issue IC50=1100nM P14324 28208018 403 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv0 F 2.4 BS02 YL5 F 2 L71 V72 E73 P74 A217 I219 P335 L64 V65 E66 P67 A208 I210 P326 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.1uM remove_due_to_license_issue IC50=1100nM P14324 28208018 404 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv0 F 2.4 BS03 YL5 F 3 Y322 Y349 K350 Y313 Y340 K341 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.1uM remove_due_to_license_issue IC50=1100nM P14324 28208018 405 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv1 F 2.3 BS01 YL6 F 1 K57 N59 R60 S205 F206 F239 Q242 D243 K45 N47 R48 S191 F192 F225 Q228 D229 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=0.86uM remove_due_to_license_issue P14324 28208018 403 VYAQEKQDFVQHFSQIVRVLTEHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv1 F 2.3 BS02 YL6 F 2 E319 Y322 A345 R346 Y349 K350 E305 Y308 A331 R332 Y335 K336 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=0.86uM remove_due_to_license_issue P14324 28208018 404 VYAQEKQDFVQHFSQIVRVLTEHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv2 F 2.3 BS02 6O3 F 1 N59 F239 L344 K347 N45 F224 L325 K328 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50~100uM remove_due_to_license_issue P14324 28208018 404 YAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv2 F 2.3 BS03 6O3 F 2 Y322 R346 Y303 R327 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50~100uM remove_due_to_license_issue P14324 28208018 405 YAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jvi E 1.12 BS06 6QC E 1 N112 A113 F114 H142 E143 H146 E166 L202 R203 H231 N112 A113 F114 H142 E143 H146 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.31uM remove_due_to_license_issue P00800 27933956 411 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5jxn E 1.38 BS06 6NN E 1 N112 A113 E143 H146 Y157 E166 L202 R203 H231 N112 A113 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.388uM remove_due_to_license_issue P00800 27933956 411 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5jxq A 1.2 BS02 6OK A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 C281 V282 D93 Y97 D143 C145 G216 L218 A219 M247 G248 C268 V269 D102 D280 C318 C320 C323 H349 D93 D267 C305 C307 C310 H336 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Ki=7nM remove_due_to_license_issue P28720 27501913 405 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSLTKQSEEGVTFKSHSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 5jy3 A 2.4 BS01 6OX A 1 F271 L274 A275 S278 E281 M312 T316 R319 F329 F340 F349 I353 F41 L44 A45 S48 E51 M82 T86 R89 F99 F110 F119 I123 ? 0003677,0004879,0006629 Ki=12nM remove_due_to_license_issue EC50=11.0nM, Ki=12nM P55055 27994765 501 QLTAAQELMIQQLVAAQLQCNKRPKVTPWPRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWD 5jyo D 2.098 BS01 63J D 1 K320 L321 F322 L323 E325 Y394 K100 L101 F102 L103 E105 Y174 S286 K289 Y414 Y466 V484 S69 K72 Y194 Y246 V264 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=5.0nM, Kd=92nM O94925 27462863 601 GSMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 5jyp A 2.74 BS01 ZBS A 1 K320 L321 F322 L323 Y394 K97 L98 F99 L100 Y171 S286 K289 Y414 Y466 V484 S68 K71 Y191 Y243 V261 3.5.1.2 0004359,0006541 remove_due_to_license_issue IC50=<100nM O94925 27462863 601 SMIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTVDGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYD 5jyy A 2.1 BS02 6PY A 1 R37 E38 D70 R71 W98 I142 E147 A166 E196 K212 R290 Y324 R37 E38 D70 R71 W98 I142 E147 A166 E196 K212 R290 Y324 D70 E197 K212 R290 Y324 D70 E197 K212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue R4NFR6 27341624 513 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCKDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 5jz9 A 2.68 BS01 6OR A 1 G44 G45 G46 S114 G154 L158 F173 M177 V243 H269 W270 G38 G39 G40 S108 G148 L152 F167 M171 V237 H263 W264 G45 G46 G48 N113 S114 L115 R192 D241 H269 W270 G39 G40 G42 N107 S108 L109 R186 D235 H263 W264 3.7.1.17,3.7.1.8 0005515,0005886,0006694,0009274,0016042,0016787,0018774,0034820,0051701,0102296 remove_due_to_license_issue P9WNH5 28380256 301 LTFESTSRFAEVDVDGPLKLHYHEAGVGNDQTVVLLHGGGPGAASWTNFSRNIAVLARHFHVLAVDQPGYGHSDKRAEHGQFNRYAAMALKGLFDQLGLGRVPLVGNSLGGGTAVRFALDYPARAGRLVLMGPGGLSINLFAPDPTEGVKRLSKFSVAPTRENLEAFLRVMVYDKNLITPELVDQRFALASTPESLTATRAMGKSFAGADFEAGMMWREVYRLRQPVLLIWGREDRVNPLDGALVALKTIPRAQLHVFGQCGHWVQVEKFDEFNKLTIEFLGGG 5jzb A 2.102 BS01 6OT A 1 G45 G46 S114 L115 G140 L158 N244 G39 G40 S108 L109 G134 L152 N238 G45 G46 G48 N113 S114 L115 R192 D241 H269 W270 G39 G40 G42 N107 S108 L109 R186 D235 H263 W264 3.7.1.17,3.7.1.8 0005515,0005886,0006694,0009274,0016042,0016787,0018774,0034820,0051701,0102296 ic50=0.41mM remove_due_to_license_issue P9WNH5 28380256 301 LTFESTSRFAEVDVDGPLKLHYHEAGVGNDQTVVLLHGGGPGAASWTNFSRNIAVLARHFHVLAVDQPGYGHSDKRAEHGQFNRYAAMALKGLFDQLGLGRVPLVGNSLGGGTAVRFALDYPARAGRLVLMGPGGLSINLFAPDPTEGVKRLSKFSVAPTRENLEAFLRVMVYDKNLITPELVDQRFALASTPESLTATRAMGKSFAGADFEAGMMWREVYRLRQPVLLIWGREDRVNPLDGALVALKTIPRAQLHVFGQCGHWVQVEKFDEFNKLTIEFLG 5jzn A 2.85 BS01 GUI A 1 V404 K419 V468 G471 L518 V26 K41 V90 G93 L140 D511 K513 E515 N516 D533 T550 D133 K135 E137 N138 D155 T172 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O15075 27545623 701 GFQIPATITERYKVGRTIGDGNFAVVKECVERSTAREYALKIIKKSKCRGKEHMIQNEVSILRRVKHPNIVLLIEEMDVPTELYLVMELVKGGDLFDAITSTNKYTERDASGMLYNLASAIKYLHSLNIVHRDIKPENLLVYEHQDGSKSLKLGDFGLATIVDGPLYTVCGTPTYVAPEIIAETGYGLKVDIWAAGVITYILLCGFPPFRGSDQEVLFDQILMGQVDFPSPYWDNVSDSAKELITMMLLVDVDQRFSAVQVLEHPWVN 5jzs B 2.27 BS01 FGZ B 1 G45 S114 G154 V155 L158 V243 G39 S108 G148 V149 L152 V237 G45 G46 G48 N113 S114 L115 R192 D241 H269 W270 G39 G40 G42 N107 S108 L109 R186 D235 H263 W264 3.7.1.17,3.7.1.8 0005515,0005886,0006694,0009274,0016042,0016787,0018774,0034820,0051701,0102296 ic50=0.54mM remove_due_to_license_issue P9WNH5 28380256 1000 LTFESTSRFAEVDVDGPLKLHYHEAGVGNDQTVVLLHGGGPGAASWTNFSRNIAVLARHFHVLAVDQPGYGHSDKRAEHGQFNRYAAMALKGLFDQLGLGRVPLVGNSLGGGTAVRFALDYPARAGRLVLMGPGGLSINLFAPDPTEGVKRLSKFSVAPTRENLEAFLRVMVYDKNLITPELVDQRFALASTPESLTATRAMGKSFAGADFEAGMMWREVYRLRQPVLLIWGREDRVNPLDGALVALKTIPRAQLHVFGQCGHWVQVEKFDEFNKLTIEFLGGG 5k00 A 1.77 BS01 6PV A 1 A38 K40 L61 L64 C70 L86 Y88 C89 G92 E93 L139 I149 D150 F151 A35 K37 L58 L61 C67 L83 Y85 C86 G89 E90 L136 I146 D147 F148 D132 K134 E136 N137 D150 S171 D129 K131 E133 N134 D147 S155 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=7nM remove_due_to_license_issue Q14680 28186750 401 MDYDELLKYYELHETIGTGAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARG 5k03 A 1.81 BS01 6P4 A 1 Y68 M89 E90 I91 A118 S119 H142 W143 Y66 M87 E88 I89 A116 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k05 A 2.14 BS01 6P5 A 1 G66 Y68 M89 E90 I91 A118 S119 Q120 H142 W143 R146 G64 Y66 M87 E88 I89 A116 S117 Q118 H140 W141 R144 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k07 A 2.0 BS01 dna B 0 K24 W26 L28 A29 P30 K31 Y49 R51 K21 W23 L25 A26 P27 K28 Y46 R48 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 27685992 101 ~ 108 GKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 5k07 A 2.0 BS02 dna C 0 V36 R51 K53 V33 R48 K50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 27685992 109 ~ 116 GKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 5k09 A 2.7 BS01 6PQ A 1 M89 E90 I91 S119 H142 W143 M88 E89 I90 S118 H141 W142 D141 K144 D169 N170 E199 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 27685665 301 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSD 5k0b A 2.36 BS01 6PS A 1 M40 G66 M89 E90 I91 S119 H142 W143 M38 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k0c A 1.95 BS01 6OZ A 1 G66 Y68 M89 E90 I91 A118 S119 H142 W143 G65 Y67 M88 E89 I90 A117 S118 H141 W142 D141 K144 D169 N170 E199 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 27685665 304 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k0f A 1.81 BS01 6P1 A 1 G66 M89 E90 I91 S119 H142 W143 G65 M88 E89 I90 S118 H141 W142 D141 K144 D169 N170 E199 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 ic50=0.47uM remove_due_to_license_issue P22734 27685665 302 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSPDK 5k0h A 2.2 BS03 6PK A 1 E97 T98 Y99 R143 E147 F174 D189 A190 C191 Q192 S195 V213 W215 G216 G219 C220 E83 T84 Y85 R132 E135 F162 D179 A180 C181 Q182 S185 V203 W205 G206 G208 C209 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 remove_due_to_license_issue Ki=29nM P00742 16848746 303 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 5k0i A 1.3 BS01 6PW A 1 Y130 Q134 Y126 Q130 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=0.002uM remove_due_to_license_issue IC50=2.0nM O14684 27554445 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5k0j A 1.94 BS01 6P2 A 1 M40 G66 Y68 M89 E90 I91 S119 H142 W143 M39 G65 Y67 M88 E89 I90 S118 H141 W142 D141 K144 D169 N170 E199 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 remove_due_to_license_issue P22734 27685665 302 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSPDKS 5k0m A 1.83 BS01 6PU A 1 P95 F97 Y148 E238 L240 D310 Y365 R367 R414 D430 P14 F16 Y67 E157 L159 D229 Y284 R286 R333 D349 ? remove_due_to_license_issue O75530 28135237 501 FKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5k0s A 2.45 BS01 0OU A 1 A11 I12 Y14 D51 H53 G54 F213 M227 Y228 V229 D232 A233 H269 A9 I10 Y12 D49 H51 G52 F211 M225 Y226 V227 D230 A231 H267 I12 H20 H23 D51 S128 D131 G150 W230 I265 I10 H18 H21 D49 S126 D129 G148 W228 I263 6.1.1.10 0000166,0004812,0004825,0005524,0005737,0006412,0006418,0006431 ic50=0.006uM remove_due_to_license_issue P59078 27500735 601 REKYYITTAIAYPNGKPHIGHAYELIATDAMARFQRLNGMDVYFLTGTDEHGIKMLQSARKEGITPRDLADRNTSAFRRMAEVLNSSNDDYIRTSEERHYKASQAIWQAMVANGDIYKGGYAGWYSVRDEAYYGEEETEVRADGVRYGPQGTPVEWVEEESYFFRLSAYQDKLLDLYENNPGFIMPAERRNEIVSFVKSGLKDLSISRTTFDWGIPVPGDEKHVMYVWVDALTNYITALGYPDTTDERWAYWPANAHIIGKDISRFHAVYWPAFLMSAQLPLPKRVFAHGFLFNRIDPFELVERYGLDQLRYFLMREVPFGQDGSYSHEAIVNRTNADLANDLGNLAQRSLSMIAKNCEGKVPQPGAFSEADKAILDQADAALETARKAMDDQALHLALGAIFAVVAEANRYFAGQEPWALRKTDPARMGTVLYVTAEVLRRVGIMVQPFIPQSAEKLLDILAVPADKRQFADVLASPLAGGTDLPAPQPVFPRYV 5k0t A 2.6 BS01 415 A 1 I12 Y14 D51 H53 G54 Y228 V229 W230 A233 I265 F268 H269 I11 Y13 D50 H52 G53 Y227 V228 W229 A232 I264 F267 H268 I12 H20 H23 D51 S128 D131 G150 W230 I265 I11 H19 H22 D50 S127 D130 G149 W229 I264 6.1.1.10 0000166,0004812,0004825,0005524,0005737,0006412,0006418,0006431 remove_due_to_license_issue P59078 27500735 601 SREKYYITTAIAYPNGKPHIGHAYELIATDAMARFQRLNGMDVYFLTGTDEHGIKMLQSARKEGITPRDLADRNTSAFRRMAEVLNSSNDDYIRTSEERHYKASQAIWQAMVANGDIYKGGYAGWYSVRDEAYYGEEETEVRADGVRYGPQGTPVEWVEEESYFFRLSAYQDKLLDLYENNPGFIMPAERRNEIVSFVKSGLKDLSISRTTFDWGIPVPGDEKHVMYVWVDALTNYITALGYPDTTDERWAYWPANAHIIGKDISRFHAVYWPAFLMSAQLPLPKRVFAHGFLFNRIDPFELVERYGLDQLRYFLMREVPFGQDGSYSHEAIVNRTNADLANDLGNLAQRSLSMIAKNCEGKVPQPGAFSEADKAILDQADAALETARKAMDDQALHLALGAIFAVVAEANRYFAGQEPWALRKTDPARMGTVLYVTAEVLRRVGIMVQPFIPQSAEKLLDILAVPADKRQFADVLASPLAGGTDLPAPQPVFPRY 5k0x A 2.231 BS01 K0X A 1 L593 A617 L671 F673 M674 K675 N728 M730 D741 L18 A39 L85 F87 M88 K89 N142 M144 D155 D723 A725 R727 N728 D741 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 ic50=4.4nM remove_due_to_license_issue IC50=<10nM Q12866 28032464 904 KLEDVVIDRNLLILGKILGEGSVMEGNLKQEDGTSLKVAVKTMKLDNSSQIEEFLSEAACMKDFSHPNVIRLLGVCIEPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFGPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESLPD 5k13 A 1.85 BS01 6Q7 A 1 W225 F228 S232 C235 L266 L269 I270 I273 F286 S287 G301 F302 V395 P407 W45 F48 S52 C55 L86 L89 I90 I93 F106 S107 G121 F122 V215 P227 ? 0003677,0004879,0005634,0006355,0048384 Ki=1.8nM remove_due_to_license_issue Ki=1.8nM P10276 27261179 501 TPEVGELIEKVRKAHQETFPALCQLGKYTTNNSSEQRVSLDIDLWDKFSELSTKCIIKTVEFAKQLPGFTTLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFAFANQLLPLEMDDAETGLLSAICLICGDRQDLEQPDRVDMLQEPLLEALKVYVRKRRPSRPHMFPKMLMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLE 5k17 A 2.1 BS01 dna C 0 K24 W26 L28 A29 P30 K31 Y49 R51 K23 W25 L27 A28 P29 K30 Y48 R50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 27685992 101 ~ 108 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 5k17 A 2.1 BS02 dna D 0 P30 V36 R51 H52 K53 P29 V35 R50 H51 K52 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 27685992 109 ~ 116 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 5k17 B 2.1 BS01 dna E 0 K24 W26 L28 A29 P30 K31 Y49 R51 K23 W25 L27 A28 P29 K30 Y48 R50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 27685992 101 ~ 108 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 5k17 B 2.1 BS02 dna F 0 P30 V36 R51 H52 K53 P29 V35 R50 H51 K52 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 27685992 109 ~ 116 SSGKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 5k1d A 1.94 BS01 5GP A 1 S65 L120 Q121 Y151 I292 L293 T313 G314 S315 I343 S67 L122 Q123 Y153 I294 L295 T313 G314 S315 I343 S65 K68 M107 E109 F122 Y151 G157 E272 K312 S315 S67 K70 M109 E111 F124 Y153 G159 E274 K312 S315 3.5.2.6 0000166,0008800,0016787,0017001,0030288,0046677,0046872 Ki=20.8uM remove_due_to_license_issue Q99QC1 28242658 401 HHGEASPVDPLRPVVDASIQPLLKEHRIPGMAVAVLKDGKAHYFNYGVANRESGAGVSEQTLFEIGSVSKTLTATLGAYAVVKGAMQLDDKASRHAPWLKGSAFDSITMGELATYSAGGLPLQFPEEVDSSEKMRAYYRQWAPVYSPGSHRQYSNPSIGLFGHLAASSLKQPFAPLMEQTLLPGLGMHHTYVNVPKQAMASYAYGYSKEDKPIRVNPGMLADEAYGIKTSSADLLRFVKANIGGVDDKALQQAISLTHQGHYSVGGMTQGLGWESYAYPVTEQTLLAGNSAKVILEANPTAAPRESQVLFNKTGSTNGFGAYVAFVPARGIGIVMLANRNYPIEARIKAAHAILAQLAG 5k1f A 1.94 BS01 IMP A 1 S65 L120 Q121 Y151 I292 T313 G314 S315 I343 S67 L122 Q123 Y153 I294 T313 G314 S315 I343 S65 K68 M107 E109 F122 Y151 G157 E272 K312 S315 S67 K70 M109 E111 F124 Y153 G159 E274 K312 S315 3.5.2.6 0000166,0008800,0016787,0017001,0030288,0046677,0046872 Ki=16.2uM remove_due_to_license_issue Q99QC1 28242658 401 HHGEASPVDPLRPVVDASIQPLLKEHRIPGMAVAVLKDGKAHYFNYGVANRESGAGVSEQTLFEIGSVSKTLTATLGAYAVVKGAMQLDDKASRHAPWLKGSAFDSITMGELATYSAGGLPLQFPEEVDSSEKMRAYYRQWAPVYSPGSHRQYSNPSIGLFGHLAASSLKQPFAPLMEQTLLPGLGMHHTYVNVPKQAMASYAYGYSKEDKPIRVNPGMLADEAYGIKTSSADLLRFVKANIGGVDDKALQQAISLTHQGHYSVGGMTQGLGWESYAYPVTEQTLLAGNSAKVILEANPTAAPRESQVLFNKTGSTNGFGAYVAFVPARGIGIVMLANRNYPIEARIKAAHAILAQLA 5k1i A 2.61 BS01 6PT A 1 Y159 M273 N321 W332 I336 F340 M357 S368 F372 Y73 M187 N232 W243 I247 F251 M268 S279 F283 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 27933955 1001 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 5k1v A 2.897 BS02 6PX A 1 D198 E200 P333 G334 A335 E337 H370 E371 H374 E393 D451 E452 Y455 Y892 D145 E147 P280 G281 A282 E284 H317 E318 H321 E340 D398 E399 Y402 Y828 E337 H370 E371 H374 E393 Q447 Y455 E284 H317 E318 H321 E340 Q394 Y402 3.4.11.- 0002250,0002474,0004175,0004177,0005515,0005615,0005737,0005783,0005788,0005789,0006508,0008217,0008237,0008270,0016020,0019885,0042277,0043171,0046872,0070006 remove_due_to_license_issue IC50=518nM Q6P179 28337326 1002 PVATNGERFPWQELRLPSVVIPLHYDLFVHPNLTSLDFVASEKIEVLVSNATQFIILHSKDLEITNATLQSEEDSRYMKPGKELKVLSYPAHEQIALLVPEKLTPHLKYYVAMDFQAKLGDGFEGFYKSTYRTLGGETRILAVTDFEPTQARMAFPCFDEPLFKANFSIKIRRESRHIALSNMPKVKTIELEGGLLEDHFETTVKMSTYLVAYIVCDFHSLSGFTSSGVKVSIYASPDKRNQTHYALQASLKLLDFYEKYFDIYYPLSKLDLIAIPDFAPGAMENWGLITYRETSLLFDPKTSSASDKLWVTRVIAHELAHQWFGNLVTMEWWNDIWLKEGFAKYMELIAVNATYPELQFDDYFLNVCFEVITKDSLNSSRPISKPAETPTQIQEMFDEVSYNKGACILNMLKDFLGEEKFQKGIIQYLKKFSYRNAKNDDLWSSLSNSCGVCHSMTSNMLAFLGENAEVKEMMTTWTLQKGIPLLVVKQDGCSLRLQQERFLQGVFQEDPEWRALQERYLWHIPLTYSTSSSNVIHRHILKSKTDTLDLPEKTSWVKFNVDSNGYYIVHYEGHGWDQLITQLNQNHTLLRPKDRVGLIHDVFQLVGAGRLTLDKALDMTYYLQHETSSPALLEGLSYLESFYHMMDRRNISDISENLKRYLLQYFKPVIDRQSWSDKGSVWDRMLRSALLKLACDLNHAPCIQKAAELFSQWMESSGKLNIPTDVLKIVYSVGAQTTAGWNYLLEQYELSMSSAEQNKILYALSTSKHQEKLLKLIELGMEGKVIKTQNLAALLHAIARRPKGQQLAWDFVRENWTHLLKKFDLGSYDIRMIISGTTAHFSSKDKLQEVKLFFESLEAQGSHLDIFQTVLETITKNIKWLEKNLPTLRTWLMVNTRHH 5k32 A 1.99 BS02 6Q2 A 1 Y159 D318 N321 F340 Q369 F372 Y72 D231 N234 F253 Q280 F283 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 29502405 1003 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 5k48 A 1.744 BS01 S5Z A 1 Y67 D118 H179 N210 H240 Y36 D87 H148 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue Q9K2N0 29271657 301 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5k4i A 1.76 BS01 6QB A 1 I31 E33 G34 G37 V39 A52 K54 Q105 M108 E109 K114 N154 L156 C166 D167 I23 E25 G26 G29 V31 A44 K46 Q97 M100 E101 K106 N146 L148 C158 D159 D149 K151 S153 N154 D167 T190 D141 K143 S145 N146 D159 T168 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=3.1nM remove_due_to_license_issue IC50=3.1nM, Kd=1.6nM P28482 27227380 401 AGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADTRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5k4j A 1.6 BS01 6QB A 1 E12 G13 Y15 G16 V18 A31 K33 F82 L83 H84 N132 L134 D145 E13 G14 Y16 G17 V19 A32 K34 F76 L77 H78 N126 L128 D139 D127 K129 Q131 N132 D145 T165 D121 K123 Q125 N126 D139 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 27227380 301 AMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5k4l A 3.179 BS04 6QN A 1 Y472 S478 F480 H483 H571 Y284 S290 F292 H295 H383 G465 Y472 H483 E485 H571 A583 G277 Y284 H295 E297 H383 A395 1.14.11.67 0003677 remove_due_to_license_issue IC50=50nM P29375 27499454 904 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRVRLDFLDQLAKFWELQGSTLKIPVVERKILDLYALSKIVASKGGFEMVTKEKKWSKVGSRLGYLPGKGTGSLLKSHYERILYPYELFQSGVSLMGVQMYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINVDISGMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCTADWLPIGRQCVNHYRRLRRHCVFSHEELIFKMAADPECLDVGLAAMVCKELTLMTEEETRLRESVVQMGVLMSEEEVFELVPDDERQCSACRTTCFLSALTCSCNPERLVCLYHPTDLCPCPMQKKCLRYRYPLEDLPSLLYGVKVRAQSYDTWVSVMLEDAEDRKYPENDLFRKLR 5k4x A 1.37 BS01 6Q9 A 1 A145 V195 M284 G285 A131 V181 M270 G271 1.1.1.205 0003824,0003938,0006164,0016491 ic50=0.38uM remove_due_to_license_issue G7CNL4 27704782 401 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 5k4z A 1.64 BS02 6Q8 A 1 T144 A145 N149 V195 M284 G285 E318 T130 A131 N135 V181 M270 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 Kd=0.7uM remove_due_to_license_issue G7CNL4 27704782 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAGL 5k51 A 2.956 BS01 6QD A 1 D117 T118 A119 T121 F166 V167 D87 T88 A89 T91 F136 V137 E113 D114 D117 F166 R179 E83 D84 D87 F136 R149 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 remove_due_to_license_issue Q07010 27786284 301 YDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGK 5k5e A 2.8 BS01 6QS A 1 W82 G115 G116 G117 E197 P285 F329 Y332 H438 W80 G113 G114 G115 E195 P283 F327 Y330 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue IC50=443nM P06276 27405689 609 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5k5h A 3.108 BS01 dna B 0 Y358 K365 R368 H369 Y386 R389 K393 R396 Q418 T421 H425 K429 R448 Y9 K16 R19 H20 Y37 R40 K44 R47 Q69 T72 H76 K80 R99 ? remove_due_to_license_issue P49711 28529057 1 ~ 13 PFKCSMCDYASVEVSKLKRHIRSHTGERPFQCSLCSYASRDTYKLKRHMRTHSGEKPYECYICHARFTQSGTMKMHILQKHTENVAKFHCPHCDTVIARKSDLGVHLRKQH 5k5h A 3.108 BS02 dna C 0 Y392 K395 Y407 S419 K423 K449 S450 R457 Y43 K46 Y58 S70 K74 K100 S101 R108 ? remove_due_to_license_issue P49711 28529057 3 ~ 15 PFKCSMCDYASVEVSKLKRHIRSHTGERPFQCSLCSYASRDTYKLKRHMRTHSGEKPYECYICHARFTQSGTMKMHILQKHTENVAKFHCPHCDTVIARKSDLGVHLRKQH 5k5n A 2.2 BS01 6QH A 1 I62 A83 K85 L132 Y134 V135 P136 R141 L188 D200 I24 A45 K47 L85 Y87 V88 P89 R94 L141 D153 D181 K183 N186 D200 S219 D134 K136 N139 D153 S172 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=9nM remove_due_to_license_issue P49841 27355874 4001 KVTTVVATPGDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQNRELQIMRKLDHCNIVRLRYFFYSSDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 5k5s A 2.6 BS01 TRP A 1 R66 W70 S147 A168 S169 S170 Y218 E297 A298 R47 W51 S113 A134 S135 S136 Y184 E263 A264 ? 0004930,0007186,0016020 remove_due_to_license_issue P41180 27434672 701 YGPDQRAQKKGDIILGGLFPIHFGVAAKDQDLKSRPESVECIRYNFRGFRWLQAMIFAIEEINSSPALLPNLTLGYRIFDTCNTVSKALEATLSFVAQNKIPSTIAVVGATGSGVSTAVANLLGLFYIPQVSYASSSRLLSNKNQFKSFLRTIPNDEHQATAMADIIEYFRWNWVGTIAADDDYGRPGIEKFREEAEERDICIDFSELISQYSDEEEIQHVVEVIQNSTAKVIVVFSSGPDLEPLIKEIVRRNITGKIWLASEAWASSSLIAMPQYFHVVGGTIGFALKAGQIPGFREFLKKVHPRKSVHNGFAKEFWEETFNCHPLCTGDENINSVETPYIDYTHLRISYNVYLAVYSIAHALQDIYTCLPGRGLFTNGSCADIKKVEAWQVLKHLRHLQFTNNMGEQVTFDECGDLVGNYSIINWHLSPEDGSIVFKEVGYYNVYAKKGERLFINEEKILWSGFSREVPFSNCSRDCLAGTRKGIIEGEPTCCFECVECPDGEYSDETDASACNKCPDDFWSNENHTSC 5k6a A 1.7 BS02 6QT A 1 S95 F97 Y174 V206 P210 W221 S94 F96 Y154 V186 P190 W201 R14 D161 Y174 K178 R13 D141 Y154 K158 ? 0000166,0016491,0047040 ic50=31uM remove_due_to_license_issue O76290 28282886 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5k6a D 1.7 BS02 6QT D 1 S95 F97 Y174 V206 P210 W221 S94 F96 Y154 V186 P190 W201 R14 D161 Y174 K178 R13 D141 Y154 K158 ? 0000166,0016491,0047040 ic50=31uM remove_due_to_license_issue O76290 28282886 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 5k76 A 2.74 BS01 6R1 A 1 M192 V200 A211 K213 Y262 V263 Y264 M265 D272 L318 M26 V30 A41 K43 Y82 V83 Y84 M85 D92 L138 D311 K313 A315 N316 D329 T351 D131 K133 A135 N136 D149 T165 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=5.0nM, Kd=0.700000nM Q9NWZ3 29172502 501 FHSFSFYELKNVTNNFDERPISGNKMGEVVYKGYVNNTTVAVKKLTEELKQQFDQEIKVMAKCQHENLVELLGFSSDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARATVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5k7h A 2.35 BS01 IVC A 1 W169 K172 W173 F174 K175 G178 R179 L180 W156 K159 W160 F161 K162 G165 R166 L167 ? 0000976,0003677,0003700,0006355 Kd=0.99uM remove_due_to_license_issue Q1D4I5 27940564 305 RYRAILETAARLICDRGYEGTSMQEIAAACRMTKAGLYHHIQNKEQLLFAIMNYGMDLFEEQVLSRVQDIANPVERLRACMRHNILLVTRGWSKEVIIILHEHATLTGETRAFIDARKKKYVDFLEEAFSQASQQGLIRPVDPTVGAFSFLGMVLWIYKWFKPDGRLTDEQIADGMVGMLFPPF 5k7h A 2.35 BS02 IVC B 1 M69 F72 K131 K132 F161 L168 M56 F59 K118 K119 F148 L155 ? 0000976,0003677,0003700,0006355 Kd=0.99uM remove_due_to_license_issue Q1D4I5 27940564 302 RYRAILETAARLICDRGYEGTSMQEIAAACRMTKAGLYHHIQNKEQLLFAIMNYGMDLFEEQVLSRVQDIANPVERLRACMRHNILLVTRGWSKEVIIILHEHATLTGETRAFIDARKKKYVDFLEEAFSQASQQGLIRPVDPTVGAFSFLGMVLWIYKWFKPDGRLTDEQIADGMVGMLFPPF 5k7h B 2.35 BS01 IVC A 1 F72 K131 K132 F161 F59 K118 K119 F148 ? 0000976,0003677,0003700,0006355 Kd=0.99uM remove_due_to_license_issue Q1D4I5 27940564 305 RYRAILETAARLICDRGYEGTSMQEIAAACRMTKAGLYHHIQNKEQLLFAIMNYGMDLFEEQVLSRVQDIANPVERLRACMRHNILLVTRGWSKEVIIILHEHATLTGETRAFIDARKKKYVDFLEEAFSQASQQGLIRPVDPTVGAFSFLGMVLWIYKWFKPDGRLTDEQIADGMVGMLFPPF 5k7h B 2.35 BS02 IVC B 1 W169 W173 F174 K175 G178 R179 L180 W156 W160 F161 K162 G165 R166 L167 ? 0000976,0003677,0003700,0006355 Kd=0.99uM remove_due_to_license_issue Q1D4I5 27940564 302 RYRAILETAARLICDRGYEGTSMQEIAAACRMTKAGLYHHIQNKEQLLFAIMNYGMDLFEEQVLSRVQDIANPVERLRACMRHNILLVTRGWSKEVIIILHEHATLTGETRAFIDARKKKYVDFLEEAFSQASQQGLIRPVDPTVGAFSFLGMVLWIYKWFKPDGRLTDEQIADGMVGMLFPPF 5k83 A 2.39 BS01 dna H 0 Y59 P60 K61 A62 H65 W94 S95 Y124 Y125 Y131 Y59 P60 K61 A62 H65 W94 S95 Y124 Y125 Y131 3.5.4.-,3.5.4.38 0003824 remove_due_to_license_issue M1GSK9 27480941 10 ~ 12 MKPQIRNMVEPMDPRTFVSNFNNRPILSGLDTVWLCCEVKTKDPSGPPLDAKIFQGKVYPKAKYHPEMRFLRWFHKWRQLHHDQEYKVTWYVSWSPCTRCANSVATFLAKDPKVTLTIFVARLYYFWKPDYQQALRILAEAGATMKIMNYNEFQDCWNKFVDGRGKPFKPWNNLPKHYTLLQATLGELLRH 5k83 C 2.39 BS01 dna I 0 Y59 P60 K61 A62 H65 W94 S95 Y124 Y125 Y59 P60 K61 A62 H65 W94 S95 Y124 Y125 3.5.4.-,3.5.4.38 0003824 remove_due_to_license_issue M1GSK9 27480941 10 ~ 12 MKPQIRNMVEPMDPRTFVSNFNNRPILSGLDTVWLCCEVKTKDPSGPPLDAKIFQGKVYPKAKYHPEMRFLRWFHKWRQLHHDQEYKVTWYVSWSPCTRCANSVATFLAKDPKVTLTIFVARLYYFWKPDYQQALRILAEAGATMKIMNYNEFQDCWNKFVDGRGKPFKPWNNLPKHYTLLQATLGELLRH 5k83 E 2.39 BS01 dna J 0 Y59 P60 K61 H65 W94 S95 Y124 Y125 Y59 P60 K61 H65 W94 S95 Y124 Y125 3.5.4.-,3.5.4.38 0003824 remove_due_to_license_issue M1GSK9 27480941 10 ~ 12 MKPQIRNMVEPMDPRTFVSNFNNRPILSGLDTVWLCCEVKTKDPSGPPLDAKIFQGKVYPKAKYHPEMRFLRWFHKWRQLHHDQEYKVTWYVSWSPCTRCANSVATFLAKDPKVTLTIFVARLYYFWKPDYQQALRILAEAGATMKIMNYNEFQDCWNKFVDGRGKPFKPWNNLPKHYTLLQATLGELLRH 5k8n A 3.225 BS01 6R6 A 1 I90 R373 I85 R368 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 501 DVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8n A 3.225 BS02 6R6 G 1 Y223 Y288 Y218 Y283 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 501 DVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8n G 3.225 BS01 6R6 A 1 Y223 R289 Y218 R284 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 501 DVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8n G 3.225 BS02 6R6 G 1 I90 N124 E158 R373 G395 I85 N119 E153 R368 G390 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 501 DVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8o A 2.893 BS02 6R7 A 1 I90 N124 E158 E196 M371 R373 G395 I87 N121 E155 E193 M368 R370 G392 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 502 SNDVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8o A 2.893 BS03 6R7 H 1 Y223 Y288 R289 Y220 Y285 R286 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 502 SNDVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8o H 2.893 BS01 6R7 A 1 Y223 Y288 R289 Y219 Y284 R285 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 502 NDVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8o H 2.893 BS03 6R7 H 1 I90 N124 E158 E196 M371 R373 G395 I86 N120 E154 E192 M367 R369 G391 3.5.99.8 0016787,0046872 remove_due_to_license_issue D3WZ85 27694799 502 NDVAKVMKTLDGMREGLIQTAVELGSIEAPTGREGAAGDYVYEWMARNGFGPERVGVFDDRFNVVGRLRGTGGGASLSFNSHLDTIMAREDTARFADANDRIYHEAWHEEGRIYGYSVVNCKGPMACWLIAAKALKEAGAALKGDVVLTAVCGEIDCEPVDEFQGHDYLAEDIGARYAISHGAISDYALVAEATNFKPAWVEAGKVFLKVTVFAGPSRYTPYVPRPVAALDSPNAIVRMAKLVEALEEWADNYEKRYTREYGGGTVVPKVAIGAIRGGVPYKIYRFPELCSIYMDIRLNPDTNPLVVQREVEAVVSKLGLKAEVKPFLFRRGYEAQGIEPLQNALEVAHREVVGRPTERPGSPECSMWRDTNPYNELGIPSLTYGCGGGAGGGNTYFLVDDMLKAAKVYAMTAMDLCNRTP 5k8s A 1.15 BS01 CMP A 1 I340 I366 Y369 F375 G376 E377 L378 A379 R386 A387 A388 I390 Y424 L428 I47 I73 Y76 F82 G83 E84 L85 A86 R93 A94 A95 I97 Y131 L135 2.7.11.11 Kd=6nM remove_due_to_license_issue Q7KQK0 27738107 501 GPGAKKRKMYEDILSHVNILKDMDPYERCKVADCLKSKSYNDGEIIIKEGEEGDTFFILIDGNAVASKDNKVIKTYTKGDYFGELALLKNKPRAATIKAQNFCQVVYLDRKSFKRLLGPIEDILHRNVENYKKVLNELGLDTTCID 5k8v A 2.25 BS01 6RE A 1 Y150 F151 Y154 G193 E215 A216 K242 E244 E258 M260 E267 M269 Y15 F16 Y19 G58 E80 A81 K107 E109 E123 M125 E132 M134 D166 E258 E267 H415 D31 E123 E132 H280 2.1.1.319 0016274,0018216 ic50=460nM remove_due_to_license_issue Q9WVG6 27879050 501 SVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 5k9w A 2.01 BS01 OTA A 1 Y46 D48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Y47 D49 K121 D182 F183 C216 S217 A218 I220 G221 R222 D181 C215 R221 S222 Q262 D182 C216 R222 S223 Q263 3.1.3.48 0004725,0006470,0016311 Kd=26uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 402 SMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHE 5ka1 A 1.84 BS01 OTA A 1 Y46 D48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Y48 D50 K122 D183 F184 C217 S218 A219 I221 G222 R223 D181 C215 R221 S222 Q262 D183 C217 R223 S224 Q264 3.1.3.48 0004725,0006470,0016311 Kd=33uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 301 ASMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIM 5ka3 A 2.141 BS01 OTA A 1 Y46 D48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Y45 D47 K119 D180 F181 C214 S215 A216 I218 G219 R220 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Kd=26uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 401 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSAATVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSH 5ka7 A 2.061 BS01 OTA A 1 Y46 D48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y47 D49 K121 D182 F183 C216 S217 A218 I220 G221 R222 Q263 D181 C215 R221 S222 Q262 D182 C216 R222 S223 Q263 3.1.3.48 0004725,0006470,0016311 Kd=45uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 303 SMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTAWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHE 5ka9 A 2.07 BS01 OTA A 1 Y46 D48 K120 C215 S216 A217 I219 G220 R221 Y51 D53 K125 C220 S221 A222 I224 G225 R226 D181 C215 R221 S222 Q262 D186 C220 R226 S227 Q267 3.1.3.48 0004725,0006470,0016311 Kd=39uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 307 GHMASMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFANFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKEL 5kab A 1.968 BS01 OTA A 1 Y46 D48 K120 C215 S216 A217 I219 G220 R221 Q262 Y46 D48 K120 C215 S216 A217 I219 G220 R221 Q262 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 306 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVGESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIM 5kad A 1.9 BS01 OTA A 1 Y46 D48 K120 D181 F182 C215 S216 A217 I219 G220 R221 Q262 Y50 D52 K124 D185 F186 C219 S220 A221 I223 G224 R225 Q266 D181 C215 R221 S222 Q262 D185 C219 R225 S226 Q266 3.1.3.48 0004725,0006470,0016311 Kd=37uM remove_due_to_license_issue IC50=500000nM, Ki=11500nM P18031 28212750 401 HMASMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLAFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFI 5kam A 2.481 BS01 IMP A 1 I115 K145 F166 V167 I81 K111 F132 V133 E113 D114 D117 F166 R179 E79 D80 D83 F132 R145 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=77.3uM remove_due_to_license_issue Q07010 27786284 3301 TSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVY 5kap A 2.95 BS01 6RH A 1 I115 D117 V167 I82 D84 V134 E113 D114 D117 F166 R179 E80 D81 D84 F133 R146 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 remove_due_to_license_issue Q07010 27786284 301 TSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVY 5kat A 2.101 BS01 P4P A 1 H117 I120 T127 V128 F133 M153 P154 H117 I120 T127 V128 F133 M153 P154 ? Kd=78.7uM remove_due_to_license_issue A0A0H3JRN6 27505298 201 MEYQLQQLASLTLVGIKETYENGRQAQQHIAGFWQRCYQEGVIADLQLKNNGDLAGILGLCIPELDGKMSYMIAVTGDNSADIAKYDVITLASSKYMVFEAQGAVPKAVQQKMEEVHHYIHQYQANTVKSAPFFELYQDGDTTSEKYITEIWMPVKGLEHHHHHH 5kau A 1.95 BS01 RHQ A 1 Q27 I30 A31 W34 Y38 V105 P106 V109 E135 Y137 Q27 I30 A31 W34 Y38 V105 P106 V109 E135 Y137 ? Kd=0.3uM remove_due_to_license_issue A0A0H3JRN6 27505298 201 MEYQLQQLASLTLVGIKETYENGRQAQQHIAGFWQRCYQEGVIADLQLKNNGDLAGILGLCIPELDGKMSYMIAVTGDNSADIAKYDVITLASSKYMVFEAQGAVPKAVQQKMEEVHHYIHQYQANTVKSAPFFELYQDGDTTSEKYITEIWMPVKGLEHHHHHH 5kax A 2.0 BS01 RHQ A 1 F35 E36 P57 Y106 Y135 L136 N138 P139 F35 E36 P57 Y106 Y135 L136 N138 P139 ? Kd=0.78uM remove_due_to_license_issue Q8KFZ1 27505298 201 MDFECQFVCELKELAPVPALLIRTQTTMSELGSLFEAGYHDILQLLAGQGKSPSGPPFARYFGMSAGTFEVEFGFPVEGGVEGSGRVVTGLTPSGKAASSLYIGPYGEIEAVYDALMKWVDDNGFDLSGEAYEIYLDNPAETAPDQLRTRVSLMLHES 5kbe A 2.5 BS02 IPH A 1 G102 P103 H106 F132 Y161 Y165 G88 P89 H92 F118 Y147 Y151 ? Kd=0.46uM remove_due_to_license_issue Q43965 27362503 602 EQNKDIQDLLDKIVFDAQHGQIWFDENRMLLMHTSILGFLRKDLYQMLGLERTKRFFIRCGYQAGMRDAEVTSKLRPNLNEAEAFMAGPQMHGIRGMVQVEVNELHLSHDLKQFYADFNWLNSFEAEVHLSEFGASDQPACWMLLGYACGYSSFVMGQTIIYQETHCVAQGDEHCRIIGKPLSEWDAVSDEIIALQAEL 5kbf A 2.0 BS01 CMP A 1 I236 L248 F257 G258 E259 L260 A261 R268 A269 A270 Y319 I77 L89 F98 G99 E100 L101 A102 R109 A110 A111 Y160 2.7.11.11 0001932,0005952,0008603 Kd=1.2nM remove_due_to_license_issue Q7KQK0 27738107 501 SVSANFIPKVYKKDEKEKAKIREALNESFLFNHLNKKEFEIIVNAFFDKNVEKGVNIINEGDYGDLLYVIDQGEVEIYKTKENNKKEVLTVLKSKDVFGELALLYNSKRAATATALTKCHLWALDRESFTYIIKDMVAKKRKMYEDILSHVNILKDMDPYERCKVADCLKSKSYNDGEIIIKEGEEGDTFFILIDGNAVASKDNKVIKTYTKGDYFGELALLKNKPRAATIKAQNFCQVVYLDRKSFKRLLGPIEDILHRNVENYKKVLNELGLDTTCIDEN 5kbf A 2.0 BS02 CMP A 2 I340 I366 Y369 F375 G376 E377 L378 A379 R386 A387 A388 I390 Y424 L428 I181 I207 Y210 F216 G217 E218 L219 A220 R227 A228 A229 I231 Y265 L269 2.7.11.11 0001932,0005952,0008603 Kd=1.2nM remove_due_to_license_issue Q7KQK0 27738107 502 SVSANFIPKVYKKDEKEKAKIREALNESFLFNHLNKKEFEIIVNAFFDKNVEKGVNIINEGDYGDLLYVIDQGEVEIYKTKENNKKEVLTVLKSKDVFGELALLYNSKRAATATALTKCHLWALDRESFTYIIKDMVAKKRKMYEDILSHVNILKDMDPYERCKVADCLKSKSYNDGEIIIKEGEEGDTFFILIDGNAVASKDNKVIKTYTKGDYFGELALLKNKPRAATIKAQNFCQVVYLDRKSFKRLLGPIEDILHRNVENYKKVLNELGLDTTCIDEN 5kbg A 2.8 BS02 JZ0 A 1 G102 P103 H106 F132 Y161 A162 Y176 G87 P88 H91 F117 Y146 A147 Y161 ? remove_due_to_license_issue Q43965 27362503 602 QNKDIQDLLDKIVFDAQHGQIWFDENRMLLMHTSILGFLRKDLYQMLGLERTKRFFIRCGYQAGMRDAEVTSKLRPNLNEAEAFMAGPQMHGIRGMVQVEVNELHLSHDLKQFYADFNWLNSFEAEVHLSEFGASDQPACWMLLGYACGYSSFVMGQTIIYQETHCVAQGDEHCRIIGKPLSEWEFMSPDAVSDEIIALQAEL 5kbh A 2.55 BS02 3CH A 1 G102 P103 H106 F132 A162 Y165 Y176 G88 P89 H92 F118 A148 Y151 Y162 ? remove_due_to_license_issue Q43965 27362503 602 EQNKDIQDLLDKIVFDAQHGQIWFDENRMLLMHTSILGFLRKDLYQMLGLERTKRFFIRCGYQAGMRDAEVTSKLRPNLNEAEAFMAGPQMHGIRGMVQVEVNELHLSHDLKQFYADFNWLNSFEAEVHLSEFGASDQPACWMLLGYACGYSSFVMGQTIIYQETHCVAQGDEHCRIIGKPLSEWENDAVSDEIIALQAELN 5kbi A 2.9 BS02 CAQ A 1 G102 P103 H106 F132 W134 Y161 G88 P89 H92 F118 W120 Y147 ? remove_due_to_license_issue Q43965 27362503 602 EQNKDIQDLLDKIVFDAQHGQIWFDENRMLLMHTSILGFLRKDLYQMLGLERTKRFFIRCGYQAGMRDAEVTSKLRPNLNEAEAFMAGPQMHGIRGMVQVEVNELHLSHDLKQFYADFNWLNSFEAEVHLSEFGASDQPACWMLLGYACGYSSFVMGQTIIYQETHCVAQGDEHCRIIGKPLSEWEPDAVSDEIIALQAELN 5kbq A 2.58 BS01 IPV A 1 I276 G277 Q278 V284 A297 K299 E315 V342 M344 Y346 L347 L396 T406 I23 G24 Q25 V31 A44 K46 E62 V89 M91 Y93 L94 L143 T153 N389 K391 D393 N394 D407 P416 T427 N136 K138 D140 N141 D154 P163 T174 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=100nM Q13153 27994749 601 LEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLDMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 5kbr A 2.36 BS01 IPW A 1 I276 V284 A297 K299 V328 V342 M344 E345 Y346 L347 L396 T406 I22 V30 A36 K38 V58 V66 M68 E69 Y70 L71 L120 T130 N389 K391 D393 N394 D407 T427 N113 K115 D117 N118 D131 T144 2.7.11.1 0004672,0005524,0006468 ic50=260nM remove_due_to_license_issue Q13153 27994749 601 EKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAEVAIKQELIINEILVMRENKNPNIVNYLDSYWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLDMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 5kby A 2.24 BS01 6RL A 1 E205 E206 Y547 S630 Y631 V656 W659 Y662 Y666 V711 E164 E165 Y506 S589 Y590 V615 W618 Y621 Y625 V670 Y547 S630 Y631 D708 H740 Y506 S589 Y590 D667 H699 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 Ki=1.5nM remove_due_to_license_issue IC50=1.3nM, Ki=5.1nM P27487 27328054 1510 RKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5kcb A 2.101 BS01 ET A 1 A32 W35 Q36 Y39 V106 Y138 A31 W34 Q35 Y38 V105 Y137 ? Kd=0.99uM remove_due_to_license_issue A0A0H3JRN6 27505298 201 MEYQLQQLASLTLVGIKETYENGRQAQQHIAGFWQRCYQEGVIADLQLKNNGDLAGILGLCIPELDGKMSYMIAVTGDNSADIAKYDVITLASSKYMVFEAQGAVPKAVQQKMEEVHHYIHQYQANTVKSAPFFELYQDGDTTSEKYITEIWMPVKGLEHHHHHH 5kcv A 2.7 BS01 6S1 A 1 N53 Q79 W80 L210 T211 V270 Y272 D274 I290 D292 N40 Q66 W67 L141 T142 V201 Y203 D205 I221 D223 D274 K276 N279 D292 D205 K207 N210 D223 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue P31749 27305487 501 IVKEGWLHKRGEYITWRPRYFLLKNDGTFIGYKERPAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYF 5kcx A 2.2 BS01 6S3 A 1 L44 V52 A65 L120 V126 L174 L11 V19 A32 L87 V93 L141 D167 K169 N172 D186 L193 T204 D134 K136 N139 D153 L160 T171 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=200nM P11309 28947155 403 LESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5kde A 2.65 BS01 6RT A 1 P63 R101 W102 V105 P112 P64 R102 W103 V106 P113 3.6.1.1 0000287,0004427,0005576,0005737,0005829,0005886,0006796,0016787,0044228,0046872 remove_due_to_license_issue IC50=1.30e+5nM P9WI55 27622287 201 AMQFDVTIEIPKGQRNKYEVDHETGRVRLDRYLYTPMAYPTDYGFIEDTLGDDGDPLDALVLLPQPVFPGVLVAARPVGMFRMVDEHGGDDKVLCVPAGDPRWDHVQDIGDVPAFELDAIKHFFVHYKDLEPGKFVKAADWVDRAEAEAEVQRSVERFKAG 5kdf A 2.45 BS01 6RU A 1 P63 W102 P64 W103 3.6.1.1 0000287,0004427,0005576,0005737,0005829,0005886,0006796,0016787,0044228,0046872 remove_due_to_license_issue IC50=5.40e+5nM P9WI55 27622287 201 AMQFDVTIEIPKGQRNKYEVDHETGRVRLDRYLYTPMAYPTDYGFIEDTLGDDGDPLDALVLLPQPVFPGVLVAARPVGMFRMVDEHGGDDKVLCVPAGDPRWDHVQDIGDVPAFELDAIKHFFVHYKDLEPGKFVKAADWVDRAEAEAEVQRSVERFKAG 5kdr A 2.6 BS01 YT5 B 1 S198 L229 S185 L216 2.1.3.15 0003824,0003989,0005524,0005737,0006633,0009317,0016740,0016743,0016874,2001295 remove_due_to_license_issue Q2FXM7 27471863 301 LDFEKPLFEIRNKIESQEEIDMLEASLERETKKIYTNLKPWDRVQIARLQERPTTLDYIPYIFDSFMELHGDRNFRDDPAMIGGIGFLNGRAVTVIGQQRGKDTKDNIYRNFGMAHPEGYRKALRLMKQAEKFNRPIFTFIDTKGAYPGKAAEERGQSESIATNLIEMASLKVPVIAIVIGEGGSGGALGIGIANKVLMLENSTYSVISPEGAAALLWKDSNLAKIAAETMKITAHDIKQLGIIDDVISEPLGGAHKDIEQQALAIKSAFVAQLDSLESLSRDEIANDRFEKFRNIGSYIE 5kdr B 2.6 BS01 YT5 B 1 M134 G166 G167 T206 G207 G208 A231 G232 V235 M106 G138 G139 T178 G179 G180 A203 G204 V207 G207 G208 G179 G180 2.1.3.15 0003989,0005524,0005737,0006633,0008270,0009317,0016740,0016743,0046872,0071768,2001295 remove_due_to_license_issue Q2FXM6 27471863 301 IMTKCPKCKKIMYTKELAENLNVCFNCDHHIALTAYKRIEAISDEGSFTEFDKGMTSANPLDFPSYLEKIEKDQQKTGLKEAVVTGTAQLDGMKFGVAVMDSRFRMGSMGSVIGEKICRIIDYCTENRLPFILFSASGGARMQEGIISLMQMGKTSVSLKRHSDAGLLYISYLTHPTTGGVSASFASVGDINLSEPKALIGFAGRRVIEQTINDFQTAEFLLEHGQLDKVVHRNDMRQTLSEILKIHQEV 5ke0 A 1.68 BS01 6S9 A 1 G35 A50 K52 Q103 D104 L105 M106 E107 L154 D165 G20 A35 K37 Q88 D89 L90 M91 E92 L139 D150 D147 K149 S151 N152 D165 T188 D132 K134 S136 N137 D150 T173 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 remove_due_to_license_issue IC50=0.200000nM P63086 27329786 401 VFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 5ke6 A 1.99 BS01 dna B 0 Y411 H416 R443 E446 R449 R471 H474 Y13 H18 R45 E48 R51 R73 H76 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 THTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDELTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5ke6 A 1.99 BS02 dna C 0 K413 S415 Y430 D445 S472 K15 S17 Y32 D47 S74 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 THTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDELTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5ke8 A 2.45 BS01 dna B 0 Y411 K413 H416 W439 F441 R443 R449 H450 K453 R471 H474 Y13 K15 H18 W41 F43 R45 R51 H52 K55 R73 H76 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 THTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDPLTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5ke8 A 2.45 BS02 dna C 0 S444 F460 S472 S46 F62 S74 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 THTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDPLTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5ke9 A 2.336 BS01 dna B 0 H416 W439 F441 R443 R449 H450 K453 R471 H474 H21 W44 F46 R48 R54 H55 K58 R76 H79 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 RTATHTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDPLTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5ke9 A 2.336 BS02 dna C 0 Y430 D445 F460 Y35 D50 F65 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 RTATHTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDPLTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5keb A 2.453 BS01 dna B 0 Y411 K413 H416 R443 R449 K453 R471 H474 Y12 K14 H17 R44 R50 K54 R72 H75 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 HTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDDLTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5keb A 2.453 BS02 dna C 0 K413 S415 Y430 K14 S16 Y31 ? remove_due_to_license_issue Q60793 27596594 1 ~ 10 HTCDYAGCGKTYTKSSHLKAHLRTHTGEKPYHCDWDGCGWKFARSDDLTRHYRKHTGHRPFQCQKCDRAFSRSDHLALHMKRHF 5kej A 2.35 BS01 GTX A 1 S14 Y16 K54 I55 E67 S68 S13 Y15 K53 I54 E66 S67 2.5.1.18 0004364,0005737,0005829,0006749,0009407,0009636,0016740 Kd=7.8uM remove_due_to_license_issue A0A1P8NWC2 28104507 301 AKSDVKLLGAWPSPYVMRARITLNVKSVDYELLEETLGSKSDLLLKSNPVHKKIPVLIHNDKPICESLIIVHYIDEFWSSGPSILPSDPYDRAIARFWAAYLDEKWYPSLKGIASAQGEEAKKAAVDQVGESLALIEDTYVKLSKGKPFFGGEKIGYLDIAFGCFLGWLRVTEKTSGVKFLNEAKTPHLAKWAVRFCADPAVKDVMPETEKLAEFAKLLAKF 5kej B 2.35 BS01 GTX B 1 S14 Y16 K54 I55 E67 S68 Y108 S13 Y15 K53 I54 E66 S67 Y107 2.5.1.18 0004364,0005737,0005829,0006749,0009407,0009636,0016740 Kd=7.8uM remove_due_to_license_issue A0A1P8NWC2 28104507 301 AKSDVKLLGAWPSPYVMRARITLNVKSVDYELLEETLGSKSDLLLKSNPVHKKIPVLIHNDKPICESLIIVHYIDEFWSSGPSILPSDPYDRAIARFWAAYLDEKWYPSLKGIASAQGEEAKKAAVDQVGESLALIEDTYVKLSKGKPFFGGEKIGYLDIAFGCFLGWLRVTEKTSGVKFLNEAKTPHLAKWAVRFCADPAVKDVMPETEKLAEFAKLLAKF 5kgw A 2.34 BS01 7SK A 1 A169 E170 H171 T174 M178 A101 E102 H103 T106 M110 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 27568085 304 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGYSAGERIVDIIATDI 5kgx A 2.67 BS01 7SK A 1 A169 E170 H171 T174 M178 A101 E102 H103 T106 M110 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0015074 remove_due_to_license_issue P12497 27568085 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKTACWWAGIKQEESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNKKRKGYSAGERIVDIIATDI 5kh3 A 1.6 BS04 6U6 A 1 W1143 G1154 R1155 W1182 Y1184 Y1189 W36 G47 R48 W75 Y77 Y82 3.5.1.-,3.5.1.98 0008270 remove_due_to_license_issue IC50=55000nM, Kd=60000nM Q9UBN7 29019676 1317 SPLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKFG 5kh7 A 1.7 BS04 6T7 A 1 W1143 R1155 W1182 Y1184 Y1189 W35 R47 W74 Y76 Y81 3.5.1.-,3.5.1.98 0008270 remove_due_to_license_issue Kd=210000nM, IC50=350000nM Q9UBN7 29019676 1304 PLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKFG 5khd A 1.7501 BS01 C2E R 1 Q113 R114 R125 D128 Q30 R31 R42 D45 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 201 KLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd A 1.7501 BS02 C2E R 2 R114 G115 D116 R31 G32 D33 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 202 KLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd A 1.7501 BS03 C2E A 1 K84 R114 S123 I124 R125 K1 R31 S40 I41 R42 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 201 KLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd A 1.7501 BS04 C2E A 2 K84 D116 N118 V121 L122 S123 K1 D33 N35 V38 L39 S40 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 202 KLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd R 1.7501 BS01 C2E R 1 K84 R114 S123 I124 R125 Q126 K2 R32 S41 I42 R43 Q44 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 201 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd R 1.7501 BS02 C2E R 2 D116 N118 V121 L122 S123 D34 N36 V39 L40 S41 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 202 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd R 1.7501 BS03 C2E A 1 I110 R114 R125 D128 I28 R32 R43 D46 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 201 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khd R 1.7501 BS04 C2E A 2 R114 G115 D116 R32 G33 D34 ? 0045892 Kd=2.5uM remove_due_to_license_issue F2RCL8 25171413 202 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDA 5khg A 2.241 BS01 CC7 A 1 V564 F580 G581 E582 I583 C584 R591 T592 R632 V122 F138 G139 E140 I141 C142 R149 T150 R190 ? Kd=20.23uM remove_due_to_license_issue O88703 27568927 701 DSSRRQYQEKYKQVEQYMSFHKLPADFRQKIHDYYEHRYQGKMFDEDSILGELNGPLREEIVNFNCRKLVASMPLFANADPNFVTAMLTKLKFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKEMKLSDGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVAIDRLDRIGKKNSIL 5khh A 1.77 BS01 6SW A 1 M572 F580 G581 E582 I583 C584 R591 T592 R632 R635 I636 M129 F137 G138 E139 I140 C141 R148 T149 R189 R192 I193 ? Kd=49.32uM remove_due_to_license_issue O88703 27568927 701 SSRRQYQEKYKQVEQYMSFHKLPADFRQKIHDYYEHRYQGKMFDEDSILGELNGPLREEIVNFNCRKLVASMPLFANADPNFVTAMLTKLKFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKEMKLSDGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVAIDRLDRIGK 5khi A 2.1 BS01 6SX A 1 V564 F580 G581 E582 I583 C584 R591 T592 R632 V122 F138 G139 E140 I141 C142 R149 T150 R190 ? Kd=0.17uM remove_due_to_license_issue O88703 27568927 701 DSSRRQYQEKYKQVEQYMSFHKLPADFRQKIHDYYEHRYQGKMFDEDSILGELNGPLREEIVNFNCRKLVASMPLFANADPNFVTAMLTKLKFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKEMKLSDGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVAIDRLDRIGKKNSIL 5khj A 2.01 BS01 6SY A 1 F580 G581 E582 I583 C584 R591 T592 R632 R635 F138 G139 E140 I141 C142 R149 T150 R190 R193 ? Kd=1.33uM remove_due_to_license_issue O88703 27568927 701 DSSRRQYQEKYKQVEQYMSFHKLPADFRQKIHDYYEHRYQGKMFDEDSILGELNGPLREEIVNFNCRKLVASMPLFANADPNFVTAMLTKLKFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKEMKLSDGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVAIDRLDRIGKKNS 5khk A 2.07 BS01 6SZ A 1 V564 M572 F580 G581 E582 I583 C584 R591 T592 A593 R632 I636 V122 M130 F138 G139 E140 I141 C142 R149 T150 A151 R190 I194 ? Kd=0.41uM remove_due_to_license_issue O88703 27568927 701 DSSRRQYQEKYKQVEQYMSFHKLPADFRQKIHDYYEHRYQGKMFDEDSILGELNGPLREEIVNFNCRKLVASMPLFANADPNFVTAMLTKLKFEVFQPGDYIIREGTIGKKMYFIQHGVVSVLTKGNKEMKLSDGSYFGEICLLTRGRRTASVRADTYCRLYSLSVDNFNEVLEEYPMMRRAFETVAIDRLDRIGKKNSIL 5khm A 1.48 BS01 XNH A 1 Y97 Y139 D145 I146 M149 Y55 Y97 D103 I104 M107 ? Ki=5.012nM remove_due_to_license_issue Ki=126nM, IC50=20nM O60885 27528113 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5khm B 1.48 BS01 XNH A 1 W81 F83 N140 D145 I146 W40 F42 N99 D104 I105 ? remove_due_to_license_issue Ki=126nM, IC50=20nM O60885 27528113 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5khx A 2.4 BS01 6TE A 1 G882 A906 E957 F958 L959 N1008 L1010 D1021 G16 A35 E81 F82 L83 N132 L134 D145 D1003 A1005 R1007 N1008 D1021 D1040 D127 A129 R131 N132 D145 D164 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=90nM P23458 27827355 4000 PTHFEKRFLKRIRDLGKVELCRYDPEGDNTGEQVAVKSLKNHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 5ki6 A 2.153 BS01 rna B 0 R277 F294 Y311 H316 H336 T337 Y338 D358 T361 I365 T368 K525 Y529 K533 Q545 C546 V547 Q548 N551 T559 N562 K566 K570 R714 H753 I756 Q757 S760 R761 Y790 R792 C793 V797 S798 Y804 Y815 R238 F255 Y272 H277 H297 T298 Y299 D318 T321 I325 T328 K485 Y489 K493 Q505 C506 V507 Q508 N511 T519 N522 K526 K530 R674 H713 I716 Q717 S720 R721 Y750 R752 C753 V757 S758 Y764 Y775 3.1.26.n2 0000340,0000932,0000993,0001046,0003676,0003723,0003725,0003727,0003729,0003743,0004519,0004521,0005515,0005634,0005654,0005737,0005829,0006355,0006412,0006413,0006417,0009791,0010501,0010586,0010628,0016020,0016442,0016891,0030422,0030425,0031047,0031054,0033962,0035194,0035196,0035197,0035198,0035278,0035279,0035925,0036464,0042985,0043232,0045727,0045766,0045944,0045947,0046872,0060213,0061980,0070062,0070551,0070578,0070922,0090128,0090624,0090625,0098794,0098808,0098978,1900153,1901165,1990904 remove_due_to_license_issue Q9UKV8 27387838 1 ~ 21 AFKPPPRPDFGTSGRTIKLQANFFEMDIPKIDIYHYELDIKPEKCPRRVNREIVEHMVQHFKTQIFGDRKPVFDGRKNLYTAMPLPIGRDKVELEVTLRIFKVSIKWVSCVSLQALHDALSGRLVPFETIQALDVVMRHLPSMRYTPVGRSFFTASNPLGGGREVWFGFHQSVRPSLWKMMLNIDVSATAFYKAQPVIEFVCEVLDFKSIEEQQKPLTDSQRVKFTKEIKGLKVEITRKYRVCNVTRRPASHQTFPLQQESGQTVECTVAQYFKDRHKLVLRYPHLPCLQVGQEQKHTYLPLEVCNIVAGQRCIKLTDNQTSTMIRATARSAPDRQEEISKLMRSADFNTDPYVREFGIMVKDEMTDVTGRVLQPPSILYGGRNKAIATPVQGVWDMRNKQFHTGIEIKVWAIACFAPQRQCTEVHLKSFTEQLRKISRDAGMPIQGQPCFCKYAQGADSVEPMFRHLKNTYAGLQLVVVILPGKTPVYAEVKRVGDTVLGMATQCVQMKNVQRTTPQTLSNLCLKINVKLGGVNNILLPQGRPPVFQQPVIFLGADVTHPPAGDGKKPSIAAVVGSMDAHPNRYCATVRVQQHRQEIIQDLAAMVRELLIQFYKSTRFKPTRIIFYRDGVSEGQFQQVLHHELLAIREACIKLEKDYQPGITFIVVQKRHHTRLFCTDKNERVGKSGNIPAGTTVDTKITHPTEFDFYLCSHAGIQGTSRPSHYHVLWDDNRFSSDELQILTYQLCHTYVRCTRSVSIPAPAYYAHLVAFRARYHLHQALAKAVQVHQDTLRTMYFA 5kit A 1.6 BS01 6TA A 1 H191 F193 R196 D219 V242 A244 S275 R311 I351 H174 F176 R179 D202 V225 A227 S258 R294 I334 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.013uM remove_due_to_license_issue IC50=47.9nM P43490 27541271 501 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 5kit B 1.6 BS01 6TA B 1 H191 F193 R196 D219 V242 A244 S275 I309 R311 H174 F176 R179 D202 V225 A227 S258 I292 R294 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=0.013uM remove_due_to_license_issue IC50=47.9nM P43490 27541271 501 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNIELE 5kj0 A 1.51 BS01 6TB A 1 W81 P82 Q85 V87 L92 Y97 Y139 N140 I146 W40 P41 Q44 V46 L51 Y56 Y98 N99 I105 ? ic50=130nM remove_due_to_license_issue IC50=100nM O60885 27862999 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5kjk A 1.93 BS04 6T1 A 1 T105 K145 I149 N180 N182 G183 F184 T185 Y240 S257 Y258 T101 K141 I145 N176 N178 G179 F180 T181 Y236 S253 Y254 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 ic50=0.012uM remove_due_to_license_issue Q9NRG4 28002961 506 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIESH 5kjm A 2.19 BS02 6TM A 1 K145 I149 N180 N182 G183 F184 T185 Y240 Y258 K141 I145 N176 N178 G179 F180 T181 Y236 Y254 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 ic50=0.065uM remove_due_to_license_issue Q9NRG4 28002961 502 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIESH 5kjn A 2.72 BS07 6TL A 1 K145 I149 V179 N180 N182 G183 F184 T185 Y240 S257 Y258 F259 K141 I145 V175 N176 N178 G179 F180 T181 Y236 S253 Y254 F255 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 remove_due_to_license_issue Q9NRG4 28002961 510 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIESH 5kk8 A 2.11 BS01 ADP A 1 K9 L61 T91 V109 N112 K9 L61 T91 V109 N112 K9 Y49 N112 H115 E126 K9 Y49 N112 H115 E126 0004550,0005524,0006166,0006183,0006228,0006241,0009165,0009202,0016301,0032261,0034214,0042802,0043531 remove_due_to_license_issue A0A3Q0KJ78 31103556 201 PERTFIMVKPDGVQRGLVGEVIQRFERRGYKLVAIKMMHASEQLLQTHYEALKSLSFFPKLVAYMSSGPVVPMVFEGRKVVENGRTMLGATKPEASCPGSIRGDYCQDVGRNVVHGSDSTESANREINLWFSPQELCQYKQAVDPWIHE 5kkq A 1.744 BS01 dna B 0 F351 K367 Y392 K395 Y407 S419 K423 S450 F35 K51 Y76 K79 Y91 S103 K107 S134 ? remove_due_to_license_issue P49711 28529057 1 ~ 17 PLGSPHKCPDCDMAFVTSGELVRHRRYKHTHEKPFKCSMCDYASVEVSKLKRHIRSHTGERPFQCSLCSYASRDTYKLKRHMRTHSGEKPYECYICHARFTQSGTMKMHILQKHTENVAKFHCPHCDTVIARKSDLGVHLRKQHSYI 5kkq A 1.744 BS02 dna C 0 F331 E336 R339 H340 Y343 K344 Y358 E362 K365 R368 H369 S372 R377 Y386 R389 K393 R396 H397 T400 K405 F416 T417 Q418 T421 H425 K429 I446 A447 R448 D451 F15 E20 R23 H24 Y27 K28 Y42 E46 K49 R52 H53 S56 R61 Y70 R73 K77 R80 H81 T84 K89 F100 T101 Q102 T105 H109 K113 I130 A131 R132 D135 ? remove_due_to_license_issue P49711 28529057 1 ~ 17 PLGSPHKCPDCDMAFVTSGELVRHRRYKHTHEKPFKCSMCDYASVEVSKLKRHIRSHTGERPFQCSLCSYASRDTYKLKRHMRTHSGEKPYECYICHARFTQSGTMKMHILQKHTENVAKFHCPHCDTVIARKSDLGVHLRKQHSYI 5kkq D 1.744 BS01 dna E 0 F351 Y392 Y407 S419 K423 K449 S450 F31 Y72 Y87 S99 K103 K129 S130 ? remove_due_to_license_issue P49711 28529057 1 ~ 17 PHKCPDCDMAFVTSGELVRHRRYKHTHEKPFKCSMCDYASVEVSKLKRHIRSHTGERPFQCSLCSYASRDTYKLKRHMRTHSGEKPYECYICHARFTQSGTMKMHILQKHTENVAKFHCPHCDTVIARKSDLGVHLRKQHSYIEQ 5kkq D 1.744 BS02 dna F 0 F331 E336 R339 H340 Y343 K344 Y358 E362 K365 R368 H369 S372 R377 Y386 R389 K393 R396 H397 T400 K405 F416 Q418 T421 H425 K429 A447 R448 D451 F11 E16 R19 H20 Y23 K24 Y38 E42 K45 R48 H49 S52 R57 Y66 R69 K73 R76 H77 T80 K85 F96 Q98 T101 H105 K109 A127 R128 D131 ? remove_due_to_license_issue P49711 28529057 1 ~ 17 PHKCPDCDMAFVTSGELVRHRRYKHTHEKPFKCSMCDYASVEVSKLKRHIRSHTGERPFQCSLCSYASRDTYKLKRHMRTHSGEKPYECYICHARFTQSGTMKMHILQKHTENVAKFHCPHCDTVIARKSDLGVHLRKQHSYIEQ 5kkr B 3.509 BS01 6U7 B 1 V680 A690 R692 F725 T739 L741 C742 F793 T802 D803 F804 V28 A38 R40 F73 T87 L89 C90 F141 T150 D151 F152 D786 K790 N791 D803 Q825 D134 K138 N139 D151 Q168 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=120nM Q6VAB6 27556948 1001 SQTSIFLQEWDIPFEQLEIGELIGFGQVYHGRWHGEVAIRLIDIERDNEDQLKAFKREVMAYRQTRHENVVLFMGACMSPPHLAIITSLCKGRTLYSVVRDAKIVLDVNKTRQIAQEIVKGMGYLHAKGILHKDLKSKNVFYDNGKVVITDFGLFSISGVLQDKLRIQNGWLCHLAPEIIRQLSPDDKLPFSKHSDVFALGTIWYELHAREWPFKTQPAEAIIWQMGTGMKPNLSQIGMGKEISDILLFCWAFEQEERPTFTKLMDMLEKLP 5kks A 3.3 BS01 6U1 A 1 R84 G85 A86 F87 G88 E89 V90 A103 K105 M153 E154 Y155 M156 L205 D216 F368 R79 G80 A81 F82 G83 E84 V85 A98 K100 M148 E149 Y150 M151 L200 D211 F363 D198 K200 N203 D216 T237 D193 K195 N198 D211 T232 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=2.0nM Q13464 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEETFPIPKAFVGNQLPFVGFTYYSNRRY 5kkt A 2.8 BS01 6U2 A 1 I82 G85 F87 G88 E89 V90 A103 K105 F120 M153 Y155 M156 L205 D216 G218 F368 I77 G80 F82 G83 E84 V85 A98 K100 F111 M144 Y146 M147 L196 D207 G209 F359 D198 K200 N203 D216 T237 D189 K191 N194 D207 T228 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=<1.000000nM Q13464 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLETFPIPKAFVGNQLPFVGFTYYSNRRY 5kl1 A 3.701 BS01 rna C 0 Q1123 R1127 F1160 N1162 Y1163 M1195 Y1196 R1199 Q1202 H1235 R1271 N1306 Y1307 Q1310 K1339 S1342 N1343 E1346 N1382 Y1383 T1415 Y1416 Q32 R36 F69 N71 Y72 M104 Y105 R108 Q111 H144 R180 N215 Y216 Q219 K248 S251 N252 E255 N291 Y292 T324 Y325 ? 0003723 remove_due_to_license_issue P25822 27482653 1 ~ 12 RSRLLEDFRNQRYPNLQLRDLANHIVEFSQDQHGSRFIQQKLERATAAEKQMVFSEILAAAYSLMTDVFGNYVIQKFFEFGTPEQKNTLGMQVKGHVLQLALQMYGCRVIQKALESISPEQQQEIVHELDGHVLKCVKDQNGNHVVQKCIECVDPVALQFIINAFKGQVYSLSTHPYGCRVIQRILEHCTAEQTTPILDELHEHTEQLIQDQYGNYVIQHVLEHGKQEDKSILINSVRGKVLVLSQHKFASNVVEKCVTHATRGERTGLIDEVCTFNDNALHVMMKDQYANYVVQKMIDVSEPTQLKKLMTKIRPHMAALRKYTYGKH 5kl1 B 3.701 BS01 rna C 0 V320 F321 N324 N325 L349 Y352 H365 T366 I367 K368 Y369 V5 F6 N9 N10 L34 Y37 H50 T51 I52 K53 Y54 ? 0003723,0008270 remove_due_to_license_issue P25724 27482653 1 ~ 12 SRHCVFCENNNEPEAVINSHSVRDNFNRVLCPKLRTYVCPICGASGDSAHTIKYCPKKPIITMEDAIKAE 5kl8 A 4.0 BS01 rna C 0 N1162 Y1163 M1195 Y1196 R1199 Q1231 H1235 Y1268 R1271 Q1274 N1306 Y1307 Q1310 S1342 N1343 E1346 N1382 Y1383 Q1386 K1413 Y1414 T1415 Y1416 N53 Y54 M86 Y87 R90 Q122 H126 Y159 R162 Q165 N197 Y198 Q201 S233 N234 E237 N273 Y274 Q277 K304 Y305 T306 Y307 ? 0003723 remove_due_to_license_issue P25822 27482653 1 ~ 11 RSRLLEDFRNQQDQHGSRFIQQKLERATAAEKQMVFSEILAAAYSLMTDVFGNYVIQKFFEFGTPEQKNTLGMQVKGHVLQLALQMYGCRVIQKALESISPEQQQEIVHELDGHVLKCVKDQNGNHVVQKCIECVDPVALQFIINAFKGQVYSLSTHPYGCRVIQRILEHCTAEQTTPILDELHEHTEQLIQDQYGNYVIQHVLEHGKQEDKSILINSVRGKVLVLSQHKFASNVVEKCVTHATRGERTGLIDEVCTFNDNALHVMMKDQYANYVVQKMIDVSEPTQLKKLMTKIRPHMAALRKYTYGK 5kl8 B 4.0 BS01 rna C 0 V320 F321 N324 N325 L349 Y352 H365 T366 I367 K368 Y369 V5 F6 N9 N10 L34 Y37 H50 T51 I52 K53 Y54 ? 0003723,0008270 remove_due_to_license_issue P25724 27482653 1 ~ 11 SRHCVFCENNNEPEAVINSHSVRDNFNRVLCPKLRTYVCPICGASGDSAHTIKYCPKKPIITMEDAIKA 5kla A 1.14 BS01 rna B 0 Q1123 R1127 Q1130 F1160 N1162 Y1163 Y1196 R1199 Q1202 H1235 C1270 R1271 Q1274 Y1304 N1306 Y1307 Q1310 K1339 S1342 N1343 E1346 N1382 Y1383 Q1386 Y1416 H1419 Q34 R38 Q41 F71 N73 Y74 Y107 R110 Q113 H146 C181 R182 Q185 Y215 N217 Y218 Q221 K250 S253 N254 E257 N293 Y294 Q297 Y327 H330 ? 0003723 remove_due_to_license_issue P25822 27482653 1 ~ 8 SGRSRLLEDFRNQRYPNLQLRDLANHIVEFSQDQHGSRFIQQKLERATAAEKQMVFSEILAAAYSLMTDVFGNYVIQKFFEFGTPEQKNTLGMQVKGHVLQLALQMYGCRVIQKALESISPEQQQEIVHELDGHVLKCVKDQNGNHVVQKCIECVDPVALQFIINAFKGQVYSLSTHPYGCRVIQRILEHCTAEQTTPILDELHEHTEQLIQDQYGNYVIQHVLEHGKQEDKSILINSVRGKVLVLSQHKFASNVVEKCVTHATRGERTGLIDEVCTFNDNALHVMMKDQYANYVVQKMIDVSEPTQLKKLMTKIRPHMAALRKYTYGKHINAKLEK 5klp A 2.002 BS01 IHP A 1 K53 K226 K229 K289 H290 S314 H317 R326 Q358 R362 K9 K178 K181 K241 H242 S266 H269 R278 Q298 R302 2.3.1.- 0000822,0005515,0005576,0016020,0016413,0016746,0020002,0030430,0035821,0042025,0044163,0090729 Kd=22.7uM remove_due_to_license_issue Q6VE93 27525589 401 TQSMRLQQKINDLKPYVRHARGPIKAYGQAALDRASGAVSFAELDATHLDAMVYIENQRNPGLNLKHFRDHYYLIQALQSDGPSAFRAIFPQTCPETGQTLKHHVMADVRLHQGAPTIIITEPAVIVGARYQQLQRHNLTLEDLSESGVPLSQVAIIETQAAATSDDCVMYSLNYAIKAHKNAAQFDDIHHGLQHGTLSTESESRARTTLGALEASSSYSVMHEGAHAAFGADVLPVDFYKHGASLTQAYYLMKRPDGRMAGRVNSEGHSEAENLVQRNQAFRVKTQFSASIDGFRLQEIKRVLAAAQR 5kly A 1.3 BS01 6UR A 1 D43 I44 N99 G105 Q106 S107 N112 H114 D32 I33 N88 G94 Q95 S96 N101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVNLHVLGGRQMHWPPG 5kly B 1.3 BS01 6UR A 1 M121 W123 M107 W109 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 GDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVNLHVLGGRQMHWPPG 5klz B 1.5 BS01 AMP B 1 D43 I44 N99 G105 S107 V108 H112 H114 D32 I33 N88 G94 S96 V97 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5km0 A 1.533 BS01 IMP A 1 I22 D43 I44 G105 Q106 S107 V108 H112 H114 I11 D32 I33 G94 Q95 S96 V97 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5km1 A 1.65 BS01 5GP A 1 I18 F41 D43 I44 N99 Q106 S107 H112 H114 I7 F30 D32 I33 N88 Q95 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5km2 A 1.25 BS01 C5P A 1 D43 I44 N99 S107 H112 H114 D32 I33 N88 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5km3 A 1.2 BS01 U5P A 1 D43 I44 N99 S107 H112 H114 D32 I33 N88 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 5km5 B 2.1 BS01 TR5 B 1 L64 F78 D80 V81 N136 S144 V145 H149 H151 L13 F27 D29 V30 N85 S93 V94 H98 H100 3.9.1.- 0003824 remove_due_to_license_issue Q9BX68 28968488 201 APTIFSRILDKSLPADILYEDQQCLVFRDVAPQAPVHFLVIPKKPIPRISQAEEEDQQLLGHLLLVAKQTAKAEGLGDGYRLVINDGKLGAQSVYHLHIHVLGGRQLQWPPG 5km9 B 1.45 BS01 ADN B 1 D80 V81 V145 D29 V30 V94 3.9.1.- 0003824 remove_due_to_license_issue Q9BX68 28968488 201 APTIFSRILDKSLPADILYEDQQCLVFRDVAPQAPVHFLVIPKKPIPRISQAEEEDQQLLGHLLLVAKQTAKAEGLGDGYRLVINDGKLGAQSVYHLHIHVLGGRQLQWPPG 5kma A 1.55 BS01 777 A 1 I18 F41 D43 I44 N99 G105 S107 V108 N112 H114 I7 F30 D32 I33 N88 G94 S96 V97 N101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVNLHVLGGRQMHWPPG 5kmf A 3.2 BS01 6U9 A 1 G1164 F1167 G164 F167 ? 0001518,0005216,0005248,0005261,0005886,0006811,0016020,0035725,0042802,0046872,0055085,0098655 remove_due_to_license_issue A8EVM5 27556947 1301 MYLRITNIVESSFFTKFIIYLIVLNGITMGLETSKTFMQSFGVYTTLFNQIVITIFTIEIILRIYVHRISFFKDPWSLFDFFVVAISLVPTSSGFEILRVLRVLRLFRLVTAVPQMRKIVSALISVIPGMLSVIALMTLFFYIFAIMATQLFGERFPEWFGTLGESFYTLFQVMTLDDWSNGIVRPLMEVYPYAYVFFIPFIFVVTFVMINLVVAIIVD 5knj A 2.88 BS01 6UX A 1 L217 E250 M254 L263 M283 Y285 C286 G289 E293 L338 A348 G349 L25 E52 M56 L65 M85 Y87 C88 G91 E95 L140 A150 G151 K331 S335 N336 G349 K133 S137 N138 G151 ? 0004672,0005524,0006468 remove_due_to_license_issue Kd=9300nM Q8NB16 27832137 501 IKEIKKEQLSGSPWILLRENEVSTLYKGEYHRAPVAIKVFKKAIVRQTFNKEIKTMKKFESPNILRIFGICIDETVTPPQFSIVMEYCELGTLRELLDREKDLTLGKRMVLVLGAARGLYRLHHSEAPELHGKIRSSNFLVTQGYQVKLAGFDRVKSTAYLSPQELEDVFYQYDVKSEIYSFGIVLWEIATGDIPFQGCNSEKIRKLVAVKRQQEPLGEDCPSELREIIDECRAHDPSVRPSVDEILKKLST 5knr A 2.864 BS01 3L5 A 1 G48 D104 I105 I106 D107 S108 G109 N110 T111 L112 K135 F156 V157 I162 G44 D95 I96 I97 D98 S99 G100 N101 T102 L103 K126 F147 V148 I153 E103 D104 D107 F156 R169 E94 D95 D98 F147 R160 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 MKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSYGTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILLD 5kns A 2.792 BS01 3L7 A 1 D107 S108 N110 T111 K135 V157 R169 D97 S98 N100 T101 K125 V147 R159 E103 D104 D107 F156 R169 E93 D94 D97 F146 R159 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 DMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILL 5kns B 2.792 BS01 3L7 B 1 D107 S108 G109 T111 K135 F156 V157 D163 R169 D98 S99 G100 T102 K126 F147 V148 D154 R160 E103 D104 D107 F156 R169 E94 D95 D98 F147 R160 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 DMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSTTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILLD 5knt A 2.55 BS01 6WB A 1 E103 D104 I105 D107 S108 G109 T111 K135 F156 V157 I162 E92 D93 I94 D96 S97 G98 T100 K124 F145 V146 I151 E103 D104 D107 F156 R169 E92 D93 D96 F145 R158 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 DMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILL 5knu A 2.808 BS01 6WA A 1 D107 S108 G109 T111 F156 V157 I162 D98 S99 G100 T102 F147 V148 I153 E103 D104 D107 F156 R169 E94 D95 D98 F147 R160 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 RDMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILLD 5knu B 2.808 BS01 6WA B 1 S73 I106 D107 S108 G109 R138 V157 I162 S71 I99 D100 S101 G102 R131 V150 I155 E103 D104 D107 F156 R169 E96 D97 D100 F149 R162 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 RDMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSYTTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILL 5knv A 2.861 BS01 6W9 A 1 I105 D107 G109 T111 K135 V157 I94 D96 G98 T100 K124 V146 E103 D104 D107 F156 R169 E92 D93 D96 F145 R158 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 MKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILL 5knv B 2.861 BS01 6W9 B 1 D107 S108 G109 T111 L112 F156 V157 I162 D97 S98 G99 T101 L102 F146 V147 I152 E103 D104 D107 F156 R169 E93 D94 D97 F146 R159 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 DMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILLD 5knx A 2.4 BS01 6WC A 1 S73 I105 D107 S108 G109 K135 R138 F156 V157 I162 S69 I97 D99 S100 G101 K127 R130 F148 V149 I154 E103 D104 D107 F156 R169 E95 D96 D99 F148 R161 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 MKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSYGSTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVILLD 5knx B 2.4 BS01 6WC B 1 S73 D107 S108 G109 K135 F156 V157 I162 S70 D104 S105 G106 K132 F153 V154 I159 E103 D104 D107 F156 R169 E100 D101 D104 F153 R166 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0032991,0042802,0046100,0046872,0051289,0052657,0097216 remove_due_to_license_issue P0A9M2 201 DMKHTVEVMIPEAEIKARIAELGRQITERYKDSGSDMVLVGLLRGSFMFMADLCREVQVSHEVDFMTASSYGSGMSTTRDVKILKDLDEDIRGKDVLIVEDIIDSGNTLSKVREILSLREPKSLAICTLLDKPSRREVNVPVEFIGFSIPDEFVVGYGIDYAQRYRHLPYIGKVIL 5ko1 A 2.16 BS01 6UY A 1 R210 E211 N212 S215 L217 A228 K230 E250 M283 C286 L338 A348 G349 R19 E20 N21 S24 L26 A37 K39 E59 M92 C95 L147 A157 G158 K331 S335 N336 G349 K140 S144 N145 G158 ? 0004672,0005524,0006468 Kd=230nM remove_due_to_license_issue Kd=230nM Q8NB16 27832137 501 QIKEIKKEQLSGSPWILLRENEVSTLYKGEYHRAPVAIKVFKKLQAGSIAIVRQTFNKEIKTMKKFESPNILRIFGICIDETVTPPQFSIVMEYCELGTLRELLDREKDLTLGKRMVLVLGAARGLYRLHHSEAPELHGKIRSSNFLVTQGYQVKLAGFELRKDRVKSTAYLSPQELEDVFYQYDVKSEIYSFGIVLWEIATGDIPFQGCNSEKIRKLVAVKRQQEPLGEDCPSELREIIDECRAHDPSVRPSVDEILKKLSTFS 5ko5 A 1.36 BS01 CYT A 1 L118 A119 G120 Y202 E203 M221 L114 A115 G116 Y198 E199 M217 S35 H66 H88 Y90 E91 L118 M221 S222 N245 S247 H259 S31 H62 H84 Y86 E87 L114 M217 S218 N241 S243 H255 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 remove_due_to_license_issue A0A0U3AGT1 30192840 301 VVANYENASMAADYIKRVSNVLPDIGIICGSGLGKLIEEIEERKVIPYINIPNFPKTTVAGHVGNLVLGSVGGRKIVAMQGRLHMYEGYSNQEIALPIRVMKLLGVRVLLITNLAGGINRKLKSGDFVLIKGHINFPGLGLNNVLVGPNQDEFGPRFPDLSNAYDRLLQQLALKIAQENDFQDLVHEGVYAFNGGPTYESPDESNMLLKLGCDVVGMSTVPEVIIACHCGIKVLAVSLIANNSILDAENDVSINHEKVLAVAEKRADLLQMWFKEIITRLPLD 5koq A 2.7 BS01 6VR A 1 T18 Q19 Y20 V36 D38 G40 Y83 T85 D226 T227 G228 A229 S230 T14 Q15 Y16 V32 D34 G36 Y79 T81 D221 T222 G223 A224 S225 D38 S41 N43 W45 D226 A229 D34 S37 N39 W41 D221 A224 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=0.580000nM P00797 27687967 402 NTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5kos A 2.41 BS01 6VS A 1 Q19 Y20 D38 G40 Y83 S84 T85 P118 V127 Y162 L224 D226 G228 A229 Q16 Y17 D35 G37 Y80 S81 T82 P115 V124 Y159 L215 D217 G219 A220 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D217 A220 3.4.23.15 0004190,0006508 ic50=1.5nM remove_due_to_license_issue IC50=0.790000nM P00797 27774132 402 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5kpk A 2.4 BS01 6VK A 1 I62 F67 Y134 V135 R141 Q185 L188 C199 I28 F33 Y97 V98 R104 Q148 L151 C162 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 ic50=0.005uM remove_due_to_license_issue IC50=5nM P49841 29515000 500 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 5kpl A 2.6 BS01 6VL A 1 I62 V70 A83 D133 Y134 V135 P136 L188 C199 I27 V35 A48 D96 Y97 V98 P99 L151 C162 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue IC50=515nM P49841 29515000 500 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 5kpm A 2.69 BS01 6VM A 1 D133 Y134 V135 P136 R141 L188 C199 D95 Y96 V97 P98 R103 L150 C161 D181 K183 N186 D200 S219 D143 K145 N148 D162 S181 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 29515000 500 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 5kq5 A 3.41 BS01 STU A 1 L22 G23 V24 G25 V30 A43 I77 M93 E94 Y95 V96 G99 E100 E143 N144 L146 D157 L13 G14 V15 G16 V21 A34 I68 M84 E85 Y86 V87 G90 E91 E134 N135 L137 D148 D139 K141 E143 N144 D157 S176 D130 K132 E134 N135 D148 S167 2.7.11.1,2.7.11.26,2.7.11.31 0004672,0004679,0005524,0006468 remove_due_to_license_issue P54645 27490827 601 RVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFAKWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDPGSHTIEFFEMCANLIKILAQ 5kqd A 2.6 BS01 PKZ A 1 G19 G20 L22 K24 G116 G191 S192 G193 V194 S195 R207 G210 T211 N322 G9 G10 L12 K14 G75 G135 S136 G137 V138 S139 R151 G154 T155 N266 2.7.1.33 0004594,0005524,0005634,0005737,0005829,0005975,0015937,0016301,0016310,0019842,0042803,1905502 remove_due_to_license_issue Q9H999 27555321 401 SPWFGMDIGGTLVKLSYFEPIEQEEVESLKSIRKYLTSNVAYRDVHLELKDLTLFNLHFIRFPTQDLPTFIQMGGGAYKFEKLHKLDELDCLVKGLLYIDSVSFNGQAECYYFANCQKMPFNLDDPYPLLVVNIGSGVSILAVHSKDNYKRVTGTSLGGGTFLGLCSLLTGCESFEEALEMASKGDSTQADKLVRDIYGGDYERFGLPGWAVASSFGNMIYKEKRESVSKEDLARATLVTITNNIGSVARMCAVNEKINRVVFVGNFLRVNTLSMKLLAYALDYWSKGQLKALFLEHEGYFGAVGALLGLPN 5kqf A 1.98 BS01 6WD A 1 D80 Y119 F156 W163 D276 G278 D34 Y73 F110 W117 D217 G219 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D217 T220 3.4.23.46 0004190,0006508,0016020 ic50=0.31uM remove_due_to_license_issue IC50=310nM P56817 27559936 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5kqg A 1.5 BS01 6VX A 1 C12 L13 G14 I16 C17 R18 Y49 D56 D129 Y131 F138 C9 L10 G11 I13 C14 R15 Y46 D53 D126 Y128 F135 C12 N15 C17 R18 S19 D129 C9 N12 C14 R15 S16 D126 3.1.3.2,3.1.3.48 0003993,0004721,0004725,0004726,0005515,0005737,0005829,0006338,0006470,0009898,0016791,0030946,0042383,0070062,0140793 Ki=3.2uM remove_due_to_license_issue P24666 27676368 200 ATKSVLFVCLGNICRSPIAEAVFRKLVTDQNISENWRVDSAATSGYEIGNPPDYRGQSCMKRHGIPMSHVARQITKEDFATFDYILCMDESNLRDLNRKSNQVKTCKAKIELLGSYDPQKQLIIEDPYYGNDSDFETVYQQCVRCCRAFLEKAH 5kql A 1.45 BS01 6VY A 1 C12 L13 G14 I16 C17 R18 Y49 D56 D129 P130 Y131 F138 C9 L10 G11 I13 C14 R15 Y46 D53 D126 P127 Y128 F135 C12 N15 C17 R18 S19 D129 C9 N12 C14 R15 S16 D126 3.1.3.2,3.1.3.48 0003993,0004721,0004725,0004726,0005515,0005737,0005829,0006338,0006470,0009898,0016791,0030946,0042383,0070062,0140793 remove_due_to_license_issue P24666 27676368 200 ATKSVLFVCLGNICRSPIAEAVFRKLVTDQNISENWRVDSAATSGYEIGNPPDYRGQSCMKRHGIPMSHVARQITKEDFATFDYILCMDESNLRDLNRKSNQVKTCKAKIELLGSYDPQKQLIIEDPYYGNDSDFETVYQQCVRCCRAFLEKAH 5kqx A 2.4 BS01 ROC A 1 N25 G27 D29 D30 G48 G49 I50 P81 I84 N25 G27 D29 D30 G48 G49 I50 P81 I84 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 Ki=3.6nM remove_due_to_license_issue C8BD48 27576689 101 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEDMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kqx B 2.4 BS01 ROC A 1 R8 N25 G48 G49 P81 I84 R8 N25 G48 G49 P81 I84 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue C8BD48 27576689 101 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEDMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kqy A 1.65 BS01 017 B 1 N25 D30 I47 G48 V82 I84 N25 D30 I47 G48 V82 I84 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue C8BD48 27576689 101 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEDMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kqy B 1.65 BS01 017 B 1 N25 G27 A28 D29 G48 I50 N25 G27 A28 D29 G48 I50 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 Ki=0.51nM remove_due_to_license_issue C8BD48 27576689 101 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEDMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr0 A 1.8 BS01 478 A 1 N25 G27 A28 D30 P81 V82 I84 N25 G27 A28 D30 P81 V82 I84 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 Ki=0.71nM remove_due_to_license_issue C8BD48 27576689 101 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEDMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr0 B 1.8 BS01 478 A 1 N25 G27 A28 D30 G48 G49 I50 N25 G27 A28 D30 G48 G49 I50 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue C8BD48 27576689 101 PQITLWKRPLVTIKIGGQLKEALLNTGADDTVIEDMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr1 A 1.6 BS01 017 B 1 N25 G27 A28 I47 G48 V82 N25 G27 A28 I47 G48 V82 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue V5YAB1 27576689 101 PQITLWKRPLVTIKVGGQLKEALLNTGADDTVIEDMNLPGKWKPKMIGGIGGFIKVKQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr1 B 1.6 BS01 017 B 1 N25 G27 A28 D29 D30 G48 I50 N25 G27 A28 D29 D30 G48 I50 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 Ki=0.32nM remove_due_to_license_issue V5YAB1 27576689 101 PQITLWKRPLVTIKVGGQLKEALLNTGADDTVIEDMNLPGKWKPKMIGGIGGFIKVKQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr2 A 1.78 BS01 ROC A 1 N25 G27 A28 D29 D30 G48 G49 I50 P81 N25 G27 A28 D29 D30 G48 G49 I50 P81 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 Ki=3.3nM remove_due_to_license_issue V5YAB1 27576689 101 PQITLWKRPLVTIKVGGQLKEALLNTGADDTVIEDMNLPGKWKPKMIGGIGGFIKVKQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr2 B 1.78 BS01 ROC A 1 N25 G48 I50 P81 I84 N25 G48 I50 P81 I84 N25 T26 G27 N25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue V5YAB1 27576689 101 PQITLWKRPLVTIKVGGQLKEALLNTGADDTVIEDMNLPGKWKPKMIGGIGGFIKVKQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5kr8 A 2.118 BS01 6WE A 1 D80 Y119 T120 Q121 F156 W163 I166 D276 G278 D34 Y73 T74 Q75 F110 W117 I120 D218 G220 D80 S83 N85 A87 Y119 D276 T279 D34 S37 N39 A41 Y73 D218 T221 3.4.23.46 0004190,0006508,0016020 ic50=150nM remove_due_to_license_issue IC50=150nM P56817 27559936 502 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5krb B 2.101 BS01 dna A 0 L85 H86 Y87 K96 K100 L14 H15 Y16 K25 K29 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue Q64249 27984042 105 ~ 120 QRTCLICGDRATGLHYGIISCEGCKGFFKRSISNKRVYRCSRDKNCVMSRKQRNRCQYCRLLKCLQMGMNRKAI 5krb B 2.101 BS02 dna E 0 E93 G94 R101 R107 R121 R124 N125 Q128 R131 E22 G23 R30 R36 R50 R53 N54 Q57 R60 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue Q64249 27984042 89 ~ 104 QRTCLICGDRATGLHYGIISCEGCKGFFKRSISNKRVYRCSRDKNCVMSRKQRNRCQYCRLLKCLQMGMNRKAI 5krb G 2.101 BS01 dna A 0 L85 H86 Y87 K96 K100 I145 R146 G149 P151 G152 R154 N155 L12 H13 Y14 K23 K27 I72 R73 G76 P78 G79 R81 N82 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue Q64249 27984042 105 ~ 120 TCLICGDRATGLHYGIISCEGCKGFFKRSISNKRVYRCSRDKNCVMSRKQRNRCQYCRLLKCLQMGMNRKAIREDGMPGGRN 5krb G 2.101 BS02 dna E 0 E93 G94 F98 R101 R107 R124 N125 Q128 R131 P151 G152 G153 R154 E20 G21 F25 R28 R34 R51 N52 Q55 R58 P78 G79 G80 R81 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue Q64249 27984042 89 ~ 104 TCLICGDRATGLHYGIISCEGCKGFFKRSISNKRVYRCSRDKNCVMSRKQRNRCQYCRLLKCLQMGMNRKAIREDGMPGGRN 5kre A 2.0 BS01 6WG A 1 S30 Y66 R80 I83 S124 M125 L181 V182 S23 Y59 R73 I76 S117 M118 L174 V175 S30 S124 N165 D179 H211 S23 S117 N158 D172 H204 3.1.2.22 0004622,0005515,0005737,0005739,0005829,0008474,0016298,0016787,0016788,0052689,0098734,0160049 remove_due_to_license_issue Q5VWZ2 27391855 301 VLQRCIVSPAGRHSASLIFLHGSGDSGQGLRMWIKQVLNQDLTFQHIKIIYPTAPPRSYTPMKGGISNVWFDRFKITNDCPEHLESIDVMCQVLTDLIDEEVKSGIKKNRILIGGFSMGGCMAMHLAYRNHQDVAGVFALSSFLNKASAVYQALQKSNGVLPELFQCHGTADELVLHSWAEETNSMLKSLGVTTKFHSFPNVYHELSKTELDILKLWILTKLPG 5ks7 A 2.9 BS01 2BA B 1 P259 V260 V280 D281 T282 Y342 T357 R358 A359 P13 V14 V34 D35 T36 Y96 T111 R112 A113 7.6.2.9 remove_due_to_license_issue Q9KHT9 27378384 500 DVTQVAQIMNTNPVSITADKSLQAAITVMKEKRVDTLLVVDEGNVLKGFIDVEQIDLNRRTATSVMDIIEKNVFYVYEDTLLRDTVQRILKRGYKYIPVVDKDKRLVGIVTRASLVDIVYDSI 5ks7 B 2.9 BS01 2BA B 1 V260 V280 D281 T282 Y342 I355 T357 R358 A359 V13 V33 D34 T35 Y95 I108 T110 R111 A112 7.6.2.9 remove_due_to_license_issue Q9KHT9 27378384 500 VTQVAQIMNTNPVSITADKSLQAAITVMKEKRVDTLLVVDEGNVLKGFIDVEQIDLNRRTATSVMDIIEKNVFYVYEDTLLRDTVQRILKRGYKYIPVVDKDKRLVGIVTRASLVDIVYDSI 5ksx F 2.65 BS02 7AM F 1 E318 Y322 R346 Y349 K350 R351 E306 Y310 R334 Y337 K338 R339 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=3700nM P14324 28208018 402 VYAQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKR 5ksx F 2.65 BS03 7AM F 2 K57 N59 F239 R346 K347 I348 K350 K46 N48 F227 R334 K335 I336 K338 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=3700nM P14324 28208018 403 VYAQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKR 5ktu A 1.38 BS01 6XB A 1 P1110 V1115 L1120 N1168 P22 V27 L32 N80 2.3.1.-,2.3.1.48 remove_due_to_license_issue IC50=620nM Q92793 27682507 1201 ELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQS 5ktw A 1.087 BS01 6XG A 1 L1109 P1110 V1115 L1120 I1122 N1168 R1173 V1174 L27 P28 V33 L38 I40 N86 R91 V92 2.3.1.-,2.3.1.48 remove_due_to_license_issue IC50=20.0nM Q92793 27682507 1201 AAFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQAL 5ktx A 1.27 BS01 6XH A 1 L1109 P1110 V1115 I1122 N1168 R1173 V1174 L27 P28 V33 I40 N86 R91 V92 2.3.1.-,2.3.1.48 remove_due_to_license_issue IC50=20nM, EC50=1900nM Q92793 27682507 1201 AAFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQAL 5ku3 A 1.14 BS01 6XH A 1 W81 L92 Y139 I146 W40 L51 Y98 I105 ? remove_due_to_license_issue IC50=10510nM O60885 27682507 211 STNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5ku6 A 1.8 BS01 MZM A 1 Q92 H94 H119 L198 T199 T200 Q95 H97 H122 L199 T200 T201 H64 H94 H96 E106 H119 T199 H70 H97 H99 E109 H122 T200 4.2.1.1 0004089,0005515,0005791,0005793,0005794,0005802,0005886,0006730,0008270,0009897,0009986,0015701,0016020,0016323,0016324,0016829,0030658,0030667,0031526,0046872,0048471,0070062,0098552 remove_due_to_license_issue Ki=6200nM, IC50=205nM P22748 28975383 301 AESHWCYEVQAESSNYPCLVPVKWGGNCQKDRQSPINIVTTKAKVDKKLGRFFFSGYDKKQTWTVQNNGHSVMMLLENKASISGGGLPAPYQAKQLHLHWSDLPYKGSEHSLDGEHFAMEMHIVHEKEKGTSDPEDEIAVLAFLVEAGTQVNEGFQPLVEALSNIPKPEMSTTMAESSLLDLLPKEEKLRHYFRYLGSLTTPTCDEKVVWTVFREPIQLHREQILAFSQKLYYDKEQTVSMKDNVRPLQQLGQRTVIKS 5ku9 A 2.2 BS01 6XJ A 1 H224 A227 M231 H252 V253 D256 R263 T266 F270 H51 A54 M58 H79 V80 D83 R90 T93 F97 3.6.1.11 0042981 ic50=1.49uM remove_due_to_license_issue P97287,Q07820 28197319 402 DDLYRQSLEIISRYLREQATGSKKPLGEAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 5kup A 1.389 BS01 6XL A 1 L408 G411 F413 V416 K430 M477 A478 G480 L528 D539 L542 S543 Y551 L15 G18 F20 V23 K37 M84 A85 G87 L135 D146 L149 S150 Y158 D521 A523 R525 N526 D539 F559 D128 A130 R132 N133 D146 F166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7.2nM remove_due_to_license_issue Q06187 27571029 706 SWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 5kv8 A 1.949 BS02 6Y6 A 1 R192 K254 E276 Y319 Y337 E409 R424 R502 Y530 R50 K112 E134 Y177 Y195 E267 R282 R360 Y388 3.2.1.18 0004308,0019031,0019058,0046789 ic50=14.5uM remove_due_to_license_issue G8G134 28674426 606 THDVGIKPLNPDDFWRCTSGLPSLMKTPKIRLMPGPGLLAMPTTVDGCVRTPSLVINDLIYAYTSNLITRGCQDIGKSYQVLQIGIITVNSDLVPDLNPRISHTFNINDNRKSCSLALLNTDVYQLCSTPKVDERSDYASSGIEDIVLDIVNHDGSISTTRFKNNNISFDQPYAALYPSVGPGIYYKGKIIFLGYGGLEHPINENAICNTTGCPGKTQRDCNQASHSPWFSDRRMVNSIIVVDKGLNSIPKLKVWTISMRQNYWGSEGRLLLLGNKIYIYTRSTSWHSKLQLGIIDITDYSDIRIKWTWHNVLSRPGNNECPWGHSCPDGCITGVYTDAYPLNPTGSIVSSVILDSQKSRVNPVITYSTATERVNELAIRNKTLSAGYTTTSCITHYNKGYCFHIVEINHKSLDTFQPMLFKTEIPKSCS 5kv9 B 2.0 BS02 I57 B 1 R192 I210 D216 K254 E276 Y319 Y337 E409 R424 R502 Y530 R52 I70 D76 K114 E136 Y179 Y197 E267 R282 R360 Y388 3.2.1.18 0004308,0019031,0019058,0046789 ic50=1.4uM remove_due_to_license_issue G8G134 28674426 605 RITHDVGIKPLNPDDFWRCTSGLPSLMKTPKIRLMPGPGLLAMPTTVDGCVRTPSLVINDLIYAYTSNLITRGCQDIGKSYQVLQIGIITVNSDLVPDLNPRISHTFNINDNRKSCSLALLNTDVYQLCSTPKVDERSDYASSGIEDIVLDIVNHDGSISTTRFKNNNISFDQPYAALYPSVGPGIYYKGKIIFLGYGGLEHPINENAICNTTGCPGKTQRDCNQASHSPWFSDRRMVNSIIVVDKNSIPKLKVWTISMRQNYWGSEGRLLLLGNKIYIYTRSTSWHSKLQLGIIDITDYSDIRIKWTWHNVLSRPGNNECPWGHSCPDGCITGVYTDAYPLNPTGSIVSSVILDSQKSRVNPVITYSTATERVNELAIRNKTLSAGYTTTSCITHYNKGYCFHIVEINHKSLDTFQPMLFKTEIPKSCS 5kva A 1.827 BS01 SAM A 1 M75 T77 G101 V102 Y103 S107 D125 I126 P153 A154 D177 A178 D179 Y186 M41 T43 G67 V68 Y69 S73 D91 I92 P119 A120 D143 A144 D145 Y152 D177 K180 G209 S210 D143 K146 G175 S176 2.1.1.104 0008168,0008171,0008757,0009809,0032259,0046872 Kd=7.32uM remove_due_to_license_issue C5Z4W3 27457122 301 KSLLKSDDLYQYILDTSVYPREPESMKELREITAKHPWNLMTTSADEGQFLNMLIKLIGAKKTMEIGVYTGYSLLATALALPEDGTILAMDINRENYELGLPCIEKAGVAHKIDFREGPALPVLDDLIADEKNHGSFDFVFVDADKDNYLNYHDRLLKLVKLGGLIGYDNTLWNGSVVLPDDAPMRKYIRFYRDFVLVLNKALAADERVEICQLPVGDGVTLCRRVK 5kw2 A 2.76 BS01 6XQ A 1 P40 Y44 G95 A99 A102 Y114 S123 V126 I130 L133 L189 L193 P194 P32 Y36 G87 A91 A94 Y106 S115 V118 I122 L125 L160 L164 P165 E1011 D1020 E194 D203 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue O14842,P00720 29695780 2401 LPPQLSFGLYVAAFALGFPLNVLAIRGATATPSAVYALNLGCSDLLLTVSLPLKAVEALASGAWPLPASLCPVFAVAHFAPLYAGGGFLAALSAARYLGAAFPLGYQAFRRPCYSWGVCAAIWALVLCHLGLVFGLEAPVCLEAWDPASAGPARFSLSLLLFFLPLAITAFCFVGCLRALARGSNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYGSLTHRRKLRAAWVAGGALLTLLLCVGPYNASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGY 5kww F 2.5 BS01 6YA F 1 F140 F488 D489 F68 F410 D411 ? 0019064 Kd=7.4nM remove_due_to_license_issue M1E1E4,P03420 28761099 613 NITEEFYQSTCSAVSKGYLSALRTGWYTSVITIELSNIKAKVKLIKQELDKYKNAVTELQLLMQFLGFLLGVGSAIASGVAVCKVLHLEGEVNKIKSALLSTNKAVVSLSNGVSVLTFKVLDLKNYIDKQLLPISISNIETVIEFQQKNNRLLEITREFSVNAGVTTPVSTYMLTNSELLSLINDMPITNDQKKLMSNNVQIVRQQSYSIMCIIKEEVLAYVVQLPLYGVIDTPCWKLHTSPLCTTNTKEGSNICLTRTDRGWYCDNAGSVSFFPQAETCKVQSNRVFCDTMNSLTLPSEVNLCNVDIFNPKYDCKIMTSKTDVSSSVITSLGAIVSCYGKTKCTASNKNRGIIKTFSNGCDYVSNKGVDTVSVGNTLYYVNKQEGKSLYVKGEPIINFYDPLVFPSDEFDASISQVNEKINQSLAFI 5kx7 B 2.8 BS01 6YD B 1 M192 V200 A211 K213 V246 Y262 Y264 M265 G268 L318 M30 V38 A49 K51 V80 Y96 Y98 M99 G102 L152 D311 K313 A315 N316 D329 T351 D145 K147 A149 N150 D163 T181 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=36nM Q9NWZ3 27476420 9901 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5kx8 A 2.671 BS01 6YE A 1 M192 V200 A211 Y262 M265 G268 A315 N316 L318 S328 D329 M30 V38 A49 Y95 M98 G101 A148 N149 L151 S161 D162 D311 K313 A315 N316 D329 T351 D144 K146 A148 N149 D162 T180 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=38nM Q9NWZ3 27476420 501 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5kxc A 1.8 BS01 6Y2 A 1 D117 G135 F159 N161 G244 L245 S246 H249 D87 G105 F129 N131 G214 L215 S216 H219 ? 0030246,0046872 remove_due_to_license_issue A0A1D5B395 27601469 303 KETTSFVFTRFSPDPQNLLLQGDTVVTSSGHLQLTQVKDGEPVYSSLGRALYYAPIHIWDSNTDTVANFVTSFSFVIDAPNKAKAADGLAFFLAPVDTEPQKPGGLLGLFHDDRHNKSNHIVAVEFDTFKNSWDPEGTHIGINVNSIVSRKTISWDLENDEVANVVISYQASTKTLTASLVYPSSSTSYILNDVVDLKQILPEYVRVGFTAASGLSKDHVETHDVLAWTFDSDLPDPS 5kxi A 3.941 BS01 NCT A 1 Y100 W156 T157 Y204 Y93 W149 T150 Y197 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue Ki=2nM, IC50=430nM, EC50=2400nM P43681 27698419 402 AHAEERLLKKLFSGYNKWSRPVANISDVVLVRFGLSIAQLIDVDEKNQMMTTNVWVKQEWHDYKLRWDPADYENVTSIRIPSELIWRPDIVLYNNADGDFAVTHLTKAHLFHDGRVQWTPPAIYKSSCSIDVTFFPFDQQNCTMKFGSWTYDKAKIDLVNMHSRVDQLDFWESGEWVIVDAVGTYNTRKYECCAEIYPDITYAFVIRRLPLFYTINLIIPCLLISCLTVLVFYLPSECGEKITLCISVLLSLTVFLLLITEIIPSTSLVIPLIGEYLLFTMIFVTLSIVITVFVLNVHHRSPRTHTMPTWVRRVFLDIVPRLLLERSVKEDWKYVAMVIDRIFLWMFIIVCLLGTVGLFLPPW 5kxi B 3.941 BS01 NCT A 1 W57 L121 W57 L121 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue IC50=3.8nM, Ki=12.0nM, EC50=132000nM P17787 27698419 402 TDTEERLVEHLLDPSRYNKLIRPATNGSELVTVQLMVSLAQLISVHEREQIMTTNVWLTQEWEDYRLTWKPEEFDNMKKVRLPSKHIWLPDVVLYNNADGMYEVSFYSNAVVSYDGSIFWLPPAIYKSACKIEVKHFPFDQQNCTMKFRSWTYDRTEIDLVLKSEVASLDDFTPSGEWDIVALPGRRNENPDDSTYVDITYDFIIRRKPLFYTINLIIPCVLITSLAILVFYLPSDCGEKMTLCISVLLALTVFLLLISKIVPPTSLDVPLVGKYLMFTMVLVTFSIVTSVCVLNVHHRSPTTHTMAPWVKVVFLEKLPALLFSEDWKYVAMVIDRLFLWIFVFVCVFGTIGMFLQPL 5kya A 2.598 BS01 6Y4 A 1 F271 L274 S278 M312 F329 L330 L345 H435 F48 L51 S55 M89 F106 L107 L122 H212 ? 0003677,0004879,0006629 remove_due_to_license_issue EC50=46nM, Ki=6.0nM P55055 27599745 501 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGSASQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDKILHRLLQD 5kyj A 2.8 BS01 6Y8 A 1 F271 L274 A275 M312 R319 F329 L330 H435 Q438 W457 F54 L57 A58 M95 R102 F112 L113 H218 Q221 W240 ? 0003677,0004879,0006629 remove_due_to_license_issue Ki=13nM, EC50=15nM P55055 27599745 501 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGADPASGSASQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVKILHRLLQD 5kyk A 2.702 BS01 6ZD A 1 C12 G13 G15 A18 F28 D30 N116 K117 D119 S145 A146 K147 C13 G14 G16 A19 F29 D31 N108 K109 D111 S137 A138 K139 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 28105276 201 GMTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDDSYRKQVVIDGETCLLDILDTAGQERDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 5kz0 A 2.3 BS01 6YL A 1 L1122 H1124 G1125 V1130 A1148 M1199 G1202 L1256 G1269 D1270 L30 H32 G33 V38 A48 M99 G102 L156 G169 D170 D1249 A1251 R1253 N1254 D1270 D149 A151 R153 N154 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=22nM remove_due_to_license_issue Ki=22nM Q9UM73 24819116 1501 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIGGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5kzi A 2.1 BS01 6YN A 1 L44 F49 V52 A65 K67 L120 R122 V126 D128 E171 L174 I185 D186 L12 F17 V20 A33 K35 L88 R90 V94 D96 E139 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.07nM remove_due_to_license_issue IC50=0.08nM P11309 27769621 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5kzq A 2.8 BS01 6YS A 1 R61 S143 Y144 S145 A166 S167 T168 Y216 R271 R36 S96 Y97 S98 A119 S120 T121 Y169 R224 ? 0004930,0007186,0016020 remove_due_to_license_issue Q14416 28002967 601 KVLTLEGDLVLGGLFPVHQKPAEDCGPVNEHRGIQRLEAMLFALDRINRDPHLLPGVRLGAHILDSCSKDTHALEQALDFVRASLPTAITGVIGGSYSDVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFFQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFELEARARNICVATSEKVGRAMSRAAFEGVVRALLQKPSARVAVLFTRSEDARELLAASQRLNASFTWVASDGWGALESVVAGSEGAAEGAITIELASYPISDFASYFQSLDPWNNSRNPWFREFWEQRFRCSFRQRDCAAHSLRAVPFEQESKIMFVVNAVYAMAHALHNMHRALCPNTTRLCDAMRPVNGRRLYKDFVLNVKFDAPFRPADTHNEVRFDRFGDGIGRYNIFTYLRAGGRYRYQKVGYWAEGLTLDTSLIPWASPSAGPLPASRCSEPCLQNEVKSVQPGEVCCWLCIPCQPYEYRLDEFTCADCGLGYWPNASLT 5l01 A 1.9 BS02 6Z4 A 1 Y235 P238 R257 Y264 T265 P266 H272 A309 E317 G333 S336 S337 Y124 P127 R146 Y153 T154 P155 H161 A198 E206 G222 S225 S226 H272 H277 E317 S336 H161 H166 E206 S225 1.14.16.4 0002576,0004497,0004510,0005506,0005515,0005737,0005829,0007623,0009072,0016714,0030279,0035902,0042427,0043005,0045600,0046849,0046872,0060749,1900046 ic50=33nM remove_due_to_license_issue IC50=33nM P17752 28041831 502 TVPWFPKKISDLDHCANRVLMYGGFKDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFQELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTIK 5l0h A 2.9 BS01 PIO A 1 W975 K979 K1103 R1107 R1128 W16 K20 K144 R148 R169 ? 0003779,0007155,0051015 remove_due_to_license_issue P18206 27503891 1202 QPVNQPILAAAQSLHWEATKWSSKGNDIIAAAKRMALLMAEMSRLVRGGSGTKRALIQCAKDIAKASDEVTRLAKEVAKQCTDKRIRTNLLQVCERIPTISTQLKILSTVKATMLGRTNISDEESEQATEMLVHNAQNLMQSVKETVREAEAASIKIRTDAGFTLRWVRKTPW 5l0m A 2.197 BS01 dna C 0 E104 S105 R112 R135 K136 R142 R162 G163 G164 R165 E22 S23 R30 R53 K54 R60 R80 G81 G82 R83 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue O00482 27984042 89 ~ 100 EELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRYTCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRAL 5l0m A 2.197 BS02 dna B 0 Y96 H97 Y98 K107 K111 V156 R157 R160 M161 R162 R165 N166 Y172 Y14 H15 Y16 K25 K29 V74 R75 R78 M79 R80 R83 N84 Y90 ? 0003677,0003700,0004879,0006355,0008270,0043565 remove_due_to_license_issue O00482 27984042 107 ~ 118 EELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRYTCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRAL 5l13 A 2.4 BS01 6ZE A 1 F170 M174 W177 F296 C301 C302 C303 D457 F459 F164 M168 W171 F290 C295 C296 C297 D451 F453 N169 K192 E268 C302 E399 E476 N163 K186 E262 C296 E393 E470 1.2.1.3 0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627 Ki=19nM remove_due_to_license_issue Ki=19nM, IC50=110nM P05091 28219011 606 AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS 5l15 A 2.4 BS02 G39 A 1 R119 E120 D152 R226 R294 R372 Y406 R37 E38 D70 R144 R212 R290 Y324 D152 E279 R294 R372 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue R4NFR6 28934455 512 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCRDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 5l17 A 2.4 BS02 ZMR A 1 R119 E120 D152 R153 W180 R226 E229 A248 E278 R294 R372 Y406 R37 E38 D70 R71 W98 R144 E147 A166 E196 R212 R290 Y324 D152 E279 R294 R372 Y406 D70 E197 R212 R290 Y324 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue R4NFR6 28934455 512 RNFNNLTKGLCTINSWHIYGKDNAVRIGESSDVLVTREPYVSCDPDECRFYALSQGTTIRGKHSNGTIHDRSQYRALISWPLSSPPTVYNSRVECIGWSSTSCHDGKSRMSICISGPNNNASAVVWYNRRPVAEINTWARNILRTQESECVCHNGVCPVVFTDGSATGPADTRIYYFKEGKILKWESLTGTAKHIEECSCYGERTGITCTCRDNWQGSNRPVIQIDPVAMTHTSQYICSPVLTDNPRPNDPNIGKCNDPYPGNNNNGVKGFSYLDGANTWLGRTISTASRSGYEMLKVPNALTDDRSKPIQGQTIVLNADWSGYSGSFMDYWAEGDCYRACFYVELIRGRPKEDKVWWTSNSIVSMCSSTEFLGQWNWPDGAKIEYFL 5l1z B 5.9 BS01 rna N 0 R259 C261 R253 C255 ? 0006357,0016538 remove_due_to_license_issue O60563 27731797 21 ~ 41 NNNKRWYFTREQLENSPSRRFGVDPDKELSYRQQAANLLQDMGQRLNVSQLTINTAIVYMHRFYMIQSFTQFPGNSVAPAALFLAAKVEEQPKKLEHVIKVAHTCLHPQESLPDTRSEAYLQQVQDLVILESIILQTLGFELTIDHPHTHVVKCTQLVRASKDLAQTSYFMATNSLHLTTFSLQYTPPVVACVCIHLACKWSNWEIPVSTDGKHWWEYVDATVTLELLDELTHEFLQILEKTPNRLKRIWNWRAC 5l1z D 5.9 BS01 rna N 0 N24 C25 Y26 N24 C25 Y26 ? 0001070,0042025,0050434 remove_due_to_license_issue P69697 27731797 21 ~ 41 MEPVDPRLEPWKHPGSQPKTACTNCYCKKCCFHCQVCFITKALGISYGR 5l26 A 3.4 BS04 URI A 1 Q154 E332 F333 F366 S371 V374 Q156 E329 F330 F363 S368 V371 ? 0005337,0005886,0015293,0016020,1901642 remove_due_to_license_issue G4CRQ5 28424521 505 PRMVVLHSLLGMAVLIAIAVLLSTDRKAINIRTVAGAFLIQVALGALVLYVPQGRDMLGEASKTISNVIAYGNNGVDFLFGGLVSEKMFEVFGGGGFVFALRVLPMIVFFSSLMAVLYYIGVMQLLIKVIGGFLQKMLGTSKAESMSAAANIFVGQTEAPLVVRPYIRRMTESELFAVMSGGLASVAGSVLAGYVQMGVPLPYLIAASFMAAPGGLLFAKLLVPETERTQNDAEVLAENEDEKPTNVIDAAASGAVTGAQIAIAVGASLLAFVALIAMINGIIGGVGGDLTLQAILGWLFSPLAWVIGVPWSEAGIAGSLIGQKVVINEFVAYSEFVKYLKPEAAVQLSDTTKAIISFALCGFANLGSIAVLVGGLSIMAPKRRKDVARLGIKAVVAGSLSNLMSAVIAGLFTGLSGAS 5l2i A 2.75 BS01 LQQ A 1 I19 A41 F98 V101 T107 Q149 L152 D163 I10 A32 F73 V76 T82 Q124 L127 D138 D145 K147 Q149 N150 D163 T182 D120 K122 Q124 N125 D138 T143 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue IC50=16nM, Ki=27nM Q00534 27496135 900 DQQYECVAEIGEGAYGKVFKARDLKNGGRFVALKRVRPLSTIREVAVLRHLETFEHPNVVRLFDVCTKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPRDVALPRQAFKSAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQ 5l2m A 1.7 BS01 6ZY A 1 F171 F290 H293 Y297 F164 F283 H286 Y290 N170 K193 E269 C303 E400 E477 N163 K186 E262 C296 E393 E470 1.2.1.19,1.2.1.28,1.2.1.3,1.2.1.36 0000166,0001523,0001758,0004029,0005096,0005497,0005515,0005737,0005829,0006081,0006629,0009449,0016491,0016620,0018479,0019145,0030392,0030424,0036438,0042572,0042995,0045202,0051287,0070062,0106373,0110095,0120163 Ki=170nM remove_due_to_license_issue Ki=170nM, IC50=130nM P00352 28219011 602 DLPVLLTDLKIQYTKIFINNEWHDSVSGKKFPVFNPATEEELCQVEEGDKEDVDKAVKAARQAFQIGSPWRTMDASERGRLLYKLADLIERDRLLLATMESMNGGKLYSNAYLNDLAGCIKTLRYCAGWADKIQGRTIPIDGNFFTYTRHEPIGVCGQIIPWNFPLVMLIWKIGPALSCGNTVVVKPAEQTPLTALHVASLIKEAGFPPGVVNIVPGYGPTAGAAISSHMDIDKVAFTGSTEVGKLIKEAAGKSNLKRVTLELGGKSPCIVLADADLDNAVEFAHHGVFYHQGQCCIAASRIFVEESIYDEFVRRSVERAKKYILGNPLTPGVTQGPQIDKEQYDKILDLIESGKKEGAKLECGGGPWGNKGYFVQPTVFSNVTDEMRIAKEEIFGPVQQIMKFKSLDDVIKRANNTFYGLSAGVFTKDIDKAITISSALQAGTVWVNCYGVVSAQCPFGGFKMSGNGRELGEYGFHEYTEVKTVTVKISQKNS 5l2n A 1.7 BS01 6ZU A 1 F171 M175 W178 H293 G294 Y297 C302 C303 I304 Y457 G458 V460 F466 F164 M168 W171 H286 G287 Y290 C295 C296 I297 Y450 G451 V453 F459 N170 K193 E269 C303 E400 E477 N163 K186 E262 C296 E393 E470 1.2.1.19,1.2.1.28,1.2.1.3,1.2.1.36 0000166,0001523,0001758,0004029,0005096,0005497,0005515,0005737,0005829,0006081,0006629,0009449,0016491,0016620,0018479,0019145,0030392,0030424,0036438,0042572,0042995,0045202,0051287,0070062,0106373,0110095,0120163 ic50=2.8uM remove_due_to_license_issue IC50=2800nM P00352 28219011 602 DLPVLLTDLKIQYTKIFINNEWHDSVSGKKFPVFNPATEEELCQVEEGDKEDVDKAVKAARQAFQIGSPWRTMDASERGRLLYKLADLIERDRLLLATMESMNGGKLYSNAYLNDLAGCIKTLRYCAGWADKIQGRTIPIDGNFFTYTRHEPIGVCGQIIPWNFPLVMLIWKIGPALSCGNTVVVKPAEQTPLTALHVASLIKEAGFPPGVVNIVPGYGPTAGAAISSHMDIDKVAFTGSTEVGKLIKEAAGKSNLKRVTLELGGKSPCIVLADADLDNAVEFAHHGVFYHQGQCCIAASRIFVEESIYDEFVRRSVERAKKYILGNPLTPGVTQGPQIDKEQYDKILDLIESGKKEGAKLECGGGPWGNKGYFVQPTVFSNVTDEMRIAKEEIFGPVQQIMKFKSLDDVIKRANNTFYGLSAGVFTKDIDKAITISSALQAGTVWVNCYGVVSAQCPFGGFKMSGNGRELGEYGFHEYTEVKTVTVKISQKNS 5l2o A 2.05 BS01 6ZW A 1 G226 G230 A231 V250 L253 G219 G223 A224 V243 L246 N170 K193 E269 C303 E400 E477 N163 K186 E262 C296 E393 E470 1.2.1.19,1.2.1.28,1.2.1.3,1.2.1.36 0000166,0001523,0001758,0004029,0005096,0005497,0005515,0005737,0005829,0006081,0006629,0009449,0016491,0016620,0018479,0019145,0030392,0030424,0036438,0042572,0042995,0045202,0051287,0070062,0106373,0110095,0120163 ic50=0.76uM remove_due_to_license_issue Ki=870nM, IC50=760nM P00352 28219011 601 DLPVLLTDLKIQYTKIFINNEWHDSVSGKKFPVFNPATEEELCQVEEGDKEDVDKAVKAARQAFQIGSPWRTMDASERGRLLYKLADLIERDRLLLATMESMNGGKLYSNAYLNDLAGCIKTLRYCAGWADKIQGRTIPIDGNFFTYTRHEPIGVCGQIIPWNFPLVMLIWKIGPALSCGNTVVVKPAEQTPLTALHVASLIKEAGFPPGVVNIVPGYGPTAGAAISSHMDIDKVAFTGSTEVGKLIKEAAGKSNLKRVTLELGGKSPCIVLADADLDNAVEFAHHGVFYHQGQCCIAASRIFVEESIYDEFVRRSVERAKKYILGNPLTPGVTQGPQIDKEQYDKILDLIESGKKEGAKLECGGGPWGNKGYFVQPTVFSNVTDEMRIAKEEIFGPVQQIMKFKSLDDVIKRANNTFYGLSAGVFTKDIDKAITISSALQAGTVWVNCYGVVSAQCPFGGFKMSGNGRELGEYGFHEYTEVKTVTVKISQKNS 5l2s A 2.27 BS01 6ZV A 1 I19 Y24 A41 K43 F98 V101 D104 L152 D163 I9 Y14 A31 K33 F73 V76 D79 L127 D138 D145 K147 Q149 N150 D163 T182 D120 K122 Q124 N125 D138 T144 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue IC50=10.0nM, Ki=8.2nM Q00534 27496135 900 QQYECVAEIGEGAYGKVFKARDLKNGGRFVALKRVRVPLSTIREVAVLRHLETFEHPNVVRLFDVCTKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLAVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPRDVALPRQAFHSKSAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQ 5l2t A 2.37 BS01 6ZZ A 1 I19 A41 F98 V101 D104 L152 D163 I9 A31 F71 V74 D77 L125 D136 D145 K147 Q149 N150 D163 T182 D118 K120 Q122 N123 D136 T142 2.7.11.22 0000082,0000122,0000307,0001726,0001954,0002244,0003323,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006468,0007165,0007219,0008285,0009615,0010389,0010468,0010628,0014002,0016301,0021542,0021670,0030097,0030154,0030332,0033077,0042063,0042127,0042995,0043697,0045596,0045638,0045646,0045656,0045668,0045786,0048146,0048699,0050680,0051301,0051726,0060218,0097131,0097132,0097133,0098770,0106310,1902036,2000145,2000773 remove_due_to_license_issue IC50=39nM Q00534 27496135 900 QQYECVAEIGEGAYGKVFKARDLKNGGRFVALKRVRVSTIREVAVLRHLETFEHPNVVRLFDVCTKLTLVFEHVDQDLTTYLDKVPEPGVPTETIKDMMFQLLRGLDFLHSHRVVHRDLKPQNILVTSSGQIKLADFGLAVTLWYRAPEVLLQSSYATPVDLWSVGCIFAEMFRRKPLFRGSSDVDQLGKILDVIGLPGEEDWPRDVALPRQAFHSKSAQPIEKFVTDIDELGKDLLLKCLTFNPAKRISAYSALSHPYFQ 5l2w A 2.8 BS01 1QK A 1 I10 A31 F80 F82 L83 Q85 L134 A144 I11 A32 F81 F83 L84 Q86 L135 A145 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 27496135 900 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLR 5l2y H 1.82 BS01 70D H 1 H57 K60A G97 T99 D189 S190 K192 S195 S214 W215 G216 G219 H41 K45 G85 T87 D186 S187 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=0.14nM remove_due_to_license_issue Ki=0.140000nM P08709 27612545 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5l2z H 1.79 BS01 70C H 1 L41 H57 G97 T99 D189 S190 K192 S195 S214 W215 G216 G219 L25 H41 G85 T87 D186 S187 K189 S192 S211 W212 G213 G215 3.4.21.21 0004252,0006508 Ki=0.06nM remove_due_to_license_issue Ki=0.060000nM P08709 27612545 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5l30 H 1.73 BS01 70A H 1 H57 C58 K60A G97 T99 D189 S190 K192 S195 S214 W215 G216 Q217 G219 H41 C42 K45 G85 T87 D183 S184 K186 S189 S208 W209 G210 Q211 G212 3.4.21.21 0004252,0006508 remove_due_to_license_issue Ki=0.12nM P08709 27612545 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5l3a A 1.98 BS01 6DP A 1 G856 V863 A880 M929 L932 L983 G16 V23 A40 M89 L92 L143 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0004713,0005524,0006468 Kd=13uM remove_due_to_license_issue Kd=12589nM, IC50=13000nM O60674 27326341 1201 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEFFKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 5l3e A 2.8 BS02 E11 A 1 L386 N535 L536 A539 W552 H564 W695 L216 N365 L366 A369 W382 H394 W525 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue Kd=243nM O60341 27626075 902 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5l3e A 2.8 BS03 E11 A 2 N383 E387 S390 D556 E559 N213 E217 S220 D386 E389 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue Kd=243nM O60341 27626075 903 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5l3e A 2.8 BS04 E11 A 3 E559 G562 E389 G392 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue Kd=243nM O60341 27626075 904 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5l3e A 2.8 BS05 E11 A 4 D557 E559 D387 E389 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue Kd=243nM O60341 27626075 905 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5l3j A 2.83 BS01 6G9 A 1 V43 N46 E50 V71 D73 R76 G77 I78 P79 V120 T165 V29 N32 E36 V57 D59 R62 G63 I64 P65 V88 T133 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue IC50=58nM, Kd=230nM P0AES6 27541007 401 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLHVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYEGGIKAFVEYLNKNKTPIHPNIFYFSTEKDGIGVEVALQWNDGFQENIYCFTNNIPQRDGGTHLAGFRAAMTRTLNAYMDKEGYSKKAKVSATGDDAREGLIAVVSVKVPDPKFSSQTKDKLVSSEVKSAVEQQMNELLAEYLLENPTDAKIVVGKIIDAARAREAARRAREMT 5l44 A 1.75 BS03 K26 A 1 R415 A418 W419 M420 H463 E464 H467 T484 R488 E492 H593 S597 Y599 Y606 R406 A409 W410 M411 H454 E455 H458 T475 R479 E483 H584 S588 Y590 Y597 H463 E464 H467 Y606 H454 E455 H458 Y597 ? 0004180,0004222,0005829,0006508,0008233,0008237,0046872 remove_due_to_license_issue A0A1L1QK30 27754586 1005 ENPFFAPSALPYGLPPFAEIREEHYVPAFERGMAEQLAEVEAIAGDTEAPTFDNTVAALERSGQVLTRVSAVFFNQSSSDTNPTVQEIQKQIIPKLTQHGDAIHLNRPLFARIKQISPDGLDAEQAWLLERYVTDFVRAGAELGAGDQERLKALNEELSTLSTRFEQNLLAHTNASAVIVDDVAQLDGLSDDSVKAAAETAKSRGLPGKYVIPLVLPTGQPGLAELTDRALRERIHRASIQRGVPDNEELIVRIATLRAERAKLLGYPTHAAYVVADQTAPTTEAVTEMLGKLTPPAVANAHREADELREQAGHDLEPWDWSFYAEKVLKERYAIDGRQMRPYFELDRVLRDGVFHAATLLYGITFTERPDLVGYHPDVRVFEVFNEDGSQLGLFLGDYYARPSKRGGAWMNSLVKQSTLEGTRPVVVNNLNIAKPPAGEPTLMTFEEVNTMFHEFGHALHGLFSEVHYPRFSGTAVPRDFVEYPSQVNEMWAVWPSVLANYARHWQTGDPMPKDLLDRMLKSQKYNQGYKTVEYLAATLLDWSWHTFQTPPENALTFEHEALTTAGVDLKLVPPRYRSTYFAHIWSSGYSAGYYSYIWSEVLDADTVDWFHENGGLLRENGDTFRQKLLSKGGSVDPMTAFQSFRGRTPRIEPLLDRRGLL 5l4h C 3.3 BS01 6JW E 1 S230 I233 S226 I229 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 27986812 402 VSPPPPIADEPLTVNTGIYLIESYSLDDCAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNCPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 5l4h D 3.3 BS01 6JW E 1 S230 I233 S226 I229 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 27986812 402 VSPPPPIADEPLTVNTGIYLIESYSLDDCAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNCPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 5l4h E 3.3 BS01 6JW E 1 S230 I233 S226 I229 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q7NDN8 27986812 402 VSPPPPIADEPLTVNTGIYLIESYSLDDCAETFKVNAFLSLSWKDRRLAFDPVRSGVRVKTYEPEAIWIPEIRFVNVENARDADVVDISVSPDGTVQYLERFSARVLSPLDFRRYPFDSQTLHIYLIVRSVDTRNIVLAVDLEKVGKNDDVFLTGWDIESFTAVVKPANFALEDRLESKLDYQLRISRQYFSYIPNIILPMLFILFISWTAFWSTSYEANVTLVVSTLIAHIAFNILVETNCPKTPYMTYTGAIIFMIYLFYFVAVIEVTVQHYLKVESQPARAASITRASRIAFPVVFLLANIILAFLFF 5l4i A 1.45 BS01 6J3 A 1 K15 L17 S117 K6 L8 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.26uM remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5l4i B 1.45 BS01 6J3 B 1 K15 L17 S117 K6 L8 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.26uM remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5l4j A 1.62 BS01 6JD A 1 L17 A108 L8 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=52uM remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5l4m A 1.581 BS01 SBK A 1 K15 L17 A108 A109 K6 L8 A99 A100 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=4.6uM remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5l4m B 1.581 BS01 SBK B 1 K15 L17 A108 A109 K6 L8 A99 A100 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=4.6uM remove_due_to_license_issue P02766 27668830 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5l6h A 2.3 BS01 6O2 B 1 A444 D470 K494 K519 V520 A542 L543 D544 N545 A548 A435 D461 K485 K510 V511 A533 L534 D535 N536 A539 R21 R481 D544 C600 T601 R603 N781 D782 R12 R472 D535 C591 T592 R594 N772 D773 6.2.1.45 0004839,0005515,0005524,0005634,0005737,0006511,0006974,0008641,0016567,0016874,0036211 remove_due_to_license_issue P22515 28578874 101 AAGEIDESLYSRQLYVLGKEAMLKMQTSNVLILGLKGLGVEIAKNVVLAGVKSMTVFDPEPVQLADLSTQFFLTEKDIGQKRGDVTRAKLAELNAYVPVNVLDSLDDVTQLSQFQVVVATDTVSLEDKVKINEFCHSSGIRFISSETRGLFGNTFVDLGDEFTVLDPTGEEPRTGMVSDIEPDGTVTMLDDNRHGLEDGNFVRFSEVEGLDKLNDGTLFKVEVLGPFAFRIGSVKEYGEYKKGGIFTEVKVPRKISFKSLKQQLSNPEFVFSDFAKFDRAAQLHLGFQALHQFAVRHNGELPRTMNDEDANELIKLVTDLSVQQPEVLGEGVDVNEDLIKELSYQARGDIPGVVAFFGGLVAQEVLKACSGKFTPLKQFMYFDSLESLPDPKNFPRNEKTTQPVNSRYDNQIAVFGLDFQKKIANSKVFLVGSGAIGCEMLKNWALLGLGSGSDGYIVVTDNDSIEKSNLNRQFLFRPKDVGKNKSEVAAEAVCAMNPDLKGKINAKIDKVGPETEEIFNDSFWESLDFVTNALDNVDARTYVDRRCVFYRKPLLESGTLGTKGNTQVIIPRLTESYSSSRDPPEKSIPLCTLRSFPNKIDHTIAWAKSLFQGYFTDSAENVNMYLTQPNFVEQTLKQSGDVKGVLESISDSLSSKPHNFEDCIKWARLEFEKKFNHDIKQLLFNFPKDAKTSNGEPFWSGAKRAPTPLEFDIYNNDHFHFVVAGASLRAYNYGIKSDDSNSKPNVDEYKSVIDHMIIPEFTPNANLKIQVNDDDPDDEIDQLVSSLPDPSTLAGFKLEPVDFEKDDDTNHHIEFITACSNCRAQNYFIETADRQKTKFIAGRIIPAIATTTSLVTGLVNLELYKLIDNKTDIEQYKNGFVNLALPFFGFSEPIASPKGEYNNKKYDKIWDRFDIKGDIKLSDLIEHFEKDEGLEITMLSYGVSLLYASFFPPKKLKERLNLPITQLVKLVTKKDIPAHVSTMILEICADDKEGEDVEVPFITIHL 5l6i A 2.76 BS01 B39 B 1 D470 N471 D472 K494 K519 V520 A542 L543 D544 A548 D461 N462 D463 K485 K510 V511 A533 L534 D535 A539 R21 R481 D544 C600 T601 R603 N781 D782 R12 R472 D535 C591 T592 R594 N772 D773 6.2.1.45 0004839,0005515,0005524,0005634,0005737,0006511,0006974,0008641,0016567,0016874,0036211 remove_due_to_license_issue P22515 28578874 101 AAGEIDESLYSRQLYVLGKEAMLKMQTSNVLILGLKGLGVEIAKNVVLAGVKSMTVFDPEPVQLADLSTQFFLTEKDIGQKRGDVTRAKLAELNAYVPVNVLDSLDDVTQLSQFQVVVATDTVSLEDKVKINEFCHSSGIRFISSETRGLFGNTFVDLGDEFTVLDPTGEEPRTGMVSDIEPDGTVTMLDDNRHGLEDGNFVRFSEVEGLDKLNDGTLFKVEVLGPFAFRIGSVKEYGEYKKGGIFTEVKVPRKISFKSLKQQLSNPEFVFSDFAKFDRAAQLHLGFQALHQFAVRHNGELPRTMNDEDANELIKLVTDLSVQQPEVLGEGVDVNEDLIKELSYQARGDIPGVVAFFGGLVAQEVLKACSGKFTPLKQFMYFDSLESLPDPKNFPRNEKTTQPVNSRYDNQIAVFGLDFQKKIANSKVFLVGSGAIGCEMLKNWALLGLGSGSDGYIVVTDNDSIEKSNLNRQFLFRPKDVGKNKSEVAAEAVCAMNPDLKGKINAKIDKVGPETEEIFNDSFWESLDFVTNALDNVDARTYVDRRCVFYRKPLLESGTLGTKGNTQVIIPRLTESYSSSRDPPEKSIPLCTLRSFPNKIDHTIAWAKSLFQGYFTDSAENVNMYLTQPNFVEQTLKQSGDVKGVLESISDSLSSKPHNFEDCIKWARLEFEKKFNHDIKQLLFNFPKDAKTSNGEPFWSGAKRAPTPLEFDIYNNDHFHFVVAGASLRAYNYGIKSDDSNSKPNVDEYKSVIDHMIIPEFTPNANLKIQVNDDDPDPDEIDQLVSSLPDPSTLAGFKLEPVDFEKDDDTNHHIEFITACSNCRAQNYFIETADRQKTKFIAGRIIPAIATTTSLVTGLVNLELYKLIDNKTDIEQYKNGFVNLALPFFGFSEPIASPKGEYNNKKYDKIWDRFDIKGDIKLSDLIEHFEKDEGLEITMLSYGVSLLYASFFPPKKLKERLNLPITQLVKLVTKKDIPAHVSTMILEICADDKEGEDVEVPFITIHL 5l6j A 2.68 BS01 61T B 1 G443 A444 D470 K494 K519 V520 A542 L543 D544 N545 D547 A548 Y551 G432 A433 D459 K483 K508 V509 A531 L532 D533 N534 D536 A537 Y540 R21 R481 D544 C600 T601 R603 N781 D782 R10 R470 D533 C589 T590 R592 N770 D771 6.2.1.45 0004839,0005515,0005524,0005634,0005737,0006511,0006974,0008641,0016567,0016874,0036211 remove_due_to_license_issue P22515 28578874 101 GEIDESLYSRQLYVLGKEAMLKMQTSNVLILGLKGLGVEIAKNVVLAGVKSMTVFDPEPVQLADLSTQFFLTEKDIGQKRGDVTRAKLAELNAYVPVNVLDSLDDVTQLSQFQVVVATDTVSLEDKVKINEFCHSSGIRFISSETRGLFGNTFVDLGDEFTVLDPTGEEPRTGMVSDIEPDGTVTMLDDNRHGLEDGNFVRFSEVEGLDKLNDGTLFKVEVLGPFAFRIGSVKEYGEYKKGGIFTEVKVPRKISFKSLKQQLSNPEFVFSDFAKFDRAAQLHLGFQALHQFAVRHNGELPRTMNDEDANELIKLVTDLSVQQPEVLGEGVDVNEDLIKELSYQARGDIPGVVAFFGGLVAQEVLKACSGKFTPLKQFMYFDSLESLPDPKNFPRNEKTTQPVNSRYDNQIAVFGLDFQKKIANSKVFLVGSGAIGCEMLKNWALLGLGSGSDGYIVVTDNDSIEKSNLNRQFLFRPKDVGKNKSEVAAEAVCAMNPDLKGKINAKIDKVGPETEEIFNDSFWESLDFVTNALDNVDARTYVDRRCVFYRKPLLESGTLGTKGNTQVIIPRLTESYSSSRDPPEKSIPLCTLRSFPNKIDHTIAWAKSLFQGYFTDSAENVNMYLTQPNFVEQTLKQSGDVKGVLESISDSLSSKPHNFEDCIKWARLEFEKKFNHDIKQLLFNFPKDAKTSNGEPFWSGAKRAPTPLEFDIYNNDHFHFVVAGASLRAYNYGIKSDDSNSKPNVDEYKSVIDHMIIPEFTPNANLKIQVNDDDPDPSDEIDQLVSSLPDPSTLAGFKLEPVDFEKDDDTNHHIEFITACSNCRAQNYFIETADRQKTKFIAGRIIPAIATTTSLVTGLVNLELYKLIDNKTDIEQYKNGFVNLALPFFGFSEPIASPKGEYNNKKYDKIWDRFDIKGDIKLSDLIEHFEKDEGLEITMLSYGVSLLYASFFPPKKLKERLNLPITQLVKLVTKKDIPAHVSTMILEICADDKEGEDVEVPFITIHL 5l6o A 1.88 BS01 6P6 A 1 A663 M686 I709 T711 F713 M714 C717 L765 A29 M52 I75 T77 F79 M80 C83 L131 D758 A760 R762 N763 D776 K799 D124 A126 R128 N129 D142 K161 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P54753 27478969 1001 CVKIEEVIGAGEVCRGRLKQPGRREVFVAIKTLKVGYTERQRRDFLSEASIMGQFDHPNIIRLEGVVTKSRPVMILTEFMENCALDSFLRLNDGQFTVIQLVGMLRGIAAGMKYLSEMNYVHRDLAARNILVNSNLVCKVSDFGLEDDPSDPTYTSSLGGKIPIRWTAPEAIAYRKFTSASDVWSYGIVMWEVMSYGERPYWDMSNQDVINAVEQDYRLPPPMDCPTALHQLMLDCWVRDRNLRPKFSQIVNTLDKLIRNPASLKVI 5l6p A 2.26 BS01 6P8 A 1 I639 A663 K665 T711 M714 C717 L765 I8 A32 K34 T80 M83 C86 L134 D758 A760 R762 N763 D776 K799 D127 A129 R131 N132 D145 K168 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P54753 27478969 1001 CVKIEEVIGAGEFGEVCRGRLKQPGRREVFVAIKTLKVGYTERQRRDFLSEASIMGQFDHPNIIRLEGVVTKSRPVMILTEFMENCALDSFLRLNDGQFTVIQLVGMLRGIAAGMKYLSEMNYVHRDLAARNILVNSNLVCKVSDFGLSRFLEDDPSDPTYTSSLGGKIPIRWTAPEAIAYRKFTSASDVWSYGIVMWEVMSYGERPYWDMSNQDVINAVEQDYRLPPPMDCPTALHQLMLDCWVRDRNLRPKFSQIVNTLDKLIRNPASLKVI 5l72 A 3.06 BS01 6PF A 1 M752 S754 P758 K779 I825 V828 M900 I910 D911 M587 S589 P593 K614 I660 V663 M735 I745 D746 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 27429068 4000 RVKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSARGNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLVEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNSLWSLEQPFSIELIEGRKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPHPVYFPALEKILELGRHGERGRITEEEQLQLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVN 5l7e A 1.86 BS02 6Q0 A 1 L769 N770 L772 A773 Q776 W806 M807 L810 S811 M845 M852 F941 C942 L33 N34 L36 A37 Q40 W70 M71 L74 S75 M109 M116 F200 C201 ? Ki=0.25uM remove_due_to_license_issue P08235 27897427 1106 SPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 5l7f A 1.8 BS07 6PJ B 1 K233 Y242 V243 R249 S251 A252 K128 Y137 V138 R144 S146 A147 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue P39900 27564088 301 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYAYVDINTFRLSADDIRGIQSLYG 5l7g A 2.01 BS02 6QE A 1 L769 N770 L772 A773 Q776 W806 M807 L810 S811 L814 F829 M845 C849 M852 L938 F941 C942 L33 N34 L36 A37 Q40 W70 M71 L74 S75 L78 F93 M109 C113 M116 L201 F204 C205 ? Ki=16nM remove_due_to_license_issue P08235 27897427 1102 SPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSPNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 5l7h A 1.84 BS02 6QG A 1 L769 N770 L772 A773 Q776 W806 M807 L810 S811 L814 M845 F941 C942 L35 N36 L38 A39 Q42 W72 M73 L76 S77 L80 M111 F206 C207 ? Ki=50nM remove_due_to_license_issue P08235 27897427 1101 YFSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSPNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 5l87 A 0.87 BS01 6RD A 1 N13 E16 D20 R22 V23 F34 K38 N9 E12 D16 R18 V19 F30 K34 ? 0005778,0016560 Ki=8.43uM remove_due_to_license_issue Q8IEW2 28360328 101 SEREKRVSNAVEFLLDSRVRRTPTSSKVHFLKSKGLSAEEICEAFTKVGQPKTLNEIKRILS 5l8a A 1.57 BS01 6RB A 1 N13 E16 F17 R22 V23 T26 F34 K38 N9 E12 F13 R18 V19 T22 F30 K34 ? 0005778,0016560 Ki=12.3uM remove_due_to_license_issue Q8IEW2 28360328 101 SEREKRVSNAVEFLLDSRVRRTPTSSKVHFLKSKGLSAEEICEAFTKVGQPKTLNEIKRILS 5l8c A 2.01 BS02 908 A 1 M785 D822 Y845 N867 E869 F877 M200 D237 Y260 N282 E284 F292 3.1.4.- 0004114,0007165,0008081 Ki=100nM remove_due_to_license_issue Ki=100nM Q8WQX9 29672041 1007 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLETR 5l8n A 2.12 BS01 6RQ A 1 E12 Y15 A32 I37 E10 Y13 A30 I35 ? 0005504,0005634,0005737,0005829,0006629,0006869,0008285,0008289,0015908,0016020 Kd=31uM remove_due_to_license_issue Kd=2800nM P51161 27500412 1001 FTGKFEMESEKNYDEFMKLLGISSDVIEKARNFKIVTEVQQDGQDFTWSQHYSGGHTMTNKFTVGKESNIQTMGGKTFKATVQMEGGKLVVNFPNYHQTSEIVGDKLVEVSTIGGVTYERVSKRL 5l8t A 1.85 BS01 6RR A 1 P1888 F1889 N1894 V1898 N1944 I1950 P33 F34 N39 V43 N89 I95 ? remove_due_to_license_issue Q9UIF8 27731638 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5l8y B 2.14 BS02 CVA B 1 M785 D822 V840 T841 F844 Y845 M861 M868 E869 L870 G873 Q874 M200 D237 V255 T256 F259 Y260 M276 M283 E284 L285 G288 Q289 3.1.4.- 0004114,0007165,0008081 Ki=400nM remove_due_to_license_issue Ki=398nM Q8WQX9 29672041 1004 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLET 5l96 A 2.15 BS01 6RZ A 1 P1888 V1893 N1894 N1944 I1950 P33 V38 N39 N89 I95 ? remove_due_to_license_issue Q9UIF8 27731638 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5l97 A 2.05 BS01 6RW A 1 W1887 P1888 P1892 V1893 N1944 W32 P33 P37 V38 N89 ? remove_due_to_license_issue Q9UIF8 27731638 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5l98 A 2.263 BS01 6RY A 1 P1888 V1893 N1944 I1950 P33 V38 N89 I95 ? remove_due_to_license_issue Q9UIF8 27731638 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5l99 A 2.0 BS01 6S0 A 1 P1888 F1889 V1893 N1944 P33 F34 V38 N89 ? remove_due_to_license_issue Q9UIF8 27731638 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5l9g A 1.75 BS01 MO0 A 1 W41 Q67 Q87 I88 G89 D92 Y130 W235 R238 D261 T297 W12 Q38 Q58 I59 G60 D63 Y101 W206 R209 D232 T268 Kd=19.8nM remove_due_to_license_issue 27609514 401 MDVVIASSGGGWQEAQDKALWAPAAKALNITYTQDTFQNWAEARAQVESGSVTWDIIQIGIADEPQAKAAGVLEKLDPDIVNKADFPPGSVTDSFVANSNYSTLIAWNKKTYGDNGPKSMADFFDVKKFPGKRALWNQPIGMIEAAALALGTPRDKVYEFLSTEEGRKAAIAKLTELAPSVSVWWESGAQAAQLIKDGEVDMIITWGGRVQGAINDGANFAYTFNDAQLGTDGYAIVKGAPHRDAAMRFLKEMSKAEYQKDLPNSFATAPANMKAYDLAKYTPEKMATMASAPENVAVQYSVDPNFWAKHAKWASEAYDNVRLSR 5l9h A 2.25 BS02 CVL A 1 N825 A837 M861 Q874 F877 F880 N240 A252 M276 Q289 F292 F295 3.1.4.- 0004114,0007165,0008081 ic50=0.4uM remove_due_to_license_issue IC50=400nM Q8WQX9 29672041 1005 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLETR 5l9i A 1.9 BS01 SNW A 1 S37 W41 Q67 Q87 Y130 W235 R238 D261 T297 S9 W13 Q39 Q59 Y102 W207 R210 D233 T269 Kd=99nM remove_due_to_license_issue 27609514 401 HMDVVIASSGGGWQEAQDKALWAPAAKALNITYTQDTFQNWAEARAQVESGSVTWDIIQIGIADEPQAKAAGVLEKLDPDIVNKADFPPGSVTDSFVANSNYSTLIAWNKKTYGDNGPKSMADFFDVKKFPGKRALWNQPIGMIEAAALALGTPRDKVYEFLSTEEGRKAAIAKLTELAPSVSVWWESGAQAAQLIKDGEVDMIITWGGRVQGAINDGANFAYTFNDAQLGTDGYAIVKGAPHRDAAMRFLKEMSKAEYQKDLPNSFATAPANMKAYDLAKYTPEKMATMASAPENVAVQYSVDPNFWAKHAKWASEAYDNVRLSR 5l9l A 1.8 BS01 GOP A 1 S37 W41 Q67 Q87 Y130 W235 R238 D261 T297 S8 W12 Q38 Q58 Y101 W206 R209 D232 T268 Kd=79.4nM remove_due_to_license_issue 27609514 401 MDVVIASSGGGWQEAQDKALWAPAAKALNITYTQDTFQNWAEARAQVESGSVTWDIIQIGIADEPQAKAAGVLEKLDPDIVNKADFPPGSVTDSFVANSNYSTLIAWNKKTYGDNGPKSMADFFDVKKFPGKRALWNQPIGMIEAAALALGTPRDKVYEFLSTEEGRKAAIAKLTELAPSVSVWWESGAQAAQLIKDGEVDMIITWGGRVQGAINDGANFAYTFNDAQLGTDGYAIVKGAPHRDAAMRFLKEMSKAEYQKDLPNSFATAPANMKAYDLAKYTPEKMATMASAPENVAVQYSVDPNFWAKHAKWASEAYDNVRL 5l9o A 1.84 BS01 GOP A 1 F96 A113 A114 G116 R121 A133 G134 T162 L163 Q164 D201 S223 A226 F61 A78 A79 G81 R86 A98 G99 T127 L128 Q129 D166 S188 A191 ? 0015276,0016020,0034220 Kd=4uM remove_due_to_license_issue Q7D447 27609514 301 DNPLGLIDPTTISVGTMGDAKPYAFTTADGNFTGFDIELFLNVAGRLGFKKEQVVFTGQEFSALMPSVANGRFDVAAAAIGTTAKRKETVDFSDGYLAGFLSVLTSEAGITDAAGLKGKRLGVVQGTLQEIYAEKNFAGTDLVKFPDNNSAVSALNNGTVDAHFLDFEAAKDYSARYPALKIAVNIPSFDAPAGFVIRKGNDALRNALDKGLKEAMQDGTWKKLHEKWFPGTPMPAAYLPK 5laq A 2.4 BS02 6M5 A 1 M519 I582 M583 Q615 F618 Y621 I622 M197 I260 M261 Q293 F296 Y299 I300 3.1.4.53 0004114,0007165,0008081 Ki=0.63nM remove_due_to_license_issue IC50=0.630957nM, Ki=0.630957nM Q07343 29672041 1005 TSISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPQS 5lav A 1.73 BS01 6SK A 1 L54 I61 M62 F86 H96 I99 Y100 L36 I43 M44 F68 H78 I81 Y82 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 27775892 201 IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5law A 1.64 BS01 6SJ A 1 L54 L57 I61 M62 Y67 F86 V93 K94 H96 I99 L37 L40 I44 M45 Y50 F69 V76 K77 H79 I82 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 27775892 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5lay A 2.71 BS01 6SS A 1 L54 I61 M62 Y67 F86 H96 I99 L38 I45 M46 Y51 F70 H80 I83 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 27775892 205 SQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5laz A 1.66 BS01 6ST A 1 L54 L57 I61 M62 Y67 F86 V93 K94 H96 I99 Y100 L37 L40 I44 M45 Y50 F69 V76 K77 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 27775892 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5lbq A 3.3 BS02 767 A 1 L386 L536 W552 D555 D556 L216 L366 W382 D385 D386 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 27626075 902 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lbq A 3.3 BS03 767 A 2 E559 G562 E389 G392 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue O60341 27626075 904 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lc0 A 2.7 BS01 6T8 A 1 S81 G82 D83 H1051 D1129 Y1130 A1132 G1133 S1135 G1151 N1152 G1153 V1154 V1155 Y1161 S34 G35 D36 H77 D155 Y156 A158 G159 S161 G177 N178 G179 V180 V181 Y187 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue A0A140DLX4 27386922 1201 MVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVKGETTDGVYRVMTRGLLGSTQVGVGVMQEGVFHTMWHVTKGSALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGHSEVQLLAVPPGERARNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQ 5lc0 A 2.7 BS02 6T8 B 1 H1051 K1054 H77 K80 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue A0A140DLX4 27386922 1201 MVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVKGETTDGVYRVMTRGLLGSTQVGVGVMQEGVFHTMWHVTKGSALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGHSEVQLLAVPPGERARNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQ 5lc0 B 2.7 BS01 6T8 A 1 H1051 K1054 H74 K77 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue A0A140DLX4 27386922 1201 MVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLETTDGVYRVMTRGLLGSTQVGVGVMQEGVFHTMWHVTKGSALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGHSEVQLLAVPPGERARNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQ 5lc0 B 2.7 BS02 6T8 B 1 S81 G82 D83 V1036 H1051 Y1130 A1132 G1133 S1135 G1151 N1152 V1154 Y1161 S34 G35 D36 V59 H74 Y153 A155 G156 S158 G174 N175 V177 Y184 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue A0A140DLX4 27386922 1201 MVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLETTDGVYRVMTRGLLGSTQVGVGVMQEGVFHTMWHVTKGSALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGHSEVQLLAVPPGERARNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQ 5lca A 1.93 BS03 B06 A 1 F62 H116 G209 N210 H240 F24 H78 G171 N172 H202 H114 H116 D118 H179 C198 Y201 N210 H240 H76 H78 D80 H141 C160 Y163 N172 H202 3.5.2.6 ic50=32.8uM remove_due_to_license_issue Q9K2N0 28451231 503 IPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHT 5lcf A 1.86 BS03 6TJ A 1 F62 Y67 W87 H116 H179 G209 N210 H240 F24 Y29 W49 H78 H141 G171 N172 H202 H114 H116 D118 H179 C198 Y201 N210 H240 H76 H78 D80 H141 C160 Y163 N172 H202 3.5.2.6 ic50=17.8uM remove_due_to_license_issue Q9K2N0 28451231 504 IPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHT 5lch A 1.94 BS03 6TU A 1 F62 Y67 W87 H116 D118 H179 G209 N210 H240 F30 Y35 W55 H84 D86 H147 G177 N178 H208 H114 H116 D118 H179 C198 Y201 N210 H240 H82 H84 D86 H147 C166 Y169 N178 H208 3.5.2.6 ic50=20.3uM remove_due_to_license_issue Q9K2N0 28451231 503 YPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5lcj A 1.78 BS01 6TS A 1 I31 V39 A52 M108 E109 K114 L156 C166 I21 V29 A42 M98 E99 K104 L146 C156 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue P28482 27385078 401 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDELDDLPKEKLKELIFEETARFQPG 5lck A 1.89 BS01 6TT A 1 I31 V39 A52 Q105 D106 M108 E109 D111 L156 C166 I21 V29 A42 Q95 D96 M98 E99 D101 L146 C156 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue P28482 27385078 405 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 5ld8 A 2.13 BS01 6U5 A 1 E120 E199 G200 P201 E203 P206 F239 I347 E117 E196 G197 P198 E200 P203 F236 I344 C171 H311 E322 K340 H345 F402 F404 C168 H308 E319 K337 H342 F399 F401 2.3.1.293 0004315,0005515,0005737,0005829,0005886,0006633,0009274,0016746,0016747,0019367,0030497,0042802 Kd=9nM remove_due_to_license_issue P9WQD9 27581223 502 PSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSACSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 5ld8 B 2.13 BS01 6U5 B 1 E120 E199 G200 P201 P206 F239 E117 E196 G197 P198 P203 F236 C171 H311 E322 K340 H345 F402 F404 C168 H308 E319 K337 H342 F399 F401 2.3.1.293 0004315,0005515,0005737,0005829,0005886,0006633,0009274,0016746,0016747,0019367,0030497,0042802 Kd=9nM remove_due_to_license_issue P9WQD9 27581223 502 PSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSACSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 5ldk B 2.099 BS01 ATP B 1 F8 H43 F48 S157 F7 H42 F47 S153 3.1.4.58 0004113,0005524,0008081,0008664,0016787,0016874 Ka=15000M^-1 remove_due_to_license_issue A0A140NFI1 28141848 201 SEPQRLFFAIDLPAEIREQIIHWRAKHFPPEAGRPVAADNLHLTLAFLGEVSAEKEKALSLLAGRIRQPGFTLTLDDAGQWLRSRVVWLGMRQPPRGLIQLANMLRSQAARSGCFRPFHPHITLLRDASEAVTIPPPGFNWSYAVTEFTLYASSFARGRTRYTPLKRWALTQ 5ldm A 2.46 BS01 2AM A 1 F8 H43 T45 F48 H125 T127 R130 F6 H41 T43 F46 H123 T125 R128 3.1.4.58 0004113,0005524,0008081,0008664,0016787,0016874 Ka=7210M^-1 remove_due_to_license_issue A0A140NFI1 28141848 201 EPQRLFFAIDLPAEIREQIIHWRAKHFPPEAGRPVAADNLHLTLAFLGEVSAEKEKALSLLAGRIRQPGFTLTLDDAGQWLRSRVVWLGMRQPPRGLIQLANMLRSQAARSGCFQSNRPFHPHITLLRDASEAVTIPPPGFNWSYAVTEFTLYASSFARGRTRYTPLKRWALTQ 5ldo A 2.752 BS01 3AM A 1 F8 H43 T45 F48 F116 H125 T127 R130 F6 H41 T43 F46 F114 H123 T125 R128 3.1.4.58 0004113,0005524,0008081,0008664,0016787,0016874 remove_due_to_license_issue A0A140NFI1 28141848 201 EPQRLFFAIDLPAEIREQIIHWRAKHFPPEAGRPVAADNLHLTLAFLGEVSAEKEKALSLLAGRIRQPGFTLTLDDAGQWLRSRVVWLGMRQPPRGLIQLANMLRSQAARSGCFQSNRPFHPHITLLRDASEAVTIPPPGFNWSYAVTEFTLYASSFARGRTRYTPLKRWALTQ 5ldp A 1.8 BS01 ATP A 1 R6 F8 H43 F48 S157 T164 Y166 R5 F7 H42 F47 S156 T163 Y165 3.1.4.58 0004113,0005524,0008081,0008664,0016787,0016874 Ka=15000M^-1 remove_due_to_license_issue A0A140NFI1 28141848 201 SEPQRLFFAIDLPAEIREQIIHWRAKHFPPEAGRPVAADNLHLTLAFLGEVSAEKEKALSLLAGRIRQPGFTLTLDDAGQWLRSRVVWLGMRQPPRGLIQLANMLRSQAARSGCFQSNRPFHPHITLLRDASEAVTIPPPGFNWSYAVTEFTLYASSFARGRTRYTPLKRWALTQ 5le1 A 1.4 BS03 6UW A 1 F62 W87 H116 D117 D118 H179 G209 N210 H240 F31 W56 H85 D86 D87 H148 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 ic50=10.6uM remove_due_to_license_issue Q9K2N0 28451231 503 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTN 5lg3 A 3.567 BS01 Z80 A 1 I20 I23 F126 V147 T149 E155 D158 W160 I162 I10 I13 F116 V137 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802 remove_due_to_license_issue E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lg3 B 3.567 BS01 Z80 B 1 N21 I23 F126 V147 T149 E155 D158 W160 I162 N11 I13 F116 V137 T139 E145 D148 W150 I152 ? 0004888,0005216,0005230,0006811,0016020,0034220,0042802 remove_due_to_license_issue E0SJQ4 27791038 401 PVDVSVSIFINKIYGVNTLEQTYKVDGYIVAQWTGKPRKTPGDKPLIVENTQIERWINNGLWVPALEFINVVGSPDTGNKRLMLFPDGRVIYNARFLGSFSNDMDFRLFPFDRQQFVLELEPFSYNNQQLRFSDIQVYTENIDNEEIDEWWIRGKASTHISDIRYDHLSSVQPNQNEFSRITVRIDAVRNPSYYLWSFILPLGLIIAASWSVFWLESFSERLQTSFTLMLTVVAYAFYTSNILPRLPYTTVIDQMIIAGYGSIFAAILLIIFAHHRQANGVEDDLLIQRCRLAFPLGFLAIGCVLVI 5lgn A 3.2 BS02 6W0 A 1 Q358 W699 Y765 Q188 W529 Y595 T335 D557 K665 T165 D387 K495 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue IC50=13400nM, Ki=43000nM O60341 28186755 902 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQADDVKVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lgo A 1.12 BS02 6VZ A 1 H57 N97 T98 L99 D189 S190 C191 Q192 G193 S195 V213 W215 G216 G219 H40 N79 T80 L81 D171 S172 C173 Q174 G175 S177 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 27476144 303 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5lgt A 3.0 BS02 6W3 A 1 F538 A539 D555 W695 A809 F368 A369 D385 W525 A639 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue Ki=2300nM, IC50=310nM O60341 28186757 902 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lgu A 3.2 BS02 6W1 A 1 A539 D555 W695 Y761 A809 A369 D385 W525 Y591 A639 T335 T165 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue IC50=22nM O60341 28186757 902 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lh4 A 1.37 BS02 6W4 A 1 F41 H57 L99 D189 S190 C191 Q192 G193 S195 V213 S214 W215 G216 F24 H40 L81 D171 S172 C173 Q174 G175 S177 V191 S192 W193 G194 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 27476144 305 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5lh8 A 1.54 BS02 6WH A 1 F41 C42 H57 L99 Y151 D189 S190 C191 Q192 G193 S195 V213 G216 G219 F24 C25 H40 L81 Y131 D171 S172 C173 Q174 G175 S177 V191 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 27476144 304 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5lhg A 3.34 BS02 6X3 A 1 V333 Q358 C360 E379 N535 F538 L677 L693 W695 T810 V163 Q188 C190 E209 N365 F368 L507 L523 W525 T640 T335 T165 1.14.99.66 0000122,0000781,0000785,0002039,0002052,0003682,0003713,0005515,0005634,0005654,0005667,0005694,0006325,0006355,0006357,0006482,0010569,0010718,0010976,0014070,0016491,0019899,0021987,0030374,0031398,0032091,0032451,0032452,0032453,0032454,0032880,0032991,0034644,0036211,0040029,0042162,0042551,0042802,0043392,0043426,0043433,0043518,0045793,0045892,0045944,0046098,0050660,0050681,0055001,0060765,0060992,0061629,0061752,0071320,0071480,0120162,0140297,0140682,0140861,0160217,1902166,1990391,1990841,2000179,2000648 remove_due_to_license_issue IC50=2500nM O60341 28186757 906 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lhg A 3.34 BS03 6X3 A 2 A539 D555 H564 A809 A369 D385 H394 A639 T335 T165 1.14.99.66 0000122,0000781,0000785,0002039,0002052,0003682,0003713,0005515,0005634,0005654,0005667,0005694,0006325,0006355,0006357,0006482,0010569,0010718,0010976,0014070,0016491,0019899,0021987,0030374,0031398,0032091,0032451,0032452,0032453,0032454,0032880,0032991,0034644,0036211,0040029,0042162,0042551,0042802,0043392,0043426,0043433,0043518,0045793,0045892,0045944,0046098,0050660,0050681,0055001,0060765,0060992,0061629,0061752,0071320,0071480,0120162,0140297,0140682,0140861,0160217,1902166,1990391,1990841,2000179,2000648 remove_due_to_license_issue IC50=2500nM O60341 28186757 907 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lhh A 3.05 BS02 6X0 A 1 V333 Q358 F538 A539 D555 H564 W695 Y761 A809 T810 V163 Q188 F368 A369 D385 H394 W525 Y591 A639 T640 T335 T165 1.14.99.66 0000122,0000781,0000785,0002039,0002052,0003682,0003713,0005515,0005634,0005654,0005667,0005694,0006325,0006355,0006357,0006482,0010569,0010718,0010976,0014070,0016491,0019899,0021987,0030374,0031398,0032091,0032451,0032452,0032453,0032454,0032880,0032991,0034644,0036211,0040029,0042162,0042551,0042802,0043392,0043426,0043433,0043518,0045793,0045892,0045944,0046098,0050660,0050681,0055001,0060765,0060992,0061629,0061752,0071320,0071480,0120162,0140297,0140682,0140861,0160217,1902166,1990391,1990841,2000179,2000648 remove_due_to_license_issue IC50=6.7nM O60341 28186757 908 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lhi A 3.4 BS02 6X5 A 1 V333 Q358 F538 A539 D555 H564 W695 Y761 A809 V163 Q188 F368 A369 D385 H394 W525 Y591 A639 T335 T165 1.14.99.66 0000122,0000781,0000785,0002039,0002052,0003682,0003713,0005515,0005634,0005654,0005667,0005694,0006325,0006355,0006357,0006482,0010569,0010718,0010976,0014070,0016491,0019899,0021987,0030374,0031398,0032091,0032451,0032452,0032453,0032454,0032880,0032991,0034644,0036211,0040029,0042162,0042551,0042802,0043392,0043426,0043433,0043518,0045793,0045892,0045944,0046098,0050660,0050681,0055001,0060765,0060992,0061629,0061752,0071320,0071480,0120162,0140297,0140682,0140861,0160217,1902166,1990391,1990841,2000179,2000648 remove_due_to_license_issue IC50=7.8nM O60341 28186757 902 PSGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGAMYTL 5lhu A 2.02 BS01 HIS A 1 Y217 D218 L275 Y217 D218 L275 2.4.2.17 0000105,0000287,0003879,0005515,0005524,0005737,0005886,0016208,0016757,0046872 remove_due_to_license_issue P9WMN1 28781362 301 MLRVAVPNKGALSEPATEILAEAGYRRRTDSKDLTVIDPVNNVEFFFLRPKDIAIYVGSGELDFGITGRDLVCDSGAQVRERLALGFGSSSFRYAAPAGRNWTTADLAGMRIATAYPNLVRKDLATKGIEATVIRLDGAVEISVQLGVADAIADVVGSGRTLSQHDLVAFGEPLCDSEAVLIERAGTDGQDQTEARDQLVARVQGVVFGQQYLMLDYDCPRSALKKATAITPGLESPTIAPLADPDWVAIRALVPRRDVNGIMDELAAIGAKAILASDIRFCRF 5li3 A 2.4 BS02 9RB A 1 T24 D101 H144 F153 D181 H183 F209 D269 Y313 T22 D99 H142 F151 D179 H181 F207 D267 Y311 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.053uM remove_due_to_license_issue Q9HXM1 27756124 404 RRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGYSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGLCPAQPL 5li3 B 2.4 BS01 9RB A 1 L340 F343 L338 F341 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.053uM remove_due_to_license_issue Q9HXM1 27756124 404 RRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGYSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGL 5li3 B 2.4 BS03 9RB B 1 T24 D101 H144 F153 D181 H183 F209 D269 Y313 T22 D99 H142 F151 D179 H181 F207 D267 Y311 3.5.1.- 0004407,0016787,0040029,0046872 ic50=0.053uM remove_due_to_license_issue Q9HXM1 27756124 404 RRTAFFFDELCLWHAAGPHALTLPVGGWVQPPAAAGHAESPETKRRLKSLLDVSGLTARLQLRSAPPASDEDLLRVHPAHYLERFKALSDAGGGSLGQDAPIGPGSYEIARLSAGLAIAALDAVLAGEADNAYSLSRPPGHHCLPDQAMGFCFFANIAVAIEAAKARHGVERVAVLDWDVHHGNGTQAIYYRRDDVLSISLHQDGCFPPGYSGAEDIGEDRGRGFNLNVPLLPGGGHDAYMQAMQRIVLPALERFRPQLIVVASGFDANAVDPLARMQLHSDSFRAMTAMVRDAAERHAGGRLVVVHEGGYSEAYVPFCGLAVIEELSGVRSAVRDPLRDFIELQQPNAAFRDFQRQRLEELAAQFGL 5lif E 1.31 BS06 6XO E 1 N112 A113 F114 H142 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 H142 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=1.34uM remove_due_to_license_issue P00800 27959500 411 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5lj0 A 1.82 BS01 6XX A 1 V1008 V1013 D1014 V1018 Y1063 N1064 G1070 D1071 I1074 R1077 V30 V35 D36 V40 Y85 N86 G92 D93 I96 R99 3.6.1.- ic50=0.00000001M remove_due_to_license_issue IC50=50nM Q6PL18 27530368 1205 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 5lj1 A 1.9 BS01 6XX A 1 W81 P82 V87 L92 L94 N140 D144 W40 P41 V46 L51 L53 N99 D103 ? ic50>0.0000316M remove_due_to_license_issue IC50=25119nM O60885 27530368 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5lj2 A 1.19 BS01 6XW A 1 W81 P82 L92 N140 D144 I146 W40 P41 L51 N99 D103 I105 ? ic50=10uM remove_due_to_license_issue O60885 27530368 204 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ljj A 3.0 BS01 AD5 A 1 I531 A551 E603 G605 N606 I607 D608 L654 Q672 P673 I17 A37 E89 G91 N92 I93 D94 L140 Q158 P159 D647 K649 N652 D664 T686 D133 K135 N138 D150 T167 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 27699881 901 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEYGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTDSQVGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 5ljq A 1.05 BS02 ANV A 1 H94 H119 F131 L198 T199 T200 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1nM remove_due_to_license_issue P00918 27933963 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ljt A 1.0 BS02 A6N A 1 H94 H119 F131 L198 T199 T200 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.2nM remove_due_to_license_issue P00918 27933963 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5lkr A 2.52 BS02 6YC A 1 N68 D70 G117 T120 S198 W231 N66 D68 G115 T118 S196 W229 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue IC50=3306nM P06276 27908752 616 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5ll4 A 1.12 BS02 6YH A 1 H94 H96 H119 F131 L198 T199 T200 P202 H94 H96 H119 F130 L197 T198 T199 P201 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=4nM P00918 306 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ll5 A 1.42 BS02 6YH A 1 H91 H93 H117 S133 L197 T198 T199 W208 H89 H91 H115 S131 L195 T196 T197 W206 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 remove_due_to_license_issue Kd=320nM, kon=280000M-1-s-1, koff=0.051s-1 O43570 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 5ll7 A 1.4 BS01 6YV A 1 C69 S70 W105 S130 E166 N170 T235 T237 C43 S44 W79 S104 E140 N144 T209 T211 S70 K73 S130 E166 K234 T237 S44 K47 S104 E140 K208 T211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue A0A0H4IUK8 29356380 301 TNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 5ll9 A 1.45 BS02 6YQ A 1 H91 H117 V119 S133 L197 T198 T199 P201 W208 H89 H115 V117 S131 L195 T196 T197 P199 W206 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 remove_due_to_license_issue Kd=833nM, kon=380000M-1-s-1, koff=0.17s-1 O43570 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 5lla B 1.5 BS02 6YQ B 1 H96 H98 H121 V123 F133 L200 T201 V202 H91 H93 H116 V118 F128 L195 T196 V197 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 remove_due_to_license_issue kon=630000M-1-s-1, koff=0.0020s-1, Kd=19nM Q8N1Q1 302 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 5llc A 1.1 BS02 V26 A 1 N62 H64 Q92 H94 H119 L198 T199 T200 N60 H62 Q90 H92 H117 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=8.2nM, kon=1300000M-1-s-1, koff=0.0082s-1 P00918 29503769 308 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5lle A 1.9 BS02 V51 A 1 Q92 H94 H96 H119 V121 F131 L198 T199 T200 P202 Q89 H91 H93 H116 V118 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=5.0nM P00918 29503769 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5llg A 1.12 BS02 VD9 A 1 H94 H96 H119 L198 T199 T200 H91 H93 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=13nM P00918 29503769 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5llg A 1.12 BS03 VD9 A 2 H4 W5 N11 H15 W16 D19 H1 W2 N8 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=13nM P00918 29503769 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5llh A 1.9 BS02 V49 A 1 Q92 H94 H96 V121 F131 L198 T199 T200 P202 Q89 H91 H93 V118 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=1.1nM P00918 29503769 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5lli C 2.4 BS01 6Z3 C 1 W88 Y98 I109 H110 S111 Y112 H115 W117 W27 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=90nM remove_due_to_license_issue Kd=90nM, IC50=88nM P40337 27811928 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQ 5llm A 3.25 BS02 6Z6 A 1 S116 G117 G120 Y127 M231 F235 F369 V373 I377 S80 G81 G84 Y91 M159 F163 F290 V294 I298 ? 0015293,0016020 remove_due_to_license_issue P43003,Q15758 28424515 603 TKEDVKSFLRRNALLLLTVLAVILGVVLGFLLRPYPLSPREVKYFAFPGELLMRMLKMLILPLIVSSLITGLASLDAKASGRLGMRAVVYYMSTTIIAVVLGIILVLIIHPEVLDCFLDLARNIFPSNLVSAAFRSYSTTPVGQEVEGMNILGLVVFSMVFGFALGKMGEQGQLLVDFFNSLNEATMKLVAIIMWYAPLGILFLIAGKIVEGGQLGMYMVTVIVGLVIHGLIVLPLIYFLITRKNPFVFIAGILQALITALGTSSSSATLPITFKCLEENNGVDKRITRFVLPVGATINMDGTALYEAVAAIFIAQQIITISITATAASIGAAGIPQAGLVTMVIVLTAVGLPTDDITLIIAVDWLLDRFRTMVNVLGDALGAGIVEHLSRKELEKQDA 5llo A 1.6 BS02 5EF A 1 N64 H91 H93 H117 A129 S130 L197 T198 T199 N62 H89 H91 H115 A127 S128 L195 T196 T197 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 remove_due_to_license_issue O43570 29503769 303 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFS 5llp A 1.48 BS02 6Z9 A 1 N64 K69 Q89 H91 H93 H117 A129 L197 T198 T199 N62 K67 Q87 H89 H91 H115 A127 L195 T196 T197 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 remove_due_to_license_issue O43570 29503769 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFS 5lm4 A 3.1 BS02 6Z6 A 1 S116 G117 G120 A123 V124 Y127 I231 I235 F369 V373 I377 S78 G79 G82 A85 V86 Y89 I151 I155 F278 V282 I286 ? 0015293,0016020 remove_due_to_license_issue P43003,Q15758 28424515 603 EDVKSFLRRNALLLLTVLAVILGVVLGFLLRPYPLSPREVKYFAFPGELLMRMLKMLILPLIVSSLITGLASLDAKASGRLGMRAVVYYMSTTIIAVVLGIILVLIIEVLDCFLDLARNIFPSNLVSAAFRSYSTQEVEGMNILGLVVFSIVFGIALGKMGEQGQLLVDFFNSLNEATMKLVAIIMWYAPLGILFLIAGKIVEGMYMVTVIVGLVIHGLIVLPLIYFLITRKNPFVFIAGILQALITALGTSSSSATLPITFKCLEENNGVDKRITRFVLPVGATINMDGTALYEAVAAIFIAQDFGQIITISITATAASIGAAGIPQAGLVTMVIVLTAVGLPTDDITLIIAVDWLLDRFRTMVNVLGDALGAGIVEHLSRKELEKQD 5lm6 A 1.17 BS03 H32 A 1 Y67 W87 H116 D117 D118 G209 N210 H240 Y36 W56 H85 D86 D87 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 ic50=7.7uM remove_due_to_license_issue Q9K2N0 28451231 504 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5lma A 1.43 BS01 6ZG A 1 L377 A400 M450 A451 G454 P455 R498 L501 D512 L15 A38 M88 A89 G92 P93 R136 L139 D150 D494 A496 R498 N499 D512 K533 D132 A134 R136 N137 D150 K169 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.25uM remove_due_to_license_issue IC50=2512nM P43405 27578246 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYD 5lmb A 1.95 BS01 6ZF A 1 L377 A400 M450 A451 G454 P455 R498 N499 L501 D512 L14 A37 M81 A82 G85 P86 R129 N130 L132 D143 D494 A496 R498 N499 D512 K533 D125 A127 R129 N130 D143 K164 2.7.10.2 0004672,0004713,0005524,0006468 ic50=16nM remove_due_to_license_issue IC50=16nM P43405 27578246 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV 5lmk A 2.4 BS01 6ZK A 1 I10 E12 A31 F80 F82 L83 H84 Q85 Q131 L134 I11 E13 A32 F79 F81 L82 H83 Q84 Q130 L133 D127 K129 Q131 N132 D145 T158 T165 D126 K128 Q130 N131 D144 T157 T164 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=37nM P24941 28039837 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5lne A 2.2 BS01 GAL C 1 F1 N44 D45 D51 D53 K132 A134 F1 N44 D45 D51 D53 K127 A129 ? 0007155,0009289 remove_due_to_license_issue A0A0H2V7F6 27667696 2 FSCNVDGGSSIGAGTTSVYVNLDPVIQPGQNLVVDLSQHISCWNDYGGWYDTDHINLVQGSAFAGLQSYKGSLYWNNVTYPFPLTTNTNVLDIGDKTPMPLPLKLYITPVGVVIKAGEVIARIHMYKIATLGSGNPRNFTWNIISNNSVVMP 5lny A 1.88 BS01 70K A 1 N51 A55 D93 G97 M98 F138 T184 N35 A39 D77 G81 M82 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=42nM remove_due_to_license_issue P07900 29701469 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5loh A 3.1 BS01 STU A 1 I41 A60 M110 Y112 L113 G116 D117 D160 L163 T173 D174 S178 I12 A27 M62 Y64 L65 G68 D69 D112 L115 T125 D126 S130 D156 K158 D160 N161 D174 T741 D108 K110 D112 N113 D126 T135 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q96GX5 27563826 901 PSIEEFSIVKPISGKVYLGQKGGKLYAVKVVKKADMLALSKSPFIVHLYYSLQSANNVYLVMEYLIGGDVKSLLHIYGYFDEEMAVKYISEVALALDYLHRHGIIHRDLKPDNMLISNEGHIKLTDFGLSKFCGTPDYLAPELLLGRAHGPAVDWWALGVCLFEFLTGIPPFNDETPQQVFQNILKRDIPWPEGEEKLSDNAQSAVEILLTIDDTKRAGMKELKRHPLFSDVDWENLQHQTMPFIPQP 5lom A 1.5 BS01 SNW A 1 F96 A113 A114 G116 R121 A133 G134 T162 L163 Q164 D201 S223 A226 F61 A78 A79 G81 R86 A98 G99 T127 L128 Q129 D166 S188 A191 ? 0015276,0016020,0034220 remove_due_to_license_issue Q7D447 27609514 301 DNPLGLIDPTTISVGTMGDAKPYAFTTADGNFTGFDIELFLNVAGRLGFKKEQVVFTGQEFSALMPSVANGRFDVAAAAIGTTAKRKETVDFSDGYLAGFLSVLTSEAGITDAAGLKGKRLGVVQGTLQEIYAEKNFAGTDLVKFPDNNSAVSALNNGTVDAHFLDFEAAKDYSARYPALKIAVNIPSFDAPAGFVIRKGNDALRNALDKGLKEAMQDGTWKKLHEKWFPGTPMPAAYLPK 5lp1 A 1.91 BS01 71H A 1 F110 L111 G152 L153 G154 A155 L159 S273 F274 W298 Q352 F357 F56 L57 G98 L99 G100 A101 L105 S219 F220 W244 Q298 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=0.398nM remove_due_to_license_issue Q13093 28105273 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINT 5lp6 A 2.9 BS03 71P B 1 S178 T179 V181 S178 T179 V181 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 27613098 504 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVDS 5lp6 B 2.9 BS02 71P B 1 C241 L248 N249 A250 L255 N258 T314 A316 I318 N350 K352 C239 L246 N247 A248 L253 N256 T306 A308 I310 N342 K344 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Q6B856 27613098 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5lpj A 1.65 BS01 XDM A 1 P1110 V1115 L1120 Y1125 Y1167 N1168 R1173 V1174 F1177 P29 V34 L39 Y44 Y86 N87 R92 V93 F96 2.3.1.-,2.3.1.48 Kd=10.1uM remove_due_to_license_issue Q92793 28766825 1201 KKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5lpk A 2.1 BS01 XDM A 1 P1074 V1079 L1084 N1132 R1137 P29 V34 L39 N87 R92 2.3.1.-,2.3.1.48 Kd=3.06uM remove_due_to_license_issue Q09472 28766825 1201 KKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKSPMDLSTIKRKLDTGQYQEPWQYVDDIWLMFNNAWLYNRKTSRVYKYCSKLSEVFEQEIDPVMQSLG 5lpl A 1.65 BS01 71X A 1 P1110 V1115 L1120 Y1125 Y1167 N1168 R1173 V1174 P32 V37 L42 Y47 Y89 N90 R95 V96 2.3.1.-,2.3.1.48 Kd=12uM remove_due_to_license_issue Q92793 28766825 1201 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5lpm A 1.5 BS01 71Y A 1 P1074 V1079 D1080 L1084 Y1089 Y1131 N1132 P29 V34 D35 L39 Y44 Y86 N87 2.3.1.-,2.3.1.48 Kd=2.77uM remove_due_to_license_issue Q09472 28766825 1201 SMIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKSPMDLSTIKRKLDTGQYQEPWQYVDDIWLMFNNAWLYNRKTSRVYKYCSKLSEVFEQEIDPVMQSLG 5lpm A 1.5 BS02 71Y A 2 L1083 L1084 L38 L39 2.3.1.-,2.3.1.48 Kd=2.77uM remove_due_to_license_issue Q09472 28766825 1202 SMIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKSPMDLSTIKRKLDTGQYQEPWQYVDDIWLMFNNAWLYNRKTSRVYKYCSKLSEVFEQEIDPVMQSLG 5lqf A 2.06 BS01 4SP A 1 I10 A31 V64 F80 E81 F82 L83 S84 M85 D86 K89 L135 D146 I13 A34 V67 F83 E84 F85 L86 S87 M88 D89 K92 L138 D149 D128 K130 Q132 N133 D146 V159 T166 D131 K133 Q135 N136 D149 V162 T164 2.7.11.22,2.7.11.23 0000082,0000086,0000226,0000307,0000781,0001618,0003682,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005789,0005813,0005819,0005829,0005856,0005876,0006260,0006281,0006338,0006357,0006468,0006915,0006974,0007077,0007095,0007098,0007344,0008353,0009410,0009636,0010628,0010629,0010971,0014038,0014070,0014075,0014823,0016020,0016301,0016477,0016579,0018105,0018107,0030261,0030332,0030496,0030544,0030855,0031100,0034501,0035173,0042307,0042542,0042752,0043066,0044772,0045471,0045740,0045931,0045995,0046686,0046688,0046718,0048144,0048511,0048678,0051301,0055015,0060045,0062033,0065003,0070062,0070301,0070371,0071407,0072686,0090166,0097121,0097122,0097125,0097472,0106310,0140833,0140834,0140835,0140836,0140837,1900182,1902423,1902850,1905448 remove_due_to_license_issue IC50=250nM P06493 28005359 301 LGSMEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRHPNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCHSRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIPIRVVTLWYRSPEVLLGSARYSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNTFPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFND 5lqq A 2.4 BS05 72P A 1 K248 F249 H251 W254 W260 F274 K193 F194 H196 W199 W205 F219 3.1.4.39 0001953,0003676,0004528,0004622,0004630,0005044,0005509,0005576,0005615,0006644,0006935,0006955,0008270,0008284,0009395,0010634,0016020,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0044849,0046872,0047391,0048714,0050731,0051894,0060326,0071276,0071392,1900026,1903165,2000394 ic50=81nM remove_due_to_license_issue Q64610 27982588 922 GSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIKVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDASFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLRLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRAKSINNSKYDPKTIIAALTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDIHLLVDRRWHVARKPLDFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPDEVSRPNYPGIMYLQSEFDLGCTCKGSTKERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWAYFQRVLVKKYASERNGVNVISGPIFDYNYDGLRDTEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCASSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5ls6 A 3.47 BS10 74D A 1 Y111 W624 Y661 C663 F665 F686 N688 Y102 W466 Y503 C505 F507 F528 N530 2.1.1.356 0006338,0042054,0046976 remove_due_to_license_issue Q15910 27739677 809 KGPVCWRKRVKSEYMRLRQLKRFRRADEVKSMFSSNRQKILERTEILNQEWKQRRIQPVHILTSVSSLRGTRECSVTSDLDFPTQVIPLKTLNAVASVPIMYSWSPLQQNFMVEDETVLHNIPYMGDEVLDQDGTFIEELIKNYDGKVHGDRECGFINDEIFVELVNALGQYNESRPPRSDKIFEAISSMFPDKGTAEELKEKYKELTQPPECTPNIDGPNAKSVQREQSLHSFHTLFCRRCFKYDCFLHPFHATPNTYKRKNTETALDNKPCGPQCYQHLEGAKEFAAALTAERIKTPNIEPPENVEWSGAEASMFRVLIGTYYDNFCAIARLIGTKTCRQVYEFRVKESSIIAPAHVYNYQPCDHPRQPCDSSCPCVIAQNFCEKFCQCSSECQNRFPGCRCKAQCNTKQCPCYLAVRECDPDLCLTCGAADHWDSKNVSCKNCSIQRGSKKHLLLAPSDVAGWGIFIKDPVQKNEFISEYCGEIISQDEADRRGKVYDKYMCSFLFNLNNDFVVDATRKGNKIRFANHSVNPNCYAKVMMVNGDHRIGIFAKRAIQTGEELFFDYRY 5lsc A 1.497 BS01 752 A 1 Y67 W87 H118 D119 D120 H196 C221 N233 H263 Y38 W58 H87 D88 D89 H150 C169 N181 H211 H116 H118 D120 H196 C221 Y224 N233 H263 H85 H87 D89 H150 C169 Y172 N181 H211 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=20uM remove_due_to_license_issue B8QIQ9 27834790 404 SGEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRSV 5lsg A 2.0 BS01 QZQ A 1 F282 C285 Q286 R288 S289 H323 I326 Y327 L330 V339 I341 M364 K367 H449 Y473 F64 C67 Q68 R70 S71 H105 I108 Y109 L112 V121 I123 M146 K149 H231 Y255 ? 0003677,0004879,0005634,0006355 Kd=4uM remove_due_to_license_issue P37231 28720829 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 5lss A 1.79 BS04 76H A 1 K1560 G1561 W1562 Y1579 H1603 Y1604 Y1605 R1625 F1626 M1627 N1628 H1629 Y1666 Q1676 C1678 F1679 L1689 K107 G108 W109 Y126 H150 Y151 Y152 R172 F173 M174 N175 H176 Y213 Q223 C225 F226 L236 Y1579 Y1666 Y126 Y213 2.1.1.-,2.1.1.359 0005634,0016279,0042054,0046975 remove_due_to_license_issue Q9BYW2 27571355 1805 LVGPSCVMDDFRDPQRWKECAKQGKMPCYFDLIEENVYLTERKMQCECTPLSKDERAQGEIACGEDCLNRLLMIECSSRCPNGDYCSNRRFQRKQHADVEVILTEKKGWGLRAAKDLPSNTFVLEYCGEVLDHKEFKARVKEYARNKNIHYYFMALKNDEIIDATQKGNCSRFMNHSCEPNCETQKWTVNGQLRVGFFTTKLVPSGSELTFDYQFQRYGKEAQKCFCGSANCRGYLG 5lsx A 2.9 BS04 76O A 1 K1560 G1561 W1562 Y1579 H1603 Y1604 Y1605 R1625 M1627 N1628 H1629 F1664 Y1666 Q1676 C1678 F1679 K103 G104 W105 Y122 H146 Y147 Y148 R168 M170 N171 H172 F207 Y209 Q216 C218 F219 Y1579 Y1666 Y122 Y209 2.1.1.-,2.1.1.359 0005634,0016279,0042054,0046975 remove_due_to_license_issue Q9BYW2 27571355 1804 GPSCVMDDFRDPQRWKECAKQGKMPCYFDLIEENVYLTEMQCECTPLSKDERAQGEIACGEDCLNRLLMIECSSRCPNGDYCSNRRFQRKQHADVEVILTEKKGWGLRAAKDLPSNTFVLEYCGEVLDHKEFKARVKEYARNKNIHYYFMALKNDEIIDATQKGNCSRFMNHSCEPNCETQKWTVNGQLRVGFFTTKLVPSGSELTFDYQFQREAQKCFCGSANCRGYLGG 5lsy A 1.62 BS04 76M A 1 K1560 G1561 W1562 Y1579 H1603 Y1604 Y1605 R1625 F1626 M1627 N1628 H1629 F1664 Y1666 Q1669 C1678 F1679 K107 G108 W109 Y126 H150 Y151 Y152 R172 F173 M174 N175 H176 F211 Y213 Q216 C225 F226 Y1579 Y1666 Y126 Y213 2.1.1.-,2.1.1.359 0005634,0016279,0042054,0046975 remove_due_to_license_issue Q9BYW2 27571355 1805 GETSVPPGSALVGPSCVMDDFRDPQRWKECAKQGKMPCYFDLIEENVYLTRMQCECTPLEIACGEDCLNRLLMIECSSRCPNGDYCSNRRFQRKQHADVEVILTEKKGWGLRAAKDLPSNTFVLEYCGEVLDHKEFKARVKEYARNKNIHYYFMALKNDEIIDATQKGNCSRFMNHSCEPNCETQKWTVNGQLRVGFFTTKLVPSGSELTFDYQFQRYGKEAQKCFCGSANCRGYLGGENRVSIRA 5lt6 A 2.05 BS04 76J A 1 K1560 G1561 W1562 Y1579 Y1605 R1625 N1628 H1629 F1664 Y1666 Q1676 C1678 F1679 L1689 K104 G105 W106 Y123 Y149 R169 N172 H173 F208 Y210 Q220 C222 F223 L233 Y1579 Y1666 Y123 Y210 2.1.1.-,2.1.1.359 0005634,0016279,0042054,0046975 remove_due_to_license_issue Q9BYW2 27571355 1805 GPSCVMDDFRDPQRWKECAKQGKMPCYFDLIEENVYLTERMQCECTPLSKDERAQGEIACGEDCLNRLLMIECSSRCPNGDYCSNRRFQRKQHADVEVILTEKKGWGLRAAKDLPSNTFVLEYCGEVLDHKEFKARVKEYARNKNIHYYFMALKNDEIIDATQKGNCSRFMNHSCEPNCETQKWTVNGQLRVGFFTTKLVPSGSELTFDYQFQRYGKEAQKCFCGSANCRGYLG 5lt9 A 3.0 BS01 ARG A 1 F99 Y101 Y109 A111 S115 L117 Y121 R126 W128 Y144 E146 P147 D173 F61 Y63 Y71 A73 S77 L79 Y83 R88 W90 Y106 E108 P109 D135 ? remove_due_to_license_issue Q9HW91 301 REDLEDYLHEMGEITASNVQNWLSGRILLIENLAQTLARDHSPETTQALLEQPLLGSTFLFTYLGQTDGTYTARPTSDLPADYDPRRRPWYNAATSAGQTTLTEPYMEPAIHELVLTIASPARQGGQPFGVVGGDLSLQTVVKIINSLDFGGMGYAFLVSGDGKILVHPDKDQVMKSLSDVYPRNTPKIGSGFSEAELHGNTRILSFSPVKGLSGLDWYIGISVDKDKAYAMLT 5ltn A 1.88 BS02 XI7 A 1 E50 D88 E51 D89 2.7.7.48,3.1.-.- remove_due_to_license_issue P14240 29765612 205 HDEIISELRELCLNYIEQDERLSRQKLNFLGQREPRMVLIEGLKLLSRCIEIDSADKSGCTHNHDDKSVETILVESGIVCPGLPLIIPDGYKLIDNSLILLECFVRSTPASFEKKFIEDTNKLACIREDLAVAGVTLVPIVDGRCDYDNSFMPEWANFKFRDLLFKLLEYSNQDEKVFEESEY 5lto A 3.459 BS01 GLN A 1 F99 Y101 Y109 S115 L117 Y121 R126 W128 Y144 E146 D173 F64 Y66 Y74 S80 L82 Y86 R91 W93 Y109 E111 D138 ? remove_due_to_license_issue Q9HW91 300 ASIREDLEDYLHEMGEITASNVQNWLSGRILLIENLAQTLARDHSPETTQALLEQPLLGSTFLFTYLGQTDGTYTARPTSDLPADYDPRRRPWYNAATSAGQTTLTEPYMEPAIHELVLTIASPARQGGQPFGVVGGDLSLQTVVKIINSLDFGGMGYAFLVSGDGKILVHPDKDQVMKSLSDVYPRNTPKIGSGFSEAELHGNTRILSFSPVKGLSGLDWYIGISVDKDKAYAMLT 5lub B 2.1 BS01 3Y7 B 1 R44 C189 S216 A218 R19 C164 S191 A193 3.4.22.34 0006508,0008233 ic50=0.7uM remove_due_to_license_issue Q99538 28345579 304 GGKHWVVIVAGSNGWYNYRHQADACHAYQIIHRNGIPDEQIVVMMYDDIAYSEDNPTPGIVINRPNGTDVYQGVPKDYTGEDVTPQNFLAVLRGDAEAVKGIGSGKVLKSGPQDHVFIYFTDHGSTGILVFPNEDLHVKDLNETIHYMYKHKMYRKMVFYIEACESGSMMNHLPDNINVYATTAANPRESSYACYYDEKRSTYLGDWYSVNWMEDSDVEDLTKETLHKQYHLVKSHTQTSHVMQYGNKTISTMKVMQFQGMK 5lud A 1.25 BS01 76X A 1 G72 N102 Q111 G72 N102 Q111 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 28396838 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 5luu A 1.61 BS01 77X A 1 W81 P82 L92 L94 N140 I146 W40 P41 L51 L53 N99 I105 ? Kd=8.63uM remove_due_to_license_issue Kd=31300nM O60885 27994766 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5lvd E 1.25 BS06 79F E 1 N112 A113 E143 H146 E166 R203 H231 N112 A113 E143 H146 E166 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=2.4mM remove_due_to_license_issue P00800 28696673 410 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5lvl A 1.4 BS01 537 A 1 L88 A109 S160 A162 G165 L212 L15 A36 S87 A89 G92 L139 D205 K207 E209 N210 D223 T245 D132 K134 E136 N137 D150 T172 2.7.11.1 0004672,0004674,0005524,0006468 Kd=1.25uM remove_due_to_license_issue O15530 27693059 401 PRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 5lvn A 1.379 BS01 ADN A 1 G89 V96 A109 A162 E166 L212 G14 V21 A34 A87 E91 L137 D205 K207 E209 N210 D223 T245 D130 K132 E134 N135 D148 T170 2.7.11.1 0004672,0004674,0005524,0006468 Kd=20uM remove_due_to_license_issue O15530 27693059 402 KKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 5lvq A 2.05 BS01 2LX A 1 F748 A757 Y809 F25 A34 Y86 2.3.1.48,2.3.1.57 0004402 Kd=73uM remove_due_to_license_issue Kd=73000nM Q92831 27994766 904 DPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 5lvr A 2.05 BS01 78Y A 1 P747 E756 Y802 N803 Y809 P24 E33 Y79 N80 Y86 2.3.1.48,2.3.1.57 0004402 Kd=250uM remove_due_to_license_issue Kd=250000nM Q92831 27994766 904 DPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 5lvx A 2.2 BS01 79B A 1 E235 S237 Q284 Y313 F316 S345 K346 W348 E235 S237 Q284 Y313 F316 S345 K346 W348 E235 E340 C342 N370 E235 E340 C342 N370 2.4.1.-,3.2.1.-,3.2.1.45,3.2.1.46 0000423,0004336,0004348,0005102,0005124,0005515,0005615,0005764,0005765,0005783,0005794,0005802,0006665,0006678,0006680,0006914,0007005,0007040,0007417,0008203,0008340,0008422,0009267,0009268,0014004,0016020,0016241,0016757,0016787,0016798,0019882,0019915,0021694,0021859,0022904,0023021,0030259,0031175,0031333,0032006,0032436,0032715,0033077,0033574,0042391,0043161,0043202,0043243,0043409,0043524,0043627,0046512,0046513,0046527,0048469,0048854,0048872,0050295,0050728,0050877,0050905,0051246,0051248,0051402,0061436,0061518,0061744,0070062,0071356,0071425,0071548,0072676,0097066,0098773,1901805,1903052,1903061,1904457,1905037,1905091,1905165 remove_due_to_license_issue P04062 29676907 507 ARPCIPKSFGYSSVVCVCNATYCDSFDPPTFPALGTFSRYESTRSGRRMELSMGPIQANHTGTGLLLTLQPEQKFQKVKGFGGAMTDAAALNILALSPPAQNLLLKSYFSEEGIGYNIIRVPMASCDFSIRTYTYADTPDDFQLHNFSLPEEDTKLKIPLIHRALQLAQRPVSLLASPWTSPTWLKTNGAVNGKGSLKGQPGDIYHQTWARYFVKFLDAYAEHKLQFWAVTAENEPSAGLLSGYPFQCLGFTPEHQRDFIARDLGPTLANSTHHNVRLLMLDDQRLLLPHWAKVVLTDPEAAKYVHGIAVHWYLDFLAPAKATLGETHRLFPNTMLFASEACVGSKFWEQSVRLGSWDRGMQYSHSIITNLLYHVVGWTDWNLALNPEGGPNWVRNFVDSPIIVDITKDTFYKQPMFYHLGHFSKFIPEGSQRVGLVASQKNDLDAVALMHPDGSAVVVVLNRSSKDVPLTIKDPAVGFLETISPGYSIHTYLWRRQ 5lwd E 1.23 BS06 79E E 1 N112 A113 F130 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F130 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.57uM remove_due_to_license_issue P00800 27959500 411 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5lwe A 2.8 BS01 79K A 1 V69 Y73 R78 T81 T83 D84 L87 I140 R144 A255 T256 V259 Y317 G321 E322 R323 F324 V26 Y30 R35 T38 T40 D41 L44 I89 R93 A185 T186 V189 Y247 G251 E252 R253 F254 ? 0004930,0004950,0006935,0006955,0007186,0016020,0016493 remove_due_to_license_issue IC50=2.8nM, Ki=3.7nM P51686 27926729 401 RQFASHFLPPLYWLVFIVGALGNSLVILVYWYCARAKTATDMFLLNLAIADLLFLVTLPFWAIATFMCKVVNSMYKMNFYSCVLLIMCICVDRYIAIAQAMRAHTWREKRLLYSKMVCFTIWVLAAALCIPEILYCTTKLKSAVLALKVILGFFLPFVVMACCYTIIIHTLIQAKKSSKHKALKATITVLTVFVLSQFPYNCILLVQTIDAYAMFISNCAVSTAIDICFQVTQAIAFFHSCLNPVLYVFVGERFRRDLVKTLKNLGAISQAAAHH 5lwm A 1.55 BS01 79T A 1 L828 V836 A853 Y904 L905 C909 R911 D912 R953 L956 L15 V23 A40 Y91 L92 C96 R98 D99 R140 L143 A949 A951 R953 N954 D967 A136 A138 R140 N141 D154 2.7.10.2 0004672,0005524,0006468 Kd=0.00134uM remove_due_to_license_issue EC50=237nM, IC50=0.130000nM P52333 27840070 1201 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 5lwn A 1.6 BS02 79R A 1 L828 A853 E903 Y904 L905 C909 R911 R953 L956 L15 A40 E90 Y91 L92 C96 R98 R140 L143 A949 A951 R953 N954 D967 A136 A138 R140 N141 D154 2.7.10.2 0004672,0005524,0006468 ic50=17nM remove_due_to_license_issue P52333 27840070 1208 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 5lws A 1.03 BS01 7B2 A 1 D15 A16 G80 D81 F116 D119 G221 T222 T223 I300 D15 A16 G80 D81 F116 D119 G221 T222 T223 I300 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 remove_due_to_license_issue P11838 28097765 409 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 5lx6 A 1.25 BS01 78P A 1 H887 G888 C907 Y919 S927 Y932 H71 G72 C91 Y103 S111 Y116 2.4.2.- 0003950 ic50=1900nM remove_due_to_license_issue IC50=43800nM Q53GL7 28001384 1101 SMNLERLAENTGEFQEVVRAFYDTLDAARSSIRVVRVERVSHPLLQQQYELYRERLLQRCERRPVEQVLYHGTTAPAVPDICAHGFNRSFCGRNATVYGKGVYFARRASLSVQDRYSPPNADGHKAVFVARVLTGDYGQGRRGLRAPPLRGPGHVLLRYDSAVDCICQPSIFVIFHDTQALPTHLITCEHV 5lxb B 2.34 BS01 7A9 B 1 Y91 W145 C188 C189 Y193 Y91 W145 C188 C189 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 27656911 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 5lxb C 2.34 BS01 7A9 B 1 R55 M114 I116 R55 M114 I116 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 27656911 301 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 5lxb C 2.34 BS02 7A9 C 1 Y91 W145 Y186 C188 C189 Y91 W145 Y186 C188 C189 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 27656911 302 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYWERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 5lxc A 2.15 BS01 7AA A 1 G156 K157 F160 V163 A176 K178 F228 L231 E279 L282 I294 G77 K78 F81 V84 A97 K99 F149 L152 E200 L203 I215 D275 K277 N280 D295 S312 D196 K198 N201 D216 S233 2.7.12.1 0004672,0004712,0005524,0006468 ic50=10.8nM remove_due_to_license_issue Q92630 27766861 501 PMTPEQAMKQYMQKLTAFEHHEIFSYPEIYFLGLNAKKRQGMTGGPNNGGYDDDQGSYVQVPHDHVAYRYEVLKVIGKGSFGQVVKAYDHKVHQHVALKMVRNEKRFHRQAAEEIRILEHLRKQDKDNTMNVIHMLENFTFRNHICMTFELLSMNLYELIKKNKFQGFSLPLVRKFAHSILQCLDALHKNRIIHCDLKPENILLKQQGRSGIKVIDFGSSCYEHQRVYTYIQSRFYRAPEVILGARYGMPIDMWSLGCILAELLTGYPLLPGEDEGDQLACMIELLGMPSQKLLDASKRAKNFVSSKGYPRYCTVTTLSDGSVVLNGGRSRRGKLRGPPESREWGNALKGCDDPLFLDFLKQCLEWDPAVRMTPGQALRHPWLR 5lxd A 2.58 BS01 7A7 A 1 G156 V163 F228 L231 L282 I294 D295 G77 V84 F149 L152 L203 I215 D216 D275 K277 N280 D295 S312 D196 K198 N201 D216 S233 2.7.12.1 0004672,0004712,0005524,0006468 remove_due_to_license_issue Q92630 27766861 501 PMTPEQAMKQYMQKLTAFEHHEIFSYPEIYFLGLNAKKRQGMTGGPNNGGYDDDQGSYVQVPHDHVAYRYEVLKVIGKGSFGQVVKAYDHKVHQHVALKMVRNEKRFHRQAAEEIRILEHLRKQDKDNTMNVIHMLENFTFRNHICMTFELLSMNLYELIKKNKFQGFSLPLVRKFAHSILQCLDALHKNRIIHCDLKPENILLKQQGRSGIKVIDFGSSCYEHQRVYTYIQSRFYRAPEVILGARYGMPIDMWSLGCILAELLTGYPLLPGEDEGDQLACMIELLGMPSQKLLDASKRAKNFVSSKGYPRYCTVTTLSDGSVVLNGGRSRRGKLRGPPESREWGNALKGCDDPLFLDFLKQCLEWDPAVRMTPGQALRHPWLRRR 5lxp A 2.07 BS01 7AG A 1 H1682 G1683 Y1714 A1716 Y1721 S1722 T1726 Y1727 H72 G73 Y95 A97 Y102 S103 T107 Y108 2.4.2.- 0003950 ic50=0.76uM remove_due_to_license_issue Q460N5 27918638 1901 DMKQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 5lyh A 2.17 BS01 7B8 A 1 H1682 G1683 T1684 S1688 F1697 N1698 S1700 V1707 T1713 Y1714 F1715 A1716 Y1721 S1722 Y1727 H71 G72 T73 S77 F86 N87 S89 V91 T97 Y98 F99 A100 Y105 S106 Y111 2.4.2.- 0003950 ic50=0.49uM remove_due_to_license_issue Q460N5 27918638 1901 MKQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 5lyr A 1.14 BS01 MAN A 1 H63 R295 E333 E336 H33 R265 E303 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 27992199 403 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 5lyr A 1.14 BS02 MNM A 1 Y46 W126 H154 E156 Y195 Y252 E333 E336 Y16 W96 H124 E126 Y165 Y222 E303 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 27992199 404 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 5lyw A 1.69 BS01 7BH A 1 F219 H231 D251 D262 H331 I338 H339 M384 Y444 F104 H116 D136 D147 H216 I223 H224 M267 Y327 D251 D262 H331 H339 E364 E459 D136 D147 H216 H224 E247 E342 3.4.11.18 0006508,0070006 ic50=0.7uM remove_due_to_license_issue P50579 27998678 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGD 5lyx A 1.9 BS01 7BF A 1 F219 H231 D251 D262 H331 I338 H339 A414 Y444 F108 H120 D140 D151 H220 I227 H228 A303 Y333 D251 D262 H331 H339 E364 E459 D140 D151 H220 H228 E253 E348 3.4.11.18 0006508,0070006 ic50=0.038uM remove_due_to_license_issue P50579 27998678 501 KVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSR 5lyy A 2.17 BS01 7BJ A 1 F110 G152 L153 G154 L159 S273 F274 W298 F322 H351 Q352 F357 F56 G98 L99 G100 L105 S219 F220 W244 F268 H297 Q298 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=14uM remove_due_to_license_issue IC50=14000nM Q13093 27933945 501 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5lz2 A 2.1 BS01 7BX A 1 F110 G152 L153 G154 Q352 A355 F357 F56 G98 L99 G100 Q298 A301 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50~1mM remove_due_to_license_issue Q13093 27933945 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5lz4 A 2.07 BS01 7BW A 1 F110 G152 L153 G154 A155 L159 S273 F274 W298 F322 H351 Q352 A355 F357 F56 G98 L99 G100 A101 L105 S219 F220 W244 F268 H297 Q298 A301 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 Kd=2uM remove_due_to_license_issue IC50=3000nM Q13093 27933945 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5lz5 A 2.05 BS01 7K4 A 1 F110 G152 L153 G154 L159 S273 F274 W298 H351 Q352 A355 F357 F56 G98 L99 G100 L105 S219 F220 W244 H297 Q298 A301 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 Kd=0.45uM remove_due_to_license_issue IC50=1600nM Q13093 27933945 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5lz7 A 2.1 BS01 7BK A 1 F110 G152 L153 G154 A155 L159 S273 F274 W298 F322 H351 Q352 A355 F357 F56 G98 L99 G100 A101 L105 S219 F220 W244 F268 H297 Q298 A301 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 Kd=0.53uM remove_due_to_license_issue IC50=1000nM Q13093 27933945 502 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5lz8 A 2.11 BS01 7BP A 1 F110 G152 L153 G154 A155 L159 H272 S273 F274 W298 F322 H351 Q352 A355 F357 F56 G98 L99 G100 A101 L105 H218 S219 F220 W244 F268 H297 Q298 A301 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=0.98uM remove_due_to_license_issue IC50=5100nM Q13093 27933945 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5lz9 A 2.06 BS01 7BR A 1 F110 G152 L153 G154 A155 S273 F274 W298 F322 H351 Q352 A355 F357 F56 G98 L99 G100 A101 S219 F220 W244 F268 H297 Q298 A301 F303 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=0.12uM remove_due_to_license_issue IC50=32nM Q13093 27933945 503 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINT 5lzg A 1.13 BS01 7BN A 1 E11 Y12 H13 E51 Q56 H57 W88 N90 K91 E11 Y12 H13 E51 Q56 H57 W88 N90 K91 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 28539625 201 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5lzg A 1.13 BS02 7BN E 1 G33 K34 G33 K34 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 28539625 201 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5lzg B 1.13 BS01 7BN A 1 G33 K34 G33 K34 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 28539625 201 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5lzg B 1.13 BS02 7BN B 1 E11 Y12 H13 E51 H57 Q61 W88 N90 K91 E11 Y12 H13 E51 H57 Q61 W88 N90 K91 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 28539625 201 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5lzj C 1.2 BS01 7BT C 1 N14 E51 Q56 H57 Q61 W88 N90 K91 N14 E51 Q56 H57 Q61 W88 N90 K91 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 28539625 202 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5lzj D 1.2 BS01 7BT D 1 H13 N14 E51 Q56 Q61 W88 N90 K91 H13 N14 E51 Q56 Q61 W88 N90 K91 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 28539625 202 TPQNITDLCAEYHNTQIYTLNDKIFSYTESLAGKREMAIITFKNGAIFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 5m04 A 1.85 BS01 GDP A 1 N169 G171 K172 S173 T174 N283 K284 D286 S314 A316 N168 G170 K171 S172 T173 N282 K283 D285 S313 A315 3.6.5.- 0000287,0003924,0005525 Kd=0.46uM remove_due_to_license_issue P42641 28223358 401 GSHMKFVDEASILVVAGDGGNGCVSFRREKYIPKGGPDGGDGGDGGDVWMEADENLNTLIDYRFEKSFRAERGQNGASRDCTGKRGKDVTIKVPVGTRVIDQGTGETMGDMTKHGQRLLVAKGGWHGLGNTRFKSTPRQKTNGTPGDKRELLLELMLLADVGMLGMPNAGKSTFIRAVSAAKPKVADYPFTTLVPSLGVVRMDNEKSFVVADIPGLIEGAAEGAGLGIRFLKHLERCRVLLHLIDIDPIDGTDPVENARIIISELEKYSQDLATKPRWLVFNKIDLLDKVEAEEKAKAIAEALGWEDKYYLISAASGLGVKDLCWDVMTFIIENPVV 5m0d A 2.4 BS06 7C8 A 1 L78 Y82 F210 L213 F249 W254 W260 F274 W275 Y306 L23 Y27 F155 L158 F194 W199 W205 F219 W220 Y251 3.1.4.39 0001953,0003676,0004528,0004622,0004630,0005044,0005509,0005576,0005615,0006644,0006935,0006955,0008270,0008284,0009395,0010634,0016020,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0044849,0046872,0047391,0048714,0050731,0051894,0060326,0071276,0071392,1900026,1903165,2000394 remove_due_to_license_issue Q64610 28165241 921 GSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIKVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDASFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLRLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRAKSINNSKYDPKTIIAALTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDIHLLVDRRWHVARKPLDFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPDEVSRPNYPGIMYLQSEFDLGCTCDGSTKERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWAYFQRVLVKKYASERNGVNVISGPIFDYNYDGLRDTEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCASSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5m0m A 2.1 BS06 7CF A 1 Y82 S169 F210 L213 K248 F249 W254 W260 F273 F274 W275 Y306 Y28 S115 F156 L159 K194 F195 W200 W206 F219 F220 W221 Y252 3.1.4.39 0001953,0003676,0004528,0004622,0004630,0005044,0005509,0005576,0005615,0006644,0006935,0006955,0008270,0008284,0009395,0010634,0016020,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0044849,0046872,0047391,0048714,0050731,0051894,0060326,0071276,0071392,1900026,1903165,2000394 remove_due_to_license_issue Q64610 28165241 925 SGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIKVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDASFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLRLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRAKSINNSKYDPKTIIAALTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDIHLLVDRRWHVARKPLFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPDEVSRPNYPGIMYLQSEFDLGCTCDSTKERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWAYFQRVLVKKYASERNGVNVISGPIFDYNYDGLRDTEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCASSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5m0s A 2.1 BS06 7CW A 1 Y82 L213 K248 F249 H251 W254 W260 F273 F274 W275 Y306 Y27 L158 K193 F194 H196 W199 W205 F218 F219 W220 Y251 3.1.4.39 0001953,0003676,0004528,0004622,0004630,0005044,0005509,0005576,0005615,0006644,0006935,0006955,0008270,0008284,0009395,0010634,0016020,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0044849,0046872,0047391,0048714,0050731,0051894,0060326,0071276,0071392,1900026,1903165,2000394 remove_due_to_license_issue Q64610 28165241 925 GSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIKVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDASFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLRLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRAKSINNSKYDPKTIIAALTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDIHLLVDRRWHVARKPLDCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPDEVSRPNYPGIMYLQSEFDLGCTCDGSTKERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWAYFQRVLVKKYASERNGVNVISGPIFDYNYDGLRDTEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCASSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5m17 A 1.03 BS01 7D1 B 1 Y46 W126 H154 E156 Y195 Y252 E336 Y16 W96 H124 E126 Y165 Y222 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 27992199 1 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 5m17 A 1.03 BS02 MAN B 1 H63 R295 E333 H335 E336 H33 R265 E303 H305 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 27992199 2 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 5m1z A 2.0 BS01 6LW B 1 W169 E170 Q195 M226 E242 Y337 W148 E149 Q174 M205 E221 Y316 3.2.1.55 0016798,0046556,0046872 remove_due_to_license_issue B8ZY56 28266777 1 GKTFSNVEIFDPPTNYRDPQVLYARPLELSDGTLLGTWENYSPEPPNVWFPIVKSKDGGKTWKEISKVKDTQNNWGLRYQPQLYELPRAFGKYPKGTVLCSGSSIPSDLSETLIEVYASRDKGYTWEFVSHVALGGEALPNPGLTPVWEPFLMTYKEKLILYYSDQRDNATHSQKLVHQTTTDLKKWSKVVDDTKYANYYARPGMPTVAKLPNNEYIYVYEYGGGPNPPAGSDYWFPVYYRLSKDPQKFLNKAHHQIVSNDGTTPAGSPYVVWTPYGGKNGTIVVSCGTRSEIFTNQALGDASAWKKWDVPQPTAYTRSLLTFQKDPDLLMIMGAGILPPAGGKNTVSASVVRLSEVMK 5m1z A 2.0 BS02 AHR B 1 E60 Q101 E39 Q80 3.2.1.55 0016798,0046556,0046872 remove_due_to_license_issue B8ZY56 28266777 2 GKTFSNVEIFDPPTNYRDPQVLYARPLELSDGTLLGTWENYSPEPPNVWFPIVKSKDGGKTWKEISKVKDTQNNWGLRYQPQLYELPRAFGKYPKGTVLCSGSSIPSDLSETLIEVYASRDKGYTWEFVSHVALGGEALPNPGLTPVWEPFLMTYKEKLILYYSDQRDNATHSQKLVHQTTTDLKKWSKVVDDTKYANYYARPGMPTVAKLPNNEYIYVYEYGGGPNPPAGSDYWFPVYYRLSKDPQKFLNKAHHQIVSNDGTTPAGSPYVVWTPYGGKNGTIVVSCGTRSEIFTNQALGDASAWKKWDVPQPTAYTRSLLTFQKDPDLLMIMGAGILPPAGGKNTVSASVVRLSEVMK 5m23 A 1.97 BS01 7DC A 1 S49 A65 G89 I90 S91 D107 F133 K259 Y260 C261 F263 I305 S17 A33 G57 I58 S59 D75 F101 K227 Y228 C229 F231 I273 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue P61964 28970883 401 PNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKS 5m25 A 2.43 BS01 7DU A 1 S49 I90 S91 D107 F133 K259 Y260 C261 F263 I305 S17 I58 S59 D75 F101 K227 Y228 C229 F231 I273 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue P61964 28970883 401 PNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKS 5m29 A 1.5 BS01 CBY A 1 P31 A32 Y50 W66 W85 G87 F162 F168 W196 D242 E245 R246 P10 A11 Y29 W45 W64 G66 F141 F147 W175 D205 E208 R209 ? 0015889,0031419,0042597 remove_due_to_license_issue P37028 28128319 301 AAPRVITLSPANTELAFAAGITPVGVSSYSDYPPQAQKIEQVSTWQGMNLERIVALKPDLVIAWRGGNAERQVDQLASLGIKVMWVDATSIEQIANALRQLAPWSPQPDKAEQAAQSLLDQYAQLKAQYADKPKKRVFLQFGINPPFTSGKESIQNQVLEVCGGENIFKDSRVPWPQVSREQVLARSPQAIVITGKIPVIPLTSDWFERASPRIILAAQQLCNALSQVD 5m2q A 1.7 BS01 CBY A 1 P31 A32 Y50 F66 W85 G87 F162 F168 W196 S241 D242 E245 R246 P9 A10 Y28 F44 W63 G65 F140 F146 W174 S203 D204 E207 R208 ? 0015889,0031419,0042597 remove_due_to_license_issue P0A910,P37028 28128319 301 APRVITLSPANTELAFAAGITPVGVSSYSDYPPQAQKIEQVSTFQGMNLERIVALKPDLVIAWRGGNAERQVDQLASLGIKVMWVDATSIEQIANALRQLAPWSPQPDKAEQAAQSLLDQYAQLKAQYADKPKKRVFLQFGINPPFTSGKESIQNQVLEVCGGENIFKDSRVPWPQVSREQVLARSPQAIVITGKIPVIPLTSDWFERASPRIILAAQQLCNALSQVD 5m2v A 3.18 BS01 7E5 A 1 Y61 P88 L89 T90 R95 S141 M189 E190 Y57 P84 L85 T86 R91 S137 M185 E186 ? 0015276,0016020 remove_due_to_license_issue P22756 28005385 301 TLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGCP 5m34 A 1.6 BS01 CBY A 1 P31 A32 Y50 Y66 W85 G87 F162 F168 W196 E245 R246 P10 A11 Y29 Y45 W64 G66 F141 F147 W175 E207 R208 ? 0015889,0031419,0042597 remove_due_to_license_issue P37028 28128319 301 AAPRVITLSPANTELAFAAGITPVGVSSYSDYPPQAQKIEQVSTYQGMNLERIVALKPDLVIAWRGGNAERQVDQLASLGIKVMWVDATSIEQIANALRQLAPWSPQPDKAEQAAQSLLDQYAQLKAQYADKPKKRVFLQFGINPPFTSGKESIQNQVLEVCGGENIFKDSRVPWPQVSREQVLARSPQAIVITKIPVIPLTSDWFERASPRIILAAQQLCNALSQVD 5m39 A 1.38 BS01 7EA A 1 W81 P82 F83 L92 N140 W40 P41 F42 L51 N99 ? remove_due_to_license_issue IC50=24000nM O60885 28910100 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 5m3a A 1.65 BS01 7E7 A 1 W81 P82 L92 N140 I146 W40 P41 L51 N99 I105 ? remove_due_to_license_issue IC50=2000nM O60885 28910100 303 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5m3b A 1.5 BS01 CBY A 1 P31 A32 Y50 W85 G87 F168 W196 S241 E245 R246 P9 A10 Y28 W63 G65 F146 W174 S203 E207 R208 ? 0015889,0031419,0042597 remove_due_to_license_issue P37028 28128319 302 APRVITLSPANTELAFAAGITPVGVSSYSDYPPQAQKIEQVSTLQGMNLERIVALKPDLVIAWRGGNAERQVDQLASLGIKVMWVDATSIEQIANALRQLAPWSPQPDKAEQAAQSLLDQYAQLKAQYADKPKKRVFLQFGINPPFTSGKESIQNQVLEVCGGENIFKDSRVPWPQVSREQVLARSPQAIVITGKIPVIPLTSDWFERASPRIILAAQQLCNALSQVD 5m44 A 2.71 BS01 7EY A 1 V53 E55 V66 I95 E114 H115 M163 I174 V51 E53 V64 I93 E112 H113 M161 I172 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 28085026 401 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 5m4c A 1.935 BS01 7EY A 1 L45 V53 V66 K68 F113 V116 M163 I174 D175 L43 V51 V64 K66 F111 V114 M161 I172 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 28085026 401 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 5m4f A 1.519 BS01 7FC A 1 V66 K68 F113 E114 H115 V116 N118 M163 I174 D175 V65 K67 F112 E113 H114 V115 N117 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 28085026 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQ 5m4i A 2.218 BS01 7FC A 1 Y50 V66 F113 H115 V116 M163 D175 Y48 V64 F111 H113 V114 M161 D173 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 28085026 401 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQAR 5m4k A 2.6 BS02 7F9 A 1 N247 R250 A251 D282 V287 T346 N232 R235 A236 D267 V272 T316 H239 E243 K246 N247 H224 E228 K231 N232 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0031670,0034614,0042593,0042803,0045254,0050848,0072332 remove_due_to_license_issue IC50=4460nM, Ki=2170nM Q15119 28199108 402 GSAPKYIEHFSKFSPSPLSMKQFLDFNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTAPYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVY 5m4q A 1.73 BS04 PRO A 1 H255 H366 R398 E412 H250 H361 R393 E407 D60 H255 D276 D287 H366 H370 H377 E412 Y416 R450 E452 D55 H250 D271 D282 H361 H365 H372 E407 Y411 R445 E447 3.4.13.9 0004181,0005515,0006508,0006520,0008233,0008237,0016805,0030145,0030574,0043069,0046872,0070006,0070062,0102009 Ki=0.31mM remove_due_to_license_issue P12955 28677335 504 GPSFWLGNETLKVPLALFALNRQRLCERLRKNPAVQAGSIVVLQGGEETQRYCTDTGVLFRQESFFHWAFGVTEPGCYGVIDVDTGKSTLFVPRLPASHATWMGKIHSKEHFKEKYAVDDVQYVDEIASVLTSQKPSVLLTLRGVNTDSGSVCREASFDGISKFEVNNTILHPEIVECRVFKTDMELEVLRYTNKISSEAHREVMKAVKVGMKEYELESLFEHYCYSRGGMRHSSYTCICGSGENSAVLHYGHAGAPNDRTIQNGDMCLFDMGGEYYCFASDITCSFPANGKFTADQKAVYEAVLRSSRAVMGAMKPGVWWPDMHRLADRIHLEELAHMGILSGSVDAMVQAHLGAVFMPHGLGHFLGIDVHDVGGYPEGVERIDEPGLRSLRTARHLQPGMVLTVEPGIYFIDHLLDEALADPARASFLNREVLQRFRGFGGVRIEEDVVVTDSGIELLTCVPRTVEEIEACMAGCDKAFTPF 5m4q B 1.73 BS04 PRO B 1 H255 H366 R398 E412 R450 H250 H361 R393 E407 R445 D60 H255 D276 D287 H366 H370 H377 E412 Y416 R450 E452 D55 H250 D271 D282 H361 H365 H372 E407 Y411 R445 E447 3.4.13.9 0004181,0005515,0006508,0006520,0008233,0008237,0016805,0030145,0030574,0043069,0046872,0070006,0070062,0102009 Ki=0.31mM remove_due_to_license_issue P12955 28677335 504 GPSFWLGNETLKVPLALFALNRQRLCERLRKNPAVQAGSIVVLQGGEETQRYCTDTGVLFRQESFFHWAFGVTEPGCYGVIDVDTGKSTLFVPRLPASHATWMGKIHSKEHFKEKYAVDDVQYVDEIASVLTSQKPSVLLTLRGVNTDSGSVCREASFDGISKFEVNNTILHPEIVECRVFKTDMELEVLRYTNKISSEAHREVMKAVKVGMKEYELESLFEHYCYSRGGMRHSSYTCICGSGENSAVLHYGHAGAPNDRTIQNGDMCLFDMGGEYYCFASDITCSFPANGKFTADQKAVYEAVLRSSRAVMGAMKPGVWWPDMHRLADRIHLEELAHMGILSGSVDAMVQAHLGAVFMPHGLGHFLGIDVHDVGGYPEGVERIDEPGLRSLRTARHLQPGMVLTVEPGIYFIDHLLDEALADPARASFLNREVLQRFRGFGGVRIEEDVVVTDSGIELLTCVPRTVEEIEACMAGCD 5m4u A 2.195 BS01 7FC A 1 L46 R48 V67 K69 F114 E115 Y116 I117 M164 I175 D176 L44 R46 V65 K67 F112 E113 Y114 I115 M162 I173 D174 I153 H155 V158 L172 V191 I151 H153 V156 L170 V189 2.7.11.1 0000785,0001669,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005829,0005956,0006302,0006338,0006468,0006915,0006974,0007283,0016055,0021987,0031519,0032435,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0097421,0106310,0140823,0140855,0140857,1901524,1903955,1905818,1990244,2001234 remove_due_to_license_issue P19784 28085026 401 GPAAGSRARVYAEVNSLRSREYWDYEAHVPSWGNQDGYQLVRKLGRGKYSEVFEAINITNNERVVVKILKPVKKKKIKREVKILENLRGGTNIIKLIDTVKDPVSKTPALVFEYINNTDFKQLYQILTDFDIRFYMYELLKALDYCHSKGIMHRDVKPHNVMIDHQQKKLRLIDWGLAEFYHPAQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRREPFFHGQDNYDQLVRIAKVLGTEELYGYLKKYHIDLDPHFNDILGQHSRKRWENFIHSENRHLVSPEALDLLDKLLRYDHQQRLTAKEAMEHPYFYPVVKEQSQ 5m51 A 1.899 BS01 NU6 A 1 K37 E87 Y88 C89 F148 K35 E85 Y86 C87 F146 D141 K143 A145 N146 D159 T179 D139 K141 A143 N144 D157 T161 2.7.11.1 0004672,0005524,0006468 ic50=19uM remove_due_to_license_issue P51955 27833088 301 SRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSDGGHTVLHRDLKPANVFLDGKQNVKLGDFVGTPYYMSPEQMNRMSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHH 5m53 A 1.9 BS01 7GJ A 1 I14 Y19 K37 E87 Y88 C89 G92 D93 F148 I8 Y13 K28 E78 Y79 C80 G83 D84 F139 D141 K143 A145 N146 D159 T179 D132 K134 A136 N137 D150 T156 2.7.11.1 0004672,0005524,0006468 ic50=0.62uM remove_due_to_license_issue P51955 27833088 301 DYEVLYTIGTGSYGRCQKIRRGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSDGGHTVLHRDLKPANVFLDGKQNVKLGDFGLVGTPYYMSPEQMNRMSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHH 5m55 A 2.4 BS01 7GG A 1 C22 E87 Y88 C89 G92 C16 E81 Y82 C83 G86 K143 A145 N146 D159 T179 K127 A129 N130 D143 T144 2.7.11.1 0004672,0005524,0006468 ic50=0.24uM remove_due_to_license_issue P51955 27833088 301 SRAEDYEVLYTIGTRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSLKPANVFLDGKQNVKLGDTPYYMSPEQMNNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 5m56 A 2.237 BS01 7FC A 1 L46 V67 K69 F114 E115 Y116 I117 M164 I175 D176 L45 V66 K68 F113 E114 Y115 I116 M163 I174 D175 I153 H155 V158 L172 V191 I152 H154 V157 L171 V190 2.7.11.1 0000785,0001669,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005829,0005956,0006302,0006338,0006468,0006915,0006974,0007283,0016055,0021987,0031519,0032435,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0097421,0106310,0140823,0140855,0140857,1901524,1903955,1905818,1990244,2001234 remove_due_to_license_issue P19784 28085026 401 PGPAAGSRARVYAEVNSLRSREYWDYEAHVPSWGNQDGYQLVRKLGRGKYSEVFEAINITNNERVVVKILKPVKKKKIKREVKILENLRGGTNIIKLIDTVKDPVSKTPALVFEYINNTDFKQLYQILTDFDIRFYMYELLKALDYCHSKGIMHRDVKPHNVMIDHQQKKLRLIDWGLAEFYHPAQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRREPFFHGQDNYDQLVRIAKVLGTEELYGYLKKYHIDLDPHFNDILGQHSRKRWENFIHSENRHLVSPEALDLLDKLLRYDHQQRLTAKEAMEHPYFYPVVKEQ 5m57 A 2.3 BS01 4SP A 1 G17 Y19 C22 K37 E87 C89 G92 F148 D159 G15 Y17 C20 K35 E85 C87 G90 F146 D157 D141 K143 A145 N146 D159 T179 D139 K141 A143 N144 D157 T161 2.7.11.1 0004672,0005524,0006468 ic50=12uM remove_due_to_license_issue P51955 27833088 301 SRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSDGGHTVLHRDLKPANVFLDGKQNVKLGDFVGTPYYMSPEQMNRMSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLILEHHHHHH 5m5d A 1.07 BS01 DGO B 1 Y46 W126 H154 E156 Y195 Y252 E333 E336 Y14 W94 H122 E124 Y163 Y220 E301 E304 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 27992199 1 LGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 5m5d A 1.07 BS02 MAN B 1 H63 R295 E333 H335 E336 H31 R263 E301 H303 E304 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 27992199 2 LGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 5m5q A 2.2 BS02 7K1 A 1 E76 V77 M78 W136 H138 H140 Y143 D151 T154 E73 V74 M75 W124 H126 H128 Y131 D139 T142 3.4.-.- 0008233,0008237 ic50=0.09uM remove_due_to_license_issue IC50=60nM Q92905 27981705 302 SGSGMAQKTWELANNMQEAQSIDEIYKYDKKQQQEILAAKPWTKDHHYFKYCKISALALLKMVMHARSGGNLEVMGLMLGKVDGETMIIMDSFALPAQAAAYEYMAAYIENAKQVGRLENAIGWYHSHPGYGCWLSGIDVSTQMLNQQFQEPFVAVVIDPTRKVNLGAFRTYPKGYKPPDEGPSEYQTIPLNKIEDFGVHCKQYYALEVSYFKSSLDRK 5m63 H 2.74 BS01 SIA A 1 Y126 H127 Y107 H108 remove_due_to_license_issue 28439022 2 QSLEESGGDLVKPGASLTLTCKASGLDLPSYFMCWVRQAPGKGLEWIACIRSSSNEILYYASWAKGRFTISKTSSTTVTLQMTSLTAADTATYFCARDYFGEGDVFYHGGVFGLWGSGTLVTVSSGQPKAPSVFPLAPCCGDTPSSTVTLGCLVKGYLPEPVTVTWNSGTLTNGVRTFPSVRQSSGLYSLSSVVSVTSSSQPVTCNVAHPATNTKVDKTVAP 5m63 L 2.74 BS01 SIA A 1 Y52 R56 Y29 R33 remove_due_to_license_issue 28439022 2 VVLTQTPSSVSAAVGGSVTISCQSSQSLYNNNRLAWYQQKAGQPPKLLIYKASTLESGVPSRFKGSGAGTQFTLTISDVVCDDAATYYCAGYKSNSDDGTAFGGGTEVVVKGDPVAPTVLIFPPAADQVATGTVTIVCVANKYFPDVTVTWEVDGTTQTTGIENSKTPQNSADCTYNLSSTLTLTSTQYNSHKEYTCKVTQGTTSVVQSFNRGDC 5m6f A 2.39 BS02 7HU A 1 G306 L307 T308 D309 W310 E314 Q319 W323 G59 L60 T61 D62 W63 E67 Q72 W76 2.3.2.27 ic50=220nM remove_due_to_license_issue P98170 28492317 403 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECL 5m6h A 2.5 BS02 7J6 A 1 K297 G306 L307 T308 D309 W310 K311 E314 Q319 W323 K50 G59 L60 T61 D62 W63 K64 E67 Q72 W76 2.3.2.27 ic50=150nM remove_due_to_license_issue P98170 28492317 403 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEEC 5m6m A 2.37 BS02 7H8 A 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 K50 G59 L60 T61 D62 W63 E67 Q72 W76 2.3.2.27 ic50=44nM remove_due_to_license_issue P98170 28492317 403 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEEC 5m6u A 2.85 BS01 7KA A 1 M752 P758 W760 Y813 E826 V828 D832 M900 I910 M659 P665 W667 Y720 E733 V735 D739 M794 I804 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue IC50=4.7nM O00329 28105286 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPLLVNVKFEGSEESFTFQVSTKDVPLALMACPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDESLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEDCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHSVTEEEQLQLREILERRGSGELYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSGGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFKTRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5m77 A 1.46 BS01 7K2 C 1 F122 D124 D125 W172 C183 D228 Y243 D294 F84 D86 D87 W134 C145 D190 Y205 D256 ? 0005975,0030246 remove_due_to_license_issue Q9Z4P9 28766587 1 SDGDTAMKAFNDTFWDPNAKMFWKDSKREKHQDFWVEAELWELVMDAYQHTSDPALKAELKTQIDDVYDGTVAKYGQDWTNNPFNDDIMWWAMGSARAYQITGNPRYLEAARDHFDFVYDTQWDEEFANGGIWWLNSDHNTKNACINFPAAQAALYLYDITKDEHYLNAATKIFRWGKTMLTDGNGKVFDRIEIEHGAVPDATHYNQGTYIGSAVGLYKATGNAVYLDDAVKAAKFTKNHLVDSNGVLNYEGPNGDLKGGKTILMRNLAHLQKTLDETGQYPEFSAEFDEWLAFNIEMAWSHQNSDHIVDGNWAGGTYESWSSAAAVQALNGI 5m77 A 1.46 BS02 7K3 C 1 D228 D239 T241 N292 D190 D201 T203 N254 ? 0005975,0030246 remove_due_to_license_issue Q9Z4P9 28766587 2 SDGDTAMKAFNDTFWDPNAKMFWKDSKREKHQDFWVEAELWELVMDAYQHTSDPALKAELKTQIDDVYDGTVAKYGQDWTNNPFNDDIMWWAMGSARAYQITGNPRYLEAARDHFDFVYDTQWDEEFANGGIWWLNSDHNTKNACINFPAAQAALYLYDITKDEHYLNAATKIFRWGKTMLTDGNGKVFDRIEIEHGAVPDATHYNQGTYIGSAVGLYKATGNAVYLDDAVKAAKFTKNHLVDSNGVLNYEGPNGDLKGGKTILMRNLAHLQKTLDETGQYPEFSAEFDEWLAFNIEMAWSHQNSDHIVDGNWAGGTYESWSSAAAVQALNGI 5m7m A 2.7 BS02 7HR A 1 I168 F211 L214 L217 F250 H252 W255 W261 F274 F275 I105 F148 L151 L154 F187 H189 W192 W198 F211 F212 3.1.4.39 0003676,0005044,0006955,0016787,0030247,0046872 remove_due_to_license_issue IC50=300nM Q13822 28731719 907 GSCKGRCFELCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFSNNAKYDPKAIIANLTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPLDCFFQGDHGFDNKVNSMQTVFVGYGPTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPEEVTRPNYPGIMYLQSDFDLGCTCSTEERHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQATSCVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 5m7s A 2.4 BS01 NHT A 1 G67 Y69 K98 D174 D175 C215 Y219 V254 W278 N280 D285 G10 Y12 K41 D117 D118 C158 Y162 V197 W221 N223 D228 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 Ki=0.9nM remove_due_to_license_issue Ki=21nM, EC50=13nM, IC50=0.410000nM O60502 28346405 1001 RRFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNVLYSPQMALKLALTEWLQEFGVPHQFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVSSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCEPWAFRGGLAGEFQRLLPI 5m7s B 2.4 BS01 NHT B 1 G67 K98 D174 D175 C215 Y219 V254 W278 N280 D285 G9 K40 D116 D117 C157 Y161 V196 W220 N222 D227 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 Ki=0.9nM remove_due_to_license_issue Ki=21nM, EC50=13nM, IC50=0.410000nM O60502 28346405 1001 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNGVRVLYSPQMALKLALTEWLQEFGVPHFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVSSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCRPWAFRGGLAGEFQRLLPI 5m7t A 2.6 BS01 GDV A 1 G67 K98 D175 Y219 F223 V254 W278 N280 D285 G9 K40 D117 Y161 F165 V196 W220 N222 D227 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue O60502 28346405 1001 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNDVLYSPQMALKLALTEWLQEFGVPHQFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVSVKDSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCRSHSQEPWAFRGGLAGEFQRLLPI 5m7t B 2.6 BS01 GDV B 1 G67 K98 D175 Y219 V254 W278 N280 D285 G9 K40 D117 Y161 V196 W220 N222 D227 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue O60502 28346405 1001 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNGVRDVLYSPQMALKLALTEWLQEFGVPHQFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVDSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCREPWAFRGGLAGEFQRLLPI 5m7u A 2.3 BS01 XHA A 1 G67 Y69 D174 D175 Y219 W278 N280 D285 N313 G9 Y11 D116 D117 Y161 W220 N222 D227 N255 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 Ki=8nM remove_due_to_license_issue O60502 28346405 1001 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNDVLYSPQMALKLALTEWLQEFGVPHQFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVSSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCLIGDQEPWAFRGGLAGEFQRLLPI 5m7u A 2.3 BS02 XHA B 1 W645 S649 W679 W406 S410 W432 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 Ki=8nM remove_due_to_license_issue O60502 28346405 1001 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNDVLYSPQMALKLALTEWLQEFGVPHQFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVSSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCLIGDQEPWAFRGGLAGEFQRLLPI 5m7u B 2.3 BS01 XHA B 1 G67 F68 Y69 D174 D175 Y219 V254 W278 N280 D285 Y286 G9 F10 Y11 D116 D117 Y161 V196 W220 N222 D227 Y228 3.2.1.169 0004415,0005634,0005737,0005829,0006044,0006493,0006516,0006517,0009100,0015929,0016020,0016231,0016798,0042802,0102571,1901135 Ki=8nM remove_due_to_license_issue O60502 28346405 1001 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNGVDVLYSPQMALKLALTEWLQEFGVPHQFVPGPNEKPLYTAEPVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVSSEKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCRDQEPWAFRGGLAGEFQRLLPI 5m8i A -1.00 BS01 rna B 0 Q22 F32 Y34 H35 K59 F61 I62 K70 F72 F74 K98 K101 R106 Q22 F32 Y34 H35 K59 F61 I62 K70 F72 F74 K98 K101 R106 ? 0003676,0003723 remove_due_to_license_issue O95319 28935965 115 ~ 119 MGSSHHHHHHSSGLVPRGSHMQKEGPEGANLFIYHLPQEFGDQDILQMFMPFGNVISAKVFIDKQTNLSKCFGFVSYDNPVSAQAAIQAMNGFQIGMKRLKVQLKRSKNDSKPW 5m9w A 1.21 BS06 7GR A 1 N112 A113 F130 E143 H146 Y157 E166 R203 H231 N112 A113 F130 E143 H146 Y157 E166 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=5.7mM remove_due_to_license_issue P00800 28696673 412 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5ma7 E 1.3 BS06 7K0 E 1 N112 A113 E143 H146 Y157 E166 R203 H231 N112 A113 E143 H146 Y157 E166 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Kd=0.336mM remove_due_to_license_issue P00800 28696673 412 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5mae A 1.0 BS01 7KN A 1 G23 C25 N66 M70 D162 H163 G23 C25 N66 M70 D162 H163 Q19 C25 H163 N187 Q19 C25 H163 N184 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 27992115 301 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 5maj A 1.0 BS01 7KH A 1 G23 C25 N66 G67 G68 D162 G23 C25 N66 G67 G68 D162 Q19 C25 H163 N187 Q19 C25 H163 N186 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 27992115 301 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTSDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 5mar A 1.89 BS03 7KE A 1 F119 L134 L138 I169 I232 V233 F66 L81 L85 I116 I179 V180 P94 D95 F96 R97 N168 D170 H187 P41 D42 F43 R44 N115 D117 H134 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=41.2uM remove_due_to_license_issue IC50=41200nM Q8IXJ6 28240897 403 HMERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPSTGLYDNLEKYHLPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGQSDPFLGMIMGLGGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQ 5mat A 2.069 BS02 7KJ A 1 I93 P94 F96 F119 A135 L138 Y139 F143 I169 F190 F235 I39 P40 F42 F63 A79 L82 Y83 F87 I113 F134 F179 P94 D95 F96 R97 N168 D170 H187 P40 D41 F42 R43 N112 D114 H131 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=0.58uM remove_due_to_license_issue IC50=580nM Q8IXJ6 28135086 402 MERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSTGLYDNLEKYHLPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGQSDPFLGMIMGLGGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5may A 1.65 BS03 FUL A 1 S22 A23 D96 D99 D101 D104 S22 A23 D96 D99 D101 D104 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 29272578 202 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5may A 1.65 BS04 PK6 A 1 G24 D96 S97 G24 D96 S97 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 29272578 203 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5may B 1.65 BS03 FUL B 1 N21 S22 A23 D96 D99 D101 D104 N21 S22 A23 D96 D99 D101 D104 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 29272578 202 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5may B 1.65 BS04 PK6 B 1 G24 R72 D96 G24 R72 D96 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 29272578 203 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5mb1 A 1.65 BS04 7KT A 1 A23 G24 D96 S97 A23 G24 D96 S97 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 29272578 204 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5mb1 B 1.65 BS04 7KT B 1 G24 D96 G24 D96 ? 0030246,0046872 remove_due_to_license_issue A0A0H2ZE85 29272578 204 ATQGVFTLPANTQFGVTAFANSAGTQTVNVQVNNETVATFTGQSTNNAIIGSKVLNSGGGGKVQILVSVNGRSSDLVSAQVILANELNFALVGSEDSTDNDYNDAVVVINWPLG 5mby A 1.55 BS04 PRO A 1 H255 H366 H377 R398 E412 R450 H250 H361 H372 R393 E407 R445 3.4.13.9 0004181,0005515,0006508,0006520,0008233,0008237,0016805,0030145,0030574,0043069,0046872,0070006,0070062,0102009 remove_due_to_license_issue P12955 30066404 504 GPSFWLGNETLKVPLALFALNRQRLCERLRKNPAVQAGSIVVLQGGEETQRYCTDTGVLFRQESFFHWAFGVTEPGCYGVIDVDTGKSTLFVPRLPASHATWMGKIHSKEHFKEKYAVDDVQYVDEIASVLTSQKPSVLLTLRGVNTDSGSVCREASFDGISKFEVNNTILHPEIVECQVFKTDMELEVLRYTNKISSEAHREVMKAVKVGMKEYELESLFEHYCYSRGGMRHSSYTCICGSGENSAVLHYGHAGAPNDRTIQNGDMCLFDMGGEYYCFASDITCSFPANGKFTADQKAVYEAVLRSSRAVMGAMKPGVWWPDMHRLADRIHLEELAHMGILSGSVDAMVQAHLGAVFMPHGLGHFLGIDVHDVGGYPEGVERIDEPGLRSLRTARHLQPGMVLTVEPGIYFIDHLLDEALADPARASFLNREVLQRFRGFGGVRIEEDVVVTDSGIELLTCVPRTVEEIEACMAGCDAFTPFS 5mby B 1.55 BS04 PRO B 1 H255 H366 H377 R398 E412 H250 H361 H372 R393 E407 3.4.13.9 0004181,0005515,0006508,0006520,0008233,0008237,0016805,0030145,0030574,0043069,0046872,0070006,0070062,0102009 remove_due_to_license_issue P12955 30066404 504 GPSFWLGNETLKVPLALFALNRQRLCERLRKNPAVQAGSIVVLQGGEETQRYCTDTGVLFRQESFFHWAFGVTEPGCYGVIDVDTGKSTLFVPRLPASHATWMGKIHSKEHFKEKYAVDDVQYVDEIASVLTSQKPSVLLTLRGVNTDSGSVCREASFDGISKFEVNNTILHPEIVECQVFKTDMELEVLRYTNKISSEAHREVMKAVKVGMKEYELESLFEHYCYSRGGMRHSSYTCICGSGENSAVLHYGHAGAPNDRTIQNGDMCLFDMGGEYYCFASDITCSFPANGKFTADQKAVYEAVLRSSRAVMGAMKPGVWWPDMHRLADRIHLEELAHMGILSGSVDAMVQAHLGAVFMPHGLGHFLGIDVHDVGGYPEGVERIDEPGLRSLRTARHLQPGMVLTVEPGIYFIDHLLDEALADPARASFLNREVLQRFRGFGGVRIEEDVVVTDSGIELLTCVPRTVEEIEACMAGCDAFTPF 5meh A 0.95 BS01 DMJ A 1 R363 P364 E365 Y423 E427 T451 E452 R339 P340 E341 Y399 E403 T427 E428 E121 R125 D249 E365 E97 R101 D225 E341 3.2.1.113 0004559,0004571,0005509,0005975,0016020,0016798,0046872 Kd=481nM remove_due_to_license_issue B0SWV2 28256791 506 ASETTPEDWKALAADVRSEFQWAWQGYVAKAWGKDEINPVSGTSRSFFIEGHDLGLSLVEALDTLWIMGLDAEFQAGVDWVKANLSFDVDGNAQVFETNIRLVGGLLSAHLASGDPVLLAKARDLADRLAKAFEASPHGLPWRYVNLRTGAVSDPETNLAEIGTYLSEFGVLSQLTGERKYFDMAKRAMRHTLDRRSKIGLMAANIHAMTGAFTSRNASIDVYADSFYEYLWDAWALFGDEDCKRWAVECVDAQLAHQAKRYDGRLWFPMVDFETGAVTGTAQSELAAYYAGLLGQVGRKAQGDDYLASFTYLQATFGVIPESIDVTTGQPRRKHTGLRPEYPDACLNLWLIDRDPRYRRLAAIHYREMKATSRAAFGYTALKDITTRPMTQDDNCPGYWWSEQMKYYYLLFSDTPRIDYGQLQLSTEANVLRGFRKV 5mek A 1.74 BS01 A3P A 1 K93 G95 T96 T97 W98 R177 S185 Y243 F284 Y311 F312 R313 K314 G315 K68 G70 T71 T72 W73 R152 S160 Y218 F259 Y286 F287 R288 K289 G290 K93 H155 S185 K68 H130 S160 2.8.2.38 0005737,0008146,0016740,0019761,0047364,0080066,0080067,0080068,0080069,0080070,0080071,0120527 remove_due_to_license_issue Q9C9C9 28646214 401 ESTEFEKNQKRYQDLISTFPHEKGWRPKEPLIEYGGYWWLPSLLEGCIHAQEFFQARPSDFLVCSYPKTGTTWLKALTFAIANRSRFDDSSNPLLKRNPHEFVPYIEIDFPFFPEVDVLKDKGNTLFSTHIPYELLPDSVVKSGCKMVYIWREPKDTFISMWTFLHKERTELGPVSNLEESFDMFCRGLSGYGPYLNHILAYWKAYQENPDRILFLKYETMRADPLPYVKSLAEFMGHGFTAEEEEKGVVEKVVNLCSFETLKNLEANKGEKDREDRPGVYANSAYFRKGKVGDWSNYLTPEMAARIDGLMEEKFKGTGLLE 5mes A 2.24 BS01 7LT A 1 H224 M231 L246 V249 M250 H252 V253 R263 T266 L267 F270 G271 H53 M60 L75 V78 M79 H81 V82 R92 T95 L96 F99 G100 ? 0042981 Kd=0.34uM remove_due_to_license_issue P97287,Q07820 28197319 401 DDLYRQSLEIISRYLREQATGSKDSKPLGEAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 5mev A 2.94 BS01 7LW A 1 H224 A227 M231 H252 V253 R263 T266 F270 H53 A56 M60 H81 V82 R92 T95 F99 ? 0042981 remove_due_to_license_issue P97287,Q07820 28197319 401 DDLYRQSLEIISRYLREQATGSKDSKPLGEAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 5mey A 2.05 BS01 dna D 0 T77 L78 L82 Q83 A85 K88 T63 L64 L68 Q69 A71 K74 ? 0005667,0006355 remove_due_to_license_issue Q13485 29234012 1 ~ 18 ACLSIVHSLMCHRQGGESETFAKRAIESLVKKLKEKKDELDSLITAITTNGAHPSKCVTIQRTLDGRLQVAGRKGFPHVIYARLWRWPDLHKNELKHVKYCQYAFDLKCDSVCVNPYHYERVVS 5mez A 2.98 BS01 dna D 0 R38 T77 L78 L82 Q83 K88 R24 T63 L64 L68 Q69 K74 ? 0005667,0006355 remove_due_to_license_issue Q13485 29234012 2 ~ 16 ACLSIVHSLMCHRQGGESETFAKRAIESLVKKLKEKKDELDSLITAITTNGAHPSKCVTIQRTLDGRLQVAGRKGFPHVIYARLWRWPDLHKNELKHVKYCQYAFDLKCDSVCVNPYHYERVVSP 5mf6 A 1.87 BS03 7M2 A 1 I61 P62 F64 F86 I52 P53 F55 F77 P62 D63 F64 R65 N114 D116 H133 P53 D54 F55 R56 N105 D107 H124 2.3.1.-,2.3.1.286,2.4.2.- 0070403 Kd=38uM remove_due_to_license_issue EC50=38000nM Q8N6T7 27990725 410 PFTADKGKCGLPEIFDPPEELERKVWELARLVWQSSSVVFHTGAGISTASGIPDFRGPHGVWTMEERGLAPKFDTTFESARPTQTHMALVQLERVGLLRFLVSQNVDGLHVRSGFPRDKLAELHGNMFVEECAKCKTQYVRDTVVGTMGLKATGRLCTVACRGELRDTILDWEDSLPDRDLALADEASRNADLSITLGTSLQIRPSGNLPLATKRRGGRLVIVNLQPTKHDRHADLRIHGYVDEVMTRLMKHLGLEIPAWDGPRVLERALPPLPRPPTPKLE 5mfr A 1.4 BS02 7MK A 1 E121 M260 M263 E264 H297 E298 H301 E320 Y376 Y381 E119 M258 M261 E262 H295 E296 H299 E318 Y374 Y379 E264 H297 E298 H301 E320 N373 Y381 E262 H295 E296 H299 E318 N371 Y379 3.4.11.2 0004177,0005515,0005886,0006508,0008237,0008270,0042802,0046872 Ki=50000nM remove_due_to_license_issue P04825 28383176 1002 QQPQAKYRHDYRAPDYQITDIDLTFDLDAQKTVVTAVSQAVRHGASDAPLRLNGEDLKLVSVHINDEPWTAWKEEEGALVISNLPERFTLKIINEISPAANTALEGLYQSGDALCTQCEAEGFRHITYYLDRPDVLARFTTKIIADKIKYPFLLSNGNRVAQGELENGRHWVQWQDPFPKPCYLFALVAGDFDVLRDTFTTRSGREVALELYVDRGNLDRAPWAMTSLKNSMKWDEERFGLEYDLDIYMIVAVDFFNMGAMENKGLNIFNSKYVLARTDTATDKDYLDIERVIGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSSDLGSRAVNRINNVRTMRGLQFAEDASPMAHPIRPDMVIEMNNFYTLTVYEKGAEVIRMIHTLLGEENFQKGMQLYFERHDGSAATCDDFVQAMEDASNVDLSHFRRWYSQSGTPIVTVKDDYNPETEQYTLTISQRTPATPDQAEKQPLHIPFAIELYDNEGKVIPLQKGGHPVNSVLNVTQAEQTFVFDNVYFQPVPALLCEFSAPVKLEYKWSDQQLTFLMRHARNDFSRWDAAQSLLATYIKLNVARHQQGQPLSLPVHVADAFRAVLLDEKIDPALAAEILTLPSVNEMAELFDIIDPIAIAEVREALTRTLATELADELLAIYNANYQSEYRVEHEDIAKRTLRNACLRFLAFGETHLADVLVSKQFHEANNMTDALAALSAAVAAQLPCRDALMQEYDDKWHQNGLVMDKWFILQATSPAANVLETVRGLLQHRSFTMSNPNRIRSLIGAFAGSNPAAFHAEDGSGYLFLVEMLTDLNSRNPQVASRLIEPLIRLKRYDAKRQEKMRAALEQLKGLENLSGDLYEKITKALA 5mfs A 1.57 BS02 7ML A 1 E121 M260 E264 H297 E298 H301 E320 Y376 Y381 E119 M258 E262 H295 E296 H299 E318 Y374 Y379 E264 H297 E298 H301 E320 N373 Y381 E262 H295 E296 H299 E318 N371 Y379 3.4.11.2 0004177,0005515,0005886,0006508,0008237,0008270,0042802,0046872 Ki=330nM remove_due_to_license_issue P04825 28383176 1002 QQPQAKYRHDYRAPDYQITDIDLTFDLDAQKTVVTAVSQAVRHGASDAPLRLNGEDLKLVSVHINDEPWTAWKEEEGALVISNLPERFTLKIINEISPAANTALEGLYQSGDALCTQCEAEGFRHITYYLDRPDVLARFTTKIIADKIKYPFLLSNGNRVAQGELENGRHWVQWQDPFPKPCYLFALVAGDFDVLRDTFTTRSGREVALELYVDRGNLDRAPWAMTSLKNSMKWDEERFGLEYDLDIYMIVAVDFFNMGAMENKGLNIFNSKYVLARTDTATDKDYLDIERVIGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSSDLGSRAVNRINNVRTMRGLQFAEDASPMAHPIRPDMVIEMNNFYTLTVYEKGAEVIRMIHTLLGEENFQKGMQLYFERHDGSAATCDDFVQAMEDASNVDLSHFRRWYSQSGTPIVTVKDDYNPETEQYTLTISQRTPATPDQAEKQPLHIPFAIELYDNEGKVIPLQKGGHPVNSVLNVTQAEQTFVFDNVYFQPVPALLCEFSAPVKLEYKWSDQQLTFLMRHARNDFSRWDAAQSLLATYIKLNVARHQQGQPLSLPVHVADAFRAVLLDEKIDPALAAEILTLPSVNEMAELFDIIDPIAIAEVREALTRTLATELADELLAIYNANYQSEYRVEHEDIAKRTLRNACLRFLAFGETHLADVLVSKQFHEANNMTDALAALSAAVAAQLPCRDALMQEYDDKWHQNGLVMDKWFILQATSPAANVLETVRGLLQHRSFTMSNPNRIRSLIGAFAGSNPAAFHAEDGSGYLFLVEMLTDLNSRNPQVASRLIEPLIRLKRYDAKRQEKMRAALEQLKGLENLSGDLYEKITKALA 5mft A 1.59 BS02 7MF A 1 E121 M260 E264 H297 E298 H301 E320 Y376 Y381 E119 M258 E262 H295 E296 H299 E318 Y374 Y379 E264 H297 E298 H301 E320 N373 Y381 E262 H295 E296 H299 E318 N371 Y379 3.4.11.2 0004177,0005515,0005886,0006508,0008237,0008270,0042802,0046872 Ki=34nM remove_due_to_license_issue P04825 28383176 1002 QQPQAKYRHDYRAPDYQITDIDLTFDLDAQKTVVTAVSQAVRHGASDAPLRLNGEDLKLVSVHINDEPWTAWKEEEGALVISNLPERFTLKIINEISPAANTALEGLYQSGDALCTQCEAEGFRHITYYLDRPDVLARFTTKIIADKIKYPFLLSNGNRVAQGELENGRHWVQWQDPFPKPCYLFALVAGDFDVLRDTFTTRSGREVALELYVDRGNLDRAPWAMTSLKNSMKWDEERFGLEYDLDIYMIVAVDFFNMGAMENKGLNIFNSKYVLARTDTATDKDYLDIERVIGHEYFHNWTGNRVTCRDWFQLSLKEGLTVFRDQEFSSDLGSRAVNRINNVRTMRGLQFAEDASPMAHPIRPDMVIEMNNFYTLTVYEKGAEVIRMIHTLLGEENFQKGMQLYFERHDGSAATCDDFVQAMEDASNVDLSHFRRWYSQSGTPIVTVKDDYNPETEQYTLTISQRTPATPDQAEKQPLHIPFAIELYDNEGKVIPLQKGGHPVNSVLNVTQAEQTFVFDNVYFQPVPALLCEFSAPVKLEYKWSDQQLTFLMRHARNDFSRWDAAQSLLATYIKLNVARHQQGQPLSLPVHVADAFRAVLLDEKIDPALAAEILTLPSVNEMAELFDIIDPIAIAEVREALTRTLATELADELLAIYNANYQSEYRVEHEDIAKRTLRNACLRFLAFGETHLADVLVSKQFHEANNMTDALAALSAAVAAQLPCRDALMQEYDDKWHQNGLVMDKWFILQATSPAANVLETVRGLLQHRSFTMSNPNRIRSLIGAFAGSNPAAFHAEDGSGYLFLVEMLTDLNSRNPQVASRLIEPLIRLKRYDAKRQEKMRAALEQLKGLENLSGDLYEKITKALA 5mg2 A 1.75 BS01 7M8 A 1 P1527 F1528 H1530 V1532 N1533 V1537 Y1582 N1583 Y1589 P29 F30 H32 V34 N35 V39 Y84 N85 Y91 2.3.1.48,2.7.11.1 0004402,0005669,0006366,0016251,0017025 Kd=17nM remove_due_to_license_issue IC50=13nM P21675 28402630 1704 SMDDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESLD 5mge A 1.95 BS01 7MX A 1 P1888 F1889 V1893 V1898 N1944 P33 F34 V38 V43 N89 ? Kd=87uM remove_due_to_license_issue Kd=87000nM Q9UIF8 28837921 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5mgf A 1.9 BS01 7MW A 1 F1889 V1893 N1944 I1950 F34 V38 N89 I95 ? Kd=54uM remove_due_to_license_issue Kd=54000nM Q9UIF8 28837921 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5mgg A 2.1 BS01 7MU A 1 P1888 F1889 V1893 N1944 I1950 P33 F34 V38 N89 I95 ? remove_due_to_license_issue Kd=>500000nM Q9UIF8 28837921 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5mgi A 1.5 BS01 6YV A 1 C69 S70 W105 S130 N132 E166 N170 T235 G236 T237 C43 S44 W79 S104 N106 E140 N144 T209 G210 T211 S70 K73 S130 E166 K234 T237 S44 K47 S104 E140 K208 T211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q848S6 29356380 301 TNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 5mgj A 2.1 BS01 7MX A 1 P1817 F1818 V1822 V1827 N1873 P22 F23 V27 V32 N78 ? Kd=51uM remove_due_to_license_issue Kd=51000nM Q9UIF9 28837921 1901 HSDLTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 5mgk A 2.301 BS01 7MW A 1 P1817 F1818 V1822 N1873 V1879 P22 F23 V27 N78 V84 ? Kd=100uM remove_due_to_license_issue Kd=100000nM Q9UIF9 28837921 1901 HSDLTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 5mgl A 2.651 BS01 7MU A 1 P1817 F1818 V1822 V1827 N1873 P19 F20 V24 V29 N75 ? remove_due_to_license_issue Kd=>500000nM Q9UIF9 28837921 1901 LTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 5mgm A 2.8 BS01 7MZ A 1 P1817 F1818 E1820 V1822 V1827 N1873 V1879 P19 F20 E22 V24 V29 N75 V81 ? remove_due_to_license_issue Kd=>500000nM Q9UIF9 28837921 1901 LTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 5mhk A 2.28 BS01 dna G 0 R307 D308 V311 S312 R480 R8 D9 V12 S13 R181 ? 0045893 remove_due_to_license_issue P08392 28505309 21 ~ 39 GAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk A 2.28 BS02 dna H 0 A304 R305 A5 R6 ? 0045893 remove_due_to_license_issue P08392 28505309 1 ~ 18 GAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk A 2.28 BS03 dna E 0 R415 S419 R460 R116 S120 R161 ? 0045893 remove_due_to_license_issue P08392 28505309 25 ~ 39 GAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk A 2.28 BS04 dna F 0 S418 R456 R457 S119 R157 R158 ? 0045893 remove_due_to_license_issue P08392 28505309 1 ~ 16 GAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk B 2.28 BS01 dna H 0 P476 R480 P188 R192 ? 0045893 remove_due_to_license_issue P08392 28505309 1 ~ 18 QPRRVELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk B 2.28 BS02 dna E 0 N393 N416 I421 R456 N107 N130 I133 R168 ? 0045893 remove_due_to_license_issue P08392 28505309 25 ~ 39 QPRRVELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk B 2.28 BS03 dna F 0 S419 M454 S455 R456 R457 S131 M166 S167 R168 R169 ? 0045893 remove_due_to_license_issue P08392 28505309 1 ~ 16 QPRRVELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk C 2.28 BS01 dna G 0 R395 R415 S417 S419 D459 R460 R104 R124 S126 S128 D168 R169 ? 0045893 remove_due_to_license_issue P08392 28505309 21 ~ 39 ELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAALT 5mhk C 2.28 BS02 dna H 0 N416 S418 R456 R457 N125 S127 R165 R166 ? 0045893 remove_due_to_license_issue P08392 28505309 1 ~ 18 ELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAALT 5mhk D 2.28 BS01 dna G 0 S417 I421 R456 S129 I133 R168 ? 0045893 remove_due_to_license_issue P08392 28505309 21 ~ 39 RRVELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhk D 2.28 BS02 dna H 0 M454 S455 R456 R457 M166 S167 R168 R169 ? 0045893 remove_due_to_license_issue P08392 28505309 1 ~ 18 RRVELDADATSGAFYARYRDGYVSGEPWPGAGPPPPGRVLYGGLGDSRPGLWGAPEAEEARRRFEASGAPAAVWAPELGDAAQQYALITRLLYTPDAEAMGWLQNPRVVPGDVALDQACFRISGAARNSSSFITGSVARAVPHLGYAMAAGRFGWGLAHAAAAVAMSRRYDRAQKGFLLTSLRRAYAPLLARENAAL 5mhp A 2.43 BS07 7NB A 1 F211 L214 H252 W255 W261 F274 F275 Y307 F153 L156 H194 W197 W203 F216 F217 Y249 3.1.4.39 0003676,0005044,0006955,0016787,0030247,0046872 Ki=15nM remove_due_to_license_issue IC50=300nM, Ki=15nM Q13822 28414242 920 WTNISGSCKGRCFELCRCDNLCKSYTSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLARGDCCTNYQVVCKGESHWVDDDCEEIKAAECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHSPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVKAGTFFWSVVIPHERRILTILQWLTLPDHERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKIVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRSKFSNNAKYDPKAIIANLTCKKPDQHFKPYLKQHLPKRLHYANNRRIEDIHLLVERRWHVARKPCFFQGDHGFDNKVNSMQTVFVGYGPTFKYKTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTFRPTMPEEVTRPNYPGIMYLQSDFDLGCTCTEERHLLYGRPAVLYRTRYDILYHTDFESGYSEIFLMPLWTSYTVSKQAEVSSVPDHLTSCVRPDVRVSPSFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWNYFQRVLVKKYASERNGVNVISGPIFDYDYDGLHDTEDKIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNEESCNSSEDESKWVEELMKMHTARVRDIEHLTSLDFFRKTSRSYPEILTLKTYLHTYE 5mhq A 1.3 BS01 8QT A 1 I10 G11 A31 K33 F80 L83 H84 Q85 Q131 N132 L134 D145 I13 G14 A34 K36 F74 L77 H78 Q79 Q125 N126 L128 D139 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T152 T159 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue IC50=30nM P24941 29063678 301 PEFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 5mi3 A 2.8 BS01 GDP A 1 D22 G24 K25 T26 T27 F47 N136 K137 D139 M140 S174 L176 D14 G16 K17 T18 T19 F39 N128 K129 D131 M132 S166 L168 ? 0003723,0003746,0003924,0005515,0005525,0005737,0005886,0006412,0006414,0032045,0046677,0097216 remove_due_to_license_issue P0CE47 29546243 402 TKPHVNVGTIGHVDHGKTTLTAAITTVLAKTYGGAARAFDQIDNAPEEKARGITINTSHVEYDTPTRHYAHVDCPGHADYVKNMITGAAQMDGAILVVAATDGPMPQTREHILLGRQVGVPYIIVFLNKCDMVDDEELLELVEMEVRELLSQYDFPGDDTPIVRGSALKALEGDAEWEAKILELAGFLDSYIPEPERAIDKPFLLPIEDVFSISGRGTVVTGRVERGIIKVGEEVEIVGIKETQKSTCTGVEMFRKLLDEGRAGENVGVLLRGIKREEIERGQVLAKPGTIKPHTKFESEVYILSKDEGGRHTPFFKGYRPQFYFRTTDVTGTIELPEGVEMVMPGDNIKMVVTLIHPIAMDDGLRFAIREGGRTVGAGVVAKVLG 5mi5 A 2.15 BS01 OAN A 1 G135 K166 D242 D243 Y282 W286 V314 N339 D344 G132 K163 D239 D240 Y279 W283 V311 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 29163914 801 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELESFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPCQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMKNLPLQVKANRVLISPAGNSEIELDAIYPGENIQINFLEISTDGKEWKTVDLKQKSRLSAGLQKAPVKFVRFTVSDRQFVLTIEK 5mi6 A 2.0 BS01 NHT A 1 G135 K166 D242 C278 Y282 W337 D344 G132 K163 D239 C275 Y279 W334 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 29163914 801 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELESFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPCQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMISNVKNLPLQVKANRVLISPANEVVKWAAGNSVEIELDAIYPGENIQINFEISTDGKEWKTVDLKQKERLSAGLQKAPVKFVRFTNVSQFVLTIEK 5mi7 A 2.1 BS01 OAN A 1 G135 K166 D242 D243 Y282 W286 V314 N339 D344 G132 K163 D239 D240 Y279 W283 V311 N336 D341 3.2.1.169 0005975,0006517,0015929,0016231,0016798,0042802,0102571,1901135 remove_due_to_license_issue Q89ZI2 29163914 801 SLQPPPQQLIVQNKTIDLPAVYQLNGGEEANPHAVKVLKELLSGKQSSKKGMLISIGEKGDKSVRKYSRQIPDHKEGYYLSVNEKEIVLAGNDERGTYYALQTFAQLLKDGKLPEVEIKDYPSVRYRGVVEGFYGTPWSHQARLSQLKFYGKNKMNTYIYGPKDDPYHSAPNWRLPYPDKEAAQLQELVAVANENEVDFVWAIHPGQDIKWNKEDRDLLLAKFEKMYQLGVRSFAVFFDDISGEGTNPQKQAELLNYIDEKFAQVKPDINQLVMCPTEYNKSWSNPNGNYLTTLGDKLNPSIQIMWTGDRVISDITRDGISWINERIKRPAYIWWNFPVSDYVRDHLLLGPVYGNDTTIAKEMSGFVTNPMEHAESSKIAIYSVASYAWNPAKYDTWQTWKDAIRTILPSAAEELESFAMHNSDLGPNGHGYRREESMDIQPAAERFLKAFKEGKNYDKADFETLQYTFERMKESADILLMNTENKPLIVEITPWVHQFKLTAEMGEEVLKMVEGRNESYFLRKYNHVKALQQQMFYIDQTSNQNPCQPGVKTATRVIKPLIDRTFATVVKFFNQKFNAHLDATTDYMPHKMIKNLPLQVKANRVLISPEIELDAIYPGENIQINFEISTDGKEWKTVDLKQKESRLSAGLQKAPVKFVRFTNQFVLTIEK 5mi9 A 3.3 BS01 GDP A 1 D22 G24 K25 T26 T27 F47 K137 S174 A175 L176 D14 G16 K17 T18 T19 F39 K129 S166 A167 L168 ? 0003723,0003746,0003924,0005515,0005525,0005737,0005886,0006412,0006414,0032045,0046677,0097216 remove_due_to_license_issue P0CE47 29546243 402 TKPHVNVGTIGHVDHGKTTLTAAITTVLAKTYGGAARAFDQIDNAPEEKARGIEINTSHVEYDTPTRHYAHVDCPGHADYVKNMITGAAQMDGAILVVAATDGPMPQTREHILLGRQVGVPYIIVFLNKCDMVDDEELLELVEMEVRELLSQYDFPGDDTPIVRGSALKALEGDAEWEAKILELAGFLDSYIPEPERAIDKPFLLPIEDVFSICGRGTVVTGRVERGIIKVGEEVEIVGIKETQKSTCTGVEMFRKLLDEGRAGENVGVLLRGIKREEIERGQVLAKPGTIKPHTKFESEVYILSKDEGGRHTPFFKGYRPQFYFRTTDVTGTIELPEGVEMVMPGDNIKMVVTLIHPIAMDDGLRFAIREGGRTVGAGVVAKVL 5mih A 1.8 BS02 7NU A 1 Y36 H50 Q53 D100 T104 N107 Y36 H50 Q53 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 ic50=64uM remove_due_to_license_issue Q05097 28960731 201 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 5mim A 1.9 BS04 1N A 1 R185 N192 D228 G229 E230 R77 N84 D120 G121 E122 D153 H194 D45 H86 3.4.21.75 0004252,0006508,0008236 Ki=0.046uM remove_due_to_license_issue P09958 28402100 609 VYQEPTDPKFPQQWYLSGVTQRDLNVKAAWAQGYTGHGIVVSILDDGIEKNHPDLAGNYDPGASFDVNDQDPDPQPRYTQMNDNRHGTRCAGEVAAVANNGVCGVGVAYNARIGGVRMLDGEVTDAVEARSLGLNPNHIHIYSASWGPEDDGKTVDGPARLAEEAFFRGVSQGRGGLGSIFVWASGNGGREHDSCNCDGYTNSIYTLSISSATQFGNVPWYSEACSSTLATTYSSGNQNEKQIVTTDLRQKCTESHTGTSASAPLAAGIIALTLEANKNLTWRDMQHLVVQTSKPAHLNANDWATNGVGRKVSHSYGYGLLDAGAMVALAQNWTTVAPQRKCIIDILTEPKDIGKRLEVRKTVTACLGEPNHITRLEHAQARLTLSYNRRGDLAIHLVSPMGTRSTLLAARPHDYSADGFNDWAFMTTHSWDEDPSGEWVLEIENTSEANNYGTLTKFTLVLYGTASGSLVPR 5mim A 1.9 BS05 1N A 2 D153 H194 L227 V231 E236 G255 D264 Y308 D45 H86 L119 V123 E128 G147 D156 Y200 D153 H194 D45 H86 3.4.21.75 0004252,0006508,0008236 Ki=0.046uM remove_due_to_license_issue P09958 28402100 610 VYQEPTDPKFPQQWYLSGVTQRDLNVKAAWAQGYTGHGIVVSILDDGIEKNHPDLAGNYDPGASFDVNDQDPDPQPRYTQMNDNRHGTRCAGEVAAVANNGVCGVGVAYNARIGGVRMLDGEVTDAVEARSLGLNPNHIHIYSASWGPEDDGKTVDGPARLAEEAFFRGVSQGRGGLGSIFVWASGNGGREHDSCNCDGYTNSIYTLSISSATQFGNVPWYSEACSSTLATTYSSGNQNEKQIVTTDLRQKCTESHTGTSASAPLAAGIIALTLEANKNLTWRDMQHLVVQTSKPAHLNANDWATNGVGRKVSHSYGYGLLDAGAMVALAQNWTTVAPQRKCIIDILTEPKDIGKRLEVRKTVTACLGEPNHITRLEHAQARLTLSYNRRGDLAIHLVSPMGTRSTLLAARPHDYSADGFNDWAFMTTHSWDEDPSGEWVLEIENTSEANNYGTLTKFTLVLYGTASGSLVPR 5mja A 2.14 BS01 7O3 A 1 I625 V633 A649 K651 E668 T697 M700 G703 L751 S761 D762 I17 V25 A41 K43 E60 T89 M92 G95 L143 S153 D154 D744 A746 R748 N749 D762 S781 D136 A138 R140 N141 D154 S167 2.7.10.1 0004672,0004713,0005524,0006468 ic50=220nM remove_due_to_license_issue P54762 28459525 901 EFAKEIDVSFVKIEEVIGAGEFGEVYKGRLKLPGKREIYVAIKTLKAGYSEKQRRDFLSEASIMGQFDHRNIIRLEGVVTKSRPVMIITEFMENGALDSFLRQNDGQFTVIQLVGMLRGIAAGMKYLSEMNYVHRDLAARNILVNSNLVCKVSDFGLSRYLPTYTSSPVRWTAPEAIAYRKFTSASDVWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPMDCPAALHQLMLDCWQKDRNSRPRFAEIVNTLDKMIRNPASLKTVA 5mjb A 2.23 BS01 7O3 A 1 I625 V633 A649 K651 E668 T697 M700 C703 L751 D762 I18 V26 A42 K44 E61 T90 M93 C96 L144 D155 D744 A746 R748 N749 D762 S781 K785 D137 A139 R141 N142 D155 S168 K172 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P54762 28459525 901 REFAKEIDVSFVKIEEVIGAGEFGEVYKGRLKLPGKREIYVAIKTLKAGYSEKQRRDFLSEASIMGQFDHRNIIRLEGVVTKSRPVMIITEFMENCALDSFLRQNDGQFTVIQLVGMLRGIAAGMKYLSEMNYVHRDLAARNILVNSNLVCKVSDFGLSRYLPTYTSSLGGKIPVRWTAPEAIAYRKFTSASDVWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPMDCPAALHQLMLDCWQKDRNSRPRFAEIVNTLDKMIRNPASLKTV 5mjn A 1.17 BS02 7O8 A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.9nM remove_due_to_license_issue Ki=2.9nM P00918 28024887 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5mkj A 2.5 BS02 4CU A 1 I268 N306 F313 R316 A327 F346 V349 C432 L436 I21 N59 F66 R69 A80 F99 V102 C185 L189 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue P19793 28691794 501 DMPVERILEAELAVEDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 5mkr A 1.87 BS01 TI8 A 1 T37 E268 K271 R272 S275 G339 R342 D366 S383 T384 R385 T37 E267 K270 R271 S274 G338 R341 D365 S382 T383 R384 D10 K71 E175 D199 D10 K71 E175 D198 ? 0005524,0140662 Ki=17uM remove_due_to_license_issue P0DMV8 28225177 401 MAKAAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILIKSTR 5mks A 1.99 BS01 TI8 A 1 E268 K271 R272 S275 G339 R342 E266 K269 R270 S273 G337 R340 D10 K71 E175 D199 D8 K69 E173 D197 ? 0005524,0140662 Ki=17uM remove_due_to_license_issue P0DMV8 28225177 401 KAAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILIKS 5mkx A 1.68 BS01 82I A 1 P747 F748 Y802 N803 Y809 P22 F23 Y77 N78 Y84 2.3.1.48,2.3.1.57 0004402 ic50=20uM remove_due_to_license_issue IC50=19953nM Q92831 28002667 901 DQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 5mky A 1.67 BS01 I0D A 1 F44 F45 V49 Y99 N100 Y106 F23 F24 V28 Y78 N79 Y85 ? ic50=2uM remove_due_to_license_issue IC50=1995nM Q9H8M2 28002667 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 5mky A 1.67 BS02 I0D A 2 L28 F32 M121 L7 F11 M100 ? ic50=2uM remove_due_to_license_issue IC50=1995nM Q9H8M2 28002667 202 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMS 5mkz A 1.62 BS01 RNK A 1 W81 V87 L92 Y139 N140 I146 W40 V46 L51 Y98 N99 I105 ? ic50=20uM remove_due_to_license_issue O60885 28002667 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ml0 A 1.64 BS01 P2L A 1 P746 F747 E755 Y759 Y801 N802 Y808 P23 F24 E32 Y36 Y78 N79 Y85 2.3.1.48,2.3.1.57 0004402 remove_due_to_license_issue Q9JHD1 28002667 901 PEQLYSTLKNILQQVKNHPNAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLRNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCASILEKFFFSKIKEAGLIDK 5ml2 B 1.6 BS01 NH6 B 1 M20 L22 W32 I53 R61 Q78 V80 W90 M117 I129 T131 F133 L147 Y149 M19 L21 W31 I52 R60 Q77 V79 W89 M111 I123 T125 F127 L141 Y143 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=13nM remove_due_to_license_issue Kd=65nM O43924 28106325 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5ml3 B 1.4 BS01 DL3 B 1 M20 L22 W32 I53 C56 R61 Q78 W90 I109 M117 I129 T131 F133 L147 Y149 M19 L21 W31 I52 C55 R60 Q77 W89 I108 M116 I128 T130 F132 L146 Y148 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=203pM remove_due_to_license_issue Kd=203nM O43924 28106325 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAAPESQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5ml4 B 2.4 BS01 RRQ B 1 M20 L22 W32 I53 L54 C56 R61 Q78 E88 W90 M117 L123 I129 T131 L147 Y149 M19 L21 W31 I52 L53 C55 R60 Q77 E87 W89 M116 L122 I128 T130 L146 Y148 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd<2nM remove_due_to_license_issue O43924 28106325 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAAPESQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5ml5 A 1.9 BS01 1VI A 1 Y35 A51 K53 L104 V105 T106 M109 F169 Y29 A45 K47 L98 V99 T100 M103 F163 D150 K152 N155 D168 T185 D144 K146 N149 D162 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=10nM remove_due_to_license_issue Q16539 28338621 404 RPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 5ml6 B 1.87 BS01 9GD B 1 M20 L22 W32 I53 L54 C56 R61 Q78 L87 W90 M117 I129 T131 F133 Y149 M19 L21 W31 I52 L53 C55 R60 Q77 L86 W89 M112 I124 T126 F128 Y144 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=358pM remove_due_to_license_issue O43924 28106325 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIESQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5ml8 B 2.6 BS01 V98 B 1 M20 L22 W32 I53 C56 R61 Q78 E88 W90 M117 I129 T131 L147 Y149 M19 L21 W31 I52 C55 R60 Q77 E87 W89 M110 I122 T124 L140 Y142 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 remove_due_to_license_issue Kd=16nM O43924 28106325 201 SAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5mli A 1.63 BS01 82I A 1 P82 F83 V87 L92 Y139 N140 P41 F42 V46 L51 Y98 N99 ? ic50=130uM remove_due_to_license_issue IC50=125893nM O60885 28002667 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5mlj A 1.8 BS01 9ST A 1 W751 P752 F753 V757 E761 Y807 N808 Y814 W23 P24 F25 V29 E33 Y79 N80 Y86 2.3.1.-,2.3.1.48 0004402 Ki=1.4nM remove_due_to_license_issue Ki=1.3nM Q92830 28002667 902 DPDQLYTTLKNLLAQIKSHPSAWPFMEPVKKSEAPDYYEVIRFPIDLKTMTERLRSRYYVTRKLFVADLQRVIANCREYNPPDSEYCRCASALEKFFYFKLKEGGLIDK 5mm9 A 1.55 BS03 8SH A 1 F61 Y67 W87 H118 D120 H196 R228 N233 H263 F31 Y36 W56 H85 D87 H148 R174 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=0.38uM remove_due_to_license_issue B5KVR9 28445786 404 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5mme A 1.35 BS01 8Q6 A 1 L1109 P1110 Q1113 V1115 L1120 N1168 V1174 L31 P32 Q35 V37 L42 N90 V96 2.3.1.-,2.3.1.48 Kd=1.4uM remove_due_to_license_issue Kd=1400nM Q92793 30258543 1201 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5mmg A 1.23 BS01 UT0 A 1 L1109 P1110 V1115 L1120 N1168 R1173 V1174 L27 P28 V33 L38 N86 R91 V92 2.3.1.-,2.3.1.48 Kd=0.97uM remove_due_to_license_issue Q92793 30258543 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5mmn A 1.9 BS01 O54 A 1 V43 N46 E50 V71 D73 I78 P79 I94 V37 N40 E44 V65 D67 I72 P73 I88 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.125uM remove_due_to_license_issue P0AES7 28406299 301 SSSIKVLKGLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLNSYKVSGGLHGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 5mmp A 2.05 BS01 G3Z A 1 N46 E50 V71 D73 R76 G77 I78 P79 I94 T165 N37 E41 V62 D64 R67 G68 I69 P70 I85 T137 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.03uM remove_due_to_license_issue P0AES7 28406299 301 IKVLKGLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 5mn1 A 0.79 BS02 2AP A 1 S190 C191 Q192 W215 G219 S172 C173 Q174 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=3.3mM remove_due_to_license_issue P00760 28371253 306 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mnb A 0.939 BS02 2AP A 1 S190 C191 G219 S172 C173 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=3.3mM remove_due_to_license_issue P00760 28371253 304 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mnc A 0.916 BS02 ANL A 1 S190 Q192 S172 Q174 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 28371253 307 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mnn A 0.859 BS02 MRZ A 1 D189 S190 C191 S195 V213 W215 G216 G219 D171 S172 C173 S177 V191 W193 G194 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue Ki=360nM P00760 30177695 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mno A 0.96 BS02 MRZ A 1 D189 S190 C191 W215 G219 D171 S172 C173 W193 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=143uM remove_due_to_license_issue Ki=360nM P00760 30177695 304 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mnr E 1.249 BS06 JC2 E 1 N111 N112 A113 F114 H142 E143 H146 Y157 E166 L202 R203 H231 N111 N112 A113 F114 H142 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 409 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5mnx A 1.42 BS02 2AP A 1 D189 S190 G219 D171 S172 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 28371253 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mny A 1.43 BS02 WOT A 1 D189 S190 D171 S172 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 28371253 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mo2 A 1.5 BS02 D86 A 1 D189 S190 C191 W215 G219 G226 D171 S172 C173 W193 G196 G204 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 30177695 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mo8 A 1.82 BS01 C98 A 1 V66 K68 F113 N118 F121 P159 H160 V162 M163 I164 I174 D175 M225 V63 K65 F110 N115 F118 P156 H157 V159 M160 I161 I171 D172 M222 D156 K158 N161 D175 P184 S194 D153 K155 N158 D172 P181 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=1.64uM remove_due_to_license_issue P68400 28495381 404 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5mob A 1.669 BS01 A8S A 1 K96 V120 F145 Y157 F196 V200 K69 V93 F118 Y130 F169 V173 Kd=90uM remove_due_to_license_issue 28736053 301 LSTITTHHLTVPPGLTPEEFQELSSSIAEFHSYRINPGQCSSLLAQRIHAPVETVWTVVRRFDKPQTYKHFIKSCSVGEDFRMTVGSTRDVTVISGLPAATSTERLDILDDDRHVTGFSIIGGEHRLRNYRSVTTVHGFERDGEIWTVVLESYVVDVPEGNTEEDTRLFADTVVKLNLQKLASVTETLAREAG 5mod A 2.08 BS01 86L A 1 N118 F121 P159 V162 I164 M225 N117 F120 P158 V161 I163 M224 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=300uM remove_due_to_license_issue IC50=3000000nM P68400 28495381 404 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVV 5moe A 1.89 BS04 OQC A 1 W24 H183 Q186 W22 H181 Q184 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Kd=520uM remove_due_to_license_issue P68400 28495381 409 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5moe A 1.89 BS05 OQC A 2 P159 V162 I164 M225 P157 V160 I162 M223 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Kd=520uM remove_due_to_license_issue P68400 28495381 410 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5moe A 1.89 BS06 OQC A 3 Q36 Y39 D103 A110 Q34 Y37 D101 A108 D156 K158 N161 D175 P184 S194 D154 K156 N159 D173 P182 S192 2.7.11.1 0004672,0004674,0005524,0006468 Kd=520uM remove_due_to_license_issue P68400 28495381 411 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5mon A 0.939 BS02 2AP A 1 D189 S190 C191 G219 D171 S172 C173 G196 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=3.3mM remove_due_to_license_issue P00760 28371253 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5moo A 1.441 BS02 WOT A 1 D189 S190 D171 S172 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Kd=48.5mM remove_due_to_license_issue P00760 28371253 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mos A 0.96 BS02 D86 A 1 D189 S190 C191 W215 G219 G226 D171 S172 C173 W193 G196 G204 H57 D102 Q192 G193 D194 S195 G196 H40 D84 Q174 G175 D176 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 30177695 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 5mpf A 2.918 BS01 dna E 0 T380 K389 F420 C421 R427 T118 K127 F153 C154 R160 ? 0003700,0006357 remove_due_to_license_issue Q9NZI5 29309642 1 ~ 12 NNFEYTLEASKSLRGDSTMTYLNKGQFYPITLKEVSKVRSVIMVVFAEDKSREDQLRHWKYWHSRQHTAKQRCIDIADYKESFNTISNVEEIAYNAISFTWDINDEAKVFISVNCLSTDFSSQKGVKGLPLNIQIDTYNNKPVHRAYCQIKVFCDKGAERKIRDEERKQSKRMDITVFKPFIDLDTQPVLFIPDVH 5mpf A 2.918 BS02 dna F 0 Q385 K386 G387 R430 Q123 K124 G125 R163 ? 0003700,0006357 remove_due_to_license_issue Q9NZI5 29309642 1 ~ 12 NNFEYTLEASKSLRGDSTMTYLNKGQFYPITLKEVSKVRSVIMVVFAEDKSREDQLRHWKYWHSRQHTAKQRCIDIADYKESFNTISNVEEIAYNAISFTWDINDEAKVFISVNCLSTDFSSQKGVKGLPLNIQIDTYNNKPVHRAYCQIKVFCDKGAERKIRDEERKQSKRMDITVFKPFIDLDTQPVLFIPDVH 5mpf B 2.918 BS01 dna E 0 Q385 K386 G387 V388 R430 Q124 K125 G126 V127 R169 ? 0003700,0006357 remove_due_to_license_issue Q9NZI5 29309642 1 ~ 12 NNFEYTLEASKSLRQKSTMTYLNKGQFYPITLKEVSSKVRSVIMVVFAEDKSREDQLRHWKYWHSRQHTAKQRCIDIADYKESFNTISNVEEIAYNAISFTWDINDEAKVFISVNCLSTDFSSQKGVKGLPLNIQIDTYSYNNRSNKPVHRAYCQIKVFCDKGAERKIRDEERKQSKRKMDITVFKPFIDLDTQPVLFIPDV 5mpf B 2.918 BS02 dna F 0 T380 C421 R427 K428 T119 C160 R166 K167 ? 0003700,0006357 remove_due_to_license_issue Q9NZI5 29309642 1 ~ 12 NNFEYTLEASKSLRQKSTMTYLNKGQFYPITLKEVSSKVRSVIMVVFAEDKSREDQLRHWKYWHSRQHTAKQRCIDIADYKESFNTISNVEEIAYNAISFTWDINDEAKVFISVNCLSTDFSSQKGVKGLPLNIQIDTYSYNNRSNKPVHRAYCQIKVFCDKGAERKIRDEERKQSKRKMDITVFKPFIDLDTQPVLFIPDV 5mpg A -1.00 BS01 rna B 0 A1 S2 K15 F17 G19 G20 L21 F23 D42 V44 M46 R55 G56 F57 F59 R82 E85 K87 A89 V90 R92 S95 R97 A1 S2 K15 F17 G19 G20 L21 F23 D42 V44 M46 R55 G56 F57 F59 R82 E85 K87 A89 V90 R92 S95 R97 ? 0003676,0003723 remove_due_to_license_issue P09651 28650318 1 ~ 7 ASKSESPKEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQR 5mpk A 1.9 BS01 0BC A 1 L1109 P1110 Q1113 V1115 L1120 N1168 R1173 V1174 L26 P27 Q30 V32 L37 N85 R90 V91 2.3.1.-,2.3.1.48 Kd=0.003uM remove_due_to_license_issue IC50=15nM, Kd=3.0nM Q92793 30258543 1201 IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQS 5mpl A -1.00 BS01 rna B 0 K106 F108 G110 G111 I112 M137 R140 R146 G147 F148 F150 E176 R178 A180 L181 S182 K183 Q184 M186 A187 K12 F14 G16 G17 I18 M43 R46 R52 G53 F54 F56 E82 R84 A86 L87 S88 K89 Q90 M92 A93 ? 0003676,0003723 remove_due_to_license_issue P09651 28650318 1 ~ 6 SQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMASASSSQRGR 5mpn A 1.23 BS01 YE5 A 1 P1110 V1115 N1168 R1173 V1174 P32 V37 N90 R95 V96 2.3.1.-,2.3.1.48 Kd=0.085uM remove_due_to_license_issue Kd=85nM, IC50=59nM Q92793 30258543 1201 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5mpn A 1.23 BS02 YE5 A 2 M1095 E1099 Y1102 M17 E21 Y24 2.3.1.-,2.3.1.48 Kd=0.085uM remove_due_to_license_issue Kd=85nM, IC50=59nM Q92793 30258543 1202 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5mpz A 1.4 BS01 4I8 A 1 P1110 F1111 V1115 N1168 V1174 P27 F28 V32 N85 V91 2.3.1.-,2.3.1.48 Kd=85uM remove_due_to_license_issue IC50=455000nM, Kd=85000nM Q92793 28410781 1201 IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVM 5mqe A 1.65 BS01 PKU A 1 V1115 L1120 N1168 V1174 V33 L38 N86 V92 2.3.1.-,2.3.1.48 Kd=4uM remove_due_to_license_issue Kd=4000nM, IC50=40000nM Q92793 28410781 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5mql A 3.25 BS02 G65 A 1 V55 M85 Y86 P89 E90 F96 Q97 F137 S144 E145 V37 M56 Y57 P60 E61 F67 Q68 F108 S115 E116 E53 R128 E35 R99 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 remove_due_to_license_issue P27707 29127277 302 TRIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNTMSQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESECMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 5mqt A 3.2 BS02 STI A 1 V55 M85 Y86 P89 Q97 F137 V36 M55 Y56 P59 Q67 F107 E53 R128 E34 R98 2.7.1.113,2.7.1.74,2.7.1.76 0004136,0004137,0004138,0005515,0005524,0005634,0005654,0005737,0005739,0005829,0006139,0006220,0008144,0009224,0016301,0019136,0042803,0043771,0106383,1901135,1901293 remove_due_to_license_issue P27707 29127277 302 RIKKISIEGNIAAGKSTFVNILKQLSEDWEVVPEPVARWSNTMSQKNGGNVLQMMYEKPERWSFTFQTYACLSRIRAQLASLNGKLKDAEKPVLFFERSVYSDRYIFASNLYESECMNETEWTIYQDWHDWMNNQFGQSLELDGIIYLQATPETCLHRIYLRGRNEEQGIPLEYLEKLHYKHESWLLHRTLKTNFDYLQEVPILTLDVNEDFKDKYESLVEKVKEFLSTL 5mqv A 2.154 BS01 D5Q A 1 I15 I23 A36 M80 M82 L85 P87 L135 L138 I148 I8 I16 A29 M73 M75 L78 P80 L128 L131 I141 D128 K130 D121 K123 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=8nM remove_due_to_license_issue P48730 28338621 301 RYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 5mqx A -1.00 BS01 APR A 1 D10 I11 G30 G31 G32 V33 C34 I113 F114 R144 W148 D10 I11 G30 G31 G32 V33 C34 I113 F114 R144 W148 2.1.1.-,2.7.7.-,2.7.7.19,2.7.7.48,3.1.3.84,3.4.22.-,3.6.1.15,3.6.1.74,3.6.4.13 remove_due_to_license_issue P36328 30825649 201 APSYHVVRGDIATATEGVIINAANSKGQPGGGVCGALYKKFPESFDLQPIEVGKARLVKGAAKHIIHAVGPNFNKVSEVEGDKQLAEAYESIAKIVNDNNYKSVAIPLLSTGIFSGNKDRLTQSLNHLLTALDTTDADVAIYCRDKKWEMTLKEAVARRE 5mqy A 1.13 BS01 GH4 A 1 G23 C25 G61 E63 N66 G67 G68 L69 A135 D162 H163 G23 C25 G61 E63 N66 G67 G68 L69 A135 D162 H163 Q19 C25 H163 N187 Q19 C25 H163 N183 3.4.22.15 0006508,0008234 remove_due_to_license_issue P07711 28287264 301 APRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV 5mra B 3.74 BS02 DM2 B 1 F134 R174 Q181 G182 F103 R143 Q150 G151 F95 G118 V120 F64 G87 V89 ? 0005509 remove_due_to_license_issue P30626 28726784 204 MDPLYGYFAAVAGQDGQIDADELQRCLTQSGIAGGYKPFNLETCRLMVSMLDRDMSGTMGFNEFKELWAVLNGWRQHFISFDTDRSGTVDPQELQKALTTMGFRLSPQAVNSIAKRYSTNGKITFDDYIACCVKLRALTDSFRRRDTAQQGVVNFPYDDFIQCVMSV 5mrb A 2.2 BS01 C5N A 1 I531 S533 A551 K553 Y604 G605 D608 S611 L654 I663 I18 S20 A38 K40 Y91 G92 D95 S98 L141 I150 D647 K649 N652 D664 T686 D134 K136 N139 D151 T168 2.7.12.1 0004672,0005524,0006468 Kd=471nM remove_due_to_license_issue P33981 28726638 901 YFQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEYGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTTSQVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 5mrd A 1.41 BS01 S26 A 1 K115 N119 Q128 K131 L155 F157 K40 N44 Q53 K56 L80 F82 D205 K207 E209 N210 D223 T245 D130 K132 E134 N135 D148 T170 2.7.11.1 0004672,0004674,0005524,0006468 ic50=36.4uM remove_due_to_license_issue O15530 28045490 401 SKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKIVEKRHVNKENKIPYVQREKDVMSRLDHPFFVKLYFCFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 5mrh A 2.5 BS01 Q9Z A 1 F281 S283 R292 F317 Y318 F217 S219 R228 F253 Y254 ? 0016020 ic50=0.0000631M remove_due_to_license_issue IC50=63096nM Q99523 28462834 805 RVRDFVAKLANNTHQHVFGSVSLSWVGDSTGVILVLTTFHVPGQSKLYRSEDYGKNFKDITDLINNTFIRTEFGMAIGPENSGKVVLTAEVSGGSRGGRIFRSSDFAKNFVQTDLPFHPLTQMMYSPQNSDYLLALSTENGLWVSKNFGGKWEEIHKAVCLAKWGSDNTIFFTTYANGSCKADLGALELWRTSDLGKSFKTIGVKIYSFGLGGRFLFASVMADKDTTRRIHVSTDQGDTWSMAQLPSVGQEQFYSILAANDDMVFMHVDEPGDTGFGTIFTSDDRGIVYSKSLDRHLYTTTGGETDFTNVTSLRGVYITSVLSEDNSIQTMITFDQGGRWTHLRKPENSECDATAKNKNECSLHIHASYSISQKLNVPMAPLSEPNAVGIVIAHGSVGDAISVMVPDVYISDDGGYSWTKMLEGPHYYTILDSGGIIVAIEHSSRPINVIKFSTDEGQCWQTYTFTRDPIYFTGLASEPGARSMNISIWGFTWVSYTIDFKDILERNCEEKDYTIWLAHSTDPEDYEDGCILGYKEQFLRLRKSSMCQNGRDYVVTKQPSICLCSLEDFLCDFGYYRPENDSKCVEQPELKGHDLEFCLHLTTNGYRKIPGDKCQGGVNPVREVKDLKKKCTSNFLSPE 5mri A 2.0 BS01 Q9Y A 1 S283 R292 F317 Y318 S230 R239 F264 Y265 ? 0016020 remove_due_to_license_issue Q99523 28462834 807 GRVRDFVAKLANNTHQHVFDDLRGSVSLSWVGDSTGVILVLTTFHVPLVIMTFGQSKLYRSEDYGKNFKDITDLINNTFIRTEFGMAIGPENSGKVVLTAEVSGGSRGGRIFRSSDFAKNFVQTDLPFHPLTQMMYSPQNSDYLLALSTENGLWVSKNFGGKWEEIHKAVCLAKWGSDNTIFFTTYANGSCKADLGALELWRTSDLGKSFKTIGVKIYSFGLGGRFLFASVMADKDTTRRIHVSTDQGDTWSMAQLPSVGQEQFYSILAANDDMVFMHVDEPGDTGFGTIFTSDDRGIVYSKSLDRHLYTTTGGETDFTNVTSLRGVYITSVLSEDNSIQTMITFDQGGRWTHLRKPENSECDATAKNKNECSLHIHASYSISQKLNVPMAPLSEPNAVGIVIAHGSVGDAISVMVPDVYISDDGGYSWTKMLEGPHYYTILDSGGIIVAIEHSSRPINVIKFSTDEGQCWQTYTFTRDPIYFTGLASEPGARSMNISIWGFTESFLTSQWVSYTIDFKDILERNCEEKDYTIWLAHSTDPEDYEDGCILGYKEQFLRLRKSSMCQNGRDYVVTKQPSICLCSLEDFLCDFGYYRPENDSKCVEQPELKGHDLEFCLYGREEHLTTNGYRKIPGDKCQGGVNPVREVKDLKKKCTSNFLSPE 5mrm A 1.8 BS01 Q9T A 1 Q158 V161 I177 A203 Q238 V239 L245 S264 V266 Q73 V76 I92 A118 Q150 V151 L157 S176 V178 2.7.7.60 0003824,0008299,0050518,0070567 ic50=9.3uM remove_due_to_license_issue P69834 28686408 401 MEKSVSVILLAPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTKTLWEMQTPQVIKPELLKKGFELVKSEGLEVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILS 5mro A 1.8 BS01 Q9P A 1 R157 I177 A203 Q238 V239 I240 D262 V263 I265 V266 V273 R73 I93 A119 Q154 V155 I156 D178 V179 I181 V182 V189 2.7.7.60 0003824,0008299,0050518,0070567 ic50=2uM remove_due_to_license_issue IC50=140nM P69834 28686408 401 EKSVSVILLAGMPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLDRKTLWEMQTPQVIKPELLKKGFELVKSEGLAVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILS 5mrp A 1.9 BS01 6BC A 1 R157 Q158 I177 A203 Q238 V239 D262 V263 I265 V266 V273 R72 Q73 I92 A118 Q148 V149 D172 V173 I175 V176 V183 2.7.7.60 0003824,0008299,0050518,0070567 ic50=3uM remove_due_to_license_issue IC50=35nM P69834 28686408 401 EKSVSVILLAGPKQYIPLLGQPIALYSFFTFSRMPEVKEIVVVCDPFFRDIFEEYEESIDVDLSFAIPGKERQDSVYSGLQEIDVNSELVCIHDSARPLVNTEDVEKVLKDGSAVGAAVLGVPAKATIKEVNSDSLVVKTLWEMQTPQVIKPELLKKGFELVKSEGLAVTDDVSIVEYLKHPVYVSQGSYTNIKVTTPDDLLLAERILS 5msb A 1.3 BS02 V13 A 1 H91 H117 V119 V141 L197 T198 T199 W208 H89 H115 V117 V139 L195 T196 T197 W206 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=35nM remove_due_to_license_issue Kd=250nM O43570 29503769 303 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 5mt0 A 1.29 BS01 QJS A 1 H40 L41 H57 I143 R151 K192 G193 S195 H24 L25 H41 I130 R137 K180 G181 S183 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd~500uM remove_due_to_license_issue Ki=500000nM, Kd=500000nM P00746 28157311 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 5mt4 A 1.65 BS01 M7O A 1 H40 L41 H57 R151 K192 G193 S195 S215 H24 L25 H41 R137 K180 G181 S183 S199 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd~500uM remove_due_to_license_issue P00746 28157311 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 5mte A 1.4 BS01 BB2 A 1 G40 I41 G42 Q47 P82 E83 G84 C85 L86 H127 E128 H131 G40 I41 G42 Q47 P82 E83 G84 C85 L86 H127 E128 H131 G42 Q47 C85 L86 H127 E128 H131 G42 Q47 C85 L86 H127 E128 H131 ? 0042586,0043686,0046872 remove_due_to_license_issue Q6VT21 29101077 201 MKILKDDAPELHAIAAEVPHGEDVKDLVLDMTAAMTAAGGIGLAGNQVGVLKRIIVLRCPTFKGCVINPIITRHTDGHVYSPEGCLSYPGKTVAKKRRNKVVVEGYDMDWQPITIAAKGLTAFCLQHEIDHLNGVTI 5mts A 2.6 BS01 XKA A 1 F1 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 N46 D47 Y48 I52 D54 Q133 N135 D140 ? 0007155,0009289 remove_due_to_license_issue P08191 28257558 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 5mtv A 2.79 BS01 AGS A 1 S71 G73 K74 T75 T76 P93 D98 D156 K223 W261 S53 G55 K56 T57 T58 P75 D80 D138 K199 W237 ? 0005509,0005515,0005524,0005525,0005737,0005768,0005783,0005886,0006907,0030100,0031901,0032456,0046872,0048471,0050731,0051260,0055038,0071363 remove_due_to_license_issue Q9EQP2 28228524 1000 GGSQTVTGGLRSLYQRKVLPLEEAYRFHEFHSPALEDADFENKPMILLVGQYSTGKTTFIRYLLEQDFPGMRIGPEPTTDSFIAVMYGETEGSTPGNALVVDPKKPFRKLSRFGNAFLNRFMCSQLPNQVLKSISIIDSPGILISRGYDFCQVLQWFAERVDRIILLFDAHKLDISDEFSEAIKAFRGQDDKIRVVLNKADQVDTQQLMRVYGALMWSLGKVINTPEVLRVYIGSFWAQPLQNTDNRRLFEAEAQDLFRDIQSLPQKAAVRKLNDLIKRARLAKVHAYIISYLKKEMPNMFGKENKKRELIYRLPEIYVQLQREYQISAGDFPEVKAMQEQLENYDFTKFHSLKPKLIEAVDNMLTNKISSLMGLISQE 5mtx A 1.8 BS01 FJI A 1 V30 A51 K53 E71 L75 L104 L108 M109 G110 A111 L167 D168 F169 V26 A45 K47 E65 L69 L98 L102 M103 G104 A105 L161 D162 F163 D150 K152 N155 D168 T185 D144 K146 N149 D162 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=17.7nM remove_due_to_license_issue IC50=1.000000nM, Kd=3.1nM Q16539 28834431 401 RPTFYRQELNKTIWEVPERYQNLSPVGSYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 5mty A 2.31 BS01 HB9 A 1 V38 A51 K53 E71 L108 M109 G110 A111 L167 D168 F169 V28 A41 K43 E61 L98 M99 G100 A101 L157 D158 F159 D150 K152 N155 D168 T185 D140 K142 N145 D158 T161 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=1.3nM remove_due_to_license_issue IC50=0.600000nM, Kd=7.5nM Q16539 28834431 401 RPTFYRQELNKTIWEVPERYQNLSPVSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 5muc A 2.6 BS01 AH2 A 1 F1 I13 N46 D47 D54 Q133 N135 D140 F1 I13 N46 D47 D54 Q133 N135 D140 ? 0007155,0009289 remove_due_to_license_issue P08191 29939458 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 5mw2 A 2.35 BS01 U52 A 1 M51 A52 C53 G55 Y58 F89 Q113 M114 E115 H116 V117 M45 A46 C47 G49 Y52 F83 Q107 M108 E109 H110 V111 ? ic50<3nM remove_due_to_license_issue P41182 28930682 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 5mw4 A 2.19 BS01 5JU A 1 S140 L143 M147 D161 G163 S164 G165 V169 E186 K187 D222 F223 F239 V240 N241 S268 S269 S117 L120 M124 D138 G140 S141 G142 V146 E163 K164 D199 F200 F216 V217 N218 S245 S246 2.1.1.360 0031151,0051726 Ki=0.002nM remove_due_to_license_issue Q8TEK3 28337327 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEKGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKN 5mw6 A 1.65 BS01 RC0 A 1 N21 R24 L25 N16 R19 L20 ? ic50=18648nM remove_due_to_license_issue P41182 28930682 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKA 5mw6 A 1.65 BS02 RC0 A 2 M51 A52 S54 G55 Y58 M46 A47 S49 G50 Y53 ? ic50=18648nM remove_due_to_license_issue P41182 28930682 202 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKA 5mw6 B 1.65 BS01 RC0 A 1 M51 A52 S54 G55 Y58 M43 A44 S46 G47 Y50 ? remove_due_to_license_issue P41182 28930682 201 IQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKA 5mw6 B 1.65 BS02 RC0 A 2 N21 R24 L25 R28 N13 R16 L17 R20 ? remove_due_to_license_issue P41182 28930682 202 IQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKA 5mwd A 1.85 BS01 TJ3 A 1 M51 A52 G55 Y58 Q113 M114 E115 M45 A46 G49 Y52 Q107 M108 E109 ? ic50=632nM remove_due_to_license_issue P41182 28930682 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 5mwg A 1.5 BS01 WGX A 1 F653 V657 P658 E661 Y707 N708 F714 F24 V28 P29 E32 Y78 N79 F85 ? ic50=1.7uM remove_due_to_license_issue IC50=1700nM P55201 29902720 801 LTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5mwh A 1.65 BS01 UWX A 1 I652 F653 V657 P658 N708 F714 I25 F26 V30 P31 N81 F87 ? Kd=1.8uM remove_due_to_license_issue Kd=2700nM, IC50=1900nM P55201 29902720 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5mwj A 2.04 BS01 EBU A 1 C488 Y532 R534 E550 A576 Y578 L636 F661 L743 C51 Y90 R92 E108 A130 Y132 L190 F215 L297 ? 0005634,0006355 Kd=24.7nM remove_due_to_license_issue Q04724 28326635 802 YFQGAMGSKPAYSFHVTQMQPVPFPPDALIGPGIPRHARQINTLNHGEVVCAVTISNPTRHVYTGGKGCVKVWDISSPVSQLDCLNRDNYIRSCKLLPDGCTLIVGGEASTLSIWDLPRIKAELTSSAPACYALAISPDSKVCFSCCSDGNIAVWDLHNQTLVRQFQGHTDGASCIDISNDGTKLWTGGLDNTVRSWDLREGRQLQQHDFTSQIFSLGYCPTGEWLAVGMESSNVEVLHVNKPDKYQLHLHESCVLSLKFAYCGKWFVSTGKDNLLNAWRTPYGASIFQSKESSSVLSCDISVDDKYIVTGSGDKKATVYEVIY 5mwo A 1.962 BS01 J6W A 1 M102 W103 G106 I107 F110 Y148 T149 W207 M81 W82 G85 I86 F89 Y127 T128 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.19mM remove_due_to_license_issue P9WMC1 28513917 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5mwo A 1.962 BS02 J6W A 2 F110 W138 M142 W145 N179 E180 F89 W117 M121 W124 N158 E159 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.19mM remove_due_to_license_issue P9WMC1 28513917 302 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5mwp A 1.82 BS02 ECV A 1 N770 L772 A773 Q776 M807 S810 S811 L814 F829 M845 M852 L938 F941 C942 T945 N36 L38 A39 Q42 M73 S76 S77 L80 F95 M111 M118 L197 F200 C201 T204 ? Ki=31.6nM remove_due_to_license_issue IC50=<10000nM, Ki=40nM, EC50=13nM P08235 29474466 1101 YFSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLSSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 5mwy A 1.75 BS02 YNU A 1 L766 L769 N770 Q776 W806 M807 S810 L814 F829 M845 M852 L938 F941 C942 T945 F956 L32 L35 N36 Q42 W72 M73 S76 L80 F95 M111 M118 L198 F201 C202 T205 F216 ? Ki=100nM remove_due_to_license_issue IC50=122nM, EC50=100nM, Ki=126nM P08235 29474466 1101 YFSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLSSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 5mwz A 1.25 BS01 KGU A 1 I652 F653 V657 P658 C704 Y707 N708 F714 I27 F28 V32 P33 C79 Y82 N83 F89 ? Kd=7.1uM remove_due_to_license_issue P55201 29902720 801 MEMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5mxf A 1.9 BS01 MFU A 1 G315 V316 G337 T338 W343 G292 V293 G314 T315 W320 ? 0046872 Kd=0.26mM remove_due_to_license_issue C7BLE4 28806750 401 MSTIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 5mxf A 1.9 BS02 MFU A 2 G171 V172 G193 T194 W199 G148 V149 G170 T171 W176 ? 0046872 Kd=0.26mM remove_due_to_license_issue C7BLE4 28806750 402 MSTIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 5mxk A 1.932 BS01 ZHA A 1 W103 G106 I107 F110 Y148 T149 N176 N179 W207 W82 G85 I86 F89 Y127 T128 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=150uM remove_due_to_license_issue P9WMC1 28513917 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5mxq A 2.0 BS03 U8K A 1 F62 Y67 W87 D118 H179 C198 R205 G209 N210 H240 F31 Y36 W56 D87 H148 C167 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=1.9uM remove_due_to_license_issue Q9K2N0 30427656 304 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5mxr A 1.75 BS03 JTY A 1 F62 W87 D118 H179 C198 R205 G209 N210 H240 F31 W56 D87 H148 C167 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=6.2uM remove_due_to_license_issue Q9K2N0 30427656 305 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5mxr A 1.75 BS04 JTY A 2 A132 H153 A101 H122 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=6.2uM remove_due_to_license_issue Q9K2N0 30427656 306 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5mxv A 1.626 BS01 K3T A 1 W103 G106 I107 F110 W145 Y148 T149 N176 N179 E180 W207 W82 G85 I86 F89 W124 Y127 T128 N155 N158 E159 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=12uM remove_due_to_license_issue P9WMC1 29018348 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5mxx A 1.75 BS01 W4A A 1 L86 A107 F165 V167 L168 G169 H170 L220 Y227 L31 A52 F110 V112 L113 G114 H115 L165 Y172 D213 D158 2.7.11.1 0004672,0005524,0006468 ic50=31nM remove_due_to_license_issue IC50=31nM Q96SB4 28135068 701 QEDPNDYCKGGYHLVKIGDLFNGRYHVIRKLGWGHFSTVWLSWDIQGKKFVAMKVVKSAEHYTETALDEIRLLKSVRNSDPNDPNREMVVQLLDDFKISGVNGTHICMVFEVLGHHLLKWIIKSNYQGLPLPCVKKIIQQVLQGLDYLHTKCRITHTDIKPENILLSVNEQYIRRLAAEATENFLVNPLEPKNAEKLKVKIADLGNACWVHKHFTEDIQTRQYRSLEVLIGSGYNTPADIWSTACMAFELATGDYLFEPHSGEEYTRDEDHIALIIELLGKVPRKLIVAGKYSKEFFTKKGDLKHITKLKPWGLFEVLVEKYEWSQEEAAGFTDFLLPMLELIPEKRATAAECLRHPWLNS 5my8 A 1.7 BS01 RXZ A 1 W88 S92 V94 A107 K109 F165 V167 L168 G169 H170 L220 V223 Y227 A496 W25 S29 V31 A44 K46 F102 V104 L105 G106 H107 L157 V160 Y164 A196 D213 D150 2.7.11.1 0004672,0005524,0006468 Kd=72nM remove_due_to_license_issue IC50=3.18nM Q96SB4 28135068 724 KGGYHLVKIGDLFNGRYHVIRKLGWGHFSTVWLSWDIQGKKFVAMKVVKSAEHYTETALDEIRLLKSVRNSDPNDPNREMVVQLLDDFKISGVNGTHICMVFEVLGHHLLKWIIKSNYQGLPLPCVKKIIQQVLQGLDYLHTKCRIIHTDIKPENILLSVNEQYIRRLAAEATEWQRFLVNPLEPKNAEKLKVKIADLGNACWVHKHFTEDIQTRQYRSLEVLIGSGYNTPADIWSTACMAFELATGDYLFEPHSGEEYTRDEDHIALIIELLGKVPRKLIVAGKYSKEFFTKKGDLKHITKLKPWGLFEVLVEKYEWSQEEAAGFTDFLLPMLELIPEKRATAAECLRHPWLNS 5myd A 2.3 BS01 DUP A 1 Q17 F20 D21 E39 E42 D70 F74 K154 N158 Q17 F20 D21 E39 E42 D70 F74 K154 N158 3.6.1.23 0004170,0046872 ic50=13.9uM remove_due_to_license_issue A0A2D0TC86 28892519 201 MTNTLTTDQLQELLQIQKEFDDRIPTLNLGDSKIAYVVEFFEWFNTLETFKNWKKKPGKPLDVQLDELADILAFGLSIANQQGFEEYDRDLFFESFDEEYFLDFPYLRNQDMIYDMMSEFYDDDLTSIRRLVIVFKIAEQLYTIDQLIDAYKKKMKRNHE 5myg A 2.3 BS01 LS8 A 1 I652 F653 V657 P658 Y707 N708 F714 I27 F28 V32 P33 Y82 N83 F89 ? Kd=31nM remove_due_to_license_issue Kd=31nM, IC50=47nM P55201 28714688 801 MEMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKMG 5myl A 1.724 BS01 Q2N A 1 W103 G106 I107 F110 W138 M142 W145 Y148 T149 V152 N176 N179 F184 W207 W82 G85 I86 F89 W117 M121 W124 Y127 T128 V131 N155 N158 F163 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=9.9uM remove_due_to_license_issue P9WMC1 29018348 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5mym B 2.28 BS01 HYV B 1 G106 F110 F114 G124 Q125 R128 W138 T149 N176 N179 E180 L183 F184 W207 G92 F96 F100 G110 Q111 R114 W124 T135 N162 N165 E166 L169 F170 W193 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=3.9uM remove_due_to_license_issue P9WMC1 29018348 301 RRTARPSGDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5myn A 1.564 BS01 ZUF A 1 W103 G106 I107 F110 W145 Y148 T149 N176 N179 W207 W82 G85 I86 F89 W124 Y127 T128 N155 N158 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=30uM remove_due_to_license_issue P9WMC1 29018348 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5myr A 1.828 BS01 UDY A 1 W103 G106 I107 F110 F114 W138 M142 W145 Y148 T149 N176 E180 L183 F184 W207 W82 G85 I86 F89 F93 W117 M121 W124 Y127 T128 N155 E159 L162 F163 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=22uM remove_due_to_license_issue P9WMC1 29018348 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5mys A 1.587 BS01 YP6 A 1 W103 G106 F110 W138 M142 W145 Y148 T149 N176 N179 F184 W207 W82 G85 F89 W117 M121 W124 Y127 T128 N155 N158 F163 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=50uM remove_due_to_license_issue P9WMC1 29018348 301 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE 5myv A 2.9 BS01 W4A A 1 L98 F177 V179 L180 G181 H182 L20 F99 V101 L102 G103 H104 D225 D147 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P78362 28135068 716 YHPVKIGDLFNGRYHVIRKLGWGHFSTVWLCWDMQGKRFVAMKVVKSAQHYTETALDEIKLLKCVRESDPSDPNKDMVVQLIDDFKISGMNGIHVCMVFEVLGHHLLKWIIKSNYQGLPVRCVKSIIRQVLQGLDYLHSKCKIIHTDIKPENILMCVDDAYVRRMAAEATEWQKLLVNPLDPRNADKIRVKIADLGNACWVHKHFTEDIQTRQYRSIEVLIGAGYSTPADIWSTACMAFELATGDYLFEPHSGEDYSRDEDHIAHIIELLGSIPRHFALSGKYSREFFNRRGELRHITKLKPWSLFDVLVEKYGWPHEDAAQFTDFLIPMLEMVPEKRASAGECLRHPWLNS 5mz3 A 2.15 BS01 8EN A 1 V38 A51 K53 E71 L74 I84 L104 T106 L108 M109 H148 L167 D168 F169 V35 A48 K50 E68 L71 I81 L101 T103 L105 M106 H145 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.0002uM remove_due_to_license_issue IC50=220nM Q16539 29107542 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 5mzg A 1.85 BS01 2GE A 1 F27 N33 F72 F74 M81 W117 D119 D120 F139 F28 N34 F73 F75 M82 W118 D120 D121 F140 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=138nM remove_due_to_license_issue P53368 29281266 201 HMSTSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADLWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVD 5n0d A 1.7 BS02 8F2 A 1 W5 Q92 H94 H119 V121 F131 L198 T199 P201 W6 Q93 H95 H120 V122 F131 L198 T199 P201 H64 H94 H96 E106 H119 T199 H65 H95 H97 E107 H120 T199 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.3nM remove_due_to_license_issue Ki=3.3nM P00918 28453941 302 GMSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 5n0e A 1.75 BS02 8F3 A 1 H64 H94 H119 L198 T199 T200 P201 P202 H61 H91 H116 L194 T195 T196 P197 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.6nM remove_due_to_license_issue Ki=3.6nM P00918 28453941 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n0f A 1.69 BS01 7K2 A 1 F122 D124 D125 W172 C183 D228 Y243 D294 F84 D86 D87 W134 C145 D190 Y205 D256 ? 0005975 Kd=0.9uM remove_due_to_license_issue Q9Z4P9 28766587 401 SDGDTAMKAFNDTFWDPNAKMFWKDSKREKHQDFWVEAELWELVMDAYQHTSDPALKAELKTQIDDVYDGTVAKYGQDWTNNPFNDDIMWWAMGSARAYQITGNPRYLEAARDHFDFVYDTQWDEEFANGGIWWLNSDHNTKNACINFPAAQAALYLYDITKDEHYLNAATKIFRWGKTMLTDGNGKVFDRIEIEHGAVPDATHYNQGTYIGSAVGLYKATGNAVYLDDAVKAAKFTKNHLVDSNGVLNYEGPNGDLKGGKTILMRNLAHLQKTLDETGQYPEFSAEFDEWLAFNIEMAWSHQNSDHIVDGNWAGGTYESWSSAAAVQALNG 5n16 A 1.76 BS01 8FN A 1 P233 F234 V238 C287 F290 N291 I297 P42 F43 V47 C96 F99 N100 I106 ? Kd=5uM remove_due_to_license_issue Q5A4W8 28516956 401 GAPKPPQEPDMNNLPENPIPQHQAKFVLNTIKAVKRNREAVPFLHPVDTVKLNVPFYYNYIPRPMDLSTIERKINLKAYEDVSQVVDDFNLMVKNCKKFNGEAAGISKMATNIQAQFEKLMVKVPPKEL 5n16 A 1.76 BS02 8FN A 2 D239 K242 L243 D48 K51 L52 ? Kd=5uM remove_due_to_license_issue Q5A4W8 28516956 404 GAPKPPQEPDMNNLPENPIPQHQAKFVLNTIKAVKRNREAVPFLHPVDTVKLNVPFYYNYIPRPMDLSTIERKINLKAYEDVSQVVDDFNLMVKNCKKFNGEAAGISKMATNIQAQFEKLMVKVPPKEL 5n17 A 1.6 BS01 8FK A 1 P233 F234 F290 N291 I297 P44 F45 F101 N102 I108 ? Kd=4.8uM remove_due_to_license_issue Q5A4W8 28516956 401 AMGAPKPPQEPDMNNLPENPIPQHQAKFVLNTIKAVKRNREAVPFLHPVDTVKLNVPFYYNYIPRPMDLSTIERKINLKAYEDVSQVVDDFNLMVKNCKKFNGEAAGISKMATNIQAQFEKLMVKVPPK 5n18 A 1.45 BS01 8HZ A 1 V415 L420 I422 Y425 F467 N468 V474 V32 L37 I39 Y42 F84 N85 V91 ? Kd=2.1uM remove_due_to_license_issue Q5A4W8 28516956 501 MGAAELRFCNQTIKELMSKKHYNYNFPFLAPVDTVALNIPNYNEIVKQPMDLGTIQSKLANNEYENADDFEKDVRLVFKNCYLFNPEGTDVNMMGHRLEAVFDKKW 5n1p A 1.448 BS01 8GK A 1 D76 H126 H130 P166 Y167 W191 H230 D9 H59 H63 P99 Y100 W124 H163 3.5.1.104 0005975,0016810 Kd=25uM remove_due_to_license_issue Q81EJ6 29257674 301 RKVAYLTFDDGPGKYTAELLNTLKQHDAKATFFLIGANVKEFPDLVKRENAEGHYVGMHSMTHNFAKLYKNGEYVNEMKEDQGLIANIIGKSPKLTRPPYGSMPGLNEGLRNKVVEGGFKVWDWTIDSLDWRYNKMPVDAAAAQIAQNVLTNATKPQEVILMHDIHPQSVAAVPAILKGLKEKGYEFEAYHEESHFPVNFWHDNRM 5n1r A 1.3 BS02 8GH A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=11nM P00918 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n1s A 1.3 BS02 8GE A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=10nM P00918 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n1v A 2.52 BS01 8GQ A 1 V53 V66 F113 V116 N117 N118 M163 D175 V52 V65 F112 V115 N116 N117 M162 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 28485934 413 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 5n1x B 1.72 BS01 8HH B 1 N21 R24 L25 N15 R18 L19 ? Kd=689uM remove_due_to_license_issue P41182 28485934 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTARKFIKA 5n1x B 1.72 BS02 8HH B 2 M51 Y58 M45 Y52 ? Kd=689uM remove_due_to_license_issue P41182 28485934 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTARKFIKA 5n1z A 1.81 BS01 8GQ A 1 M51 A52 G55 Y58 Q113 M114 E115 M46 A47 G50 Y53 Q108 M109 E110 ? Kd=0.0065uM remove_due_to_license_issue IC50=1995nM P41182 28485934 202 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 5n20 A 1.38 BS01 8GN A 1 M51 A52 C53 S54 Y58 S59 M46 A47 C48 S49 Y53 S54 ? ic50=61uM remove_due_to_license_issue P41182 28485934 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 5n21 A 1.58 BS01 8HN A 1 M51 C53 G55 Y58 Q113 E115 M45 C47 G49 Y52 Q107 E109 ? Kd=1.1uM remove_due_to_license_issue Kd=1100nM P41182 28485934 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 5n21 A 1.58 BS02 8HN B 1 N21 R24 L25 N15 R18 L19 ? Kd=1.1uM remove_due_to_license_issue Kd=1100nM P41182 28485934 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 5n24 A 1.5 BS02 8HE A 1 H94 H119 F131 L198 T199 T200 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=1.2nM P00918 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n24 A 1.5 BS03 8HE A 2 H3 H4 W5 H10 N11 W16 D19 H1 H2 W3 H8 N9 W14 D17 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=1.2nM P00918 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n25 A 1.4 BS02 8HK A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=17nM P00918 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n25 A 1.4 BS03 8HK A 2 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=17nM P00918 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5n2d A 2.35 BS01 8J8 B 1 F19 Y56 M115 I116 S117 A121 D122 Y123 F2 Y39 M98 I99 S100 A104 D105 Y106 ? remove_due_to_license_issue Kd=<1000nM, IC50=6.0nM Q9NZQ7 28613862 201 AFTVTVPKDLYVVEYGSNMTIECKFPVEKQLDLAALIVYWEMEDKNIIQFVHGEEDLKVQHSSYRQRARLLKDQLSLGNAALQITDVKLQDAGVYRCMISYGGADYKRITVKVNAPYAAALEHHH 5n2d B 2.35 BS01 8J8 B 1 Y56 Q66 M115 I116 S117 Y39 Q49 M98 I99 S100 ? ic50~50uM remove_due_to_license_issue Kd=<1000nM, IC50=6.0nM Q9NZQ7 28613862 201 AFTVTVPKDLYVVEYGSNMTIECKFPVEKQLDLAALIVYWEMEDKNIIQFVHGEEDLKVQHSSYRQRARLLKDQLSLGNAALQITDVKLQDAGVYRCMISYGGADYKRITVKVNAPYAAALEHH 5n2f A 1.7 BS01 8HW B 1 Y56 M115 A121 D122 Y39 M98 A104 D105 ? remove_due_to_license_issue Q9NZQ7 28613862 201 AFTVTVPKDLYVVEYGSNMTIECKFPVEKQLDLAALIVYWEMEDKNIIQFVHGEEDLKVQHSSYRQRARLLKDQLSLGNAALQITDVKLQDAGVYRCMISYGGADYKRITVKVNAPYAAALEHHHH 5n2f B 1.7 BS01 8HW B 1 I54 Y56 Q66 M115 I116 A121 D122 I37 Y39 Q49 M98 I99 A104 D105 ? ic50=80nM remove_due_to_license_issue Q9NZQ7 28613862 201 AFTVTVPKDLYVVEYGSNMTIECKFPVEKQLDLAALIVYWEMEDKNIIQFVHGEEDLKVQHSSYRQRARLLKDQLSLGNAALQITDVKLQDAGVYRCMISYGGADYKRITVKVNAPYAAALEHH 5n2t E 1.379 BS06 8KK E 1 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 410 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n2x E 1.209 BS06 8KN E 1 N111 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 N111 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 409 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n2z E 1.37 BS06 8JH E 1 N111 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 N111 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 410 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n31 E 1.368 BS06 8LB E 1 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 410 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n34 E 1.22 BS06 8JQ E 1 N112 A113 F114 N116 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 N116 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 412 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n3v E 1.12 BS06 8L5 E 1 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 406 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n3w A 2.3 BS02 8KW A 1 Q136 A137 Y267 W311 F314 V367 P374 D375 A377 Y378 Q133 A134 Y264 W308 F311 V364 P371 D372 A374 Y375 E271 H295 E296 H299 E318 D375 Y383 E268 H292 E293 H296 E315 D372 Y380 3.3.2.6,3.4.11.4 0003723,0004177,0004301,0004463,0005515,0005576,0005634,0005654,0005737,0005829,0006508,0006629,0006691,0008233,0008237,0008270,0010043,0019370,0019538,0043171,0043434,0045148,0046872,0060509,0070006,0070062,1904724,1904813 ic50=0.5uM remove_due_to_license_issue P09960 28303931 704 VDTCSLASPASVCRTKHLHLRCSVDFTRRTLTGTAALTVQSQEDNLRSLVLDTKDLTIEKVVINGQEVKYALGERQSYKGSPMEISLPIALSKNQEIVIEISFETSPKSSALQWLTPEQTSGKEHPYLFSQCQAIHCRAILPCQDTPSVKLTYTAEVSVPKELVALMSAIRDGETPDPEDPSRKIYKFIQKVPIPCYLIALVVGALESRQIGPRTLVWSEKEQVEKSAYEFSETESMLKIAEDLGGPYVWGQYDLLVLPPSFPYGGMENPCLTFVTPTLLAGDKSLSNVIAHEISHSWTGNLVTNKTWDHFWLNEGHTVYLERHICGRLFGEKFRHFNALGGWGELQNSVKTFGETHPFTKLVVDLTDIDPDVAYSSVPYEKGFALLFYLEQLLGGPEIFLGFLKAYVEKFSYKSITTDDWKDFLYSYFKDKVDVLNQVDWNAWLYSPGLPPIKPNYDMTLTNACIALSQRWITAKEDDLNSFNATDLKDLSSHQLNEFLAQTLQRAPLPLGHIKRMQEVYNFNAINNSEIRFRWLRLCIQSKWEDAIPLALKMATEQGRMKFTRPLFKDLAAFDKSHDQAVRTYQEHKASMHPVTAMLVGKDLKV 5n3y E 1.339 BS06 8L2 E 1 N112 A113 F114 N116 H142 E143 H146 Y157 E166 L202 R203 H231 N112 A113 F114 N116 H142 E143 H146 Y157 E166 L202 R203 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 remove_due_to_license_issue P00800 28590130 411 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGNGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSQMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5n49 B 1.94 BS01 8LW B 1 R585 I586 Q589 V591 S592 Y641 N642 F648 R27 I28 Q31 V33 S34 Y83 N84 F90 ? ic50=450nM remove_due_to_license_issue O95696 28402630 701 AMELRLTELTRLLRSVLDQLQDKDPARIFAQPVSLKEVPDYLDHIKHPMDFATMRKRLEAQGYKNLHEFEEDFDLIIDNCMKYNARDTVFYRAAVRLRDQGGVVLRQARREVDS 5n4s A 1.2 BS03 R38 A 1 Y67 H116 D118 H179 R205 G209 N210 H240 Y36 H85 D87 H148 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=0.055uM remove_due_to_license_issue Q9K2N0 28470248 504 AYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4s A 1.2 BS04 R38 B 1 G64 A65 G33 A34 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=0.055uM remove_due_to_license_issue Q9K2N0 28470248 504 AYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5n4t A 1.16 BS03 R59 A 1 Y67 W87 D118 H179 R205 N210 H240 Y38 W58 D89 H150 R176 N181 H211 H114 H116 D118 H179 C198 Y201 N210 H240 H85 H87 D89 H150 C169 Y172 N181 H211 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=1.06uM remove_due_to_license_issue Q9K2N0 28470248 504 SGEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 5n53 B 1.48 BS01 8NB B 1 Y174 P176 T207 P208 T213 Y75 P77 T108 P109 T114 N102 R236 D260 E265 H283 N3 R137 D161 E166 H184 1.1.1.37,1.1.1.399,1.1.1.95 0051287 Kd=2.8mM remove_due_to_license_issue Kd=2800000nM O43175 29568346 301 NGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSR 5n55 A 1.99 BS02 8NN A 1 F62 Y67 P68 W87 H116 D118 R205 G209 N210 H240 F31 Y36 P37 W56 H85 D87 R174 G178 N179 H209 H114 H116 D118 H179 C198 L201 N210 H240 H83 H85 D87 H148 C167 L170 N179 H209 3.5.2.6 Kd=1.03uM remove_due_to_license_issue Q8GKX2 28470248 502 EYPTVNEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRKAGVATYASPSTRRLAEAEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSANVLYGGCAVLALSRTSAGNVADADLAEWPTSVERIQKHYPEAEVVIPGHGLPGGLDLLQHTANVVTAHKN 5n55 A 1.99 BS03 8NN B 1 D63 G64 D32 G33 H114 H116 D118 H179 C198 L201 N210 H240 H83 H85 D87 H148 C167 L170 N179 H209 3.5.2.6 Kd=1.03uM remove_due_to_license_issue Q8GKX2 28470248 502 EYPTVNEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRKAGVATYASPSTRRLAEAEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSANVLYGGCAVLALSRTSAGNVADADLAEWPTSVERIQKHYPEAEVVIPGHGLPGGLDLLQHTANVVTAHKN 5n58 A 1.957 BS02 93W A 1 Y67 S204 R205 T206 S207 H240 Y29 S166 R167 T168 S169 H202 H114 H116 D118 H179 C198 L201 N210 H240 H76 H78 D80 H141 C160 L163 N172 H202 3.5.2.6 Kd=0.8uM remove_due_to_license_issue Q8GKX2 28470248 502 IPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRKAGVATYASPSTRRLAEAEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSANVLYGGCAVLALSRTSAGNVADADLAEWPTSVERIQKHYPEAEVVIPGHGLPGGLDLLQHTANVVTA 5n69 A 2.45 BS03 2OW A 1 K146 Y164 T167 D168 H666 P710 N711 R712 Y722 L770 E774 K143 Y161 T164 D165 H619 P663 N664 R665 Y675 L720 E724 S180 G181 T185 N238 S241 S242 G464 E466 S177 G178 T182 N221 S224 S225 G441 E443 ? 0003774,0005524,0016459,0051015 Kd=0.29uM remove_due_to_license_issue Q9BE39 28775348 904 AEMAAFGEAAPYLRKSEKERLEAQTRPFDLKKDVFVPDDKEEFVKATILSREGGKVTAETEHGKTVTVKEDQVLQQNPPKFDKIEDMAMLTFLHEPAVLYNLKERYASWMIYTYSGLFCVTINPYKWLPVYNAEVVAAYRGKKRSEAPPHIFSISDNAYQYMLTDRENQSILITGESGAGKTVNTKRVIQYFAVIAATLEDQIIQANPALEAFGNAKTVRNDNSSRFGKFIRIHFGATGKLASADIETYLLEKSRVIFQLKAERDYHIFYQILSNKKPELLDMLLITNNPYDYAFISQGETTVASIDDAEELMATDNAFDVLGFTTEEKNSMYKLTGAIMHFGNMKFKLKQREEQAEPDGTEEADKSAYLMGLNSADLLKGLCHPRVVTKGQNVQQVVYAKGALAKAVYERMFNWMVTRINATLETKQPRQYFIGVLDIAGFEIFDFNSFEQLCINFTNEKLQQFFNHHMFVLEQEEYKKEGIEWEFIDFGMDLQACIDLIEKPMGIMSILEEECMFPKATDMTFKAKLFDNHLGKSSNFQKPRNIKPEAHFSLIHYAGTVDYNIIGWLQKNKDPLNETVVDLYKKSSLKMLSSLFAQTVSALHRENLNKLMTNLRSTHPHFVRCIIPNETKSPGVIDNPLVMHQLRCNGVLEGIRICRKGFPNRILYGDFRQRYRILNPAAIPEIDSRKGAEKLLGSLDIDHNQYKFGHTKVFFKAGLLGLLEEMRDERLSRIITRIQAQSRGVLSRMEFKKLLERRDS 5n6s A 2.1 BS01 8P5 A 1 Q20 H121 W122 N165 E166 W168 V169 E351 W398 E405 W406 F414 Q18 H119 W120 N163 E164 W166 V167 E349 W396 E403 W404 F412 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E349 3.2.1.21 0004553,0005975,0008422,0016798,0030245 remove_due_to_license_issue Q08638 28463498 507 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 5n7v A 2.52 BS01 8PT A 1 I531 V539 A551 I586 C604 G605 L654 P673 I16 V24 A36 I71 C89 G90 L139 P158 D647 K649 N652 D664 T686 D132 K134 N137 D149 T164 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.8nM P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDSQVGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5n84 A 2.3 BS01 8Q5 A 1 K553 I586 M602 G605 N606 L654 I663 K38 I71 M87 G90 N91 L139 I148 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 Kd=11nM remove_due_to_license_issue IC50=10.0nM P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQQVGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5n87 A 2.29 BS01 N66 A 1 I531 S533 S537 K553 C604 G605 I607 D608 L654 I663 I16 S18 S22 K38 C89 G90 I92 D93 L139 I148 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 Kd=0.56nM remove_due_to_license_issue P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQQVGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5n8v A 1.55 BS01 KZZ A 1 N13 A14 F17 T26 F34 K38 N10 A11 F14 T23 F31 K35 ? 0005778,0016560 Ki=0.207uM remove_due_to_license_issue Q8IEW2 28360328 101 HSEREKRVSNAVEFLLDSRVRRTPTSSKVHFLKSKGLSAEEICEAFTKVGQPKTLNEIKRILS 5n93 A 2.1 BS01 8QE A 1 I531 A551 M602 E603 C604 I607 L654 I663 M671 I16 A36 M87 E88 C89 I92 L139 I148 M156 D647 K649 N652 D664 T686 D132 K134 N137 D149 T162 2.7.12.1 0004672,0005524,0006468 Kd=2.2nM remove_due_to_license_issue IC50=6.4nM P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDVGTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5n9k A 1.643 BS01 8QK A 1 L45 V66 K68 I95 F113 V116 M163 I174 D175 L44 V65 K67 I94 F112 V115 M162 I173 D174 D156 K158 N161 D175 S194 D155 K157 N160 D174 S193 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.46nM remove_due_to_license_issue P68400 29462988 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 5n9l A 1.79 BS01 8QH A 1 R47 G48 S51 V53 V66 K68 F113 V116 M163 I174 D175 R46 G47 S50 V52 V65 K67 F112 V115 M162 I173 D174 D156 K158 N161 D175 S194 D155 K157 N160 D174 S193 2.7.11.1 0004672,0004674,0005524,0006468 Ki=15nM remove_due_to_license_issue IC50=30nM P68400 29462988 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 5n9r A 2.23 BS01 8RN A 1 Y224 D295 Q297 L406 M407 R408 F409 K420 H456 N460 H461 Y465 Y514 Y19 D90 Q92 L201 M202 R203 F204 K215 H251 N255 H256 Y260 Y308 3.4.19.12 0004843,0016579 Kd=2.6uM remove_due_to_license_issue IC50=300nM Q93009 29200206 1003 MSKKHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHDDLSVRHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQKRKERQEHH 5n9s A 2.3 BS01 8QW A 1 I531 A551 K553 Y568 M600 M602 G605 N606 L654 I663 I16 A36 K38 Y53 M85 M87 G90 N91 L139 I148 D647 K649 N652 D664 T686 D132 K134 N137 D149 T164 2.7.12.1 0004672,0005524,0006468 Kd=2.4nM remove_due_to_license_issue IC50=<1.000nM P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDSQVGTVNYMPPEAIKDKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5n9t A 1.73 BS01 8QQ A 1 Y224 D295 Q297 Q351 L406 M407 R408 F409 K420 H456 N460 H461 Y465 Y514 Y18 D89 Q91 Q145 L200 M201 R202 F203 K214 H250 N254 H255 Y259 Y308 3.4.19.12 0004843,0016579 ic50=22nM remove_due_to_license_issue IC50=22nM Q93009 29200206 1005 SKKHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHDDDLSVRHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQKRKERQEHHH 5na0 A 2.9 BS01 8QZ A 1 I531 G534 S537 K553 Y568 M600 G605 N606 S611 K615 L654 D664 I16 G19 S22 K38 Y53 M85 G90 N91 S96 K100 L139 D149 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMVGTVNYMPPEAIKDISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5nad A 2.8 BS01 8RH A 1 I531 Q541 E571 I586 M602 C604 G605 A651 L654 I663 M671 P673 I16 Q26 E56 I71 M87 C89 G90 A136 L139 I148 M156 P158 D647 K649 N652 D664 T686 D132 K134 N137 D149 T160 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.000000nM P33981 28539250 901 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 5nai A 1.15 BS03 93W A 1 F62 Y67 S204 R205 T206 S207 G209 H240 F32 Y37 S174 R175 T176 S177 G179 H210 H114 H116 D118 H179 C198 L201 N210 H240 H84 H86 D88 H149 C168 L171 N180 H210 3.5.2.6 remove_due_to_license_issue Q8GKX2 28470248 304 GEYPTVNEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRKAGVATYASPSTRRLAEAEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSANVLYGGCAVLALSRTSAGNVADADLAEWPTSVERIQKHYPEAEVVIPGHGLPGGLDLLQHTANVVTAHKN 5nap A 2.17 BS01 DZ7 A 1 Y70 W84 E199 W279 F330 F331 Y334 Y67 W81 E196 W276 F327 F328 Y331 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=11.12nM remove_due_to_license_issue P04058 29651884 611 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 5nar A 1.55 BS01 8RW A 1 H40 L41 C42 R151 C191 K192 G193 S195 T214 S215 G216 S217 R218 C220 H24 L25 C26 R133 C166 K167 G168 S170 T185 S186 G187 S188 R189 C191 H57 D102 K192 G193 D194 S195 G196 H41 D85 K167 G168 D169 S170 G171 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=0.5uM remove_due_to_license_issue IC50=500nM P00746 28621538 302 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNTERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 5nau A 2.25 BS01 DZ0 A 1 W84 Y121 E199 W279 F330 F331 Y334 H440 W81 Y118 E196 W276 F327 F328 Y331 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 Ki=29.86nM remove_due_to_license_issue P04058 29651884 611 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 5naw A 1.25 BS01 8RZ A 1 H40 L41 C42 H57 C58 R151 C191 K192 G193 S195 T214 S215 G216 R218 C220 H24 L25 C26 H41 C42 R137 C179 K180 G181 S183 T198 S199 G200 R202 C204 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=0.05uM remove_due_to_license_issue IC50=50nM P00746 28621538 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 5nb6 A 1.75 BS01 8S2 A 1 H40 L41 C42 R151 C191 K192 G193 S195 T214 S215 G216 R218 H24 L25 C26 R133 C165 K166 G167 S169 T184 S185 G186 R188 H57 D102 K192 G193 D194 S195 G196 H41 D85 K166 G167 D168 S169 G170 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=0.5uM remove_due_to_license_issue IC50=667nM P00746 28621538 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 5nb7 A 1.33 BS01 8NQ A 1 L41 C42 H57 C58 W141 G142 C191 K192 G193 S195 S215 G216 S217 R218 L25 C26 H41 C42 W128 G129 C179 K180 G181 S183 S199 G200 S201 R202 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=0.006uM remove_due_to_license_issue IC50=9nM P00746 28621538 303 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 5nba A 1.87 BS01 8S5 A 1 H40 L41 H57 C58 R151 C191 K192 G193 S195 T214 S215 G216 S217 R218 C220 H24 L25 H41 C42 R132 C174 K175 G176 S178 T193 S194 G195 S196 R197 C199 H57 D102 K192 G193 D194 S195 G196 H41 D84 K175 G176 D177 S178 G179 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=0.05uM remove_due_to_license_issue IC50=50nM P00746 28621538 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 5nbw H 2.4 BS01 8SK L 1 E35 K99 Y100 G101 W104 E35 K99 Y100 G101 W104 remove_due_to_license_issue 28603847 301 EVKLHQSGAELVNPGASVKISCKAPGYTFNNYWIEWVKQRPGHGLEWIGEILPGSGRINYNEKFKDKATFTADTSSNTAYMQLSSLTSDDSAVYYCAKKYGDYWGQGTTVTVSSAKTTPPSVYPLAPGSAAQTNSMVTLGCLVKGYFPEPVTVTWNSGSLSSGVHTFPAVLQSDLYTLSSSVTVPSSTWPSETVTCNVAHPASSTKVDKKIVPRDC 5nbw L 2.4 BS01 8SK L 1 N34 F36 Y49 L89 Y91 N34 F36 Y49 L89 Y91 remove_due_to_license_issue 28603847 301 DIELTQSPSSMYASLGERVTITCKASQDINSYLNWFQQKPGKSPKTLIYHTNRLVDGVPSRFSGSGSGQDYSLIISSLEFEDMGIYYCLQYDEFPYTFGGGTKLELKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC 5ncq A 3.0 BS02 8T8 A 1 D59 L61 L65 N101 L253 D254 E309 P312 I315 D59 L61 L65 N101 L253 D254 E299 P302 I305 D351 D703 D707 D341 D693 D697 7.2.2.10 0000166,0005215,0005388,0005509,0005524,0006816,0016020,0016529,0016887,0031448,0033017,0046872,0070588,0106134,1901896,1902082,1990036 remove_due_to_license_issue P04191 29293507 1005 MEAAHSKSTEECLAYFGVSETTGLTPDQVKRHLEKYGHNELPAEEGKSLWELVIEQFEDLLVRILLLAACISFVLAWFEEGEETITAFVEPFVILLILIANAIVGVWQERNAENAIEALKEYEPEMGKVYRADRKSVQRIKARDIVPGDIVEVAVGDKVPADIRILSIKSTTLRVDQSILTGESVSVIKHTEPVPDPRAVNQDKKNMLFSGTNIAAGKALGIVATTGVSTEIGKIRDQMAATEQDKTPLQQKLDEFGEQLSKVISLICVAVWLINIGWIRGAIYYFKIAVALAVAAIPEGLPAVITTCLALGTRRMAKKNAIVRSLPSVETLGCTSVICSDKTGTLTTNQMSVCKMFIIDKVDGDFCSLNEFSITGSTYAPEGEVLKNDKPIRSGQFDGLVELATICALCNDSSLDFNETKGVYEKVGEATETALTTLVEKMNVFNTEVRNLSKVERANACNSVIRQLMKKEFTLEFSRDRKSMSVYCSPAKSSRAAVGNKMFVKGAPEGVIDRCNYVRVGTTRVPMTGPVKEKILSVIKEWGTGRDTLRCLALATRDTPPKREEMVLDDSSRFMEYETDLTFVGVVGMLDPPRKEVMGSIQLCRDAGIRVIMITGDNKGTAIAICRRIGIFGENEEVADRAYTGREFDDLPLAEQREACRRACCFARVEPSHKSKIVEYLQSYDEITAMTGDGVNDAPALKKAEIGIAMGSGTAVAKTASEMVLADDNFSTIVAAVEEGRAIYNNMKQFIRYLISSNVGEVVCIFLTAALGLPEALIPVQLLWVNLVTDGLPATALGFNPPDLDIMDRPPRSPKEPLISGWLFFRYMAIGGYVGAATVGAAAWWFMYAEDGPGVTYHQLTHFMQCTEDHPHFEGLDCEIFEAPEPMTMALSVLVTIEMCNALNSLSENQSLMRMPPWVNIWLLGSICLSMSLHFLILYVDPLPMIFKLKALDLTQWLMVLKISLPVIGLDEILKFIARNYLEG 5ncy A 1.9 BS01 8TK A 1 F751 M752 P758 W760 I777 Y813 I825 E826 V827 V828 M900 I910 F560 M561 P567 W569 I586 Y622 I634 E635 V636 V637 M709 I719 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=0.4nM remove_due_to_license_issue O35904 28520415 1104 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELGRITEEELREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5ncz A 1.94 BS01 8TN A 1 F751 M752 P758 W760 I777 Y813 I825 V827 V828 D832 M900 I910 F560 M561 P567 W569 I586 Y622 I634 V636 V637 D641 M709 I719 2.7.1.137,2.7.1.153 0001782,0002250,0005524,0005737,0005829,0006629,0006935,0006954,0007166,0010628,0016301,0016303,0030154,0036092,0042113,0043491,0045087,0045766,0046854,0046934,0048872,0050832 ic50=0.79nM remove_due_to_license_issue O35904 28520415 1105 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELGRITEEELREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5ndb A 2.38 BS04 8TW A 1 Y59 F79 D110 H195 C220 K223 Y232 H262 Y27 F48 D79 H164 C183 K186 Y192 H220 H106 H108 D110 H195 C220 K223 Y232 H262 H75 H77 D79 H164 C183 K186 Y192 H220 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue Q8G9Q0 29250863 412 DHVDLPYNLTATKIDSDVFVVTDRDFYSSNVLVAKMLDGTVVIVSSPFENLGTQTLMDWVAKTMKPKKVVAINTHFHLDGTGGNEIYKKMGAETWSSDLTKQLRLEENKKDRIKAAEFYKNEDLKRRILSSHPVPADNVFDLKQGKVFSFSNELVEVSFPGPAHSPDNVVVYFPKKKLLFGGCMIKPKELGYLGDANVKAWPDSARRLKKFDAKIVIPGHGEWGGPEMVNKTIKVAEKAVGEMR 5ndd A 2.801 BS01 8TZ A 1 Y82 Y134 H135 W141 F155 C226 H227 D228 I327 L330 Y190 Y242 H243 W249 F263 C334 H335 D336 I535 L538 E1011 D1020 E12 D21 3.2.1.17 0003796,0004930,0005506,0007186,0009055,0009253,0016020,0016798,0016998,0020037,0022900,0030430,0031640,0042597,0042742,0044659,0046872 remove_due_to_license_issue P00720,P0ABE7,P55085 28445455 2201 ASNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYIYEFFSVDEFSASVLTGKLTTVFLPIVYTIVFVVALPSNGMALWVFLFRTKKKAPAVIYMANLALADLLSVIWFPLKIAYHIHGNNWIYGEALCNVLIGFFYANMYCSILFLTCLSVQRAWEIVNPMGHSRKKANIAIGISLAIWLLILLVTIPLYVVKQTIFIPALQITTCHDVLPEQLLVGDMFNYFLSLAIGVFLFPAFLTASAYVLMIRALADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLENSEKKRKRAIKLAVTVAAMYLICFTPSNLLLVVHYFLIKSQGQSHVYALYIVALCLSTLNSCIDPFVYYFVSHDFRDHAKNAL 5ndf A 2.3 BS03 LU2 A 1 I253 L270 W282 F361 I179 L196 W208 F287 2.4.1.41 0000139,0004653,0005515,0005576,0005789,0005794,0005795,0006486,0006493,0016020,0016266,0016757,0018242,0018243,0030145,0030246,0032580,0046872,0048471,0051604 Ki=1.4uM remove_due_to_license_issue Q10471 29061849 608 KVRWPDFNQEAYVGGTMVRSGQDPYARNKFNQVESDKLRMDRAIPDTRHDQCQRKQWRVDLPATSVVITFHNEARSALLRTVVSVLKKSPPHLIKEIILVDDYSNDPEDGALLGKIEKVRVLRNDRREGLMRSRVRGADAAQAKVLTFLDSHCECNEHWLEPLLERVAEDRTRVVSPIIDVINMDNFQYVGASADLKGGFDWNLVFKWDYMTPEQRRSRQGNPVAPIKTPMIAGGLFVMDKFYFEELGKYDMMMDVWGGENLEISFRVWQCGGSLEIIPCSRVGHVFRKQHPYTFPGGSGTVFARNTRRAAEVWMDEYKNFYYAAVPSARNVPYGNIQSRLELRKKLSCKPFKWYLENVYPELRVPDHQDIAFGALQQGTNCLDTLGHFADGVVGVYECHNAGGNQEWALTKEKSVKHMDLCLTVVDRAPGSLIKLQGCREDDSRQKWEQIEGNSKLRHVGSNLCLDSRTAKSGGLSVEVCGPALSQQWKFTLNL 5ne1 B 2.09 BS01 OK3 B 1 S70 H105 S130 N132 N170 T235 G236 S237 N238 G240 S50 H85 S110 N112 N150 T215 G216 S217 N218 G219 S70 K73 S130 E166 K234 S237 S50 K53 S110 E146 K214 S217 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9RBQ1 28876489 302 NAPTDAAITAASDFAALEKACAGRLGVTLLDTASGRRIGHRQDERFPMCSTFKSMLAATVLSQAERMPALLDRRVPVGEADLLSHAPVTRRHAGKDMTVRDLCRATIITSDNTAANLLFGVVGGPPAVTAFLRASGDTVSRSDRLEPELNSFAKGDPRDTTTPAAMAATLQRVVLGEVLQPASRQQLADWLIDNETGDACLRAGLGKRWRVGDKTGSNGEDARNDIAVLWPVAGGAPWVLTAYLQAGAISYEQRASVLAQVGRIADRLIG 5ne3 A 1.35 BS01 NXL A 1 S69 H104 S129 N131 N169 T215 T234 G235 S236 S49 H84 S109 N111 N149 T195 T214 G215 S216 S69 K72 S129 E165 K233 S236 S49 K52 S109 E145 K213 S216 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue B2FRP5 28876489 301 APTDAAITAASDFAALEKACAGRLGVTLLDTASGRRIGHRQDERFPMCSTFKSMLAATVLSQAERMPALLDRRVPVGEADLLSHAPVTRRHAGKDMTVRDLCRATIITSDNTAANLLFGVVGGPPAVTAFLRASGDTVSRSDRLEPELNSFAKGDPRDTTTPAAMAATLQRVVLGEVLQPASRQQLADWLIDNETGDACLRAGLGKRWRVGDKTGSNGEDARNDIAVLWPVAGGAPWVLTAYLQAGAISYEQRASVLAQVGRIADRLIG 5ne5 A 1.05 BS01 KIF A 1 L310 R363 P364 E365 Y423 E427 T451 E452 L281 R334 P335 E336 Y394 E398 T422 E423 E121 R125 D249 E365 E92 R96 D220 E336 3.2.1.113 0004559,0004571,0005509,0005975,0016020,0016798,0046872 Kd=39nM remove_due_to_license_issue B0SWV2 28493500 501 PEDWKALAADVRSEFQWAWQGYVAKAWGKDEINPVSGTSRSFFIEGHDLGLSLVEALDTLWIMGLDAEFQAGVDWVKANLSFDVDGNAQVFETNIRLVGGLLSAHLASGDPVLLAKARDLADRLAKAFEASPHGLPWRYVNLRTGAVSDPETNLAEIGTYLSEFGVLSQLTGERKYFDMAKRAMRHTLDRRSKIGLMAANIHAMTGAFTSRNASIDVYADSFYEYLWDAWALFGDEDCKRWAVECVDAQLAHQAKRYDGRLWFPMVDFETGAVTGTAQSELAAYYAGLLGQVGRKAQGDDYLASFTYLQATFGVIPESIDVTTGQPRRKHTGLRPEYPDACLNLWLIDRDPRYRRLAAIHYREMKATSRAAFGYTALKDITTRPMTQDDNCPGYWWSEQMKYYYLLFSDTPRIDYGQLQLSTEANVLRGFRK 5nea A 1.3 BS02 8V8 A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.05nM remove_due_to_license_issue Ki=0.050000nM P00918 28728897 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nea A 1.3 BS03 8V8 A 2 H4 W5 N11 H15 W16 D19 H1 W2 N8 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.05nM remove_due_to_license_issue Ki=0.050000nM P00918 28728897 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5neb A 2.05 BS01 8VE A 1 Y61 P88 T90 R95 G140 S141 T142 E190 Y61 P88 T90 R95 G140 S141 T142 E190 ? 0015276,0016020 Ki=17nM remove_due_to_license_issue P22756 28691798 307 GANRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGC 5nee A 1.7 BS02 8V5 A 1 Q92 H94 H96 F131 L198 T199 T200 Q89 H91 H93 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.02nM remove_due_to_license_issue Ki=0.020000nM P00918 28728897 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nev A 2.97 BS01 72L A 1 G11 E12 A31 V64 F80 E81 F82 L83 H84 Q85 D86 K89 Q131 L134 G12 E13 A32 V65 F81 E82 F83 L84 H85 Q86 D87 K90 Q132 L135 D127 K129 Q131 N132 D145 T158 T165 D128 K130 Q132 N133 D146 T159 T166 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 28005359 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPH 5nf5 B 2.85 BS01 8VN B 1 Y61 P88 T90 R95 S141 T142 E190 Y59 P86 T88 R93 S139 T140 E188 ? 0015276,0016020 remove_due_to_license_issue P22756 28691798 303 NRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 5nf6 A 2.55 BS03 8VN A 1 Y61 P88 T90 R95 G140 A141 T142 E189 Y59 P86 T88 R93 G138 A139 T140 E187 ? 0015276,0016020 remove_due_to_license_issue P42264 28691798 304 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 5nf9 A 1.87 BS01 8VW A 1 H158 R162 E165 N174 W181 E184 R186 H46 R50 E53 N62 W69 E72 R74 ? 0030246 Kd=4.7uM remove_due_to_license_issue P17931 28554839 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5nfb A 1.59 BS01 8VT A 1 R144 H158 R162 E165 N174 W181 E184 R186 R32 H46 R50 E53 N62 W69 E72 R74 ? 0030246 Kd=0.77uM remove_due_to_license_issue P17931 28554839 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5ng9 A 1.15 BS01 8VN A 1 Y61 P89 T91 R96 L138 G141 S142 T143 E193 Y61 P89 T91 R96 L138 G141 S142 T143 E193 ? 0015276,0016020 Ki=191nM remove_due_to_license_issue P19491 28691798 304 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECGS 5ngb A 2.9 BS01 8WH A 1 K708 M752 W760 Y813 E826 V827 V828 M900 I910 K512 M556 W564 Y617 E630 V631 V632 M697 I707 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28857471 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLTAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5nge A 2.35 BS01 8WK A 1 Y224 D295 Q297 Q351 L406 M407 R408 F409 H456 D459 N460 H461 Y465 Y514 Y13 D84 Q86 Q140 L195 M196 R197 F198 H245 D248 N249 H250 Y254 Y295 N218 C223 H464 D481 N7 C12 H253 D270 3.4.19.12 0004843,0016579 Kd=65nM remove_due_to_license_issue Q93009 29045389 601 GYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQKRK 5ngf A 2.33 BS01 8WN A 1 C223 Y224 M292 D295 Q297 M407 F409 Y465 C15 Y16 M84 D87 Q89 M199 F201 Y251 N218 C223 H464 D481 N10 C15 H250 D267 3.4.19.12 0004843,0016579 remove_due_to_license_issue Q93009 29045389 601 KHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQK 5ngr A 2.2 BS01 8WT A 1 L9 N33 F72 M81 W117 D119 D120 L7 N31 F70 M79 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=24uM remove_due_to_license_issue P36639 28929756 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5ngs A 1.85 BS01 8WW A 1 Y7 F27 N33 F72 W117 D119 D120 Y5 F25 N31 F70 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=170nM remove_due_to_license_issue P36639 28929756 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5ngt A 1.54 BS01 8WZ A 1 N33 F72 F74 M81 W117 D119 D120 N31 F70 F72 M79 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue P36639 28929756 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5ngu A 2.74 BS01 8X2 A 1 I31 Y36 A52 K54 D106 M108 D111 L156 C166 D167 I21 Y26 A42 K44 D96 M98 D101 L146 C156 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue IC50=36nM P28482 28376306 403 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDLPKEKLKELIFEETARFQ 5ngz A 2.4 BS01 2BG A 1 F70 P73 I74 S81 W146 F69 P72 I73 S80 W145 C86 C85 2.3.2.23 0000209,0003682,0004842,0005515,0005524,0005634,0005654,0005730,0006281,0006513,0006974,0016567,0016740,0019787,0031625,0032446,0035519,0044314,0051865,0061631,0070534,0070936,0070979,0085020 Kd=1.3mM remove_due_to_license_issue Kd=1300000nM Q9NPD8 28437106 201 QRASRLKRELHMLATEPPPGITCWQDKDQMDDLRAQILGGANTPYEKGVFKLEVIIPERYPFEPPQIRFLTPIYHPNIDSAGRICLDVLKLPPKGAWRPSLNIATVLTSIQLLMSEPNPDDPLMADISSEFKYNKPAFLKNARQWTEKHARQ 5nhf A 2.14 BS01 8X5 A 1 I31 G34 G37 V39 K54 M108 T110 L156 I20 G23 G26 V28 K43 M97 T99 L145 D149 K151 S153 N154 D167 T190 D138 K140 S142 N143 D156 T179 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50<0.00032uM remove_due_to_license_issue IC50=80nM P28482 28376306 402 EMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDDLPKEKLKELIFEETARFQ 5nhh A 1.94 BS01 8XH A 1 I31 G37 V39 A52 K54 M108 T110 K114 L156 D167 I21 G27 V29 A42 K44 M98 T100 K104 L146 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50<0.00113uM remove_due_to_license_issue IC50=4.8nM P28482 28376306 404 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY 5nhj A 2.12 BS01 8XE A 1 I31 G37 V39 A52 K54 M108 E109 D111 L156 C166 D167 I21 G27 V29 A42 K44 M98 E99 D101 L146 C156 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.00539uM remove_due_to_license_issue IC50=1600nM P28482 28376306 403 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQ 5nhl A 2.07 BS01 8XB A 1 G34 G37 V39 A52 K54 M108 K114 L156 D167 G24 G27 V29 A42 K44 M98 K104 L146 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50<0.0003uM remove_due_to_license_issue IC50=<0.300000nM P28482 28376306 402 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQ 5nho A 2.24 BS01 8XN A 1 I31 G37 V39 A52 K54 M108 T110 D111 L156 C166 D167 I21 G27 V29 A42 K44 M98 T100 D101 L146 C156 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50<0.0003uM remove_due_to_license_issue IC50=<0.300000nM P28482 28376306 402 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQ 5nhp A 1.99 BS01 8XK A 1 I31 G37 A52 K54 M108 T110 K114 L156 C166 D167 I21 G27 A42 K44 M98 T100 K104 L146 C156 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.023uM remove_due_to_license_issue IC50=>10000nM P28482 28376306 403 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKLPKEKLKELIFEETARFQ 5nhv A 2.0 BS01 8QB A 1 I31 Y36 A52 K54 M108 T110 L156 C166 D167 I21 Y26 A42 K44 M98 T100 L146 C156 D157 D149 K151 S153 N154 D167 T190 D139 K141 S143 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.0028uM remove_due_to_license_issue IC50=2.8nM P28482 28376306 402 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQ 5nhy A 1.72 BS01 8XT A 1 L9 N33 G34 F72 M81 W117 D119 D120 F124 L7 N31 G32 F70 M79 W115 D117 D118 F122 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=2.3nM remove_due_to_license_issue IC50=2.3nM P36639 28679043 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 5nhz A 1.85 BS03 8XZ A 1 Y67 W87 D120 H196 C221 R228 N233 H263 Y36 W56 D87 H148 C167 R174 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 ic50=4.7uM remove_due_to_license_issue IC50=4700nM Q9K2N0 28445786 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTN 5ni0 A 1.673 BS03 8XW A 1 Y67 W87 D120 H196 C221 H263 Y36 W56 D87 H148 C167 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 ic50=1.8uM remove_due_to_license_issue IC50=1800nM Q9K2N0 28445786 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTN 5ni5 A 2.3 BS02 8YB A 1 Q286 L287 C320 H323 L324 R364 M365 R367 A368 V376 F377 F378 F388 I400 F401 Q29 L30 C63 H66 L67 R107 M108 R110 A111 V119 F120 F121 F131 I143 F144 ? 0003677,0004879,0005634,0006355 ic50=0.009uM remove_due_to_license_issue IC50=10.0nM, EC50=8.0nM, Ki=40nM P51449 30095900 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5ni7 A 2.45 BS02 8Y8 A 1 Q286 L287 H323 R364 M365 R367 A368 V376 F377 F378 F388 I397 I400 F401 Q29 L30 H66 R107 M108 R110 A111 V119 F120 F121 F131 I140 I143 F144 ? 0003677,0004879,0005634,0006355 ic50=0.02uM remove_due_to_license_issue IC50=20nM P51449 30095900 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5ni8 A 1.94 BS02 8Y2 A 1 Q286 L287 C320 H323 R364 M365 R367 A368 F377 F378 F388 I400 F401 Q29 L30 C63 H66 R107 M108 R110 A111 F120 F121 F131 I143 F144 ? 0003677,0004879,0005634,0006355 ic50=0.02uM remove_due_to_license_issue IC50=20nM P51449 30095900 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5nib A 1.82 BS02 8Y5 A 1 Q286 L287 C320 H323 L324 M358 R364 M365 R367 A368 F377 F378 F388 L391 I397 I400 F401 H479 Q29 L30 C63 H66 L67 M101 R107 M108 R110 A111 F120 F121 F131 L134 I140 I143 F144 H222 ? 0003677,0004879,0005634,0006355 ic50=0.019uM remove_due_to_license_issue IC50=19nM P51449 30095900 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 5nih A 1.3 BS01 8VE A 1 E13 Y61 P89 T91 R96 L138 G141 S142 T143 E193 M196 E13 Y61 P89 T91 R96 L138 G141 S142 T143 E193 M196 ? 0015276,0016020 Ki=134nM remove_due_to_license_issue P19491 28691798 304 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 5niy A 1.7 BS01 GNP A 1 N302 G303 G305 T307 T308 R333 T446 K447 D449 G472 E475 N106 G107 G109 T111 T112 R137 T250 K251 D253 G276 E279 3.6.5.4 0005525,0006614,0016887 remove_due_to_license_issue P10121 30146170 601 ARLKRSLLKTKENLGSGFISLFRGKKIDDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFARE 5nj8 A 3.3 BS01 dna E 0 R40 D65 K66 R7 D32 K33 ? 0006355,0006805,0009410,0046983 remove_due_to_license_issue P35869 28602820 1 ~ 12 NPSKRHRDRLNTELDRLASLLPFPQDVINKLDKLSVLRLSVSYLRAKSFFDVALKGLNLQEGEFLLQALNGFVLVVTTDALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQLHWPPENSPLMERCFICRLRCLLDSSGFLAMNFQGKLKYLHGQKPQLALFAIATPL 5nj8 A 3.3 BS02 dna F 0 R38 H39 R42 R5 H6 R9 ? 0006355,0006805,0009410,0046983 remove_due_to_license_issue P35869 28602820 1 ~ 12 NPSKRHRDRLNTELDRLASLLPFPQDVINKLDKLSVLRLSVSYLRAKSFFDVALKGLNLQEGEFLLQALNGFVLVVTTDALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQLHWPPENSPLMERCFICRLRCLLDSSGFLAMNFQGKLKYLHGQKPQLALFAIATPL 5nj8 B 3.3 BS01 dna E 0 E98 R101 E14 R17 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P27540 28602820 1 ~ 12 DKERLARENHSEIERRRRNKMTAYITELSDMVPTCPDKLTILRMAVSHMKSLRGSYKPSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSSRRSFICRMRCHFVVVHCTGYIKAWPDDDPEAKFCLVAIGRLQV 5nj8 B 3.3 BS02 dna F 0 R88 H94 R102 D127 K128 R4 H10 R18 D37 K38 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P27540 28602820 1 ~ 12 DKERLARENHSEIERRRRNKMTAYITELSDMVPTCPDKLTILRMAVSHMKSLRGSYKPSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSSRRSFICRMRCHFVVVHCTGYIKAWPDDDPEAKFCLVAIGRLQV 5nj8 C 3.3 BS01 dna G 0 R40 N44 D65 K66 R9 N13 D34 K35 ? 0006355,0006805,0009410,0046983 remove_due_to_license_issue P35869 28602820 1 ~ 12 KSNPSKRHRDRLNTELDRLASLLPFPQDVINKLDKLSVLRLSVSYLRAKSFFDVALKREGLNLQEGEFLLQALNGFVLVVTTDALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQENSPLMERCFICRLRCLFLAMNFQGKLKYLHGQKKDGSILPPQLALFAIATP 5nj8 C 3.3 BS02 dna H 0 R38 H39 R42 R7 H8 R11 ? 0006355,0006805,0009410,0046983 remove_due_to_license_issue P35869 28602820 1 ~ 12 KSNPSKRHRDRLNTELDRLASLLPFPQDVINKLDKLSVLRLSVSYLRAKSFFDVALKREGLNLQEGEFLLQALNGFVLVVTTDALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQENSPLMERCFICRLRCLFLAMNFQGKLKYLHGQKKDGSILPPQLALFAIATP 5nj8 D 3.3 BS01 dna G 0 I97 E98 R101 I14 E15 R18 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P27540 28602820 1 ~ 12 ADKERLARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLRGTSTDGSYKPSFLTDQELKHLILEAADFLFYVSDSVTPVQPQSESTLYDSRRSFICRMRCHCTGYIKALVAIGR 5nj8 D 3.3 BS02 dna H 0 H94 R102 D127 K128 H11 R19 D44 K45 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P27540 28602820 1 ~ 12 ADKERLARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLRGTSTDGSYKPSFLTDQELKHLILEAADFLFYVSDSVTPVQPQSESTLYDSRRSFICRMRCHCTGYIKALVAIGR 5njz A 1.768 BS01 8ZH A 1 A644 I645 K646 E663 I690 T692 Y694 M695 G698 L746 A38 I39 K40 E57 I84 T86 Y88 M89 G92 L140 D739 A741 R743 N744 D757 P780 D133 A135 R137 N138 D151 P157 2.7.10.1 0004672,0004713,0005524,0006468 Kd=16.6nM remove_due_to_license_issue P29317 28544567 1001 FTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nk2 A 1.649 BS01 8ZZ A 1 I619 A644 I645 K646 E663 I690 T692 M695 G698 L746 I22 A42 I43 K44 E61 I88 T90 M93 G96 L144 D739 A741 R743 N744 D757 D766 P780 D137 A139 R141 N142 D155 D164 P174 2.7.10.1 0004672,0004713,0005524,0006468 Kd=0.182uM remove_due_to_license_issue P29317 28544567 1001 NQAVLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nk3 A 1.586 BS01 92Q A 1 I619 A644 I645 K646 M667 I690 T692 Y694 M695 G698 A699 L746 I19 A40 I41 K42 M63 I86 T88 Y90 M91 G94 A95 L142 D739 A741 R743 N744 D757 D766 P780 D135 A137 R139 N140 D153 D162 P173 2.7.10.1 0004672,0004713,0005524,0006468 Kd=38.02nM remove_due_to_license_issue P29317 28544567 1001 VLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFD 5nk4 A 1.45 BS01 90E A 1 I619 A644 I645 K646 E663 I690 T692 Y694 M695 E696 N697 G698 L746 I19 A38 I39 K40 E57 I84 T86 Y88 M89 E90 N91 G92 L140 D739 A741 R743 N744 D757 D766 P780 D133 A135 R137 N138 D151 D160 P174 2.7.10.1 0004672,0004713,0005524,0006468 Kd=1.995nM remove_due_to_license_issue P29317 28544567 1001 VLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTSGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nk6 A 1.267 BS01 90W A 1 A644 K646 E663 I690 T692 Y694 M695 G698 L746 A35 K37 E54 I81 T83 Y85 M86 G89 L137 D739 A741 R743 N744 D757 D766 P780 D130 A132 R134 N135 D148 D157 P168 2.7.10.1 0004672,0004713,0005524,0006468 Kd=0.158uM remove_due_to_license_issue P29317 28544567 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nk7 A 1.889 BS01 8ZZ A 1 I619 A644 I645 K646 E663 I690 T692 Y694 M695 G698 L746 I16 A36 I37 K38 E55 I82 T84 Y86 M87 G90 L138 D739 A741 R743 N744 D757 D766 P780 D131 A133 R135 N136 D149 D158 P168 2.7.10.1 0004672,0004713,0005524,0006468 Kd=0.468nM remove_due_to_license_issue P29317 28544567 1001 FTTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nk8 A 1.761 BS01 90Z A 1 I619 A644 K646 I690 T692 M695 E696 G698 E706 L746 S756 I15 A36 K38 I82 T84 M87 E88 G90 E98 L138 S148 D739 A741 R743 N744 D757 P780 D131 A133 R135 N136 D149 P152 2.7.10.1 0004672,0004713,0005524,0006468 Kd=0.229uM remove_due_to_license_issue P29317 28544567 1001 TTEIHPSCVTRQKVIGGEVYKGMLKTSSGKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIR 5nk9 A 1.588 BS01 912 A 1 I619 A644 K646 E663 I690 T692 Y694 M695 G698 K702 L746 I15 A35 K37 E54 I81 T83 Y85 M86 G89 K93 L137 D739 A741 R743 N744 D757 D766 P780 D130 A132 R134 N135 D148 D157 P169 2.7.10.1 0004672,0004713,0005524,0006468 Kd=0.724uM remove_due_to_license_issue P29317 28544567 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nka A 1.377 BS01 91H A 1 K617 I619 A644 I645 K646 E663 I690 T692 Y694 M695 G698 L746 K13 I15 A40 I41 K42 E59 I86 T88 Y90 M91 G94 L142 D739 A741 R743 N744 D757 P780 D135 A137 R139 N140 D153 P158 2.7.10.1 0004672,0004713,0005524,0006468 Kd=3.47uM remove_due_to_license_issue P29317 28544567 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKTSSGKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDVSIRL 5nkb A 1.5 BS01 8ZT A 1 I619 A644 K646 E663 I690 T692 M695 E696 G698 L746 S756 I15 A35 K37 E54 I81 T83 M86 E87 G89 L137 S147 D739 A741 R743 N744 D757 D766 P780 D130 A132 R134 N135 D148 D157 P169 2.7.10.1 0004672,0004713,0005524,0006468 Kd=0.759nM remove_due_to_license_issue P29317 28544567 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nkc A 1.448 BS01 90T A 1 I619 A644 K646 E663 I690 T692 Y694 M695 G698 L746 I19 A39 K41 E58 I85 T87 Y89 M90 G93 L141 D739 A741 R743 N744 D757 D766 P780 D134 A136 R138 N139 D152 D161 P170 2.7.10.1 0004672,0004713,0005524,0006468 Kd=18.62nM remove_due_to_license_issue P29317 28544567 1001 VLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nkd A 1.408 BS01 91K A 1 K617 I619 A644 K646 E663 I690 T692 Y694 M695 G698 L746 K18 I20 A39 K41 E58 I85 T87 Y89 M90 G93 L141 D739 A741 R743 N744 D757 D766 P780 D134 A136 R138 N139 D152 D161 P171 2.7.10.1 0004672,0004713,0005524,0006468 Kd=26.3nM remove_due_to_license_issue P29317 28544567 1001 AVLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nkg A 1.1 BS01 8ZK A 1 I619 A644 K646 E663 I690 T692 Y694 M695 E696 N697 G698 L746 I15 A40 K42 E59 I86 T88 Y90 M91 E92 N93 G94 L142 D739 A741 R743 N744 D757 D766 P780 D135 A137 R139 N140 D153 D162 P176 2.7.10.1 0004672,0004713,0005524,0006468 Kd=20.89nM remove_due_to_license_issue P29317 28544567 1001 TTEIHPSCVTRQKVIGAGEFGEVYKGMLKTSSGKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTSGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nkh A 1.29 BS01 8ZQ A 1 I619 G620 A644 K646 I690 T692 Y694 M695 E696 G698 L746 I19 G20 A44 K46 I90 T92 Y94 M95 E96 G98 L146 D739 A741 R743 N744 D757 D766 P780 D139 A141 R143 N144 D157 D166 P180 2.7.10.1 0004672,0004713,0005524,0006468 Kd=25.7nM remove_due_to_license_issue P29317 28544567 1001 VLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKTSSGKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSRVLEDDPEATYTTSGGKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRL 5nki A 1.675 BS01 8ZW A 1 A644 K646 E663 I690 T692 M695 E696 G698 L746 A36 K38 E55 I82 T84 M87 E88 G90 L138 D739 A741 R743 N744 D757 P780 D131 A133 R135 N136 D149 P152 2.7.10.1 0004672,0004713,0005524,0006468 Kd=18.62nM remove_due_to_license_issue P29317 28544567 1001 FTTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLP 5nkk F 2.64 BS01 GDP F 1 Q95 G98 K99 S100 T101 P122 K241 E284 Q37 G40 K41 S42 T43 P64 K153 E196 ? 0000184 remove_due_to_license_issue Q9XWJ1 28389433 401 MKESVRFLTDFGEISDAISDLLTSSPNFNVISAIGPQGAGKSTLLSMLAGNNSRQMYREYVFRPVSTIQIDIYIVNHQIFLDCDDSTAMSDTLRLTAFLLYVSHTVLVVSETHYDKVIIDTLRVAEQIRPYLAIFRPKLAIDRKTNLVFIKTKASSIDLAPTVIREREELLRLSFQDSRWLKVSQEPFKTLIVLEEFDEQIAELREELQKNREDFTVETAAMDEKKWLDMCREVIRDKTLHKTLKEYQRAMTD 5nkn A 2.2 BS01 LOC A 1 F41 F68 K70 F71 W106 F134 F37 F64 K66 F67 W102 F130 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 Kd=120pM remove_due_to_license_issue P80188 30517073 201 SDLIPAPPLSKVPLQQNFQDNQFHGKWYVVGVAGNGFLREDKDPIKMAATIYELKEDKSYNVTFQKFPMKKCQYMTDTLVPGSQPGEFTLGNIKSEPGYTSWLVRVVSTNYNQHAMVFFKAVQQNREDFFITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCI 5nlk A 1.8 BS01 92E A 1 P1106 L1109 P1110 Q1113 V1115 L1120 N1168 R1173 V1174 P24 L27 P28 Q31 V33 L38 N86 R91 V92 2.3.1.-,2.3.1.48 Kd=0.035uM remove_due_to_license_issue Kd=35nM, IC50=19nM Q92793 29532017 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5nn0 A 2.1 BS03 92H A 1 L236 V294 G296 M302 L234 V292 G294 M300 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 Kd=11.1pM remove_due_to_license_issue IC50=1.0nM P06276 29227101 626 DIIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5nn0 A 2.1 BS04 92H A 2 I69 D70 W82 G116 G117 W231 L286 F329 Y332 I67 D68 W80 G114 G115 W229 L284 F327 Y330 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 Kd=11.1pM remove_due_to_license_issue IC50=1.0nM P06276 29227101 627 DIIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 5nn4 A 1.83 BS01 SC2 A 1 H432 G435 R436 R437 H339 G342 R343 R344 3.2.1.20 0000023,0002026,0002086,0003007,0003824,0004553,0004558,0005764,0005765,0005886,0005975,0005977,0005980,0005985,0006006,0006941,0007040,0007626,0009888,0016020,0016798,0030246,0035577,0035904,0043181,0043202,0043231,0046716,0050884,0050885,0060048,0061723,0070062,0070821,0090599,0101003,0120282 Kd=11.57mM remove_due_to_license_issue P10253 29061980 1016 QCDVPPNSRFDCAPDKAITQEQCEARGCCYIPAKQGQPWCFFPPSYPSYKLENLSSSEMGYTATLTRTTPTFFPKDILTLRLDVMMETENRLHFTIKDPANRRYEVPLETAPSPLYSVEFSEEPFGVIVHRQLDGRVLLNTTVAPLFFADQFLQLSTSLPSQYITGLAEHLSPLMLSTSWTRITLWNRDLAPTPGANLYGSHPFYLALEDGGSAHGVFLLNSNAMDVVLQPSPALSWRSTGGILDVYIFLGPEPKSVVQQYLDVVGYPFMPPYWGLGFHLCRWGYSSTAITRQVVENMTRAHFPLDVQWNDLDYMDSRRDFTFNKDGFRDFPAMVQELHQGGRRYMMIVDPAISSSGPAGSYRPYDEGLRRGVFITNETGQPLIGKVWPGSTAFPDFTNPTALAWWEDMVAEFHDQVPFDGMWIDMNEPSNFIRGSEDGCPNNELENPPYVPGVVGGTLQAATICASSHQFLSTHYNLHNLYGLTEAIASHRALVKARGTRPFVISRSTFAGHGRYAGHWTGDVWSSWEQLASSVPEILQFNLLGVPLVGADVCGFLGNTSEELCVRWTQLGAFYPFMRNHNSLLSLPQEPYSFSEPAQQAMRKALTLRYALLPHLYTLFHQAHVAGETVARPLFLEFPKDSSTWTVDHQLLWGEALLITPVLQAGKAEVTGYFPLGTWYDLQTVPIEREPAIHSEGQWVTLPAPLDTINVHLRAGYIIPLQGPGLTTTESRQQPMALAVALTKGGEARGELFWDDGESLEVLERGAYTQVIFLARNNTIVNELVRVTSEGAGLQLQKVTVLGVATAPQQVLSNGVPVSNFTYSPDTKVLDICVSLLMGEQFLVSWC 5nn4 A 1.83 BS02 SC2 A 2 H742 Q757 H649 Q664 3.2.1.20 0000023,0002026,0002086,0003007,0003824,0004553,0004558,0005764,0005765,0005886,0005975,0005977,0005980,0005985,0006006,0006941,0007040,0007626,0009888,0016020,0016798,0030246,0035577,0035904,0043181,0043202,0043231,0046716,0050884,0050885,0060048,0061723,0070062,0070821,0090599,0101003,0120282 Kd=11.57mM remove_due_to_license_issue P10253 29061980 1017 QCDVPPNSRFDCAPDKAITQEQCEARGCCYIPAKQGQPWCFFPPSYPSYKLENLSSSEMGYTATLTRTTPTFFPKDILTLRLDVMMETENRLHFTIKDPANRRYEVPLETAPSPLYSVEFSEEPFGVIVHRQLDGRVLLNTTVAPLFFADQFLQLSTSLPSQYITGLAEHLSPLMLSTSWTRITLWNRDLAPTPGANLYGSHPFYLALEDGGSAHGVFLLNSNAMDVVLQPSPALSWRSTGGILDVYIFLGPEPKSVVQQYLDVVGYPFMPPYWGLGFHLCRWGYSSTAITRQVVENMTRAHFPLDVQWNDLDYMDSRRDFTFNKDGFRDFPAMVQELHQGGRRYMMIVDPAISSSGPAGSYRPYDEGLRRGVFITNETGQPLIGKVWPGSTAFPDFTNPTALAWWEDMVAEFHDQVPFDGMWIDMNEPSNFIRGSEDGCPNNELENPPYVPGVVGGTLQAATICASSHQFLSTHYNLHNLYGLTEAIASHRALVKARGTRPFVISRSTFAGHGRYAGHWTGDVWSSWEQLASSVPEILQFNLLGVPLVGADVCGFLGNTSEELCVRWTQLGAFYPFMRNHNSLLSLPQEPYSFSEPAQQAMRKALTLRYALLPHLYTLFHQAHVAGETVARPLFLEFPKDSSTWTVDHQLLWGEALLITPVLQAGKAEVTGYFPLGTWYDLQTVPIEREPAIHSEGQWVTLPAPLDTINVHLRAGYIIPLQGPGLTTTESRQQPMALAVALTKGGEARGELFWDDGESLEVLERGAYTQVIFLARNNTIVNELVRVTSEGAGLQLQKVTVLGVATAPQQVLSNGVPVSNFTYSPDTKVLDICVSLLMGEQFLVSWC 5nn5 A 2.0 BS01 NOJ A 1 W376 D404 L405 D518 R600 W613 D616 F649 H674 W283 D311 L312 D425 R507 W520 D523 F556 H581 3.2.1.20 0000023,0002026,0002086,0003007,0003824,0004553,0004558,0005764,0005765,0005886,0005975,0005977,0005980,0005985,0006006,0006941,0007040,0007626,0009888,0016020,0016798,0030246,0035577,0035904,0043181,0043202,0043231,0046716,0050884,0050885,0060048,0061723,0070062,0070821,0090599,0101003,0120282 Ki=3.4uM remove_due_to_license_issue P10253 29061980 1016 QCDVPPNSRFDCAPDKAITQEQCEARGCCYIPAKQGQPWCFFPPSYPSYKLENLSSSEMGYTATLTRTTPTFFPKDILTLRLDVMMETENRLHFTIKDPANRRYEVPLETAPSPLYSVEFSEEPFGVIVHRQLDGRVLLNTTVAPLFFADQFLQLSTSLPSQYITGLAEHLSPLMLSTSWTRITLWNRDLAPTPGANLYGSHPFYLALEDGGSAHGVFLLNSNAMDVVLQPSPALSWRSTGGILDVYIFLGPEPKSVVQQYLDVVGYPFMPPYWGLGFHLCRWGYSSTAITRQVVENMTRAHFPLDVQWNDLDYMDSRRDFTFNKDGFRDFPAMVQELHQGGRRYMMIVDPAISSSGPAGSYRPYDEGLRRGVFITNETGQPLIGKVWPGSTAFPDFTNPTALAWWEDMVAEFHDQVPFDGMWIDMNEPSNFIRGSEDGCPNNELENPPYVPGVVGGTLQAATICASSHQFLSTHYNLHNLYGLTEAIASHRALVKARGTRPFVISRSTFAGHGRYAGHWTGDVWSSWEQLASSVPEILQFNLLGVPLVGADVCGFLGNTSEELCVRWTQLGAFYPFMRNHNSLLSLPQEPYSFSEPAQQAMRKALTLRYALLPHLYTLFHQAHVAGETVARPLFLEFPKDSSTWTVDHQLLWGEALLITPVLQAGKAEVTGYFPLGTWYDLQTVPIEEPAIHSEGQWVTLPAPLDTINVHLRAGYIIPLQGPGLTTTESRQQPMALAVALTKGGEARGELFWDDGESLEVLERGAYTQVIFLARNNTIVNELVRVTSEGAGLQLQKVTVLGVATAPQQVLSNGVPVSNFTYSPDTKVLDICVSLLMGEQFLVSWC 5nn6 A 2.0 BS01 MIG A 1 W376 D404 L405 W481 D518 M519 R600 W613 D616 F649 H674 W281 D309 L310 W386 D423 M424 R505 W518 D521 F554 H579 3.2.1.20 0000023,0002026,0002086,0003007,0003824,0004553,0004558,0005764,0005765,0005886,0005975,0005977,0005980,0005985,0006006,0006941,0007040,0007626,0009888,0016020,0016798,0030246,0035577,0035904,0043181,0043202,0043231,0046716,0050884,0050885,0060048,0061723,0070062,0070821,0090599,0101003,0120282 Ki=3uM remove_due_to_license_issue IC50=2000nM P10253 29061980 1013 QCDVPPNSRFDCAPDKAITQEQCEARGCCYIPAKQGQPWCFFPPSYPSYKLENLSSSEMGYTATLTRTTPTFFPKDILTLRLDVMMETENRLHFTIKDPANRRYEVPLAPSPLYSVEFSEEPFGVIVHRQLDGRVLLNTTVAPLFFADQFLQLSTSLPSQYITGLAEHLSPLMLSTSWTRITLWNRDLAPTPGANLYGSHPFYLALEDGGSAHGVFLLNSNAMDVVLQPSPALSWRSTGGILDVYIFLGPEPKSVVQQYLDVVGYPFMPPYWGLGFHLCRWGYSSTAITRQVVENMTRAHFPLDVQWNDLDYMDSRRDFTFNKDGFRDFPAMVQELHQGGRRYMMIVDPAISSSGPAGSYRPYDEGLRRGVFITNETGQPLIGKVWPGSTAFPDFTNPTALAWWEDMVAEFHDQVPFDGMWIDMNEPSNFIRGSEDGCPNNELENPPYVPGVVGGTLQAATICASSHQFLSTHYNLHNLYGLTEAIASHRALVKARGTRPFVISRSTFAGHGRYAGHWTGDVWSSWEQLASSVPEILQFNLLGVPLVGADVCGFLGNTSEELCVRWTQLGAFYPFMRNHNSLLSLPQEPYSFSEPAQQAMRKALTLRYALLPHLYTLFHQAHVAGETVARPLFLEFPKDSSTWTVDHQLLWGEALLITPVLQAGKAEVTGYFPLGTWYDLQTVPIEREPAIHSEGQWVTLPAPLDTINVHLRAGYIIPLQGPGLTTTESRQQPMALAVALTKGGEARGELFWDDGESLEVLERGAYTQVIFLARNNTIVNELVRVTSEGAGLQLQKVTVLGVATAPQQVLSNGVPVSNFTYSPDTKVLDICVSLLMGEQFLVSWC 5nob A 1.85 BS01 92T A 1 S1033 F1035 I1039 F1044 D1045 H1048 Y1060 Y1071 I1075 S82 F84 I88 F93 D94 H97 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=0.0063uM remove_due_to_license_issue IC50=6.3nM Q9H2K2 29155568 1301 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSMAHSPPGHHSVTGRPLALAEYVIYRGEQAYPEYLITYQIMRPE 5npb A 1.9 BS03 93Z A 1 F271 D299 F377 W410 D412 R463 W477 D480 F513 H540 F234 D262 F340 W373 D375 R426 W440 D443 F476 H503 2.4.1.161 0003824,0004553,0005975,0016757,0030246,0033825 remove_due_to_license_issue B3PEE6 28776021 907 AVFYKEHKLRNDGLVITTNQGNIRLQFKSEAAIEVLYRADSKQLPSFALAQPESAIKAQLTETENHLQFSGGTLTARIQKRPFAISYYRDSELLLAEESGFQVKINFRFYLSPGEKILGGGQRILGMDRRGQRFPLYNRAHYGYSDHSGQMYFGLPAIMSSKQYILVFDNSASGAMDIGKTESDILQLEAKSGRSAYILVAGNSYPSLIENFTQVTGRQPLPPRWALGSFASRFGYRSEAETRATVQKYKTEDFPLDTIVLDLYWFGKDIKGHMGNLDWDKENFPTPLDMMADFKQQGVKTVLITEPFVLTSSKRWDDAVKAKALAKDPQGQPKAFELYFGNGGIIDVFSKEGSRWFSSIYKDLSKQGVAGWWGDLGEPEMHPEDTQHAIGDADTVHNAYGHRWAEMLYQQQLDQFPELRPFIMMRAGFVGSQRYGMIPWTGDVSRTWGGLASQVELALQMSLLGFGYIHSDLGGFADGETLDKEMYIRWLQYGVFQPVYRPHGQDHIPSEPVFQDEETKAILRPLVKLRYRMLPYIYTAAYQNTLTGMPLMRPLFFSDEKNPALIDNKTSYFWGDSLLVTPITQAGVESVSIPAPKGVWFDFWKDTRYQTDGAPLTLPTDLHTIPVLVKAGAFMPYVPAVSTTEDYRSDSLEIHYYADASVPLAQGEIFEDDGKDPNSIKRNQFDLLTLQATHTDNQLHFQLARTGKGYRGMPERRATTLVIHNASDQYQHLDINGKTIAIAQADCASTPALACYDQERRQLQLVFTWGREALNLRLHK 5npc A 1.96 BS06 94E A 1 F271 D299 W410 N412 R463 D480 F513 H540 F234 D262 W373 N375 R426 D443 F476 H503 2.4.1.161 0003824,0004553,0005975,0016757,0030246,0033825 remove_due_to_license_issue B3PEE6 28776021 922 AVFYKEHKLRNDGLVITTNQGNIRLQFKSEAAIEVLYRADSKQLPSFALAQPESAIKAQLTETENHLQFSGGTLTARIQKRPFAISYYRDSELLLAEESGFQVKINFRFYLSPGEKILGGGQRILGMDRRGQRFPLYNRAHYGYSDHSGQMYFGLPAIMSSKQYILVFDNSASGAMDIGKTESDILQLEAKSGRSAYILVAGNSYPSLIENFTQVTGRQPLPPRWALGSFASRFGYRSEAETRATVQKYKTEDFPLDTIVLDLYWFGKDIKGHMGNLDWDKENFPTPLDMMADFKQQGVKTVLITEPFVLTSSKRWDDAVKAKALAKDPQGQPKAFELYFGNGGIIDVFSKEGSRWFSSIYKDLSKQGVAGWWGNLGEPEMHPEDTQHAIGDADTVHNAYGHRWAEMLYQQQLDQFPELRPFIMMRAGFVGSQRYGMIPWTGDVSRTWGGLASQVELALQMSLLGFGYIHSDLGGFADGETLDKEMYIRWLQYGVFQPVYRPHGQDHIPSEPVFQDEETKAILRPLVKLRYRMLPYIYTAAYQNTLTGMPLMRPLFFSDEKNPALIDNKTSYFWGDSLLVTPITQAGVESVSIPAPKGVWFDFWKDTRYQTDGAPLTLPTDLHTIPVLVKAGAFMPYVPAVSTTEDYRSDSLEIHYYADASVPLAQGEIFEDDGKDPNSIKRNQFDLLTLQATHTDNQLHFQLARTGKGYRGMPERRATTLVIHNASDQYQHLDINGKTIAIAQADCASTPALACYDQERRQLQLVFTWGREALNLRLHK 5npd A 1.95 BS05 94B A 1 F271 D299 N412 R463 D480 F513 H540 F234 D262 N375 R426 D443 F476 H503 2.4.1.161 0003824,0004553,0005975,0016757,0030246,0033825 remove_due_to_license_issue B3PEE6 28776021 915 AVFYKEHKLRNDGLVITTNQGNIRLQFKSEAAIEVLYRADSKQLPSFALAQPESAIKAQLTETENHLQFSGGTLTARIQKRPFAISYYRDSELLLAEESGFQVKINFRFYLSPGEKILGGGQRILGMDRRGQRFPLYNRAHYGYSDHSGQMYFGLPAIMSSKQYILVFDNSASGAMDIGKTESDILQLEAKSGRSAYILVAGNSYPSLIENFTQVTGRQPLPPRWALGSFASRFGYRSEAETRATVQKYKTEDFPLDTIVLDLYWFGKDIKGHMGNLDWDKENFPTPLDMMADFKQQGVKTVLITEPFVLTSSKRWDDAVKAKALAKDPQGQPKAFELYFGNGGIIDVFSKEGSRWFSSIYKDLSKQGVAGWWGNLGEPEMHPEDTQHAIGDADTVHNAYGHRWAEMLYQQQLDQFPELRPFIMMRAGFVGSQRYGMIPWTGDVSRTWGGLASQVELALQMSLLGFGYIHSDLGGFADGETLDKEMYIRWLQYGVFQPVYRPHGQDHIPSEPVFQDEETKAILRPLVKLRYRMLPYIYTAAYQNTLTGMPLMRPLFFSDEKNPALIDNKTSYFWGDSLLVTPITQAGVESVSIPAPKGVWFDFWKDTRYQTDGAPLTLPTDLHTIPVLVKAGAFMPYVPAVSTTEDYRSDSLEIHYYADASVPLAQGEIFEDDGKDPNSIKRNQFDLLTLQATHTDNQLHFQLARTGKGYRGMPERRATTLVIHNASDQYQHLDINGKTIAIAQADCASTPALACYDQERRQLQLVFTWGREALNLRLHK 5npe A 1.95 BS04 948 A 1 F271 D299 W410 D412 R463 W477 D480 F513 H540 F234 D262 W373 D375 R426 W440 D443 F476 H503 2.4.1.161 0003824,0004553,0005975,0016757,0030246,0033825 remove_due_to_license_issue B3PEE6 28776021 910 AVFYKEHKLRNDGLVITTNQGNIRLQFKSEAAIEVLYRADSKQLPSFALAQPESAIKAQLTETENHLQFSGGTLTARIQKRPFAISYYRDSELLLAEESGFQVKINFRFYLSPGEKILGGGQRILGMDRRGQRFPLYNRAHYGYSDHSGQMYFGLPAIMSSKQYILVFDNSASGAMDIGKTESDILQLEAKSGRSAYILVAGNSYPSLIENFTQVTGRQPLPPRWALGSFASRFGYRSEAETRATVQKYKTEDFPLDTIVLDLYWFGKDIKGHMGNLDWDKENFPTPLDMMADFKQQGVKTVLITEPFVLTSSKRWDDAVKAKALAKDPQGQPKAFELYFGNGGIIDVFSKEGSRWFSSIYKDLSKQGVAGWWGDLGEPEMHPEDTQHAIGDADTVHNAYGHRWAEMLYQQQLDQFPELRPFIMMRAGFVGSQRYGMIPWTGDVSRTWGGLASQVELALQMSLLGFGYIHSDLGGFADGETLDKEMYIRWLQYGVFQPVYRPHGQDHIPSEPVFQDEETKAILRPLVKLRYRMLPYIYTAAYQNTLTGMPLMRPLFFSDEKNPALIDNKTSYFWGDSLLVTPITQAGVESVSIPAPKGVWFDFWKDTRYQTDGAPLTLPTDLHTIPVLVKAGAFMPYVPAVSTTEDYRSDSLEIHYYADASVPLAQGEIFEDDGKDPNSIKRNQFDLLTLQATHTDNQLHFQLARTGKGYRGMPERRATTLVIHNASDQYQHLDINGKTIAIAQADCASTPALACYDQERRQLQLVFTWGREALNLRLHK 5npf A 1.38 BS02 945 A 1 E441 Y445 D452 H507 Y523 T591 D593 E777 R786 E403 Y407 D414 H469 Y485 T553 D555 E739 R748 3.2.1.45 0004348,0004553,0005975,0006680,0008422,0016020,0016798,0046872 remove_due_to_license_issue F6BL85 28776021 915 DKISHKIDIPDSAWTIGIGEKFKNAGHPNVKYPMIDDSYVQGAPLGGFGAGTIGRTYNGGFSRWHLEIGKNKYTTVYANQFSVFQKVEGNKDGVAQVLYAGEPGYLSSWKWDYPKESGMYYALYPNSWYTYTNKDLPVQLAVKQFSPIIPYNYKETSYPVAVFKWTAYNPTNKNVDVSIMFTWQNMIGFFGKQVNVNSGNFNKIIKDKSEIVAAVMGNISNDNEEWNGEYSIGVKKVPGVDISYKAKFVTTGDGSDLWHEFSKNGILDNKDDETPTKQDGIGSAIAVNFKLQPGQTIEVPFALSWDLPIMKFGGGDKWYKMYTKYFGKNGKNSFAILKEALNNYQKWEKMIDDWQKPILSNKSKPDWYKTALFNELYYLADGGTAWENGKVGERTNNMFGLLECFDYNYYETLDVRFYGSFPLVMLWPDIEKQVMRQFADTINVQDSSEFKVGSNGAMAVKKVQGMIPHDLGSSYALPWIKINAYDWQNPNIWKDLNSKYVLLVYRDYVLTGKTDKEFLKYTWKSVKTALDKLKEMDKDNDGIPDNEGIPDQTYDTWSMKGTSAYCGSLWLAALKAAQEIGKVLKDNEAYIKYNEWYKIAQQNFEKELWNGEYYNFDTESDHKDSIMADQLAGQWYADILRLGDILPKDHVQKALKKIYEFNVMKFENGKMGAVNGMRPDGIVDESDIQAQEVWTGVTYALASFMKYRGMTEEAYNTAYGVYKMTYDKSGKGYWFRTPEAWTKDGNYRASMYMRPLSIWSMEV 5npr A 1.85 BS02 94T E 1 Q839 K842 L866 V895 A896 K898 H901 H920 T921 T922 D925 Q506 K509 L533 V562 A563 K565 H568 H587 T588 T589 D592 2.4.1.255 0006493,0016757 remove_due_to_license_issue O15294 29723473 101 THADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMI 5nps A 1.68 BS02 94T D 1 H496 P559 T633 Q839 K842 L866 V895 A896 K898 H901 H920 T921 T922 D925 H183 P246 T320 Q506 K509 L533 V561 A562 K564 H567 H586 T587 T588 D591 2.4.1.255 0006493,0016757 remove_due_to_license_issue O15294 29723473 101 PTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMI 5nq5 A 2.85 BS01 952 A 1 F36 L52 M66 F70 R74 R95 N100 Y103 R107 F36 L52 M66 F70 R74 R95 N100 Y103 R107 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 remove_due_to_license_issue P9WKE1 29510037 301 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLARDNYERDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAPPDV 5nqe A 2.71 BS01 94Z A 1 H1682 G1683 Y1714 F1715 A1716 Y1721 S1722 Y1727 G1751 N1752 H1753 T1774 L1782 H71 G72 Y93 F94 A95 Y100 S101 Y106 G130 N131 H132 T153 L161 2.4.2.- 0003950 remove_due_to_license_issue Q460N5 28495083 1901 MKQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 5nqr A 2.2 BS01 958 A 1 W28 R51 D60 G61 W15 R38 D47 G48 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 ic50=70nM remove_due_to_license_issue Q9UKK9 29343827 301 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nqr A 2.2 BS02 958 A 2 W28 R51 L98 W15 R38 L85 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 ic50=70nM remove_due_to_license_issue Q9UKK9 29343827 302 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nqr A 2.2 BS03 958 A 3 W46 E47 W33 E34 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 ic50=70nM remove_due_to_license_issue Q9UKK9 29343827 303 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nqr B 2.2 BS01 958 A 1 W46 E47 W33 E34 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 remove_due_to_license_issue Q9UKK9 29343827 301 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nqr B 2.2 BS02 958 A 2 W46 E47 W33 E34 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 remove_due_to_license_issue Q9UKK9 29343827 302 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nqr B 2.2 BS03 958 A 3 W28 R51 D60 G61 W15 R38 D47 G48 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 remove_due_to_license_issue Q9UKK9 29343827 303 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nr7 A 2.35 BS01 YUI A 1 P37 L52 H53 F70 R74 R95 S99 N100 Y103 P37 L52 H53 F70 R74 R95 S99 N100 Y103 2.7.4.9 0000287,0004798,0005524,0005525,0005737,0005829,0006227,0006233,0006235,0009165,0016301,0042803,0046044,0046872,0046940 ic50=0.95uM remove_due_to_license_issue P9WKE1 29510037 301 MLIAIEGVDGAGKRTLVEKLSGAFRAAGRSVATLAFPRYGQSVAADIAAEALHGEHGDLASSVYAMATLFALDRAGAVHTIQGLCRGYDVVILDRYVASNAAYSAARLHENAAGKAAAWVQRIEFARLGLPKPDWQVLLAVSAELRDAELQQRTGAVYAELAAQGWGGRWLVVGADVDPGRLAATLAP 5nr8 A 1.349 BS01 95N A 1 Y27 W99 A183 M210 Y212 D213 Y267 T295 M300 M356 W358 Y6 W78 A162 M189 Y191 D192 Y246 T274 M279 M335 W337 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 ic50=175nM remove_due_to_license_issue IC50=175nM Q13231 29283260 401 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEESGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQELSLVPRGSHHHHHH 5nra A 1.267 BS01 95K A 1 Y27 W99 A183 M210 Y212 D213 Y267 T295 M300 M356 W358 Y6 W78 A162 M189 Y191 D192 Y246 T274 M279 M335 W337 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 ic50=123nM remove_due_to_license_issue Q13231 29283260 401 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEESGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQELSLVPRGSHHHHHH 5nrf A 1.447 BS01 95Q A 1 Y27 W99 A183 M210 Y212 D213 Y267 R269 T295 E297 M300 M356 W358 Y6 W78 A162 M189 Y191 D192 Y246 R248 T274 E276 M279 M335 W337 D136 D138 E140 Y212 D115 D117 E119 Y191 3.2.1.14 0004553,0005975,0008061 ic50=163nM remove_due_to_license_issue IC50=163nM Q13231 29283260 401 AKLVCYFTNWAQYRQGEARFLPKDLDPSLCTHLIYAFAGMTNHQLSTTEWNDETLYQEFNGLKKMNPKLKTLLAIGGWNFGTQKFTDMVATANNRQTFVNSAIRFLRKYSFDGLDLDWEYPGSQGSPAVDKERFTTLVQDLANAFQQEAQTSGKERLLLSAAVPAGQTYVDAGYEVDKIAQNLDFVNLMAYDFHGSWEKVTGHNSPLYKRQEESGAAASLNVDAAVQQWLQKGTPASKLILGMPTYGRSFTLASSSDTRVGAPATGSGTPGPFTKEGGMLAYYEVCSWKGATKQRIQDQKVPYIFRDNQWVGFDDVESFKTKVSYLKQKGLGGAMVWALDLDDFAGFSCNQGRYPLIQTLRQELSLVPRGSHHHHHH 5nsp B 2.3 BS02 97E B 1 H1031 S1033 F1035 I1039 F1044 D1045 H1048 A1049 I1051 Y1060 Y1071 I1075 H80 S82 F84 I88 F93 D94 H97 A98 I100 Y109 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=0.34uM remove_due_to_license_issue IC50=>10000nM Q9H2K2 29155568 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 5nsx A 1.8 BS02 97K A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=400nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nt0 A 1.75 BS02 97H A 1 H1031 G1032 S1033 Y1050 Y1060 A1062 S1068 Y1071 I1075 H80 G81 S82 Y99 Y109 A111 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=280nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nt4 A 1.9 BS02 97Z A 1 H1031 G1032 H1048 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 H97 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=17nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5ntk A 1.9 BS01 99N A 1 C285 Q286 L287 M313 W317 M365 R367 L391 C393 H479 C21 Q22 L23 M49 W53 M101 R103 L127 C129 H215 ? 0003677,0004879,0005634,0006355 ic50=9.7nM remove_due_to_license_issue P51449 28590087 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHL 5ntp A 1.7 BS01 98E A 1 L287 H323 M365 A368 V376 F377 F388 S404 H479 F486 L25 H61 M103 A106 V114 F115 F126 S142 H217 F224 ? 0003677,0004879,0005634,0006355 ic50=0.7nM remove_due_to_license_issue P51449 28590087 501 PYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPI 5ntq A 2.26 BS01 444 A 1 W317 C320 H323 L324 V361 M365 V376 F388 I400 H479 W53 C56 H59 L60 V97 M101 V112 F124 I136 H215 ? 0003677,0004879,0005634,0006355 ic50=33.8nM remove_due_to_license_issue IC50=60nM, EC50=54nM, Ki=51nM P51449 28590087 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAF 5ntt A 2.75 BS01 SVE A 1 I531 S537 A551 K553 M602 Y604 G605 N606 D608 S611 L654 I663 I21 S27 A41 K43 M92 Y94 G95 N96 D98 S101 L144 I153 D647 K649 N652 D664 D674 T686 D137 K139 N142 D154 D164 T176 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=182nM P33981 28726638 801 ENLYFQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEYGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTTSVVKDSQVGTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQTHP 5ntw A 1.64 BS03 98N A 1 Q286 L287 W317 C320 R364 M365 R367 A368 F377 F378 F388 L396 I400 H479 Q23 L24 W54 C57 R101 M102 R104 A105 F114 F115 F125 L133 I137 H216 ? 0003677,0004879,0005634,0006355 ic50=0.6nM remove_due_to_license_issue IC50=<100nM, Ki=<100nM P51449 28590087 601 YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFST 5nu1 A 1.85 BS02 8YB A 1 Q286 L287 C320 H323 L324 R364 M365 R367 A368 V376 F377 F378 F388 I400 F401 Q23 L24 C57 H60 L61 R101 M102 R104 A105 V113 F114 F115 F125 I137 F138 ? 0003677,0004879,0005634,0006355 ic50=1nM remove_due_to_license_issue IC50=10.0nM, EC50=8.0nM, Ki=40nM P51449 28590087 601 YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFST 5nu3 A 1.75 BS01 99E A 1 P1110 F1111 V1115 L1120 Y1125 Y1167 N1168 R1173 V1174 P32 F33 V37 L42 Y47 Y89 N90 R95 V96 2.3.1.-,2.3.1.48 Kd=0.23uM remove_due_to_license_issue Q92793 28766825 1201 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5nu5 A 1.6 BS01 99E A 1 L1073 P1074 V1079 L1084 Y1131 N1132 R1137 L28 P29 V34 L39 Y86 N87 R92 2.3.1.-,2.3.1.48 Kd=0.47uM remove_due_to_license_issue Q09472 28766825 1201 SMIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKSPMDLSTIKRKLDTGQYQEPWQYVDDIWLMFNNAWLYNRKTSRVYKYCSKLSEVFEQEIDPVMQSLG 5nud A 2.5 BS01 99K A 1 L473 R483 V550 E551 C552 A553 A554 L619 L21 R29 V96 E97 C98 A99 A100 L150 D612 R616 N617 D630 D143 R147 N148 D161 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 30108871 801 DLPLDPLWEFPRDRLVLGKPLGEGGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGRLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAVSEE 5nut A 1.6 BS02 9A8 A 1 H1031 G1032 P1034 Y1050 Y1060 K1067 S1068 Y1071 I1075 H80 G81 P83 Y99 Y109 K116 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=12nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5nvc A 1.6 BS02 9AN A 1 H1031 G1032 Y1050 Y1060 K1067 S1068 Y1071 I1075 H80 G81 Y99 Y109 K116 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=650nM remove_due_to_license_issue Q9H2K2 29374194 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nve A 1.5 BS02 9AQ A 1 H1031 G1032 Y1050 Y1060 K1067 S1068 Y1071 H80 G81 Y99 Y109 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=35nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM 5nvf A 1.55 BS02 9AW A 1 H1031 G1032 F1035 H1048 A1049 Y1050 Y1060 S1068 Y1071 I1075 H80 G81 F84 H97 A98 Y99 Y109 S117 Y120 I124 2.4.2.-,2.4.2.30 0003950 ic50=16nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nvh A 1.6 BS02 9B2 A 1 H1031 G1032 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=15nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nvv C 2.1 BS01 9BT C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=105nM remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nvw C 2.2 BS01 9BW C 1 R69 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 R8 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=132nM remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nvx C 2.2 BS01 4YY C 1 R69 W88 Y98 I109 H110 S111 Y112 H115 W117 R8 W27 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=44nM remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nvy C 2.9 BS01 9B5 C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue IC50=21200nM P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nvz C 2.7 BS01 9BN C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQ 5nw0 C 2.3 BS01 9BK C 1 R69 W88 Y98 I109 H110 S111 Y112 H115 W117 R8 W27 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=128nM remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nw1 C 2.1 BS01 9BH C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=210nM remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nw2 C 2.2 BS01 9B8 C 1 R69 W88 Y98 I109 H110 S111 Y112 H115 W117 R8 W27 Y37 I48 H49 S50 Y51 H54 W56 ? Kd=232nM remove_due_to_license_issue P40337 28853884 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 5nw5 A 6.502 BS01 dna C 0 K319 K451 K135 K267 ? remove_due_to_license_issue P29539 28604726 1 ~ 30 ETRVNPRALEYWVSGEIHGLVDNESVSEFKEIIEGGLGILRQESEDYVARRFEVYATFNNIIPILTTKNVNEVDQKFNILIVNIESIIEICIPHLQIAQDTLLSSSEKKNPFVIRLYVQIVRFFSAIMSNFKIVKWLTKRPDLVNKLKVIYRWTTGALRNENSNKIIITAQVSFLRDEKFGTFFLSNEEIKPIISTFTEIMEINSHNLIYEKLLLIRGFLSKYPKLMIETVTSWLPGEVLPRIIIGDEIYSMKILITSIVVLLELLKKCLDFVDEHERIYQCIMLSPVCETIPEKFLSKLPLNSYDSANLDKVTIGHLLTQQIKNYIVVKNDNKIAMDLWLSMTGLLYDSGKRVYDLTSESNKVWFDLNNLCFINNHPKTRLMSIKVWRIITYCICTKISQKNQEGNKSLLSLLRTPFQMTLPYVNDPSAREGIIYHLLGVVYTAFTSNKNLSTDMFELFWDHLITPIYEDYVFKYDSIHLQNVLFTVLHLLIGGKNADVALERKHIHPMSVIASEGVKLKDISSLPPQIIKREYDKIMKVVFQAVEVAISNVNLAHDLILTSLKHLPEDRKDQTHLESFSSLILKVTQNNKDTPIFRDFFGAVTSSFVYTFLDLFLRKNDSSLVNFNIQISKVGISQGNMTLDLLKDVIRKARNETSEFLIIEKFLELDDKKTEVYAQNWVGSTLLPPNISFREFQSLANIVNKVPNENSIENFLDLCLKLSFPVNLFTLLHVSMWSNNNFIYFIQSYVSKNENKLNVDLITLLKTSLPGNPELFSGLLPFLRRNKFMDILEYCIHSNPNLLNSIPDLNSDLLLKLLPRSRASYFAANIKLFKCSEQLTLVRWLLKGQQLEQLNQNFSEIENVLQNASDSELEKSEIIRELLHLAMANPIEPLFSGLLNFCIKNNMADHLDEFCGNMTSEVLFKISPELLLKLLTYKEKPNGKLLAAVIEKIENGDDDYILELLEKIIIQKEIQILEKLKEPLLVFFLNPVSSNMQKHKKSTNMLRELVLLYLTKPLSRSAAKKFFSMLISILPPNPNYQTIDMVNLLIDLIKSHNRKFKDKRTYNATLKTIGKWIQESGVVHQ 5nw5 B 6.502 BS01 dna C 0 K1203 S1206 R1207 S1208 K1016 S1019 R1020 S1021 ? remove_due_to_license_issue P29539 28604726 1 ~ 30 ETRVNPRALEYWVSGEIHGLVDNESVSEFKEIIEGGLGILRQESEDYVARRFEVYATFNNIIPILTTKNVNEVDQKFNILIVNIESIIEICIPHLQIAQDTLLSSSEKKNPFVIRLYVQIVRFFSAIMSNFKIVKWLTKRPDLVNKLKVIYRWTTGALRNENSNKIIITAQVSFLRDEKFGTFFLSNEEIKPIISTFTEIMEINSHNLIYEKLLLIRGFLSKYPKLMIETVTSWLPGEVLPRIIIGDEIYSMKILITSIVVLLELLKKCLDFVDEHERIYQCIMLSPVCETIPEKFLSKLPLNSYDSANLDKVTIGHLLTQQIKNYIVVKNDNKIAMDLWLSMTGLLYDSGKRVYDLTSESNKVWFDLNNLCFINNHPKTRLMSIKVWRIITYCICTKISQKNQEGNKSLLSLLRTPFQMTLPYVNDPSAREGIIYHLLGVVYTAFTSNKNLSTDMFELFWDHLITPIYEDYVFKYDSIHLQNVLFTVLHLLIGGKNADVALEKKHIHPMSVIASEGVKLKDISSLPPQIIKREYDKIMKVVFQAVEVAISNVNLAHDLILTSLKHLPEDRKDQTHLESFSSLILKVTQNNKDTPIFRDFFGAVTSSFVYTFLDLFLRKNDSSLVNFNIQISKVGISQGNMTLDLLKDVIRKARNETSEFLIIEKFLELDDKKTEVYAQNWVGSTLLPPNISFREFQSLANIVNKVPNENSIENFLDLCLKLSFPVNLFTLLHVSMWSNNNFIYFIQSYVSKNENKLNVDLITLLKTSLPGNPELFSGLLPFLRRNKFMDILEYCIHSNPNLLNSIPDLNSDLLLKLLPRSRASYFAANIKLFKCSEQLTLVRWLLKGQQLEQLNQNFSEIENVLQNASDSELEKSEIIRELLHLAMANPIEPLFSGLLNFCIKNNMADHLDEFCGNMTSEVLFKISPELLLKLLTYKEKPNGKLLAAVIEKIENGDDDYILELLEKIIIQKEIQILEKLKEPLLVFFLNPVSSNMQKHKKSTNMLRELVLLYLTKPLSRSAAKKFFSMLISILPPNPNYQTIDMVNLLIDLIKSHNRKFKDKRTYNATLKTIGKWIQESGVVHQ 5nw7 A 1.85 BS02 9C2 A 1 W18 E48 K100 L108 S109 Q111 H113 K136 E138 H285 Y287 E294 K310 W17 E47 K99 L107 S108 Q110 H112 K135 E137 H284 Y286 E293 K309 5.3.1.8 0000032,0004476,0005575,0005737,0005829,0005975,0006486,0008270,0009298,0016853,0031505,0046872 Ki=1.7uM remove_due_to_license_issue P34948 29687459 502 SSEKLFRIQCGYQNYDWGKIGSSSAVAQFVHNSDPSITIDETKPYAELWMGTHPSVPSKAIDLNNQTLRDLVTAKPQEYLGESIITKFGSSKELPFLFKVLSIEKVLSIQAHPDKKLGAQLHAADPKNYPDDNHKPEMAIAVTDFEGFCGFKPLDQLAKTLATVPELNEIIGQELVDEFISGIKLPAEVGSQDDVNNRKLLQKVFGKLMNTDDDVIKQQTAKLLERTDREPQVFKDIDSRLPELIQRLNKQFPNDIGLFCGCLLLNHVGLNKGEAMFLQAKDPHAYISGDIIECMAASDNVVRAGFTPKFKDVKNLVEMLTYSYESVEKQKMPLQEFPRSKGDAVKSVLYDPPIAEFSVLQTIFDKSKGGKQVIEGLNGPSIVIATNGKGTIQITGDDSTKQKIDTGYVFFVAPGSSIELTADSANQDQDFTTYRAFVEA 5nwb A 1.6 BS02 9C5 A 1 H1031 G1032 H1048 A1049 Y1050 Y1060 K1067 S1068 Y1071 H80 G81 H97 A98 Y99 Y109 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=16nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nwc A 1.5 BS02 9CE A 1 H1031 G1032 Y1050 Y1060 K1067 S1068 Y1071 H80 G81 Y99 Y109 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=700nM remove_due_to_license_issue Q9H2K2 29374194 1204 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nwd A 1.45 BS01 9C8 A 1 H1031 G1032 F1035 H1048 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 F84 H97 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=10nM remove_due_to_license_issue Q9H2K2 29374194 1201 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSA 5nwe A 2.0 BS03 G39 A 1 E119 D151 R152 I223 E277 R293 R368 Y402 E38 D70 R71 I142 E196 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Kd=13200nM remove_due_to_license_issue C3W6G3 29933553 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYYYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTIDK 5nwg A 1.4 BS02 9CB A 1 H1031 G1032 F1035 Y1050 Y1060 K1067 S1068 Y1071 H80 G81 F84 Y99 Y109 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=660nM remove_due_to_license_issue Q9H2K2 29374194 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFS 5nwh A 2.6 BS01 9CH A 1 W28 R51 R84 L98 I141 W15 R38 R71 L85 I128 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 remove_due_to_license_issue Q9UKK9 29343827 301 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nwh A 2.6 BS02 9CH A 2 W46 E47 W33 E34 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 remove_due_to_license_issue Q9UKK9 29343827 302 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nwh B 2.6 BS01 9CH A 2 W28 R51 I141 W15 R38 I128 2.7.7.96,3.6.1.13,3.6.1.58 0000287,0003723,0005515,0005634,0005829,0006139,0006338,0006753,0009117,0009191,0016462,0016740,0016779,0016787,0017110,0019144,0019303,0019693,0030515,0042802,0042803,0044715,0044716,0046872,0047631,0055086,0070062,0140933,1990966 remove_due_to_license_issue Q9UKK9 29343827 302 KQYIISEELISEGKWVKLEKTTYMDPTGKTRTWESVKRTTRKEQTADGVAVIPVLQRTLHYECIVLVKQFRPPMGGYCIEFPAGLIDDGETPEAAALRELEEETGYKGDIAECSPAVCMDPGLSNCTIHIVTVTINGDDAENARPKPKPGDGEFVEVISLPKNDLLQRLDALVAEEHLTVDARVYSYALALKHAN 5nwz A 2.37 BS01 9CT A 1 L473 G474 C477 A501 K503 E520 M524 I534 V550 A553 G556 N557 L619 D630 F631 L20 G21 C24 A48 K50 E67 M71 I81 V97 A100 G103 N104 L156 D167 F168 D612 R616 N617 D630 D149 R153 N154 D167 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 30108871 801 LPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPDLPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAVSE 5nx9 A 2.3 BS01 AMP A 1 R85 H86 D87 S112 Q241 L331 S334 A335 R338 R77 H78 D79 S104 Q233 L317 S320 A321 R324 H86 T158 H159 K295 E302 H78 T150 H151 K281 E288 4.3.2.2 0000166,0003824,0004018,0005829,0006164,0006189,0009152,0009168,0016829,0044208,0070626 remove_due_to_license_issue A0A384E0N4 30573755 503 SPDSYRSPLASRYASPEMCFVFSDRYKFRTWRQLWLWLAEAEQTLGLPITDEQIQEMKSNLENIDFKMAAEEEKRLRHDVMAHVHTFGHCCPKAAGIIHLGATSCYVGDNTDLIILRNALDLLLPKLARVISRLADFAKERASLPTLGFTHFQPAQLTTVGKRCCLWIQDLCMDLQNLKRVRDDLRFRGVKGTTGTQASFLQLFEGDDHKVEQLDKMVTEKAGFKRAFIITGQTYTRKVDIEVLSVLASLGASVHKICTDIRLLANLKEMEEPFEKQQIGKRNPMRSERCCSLARHLMTLVMDPLQTASVQWFERTLDDSANRRICLAEAFLTADTILNTLQNISEGLVVYPKVIERRIRQELPFMATENIIMAMVKAGGSRQDCHEKIRVLSQQAASVVKQEGGDNDLIERIQADAYFSPIHSQLDHLLDPSSFTGRASQQVQRFLEEEVYPLLKPYESVMKVKA 5nx9 A 2.3 BS04 AMP D 1 R20 Y21 R303 R12 Y13 R289 H86 T158 H159 K295 E302 H78 T150 H151 K281 E288 4.3.2.2 0000166,0003824,0004018,0005829,0006164,0006189,0009152,0009168,0016829,0044208,0070626 remove_due_to_license_issue A0A384E0N4 30573755 502 SPDSYRSPLASRYASPEMCFVFSDRYKFRTWRQLWLWLAEAEQTLGLPITDEQIQEMKSNLENIDFKMAAEEEKRLRHDVMAHVHTFGHCCPKAAGIIHLGATSCYVGDNTDLIILRNALDLLLPKLARVISRLADFAKERASLPTLGFTHFQPAQLTTVGKRCCLWIQDLCMDLQNLKRVRDDLRFRGVKGTTGTQASFLQLFEGDDHKVEQLDKMVTEKAGFKRAFIITGQTYTRKVDIEVLSVLASLGASVHKICTDIRLLANLKEMEEPFEKQQIGKRNPMRSERCCSLARHLMTLVMDPLQTASVQWFERTLDDSANRRICLAEAFLTADTILNTLQNISEGLVVYPKVIERRIRQELPFMATENIIMAMVKAGGSRQDCHEKIRVLSQQAASVVKQEGGDNDLIERIQADAYFSPIHSQLDHLLDPSSFTGRASQQVQRFLEEEVYPLLKPYESVMKVKA 5nx9 D 2.3 BS01 AMP A 1 R20 Y21 R303 R13 Y14 R296 H86 T158 H159 S290 K295 E302 H79 T151 H152 S283 K288 E295 4.3.2.2 0000166,0003824,0004018,0005829,0006164,0006189,0009152,0009168,0016829,0044208,0070626 remove_due_to_license_issue A0A384E0N4 30573755 503 GSPDSYRSPLASRYASPEMCFVFSDRYKFRTWRQLWLWLAEAEQTLGLPITDEQIQEMKSNLENIDFKMAAEEEKRLRHDVMAHVHTFGHCCPKAAGIIHLGATSCYVGDNTDLIILRNALDLLLPKLARVISRLADFAKERASLPTLGFTHFQPAQLTTVGKRCCLWIQDLCMDLQNLKRVRDDLRFRGVKGTTGTQASFLQLFEGDDHKVEQLDKMVTEKAGFKRAFIITGQTYTRKVDIEVLSVLASLGASVHKICTDIRLLANLKEMEEPFEKQQIGSSAMPYKRNPMRSERCCSLARHLMTLVMDPLQTASVQWFERTLDDSANRRICLAEAFLTADTILNTLQNISEGLVVYPKVIERRIRQELPFMATENIIMAMVKAGGSRQDCHEKIRVLSQQAASVVKQEGGDNDLIERIQADAYFSPIHSQLDHLLDPSSFTGRASQQVQRFLEEEVYPLLKPYESVMKVKAELCL 5nx9 D 2.3 BS04 AMP D 1 R85 H86 D87 S112 Q241 L331 S334 A335 R338 R78 H79 D80 S105 Q234 L324 S327 A328 R331 H86 T158 H159 S290 K295 E302 H79 T151 H152 S283 K288 E295 4.3.2.2 0000166,0003824,0004018,0005829,0006164,0006189,0009152,0009168,0016829,0044208,0070626 remove_due_to_license_issue A0A384E0N4 30573755 502 GSPDSYRSPLASRYASPEMCFVFSDRYKFRTWRQLWLWLAEAEQTLGLPITDEQIQEMKSNLENIDFKMAAEEEKRLRHDVMAHVHTFGHCCPKAAGIIHLGATSCYVGDNTDLIILRNALDLLLPKLARVISRLADFAKERASLPTLGFTHFQPAQLTTVGKRCCLWIQDLCMDLQNLKRVRDDLRFRGVKGTTGTQASFLQLFEGDDHKVEQLDKMVTEKAGFKRAFIITGQTYTRKVDIEVLSVLASLGASVHKICTDIRLLANLKEMEEPFEKQQIGSSAMPYKRNPMRSERCCSLARHLMTLVMDPLQTASVQWFERTLDDSANRRICLAEAFLTADTILNTLQNISEGLVVYPKVIERRIRQELPFMATENIIMAMVKAGGSRQDCHEKIRVLSQQAASVVKQEGGDNDLIERIQADAYFSPIHSQLDHLLDPSSFTGRASQQVQRFLEEEVYPLLKPYESVMKVKAELCL 5nxg A 1.2 BS02 RA1 A 1 Q92 H94 H119 F131 L198 T199 T200 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.8nM remove_due_to_license_issue P00918 29316128 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxi A 1.16 BS02 9DE A 1 H94 H119 F131 L198 T199 T200 H93 H118 F129 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=217.4nM remove_due_to_license_issue P00918 29316128 302 AHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxo A 1.2 BS02 9HK A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=4.9nM remove_due_to_license_issue P00918 29316128 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxo A 1.2 BS03 9HK A 2 H3 W5 H10 N11 H15 W16 D19 H1 W3 H8 N9 H13 W14 D17 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=4.9nM remove_due_to_license_issue P00918 29316128 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxp A 1.25 BS02 9DH A 1 Q92 H94 H119 F131 L198 T199 T200 P202 Q90 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=10.2nM remove_due_to_license_issue P00918 29316128 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxv A 1.1 BS02 9E2 A 1 H94 H119 F131 L198 T199 T200 H92 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.5nM remove_due_to_license_issue P00918 29316128 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxw A 1.1 BS02 RA9 A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=57.4nM remove_due_to_license_issue P00918 29316128 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxw A 1.1 BS03 RA9 A 2 H4 W5 N11 H15 D19 H1 W2 N8 H12 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=57.4nM remove_due_to_license_issue P00918 29316128 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nxx C 2.2 BS01 3Q7 C 1 S25 G26 I27 W72 W178 W225 T229 H230 S18 G19 I20 W65 W171 W218 T222 H223 ? 0005886,0006865,0022857,0043190,0045121,0055085 remove_due_to_license_issue P46922 29159878 301 ASAAEQVNKTIIGIDPGSGIMSLTDKAMKDYDLNDWTLISASSAAMTATLKKSYDRKKPIIITGWTPHWMFSRYKLKYLDDPKQSYGSAEEIHTITRKGFSKEQPNAAKLLSQFKWTQDEMGEIMIKVEEGEKPAKVAAEYVNKHKDQIAEWTKGVQKVKGDKINLAYVAWDSEIASTNVIGKVLEDLGYEVTLTQVEAGPMWTAIATGSADASLSAWLPNTHKAYAAKYKGKYDDIGTSMTGVKMGLVVPQYMKNVNSIEDLKK 5nxy A 1.9 BS01 1Y8 A 1 D66 N107 Y109 Y189 Y213 D63 N104 Y106 Y186 Y210 ? 0005886,0006865,0022857,0043190,0055085 remove_due_to_license_issue Q45462 29159878 301 QTIKIGAQSMSESEIIASMQGQLIEHHTDLKTTTIKNLGSNAVQQQALMNGEIDIAATRYTGDALTGTLRMEPEKDPDKALALTQREFKKRYDLKWYDSYGFDNTYAFTVSKELADQYHLETVSDVKKWAPQLKLGVDNYWMKLKGNGYQDFTKTYGMTFGGTYPMQIGLVYDAVKSGKMDIVLAYSTDGRIKSYGLKMLKDDKQFFPPYDCSPVVPEKVLKEHPELEGIIKKMLGKIDTATMQELNYEVDGNLKEPSVVAKEYLEKHRYFE 5ny1 A 1.1 BS02 9E5 A 1 H94 H119 F131 L198 T199 T200 P202 H91 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=366.7nM remove_due_to_license_issue P00918 29316128 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ny3 A 1.4 BS02 9E8 A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=33.9nM remove_due_to_license_issue P00918 29316128 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ny6 A 1.1 BS03 R92 A 1 P155 Q158 K159 P152 Q155 K156 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=13.5nM remove_due_to_license_issue P00918 29316128 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nya A 1.2 BS02 FB2 A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=415.6nM remove_due_to_license_issue Ki=1103nM, Kd=1149700nM P00918 29316128 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5nyh A 1.65 BS01 9EK A 1 N51 A55 D93 G97 M98 L107 F138 T184 N36 A40 D78 G82 M83 L92 F123 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=18.7nM remove_due_to_license_issue P07900 29701469 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5nyz A 2.5 BS01 DUP A 1 G78 I80 D81 Y84 G89 G78 I80 D81 Y84 G89 A25 R64 G66 L73 D81 A25 R64 G66 L73 D81 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 remove_due_to_license_issue A4ZF98 28894239 201 MTNTLQVKLLSKNARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNEHEDDKMQTIFLRNIDNEKIFEKERHLYKLGSYRIEKGERIAQLVIVPIWTPELKQVEEFESVERGEKGFGSS 5nz2 A 2.85 BS01 DUP A 1 G78 D81 Y84 G89 G77 D80 Y83 G88 A25 R64 G66 L73 D81 A24 R63 G65 L72 D80 3.6.1.23 0000287,0004170,0006226,0009117,0016787,0046081,0046872 remove_due_to_license_issue A4ZF98 28894239 201 TNTLQVKLLSKNARMPERNHKTDAGYDIFSAETVVLEPQEKAVIKTDVAVSIPEGYVGLLTSRSGVSSKTHLVIETGKIDAGYHGNLGINIKNEHEDDKMQTIFLRNIDNEKIFEKERHLYKLGSYRIEKGERIAQLVIVPIWTPELKQVEEFES 5nz4 B 1.36 BS03 G39 B 1 R118 E119 D151 R152 R225 E277 R293 N295 R368 Y402 R37 E38 D70 R71 R144 E196 R212 N214 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Kd=520nM remove_due_to_license_issue C3W6G3 29933553 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNVLRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 5nze B 1.69 BS03 G39 B 1 R118 E119 D151 R152 R225 E277 R293 R368 Y402 R37 E38 D70 R71 R144 E196 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Kd=410nM remove_due_to_license_issue C3W6G3 29933553 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPNNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 5nzf A 1.75 BS03 G39 A 1 E119 D151 R152 W179 E277 R293 R368 Y402 E38 D70 R71 W98 E196 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=94000nM remove_due_to_license_issue C3W6G3 29933553 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNVLRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYYYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 5nzm A 2.35 BS01 9ET A 1 R248 R373 R243 R368 2.7.7.9 0003983,0005737,0005829,0005977,0006011,0016779,0031981,0070569,0097014 remove_due_to_license_issue Q4QDU3 601 KSLSAAAQACVKKMRDAKVNEACIRTFIAQHVMVSKGETGSIPDSAIMPVDSLDALDSLTIECDNAVLQSTVVLKLNGGLGTGMGLCDAKTLLEVKDGKTFLDFTALQVQYLRQHCSEHLRFMLMDSFNTSASTKSFLKARYPWLYQVFDSEVELMQNQVPKILQDTLEPAAWAENPAYEWAPPGHGDIYTALYGSGKLQELVEQGYRYMFVSNGDNLGATIDKRVLAYMEKEKIDFLMEVCRRTESDKKGGHLARQTVYVKGKDGQPDAEKRVLLLRESAQCPKADMESFQDINKYSFFNTNNLWIRLPVLLETMQEHGGTLPLPVIRNEKTVDSSNSASPKVYQLETAMGAAIAMFESASAIVVPRSRFAPVKTCADLLALRSDAYVVTDDFRLVLDDRCHGHPPVVDLDSAHYKMMNGFEKLVQHGVPSLVECKRVTVKGLVQFGAGNVLTGTVTIENTDSASAFVIPDGAKLNDTTASP 5nzn A 1.73 BS03 G39 A 1 R118 E119 D151 R152 W179 E277 R293 R368 Y402 R37 E38 D70 R71 W98 E196 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=220000nM remove_due_to_license_issue C3W6G3 29933553 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPNNGQASYKIFRIEKGKIVKSVEMNAPNYYYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 5nzo B 1.29 BS01 9EZ B 1 Y174 P176 T207 P208 T213 Y75 P77 T108 P109 T114 N102 R236 D260 E265 H283 N3 R137 D161 E166 H184 1.1.1.37,1.1.1.399,1.1.1.95 0051287 remove_due_to_license_issue Kd=5800000nM O43175 29568346 301 NGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSR 5nzp B 1.3 BS01 9EW B 1 Y174 P176 T207 S212 T213 Y75 P77 T108 S113 T114 N102 R236 D260 E265 H283 N3 R137 D161 E166 H184 1.1.1.37,1.1.1.399,1.1.1.95 0051287 Kd=6.5mM remove_due_to_license_issue Kd=6500000nM O43175 29568346 301 NGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSR 5nzq B 1.5 BS01 5AO B 1 Y174 P176 T207 P208 L216 Y75 P77 T108 P109 L117 N102 R236 D260 E265 H283 N3 R137 D161 E166 H184 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 remove_due_to_license_issue Kd=9300000nM O43175 29568346 401 NGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSR 5o07 A 1.8 BS02 1VQ A 1 Q92 H94 H96 V121 L198 T199 T200 Q89 H91 H93 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=33.8nM remove_due_to_license_issue Ki=34nM P00918 28738704 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 5o0a A 1.805 BS01 9FH A 1 T14 G16 H17 R90 T118 Y122 S126 S127 T14 G16 H17 R90 T118 Y122 S126 S127 H17 R90 S127 H17 R90 S127 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 Kd=0.58mM remove_due_to_license_issue B1MDL6 28648615 201 MTGAVCPGSFDPVTLGHLDVFERAAAQFDEVIVAVLINPNKAGMFTVDERIEMIRESTADLPNLRVESGQGLLVDFVRERGLNAIVKGLRTGTDFEYELQMAQMNKHIAGVDTFFVATAPAYSFVSSSLAKEVATYGGDVSALLPASVHQRLLGKLR 5o0a B 1.805 BS01 9FH B 1 T14 G16 H17 R90 T118 Y122 V125 S126 S127 T14 G16 H17 R88 T116 Y120 V123 S124 S125 H17 R90 S127 H17 R88 S125 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 Kd=0.58mM remove_due_to_license_issue B1MDL6 28648615 201 MTGAVCPGSFDPVTLGHLDVFERAAAQFDEVIVAVLINPAGMFTVDERIEMIRESTADLPNLRVESGQGLLVDFVRERGLNAIVKGLRTGTDFEYELQMAQMNKHIAGVDTFFVATAPAYSFVSSSLAKEVATYGGDVSALLPASVHQRLLGKLR 5o0b A 1.735 BS01 9FE A 1 G8 S9 F10 H17 V20 G88 G8 S9 F10 H17 V20 G88 H17 R90 S127 H17 R90 S127 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 Kd=66uM remove_due_to_license_issue B1MDL6 28648615 201 MTGAVCPGSFDPVTLGHLDVFERAAAQFDEVIVAVLINPNKAGMFTVDERIEMIRESTADLPNLRVESGQGLLVDFVRERGLNAIVKGLRTGTDFEYELQMAQMNKHIAGVDTFFVATAPAYSFVSSSLAKEVATYGGDVSALLPASVHQRLLGKLR 5o0b A 1.735 BS02 9FE A 2 G16 H17 G88 R90 S126 S127 G16 H17 G88 R90 S126 S127 H17 R90 S127 H17 R90 S127 2.7.7.3 0003824,0004595,0005524,0005737,0009058,0015937,0016779 Kd=66uM remove_due_to_license_issue B1MDL6 28648615 202 MTGAVCPGSFDPVTLGHLDVFERAAAQFDEVIVAVLINPNKAGMFTVDERIEMIRESTADLPNLRVESGQGLLVDFVRERGLNAIVKGLRTGTDFEYELQMAQMNKHIAGVDTFFVATAPAYSFVSSSLAKEVATYGGDVSALLPASVHQRLLGKLR 5o0j A 1.81 BS01 8BR A 1 E198 N295 H345 T346 Y347 V431 V432 P435 I441 E194 N291 H341 T342 Y343 V427 V428 P431 I437 2.7.1.-,2.7.1.147 0000287,0004340,0005737,0005975,0006006,0006096,0016301,0016773,0043843,0046872,0051156 Kd=16.85uM remove_due_to_license_issue O58328 29784881 501 TNWESLYEKALDKVEASIRKVRGVLLAYNTNIDAIKYLKREDLEKRIEKVGKEEVLRYSEELPKEIETIPQLLGSILWSIKRGKAAELLVVSREVREYMRKWGWDELRMGGQVGIMANLLGGVYGIPVIAHVPQLSELQASLFLDGPIYVPTFERGELRLIHPREFRKGEEDCIHYIYEFPRNFKVLDFEAPRENRFIGAADDYNPILYVREEWIERFEEIAKRSELAIISGLHPLTQENHGKPIKLVREHLKILNDLGIRAHLEFAFTPDEVVRLEIVKLLKHFYSVGLNEVELASVVSVMGEKELAERIISKDPADPIAVIEGLLKLIKETGVKRIHFHTYGYYLALTREKGEHVRDALLFSALAAATKAMKGNIEKLSDIREGLAVPIGEQGLEVEKILEKEFSLRDGIGSIEDYQLTFIPTKVVKKPKSTVGIGDTISSSAFVSEFSLH 5o0j A 1.81 BS02 8BR A 2 W82 R86 K88 F272 W78 R82 K84 F268 2.7.1.-,2.7.1.147 0000287,0004340,0005737,0005975,0006006,0006096,0016301,0016773,0043843,0046872,0051156 Kd=16.85uM remove_due_to_license_issue O58328 29784881 502 TNWESLYEKALDKVEASIRKVRGVLLAYNTNIDAIKYLKREDLEKRIEKVGKEEVLRYSEELPKEIETIPQLLGSILWSIKRGKAAELLVVSREVREYMRKWGWDELRMGGQVGIMANLLGGVYGIPVIAHVPQLSELQASLFLDGPIYVPTFERGELRLIHPREFRKGEEDCIHYIYEFPRNFKVLDFEAPRENRFIGAADDYNPILYVREEWIERFEEIAKRSELAIISGLHPLTQENHGKPIKLVREHLKILNDLGIRAHLEFAFTPDEVVRLEIVKLLKHFYSVGLNEVELASVVSVMGEKELAERIISKDPADPIAVIEGLLKLIKETGVKRIHFHTYGYYLALTREKGEHVRDALLFSALAAATKAMKGNIEKLSDIREGLAVPIGEQGLEVEKILEKEFSLRDGIGSIEDYQLTFIPTKVVKKPKSTVGIGDTISSSAFVSEFSLH 5o0s A 1.16 BS02 9FQ A 1 E441 Y445 D452 H507 Y523 T591 D593 E777 R786 E408 Y412 D419 H474 Y490 T558 D560 E744 R753 3.2.1.45 0004348,0004553,0005975,0006680,0008422,0016020,0016798,0046872 remove_due_to_license_issue F6BL85 28776021 911 DKISHKIDIPDSAWTIGIGEKFKNAGHPNVKYPMIDDSYVQGAPLGGFGAGTIGRTYNGGFSRWHLEIGKNKYTTVYANQFSVFQKVEGNKDGVAQVLYAGEPENGYLSSWKWDYPKESGMYYALYPNSWYTYTNKDLPVQLAVKQFSPIIPYNYKETSYPVAVFKWTAYNPTNKNVDVSIMFTWQNMIGFFGKQVNVNSGNFNKIIKDKSKDSEIVAAVMGNISNDNEEWNGEYSIGVKKVPGVDISYKAKFVTTGDGSDLWHEFSKNGILDNKDDETPTKQDGIGSAIAVNFKLQPGQTIEVPFALSWDLPIMKFGGGDKWYKMYTKYFGKNGKNSFAILKEALNNYQKWEKMIDDWQKPILSNKSKPDWYKTALFNELYYLADGGTAWENGKVGERTNNMFGLLECFDYNYYETLDVRFYGSFPLVMLWPDIEKQVMRQFADTINVQDSSEFKVGSNGAMAVKKVQGMIPHDLGSSYALPWIKINAYDWQNPNIWKDLNSKYVLLVYRDYVLTGKTDKEFLKYTWKSVKTALDKLKEMDKDNDGIPDNEGIPDQTYDTWSMKGTSAYCGSLWLAALKAAQEIGKVLKDNEAYIKYNEWYKIAQQNFEKELWNGEYYNFDTESDHKDSIMADQLAGQWYADILRLGDILPKDHVQKALKKIYEFNVMKFENGKMGAVNGMRPDGIVDESDIQAQEVWTGVTYALASFMKYRGMTEEAYNTAYGVYKMTYDKSGKGYWFRTPEAWTKDGNYRASMYMRPLSIWSMEV 5o11 A 2.4 BS01 3NG A 1 L44 G45 S46 V52 A65 K67 R122 L174 I185 D186 L11 G12 S13 V17 A30 K32 R87 L139 I150 D151 D167 K169 N172 D186 L193 T204 D132 K134 N137 D151 L158 T169 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 ic50=0.216uM remove_due_to_license_issue IC50=48nM P11309 29042609 401 LESQYQVGPLLGSGGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 5o1a A 1.44 BS02 9H5 A 1 L145 V147 T150 P151 C220 E221 P222 P223 T230 L50 V52 T55 P56 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=30uM remove_due_to_license_issue Kd=30000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5o1b A 1.43 BS02 9H2 A 1 L145 V147 T150 C220 E221 P222 P223 T230 L50 V52 T55 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=20uM remove_due_to_license_issue Kd=20000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 5o1c A 1.32 BS02 9GZ A 1 L145 V147 T150 P151 C220 E221 P222 P223 T230 L50 V52 T55 P56 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=113uM remove_due_to_license_issue Kd=113000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 5o1d A 1.36 BS02 9GW A 1 L145 V147 T150 P151 C220 E221 P223 T230 L50 V52 T55 P56 C125 E126 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=22uM remove_due_to_license_issue Kd=22000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 5o1e A 1.3 BS02 9GT A 1 L145 V147 T150 P151 C220 E221 P223 T230 L50 V52 T55 P56 C125 E126 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=33uM remove_due_to_license_issue Kd=33000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 5o1f A 1.38 BS02 9GQ A 1 L145 V147 T150 P151 C220 E221 P223 T230 L50 V52 T55 P56 C125 E126 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=30uM remove_due_to_license_issue Kd=30000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5o1g A 1.35 BS02 9GK A 1 L145 V147 T150 P151 P153 V157 C220 E221 P223 T230 L50 V52 T55 P56 P58 V62 C125 E126 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=116uM remove_due_to_license_issue Kd=116000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5o1h A 1.32 BS02 9GN A 1 L145 V147 T150 P151 C220 P223 T230 L50 V52 T55 P56 C125 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=14uM remove_due_to_license_issue Kd=14000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5o1i A 1.4 BS02 9GH A 1 L145 V147 T150 P152 V157 C220 E221 P222 P223 T230 L50 V52 T55 P57 V62 C125 E126 P127 P128 T135 ? 0000976,0003677,0003700,0005634,0006355,0006915 Kd=4uM remove_due_to_license_issue Kd=4000nM P04637 29702446 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 5o1s A 1.9 BS01 9HB A 1 C599 W602 C177 W180 D539 K541 N544 D561 D120 K122 N125 D142 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P18654 30341347 802 SIQFTDGYEVKEDISVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCNFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNR 5o1s A 1.9 BS02 9HB A 2 C436 A449 K451 C17 A30 K32 D539 K541 N544 D561 D120 K122 N125 D142 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue P18654 30341347 803 SIQFTDGYEVKEDISVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCNFVAPEVLERQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNR 5o22 A 2.1 BS01 C3R A 1 Y50 K54 I232 P260 G261 G264 P265 Y44 K48 I226 P254 G255 G258 P259 1.5.1.5,3.5.4.9 0000105,0003824,0004477,0004488,0005829,0006164,0006730,0009086,0016491,0016787,0035999,0042803 Kd=10nM remove_due_to_license_issue P24186 29142318 301 AAKIIDGKTIAQQVRSEVAQKVQARIAAGLRAPGLAVVLVGSNYVASKRKACEEVGFVSRSYDLPETTSEAELLELIDTLNADNTIDGILVQLPLPAGIDNVKVLERIHPDKDVDGFHPYNVGRLCQRAPRLRPCTPRGIVTLLERYNIDTFGLNAVVIGASNIVGRPMSMELLLAGCTTTVTHRFTKNLRHHVENADLLIVAVGKPGFIPGDWIKEGAIVIDVGINRLENGKVVGDVVFEDAAKRASYITPVPGGVGPMTVATLIENTLQACVEYHDPQ 5o2d A 1.6 BS01 9HH A 1 V1032 F1129 P1130 A1131 I1132 G1133 F1144 I1148 N1178 F1182 V31 F128 P129 A130 I131 G132 F143 I147 N177 F181 2.4.2.- remove_due_to_license_issue IC50=900nM, Kd=2100nM Q460N5 28991428 1201 SWEKGSLVSPGGLQMLLVKEGVQNAKTDVVVNSVPLDLVLSRGPLSSSLLEKAGPELQEELDTVGQGVAVSMGTVLKTSSWNLDCRYVLHVVAPEWRNGSTSSLKIMEDIIRECMEITESLSLKSIAFPAIGTGNLGFPKNIFAELIISEVFSFSSSNQLSTLQEVHFLLHPSDHENIQAFSDEFARRA 5o3q A 1.75 BS01 CMP A 1 G31 Y32 T33 L65 G30 Y31 T32 L52 ? 0005886,0006808,0009579,0030234,0031676 Kd=2.1uM remove_due_to_license_issue P73954 29735650 200 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGSDIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGCS 5o3q A 1.75 BS02 CMP B 1 V11 G39 K40 N59 A88 G89 I90 V10 G38 K39 N46 A75 G76 I77 ? 0005886,0006808,0009579,0030234,0031676 Kd=2.1uM remove_due_to_license_issue P73954 29735650 201 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGSDIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGCS 5o3q C 1.75 BS01 CMP A 1 V11 K40 N59 A88 I90 V10 K39 N44 A73 I75 ? 0005886,0006808,0009579,0030234,0031676 remove_due_to_license_issue P73954 29735650 200 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGCSAWS 5o3q C 1.75 BS02 CMP B 2 G31 Y32 T33 L65 G30 Y31 T32 L50 ? 0005886,0006808,0009579,0030234,0031676 remove_due_to_license_issue P73954 29735650 202 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGCSAWS 5o3r A 1.9 BS01 AMP A 1 G39 K40 G41 N59 A88 G89 I90 G38 K39 G40 N45 A74 G75 I76 ? 0005886,0006808,0009579,0030234,0031676 Kd=10.1uM remove_due_to_license_issue P73954 29735650 201 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGDIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGC 5o3r A 1.9 BS02 AMP A 2 G31 Y32 T33 L65 H102 G30 Y31 T32 L51 H88 ? 0005886,0006808,0009579,0030234,0031676 Kd=10.1uM remove_due_to_license_issue P73954 29735650 202 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGDIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGC 5o3r B 1.9 BS01 AMP A 1 G31 Y32 T33 I64 L65 H102 G30 Y31 T32 I51 L52 H89 ? 0005886,0006808,0009579,0030234,0031676 remove_due_to_license_issue P73954 29735650 201 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGSDIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGCSAWS 5o3r B 1.9 BS02 AMP C 1 N59 A88 G89 I90 N46 A75 G76 I77 ? 0005886,0006808,0009579,0030234,0031676 remove_due_to_license_issue P73954 29735650 200 AKPANKLVIVTEKILLKKIAKIIDESGAKGYTVMNTGGKGSDIEANIKFEILTETREMAEEIADRVAVKYFNDYAGIIYICSAEVLYGHTFCGPEGCSAWS 5o48 A 1.69 BS02 9K2 A 1 F105 T197 Y211 Y334 N365 A366 L367 L388 L410 F80 T172 Y186 Y309 N340 A341 L342 L363 L385 N161 F162 L163 T197 L410 N136 F137 L138 T172 L385 2.3.1.97 0004379,0005737,0006499,0016746,0046872 remove_due_to_license_issue A5K1A2 29760414 502 IDYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 5o4f B 2.1 BS01 8VE B 1 Y61 P88 T90 R95 A141 T142 E189 Y58 P85 T87 R92 A138 T139 E186 ? 0015276,0016020 Ki=208uM remove_due_to_license_issue P42264 28691798 305 RSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGC 5o4s A 1.75 BS01 9KW A 1 I652 F653 V657 P658 E661 N708 F714 I25 F26 V30 P31 E34 N81 F87 ? ic50=3.4uM remove_due_to_license_issue Kd=2500nM, IC50=3400nM P55201 29902720 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o4t A 1.5 BS01 9KT A 1 V662 Y707 N708 F714 V36 Y81 N82 F88 ? remove_due_to_license_issue IC50=>400000nM P55201 29902720 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o4z A 1.7 BS01 A A 1 H105 H263 S265 R267 G283 G284 H286 G291 H108 H266 S268 R270 G286 G287 H289 G294 ? 0000166,0003676,0046872 remove_due_to_license_issue Q9X1T1 29107484 401 GSGMDEIVKVLSQHDRILVVGHIMPDGDCVSSVLSLTLGLEKLGKEVKAAVDYKIPYVFEKFPYIDKIEENPNFDPELLVVVNASSPDRIGKFQDLLDKVPSVVIDHHSTNTNFGNWNWVDPSFAATAQMIFRINKALGVEYDSNLATLNYLGIATNTGFFRHSNADVRVFEDAYKLVKMGADAHFVAKEILENKRFEQFKLFAEVLERLQLLENGKIAYSYIDYDTYLRHNCTDEDSAGFVGELRSIRGVEVAVLFMEFPRGKIHVSMRSKDWFNVNEVAFELGGGGHPRAAGVTFEGKKIEEVIPRVINHLLKKFKEGVES 5o4z A 1.7 BS02 A A 2 H104 H105 N154 H160 N162 R267 H286 A289 H107 H108 N157 H163 N165 R270 H289 A292 ? 0000166,0003676,0046872 remove_due_to_license_issue Q9X1T1 29107484 402 GSGMDEIVKVLSQHDRILVVGHIMPDGDCVSSVLSLTLGLEKLGKEVKAAVDYKIPYVFEKFPYIDKIEENPNFDPELLVVVNASSPDRIGKFQDLLDKVPSVVIDHHSTNTNFGNWNWVDPSFAATAQMIFRINKALGVEYDSNLATLNYLGIATNTGFFRHSNADVRVFEDAYKLVKMGADAHFVAKEILENKRFEQFKLFAEVLERLQLLENGKIAYSYIDYDTYLRHNCTDEDSAGFVGELRSIRGVEVAVLFMEFPRGKIHVSMRSKDWFNVNEVAFELGGGGHPRAAGVTFEGKKIEEVIPRVINHLLKKFKEGVES 5o55 A 1.45 BS01 9L5 A 1 I652 V657 P658 Y707 N708 F714 I26 V31 P32 Y81 N82 F88 ? remove_due_to_license_issue Kd=20000nM P55201 29902720 802 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o5a A 1.6 BS01 9LN A 1 I652 E655 V657 P658 E661 C704 Y707 N708 F714 I26 E29 V31 P32 E35 C78 Y81 N82 F88 ? remove_due_to_license_issue Kd=17000nM P55201 29902720 802 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o5f A 1.302 BS01 9LT A 1 I652 V657 P658 E661 Y707 N708 F714 I26 V31 P32 E35 Y81 N82 F88 ? remove_due_to_license_issue Kd=>50000nM P55201 29902720 801 EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o5h A 1.85 BS01 9LK A 1 F653 V657 P658 Y707 N708 F714 F26 V30 P31 Y80 N81 F87 ? remove_due_to_license_issue Kd=>75000nM P55201 29902720 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o5h A 1.85 BS02 9LK A 2 F653 V657 E661 Y707 F714 F26 V30 E34 Y80 F87 ? remove_due_to_license_issue Kd=>75000nM P55201 29902720 802 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5o5m A 1.583 BS02 9LQ A 1 T51 G52 G55 V57 A70 K72 Y122 V123 L173 D184 F327 T43 G44 G47 V49 A62 K64 Y114 V115 L165 D176 F317 D166 K168 N171 D184 T201 D158 K160 N163 D176 T193 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P25321 401 GSEQESVKEFLAKAKEEFLKKWESPSQNTAQLDHFDRIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGDTSNFDDYEEEEIRVSINEKCGKEFTEF 5o7e A 1.87 BS03 9NB A 1 M427 Y428 E430 H455 H459 W471 E486 E487 M86 Y87 E89 H114 H118 W130 E145 E146 3.4.24.3 0004222,0005576,0006508,0008270 ic50=0.017uM remove_due_to_license_issue IC50=17nM Q46085 28820255 803 YCPKTYTFDDGKVIIKAGARVEEEKVKRLYWASKEVNSQFFRVYGIDKPLEEGNPDDILTMVIYNSPEEYKLNSVLYGYDTNNGGMYIEPEGTFFTYEREAQESTYTLEELFRHEYTHYLQGRYAVPGQWGRTKLYDNDRLTWYEEGGAELFAGSTRTSGILPRKSIVSNIHNTTRNNRYKLSDTVHSKYGASFEFYNYACMFMDYMYNKDMGILNKLNDLAKNNDVDGYDNYIRDLSSNHALNDKYQDHMQERIDNYENLTVPFVADDYLVRHAYKNPNEIYSEISEVAKLKDAKSEVKKSQYFSTFTLRGSYTGGVSKGKLEDQKAMNKFIDDSLKKLDTYSWSGYKTLTAYFTNYKVDSSNKVTYDVVFHGYLPNEG 5o83 A 2.9 BS01 9NQ A 1 M752 P758 W760 K779 D787 I825 V828 M900 I910 D911 M537 P543 W545 K564 D572 I610 V613 M678 I688 D689 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue IC50=101nM O35904 28947947 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSLTPHLTMVHSSSILAMRDEQSNWSLEQPFSILIEGRKVNADMKLVVQAGLFHGNEMLCKTVSSSECSEPVWEFDISVCDLPRMARLCFALYAVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5o87 A 2.2 BS01 NCT A 1 Y110 W164 V165 C207 Y212 Y91 W145 V146 C188 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=598nM Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 5o87 A 2.2 BS02 NCT E 1 Y72 I135 Y53 I116 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=598nM Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 5o87 B 2.2 BS01 NCT B 1 Y110 W164 V165 C207 Y212 Y91 W145 V146 C188 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=598nM Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERRAGNGFF 5o8t A 2.2 BS01 SY9 A 1 Y110 W164 Y205 C207 C208 Y212 Y91 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 5o8t A 2.2 BS02 SY9 E 1 Y72 Q74 I135 Y53 Q55 I116 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 5o8t B 2.2 BS01 SY9 B 1 Y110 W164 Y205 C207 C208 Y212 Y91 W145 Y186 C188 C189 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFTLQDIVKVDSSTNEVDLVYYEQQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAYSSTRPVQVLSPQIAVVTHDGSVMFIPAQRLSFMCDPTGVDSEEGVTCAVKFGSWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRER 5o91 A 3.2 BS01 C5N A 1 I531 S537 K553 W604 G605 I607 S611 L654 I663 I18 S24 K40 W91 G92 I94 S98 L141 I150 D647 K649 N652 D664 T686 D134 K136 N139 D151 T167 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P33981 28726638 901 YFQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEWGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTTQVGTVNYMPPEAIKDSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQTH 5o9h A 2.7 BS01 9P2 A 1 A128 T129 L156 V159 L163 L209 W213 P214 T217 A98 T99 L126 V129 L133 L177 W181 P182 T185 ? 0004875,0004930,0006935,0007186,0016020 remove_due_to_license_issue P21730 29300009 401 NTLRVPDILALVIFAVVFLVGVLGNALVVWVTAFEAKRTINAIWFLNLAVADFLACLALPALFTSIVQHHHWPFGGAACSILPSLILLNMYASILLLATISADRFLLVFKPAWCQRFRGAGLAWILCAVAWGLALLLTIPSALYRVVREEYFPPKVLCGVDHDKRRERAVAIVRLVLGFLWPLLTLTICYTFILLRTWSARETRSTKTLKVVVAVVASFFIFWLPYQVTGIMMSFLEPSSPTFLLLKKLDSLCVSFAYINCCINPIIYVVAGQGFQKSLPELLREVLTEESVVR 5o9h B 2.7 BS01 9P2 A 1 A158 G162 L166 A128 G132 L136 ? 0004875,0004930,0006935,0007186,0016020 remove_due_to_license_issue P21730 29300009 401 NTLRVPDILALVIFAVVFLVGVLGNALVVWVTAFEAKRTINAIWFLNLAVADFLACLALPALFTSIVQHHHWPFGGAACSILPSLILLNMYASILLLATISADRFLLVFKPAWCQRFRGAGLAWILCAVAWGLALLLTIPSALYRVVREEYFPPKVLCGVDYSHDKRRERAVAIVRLVLGFLWPLLTLTICYTFILLRTWSARETRSTKTLKVVVAVVASFFIFWLPYQVTGIMMSFLEPSSPTFLLLKKLDSLCVSFAYINCCINPIIYVVAGQRKSLPELLREVLTEESVVRE 5o9h B 2.7 BS02 9P2 B 1 L125 A128 T129 L156 V159 L209 W213 P214 T217 L95 A98 T99 L126 V129 L179 W183 P184 T187 ? 0004875,0004930,0006935,0007186,0016020 remove_due_to_license_issue P21730 29300009 401 NTLRVPDILALVIFAVVFLVGVLGNALVVWVTAFEAKRTINAIWFLNLAVADFLACLALPALFTSIVQHHHWPFGGAACSILPSLILLNMYASILLLATISADRFLLVFKPAWCQRFRGAGLAWILCAVAWGLALLLTIPSALYRVVREEYFPPKVLCGVDYSHDKRRERAVAIVRLVLGFLWPLLTLTICYTFILLRTWSARETRSTKTLKVVVAVVASFFIFWLPYQVTGIMMSFLEPSSPTFLLLKKLDSLCVSFAYINCCINPIIYVVAGQRKSLPELLREVLTEESVVRE 5o9o A 1.9 BS01 9PB A 1 Y107 S134 P136 S139 I140 R142 Y244 E275 Y307 Y316 Y65 S92 P94 S97 I98 R100 Y202 E233 Y265 Y274 2.4.1.- Kd=13uM remove_due_to_license_issue Q06135 29164827 601 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQTSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYESVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPFGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKLYCKIGANDRHCPLNDKNVYFNLESLQPC 5o9p A 1.75 BS01 9P8 A 1 Y107 D132 S134 P136 S139 I140 R142 V177 Y244 E275 Y307 Y316 Y71 D96 S98 P100 S103 I104 R106 V141 Y208 E239 Y271 Y280 2.4.1.- Kd=8.06uM remove_due_to_license_issue Q06135 29164827 601 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQRSGAFETSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYLTESVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKLYCKIGANDRHCPLNDKNVYFNLESLQPC 5o9q A 1.4 BS04 9PH A 1 Y107 S134 P136 S139 I140 R142 Y244 E275 Y307 Y316 Y71 S98 P100 S103 I104 R106 Y208 E239 Y271 Y280 2.4.1.- Kd=6.2uM remove_due_to_license_issue Q06135 29164827 604 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQRSGAFETSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYLTESVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPFGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKYCIGANDRHCPLNDKNVYFNLESLQPC 5o9r A 1.7 BS04 9PK A 1 Q60 Y107 S134 P136 S139 I140 R142 Y244 E275 Y307 Q32 Y66 S93 P95 S98 I99 R101 Y203 E234 Y266 2.4.1.- Kd=4.09uM remove_due_to_license_issue Q06135 29164827 604 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQRSSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYLTSVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKLYCKIGANDRHCPLNDKNVYFNLESLQPC 5o9y A 1.57 BS01 9PN A 1 Y107 S134 P136 S139 I140 R142 Y244 Y307 Y316 Y67 S94 P96 S99 I100 R102 Y204 Y267 Y276 2.4.1.- Kd=4.6uM remove_due_to_license_issue Q06135 29164827 601 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQRSTSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYLTVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPFGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKLYCKIGANDRHCPLNDKNVYFNLESLQC 5oa2 C 2.15 BS04 9PW C 1 Y107 S134 P136 S139 I140 N141 R142 V177 Y244 E275 Y307 Y64 S91 P93 S96 I97 N98 R99 V134 Y201 E232 Y264 2.4.1.- Kd=9.8uM remove_due_to_license_issue Q06135 29164827 604 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYLTESVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPFESGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKLYCKIGANDRHCPLNDKNVYFNLESLQPCKNVF 5oa6 A 1.94 BS01 9PT A 1 Y107 S134 P136 S139 I140 R142 Y244 E275 Y307 Y67 S94 P96 S99 I100 R102 Y204 E235 Y267 2.4.1.- Kd=3.1uM remove_due_to_license_issue Q06135 29164827 601 SFEKTPAIKIVGNKFFDSESGEQFFIKGIAYQLQRSTSYIDALADPKICLRDIPFLKMLGVNTLRVYAIDPTKSHDICMEALSAEGMYVLLDLSEPDISINRENPSWDVHIFERYKSVIDAMSSFPNLLGYFAGNEVTNDHTNTFASPFVKAAIRDAKEYISHSNHRKIPVGYSTNDDAMTRDNLARYFVCGDVKADFYGINMYEWCGYSTYGTSGYRERTKEFEGYPIPVFFSEFGCNLVRPRPFTEVSALYGNKMSSVWSGGLAYMYFEEENEYGVVKINDNDGVDILPDFKNLKKEFAKADPKGITEEEYLTSVECPHIAVGVWEANEKLPETPDRSKCACLDEILPCEIVPGKYEEYFSYLCSKVDCSDILANGKTGEYGEFSDCSVEQKLSLQLSKLYCKIGANDRHCPLNDKNVYFNLESLQPC 5oae A 2.7 BS03 SVF A 1 H42 H60 P201 H204 N205 H208 R209 V218 H39 H57 P198 H201 N202 H205 R206 V215 ? 0016491,0046872 remove_due_to_license_issue B2ZB02 29634898 303 KYRVRKNVLHLTDTEKRDFVRTVLILKEKGIYDRYIAWHGAAGKFHTPPGSDRNAAHMSSAFLPWHREYLLRFERDLQSINPEVTLPYWEWETDAQMQDPSQSQIWSADFMGGNGNPIKDFIVDTGPFAAGRWTTIDEQGNPSGGLKRNFGATKEAPTLPTRDDVLNALKITQYDTPPWDMTSQNSFRNQLEGFINGPQLHNRVHRWVGGQMGVVPTAPNDPVFFLHHANVDRIWAVWQIIHRNQNYQPMKNGPFGQNFRDPMYPWNTTPEDVMNHRKLGYVYDIEL 5oah A 1.8 BS02 95B A 1 Q98 R118 K121 R205 H227 R249 Y288 Q76 R96 K99 R183 H205 R227 Y266 ? 0006826,0030288,0030313,0046872,1901678 remove_due_to_license_issue Q0P8Q4 402 MLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5oai A 2.0 BS01 B5K A 1 L54 G58 I61 F86 V93 H96 I99 L38 G42 I45 F70 V77 H80 I83 2.3.2.27 0005634,0043066,0051726 Ki=0.1uM remove_due_to_license_issue Ki=0.13nM Q00987 30715803 201 MQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVNQQ 5oaj D 2.47 BS01 TKT E 1 E162 W164 C207 C208 Y212 E143 W145 C188 C189 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFFLQDIVKVDSSTNEVDLVYYERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAASSTRPVQVLSPQIAVVTHDGSVMFSPAQRLSFMCDPTGVDSEEGVTCAVKFESWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYSCCPEPYIDVNLVVKFRERR 5oax A 1.2 BS01 9Q5 A 1 R144 H158 R162 W181 E184 R186 R32 H46 R50 W69 E72 R74 ? 0030246 Kd=27nM remove_due_to_license_issue P17931 29284090 301 MLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5obg A 2.0 BS01 SY9 A 1 E162 S163 W164 S167 Y205 Y212 E143 S144 W145 S148 Y186 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFFLQDIVKVDSSTNEVDLVYYERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAASSTRPVQVLSPQIAVVTHDGSVMFSPAQRLSFMCDPTGVDSEEGVTCAVKFESWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYKGTGEPYIDVNLVVKFRERR 5obg B 2.0 BS01 SY9 B 1 W164 V165 Y205 E210 Y212 W145 V146 Y186 E191 Y193 ? 0004888,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Q8WSF8 31709057 601 QANLMRLKSDLFNRSPMYPGPTKDDPLTVTLGFFLQDIVKVDSSTNEVDLVYYERQRWKLNSLMWDPNEYGNITDFRTSAADIWTPDITAASSTRPVQVLSPQIAVVTHDGSVMFSPAQRLSFMCDPTGVDSEEGVTCAVKFESWVYSGFEIDLKTDTDQVDLSSYYASSKYEILSATQTRQVQHYKGTGEPYIDVNLVVKFRERRFF 5obj A 2.901 BS02 9QK A 1 K166 L169 E175 L178 R179 Y199 V206 K40 L43 E49 L52 R53 Y73 V80 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T162 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 28787041 405 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 5obr A 2.62 BS01 9QT A 1 K166 E175 L178 R179 Y199 H201 V206 K41 E50 L53 R54 Y74 H76 V81 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 28787041 401 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKP 5oci A 1.62 BS01 9R8 A 1 N51 A55 D93 G97 M98 L107 G135 F138 W162 T184 N35 A39 D77 G81 M82 L89 G115 F118 W142 T164 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=9nM remove_due_to_license_issue P07900 29701469 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLNLIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5ocj A 1.8 BS01 9SW A 1 L40 S124 W265 L33 S117 W258 2.3.1.122,2.3.1.20 0004144,0005576,0006869,0009247,0009274,0016020,0016746,0016747,0035375,0046677,0050348,0071769 remove_due_to_license_issue P9WQN9 29301937 401 VEYLQVPSASMGRDIKVQFQGGGPHAVYLLDGLRAQDDYNGWDINTPAFEEYYQSGLSVIMPVGGQSSFYTDWYQPSQSNGQNYTYKWETFLTREMPAWLQANKGVSPTGNAAVGLSMSGGSALILAAYYPQQFPYAASLSGFLNPSEGWWPTLIGLAMNDSGGYNANSMWGPSSDPAWKRNDPMVQIPRLVANNTRIWVYCGNGTPSDLGGDNIPAKFLEGLTLRTNQTFRDTYAADGGRNGVFNFPPNGTHSWPYWNEQLVAMKADIQHVLNG 5ocj A 1.8 BS02 9SW B 1 I222 P223 F226 I215 P216 F219 2.3.1.122,2.3.1.20 0004144,0005576,0006869,0009247,0009274,0016020,0016746,0016747,0035375,0046677,0050348,0071769 remove_due_to_license_issue P9WQN9 29301937 401 VEYLQVPSASMGRDIKVQFQGGGPHAVYLLDGLRAQDDYNGWDINTPAFEEYYQSGLSVIMPVGGQSSFYTDWYQPSQSNGQNYTYKWETFLTREMPAWLQANKGVSPTGNAAVGLSMSGGSALILAAYYPQQFPYAASLSGFLNPSEGWWPTLIGLAMNDSGGYNANSMWGPSSDPAWKRNDPMVQIPRLVANNTRIWVYCGNGTPSDLGGDNIPAKFLEGLTLRTNQTFRDTYAADGGRNGVFNFPPNGTHSWPYWNEQLVAMKADIQHVLNG 5od5 A 1.9 BS02 95B A 1 Q98 R118 K121 R205 R249 Y288 Q76 R96 K99 R183 R227 Y266 ? 0006826,0030288,0030313,0046872,1901678 remove_due_to_license_issue Q0P8Q4 403 MLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5od5 A 1.9 BS03 9RT A 1 T226 H227 T204 H205 ? 0006826,0030288,0030313,0046872,1901678 remove_due_to_license_issue Q0P8Q4 404 MLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTHGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5odu F 1.56 BS01 AMG F 1 Y38 E44 Q57 I61 D96 V97 T100 D103 Y37 E43 Q56 I60 D95 V96 T99 D102 ? 0030246,0046872 ic50=0.52mM remove_due_to_license_issue Q7N561 28972138 201 SDWSGSVPANAENGKSTGLILKQGDTISVVAHGWVKYGRDNVEWAAPDGPVPNNPQPSSIATLVAKIANKKFAIGNGVLHKTVPVDGELILLFNDVPGTFGDNSGEFQVEVIIESRYSPLK 5odx A 1.82 BS01 9RZ A 1 N51 D54 A55 D93 G97 M98 G135 F138 W162 T184 N36 D39 A40 D78 G82 M83 G120 F123 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=195nM remove_due_to_license_issue P07900 29701469 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 5ody A 1.149 BS01 9SK A 1 R144 I145 A146 H158 N160 R162 W181 E184 R186 S237 G238 R32 I33 A34 H46 N48 R50 W69 E72 R74 S125 G126 ? 0030246 Kd=4nM remove_due_to_license_issue P17931 29284090 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 5oei A 1.78 BS01 OOG A 1 F48 T54 S169 S173 T174 S198 N216 S261 F13 T19 S134 S138 T139 S163 N181 S226 ? Kd=1.6uM remove_due_to_license_issue Q6N193 29082669 401 DWPTRQVTLVVPFTSGGTTDMLARLIAARLSEHYGQSFVIDNRSGESGNIAASYVAKVPADGYTFIIGTPGIHATNRLVYRTMGYDPATDFTPVIVIARVPNLLSVTKSLPVTSVADLISYARQRPRELFYGVSALGSTGHLSTELFKTMTGVEITAVPYKGSAPMLRDLAEGRVHLTIDNLPASKPLLEAGEIRPLAVTTAKRWPPLSHLPTIAEAGVPGYETASWFTVGAPRGTPTEIVTSLNTTVAAFLGSDSGTVKLREIGAEPGGGSPQDMQRHVEAEIARWEKVAKTAGIAPL 5of0 A 1.48 BS05 9TB A 1 R210 M424 L428 R463 D465 G518 N519 R534 R536 F546 Y552 H553 K699 Y700 R156 M370 L374 R409 D411 G464 N465 R480 R482 F488 Y494 H495 K641 Y642 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue IC50=2.3nM Q04609 30429952 822 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAMEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 5ofi C 2.0 BS02 9TQ C 1 Y38 E44 Q57 I61 D96 V97 G99 T100 D103 Y37 E43 Q56 I60 D95 V96 G98 T99 D102 ? 0030246,0046872 Kd=62.7uM remove_due_to_license_issue Q7N561 28972138 202 SDWSGSVPANAENGKSTGLILKQGDTISVVAHGWVKYGRDNVEWAAPDGPVPNNPQPSSIATLVAKIANKKFAIGNGVLHKTVPVDGELILLFNDVPGTFGDNSGEFQVEVIIESRYSPLK 5ofu A 2.62 BS01 AMP A 1 I16 S19 Q20 P21 S24 R25 G26 F28 Y113 I10 S13 Q14 P15 S18 R19 G20 F22 Y97 D74 E97 E98 D118 L120 D121 E284 D58 E81 E82 D102 L104 D105 E268 3.1.3.11 0000166,0005737,0005829,0005975,0006000,0006002,0006094,0016787,0016791,0020015,0030388,0042132,0042578,0046872 remove_due_to_license_issue O97193 28882541 401 PTPTTLTQYIIKSQPPHSRGDFTLLMMAIQTSVKVIEKNIRRAGMKGMLGYIAGAKLDVISNIAFKAYLLSSTSVCVLGSEEEEQMIIAESGRRGDYLIFFDPLDGSSNIDANVSVGSIWGVWRLPKDTTINSVEDANAVIRMLKGTDMVSAGYAVYGSATNLVLTSGHGVDGFTLDPNIGEFILTHPHISIPKKRSIYSVNEGNYGKWEPWFKEYIDYLKMNKTTRYSARYIGSMVGDIHRTLLYGGIFCYPKDANQVEGKLRLLYEAAPMAMIVEQAGGKAVGSNGRILEQSITRLHQRTPVYFGSRQEVDLCMAFRDRN 5ofv B 1.5 BS01 9TZ B 1 Y174 P176 T207 T213 Y75 P77 T108 T114 N102 R236 D260 E265 H283 N3 R137 D161 E166 H184 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 Kd=26.2mM remove_due_to_license_issue O43175 29568346 401 NGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSR 5ofw B 1.5 BS01 9TW B 1 G152 Y174 P176 T207 S212 T213 G53 Y75 P77 T108 S113 T114 N102 R236 D260 E265 H283 N3 R137 D161 E166 H184 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 Kd=1.6mM remove_due_to_license_issue Kd=1500000nM O43175 29568346 401 NGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSR 5ogk A 3.6 BS01 GDD A 1 Y28 M35 Y114 I265 S266 S269 Y281 K289 Y10 M17 Y93 I224 S225 S228 Y240 K248 ? 0000139,0005458,0005739,0005783,0005789,0005794,0015297,0016020,0030659,0031410,0055085,1990570 remove_due_to_license_issue P40107 29143814 401 NSGPISILSYCGSSILMTVTNKFVVNLKDFNMNFVMLFVQSLVCTITLIILRILGFRSLNKTDAKNWFPISFLLVLMIYTSSKALQYLAVPIYTIFKNLTIILIAYGEVLFFGGSVTSMELSSFLLMVLSSVVATWGDQQNPGYFWMFTNCITSALFVLIMRKRIKLTNFKDFDTMFYNNVLALPILLLFSFCVEDWSSVNLTNNFSNDSLTAMIISGVASVGISYCSGWCVRVTSSTTYSMVGALNKLPIALSGLIFFDAPRNFLSILSIFIGFLSGIIYAVAKQKKQQAQ 5ogl A 2.7 BS04 9UB A 1 D56 F60 Y79 Y196 S198 Q289 Y293 M368 R375 F376 Y379 Y468 D55 F59 Y78 Y195 S197 Q288 Y292 M367 R374 F375 Y378 Y467 2.4.99.19 0000287,0004576,0005886,0006486,0016020,0016757,0018279,0046872 remove_due_to_license_issue B9KDD4 29058712 803 ELQQNFTDNNSIKYTAILILIAFAFSVLARLYWVAWASEFYEFFFNDQLMITTNDGYAFAEGARDMIAGFHQPNDLSYFGSSLSTLTYWLYSILPFSFESIILYMSTFFASLIVVPIILIAREYKLTTYGFIAALLGSIANSYYNRTMSGYYDTDMLVLVLPMLILLTFIRLTINKDIFTLLLSPVFIMIYLWWYPSSYSLNFAMIGLFGLYTLVFHRKEKIFYLTIALMIIALSMLAWQYKLALIVLLFAIFAFKEEKINFYMIWALIFISILILHLSGGLDPVLYQLKFYVFKASDVQNLKDAAFMYFNVNETIMEVNTIDPEVFMQRISSSVLVFILSFIGFILLLKDHKSMLLALPMLALGFMALRAGLRFTIYAVPVMALGFGYFLYAFFNFLEKKQIKLSLRNKNILLILIAFFSISPALMHIYYYKSSTVFTSYEASILNDLKNKAQREDYVVAWWDYGYPIRYYSDVKTLIDGGKHLGKDNFFSSFVLSKEQIPAANMARLSVEYTEKSFKENYPDVLKAMVKDYQKTSAKDFLESLNDPNFKIDTPKTRDVYIYMPYRMLRIMPVVAQFANTNPDNGEQEKSLFFSQANPLDQDGSITLDNGVEISNDYRSLKIEGNSIPLKAFVDIESITNGKFYYNEIDSKAQIYLLYLREYKSYVILDESLYNSSYIQMFLLNQYDQDLFEQITNDTRAKIYRLK 5oh1 C 1.7 BS02 9UQ C 1 E76 F77 W79 W85 W99 Y101 E53 F54 W56 W62 W76 Y78 ? 0046872 remove_due_to_license_issue A4TVL0 31459225 202 GASIFRCRQCGQTISRRDWLLEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5oh2 A 1.9 BS02 BAQ A 1 F77 W79 W85 W99 Y101 F59 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue A4TVL0 31459225 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5oh3 A 2.1 BS02 9V2 A 1 N50 F77 W79 W85 W99 Y101 N32 F59 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue A4TVL0 31459225 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5oh4 A 2.3 BS02 9UZ A 1 F77 S78 W79 W85 W99 Y101 F59 S60 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue Ki=28000nM, IC50=48900nM A4TVL0 31459225 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5oh7 A 1.85 BS02 HYN A 1 F77 W79 W85 W99 Y101 F59 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue A4TVL0 31459225 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5oh9 A 1.65 BS02 9UT A 1 F77 W79 W85 W99 Y101 F60 W62 W68 W82 Y84 ? 0046872 remove_due_to_license_issue A4TVL0 31459225 202 GASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5oha A 1.55 BS02 9UW A 1 F77 W79 W85 W99 Y101 F59 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue A4TVL0 31459225 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 5ohi A 1.66 BS06 9V8 A 1 D171 T209 F210 L213 Y214 L243 W260 F273 F274 W275 Y306 D311 D121 T159 F160 L163 Y164 L193 W210 F223 F224 W225 Y256 D261 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 remove_due_to_license_issue Q9R1E6 29259743 920 WTNTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPLDCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5ohj A 1.6 BS02 9VE A 1 M519 D564 N567 Y575 W578 T579 I582 F586 Q589 M603 C604 S614 Q615 F618 I622 M197 D242 N245 Y253 W256 T257 I260 F264 Q267 M281 C282 S292 Q293 F296 I300 3.1.4.53 0004114,0007165,0008081 ic50=0.0378nM remove_due_to_license_issue Q07343 29200281 801 TSISRFGVNTENEDHLAKELEDLNKWGLNIFNVAGYSHNRPLTCIMYAIFQERDLLKTFRISSDTFITYMMTLEDHYHSDVAYHNSLHAADVAQSTHVLLSTPALDAVFTDLEILAAIFAAAIHDVDHPGVSNQFLINTNSELALMYNDESVLENHHLAVGFKLLQEEHCDIFMNLTKKQRQTLRKMVIDMVLATDMSKHMSLLADLKTMVETKKVTSSGVLLLDNYTDRIQVLRNMVHCADLSNPTKSLELYRQWTDRIMEEFFQQGDKERERGMEISPMCDKHTASVEKSQVGFIDYIVHPLWETWADLVQPDAQDILDTLEDNRNWYQSMIPQ 5oje A 1.579 BS01 VSK A 1 D33 D35 Y79 G80 D81 F116 D219 G221 T222 I300 D33 D35 Y79 G80 D81 F116 D219 G221 T222 I300 D35 S38 D40 W42 Y79 D219 T222 D35 S38 D40 W42 Y79 D219 T222 3.4.23.22 0004190,0006508 Ki=6.1uM remove_due_to_license_issue P11838 30178575 401 STGSATTTPIDSLDDAYITPVQIGTPAQTLNLDFDTGSSDLWVFSSETTASEVDGQTIYTPSKSTTAKLLSGATWSISYGDGSSSSGDVYTDTVSVGGLTVTGQAVESAKKVSSSFTEDSTIDGLLGLAFSTLNTVSPTQQKTFFDNAKASLDSPVFTADLGYHAPGTYNFGFIDTTAYTGSITYTAVSTKQGFWEWTSTGYAVGSGTFKSTSIDGIADTGTTLLYLPATVVSAYWAQVSGAKSSSSVGGYVFPCSATLPSFTFGVGSARIVIPGDYIDFGPISTGSSSCFGGIQSSAGIGINIFGDVALKAAFVVFNGATTPTLGFASK 5okt A 2.13 BS01 9XK A 1 I15 L25 A36 L85 G86 L135 I12 L22 A33 L82 G83 L132 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=317nM remove_due_to_license_issue P48730 29630366 301 RVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 5oku A 2.07 BS01 0L1 A 1 F48 T54 P105 S173 T174 S198 N216 S261 F13 T19 P70 S138 T139 S163 N181 S226 ? Kd=0.55uM remove_due_to_license_issue Q6N193 29082669 401 DWPTRQVTLVVPFTSGGTTDMLARLIAARLSEHYGQSFVIDNRSGESGNIAASYVAKVPADGYTFIIGTPGIHATNRLVYRTMGYDPATDFTPVIVIARVPNLLSVTKSLPVTSVADLISYARQRPRELFYGVSALGSTGHLSTELFKTMTGVEITAVPYKGSAPMLRDLAEGRVHLTIDNLPASKPLLEAGEIRPLAVTTAKRWPPLSHLPTIAEAGVPGYETASWFTVGAPRGTPTEIVTSLNTTVAAFLGSDSGTVKLREIGAEPGGGSPQDMQRHVEAEIARWEKVAKTAGIAPL 5olb A 1.82 BS05 6ZO A 1 D171 T209 L213 L243 F273 F274 W275 Y306 D311 H315 D121 T159 L163 L193 F223 F224 W225 Y256 D261 H265 3.1.4.39 0003676,0004528,0004551,0004622,0004630,0005044,0005509,0005576,0005615,0005886,0006644,0006935,0006955,0008270,0009395,0010634,0016042,0016192,0016787,0016788,0030149,0030247,0030334,0034638,0046872,0047391,0050731,2000394 remove_due_to_license_issue IC50=2.8nM Q9R1E6 29259743 925 WTNTSGSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKDRCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIRVPECPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVYPTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDATFHLRGREKFNHRWWGGQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAFYSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLKLHRCVNVIFVGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRPKIPNNLKYDPKAIIANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDLHLLVERRWHVARKPLDKCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIELYNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTLPEEVSRPNYPGIMYLQSDFDLGCTCDDKGSTEERHLLYGRPAVLYRTSYDILYHTDFESGYSEIFLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQMSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWTYFQRVLVKKYASERNGVNVISGPIFDYNYNGLRDIEDEIKQYVEGSSIPVPTHYYSIITSCLDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTARVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE 5olk A 2.45 BS01 DTP A 1 I9 K11 R12 F19 V20 K23 I24 V68 V71 Q72 I5 K7 R8 F15 V16 K19 I20 V64 V67 Q68 1.17.4.1 0004748,0005524,0009263,0016491,0046872 Kd=1uM remove_due_to_license_issue A3XHF9 29388911 1001 EIKKIIKRDYSTAPFVLEKITNAIANAMAALGHGSEQDAKLISMQVYESLLNNKEQESEYIPTVEQVQDMVEDKLMSSEFHDVAKAYIIYRNKRALERKTNIFEKRINLKPYEYPELNEYVAAIRHSYWIHTEFNFTSDIQDFKTGLSEVERSAIKNTMLAISQIEVAVKTFWGDVHHRLPKPEIAAVGATFAESEVRHHDAYSHLLEILGLNEEFKELKKKPVIMKRVHYLETSLKHAKSDDDREYTESILLFALFIEHVSLFSQFLIIMAFNKHKNMLKGISNAVEATSKEEQIHGDFGVDIINIIKKENPEWFDEEHNNLIKEMCLNSFEAESKVVDWIFEKGELDFLPKAVINEFLKNRFNKSLEAIGLEKLFDIDEALLQETEWFDDEII 5olk A 2.45 BS02 DTP A 2 R12 A27 N30 A31 A90 Y91 Y94 R98 R102 R8 A23 N26 A27 A86 Y87 Y90 R94 R98 1.17.4.1 0004748,0005524,0009263,0016491,0046872 Kd=1uM remove_due_to_license_issue A3XHF9 29388911 1002 EIKKIIKRDYSTAPFVLEKITNAIANAMAALGHGSEQDAKLISMQVYESLLNNKEQESEYIPTVEQVQDMVEDKLMSSEFHDVAKAYIIYRNKRALERKTNIFEKRINLKPYEYPELNEYVAAIRHSYWIHTEFNFTSDIQDFKTGLSEVERSAIKNTMLAISQIEVAVKTFWGDVHHRLPKPEIAAVGATFAESEVRHHDAYSHLLEILGLNEEFKELKKKPVIMKRVHYLETSLKHAKSDDDREYTESILLFALFIEHVSLFSQFLIIMAFNKHKNMLKGISNAVEATSKEEQIHGDFGVDIINIIKKENPEWFDEEHNNLIKEMCLNSFEAESKVVDWIFEKGELDFLPKAVINEFLKNRFNKSLEAIGLEKLFDIDEALLQETEWFDDEII 5om2 A 1.47 BS01 DXT B 1 L273 A274 F277 D278 L251 A252 F255 D256 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 remove_due_to_license_issue P01011 29760101 501 DRGLASANVDFAFSLYKQLVLKAPDKNVIFSPLSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNQSSDELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKFEMPFDPQDTHQSRFYLSKKKYVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASALFILPDQDKMEEVEAMLSQETLARFFDSLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTEASAATALEVLFQ 5om2 B 1.47 BS01 DXT B 1 H383 W386 H16 W19 ? remove_due_to_license_issue P01011 29760101 501 TIVRFNRPFLMIIVDHFTWSIFFMSKVTNPK 5om3 A 2.0 BS01 DXT B 1 L273 S274 F277 D278 L248 S249 F252 D253 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 remove_due_to_license_issue P01011 29760101 501 VDRGLASANVDFAFSLYKQLVLKAPDKNVIFSPLSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKFEMPFDPQDTHQSRFYLSKKKYVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASALFILPDQDKMEEVEAMLSQETLSRFFDSLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTEASAATALFIPLS 5om3 B 2.0 BS01 DXT B 1 H383 W386 H17 W20 ? remove_due_to_license_issue P01011 29760101 501 RTIVRFNRPFLMIIVDHFTWSIFFMSKVTNPKQ 5om7 A 1.727 BS01 DM2 A 1 Q242 L273 F277 E278 Q220 L251 F255 E256 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 remove_due_to_license_issue P01011 29760101 501 DRGLASANVDFAFSLYKQLVLKAPDKNVIFSPLSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNQSSDELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKFEMPFDPQDTHQSRFYLSKKKYVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASALFILPDQDKMEEVEAMLSQETLSRFFESLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTEASAATALEVLFQ 5om7 B 1.727 BS01 DM2 A 1 V381 N383 W386 V15 N17 W20 ? remove_due_to_license_issue P01011 29760101 501 RTIVRFNRPFLMIIVDNFTWSIFFMSKVTNPKQ 5om9 A 1.8 BS01 O2S A 1 H69 R127 N144 R145 Y248 E270 H157 R215 N232 R233 Y336 E358 H69 E72 R127 H196 E270 H157 E160 R215 H284 E358 3.4.17.1 0004181,0006508,0008270 remove_due_to_license_issue P15085 29057062 401 KEDFVGHQVLRISVADEAQVQKVKELEDLEHLQLDFWRGPAHPGSPIDVRVPFPSIQAVKIFLESHGISYETMIEDVQSLLDEEQEQMFRSTDTFNYATYHTLEEIYDFLDLLVAENPHLVSKIQIGNTYEGRPIYVLKFSTGGSKRPAIWIDTGIHSREWVTQASGVWFAKKITQDYGQDAAFTAILDTLDIFLEIVTNPDGFAFTHSTNRMWRKTRSHTAGSLCIGVDPNRNWDAGFGLSGASSNPCSETYHGKFANSEVEVKSIVDFVKDHGNIKAFISIHSYSQLLMYPYGYKTEPVPDQDELDQLSKAAVTALASLYGTKFNYGSIIKAIYQASGSTIDWTYSQGIKYSFTFELRDTGRYGFLLPASQIIPTAKETWLALLTIMEHTLNHP 5one A 2.6 BS01 9YQ A 1 L194 L210 E211 A213 G216 R220 L263 A273 L68 L84 E85 A87 G90 R94 L137 A147 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue EC50=38nM, IC50=52nM O14965 28818446 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5oot A 2.1 BS01 4K4 A 1 T14 V23 A36 M84 L86 A87 G90 L137 T11 V20 A33 M74 L76 A77 G80 L127 D130 K132 H134 N135 D148 T170 D120 K122 H124 N125 D138 T160 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.0285uM remove_due_to_license_issue O14757 29023112 301 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5op2 A 1.9 BS01 A0Q A 1 L15 G16 E17 V23 A36 M84 E85 A87 G90 L137 L12 G13 E14 V20 A33 M76 E77 A79 G82 L129 D130 K132 H134 N135 D148 T170 D122 K124 H126 N127 D140 T162 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.24uM remove_due_to_license_issue O14757 29023112 301 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMCPENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 5op4 A 2.0 BS01 A0T A 1 L15 V23 A36 M84 L86 A87 S88 G90 L137 L13 V21 A34 M73 L75 A76 S77 G79 L126 D130 K132 H134 N135 D148 T170 D119 K121 H123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.194uM remove_due_to_license_issue O14757 29023112 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5op5 A 1.9 BS01 3FE A 1 V23 A36 M84 E85 L86 A87 L137 D148 V20 A33 M73 E74 L75 A76 L126 D137 D130 K132 H134 N135 D148 T170 D119 K121 H123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.216uM remove_due_to_license_issue O14757 29023112 301 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5op6 A 2.45 BS02 A0W A 1 Y93 L101 Y102 Y145 Q147 L188 T196 H199 D201 F207 K214 R238 I281 Y79 L87 Y88 Y129 Q131 L172 T180 H183 D185 F191 K198 R222 I265 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=21uM remove_due_to_license_issue IC50=21000nM Q9NWT6 29435217 404 EPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 5op8 A 2.3 BS02 A1H A 1 Y93 Q147 L188 H199 D201 F207 K214 H279 I281 W296 Y79 Q133 L174 H185 D187 F193 K200 H265 I267 W282 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=66uM remove_due_to_license_issue IC50=31000nM Q9NWT6 29435217 402 EPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 5opb A 1.55 BS01 A1N A 1 L15 E17 A36 M84 E85 L86 A87 G90 L137 L11 E13 A32 M75 E76 L77 A78 G81 L128 D130 K132 H134 N135 D148 T170 D121 K123 H125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.0241uM remove_due_to_license_issue O14757 29023112 301 FVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMCPENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 5opc A 2.3 BS02 A1Z A 1 L186 L188 T196 H199 D201 F207 I281 W296 L176 L178 T186 H189 D191 F197 I271 W286 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0030947,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=29uM remove_due_to_license_issue IC50=29000nM Q9NWT6 29435217 412 SGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 5opr A 1.95 BS01 A3E A 1 L15 A36 M84 L86 A87 G90 L137 L12 A33 M72 L74 A75 G78 L125 D130 K132 H134 N135 D148 T170 D118 K120 H122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=2.56uM remove_due_to_license_issue O14757 29023112 301 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5ops A 2.0 BS01 A3Q A 1 L15 V23 A36 M84 E85 A87 L137 L13 V21 A34 M72 E73 A75 L125 D130 K132 H134 N135 D148 T170 D118 K120 H122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.863uM remove_due_to_license_issue O14757 29023112 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5opu A 1.55 BS01 A3K A 1 V23 A36 M84 E85 A87 L137 V21 A34 M74 E75 A77 L127 D130 K132 H134 N135 D148 T170 D120 K122 H124 N125 D138 T160 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.053uM remove_due_to_license_issue O14757 29023112 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 5opv A 1.9 BS01 A3H A 1 V23 A36 M84 E85 A87 G90 L137 V21 A34 M75 E76 A78 G81 L128 D130 K132 H134 N135 D148 T170 D121 K123 H125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.0515uM remove_due_to_license_issue O14757 29023112 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5oq4 A 2.7 BS01 A3W A 1 I831 K833 D836 E880 I881 V882 K890 D964 I585 K587 D590 E634 I635 V636 K644 D717 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue Kd=25nM, IC50=708nM P48736 28829592 1201 EESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCRLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHILGERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 5oq5 A 1.4 BS01 4K4 A 1 V23 A36 A87 S88 G89 G90 L137 V21 A34 A82 S83 G84 G85 L132 D130 K132 H134 N135 D148 T170 D125 K127 H129 N130 D143 T165 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.02uM remove_due_to_license_issue O14757 29023112 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5oq6 A 1.95 BS01 4K4 A 1 T14 L15 V23 A36 L86 A87 S88 L137 T10 L11 V19 A32 L73 A74 S75 L124 D130 K132 H134 N135 D148 T170 D117 K119 H121 N122 D135 T157 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.0277uM remove_due_to_license_issue O14757 29023112 301 FVEDWDLVQTLGEGSFGEVQLAVNRVTEEAVAVKIVDNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5oq7 A 2.1 BS01 A0Q A 1 G16 E17 V23 I68 M84 E85 A87 G90 L137 G9 E10 V16 I56 M72 E73 A75 G78 L125 D130 K132 H134 N135 D148 T170 D118 K120 H122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.322uM remove_due_to_license_issue O14757 29023112 301 DWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMCPENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK 5oq8 A 2.0 BS01 A0Q A 1 L15 A36 M84 E85 L86 A87 G90 L137 L12 A33 M75 E76 L77 A78 G81 L128 D130 K132 H134 N135 D148 T170 D121 K123 H125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=1.41uM remove_due_to_license_issue O14757 29023112 301 PFVEDWDLVQTLGEGSFGEVQLAVNRVTEEAVAVKIVDMPENIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK 5oqu A 2.324 BS02 A4B A 1 L124 P159 V162 M221 M225 L121 P156 V159 M218 M222 D156 K158 N161 D175 S194 D153 K155 N158 D172 S191 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=493000nM P68400 29732088 402 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5oqw A 2.31 BS02 A4E A 1 L292 K299 G306 L307 T308 D309 W310 E314 Q319 W323 Y324 L44 K51 G58 L59 T60 D61 W62 E66 Q71 W75 Y76 2.3.2.27 ic50<40nM remove_due_to_license_issue P98170 29695633 403 NFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5oqw B 2.31 BS02 A4E B 1 K297 G306 L307 T308 D309 W310 E314 Q319 W323 Y324 K50 G59 L60 T61 D62 W63 E67 Q72 W76 Y77 2.3.2.27 ic50<40nM remove_due_to_license_issue P98170 29695633 402 MNFPNSTNLPRNPSMADYEARIFTFGTWIYSVNKEQLARAGFYALGEGDKVKCFHCGGGLTDWKPSEDPWEQHAKWYPGCKYLLEQKGQEYINNIHLTHSLEECLVR 5or9 A 2.0 BS01 JR5 A 1 W1887 P1888 F1889 L1891 P1892 V1893 N1944 I1950 W32 P33 F34 L36 P37 V38 N89 I95 ? ic50=88uM remove_due_to_license_issue Q9UIF8 28862840 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5orb A 2.103 BS01 JR6 A 1 P1888 F1889 V1893 F1943 N1944 P33 F34 V38 F88 N89 ? remove_due_to_license_issue Q9UIF8 28862840 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 5org A 1.99 BS01 6DB A 1 E30 Y33 W71 A88 A89 M90 S91 R96 N111 Q159 T162 T163 N202 E11 Y14 W52 A69 A70 M71 S72 R77 N92 Q140 T143 T144 N183 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=0.009uM remove_due_to_license_issue P0A4F8 29269740 321 MQEKSITIATEGGYAPWNFSGPGGKLDGFEIDLANALCEKMKAKCQIVAQNWDGIMPSLTGKKYDAIMAAMSVTPKRQEVIGFSIPYAAGINGFAVMGDSKLAEMPGLGETYSLDSQADAAKKAIADISSFLNGTTVGVQGSTTASTFLDKYFKGSVDIKEYKSVEEHNLDLTSGRLDAVLANATVLAAAIEKPEMKGAKLVGPLFSGGEFGVVAVGLRKEDTALKADFDAAIKAASEDGTIKTLSLKWFKVDVTPQ 5orh A 1.75 BS01 A4N A 1 Q36 Y39 K102 D103 T108 A110 Q33 Y36 K99 D100 T105 A107 D156 K158 N161 D175 S194 D153 K155 N158 D172 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=41uM remove_due_to_license_issue IC50=208000nM P68400 29732088 401 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5orh A 1.75 BS02 A4N A 2 F121 L124 M137 P159 V162 I164 M221 M225 F118 L121 M134 P156 V159 I161 M218 M222 D156 K158 N161 D175 S194 D153 K155 N158 D172 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=41uM remove_due_to_license_issue IC50=208000nM P68400 29732088 402 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5orj B 1.99 BS04 A4Q B 1 F121 P159 V162 M221 M225 F118 P156 V159 M218 M222 D156 K158 N161 D175 S194 D153 K155 N158 D172 S191 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=160000nM P68400 29732088 404 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5ork A 2.143 BS03 A4T A 1 F121 L124 L128 P159 V162 I164 M221 M225 F118 L121 L125 P156 V159 I161 M218 M222 D156 K158 N161 D175 S194 D153 K155 N158 D172 S191 2.7.11.1 0004672,0004674,0005524,0006468 Kd=234uM remove_due_to_license_issue IC50=150000nM P68400 29732088 404 PVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5orl A 1.69 BS03 A4W A 1 E183 L188 C247 V252 H280 E57 L62 C121 V126 H154 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 29045126 407 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5orr A 2.09 BS03 A5Q A 1 K166 E175 L178 R179 Y199 K40 E49 L52 R53 Y73 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=170uM remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5ort A 2.56 BS03 A5Z A 1 E175 R179 Y199 H201 V206 E49 R53 Y73 H75 V80 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 29045126 406 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5orv A 1.88 BS03 A65 A 1 K166 R179 Y199 K40 R53 Y73 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=1297uM remove_due_to_license_issue O14965 29045126 406 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5orw A 2.0 BS03 A6E A 1 E175 R179 Y199 H201 E49 R53 Y73 H75 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=796uM remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5orx A 1.88 BS03 A6H A 1 E175 L178 Y199 H201 E49 L52 Y73 H75 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 ic50=308uM remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5ory A 1.99 BS03 AY4 A 1 E175 R179 Y199 H201 E49 R53 Y73 H75 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=357uM remove_due_to_license_issue O14965 29045126 406 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5orz A 1.92 BS03 A6W A 1 K166 L178 Y199 K40 L52 Y73 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=432uM remove_due_to_license_issue O14965 29045126 407 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5os0 A 1.74 BS03 A6Z A 1 Y199 H201 Y73 H75 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=2792uM remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5os1 A 1.9 BS03 A7H A 1 K166 E175 V182 Y199 K40 E49 V56 Y73 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=494uM remove_due_to_license_issue O14965 29045126 407 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5os2 A 1.92 BS03 A7K A 1 K166 Y199 H201 K40 Y73 H75 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T162 2.7.11.1 0004672,0005524,0006468 Kd=1821uM remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5os3 A 1.81 BS03 A7N A 1 L178 R179 Y199 L52 R53 Y73 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5os4 A 1.88 BS03 A8H A 1 E175 V182 Y199 E49 V56 Y73 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5os5 A 1.74 BS03 A8K A 1 E175 L178 R179 V182 E183 Y199 V206 E51 L54 R55 V58 E59 Y75 V82 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0004672,0005524,0006468 Kd=410uM remove_due_to_license_issue O14965 29045126 404 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPSN 5os7 B 1.66 BS01 A8Q B 1 N118 F121 L124 Y136 P159 V162 I164 M221 M225 N116 F119 L122 Y134 P157 V160 I162 M219 M223 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 402 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 5os8 A 1.55 BS01 J27 A 1 P159 V162 I164 M221 L222 M225 P157 V160 I162 M219 L220 M223 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 404 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5os8 A 1.55 BS02 J27 A 2 E52 I69 K71 P72 D103 S106 E50 I67 K69 P70 D101 S104 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 405 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5os8 A 1.55 BS03 J27 A 3 E282 V285 Q290 V293 P295 E280 V283 Q288 V291 P293 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 406 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5osd A 1.99 BS03 A9B A 1 W128 F133 E152 Y197 W4 F9 E28 Y73 D256 K258 E260 N261 D274 T292 D132 K134 E136 N137 D150 T168 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14965 29045126 404 KRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5ose A 1.9 BS03 A98 A 1 W128 E152 Y197 W2 E26 Y71 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 Kd=681uM remove_due_to_license_issue O14965 29045126 404 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 5osk A 2.11 BS02 A9Q B 1 S178 T179 A180 V181 S178 T179 A180 V181 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 29227648 507 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGV 5osk B 2.11 BS02 A9Q B 1 L242 L248 A250 L255 N258 M259 A317 I318 K352 A354 L240 L246 A247 L252 N255 M256 A309 I310 K344 A346 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 ic50=2.5uM remove_due_to_license_issue Q6B856 29227648 507 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLADLRKLAVNMVPFPRLHFFMPGFAPLTQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQD 5osl A 1.95 BS03 A9K A 1 N118 L124 P159 V162 I164 M221 M225 N117 L123 P158 V161 I163 M220 M224 D156 K158 N161 D175 S194 D155 K157 N160 D174 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 406 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5osl A 1.95 BS04 A9K A 2 E52 I69 P72 S106 E51 I68 P71 S105 D156 K158 N161 D175 S194 D155 K157 N160 D174 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 407 SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5oss B 1.7 BS01 AEZ B 1 Q20 H121 E166 Y295 E351 W398 E405 W406 F414 Q18 H119 E164 Y293 E349 W396 E403 W404 F412 R77 H121 E166 V169 N293 Y295 E351 R75 H119 E164 V167 N291 Y293 E349 3.2.1.21 0004553,0005975,0008422,0016798,0030245 Kd=28.3uM remove_due_to_license_issue Q08638 29601200 505 VKKFPEGFLWGVATASYQIEGSPLADGAGMSIWHTFSHTPGNVKNGDTGDVACDHYNRWKEDIEIIEKLGVKAYRFSISWPRILPEGTGRVNQKGLDFYNRIIDTLLEKGITPFVTIYHWDLPFALQLKGGWANREIADWFAEYSRVLFENFGDRVKNWITLNEPWVVAIVGHLYGVHAPGMRDIYVAFRAVHNLLRAHARAVKVFRETVKDGKIGIVFNNGYFEPASEKEEDIRAVRFMHQFNNYPLFLNPIYRGDYPELVLEFAREYLPENYKDDMSEIQEKIDFVGLNYYSGHLVKFDPDAPAKVSFVERDLPKTAMGWEIVPEGIYWILKKVKEEYNPPEVYITENGAAFDDVVSEDGRVHDQNRIDYLKAHIGQAWKAIQEGVPLKGYFVWSLLDNFEWAEGYSKRFGIVYVDYSTQKRIVKDSGYWYSNVVKNNGLE 5ost A 2.1 BS02 AEZ A 1 E441 Y445 D452 H507 Y523 T591 D593 E777 R786 E402 Y406 D413 H468 Y484 T552 D554 E738 R747 3.2.1.45 0004348,0004553,0005975,0006680,0008422,0016020,0016798,0046872 Kd=27.3uM remove_due_to_license_issue F6BL85 29601200 915 HKIDIPDSAWTIGIGEKFKNAGHPNVKYPMIDDSYVQGAPLGGFGAGTIGRTYNGGFSRWHLEIGKNKYTTVYANQFSVFQKVEGNKDGVAQVLYAGEPGYLSSWKWDYPKESGMYYALYPNSWYTYTNKDLPVQLAVKQFSPIIPYNYKETSYPVAVFKWTAYNPTNKNVDVSIMFTWQNMIGFFGKQVNVNSGNFNKIIKDKSKDSEIVAAVMGNISNDNEEWNGEYSIGVKKVPGVDISYKAKFVTTGDGSDLWHEFSKNGILDNKDDETPTKQDGIGSAIAVNFKLQPGQTIEVPFALSWDLPIMKFGGGDKWYKMYTKYFGKNGKNSFAILKEALNNYQKWEKMIDDWQKPILSNKSKPDWYKTALFNELYYLADGGTAWENGKVGERTNNMFGLLECFDYNYYETLDVRFYGSFPLVMLWPDIEKQVMRQFADTINVQDSSEFKVGSNGAMAVKKVQGMIPHDLGSSYALPWIKINAYDWQNPNIWKDLNSKYVLLVYRDYVLTGKTDKEFLKYTWKSVKTALDKLKEMDKDNDGIPDNEGIPDQTYDTWSMKGTSAYCGSLWLAALKAAQEIGKVLKDNEAYIKYNEWYKIAQQNFEKELWNGEYYNFDTESDHKDSIMADQLAGQWYADILRLGDILPKDHVQKALKKIYEFNVMKFENGKMGAVNGMRPDGIVDESDIQAQEVWTGVTYALASFMKYRGMTEEAYNTAYGVYKMTYDKSGKGYWFRTPEAWTKDGNYRASMYMRPLSIWSMEV 5osy A 2.06 BS01 AJQ A 1 R54 D59 I61 E85 K142 Y143 W175 E185 D205 L206 K207 Y217 H268 S272 Y273 P288 R294 R18 D23 I25 E49 K106 Y107 W139 E149 D169 L170 K171 Y181 H232 S236 Y237 P252 R258 3.6.1.59 0000290,0016787 ic50=0.0447uM remove_due_to_license_issue Q96C86 29676910 400 SAPVRLPFSGFRLQKVLRESARDKIIFLHGKVNEASGDGDGEDAVVILEKTPFQVEQVAQLLTGSPELQLQFSNDIYSTYHLFPPRQLNDVKTTVVYPATEKHLQKYLRQDLRLIRETGDDYRNITLPHLESQSLSIQWVYNILDKKAEADRIVFENPDPSDGFVLIPDLKWNQQQLDDLYLIAICHRRGIRSLRDLTPEHLPLLRNILHQGQEAILQRYRMKGDHLRVYLHYLPSYYHLHVHFTALGFEAPGSGVERAHLLAEVIENLECDPRHYQQRTLTFALRADDPLLKLLQEAQQ 5osy B 2.06 BS01 AJQ B 1 W175 E185 L206 W130 E140 L161 3.6.1.59 0000290,0016787 ic50=0.0447uM remove_due_to_license_issue Q96C86 29676910 401 VRLPFSGFRLQKVLRESARDKIIFLHGKVNEGEDAVVILEKTPFQVEQVAQLLTGSPELQLQFSNDIYSTYHLFPPRQLNDVKTTVVYPATEKHLQKYLRQDLRLIRETGDDYRNITLPHLESQSLSIQWVYNILDKKAEADRIVFENPDPSDGFVLIPDLKWNQQQLDDLYLIAICHRRGIRSLRDLTPEHLPLLRNILHQGQEAILQRYRMKGDHLRVYLHYLPSYYHLHVHFTALGFEAPGSGVERAHLLAEVIENLECDPRHYQQRTLTFALRADDPLLKLLQEAQQ 5ot3 A 2.04 BS02 9LQ A 1 G52 G55 V57 A70 K72 M120 Y122 V123 L173 T183 D184 F327 G41 G44 V46 A59 K61 M109 Y111 V112 L162 T172 D173 F316 D166 K168 N171 D184 T201 D155 K157 N160 D173 T190 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007189,0007193,0016607,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P25321 401 QESVKEFLAKAKEEFLKKWESPSQNTAQLDHFDRIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 5ot8 A 2.35 BS01 6DB A 1 E36 Y39 W77 A94 A95 S97 R102 M117 Q165 T168 S169 H170 S207 E10 Y13 W51 A68 A69 S71 R76 M91 Q139 T142 S143 H144 S181 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=52uM remove_due_to_license_issue P35120 29269740 301 DYKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMSIQPAREKVIAFSRPYLLTPMTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASPK 5ot9 A 2.45 BS01 AOZ A 1 E36 Y39 W77 A94 A95 R102 M117 Q165 T168 S169 H170 S207 E9 Y12 W50 A67 A68 R75 M90 Q138 T141 S142 H143 S180 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=84.4uM remove_due_to_license_issue P35120 29269740 303 YKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPMTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASP 5ota A 2.1 BS01 AQQ A 1 E36 Y39 W77 A95 G97 R102 M117 Q165 T168 S169 H170 S207 E9 Y12 W50 A68 G70 R75 M90 Q138 T141 S142 H143 S180 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=4.4uM remove_due_to_license_issue P35120 29269740 301 YKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPMTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASP 5otc A 2.2 BS01 AQK A 1 E36 Y39 W77 A95 G97 R102 Q165 T168 S169 H170 S207 E9 Y12 W50 A68 G70 R75 Q138 T141 S142 H143 S180 ? 0015276,0016020,0030288,0034220,0042597,0071705 Kd=23uM remove_due_to_license_issue P35120 29269740 301 YKSITIATEGSYAPYNFKDAGGKLIGFDIDLGNDLCKRMNIECKFVEQAWDGIIPSLTAGRYDAIMAAMGIQPAREKVIAFSRPYLLTPMTFLTTADSPLLKTQVAIENLPLDNITPEQKAELDKFTKIFEGVKFGVQAGTSHEAFMKQMMPSVQISTYDTIDNVVMDLKAGRIDASLASVSFLKPLTDKPDNKDLKMFGPRMTGGLFGKGVGVGIRKEDADLKALFDKAIDAAIADGTVQKLSQQWFGYDASPKQ 5otr A 1.52 BS01 AU8 A 1 L124 Y125 P159 V162 I164 M221 M225 L122 Y123 P157 V160 I162 M219 M223 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 403 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5otr A 1.52 BS02 AU8 A 2 E282 V285 Q290 V293 P295 E280 V283 Q288 V291 P293 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 405 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5otz A 1.46 BS02 AUT A 1 F121 L124 Y125 P159 V162 I164 M221 M225 F119 L122 Y123 P157 V160 I162 M219 M223 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 Kd=6.5uM remove_due_to_license_issue P68400 29732088 404 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5ou1 A 1.78 BS02 AUQ A 1 A145 G285 E318 A131 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 Ki=0.86uM remove_due_to_license_issue G7CNL4 29547284 502 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 5ou2 A 1.45 BS02 36Y A 1 H146 N149 E318 H132 N135 E280 1.1.1.205 0003824,0003938,0006164,0016491 Ki=609uM remove_due_to_license_issue G7CNL4 29547284 502 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 5ou2 A 1.45 BS03 36Y A 2 A145 N173 E318 A131 N159 E280 1.1.1.205 0003824,0003938,0006164,0016491 Ki=609uM remove_due_to_license_issue G7CNL4 29547284 503 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 5ou3 A 1.6 BS02 AUN A 1 D143 H146 N173 G285 E318 D130 H133 N160 G272 E282 1.1.1.205 0003824,0003938,0006164,0016491 Ki=0.61uM remove_due_to_license_issue G7CNL4 29547284 401 PVPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQGVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAGL 5oug A 2.57 BS02 9Z0 A 1 L54 I88 R96 L55 I89 R97 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 1104 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug A 2.57 BS03 9Z0 A 2 Y7 E9 L10 L63 Q64 Y70 V107 Y8 E10 L11 L64 Q65 Y71 V108 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 1105 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oug A 2.57 BS05 9Z0 E 1 L100 T101 L101 T102 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 301 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5ouh A 2.5 BS01 L0B A 1 Y91 W145 C186 Y191 Y92 W146 C187 Y192 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5ouh A 2.5 BS02 L0B E 1 W53 L106 L116 W54 L107 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 304 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5ouh B 2.5 BS01 L0B A 1 W53 L106 Q114 L116 W54 L107 Q115 L117 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5ouh B 2.5 BS02 L0B C 1 Y91 W145 Y92 W146 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 304 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oui A 3.1 BS01 AVB A 1 E158 A159 V175 T176 Q177 F196 E159 A160 V176 T177 Q178 F197 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue 29237730 306 GEFQRKLYKELVKNYNPDVIPTQRDRPVTVYFSLSLLQIMDVDEKNQVVDVVIWLQMSWTDHYLQWNVSEYPGVKQVSVPISSLWKPDILLYNAIERPEVLTPQLALVNSSGHVQYLPSIRQRFSCDVSGVDTESGATCKLKFGSWTHHSRELDLQMQEADISGYIPYSRFELVGVTQKRSERFYECCKEPYPDVTFTVTFRKKG 5oul A 1.34 BS01 AWE A 1 L128 I133 M137 P159 V162 I164 M221 M225 L126 I131 M135 P157 V160 I162 M219 M223 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 403 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5oul A 1.34 BS02 AWE A 2 Q290 V293 P295 L298 Q288 V291 P293 L296 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 404 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5oul A 1.34 BS03 AWE A 3 E282 R283 V285 Q290 E280 R281 V283 Q288 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 405 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5oul A 1.34 BS04 AWE A 4 E52 I69 K71 P72 D103 S106 E50 I67 K69 P70 D101 S104 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 406 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5oul A 1.34 BS05 AWE A 5 L45 V66 V116 N118 M163 L43 V64 V114 N116 M161 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 407 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5oul A 1.34 BS06 AWE A 6 H160 N161 H158 N159 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29732088 408 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 5ov8 A 1.8 BS01 AXN A 1 I652 F653 V657 P658 E661 Y707 N708 F714 I24 F25 V29 P30 E33 Y79 N80 F86 ? Kd=18uM remove_due_to_license_issue Kd=18000nM, IC50=11000nM P55201 29902720 801 QLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5ov9 A 2.4 BS01 CVI A 1 D74 L76 Y341 D74 L76 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=2.2uM remove_due_to_license_issue P21836 28867801 608 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 5ov9 A 2.4 BS02 CVI A 2 Y72 D283 W286 H287 Y341 Y72 D276 W279 H280 Y334 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G121 G122 G154 S203 A204 G242 F290 F292 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 ic50=2.2uM remove_due_to_license_issue P21836 28867801 609 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLS 5ove A 1.85 BS01 AXE A 1 M878 N879 Y884 F890 K898 L901 H905 M306 N307 Y312 F318 K326 L329 H333 ? 0005085,0007264 ic50=320nM remove_due_to_license_issue Q07889 30683722 1104 GAMAEEQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIARDTFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSN 5ovf A 2.01 BS01 AWT A 1 M878 N879 Y884 F890 K898 E902 H905 M305 N306 Y311 F317 K325 E329 H332 ? 0005085,0007264 ic50=140nM remove_due_to_license_issue Q07889 30683722 1101 GAMAEEQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIARDFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 5ovg A 2.3 BS01 AWZ A 1 N879 Y884 D887 F890 L901 E902 H905 N290 Y295 D298 F301 L312 E313 H316 ? 0005085,0007264 ic50=400nM remove_due_to_license_issue Q07889 30683722 1101 AEEQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIARDTFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSN 5ovh A 2.3 BS01 AWW A 1 M878 N879 V883 Y884 F890 E902 H905 M288 N289 V293 Y294 F300 E312 H315 ? 0005085,0007264 ic50=280nM remove_due_to_license_issue Q07889 30683722 1101 GAMAEEQMRLPSADVYRFAEPDSEENIIFEAGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIARDITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNP 5ovi A 2.2 BS01 AXH A 1 N879 V883 Y884 D887 F890 L901 E902 H905 N301 V305 Y306 D309 F312 L323 E324 H327 ? 0005085,0007264 ic50=21nM remove_due_to_license_issue Q07889 30683722 2001 QMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIARDTFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSN 5ovr A 2.15 BS01 AXK A 1 N376 E378 E379 S434 W435 P436 D437 K439 R443 R478 Q520 N126 E128 E129 S184 W185 P186 D187 K189 R193 R228 Q270 D437 C472 R478 T479 Q516 D187 C222 R228 T229 Q266 3.1.3.48 0004725,0006470,0016311 Kd=27.2uM remove_due_to_license_issue P54829 29116812 601 NLYFQSMSRVLQAEELHEKALDPFLLQAEFFEIPMNFVDPKEYDIPGLVRKNRYKTILPNPHSRVCLTSPDPDDPLSSYINANYIRGYGGEEKVYIATQGPIVSTVADFWRMVWQEHTPIIVMITNIEEMNEKCTEYWPEEQVAYDGVEITVQKVIHTEDYRLRLISLKSGTEERGLKHYWFTSWPDQKTPDRAPPLLHLVREVEEAAQQEGPHCAPIIVHCSAGIGRTGCFIATSICCQQLRQEGVVDILKTTCQLRQDRGGMIQTCEQYQFVHHVMSLYEKQLSH 5ovx A 2.1 BS01 AY5 A 1 N376 E378 E379 S434 W435 P436 D437 K439 R443 R478 Q520 N126 E128 E129 S184 W185 P186 D187 K189 R193 R228 Q270 D437 C472 R478 T479 Q516 D187 C222 R228 T229 Q266 3.1.3.48 0004725,0006470,0016311 Kd=31.4uM remove_due_to_license_issue P54829 29116812 601 NLYFQSMSRVLQAEELHEKALDPFLLQAEFFEIPMNFVDPKEYDIPGLVRKNRYKTILPNPHSRVCLTSPDPDDPLSSYINANYIRGYGGEEKVYIATQGPIVSTVADFWRMVWQEHTPIIVMITNIEEMNEKCTEYWPEEQVAYDGVEITVQKVIHTEDYRLRLISLKSGTEERGLKHYWFTSWPDQKTPDRAPPLLHLVREVEEAAQQEGPHCAPIIVHCSAGIGRTGCFIATSICCQQLRQEGVVDILKTTCQLRQDRGGMIQTCEQYQFVHHVMSLYEKQLSH 5ow1 A 2.05 BS01 AY8 A 1 Y304 W435 K439 A474 R478 Q516 Q520 Y54 W182 K186 A221 R225 Q263 Q267 D437 C472 R478 T479 Q516 D184 C219 R225 T226 Q263 3.1.3.48 0004725,0006470,0016311 Kd=70.4uM remove_due_to_license_issue Kd=70400nM, Ki=20000nM P54829 29116812 601 NLYFQSMSRVLQAEELHEKALDPFLLQAEFFEIPMNFVDPKEYDIPGLVRKNRYKTILPNPHSRVCLTSPDPDDPLSSYINANYIRGYGGEEKVYIATQGPIVSTVADFWRMVWQEHTPIIVMITNIEEMCTEYWPEEQVAYDGVEITVQKVIHTEDYRLRLISLKSGTEERGLKHYWFTSWPDQKTPDRAPPLLHLVREVEEAAQQEGPHCAPIIVHCSAGIGRTGCFIATSICCQQLRQEGVVDILKTTCQLRQDRGGMIQTCEQYQFVHHVMSLYEKQLSH 5ow8 A 1.9 BS02 AYN A 1 I2 L5 Y20 G28 L29 C43 H46 D47 I2 L5 Y20 G28 L29 C43 H46 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 ic50=6.9uM remove_due_to_license_issue IC50=6900nM O15496 30034585 206 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD 5owa A 1.95 BS01 B0H A 1 F653 V657 P658 Y707 N708 F714 F24 V28 P29 Y78 N79 F85 ? Kd=3.5uM remove_due_to_license_issue IC50=30600nM, Kd=3500nM P55201 29902720 801 LTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5owc A 1.75 BS02 AYZ A 1 L5 P17 Y20 G28 L29 G30 C43 H46 D47 L5 P17 Y20 G28 L29 G30 C43 H46 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0001516,0001669,0002532,0003847,0004620,0004623,0005509,0005515,0005543,0005576,0005615,0005764,0006629,0006644,0006658,0007411,0009566,0010744,0010884,0016042,0016787,0019369,0031069,0031410,0032308,0034374,0034638,0036335,0042116,0042632,0043030,0043249,0043433,0046337,0046470,0046471,0046473,0046872,0047498,0047499,0050482,0050728,0051247,0051607,0051977,0062234,0090238,0090370,1900016,1990830,2000344 ic50=0.026uM remove_due_to_license_issue IC50=26nM O15496 30034585 202 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKC 5owf A 1.91 BS01 GLN A 1 Y35 F73 S90 S91 S93 R98 K138 S141 T142 D182 Y11 F49 S66 S67 S69 R74 K114 S117 T118 D158 ? 0006865,0030288,0042597,0071705 Kd=1.59uM remove_due_to_license_issue P02911 29524280 320 QTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVKQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 5owh A 2.3 BS01 B0K A 1 V53 K68 F113 N118 M163 I174 D175 W176 V52 K67 F112 N117 M162 I173 D174 W175 D156 K158 N161 D175 S194 D155 K157 N160 D174 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29966873 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARMG 5owl A 2.23 BS01 B0K A 1 V53 V66 K68 F113 V116 M163 I174 D175 V52 V65 K67 F112 V115 M162 I173 D174 D156 K158 N161 D175 S194 D155 K157 N160 D174 S193 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29966873 401 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 5owt A 2.2 BS01 F37 A 1 H1031 G1032 P1034 F1035 H1048 A1049 Y1050 Y1060 S1068 Y1071 H80 G81 P83 F84 H97 A98 Y99 Y109 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 29374194 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5owt B 2.2 BS01 F37 B 1 H1031 G1032 F1035 H1048 A1049 Y1050 Y1060 A1062 S1068 Y1071 H80 G81 F84 H97 A98 Y99 Y109 A111 S117 Y120 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue Q9H2K2 29374194 1203 GTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE 5ox5 A 2.251 BS02 B2E A 1 D254 M299 Y303 Y310 H313 Y329 L343 H374 V376 R383 D67 M112 Y116 Y123 H126 Y142 L156 H187 V189 R196 1.14.11.29 0005506,0016705,0031418 ic50=2.6uM remove_due_to_license_issue Q9GZT9 29435217 502 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYVRVEL 5ox6 A 1.99 BS02 A1Z A 1 M299 Y303 Y310 H313 D315 Y329 H374 V376 R383 M112 Y116 Y123 H126 D128 Y142 H187 V189 R196 1.14.11.29 0005506,0016705,0031418 ic50=0.029uM remove_due_to_license_issue IC50=410nM Q9GZT9 29435217 502 LPALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYLKGVRV 5oxg A 2.13 BS01 B4B A 1 V214 V222 A233 K235 L263 T283 H286 E287 G289 D293 L343 V12 V20 A31 K33 L61 T78 H81 E82 G84 D88 L138 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=26nM Q04771 28918311 501 TVARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKI 5oxk A 2.38 BS14 ALA A 1 N156 N328 E400 N151 N311 E379 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 518 KTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMIVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAWPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPNSQMMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFLS 5oxk A 2.38 BS15 GLN A 1 R26 Y30 Y68 K126 I155 W296 W427 S431 R21 Y25 Y63 K121 I150 W279 W392 S396 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 519 KTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMIVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAWPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPNSQMMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFLS 5oxl A 2.66 BS09 ALA A 1 Y30 N156 N328 Y26 N152 N316 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 516 GKTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMTEHLRVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAWPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPVGLSVAFNSQMMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFL 5oxl A 2.66 BS10 LEU A 1 R26 Y30 K126 I155 W296 W427 R22 Y26 K122 I151 W284 W404 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 517 GKTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMTEHLRVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAWPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPVGLSVAFNSQMMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFL 5oxm A 2.295 BS19 ASP A 1 Y30 E299 N328 Y25 E287 N316 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 521 KTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMSTEHLRVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAQPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPVMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFLS 5oxm A 2.295 BS20 GLU A 1 R26 Y30 Y68 K126 I155 S431 R21 Y25 Y63 K121 I150 S398 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 522 KTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMSTEHLRVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAQPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPVMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFLS 5oxn A 2.196 BS13 PHE A 1 Y30 E299 N328 E400 Y26 E290 N319 E391 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 516 GKTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMISSTEHLRVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAWKKNQPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPVGLSVTTKLSQMMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFLSKRIQGL 5oxn A 2.196 BS14 ALA A 1 Y68 W296 Y64 W287 ? 0005886,0006857,0015833,0016020,0022857,0042802,0055085,1904680 remove_due_to_license_issue Q5M4H8 29429879 517 GKTFFGQPLGLSTLFMTEMWERFSYYGMRAILLYYMWFLISTGDLHITRATAASIMAIYASMVYLSGTIGGFVADRIIGARPAVFWGGVLIMLGHIVLALPFGASALFGSIILIIIGTGFLKPNVSTLVGTLYDEHDRRRDAGFSIFVFGINLGAFIAPLIVGAAQEAAGYHVAFSLAAIGMFIGLLVYYFGGKKTLDPHYLRPTDPLAPEEVKPLLVKVSLAVAGFIAIIVVMNLVGWNSLPAYINLLTIVAIAIPVFYFAWMISSTEHLRVVSYIPLFIAAVLFWAIEEQGSVVLATFAAERVDSSWFPVSWFQSLNPLFIMLYTPFFAWLWTAWKKNQPSSPTKFAVGLMFAGLSFLLMAIPGALYGTSGKVSPLWLVGSWALVILGEMLISPVGLSVTTKLSQMMSMWFLSSSVGSALNAQLVTLYNAKSEVAYFSYFGLGSVVLGIVLVFLSKRIQGL 5oyd A 2.1 BS01 NBG C 1 H208 N254 E255 H323 Y325 E390 W432 H113 N159 E160 H228 Y230 E295 W337 3.2.1.4 0000272,0004553 remove_due_to_license_issue B3PD52 29467823 1 GLYPSYNTSPAAPDSTGMQSTAVQLAGKIRLGWNIGNTMEAIGGETAWGNPMVSNELLKLVKDSGFDAVRIPVAWDQYANQESAEISAAWLNRVKQVVQMAIDNELYVLINIHWDGGWLENNITPAKKDENNAKQKAFWEQIATHLRDFDEHLLFAGTNEPNAENAEQMDVLNSYLQTFVDAVRSTGGKNAYRVLVLQGPVTDIEKTNELWTHMPADTATDRLMAEVHFYTPYNFALMRQDESWGKQFYYWGEGFLSTTDTERNPTWGEEATIDQLFDLMKTKFVDQGIPVVLGEFSAMRRTNLTGDALTLHLAGRAYYHKYVTQQALARGLLPFYWDNGGNDNFSSGIFNRQQNTVFDQQVLDALLEGA 5oyd A 2.1 BS02 BGC C 1 N132 W143 N434 N37 W48 N339 3.2.1.4 0000272,0004553 remove_due_to_license_issue B3PD52 29467823 2 GLYPSYNTSPAAPDSTGMQSTAVQLAGKIRLGWNIGNTMEAIGGETAWGNPMVSNELLKLVKDSGFDAVRIPVAWDQYANQESAEISAAWLNRVKQVVQMAIDNELYVLINIHWDGGWLENNITPAKKDENNAKQKAFWEQIATHLRDFDEHLLFAGTNEPNAENAEQMDVLNSYLQTFVDAVRSTGGKNAYRVLVLQGPVTDIEKTNELWTHMPADTATDRLMAEVHFYTPYNFALMRQDESWGKQFYYWGEGFLSTTDTERNPTWGEEATIDQLFDLMKTKFVDQGIPVVLGEFSAMRRTNLTGDALTLHLAGRAYYHKYVTQQALARGLLPFYWDNGGNDNFSSGIFNRQQNTVFDQQVLDALLEGA 5oyd A 2.1 BS03 BGC C 2 A142 W143 A47 W48 3.2.1.4 0000272,0004553 remove_due_to_license_issue B3PD52 29467823 4 GLYPSYNTSPAAPDSTGMQSTAVQLAGKIRLGWNIGNTMEAIGGETAWGNPMVSNELLKLVKDSGFDAVRIPVAWDQYANQESAEISAAWLNRVKQVVQMAIDNELYVLINIHWDGGWLENNITPAKKDENNAKQKAFWEQIATHLRDFDEHLLFAGTNEPNAENAEQMDVLNSYLQTFVDAVRSTGGKNAYRVLVLQGPVTDIEKTNELWTHMPADTATDRLMAEVHFYTPYNFALMRQDESWGKQFYYWGEGFLSTTDTERNPTWGEEATIDQLFDLMKTKFVDQGIPVVLGEFSAMRRTNLTGDALTLHLAGRAYYHKYVTQQALARGLLPFYWDNGGNDNFSSGIFNRQQNTVFDQQVLDALLEGA 5prc L 2.35 BS04 ATZ L 1 E212 F216 V220 Y222 S223 I224 G225 I229 E212 F216 V220 Y222 S223 I224 G225 I229 ? 0009772,0015979,0016020,0019684,0030077,0042314,0042717,0045156,0046872 remove_due_to_license_issue P06009 10024457 502 ALLSFERKYRVRGGTLIGGDLFDFWVGPYFVGFFGVSAIFFIFLGVSLIGYAASQGPTWDPFAISINPPDLKYGLGAAPLLEGGFWQAITVCALGAFISWMLREVEISRKLGIGWHVPLAFCVPIFMFCVLQVFRPLLLGSWGHAFPYGILSHLDWVNNFGYQYLNWHYNPGHMSSVSFLFVNAMALGLHGGLILSVANPGDGDKVKTAEHENQYFRDVVGYSIGALSIHRLGLFLASNIFLTGAFGTIASGPFWTRGWPEWWGWWLDIPFWS 5pzn A 2.25 BS02 8XP A 1 F193 P197 R200 L204 L314 I363 S365 C366 S368 M414 Y448 Y452 F165 P169 R172 L176 L286 I335 S337 C338 S340 M386 Y420 Y424 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 28430437 602 SMSYTWTGALITPCVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSLSRARPRWFM 5q0d A 2.12 BS01 9EY A 1 R39 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=1nM remove_due_to_license_issue Ki=<5nM P03951 28687203 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5q0e A 2.12 BS01 9FD A 1 R39 H40 L41 H57 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.69nM remove_due_to_license_issue Ki=0.690000nM P03951 28687203 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5q0f A 2.12 BS02 9FA A 1 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.13nM remove_due_to_license_issue Ki=0.130000nM P03951 28687203 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5q0g A 2.6 BS01 9F7 A 1 R39 H40 L41 H57 C58 I151 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 C45 I141 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue Ki=0.180000nM P03951 28687203 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5q0h A 2.5 BS01 9F1 A 1 R39 H40 L41 H57 I151 C191 K192 G193 S195 S214 W215 G216 R26 H27 L28 H44 I141 C184 K185 G186 S188 S207 W208 G209 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=12nM remove_due_to_license_issue Ki=12nM P03951 28687203 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5q0i A 1.7 BS02 0X0 A 1 N287 L291 M294 H298 M332 F333 S336 I339 I356 F370 Y373 W458 N41 L45 M48 H52 M86 F87 S90 I93 I110 F124 Y127 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=56100nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNKFTPLLCEIWDV 5q0j A 2.0 BS02 9KV A 1 M294 H298 M332 F333 R335 S336 I339 Y373 L455 M48 H52 M86 F87 R89 S90 I93 Y127 L209 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=239nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0l A 2.5 BS02 9KY A 1 I273 N287 M294 H298 M332 F333 S336 I339 I356 M369 Y373 M454 I27 N41 M48 H52 M86 F87 S90 I93 I110 M123 Y127 M208 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=5240nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0m A 2.2 BS02 9L1 A 1 M269 T274 T292 M294 R335 I339 H451 M23 T28 T46 M48 R89 I93 H205 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=7.900000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWKFTPLLCEIWD 5q0n A 2.4 BS02 9L4 A 1 I273 I277 L291 M294 A295 M332 F333 R335 S336 I339 F340 I356 M369 Y373 I27 I31 L45 M48 A49 M86 F87 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue EC50=300nM, IC50=9nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDV 5q0o A 1.9 BS02 9L7 A 1 N287 M294 H298 M332 F333 S336 I339 I356 Y373 H451 L455 W458 W473 N41 M48 H52 M86 F87 S90 I93 I110 Y127 H205 L209 W212 W227 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=24.400000nM Q96RI1 29204945 502 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0p A 1.8 BS02 9LA A 1 I273 I277 M294 M332 F333 R335 S336 I339 F340 I356 S359 M369 Y373 I27 I31 M48 M86 F87 R89 S90 I93 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=39nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0q A 2.6 BS02 9LD A 1 M269 F288 L291 T292 M294 A295 H298 M332 R335 S336 I339 L352 H451 M454 W473 M23 F42 L45 T46 M48 A49 H52 M86 R89 S90 I93 L106 H205 M208 W220 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=785nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSFTPLLCEIWD 5q0r A 1.91 BS02 9LG A 1 F288 L291 T292 M294 A295 H298 M332 S336 I339 F340 S349 L352 E353 I356 M369 Y373 H451 W473 F42 L45 T46 M48 A49 H52 M86 S90 I93 F94 S103 L106 E107 I110 M123 Y127 H205 W223 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=27100nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWHKFTPLLCEIWD 5q0s A 2.5 BS02 9LJ A 1 I277 N287 L291 M294 M332 F333 S336 I339 F340 I356 S359 M369 Y373 I31 N41 L45 M48 M86 F87 S90 I93 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=62nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0t A 2.14 BS02 9LM A 1 F288 L291 T292 M294 A295 M332 R335 S336 I339 L352 I356 Y373 H451 F465 W473 F42 L45 T46 M48 A49 M86 R89 S90 I93 L106 I110 Y127 H205 F212 W220 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=29000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLHKFTPLLCEIWDV 5q0u A 1.9 BS02 9LP A 1 Q267 R268 I273 I277 L291 M294 H298 M332 F333 R335 S336 F340 I356 M369 Y373 Q21 R22 I27 I31 L45 M48 H52 M86 F87 R89 S90 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=175nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0v A 1.87 BS02 9LS A 1 I277 N287 L291 M294 H298 M332 S336 I339 F340 I356 M369 Y373 I31 N41 L45 M48 H52 M86 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=20.500000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0w A 1.9 BS02 9LV A 1 Q267 M269 L291 M294 N297 H298 V301 M332 F333 S336 I339 M369 H451 M454 W458 W473 Q21 M23 L45 M48 N51 H52 V55 M86 F87 S90 I93 M123 H205 M208 W212 W227 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=58nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWD 5q0x A 2.26 BS02 643 A 1 M269 F288 L291 M294 A295 F333 R335 S336 I339 M369 Y373 M23 F42 L45 M48 A49 F87 R89 S90 I93 M118 Y122 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=94nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVHKFTPLLCEIWDV 5q0y A 2.2 BS02 9LY A 1 I277 N287 L291 M294 H298 M332 F333 S336 I339 F340 I356 S359 M369 Y373 M454 L455 I31 N41 L45 M48 H52 M86 F87 S90 I93 F94 I110 S113 M123 Y127 M208 L209 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=1870nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q0z A 2.26 BS02 9M1 A 1 I273 L291 M294 A295 M332 S336 F340 I356 M369 Y373 L455 W458 I27 L45 M48 A49 M86 S90 F94 I110 M123 Y127 L209 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue Q96RI1 29204945 500 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q10 A 2.2 BS02 9M4 A 1 F288 L291 T292 A295 M332 F333 Y365 M369 Y373 H451 M454 T466 W473 F42 L45 T46 A49 M86 F87 Y119 M123 Y127 H205 M208 T220 W227 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=6280nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIW 5q11 A 2.2 BS02 9M7 A 1 F288 L291 T292 M294 A295 M332 F333 S336 L352 Y365 M369 Y373 M454 W473 F42 L45 T46 M48 A49 M86 F87 S90 L106 Y119 M123 Y127 M207 W221 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=7190nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPNPQHFACLLGRLTELRTFNHHHAEMLMSHKFTPLLCEIW 5q12 A 2.0 BS02 9MA A 1 F288 L291 T292 A295 M332 F333 S336 M369 H451 L455 T466 L469 F42 L45 T46 A49 M86 F87 S90 M123 H205 L209 T220 L223 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=4640nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWD 5q13 A 1.9 BS02 9MD A 1 I273 L291 M294 H298 M332 F333 R335 S336 I339 F340 L352 I356 S359 M369 Y373 M454 I29 L47 M50 H54 M88 F89 R91 S92 I95 F96 L108 I112 S115 M125 Y129 M210 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=91nM Q96RI1 29204945 501 SHMELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q14 A 1.85 BS02 9MM A 1 I277 N287 M294 H298 M332 F333 R335 S336 I339 F340 I356 S359 M369 Y373 I31 N41 M48 H52 M86 F87 R89 S90 I93 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=21nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q15 A 1.9 BS02 9MP A 1 I277 N287 L291 H298 M332 S336 I339 F340 I356 S359 I361 M369 Y373 W458 I31 N41 L45 H52 M86 S90 I93 F94 I110 S113 I115 M123 Y127 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=8.900000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q16 A 2.0 BS02 9MS A 1 N287 L291 M294 H298 M332 F333 S336 I339 I356 S359 Y373 M454 L455 W458 N41 L45 M48 H52 M86 F87 S90 I93 I110 S113 Y127 M208 L209 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=13.500000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q17 A 2.1 BS02 9MV A 1 M269 P270 L291 M294 H298 M332 S336 I339 W473 M24 P25 L46 M49 H53 M87 S91 I94 W223 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=5640nM Q96RI1 29204945 501 HMELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSHKFTPLLCEIWD 5q18 A 1.9 BS02 9MY A 1 I277 H298 M332 S336 F340 I356 S359 I361 M369 Y373 W458 I31 H52 M86 S90 F94 I110 S113 I115 M123 Y127 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=67.500000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q19 A 1.98 BS02 9N1 A 1 N287 L291 M294 H298 M332 F333 S336 I339 I356 S359 I361 M369 Y373 M454 W458 N41 L45 M48 H52 M86 F87 S90 I93 I110 S113 I115 M123 Y127 M208 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=59.600000nM Q96RI1 29204945 500 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q1a A 2.0 BS02 9N4 A 1 N287 L291 M294 H298 M332 F333 S336 I356 S359 M369 Y373 M454 N41 L45 M48 H52 M86 F87 S90 I110 S113 M123 Y127 M208 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=9.600000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q1b A 2.3 BS02 9N7 A 1 I273 I277 L291 M294 M332 F333 R335 S336 F340 I356 Y373 L455 I27 I31 L45 M48 M86 F87 R89 S90 F94 I110 Y127 L209 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=48.700000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q1c A 2.3 BS02 9NA A 1 I273 I277 N287 L291 M294 M332 F333 S336 I339 F340 I356 I361 M369 Y373 I26 I30 N40 L44 M47 M85 F86 S89 I92 F93 I109 I114 M122 Y126 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=8.400000nM Q96RI1 29204945 501 ELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q1d A 1.89 BS02 9ND A 1 I277 N287 L291 M294 H298 M332 F333 S336 I339 F340 I356 M369 Y373 I31 N41 L45 M48 H52 M86 F87 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=760nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 5q1e A 1.85 BS02 9NG A 1 Q267 M269 P270 L291 M294 N297 V301 M332 S336 I339 F340 L352 W473 Q21 M23 P24 L45 M48 N51 V55 M86 S90 I93 F94 L106 W223 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRKFTPLLCEIWD 5q1f A 2.3 BS02 9NJ A 1 I273 I277 N287 L291 M294 H298 M332 R335 S336 I339 F340 I356 M369 Y373 I27 I31 N41 L45 M48 H52 M86 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=72.500000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDV 5q1g A 2.0 BS02 9NM A 1 L291 M294 M332 S336 I339 F340 I356 Y373 H451 W458 W473 L40 M43 M81 S85 I88 F89 I105 Y122 H200 W207 W222 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=263000nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDV 5q1h A 2.2 BS02 9NP A 1 N287 L291 M294 H298 M332 F333 S336 I339 I356 S359 I361 Y373 H451 M454 L455 W458 N41 L45 M48 H52 M86 F87 S90 I93 I110 S113 I115 Y127 H205 M208 L209 W212 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=6250nM Q96RI1 29204945 500 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDV 5q1i A 1.95 BS02 9O1 A 1 L291 M294 A295 H298 M332 F333 S336 I339 L352 I356 M369 Y373 W473 L45 M48 A49 H52 M86 F87 S90 I93 L105 I109 M122 Y126 W226 ? 0003677,0004879,0006355,0032052,0038183 remove_due_to_license_issue IC50=570nM Q96RI1 29204945 501 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWD 5qa4 A 1.95 BS01 TI7 A 1 Y117 Y211 R250 Y94 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=170uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qa5 A 1.95 BS01 L5D A 1 I102 Y211 R250 I79 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=300uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qa6 A 1.95 BS01 AUV A 1 I102 Y211 R250 I79 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=175uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qa7 A 1.82 BS01 IQQ A 1 I102 Y211 R250 I79 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=110uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qa8 A 2.5 BS01 JSX A 1 I102 T209 Y211 L247 R250 I79 T186 Y188 L224 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=170uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qa9 A 1.9 BS01 QKU A 1 I102 Y211 R250 I79 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=230uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qaa A 1.95 BS01 EAJ A 1 I102 Y211 R250 I79 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=123uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qab A 2.15 BS01 XEV A 1 Y211 R250 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=226uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qac A 2.0 BS01 U4J A 1 Y211 R250 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=250uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qad A 1.75 BS01 WVV A 1 Y211 R250 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=170uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qae A 2.1 BS01 Q4G A 1 Y211 R250 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=240uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qaf A 2.15 BS01 S1D A 1 T209 R250 T186 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=312uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qag A 2.3 BS01 Q2R A 1 Y211 R250 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=200uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qah A 1.95 BS01 EFX A 1 S70 T209 G210 Y211 L247 R250 S47 T186 G187 Y188 L224 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=144uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qai A 1.9 BS01 VM7 A 1 I102 R250 I79 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=150uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qaj A 2.0 BS01 VBC A 1 T209 R250 T186 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=330uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qak A 1.9 BS01 AV4 A 1 I102 R250 I79 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=220uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qal A 1.95 BS01 TVZ A 1 Y117 T209 R250 Y94 T186 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=350uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qam A 1.87 BS01 GA6 A 1 S70 S118 T209 G210 Y211 S244 R250 S47 S95 T186 G187 Y188 S221 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=100uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qan A 2.3 BS01 M8Q A 1 I102 T209 Y211 T213 R250 I79 T186 Y188 T190 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=110uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qao A 2.0 BS01 Z8R A 1 I102 Y211 R250 I79 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=240uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qap B 1.79 BS01 AV7 B 1 S70 V120 L158 R214 R250 S47 V97 L135 R191 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=100uM remove_due_to_license_issue Q6XEC0 29348071 302 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qaq B 2.4 BS01 S1C B 1 Y117 T209 Y211 R250 Y94 T186 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=290uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qar A 2.1 BS01 QIU A 1 S70 I102 S118 T209 G210 Y211 R250 S47 I79 S95 T186 G187 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=170uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qas A 1.9 BS01 CVF A 1 D101 I102 R250 D78 I79 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=190uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qat A 1.9 BS01 T7O A 1 Y211 T213 R250 Y188 T190 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=140uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qau C 1.75 BS01 V7V C 1 S70 S118 T209 G210 Y211 R250 S47 S95 T186 G187 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=70uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qav C 1.72 BS01 L43 C 1 W105 L158 R214 R250 W82 L135 R191 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=70uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qaw A 2.2 BS01 TVC A 1 S70 S118 T209 G210 Y211 S244 R250 S47 S95 T186 G187 Y188 S221 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=400uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qax A 2.31 BS01 Q92 A 1 S118 T209 G210 Y211 S244 L247 R250 S95 T186 G187 Y188 S221 L224 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=160uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qay A 1.7 BS01 X6P A 1 T209 Y211 R250 T186 Y188 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=590uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qaz A 2.2 BS01 Q2S A 1 T209 S244 R250 T186 S221 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=400uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qb0 A 1.95 BS01 AVA A 1 I102 T104 Y117 R250 I79 T81 Y94 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=159uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qb1 B 1.8 BS01 F1C B 1 S70 V120 Y211 R214 S244 R250 S47 V97 Y188 R191 S221 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=20uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qb2 A 1.75 BS01 U3M A 1 S70 I102 T104 W105 Y117 V120 L158 T209 G210 R250 S47 I79 T81 W82 Y94 V97 L135 T186 G187 R227 S70 K73 S118 Y123 W157 Y211 S47 K50 S95 Y100 W134 Y188 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=70uM remove_due_to_license_issue Q6XEC0 29348071 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qb3 A 2.0 BS01 AVM A 1 S70 V120 L158 T209 Y211 R214 S244 L247 R250 S46 V96 L134 T185 Y187 R190 S220 L223 R226 S70 K73 S118 Y123 W157 Y211 S46 K49 S94 Y99 W133 Y187 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0046677,0046872,0071555 Kd=49uM remove_due_to_license_issue Q6XEC0 29348071 301 WQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLPASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 5qbv A 1.796 BS01 N2D A 1 G62 G68 G69 F70 T73 V162 G165 F211 G63 G69 G70 F71 T74 V163 G166 F212 Q19 S25 H164 N184 Q20 S26 H165 N185 3.4.22.27 0006508,0008234 remove_due_to_license_issue IC50=430nM P25774 20541404 901 ILPDSVDWREKGCVTEVKYQGSCGASWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEILQ 5qby A 2.25 BS01 N2A A 1 G62 K64 G68 G69 F70 M71 T73 E115 V162 G165 F211 G63 K65 G69 G70 F71 M72 T74 E116 V163 G166 F212 Q19 S25 H164 N184 Q20 S26 H165 N185 3.4.22.27 0006508,0008234 remove_due_to_license_issue IC50=40nM P25774 20541404 901 ILPDSVDWREKGCVTEVKYQGSCGASWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEIL 5qc4 A 2.0 BS01 BC7 A 1 K64 N67 G68 G69 F70 M71 V162 N163 H164 G165 F211 K65 N68 G69 G70 F71 M72 V163 N164 H165 G166 F212 Q19 S25 H164 N184 Q20 S26 H165 N185 3.4.22.27 0006508,0008234 ic50=0.15uM remove_due_to_license_issue IC50=150nM P25774 20188543 901 ILPDSVDWREKGCVTEVKYQGSCGASWAFSAVGALEAQLKLKTGKLVSLSAQNLVDCSTEKYGNKGCNGGFMTTAFQYIIDNKGIDSDASYPYKAMDQKCQYDSKYRAATCSKYTELPYGREDVLKEAVANKGPVSVGVDARHPSFFLYRSGVYYEPSCTQNVNHGVLVVGYGDLNGKEYWLVKNSWGHNFGEEGYIRMARNKGNHCGIASFPSYPEILQG 5qck A 2.64 BS01 BUV A 1 R39 L41 C42 H57 C58 Y143 I151 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 V227 R26 L28 C29 H44 C45 Y134 I141 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue Ki=23nM P03951 29077405 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qcl A 2.11 BS01 BUY A 1 H57 Y143 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 H44 Y134 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=11nM remove_due_to_license_issue Ki=10.32nM P03951 29077405 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qcm A 2.2 BS01 BVJ A 1 H57 I151 A190 C191 K192 G193 S195 T213 S214 W215 G216 G218 C219 V227 H44 I141 A183 C184 K185 G186 S188 T206 S207 W208 G209 G211 C212 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=110nM remove_due_to_license_issue Ki=110nM P03951 29077405 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qcn A 2.3 BS01 BVM A 1 R39 H57 Y143 I151 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 V227 R26 H44 Y134 I141 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=6nM remove_due_to_license_issue P03951 29077405 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qik A 1.58 BS01 J2M A 1 I211 A230 K232 L260 S280 H283 G286 K337 L340 D351 I15 A34 K36 L64 S84 H87 G90 K141 L144 D155 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue P36897 30429955 601 GHMTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQE 5qil A 1.98 BS01 J2V A 1 I211 K213 G214 V219 A230 K232 L260 S280 Y282 H283 G286 L340 D351 I15 K17 G18 V23 A34 K36 L64 S84 Y86 H87 G90 L144 D155 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=3.0nM P36897 30429955 601 GHMTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQE 5qim A 1.75 BS01 J2Y A 1 G214 V219 A230 K232 L260 L278 S280 Y282 H283 G286 L340 G17 V22 A33 K35 L63 L81 S83 Y85 H86 G89 L143 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=6.0nM P36897 30429955 601 GGTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEGI 5qin A 1.57 BS01 J2V A 1 V258 A275 K277 F294 L305 L323 T325 F327 H328 G331 L386 C396 D397 V19 A31 K33 F50 L61 L79 T81 F83 H84 G87 L142 C152 D153 D379 K381 N384 D397 T421 D135 K137 N140 D153 T175 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=40nM P37173 30429955 601 ELLPIELDTLVGKGRFAEVYKAKLKQFETVAVKIFPYEEYASWKTEKDIFSDINLKHENILQFLTAEERKTELGKQYWLITAFHAKGNLQEYLTRHVISWEDLRKLGSSLARGIAHLHSDHTPCGRPKMPIVHRDLKSSNILVKNDLTCCLCDFGLSLRLDPTLSVDDLANQVGTARYMAPEVLASAMNLENVESFKQTDVYSMALVLWEMTSRCNAVGEVKDYEPPFGSKVREHPCVASMADNVLADAGRPEIPSFWLNHQGIQMVCETLTECWDHDPEARLTAQCVAERFSEL 5qj2 A 2.82 BS02 JXS B 1 H95 F99 H95 F99 Q91 D94 H95 D96 Q91 D94 H95 D96 1.11.2.2 0004601,0006979,0020037 remove_due_to_license_issue P05164 30613322 613 CPEQDKYRTITGMCNNRRSPTLGASNRAFVRWLPAEYEDGFSLPYGWTPGVKRNGFPVALARAVSNEIVRFPTDQLTPDQERSLMFMQWGQLLDHDLDFTPEP 5qj2 B 2.82 BS05 JXS B 1 T238 R239 F366 F407 T126 R127 F254 F295 1.11.2.2 0004601,0006979,0020037 remove_due_to_license_issue P05164 30613322 613 VNCETSCVQQPPCFPLKIPPNDPRIKNQADCIPFFRSCPACPGSNITIRNQINALTSFVDASMVYGSEEPLARNLRNMSNQLGLLAVNQRFQDNGRALLPFDNLHDDPCLLTNRSARIPCFLAGDTRSSEMPELTSMHTLLLREHNRLATELKSLNPRWDGERLYQEARKIVGAMVQIITYRDYLPLVLGPTAMRKYLPTYRSYNDSVDPRIANVFTNAFRYGHTLIQPFMFRLDNRYQPMEPNPRVPLSRVFFASWRVVLEGGIDPILRGLMATPAKLNRQNQIAVDEIRERLFEQVMRIGLDLPALNMQRSRDHGLPGYNAWRRFCGLPQPETVGQLGTVLRNLKLARKLMEQYGTPNNIDIWMGGVSEPLKRKGRVGPLLACIIGTQFRKLRDGDRFWWENEGVFSMQQRQALAQISLPRIICDNTGITTVSKNNIFMSNSYPRDFVNCSTLPALNLASWRE 5qj3 B 2.76 BS04 JXP B 1 P220 T238 R239 F366 F407 V410 M411 P107 T125 R126 F253 F294 V297 M298 1.11.2.2 0004601,0006979,0020037 remove_due_to_license_issue P05164 30613322 613 NCETSCVQQPPCFPLKIPPNDPRIKNQADCIPFFRSCPACPGSNITIRNQINALTSFVDASMVYGSEEPLARNLRNMSNQLGLLAVNQRFQDNGRALLPFDNLHDDPCLLTNRSARIPCFLAGDTRSSEMPELTSMHTLLLREHNRLATELKSLNPRWDGERLYQEARKIVGAMVQIITYRDYLPLVLGPTAMRKYLPTYRSYNDSVDPRIANVFTNAFRYGHTLIQPFMFRLDNRYQPMEPNPRVPLSRVFFASWRVVLEGGIDPILRGLMATPAKLNRQNQIAVDEIRERLFEQVMRIGLDLPALNMQRSRDHGLPGYNAWRRFCGLPQPETVGQLGTVLRNLKLARKLMEQYGTPNNIDIWMGGVSEPLKRKGRVGPLLACIIGTQFRKLRDGDRFWWENEGVFSMQQRQALAQISLPRIICDNTGITTVSKNNIFMSNSYPRDFVNCSTLPALNLASWRE 5qqo A 2.0 BS02 NRJ A 1 H40 L41 H57 I151 D189 A190 C191 K192 G193 S195 T213 W215 G226 V227 Y228 H27 L28 H44 I141 D182 A183 C184 K185 G186 S188 T206 W208 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=17nM remove_due_to_license_issue Ki=17nM P03951 31445854 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qqp A 2.08 BS01 NR7 A 1 R39 H40 L41 H57 I151 D189 A190 C191 K192 G193 S195 T213 W215 G226 V227 Y228 R26 H27 L28 H44 I141 D182 A183 C184 K185 G186 S188 T206 W208 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=5.3nM remove_due_to_license_issue Ki=5.3nM P03951 31445854 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qtt A 2.23 BS01 QEY A 1 R39 H40 L41 I151 D189 A190 C191 K192 G193 S195 T213 S214 W215 G216 G226 V227 Y228 R26 H27 L28 I141 D182 A183 C184 K185 G186 S188 T206 S207 W208 G209 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=3.4nM remove_due_to_license_issue P03951 31833761 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5qtu A 2.53 BS02 QEV A 1 R39 H40 L41 I151 D189 A190 C191 K192 G193 S195 T213 W215 G218 G226 V227 Y228 R26 H27 L28 I141 D182 A183 C184 K185 G186 S188 T206 W208 G211 G219 V220 Y221 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 remove_due_to_license_issue P03951 31833761 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5std A 1.95 BS02 UNN A 1 F53 M69 V75 V108 N131 P149 I151 F158 F45 M61 V67 V100 N123 P141 I143 F150 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=32pM remove_due_to_license_issue Ki=32nM P56221 10382670 175 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFGDK 5std B 1.95 BS02 UNN B 1 Y50 F53 M69 V75 V108 N131 P149 I151 Y42 F45 M61 V67 V100 N123 P141 I143 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=32pM remove_due_to_license_issue Ki=32nM P56221 10382670 173 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFGDK 5svk A 2.773 BS02 ATP A 1 V274 S275 N279 R281 K299 V268 S269 N273 R275 K293 ? 0001614,0001666,0004931,0005216,0005524,0005886,0006811,0006812,0007165,0007268,0007274,0009266,0009408,0009409,0009612,0009743,0010524,0014832,0015267,0016020,0030424,0030432,0033198,0034220,0035590,0043005,0043235,0046872,0048167,0048266,0050804,0050850,0050909,0051649,0060079,0070207,0070588,0071318,0098655,0098662,0098685,0098686,0098794 remove_due_to_license_issue EC50=340nM P56373 27626375 401 FFTYETPKVIVVKSWTIGIINRVVQLLIISYFVGWVFLHEKAYQVRDTAIESSVVTKVKGSGLYANRVMDVSDYVTPPQGTSVFVIITKMIVTENQMQGFCPESEEKYRCVSDSQCGPERLPGGGILTGRCVNYSSVLRTCEIQGWCPTEVDTVETPIMMEAENFTIFIKNSIRFPLFNFEKGNLLPNLTARDMKTCRFHPDKDPFCPILRVGDVVKFAGQDFAKLARTGGVLGIKIGWVCDLDKAWDQCIPKYSFTRLDSVSEKSSVSPGYNFRFAKYYKMENGSEYRTLLKAFGIRFDVLVYGNAGKFNIIPTIISSVAAFTSVGVGTVLCDIILLNFLKGADQYKAKKFEEVNE 5svl A 2.9 BS01 ATP A 1 V274 S275 N279 R281 K299 V261 S262 N266 R268 K286 ? 0001614,0001666,0004931,0005216,0005524,0005886,0006811,0006812,0007165,0007268,0007274,0009266,0009408,0009409,0009612,0009743,0010524,0014832,0015267,0016020,0030424,0030432,0033198,0034220,0035590,0043005,0043235,0046872,0048167,0048266,0050804,0050850,0050909,0051649,0060079,0070207,0070588,0071318,0098655,0098662,0098685,0098686,0098794 remove_due_to_license_issue P56373 27626375 401 KSVVVKSWTIGIINRVVQLLIISYFVGWVFLHEKAYQVRDTAIESSVVTKVKGSGLYANRVMDVSDYVTPPQGTSVFVIITKMIVTENQMQGFCPESEEKYRCVSDSQCGPERLPGGGILTGRCVNYSSVLRTCEIQGWCPTEVDTVETPIMMEAENFTIFIKNSIRFPLFNFEKGNLLPNLTARDMKTCRFHPDKDPFCPILRVGDVVKFAGQDFAKLARTGGVLGIKIGWVCDLDKAWDQCIPKYSFTRLDSVSEKSSVSPGYNFRFAKYYKMENGSEYRTLLKAFGIRFDVLVYGNAGKFNIIPTIISSVAAFTSVGVGTVLCDIILLNF 5sxk B 3.55 BS01 71K B 1 N377 N378 N46 N47 ? remove_due_to_license_issue P27986 28129991 701 LQDAEWYWGSREEVNEKLRDTADGTFLVRDTKMHGDYTLTLRKGGNNKLIKIDGKYGFSDPLTFSSVVELINHYRNESLAQYNPKLDVKYPVSQVVKEDNIEAVGKKLHEYNTQFQEKSREYDRLYEEYTRTSQEIQMKRTAIEAFNETIKIFEEQCQTQERYSKEYIEKFKREGNEKEIQRIMHNYDKLKSRISEIIDSRRRLEEDLKKQAAEYREIDKRMNSIKPDLIQLRKTRDQYLMWLTQKGVRQKKLNEWL 5sxn A 2.1 BS01 74U A 1 T18 Y20 V36 Y83 P118 L121 A122 F124 T227 G228 A229 S230 T17 Y19 V35 Y82 P117 L120 A121 F123 T223 G224 A225 S226 D38 S41 N43 W45 Y83 D226 A229 D37 S40 N42 W44 Y82 D222 A225 3.4.23.15 0004190,0006508 ic50=11uM remove_due_to_license_issue IC50=11000nM P00797 27687967 403 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSNSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5sy2 A 2.25 BS01 74V A 1 T18 Q19 Y20 V36 D38 G40 Y83 T85 F124 D226 T227 G228 A229 S230 T17 Q18 Y19 V35 D37 G39 Y82 T84 F123 D221 T222 G223 A224 S225 D38 S41 N43 W45 D226 A229 D37 S40 N42 W44 D221 A224 3.4.23.15 0004190,0006508 ic50=11uM remove_due_to_license_issue P00797 27687967 402 TLGNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5sy3 A 2.3 BS01 74Z A 1 T18 Y20 V36 Y83 F119 F124 V127 T227 G228 A229 S230 T15 Y17 V33 Y80 F116 F121 V124 T220 G221 A222 S223 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 ic50=43uM remove_due_to_license_issue IC50=43000nM P00797 27687967 402 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5sy7 A 4.2 BS01 dna C 0 R91 H94 S95 R99 R102 D127 K128 R3 H6 S7 R11 R14 D39 K40 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P53762 27782878 1 ~ 21 LARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLPSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSSRRSFICRMRCGTNGLGSVKEGEPHFVVVHCTGYLVAIGRLQVTSSPEFISRHNIEGIFTFVDHRCVATVGYQPQELLGKNIVEFCHPEDQQLLRDSFQQVVKLKGQVLSVMFRFRSKTREWLWMRTSSFTFQNPYSDEIEYIICTNTN 5sy7 A 4.2 BS02 dna D 0 H94 E98 R101 H6 E10 R13 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P53762 27782878 1 ~ 21 LARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLPSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQPQSEWFGSTLYDQVHPDDVDKLREQLSTSSRRSFICRMRCGTNGLGSVKEGEPHFVVVHCTGYLVAIGRLQVTSSPEFISRHNIEGIFTFVDHRCVATVGYQPQELLGKNIVEFCHPEDQQLLRDSFQQVVKLKGQVLSVMFRFRSKTREWLWMRTSSFTFQNPYSDEIEYIICTNTN 5sy7 B 4.2 BS01 dna C 0 K62 R70 K4 R12 ? 0006355,0046983 remove_due_to_license_issue Q9QZQ0 27782878 1 ~ 21 RKEKSRDAARSRRGKENFEFYELAKLLPLPAAITSQLDKASIIRLTISYLKMRDFANQGDIEVFEAHLGSHILQSLDGFVFALNQEGKFLYISETVSIYLGLSQVELTGSSVFDYVHPGDHVEMAEQLGMLERSFFIRMKSTLGYKVIHITGRLRMGLVVVAHALPHMFVTRVNMDLNIIYCENRISDYMDLTPVDIVGKRCYHFIHAEDVEGIRHSHLDLLNKGQCVTKYYRWMQKNGGYIWIQSSATIAKNIIWVNYLLSNPEYKDTPMDIAQL 5sy7 B 4.2 BS02 dna D 0 K60 R64 R71 N75 K97 K2 R6 R13 N17 K39 ? 0006355,0046983 remove_due_to_license_issue Q9QZQ0 27782878 1 ~ 21 RKEKSRDAARSRRGKENFEFYELAKLLPLPAAITSQLDKASIIRLTISYLKMRDFANQGDIEVFEAHLGSHILQSLDGFVFALNQEGKFLYISETVSIYLGLSQVELTGSSVFDYVHPGDHVEMAEQLGMLERSFFIRMKSTLGYKVIHITGRLRMGLVVVAHALPHMFVTRVNMDLNIIYCENRISDYMDLTPVDIVGKRCYHFIHAEDVEGIRHSHLDLLNKGQCVTKYYRWMQKNGGYIWIQSSATIAKNIIWVNYLLSNPEYKDTPMDIAQL 5sym A 1.55 BS01 71Q A 1 I75 G77 L78 S79 P80 W145 R149 L176 F181 T185 I68 G70 L71 S72 P73 W138 R142 L169 F174 T178 L30 S119 N161 D174 H208 L23 S112 N154 D167 H201 3.1.2.-,3.1.2.22 0002084,0004620,0004622,0005515,0005634,0005654,0005737,0005739,0005783,0005829,0005886,0006631,0008474,0015908,0016298,0016787,0031965,0042997,0052689,0070062,1905336 Ki=280nM remove_due_to_license_issue Ki=300nM O75608 27748579 301 TPLPAIVPAARKATAAVIFLHGLGDTGHGWAEAFAGIRSSHIKYICPHAPVRPVTLNMNVAMPSWFDIIGLSPDSQEDESGIKQAAENIKALIDQEVKNGIPSNRIILGGFSQGGALSLYTALTTQQKLAGVTALSCWLPLRASFPQGPIGGANRDISILQCHGDCDPLVPLMFGSLTVEKLKTLVNPANVTFKTYEGMMHSSCQQEMMDVKQFIDKLLPPID 5syn A 1.64 BS01 71T A 1 L33 L78 G80 L81 P83 S122 W148 H152 M178 F183 L186 T187 L25 L70 G72 L73 P75 S114 W140 H144 M170 F175 L178 T179 L33 S122 A163 D176 H210 L25 S114 A155 D168 H202 3.1.2.-,3.1.2.22 0002084,0004622,0005515,0005654,0005737,0005795,0005829,0006631,0007411,0008474,0016787,0045296,0046464,0052689,0070062,1905344 Kd=240nM remove_due_to_license_issue Ki=120nM, Kd=240nM, IC50=1.1e+3nM O95372 27748579 301 PLLTDAATVSGAERETAAVIFLHGLGDTGHSWADALSTIRLPHVKYICPHAPRIPVTLNMKMVMPSWFDLMGLSPDAPEDEAGIKKAAENIKALIEHEMKNGIPANRIVLGGFSQGGALSLYTALTCPHPLAGIVALSCWLPLHRAFPQAANGSAKDLAILQCHGELDPMVPVRFGALTAEKLRSVVTPARVQFKTYPGVMHSSCPQEMAAVKEFLEKLLPPV 5sz0 A 1.63 BS02 72D A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.8nM remove_due_to_license_issue Ki=0.8nM P00918 27860128 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz1 A 1.55 BS02 72E A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.2nM remove_due_to_license_issue Ki=1.2nM P00918 27860128 307 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz2 A 1.63 BS02 72G A 1 H4 H10 H15 W16 D19 H1 H7 H12 W13 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2nM remove_due_to_license_issue Ki=2.0nM P00918 27860128 307 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz2 A 1.63 BS03 72G A 2 Q92 H94 H96 H119 L198 T199 T200 Q89 H91 H93 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2nM remove_due_to_license_issue Ki=2.0nM P00918 27860128 308 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz3 A 1.689 BS02 72H A 1 H94 L198 T199 T200 H91 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.5nM remove_due_to_license_issue Ki=2.5nM P00918 27860128 307 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz4 A 1.6 BS02 72D A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=0.8nM P00918 27860128 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz5 A 1.274 BS02 72E A 1 H94 H119 V121 L198 T199 T200 H91 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=1.2nM P00918 27860128 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz6 A 1.15 BS02 72G A 1 H94 H119 L198 T199 T200 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=2.0nM P00918 27860128 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz7 A 1.776 BS02 72H A 1 H94 H119 V135 L198 T199 T200 H91 H116 V131 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=2.5nM P00918 27860128 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5sz9 A 2.85 BS01 74Y A 1 T18 Q19 Y20 V36 Y83 L121 F124 V127 T227 G228 A229 T15 Q16 Y17 V33 Y80 L118 F121 V124 T221 G222 A223 D38 S41 N43 W45 Y83 D226 A229 D35 S38 N40 W42 Y80 D220 A223 3.4.23.15 0004190,0006508 remove_due_to_license_issue IC50=38000nM P00797 27687967 402 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5sze A 1.5 BS01 rna C 0 N14 R17 S39 F40 N12 R15 S37 F38 ? 0003723,0005829,0006355,0043487,0045974 remove_due_to_license_issue O66512 28375142 1 ~ 3 HMPYKLQESFLNTARKKRVKVSVYLVNGVRLQGRIRSFDLFTILLEDGKQQTLVYKHAITTIVPHERLEIE 5szx A 2.251 BS01 dna C 0 R179 N182 R183 S186 R187 R190 K194 R5 N8 R9 S12 R13 R16 K20 ? 0003700,0006355 remove_due_to_license_issue P03206 28158710 1 ~ 18 LEIKRYKNRVASRKSRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPD 5szx A 2.251 BS02 dna D 0 A185 S186 K188 S189 K192 A11 S12 K14 S15 K18 ? 0003700,0006355 remove_due_to_license_issue P03206 28158710 102 ~ 119 LEIKRYKNRVASRKSRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPD 5szx B 2.251 BS01 dna C 0 S186 S189 S12 S15 ? 0003700,0006355 remove_due_to_license_issue P03206 28158710 1 ~ 18 LEIKRYKNRVASRKSRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPD 5szx B 2.251 BS02 dna D 0 R179 N182 R183 R187 R190 K194 R5 N8 R9 R13 R16 K20 ? 0003700,0006355 remove_due_to_license_issue P03206 28158710 102 ~ 119 LEIKRYKNRVASRKSRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPD 5t01 A 1.89 BS01 dna C 0 R259 R263 R270 R8 R12 R19 ? 0003677,0003700,0006355 remove_due_to_license_issue P05412 28158710 1 ~ 18 HMKAERKRMRNRIAASKSRKRKLERIARLEEKVKTLKAQNSELASTANMLREQVAQLKQKVM 5t01 A 1.89 BS02 dna D 0 H252 M253 H1 M2 ? 0003677,0003700,0006355 remove_due_to_license_issue P05412 28158710 23 ~ 41 HMKAERKRMRNRIAASKSRKRKLERIARLEEKVKTLKAQNSELASTANMLREQVAQLKQKVM 5t01 B 1.89 BS01 dna C 0 H252 R261 A265 S269 R272 K273 H1 R10 A14 S18 R21 K22 ? 0003677,0003700,0006355 remove_due_to_license_issue P05412 28158710 1 ~ 18 HMKAERKRMRNRIAASKSRKRKLERIARLEEKVKTLKAQNSELASTANMLREQVAQLKQKVM 5t01 B 1.89 BS02 dna D 0 R259 N262 R263 R270 R8 N11 R12 R19 ? 0003677,0003700,0006355 remove_due_to_license_issue P05412 28158710 23 ~ 41 HMKAERKRMRNRIAASKSRKRKLERIARLEEKVKTLKAQNSELASTANMLREQVAQLKQKVM 5t18 A 1.5 BS01 73T A 1 T410 V416 A428 K430 Y476 M477 A478 G480 C481 N484 R525 L528 T17 V23 A35 K37 Y83 M84 A85 G87 C88 N91 R128 L131 D521 A523 R525 N526 D539 F559 D124 A126 R128 N129 D142 F162 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.5nM remove_due_to_license_issue IC50=0.410nM Q06187 27583770 701 HMEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 5t19 A 2.1001 BS01 73U A 1 Y46 V49 F182 C215 S216 A217 I219 G220 R221 Q262 Y48 V51 F184 C217 S218 A219 I221 G222 R223 Q264 D181 C215 R221 S222 Q262 D183 C217 R223 S224 Q264 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P18031 28345882 402 GHMEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED 5t1a A 2.806 BS02 VT5 A 1 L81 A241 V244 Y305 G309 E310 K311 F312 L45 A366 V369 Y430 G434 E435 K436 F437 E1011 D1020 E207 D216 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P41597 27926736 1202 VKQIGAQLLPPLYSLVFIFGFVGNMLVVLILINCKKLKCLTDIYLLNLAISDLLFLITLPLWAHSAANEWVFGNAMCKLFTGLYHIGYFGGIFFIILLTIDRYLAIVHAVFALKARTVTFGVVTSVITWLVAVFASVPGIIFTKCQKEDSVYVCGPYFPRGWNNFHTIMRNILGLVLPLLIMVICYSGISRASKSRINIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYPPPSREKKAVRVIFTIMIVYFLFWTPYNIVILLNTFQEFFGLSNCESTSQLDQATQVTETLGMTHCCINPIIYAFVGEKFRRYLSVFF 5t1j A 2.947 BS01 dna E 0 R198 N246 S262 T303 P319 G323 R63 N111 S127 T168 P184 G188 ? 0000978,0003700,0005634,0006355,0045893 remove_due_to_license_issue Q9JKD8 27791029 501 ~ 524 KLRVALSNHLLWSKFNQHQTEMIITKQGRRMFPFLSFTVAGLEPTSHYRMFVDVVLVDQHHWRYQSGKWVQCGKAEGSMPGNRLYVHPDSPNTGAHWMRQEVSFGKLKLTNNKGASNNVTQMIVLQSLHKYQPRLHIVEVNDGEPEAACSASNTHVFTFQETQFIAVTAYQNAEITQLKIDNNPFAKGFREN 5t1j A 2.947 BS02 dna F 0 R164 R165 K243 Y305 T311 F320 R29 R30 K108 Y170 T176 F185 ? 0000978,0003700,0005634,0006355,0045893 remove_due_to_license_issue Q9JKD8 27791029 501 ~ 524 KLRVALSNHLLWSKFNQHQTEMIITKQGRRMFPFLSFTVAGLEPTSHYRMFVDVVLVDQHHWRYQSGKWVQCGKAEGSMPGNRLYVHPDSPNTGAHWMRQEVSFGKLKLTNNKGASNNVTQMIVLQSLHKYQPRLHIVEVNDGEPEAACSASNTHVFTFQETQFIAVTAYQNAEITQLKIDNNPFAKGFREN 5t1j B 2.947 BS01 dna C 0 R198 N246 S262 T303 P319 G323 F324 E326 R63 N111 S127 T168 P184 G188 F189 E191 ? 0000978,0003700,0005634,0006355,0045893 remove_due_to_license_issue Q9JKD8 27791029 501 ~ 524 KLRVALSNHLLWSKFNQHQTEMIITKQGRRMFPFLSFTVAGLEPTSHYRMFVDVVLVDQHHWRYQSGKWVQCGKAEGSMPGNRLYVHPDSPNTGAHWMRQEVSFGKLKLTNNKGASNNVTQMIVLQSLHKYQPRLHIVEVNDGEPEAACSASNTHVFTFQETQFIAVTAYQNAEITQLKIDNNPFAKGFREN 5t1j B 2.947 BS02 dna D 0 R164 R165 Y305 T311 K314 N318 F320 R29 R30 Y170 T176 K179 N183 F185 ? 0000978,0003700,0005634,0006355,0045893 remove_due_to_license_issue Q9JKD8 27791029 501 ~ 524 KLRVALSNHLLWSKFNQHQTEMIITKQGRRMFPFLSFTVAGLEPTSHYRMFVDVVLVDQHHWRYQSGKWVQCGKAEGSMPGNRLYVHPDSPNTGAHWMRQEVSFGKLKLTNNKGASNNVTQMIVLQSLHKYQPRLHIVEVNDGEPEAACSASNTHVFTFQETQFIAVTAYQNAEITQLKIDNNPFAKGFREN 5t1s A 2.3 BS01 76Q A 1 M192 A211 K213 V246 Y262 Y264 M265 P266 N267 G268 D272 L318 S328 D329 M25 A44 K46 V73 Y89 Y91 M92 P93 N94 G95 D99 L145 S155 D156 D311 K313 A315 N316 D329 T351 D138 K140 A142 N143 D156 T175 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=84nM remove_due_to_license_issue Q9NWZ3 28501511 9901 TRFHSFSFYELKNVTNNFDERPIKMGEGGFGVVYKGYVNNTTVAVKKLTTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5t1t A 2.34 BS01 76P A 1 M192 A211 K213 Y262 M265 D272 L318 M30 A49 K51 Y95 M98 D105 L151 D311 K313 A315 N316 D329 T351 D144 K146 A148 N149 D162 T178 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=58nM remove_due_to_license_issue IC50=58nM Q9NWZ3 28501511 9901 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARATVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5t1u A 1.78 BS01 P6U A 1 G13 D32 Y71 F108 W115 D228 G230 T231 T232 G17 D36 Y75 F112 W119 D223 G225 T226 T227 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=0.069uM remove_due_to_license_issue IC50=69nM P56817 27997172 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5t1w A 2.96 BS01 74B A 1 G11 Q12 G13 L30 D32 Y71 F108 W115 D228 G230 G15 Q16 G17 L34 D36 Y75 F112 W119 D221 G223 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=77nM P56817 27997172 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5t23 A 2.78 BS01 74F A 1 M804 W812 I879 E880 I881 V882 A885 T887 K890 M953 I963 M550 W558 I625 E626 I627 V628 A631 T633 K636 M690 I700 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue IC50=1585nM P48736 28017532 1201 ESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRTTSQTIKVSPDDTPGAILQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKVSLWDCDRKFRVKIRGIDIPVTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCQLLYYVNLLLIDHRFLLRRGEYVLHMWQISFNADKLTSATNPDKENSMSISILLDNYCHPIALPKRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSASSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHERVPFVLTPDFLFVMGTSGTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWF 5t27 A 2.6 BS01 74F A 1 M752 W760 I777 V828 M900 I910 M561 W569 I586 V637 M704 I714 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNARMKLVVQAGLFHGNEMLCKTVSSSEVNVEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELGRTEEELREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKTAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLATEEEALKHFRVKFNEALRESW 5t28 A 2.8 BS01 74Q A 1 M752 W760 I777 I825 V828 M900 I910 M556 W564 I581 I629 V632 M704 I714 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2b A 2.3 BS01 74O A 1 W760 I777 V828 S831 M900 I910 W562 I579 V630 S633 M702 I712 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=5nM remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2d A 2.9 BS01 74L A 1 W760 I777 I825 V828 S831 M900 I910 W562 I579 I627 V630 S633 M702 I712 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2g A 2.55 BS01 74K A 1 M752 W760 I777 I825 E826 V828 S831 M900 I910 D911 M554 W562 I579 I627 E628 V630 S633 M702 I712 D713 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2i A 2.3 BS01 74J A 1 W760 I777 I825 V827 V828 M900 I910 W562 I579 I627 V629 V630 M702 I712 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=2nM remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2l A 2.55 BS01 74H A 1 M752 W760 I777 Y813 I825 V828 N836 M900 I910 D911 M564 W572 I589 Y625 I637 V640 N648 M712 I722 D723 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELGRHEEQLQLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2m A 2.8 BS01 74N A 1 T750 W760 I777 K779 I825 V828 S831 M900 I910 T552 W562 I579 K581 I627 V630 S633 M702 I712 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 28017532 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 5t2p A 1.693 BS01 K89 A 1 P25 L30 T33 W102 I105 S106 F110 Y118 L140 P25 L30 T33 W102 I105 S106 F110 Y118 L140 ? 0005198 ic50=1.9uM remove_due_to_license_issue L7R9I1 28205569 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHCSPHHTALRQAILCWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISCLTFGRETVLEYLVSFGVWIRTPPAARPPNAPILSVENLYFQ 5t2p A 1.693 BS02 K89 F 1 V124 W125 T128 P134 V124 W125 T128 P134 ? 0005198 ic50=1.9uM remove_due_to_license_issue L7R9I1 28205569 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHCSPHHTALRQAILCWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISCLTFGRETVLEYLVSFGVWIRTPPAARPPNAPILSVENLYFQ 5t2t A 1.967 BS02 0N8 A 1 K43 R47 L84 I86 D88 K114 K44 R48 L85 I87 D89 K115 2.7.7.48,3.1.-.- remove_due_to_license_issue P14240 29765612 203 HDEIISELRELCLNYIEQDERLSRQKLNFLGQREPRMVLIEGLKLLSRCIEIDSADKSGCTHNHDDKSVETILVESGIVCPGLPLIIPDGYKLIDNSLILLECFVRSTPASFEKKFIEDTNKLACIREDLAVAGVTLVPIVDGRCDYDNSFMPEWANFKFRDLLFKLLEYSNQDEKVFEESEYFRLCES 5t2y A 1.94 BS01 753 A 1 S136 F152 G154 I155 G173 V188 S133 F149 G151 I152 G170 V185 2.3.1.203 0006486,0016746,0016747,0018279 ic50=2.2uM remove_due_to_license_issue IC50=2200nM Q0P9D1 28182413 201 ARTEKIYIYGASGHGLVCEDVAKNMGYKECIFLDDFMKFESTLPKYDFFIAIGNNEIRKKIYQKISENGFKIVNLIHKSALISPSAIVEENAGILIMPYVVINAKAKIEKGVILNTSSVIEHECVIGEFSHVSVGAKCAGNVKIGKNCFLGINSCVLPNLSLADDSILGGGATLVKNQDEKGVFVGVPAKRM 5t2y B 1.94 BS01 753 B 1 S136 F152 G154 I155 G173 V188 S133 F149 G151 I152 G170 V185 2.3.1.203 0006486,0016746,0016747,0018279 ic50=2.2uM remove_due_to_license_issue IC50=2200nM Q0P9D1 28182413 201 ARTEKIYIYGASGHGLVCEDVAKNMGYKECIFLDDFMKFESTLPKYDFFIAIGNNEIRKKIYQKISENGFKIVNLIHKSALISPSAIVEENAGILIMPYVVINAKAKIEKGVILNTSSVIEHECVIGEFSHVSVGAKCAGNVKIGKNCFLGINSCVLPNLSLADDSILGGGATLVKNQDEKGVFVGVPAKRM 5t35 A 2.7 BS01 759 D 1 W374 A384 L385 L387 N433 H437 E438 V439 W26 A36 L37 L39 N85 H89 E90 V91 ? remove_due_to_license_issue O60885 28288108 301 KVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMPD 5t35 D 2.7 BS01 759 D 1 W88 Y98 P99 R107 I109 H110 S111 Y112 H115 W117 W28 Y38 P39 R47 I49 H50 S51 Y52 H55 W57 ? remove_due_to_license_issue P40337 28288108 301 PVLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQERIAHQ 5t36 A 1.4 BS01 755 A 1 P124 S127 T131 P119 S122 T126 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=0.043uM remove_due_to_license_issue IC50=8910nM O14684 28190634 201 LVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5t37 A 1.761 BS01 758 A 1 P124 S127 P120 S123 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=0.241uM remove_due_to_license_issue IC50=0.744000nM O14684 28190634 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5t3n A 2.4 BS01 75G A 1 I366 Y369 F375 G376 E377 L378 A379 R386 A387 I390 Y424 L428 I438 I80 Y83 F89 G90 E91 L92 A93 R100 A101 I104 Y138 L142 I152 2.7.11.11 Kd=9.1nM remove_due_to_license_issue Q7KQK0 27738107 503 HHEVLFQGPGAKKRKMYEDILSHVNILKDMDPYERCKVADCLKSKSYNDGEIIIKEGEEGDTFFILIDGNAVASKDNKVIKTYTKGDYFGELALLKNKPRAATIKAQNFCQVVYLDRKSFKRLLGPIEDILHRNVENYKKVLNELGLDTTCID 5t4b A 1.76 BS01 75N A 1 E205 E206 Y547 W629 S630 Y631 Y662 Y666 H740 E167 E168 Y509 W591 S592 Y593 Y624 Y628 H702 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=0.42nM remove_due_to_license_issue P27487 27670099 810 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5t4e A 1.77 BS01 75L A 1 E205 E206 Y547 W629 S630 Y631 Y662 Y666 E167 E168 Y509 W591 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=4376nM remove_due_to_license_issue IC50=4376nM P27487 27670099 810 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5t4f A 1.9 BS01 75M A 1 E205 E206 Y547 W629 S630 Y631 Y662 Y666 E167 E168 Y509 W591 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 ic50=10nM remove_due_to_license_issue P27487 27670099 812 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5t4h A 2.61 BS01 75J A 1 E205 E206 Y547 K554 W629 S630 Y631 Y662 Y666 E167 E168 Y509 K516 W591 S592 Y593 Y624 Y628 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 27670099 810 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 5t4u A 1.5 BS01 12Q A 1 V657 P658 N708 F714 V30 P31 N81 F87 ? ic50=4800nM remove_due_to_license_issue IC50=4800nM P55201 28068087 802 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5t4v A 1.65 BS01 N48 A 1 V657 P658 E661 N708 F714 V30 P31 E34 N81 F87 ? ic50=60nM remove_due_to_license_issue IC50=60nM P55201 28068087 801 MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKM 5t54 A 1.65 BS01 FUC C 1 V123 N124 T125 E126 V123 N124 T125 E126 ? 0005576,0030246,0046872 remove_due_to_license_issue P86993 27973758 2 SELSFNYPNFQSVEDITFQGGASPRNETLQLTPTDSNGIPIRQRAGHAVYSQPFQLRDTSFYTTFTFVIRTTSNSPADGFAIFIAPPDFPVKRYGGYLGLFEPNTATNTSANKVVAVEFDTWVNTEWKEPRYRHIGIDVNSIVSVRVTRWQDKDVFSRSIATAHVGYDGISKILTAFVTYPDGGNYVLSHVVDLAEIFPGDVRIGFSGATGQYETQYIHSWSFSSTSTN 5t5c A 1.851 BS01 dna C 0 R109 R138 G139 A140 G145 K148 F168 N171 S172 N176 R314 R49 R78 G79 A80 G85 K88 F108 N111 S112 N116 R254 C112 A140 N162 N171 E179 C52 A80 N102 N111 E119 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 28466855 1 ~ 8 VLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKA 5t5c A 1.851 BS02 dna D 0 S172 L311 R320 S112 L251 R260 C112 A140 N162 N171 E179 C52 A80 N102 N111 E119 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 28466855 3 ~ 10 VLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKA 5t5c B 1.851 BS01 dna E 0 R109 S137 R138 G145 K148 F168 N171 S172 N176 R49 S77 R78 G85 K88 F108 N111 S112 N116 C112 A140 N162 N171 E179 C52 A80 N102 N111 E119 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 28466855 1 ~ 8 VLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKA 5t5c B 1.851 BS02 dna F 0 K113 S172 K315 R320 R324 K53 S112 K255 R260 R264 C112 A140 N162 N171 E179 C52 A80 N102 N111 E119 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 28466855 3 ~ 10 VLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKA 5t5g A 2.1 BS01 75P A 1 Y286 C311 Y312 M313 R336 L337 N339 T348 Y375 Y377 Y52 C77 Y78 M79 R102 L103 N105 T114 Y141 Y143 2.1.1.-,2.1.1.361 0042799 remove_due_to_license_issue Q9NQR1 27804297 407 SKAELQSEERKRIDELIESGKEEGMKIDLIDGKGRGVIATKQFSRGDFVVEYHGDLIEITDAKKREALYAQDPSTGCYMYYFQYLSKTYCVDATRETNRLGRLINHSKSGNCQTKLHDIDGVPHLILIASRDIAAGEELLYDY 5t66 A 1.951 BS01 C6S A 1 S73 N107 Y108 S133 N135 N173 T238 G239 S240 S43 N77 Y78 S103 N105 N143 T208 G209 S210 S73 K76 S133 E169 K237 S240 S43 K46 S103 E139 K207 S210 3.5.2.6 0008800,0016020,0016787,0017001,0030655,0046677 remove_due_to_license_issue G3G192 28115348 300 ADVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTDGL 5t68 A 2.93 BS01 77V A 1 L377 A400 M450 A451 L453 G454 L501 L15 A38 M83 A84 L86 G87 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=23nM, EC50=34nM P43405 27789138 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEG 5t68 B 2.93 BS01 77V B 1 L377 A400 V433 M448 M450 A451 L453 G454 L501 L15 A38 V66 M81 M83 A84 L86 G87 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=23nM, EC50=34nM P43405 27789138 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 5t6f A 1.9 BS01 N38 A 1 E54 I109 Q110 R112 T134 I135 P136 C139 H157 A158 A159 A160 T161 V168 E55 I110 Q111 R113 T126 I127 P128 C131 H149 A150 A151 A152 T153 V160 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 27914364 201 HAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 5t6g A 2.45 BS01 N40 A 1 H30 E54 I109 Q110 R112 V114 T134 C139 H157 A158 A159 A160 H32 E56 I111 Q112 R114 V116 T136 C141 H159 A160 A161 A162 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 27914364 201 HHAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGMDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQ 5t8d A 2.15 BS01 dna B 0 R42 I68 N71 N72 G73 I80 T82 R83 F84 W140 G177 E178 G179 H180 E184 K187 E201 A203 Q204 H205 R232 W234 R236 K262 K294 N298 K299 R33 I59 N62 N63 G64 I71 T73 R74 F75 W131 G168 E169 G170 H171 E175 K178 E192 A194 Q195 H196 R223 W225 R227 K253 K285 N289 K290 0004519 remove_due_to_license_issue 28873986 1 ~ 26 ASSINPWILTGFADAEGSFGLYIINRNIRYTTRLKFTITLHNKDKSILENIQSTWKVGIIANNGDNAVSLIVTRFEDLKVIIDHFEKYPLITQKLGDYKLFKQAFSVMENKEHLKENGIKELVRIKAKMNWGLTDELKKAFPGNISRERPLINKNIPNFKWLAGFTSGEGHFGVELIKNSRNSRVHVRLRFEIAQHVRDKNLMNSLITYLGCGYIYEQNYSERSWLRFSVSKFSDINDKIIPVFQENTLIGVKLEDFEDWCKVAKLIEEKKHLTESGLDEIKKIKLNMNKGR 5t8d A 2.15 BS02 dna C 0 A21 E22 G23 S24 Y28 T48 L49 H50 K103 N139 W140 T143 R190 H195 R197 R199 Y223 Y225 Q227 Y229 W234 R236 K241 F242 H281 A15 E16 G17 S18 Y22 T39 L40 H41 K94 N130 W131 T134 R181 H186 R188 R190 Y214 Y216 Q218 Y220 W225 R227 K232 F233 H272 0004519 remove_due_to_license_issue 28873986 1 ~ 26 ASSINPWILTGFADAEGSFGLYIINRNIRYTTRLKFTITLHNKDKSILENIQSTWKVGIIANNGDNAVSLIVTRFEDLKVIIDHFEKYPLITQKLGDYKLFKQAFSVMENKEHLKENGIKELVRIKAKMNWGLTDELKKAFPGNISRERPLINKNIPNFKWLAGFTSGEGHFGVELIKNSRNSRVHVRLRFEIAQHVRDKNLMNSLITYLGCGYIYEQNYSERSWLRFSVSKFSDINDKIIPVFQENTLIGVKLEDFEDWCKVAKLIEEKKHLTESGLDEIKKIKLNMNKGR 5t8e A 2.71 BS01 77U A 1 L704 N705 L707 Q711 M745 F764 L873 T877 L34 N35 L37 Q41 M75 F94 L203 T207 ? remove_due_to_license_issue IC50=0.720000nM, EC50=0.190000nM P10275 28363748 1003 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 5t8j A 2.7 BS01 77T A 1 L704 L707 G708 Q711 M742 F764 M780 L873 T877 L34 L37 G38 Q41 M72 F94 M110 L203 T207 ? remove_due_to_license_issue IC50=1.000000nM, EC50=0.290000nM P10275 28363748 1002 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 5t8o A 2.41 BS01 76Z A 1 V416 A429 E442 M471 E472 L474 L524 C535 D536 F537 V69 A82 E95 M124 E125 L127 L177 C188 D189 F190 D517 K519 N522 D536 L553 T561 D170 K172 N175 D189 L202 T210 2.7.11.25 0004672,0004674,0005524,0006468 Ki=0.31uM remove_due_to_license_issue Q9WUL6 28005357 705 PVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQGKSLLTGDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 5t8p A 2.32 BS01 774 A 1 V416 A429 M471 L473 D521 L524 C535 D536 V70 A83 M125 L127 D175 L178 C189 D190 D517 K519 N522 D536 L553 T561 D171 K173 N176 D190 L205 T213 2.7.11.25 0004672,0004674,0005524,0006468 Ki=1.28uM remove_due_to_license_issue Q9WUL6 28005357 701 VPVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQPDGLSLLTGDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 5t8q A 2.63 BS01 76Y A 1 R410 V416 R418 L473 L474 L524 R63 V69 R71 L126 L127 L177 D517 K519 N522 D536 L553 T561 D170 K172 N175 D189 L201 T209 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 28005357 706 PVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQPSLLTGDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 5t92 A 2.22 BS01 77W A 1 T347 A350 E353 L384 L387 M388 M421 I424 H524 T30 A33 E36 L67 L70 M71 M95 I98 H182 ? ic50=16nM remove_due_to_license_issue P03372 28296398 601 LTADQMVSALLDAEPPILYSSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHL 5t97 A 3.0 BS01 782 A 1 T347 A350 D351 E353 M388 F404 M421 I424 H524 T24 A27 D28 E30 M65 F81 M89 I92 H176 ? remove_due_to_license_issue IC50=34nM P03372 28296398 601 LTADQMVSALLDAEPPILYMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHL 5t9u A 2.301 BS01 7HG A 1 R55 M61 Q63 A101 N102 Q111 F113 H126 R54 M60 Q62 A100 N101 Q110 F112 H125 R55 F60 Q63 N102 F113 L122 H126 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Kd=25nM remove_due_to_license_issue Kd=25nM, Ki=16nM P62937 28075591 300 VNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQL 5t9w A 2.0 BS01 78E A 1 R55 I57 F60 Q63 A101 N102 A103 Q111 F113 K125 H126 R54 I56 F59 Q62 A100 N101 A102 Q110 F112 K124 H125 R55 F60 Q63 N102 F113 L122 H126 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Kd=2600nM remove_due_to_license_issue Kd=2600nM, Ki=795nM P62937 28075591 300 VNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 5t9z A 1.4 BS01 78R A 1 R55 F60 M61 Q63 A101 N102 Q111 F113 R54 F59 M60 Q62 A100 N101 Q110 F112 R55 F60 Q63 N102 F113 L122 H126 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Kd=64nM remove_due_to_license_issue Kd=64nM, Ki=14nM P62937 28075591 300 VNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQL 5ta2 A 1.48 BS01 78X A 1 R55 I57 M61 Q63 A101 N102 Q111 F113 H126 R54 I56 M60 Q62 A100 N101 Q110 F112 H125 R55 F60 Q63 N102 F113 L122 H126 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Kd=11nM remove_due_to_license_issue Kd=11nM, Ki=4.0nM P62937 28075591 300 VNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQL 5ta4 A 1.5 BS01 838 A 1 R55 I57 M61 Q63 A101 N102 Q111 F113 R54 I56 M60 Q62 A100 N101 Q110 F112 R55 F60 Q63 N102 F113 L122 H126 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 Kd=24nM remove_due_to_license_issue Kd=24nM, Ki=7.0nM P62937 28075591 201 VNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 5ta6 A 2.5 BS01 79D A 1 L59 K61 C67 V114 L130 L132 C133 R134 R136 F183 D194 L23 K25 C31 V78 L94 L96 C97 R98 R100 F147 D158 D176 K178 G180 N181 D194 T214 D140 K142 G144 N145 D158 T178 2.7.11.21 0004672,0005524,0006468 ic50=1.5nM remove_due_to_license_issue IC50=1.5nM P53350 28169164 1000 AKEIPEVLVDPRSRRRYVRGRFLGKGGFAKCFEISDADTKEVFAGKIVPKSLLLKPHQREKMSMEISIHRSLAHQHVVGFHGFFEDNDFVFVVLELCRRRSLLELHKRRKALTEPEARYYLRQIVLGCQYLHRNRVIHRDLKLGNLFLNEDLEVKIGDFGLATKVEYDGERKKVLCGTPNYIAPEVLSKKGHSFEVDVWSIGCIMYTLLVGKPPFETSCLKETYLRIKKNEYSIPKHINPVAASLIQKMLQTDPTARPTINELLNDEFFTSGYIPARLPITCLTIPPRFSIAPS 5tb6 A 1.79 BS01 77X A 1 P1110 F1111 V1115 L1120 N1168 V1174 P32 F33 V37 L42 N90 V96 2.3.1.-,2.3.1.48 Kd=1.53uM remove_due_to_license_issue Kd=3650nM Q92793 27994766 1201 SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5tbe A 2.44 BS01 78L A 1 V30 A51 K53 E71 L75 I84 T106 L108 M109 G110 A111 L167 D168 F169 V26 A45 K47 E65 L69 I78 T100 L102 M103 G104 A105 L161 D162 F163 D150 K152 N155 D168 D144 K146 N149 D162 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=4.4nM remove_due_to_license_issue Kd=2.7nM, IC50=1.000000nM Q16539 28397331 401 RPTFYRQELNKTIWEVPERYQNLSPVGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKIESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 5tbj A 2.32 BS01 LHD A 1 Y150 Y154 Q159 M163 G193 E215 A216 E258 M260 M269 W416 Y15 Y19 Q24 M28 G58 E80 A81 E123 M125 M134 W281 D166 E258 E267 H415 D31 E123 E132 H280 2.1.1.319 0016274,0018216 remove_due_to_license_issue Q9WVG6 29685976 501 SVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 5tbm A 1.85 BS01 79A A 1 F244 H248 M252 A277 Y281 H293 L296 V302 Y307 M309 T321 I337 C339 N341 F6 H10 M14 A39 Y43 H55 L58 V64 Y69 M71 T83 I95 C97 N99 ? Kd=0.049uM remove_due_to_license_issue EC50=27nM, IC50=12nM Q99814 27635045 401 LDSKTFLSEHSMDMKFTYCDDRITELIGYHPEELLGRSAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGGYVWLETQGTVIYNPPQCIMCVNYVLSEIE 5tbp A 2.6 BS01 7A4 A 1 A272 Q275 L276 L301 R302 W305 A10 Q13 L14 L39 R40 W43 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue Kd=2380nM, IC50=2400nM P19793 28714476 501 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp A 2.6 BS02 7A4 A 2 A271 A272 Q275 R316 L326 A327 A9 A10 Q13 R54 L64 A65 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue Kd=2380nM, IC50=2400nM P19793 28714476 502 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp A 2.6 BS03 7A4 A 3 F439 I447 F177 I185 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue Kd=2380nM, IC50=2400nM P19793 28714476 503 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp C 2.6 BS01 7A4 A 3 D273 R302 W305 D28 R57 W60 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue Kd=2380nM, IC50=2400nM P19793 28714476 503 EDMPVERILEAELAVPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 5tc0 A 2.24 BS01 79Y A 1 A617 K619 L671 P672 F673 M674 G677 N728 M730 A740 D741 A40 K42 L74 P75 F76 M77 G80 N131 M133 A143 D144 D723 A725 R727 N728 D741 M762 D126 A128 R130 N131 D144 M146 2.7.10.1 0004672,0004713,0005524,0006468 ic50=25nM remove_due_to_license_issue Q12866 28082036 1100 EDVVIDRNLLILGKILGEGEFGSVMEGNLKQEDGTSLKVAVKTMKDFSHPNVMRLLGVCIEMSSQGIPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFMPVKWIAIETSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESL 5tca A 3.15 BS01 J55 A 1 L40 C41 R152 C194 K195 G196 S198 T213 S214 S216 R217 L25 C26 R137 C179 K180 G181 S183 T198 S199 S201 R202 H56 D104 K195 G196 D197 S198 G199 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 remove_due_to_license_issue Kd=19nM, IC50=19nM P00746 27994744 500 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 5tcc A 3.37 BS01 J56 A 1 L40 C41 H56 C57 R152 K195 G196 S198 S214 G215 S216 R217 L25 C26 H41 C42 R137 K180 G181 S183 S199 G200 S201 R202 H56 D104 K195 G196 D197 S198 G199 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 remove_due_to_license_issue IC50=77nM, Kd=2210nM P00746 27994744 500 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 5tci A 2.45 BS01 79V B 1 D64 G66 D136 D57 G59 D129 E57 D68 Y181 E50 D61 Y174 4.2.1.20 0000162,0004834,0005829,0005886,0006568,0016829 remove_due_to_license_issue P9WFY1 28671682 501 EASRLGPVFDSCRANNRAALIGYLPTGYPDVPASVAAMTALVESGCDIIEVGVPYSDPGMDGPTIARATEAALRGGVRVRDTLAAVEAISIAGGRAVVMTYWNPVLRYGVDAFARDLAAAGGLGLITPDLIPDEAQQWLAASEEHRLDRIFLVAPSSTPERLAATVEASRGFVYAASSQAAPELVGRVKAVSDIPVGVGLGVRSRAQAAQIAQYADGVIVGSALVTALTEGLPRLRALTGELAAGVRLG 5tci B 2.45 BS01 79V B 1 P31 Y200 F202 P208 F211 H294 G295 P27 Y196 F198 P204 F207 H290 G291 K101 E123 S390 K97 E119 S386 4.2.1.20 0000162,0004834,0005737,0006568,0016829 Kd=132nM remove_due_to_license_issue P9WFX9 28671682 501 IAEPTSHDPDSGGHFGGPSGWGGRYVPEALMAVIEEVTAAYQKERVSQDFLDDLDRLQANYAGRPSPLYEATRLSQHAGSARIFLKREDLNHTGSHKINNVLGQALLARRMGKTRVIAETGAGQHGVATATACALLGLDCVIYMGGIDTARQALNVARMRLLGAEVVAVQTGSKTLKDAINEAFRDWVANADNTYYCFGTAAGPHPFPTMVRDFQRIIGMEARVQIQGQAGRLPDAVVACVGGGSNAIGIFHAFLDDPGVRLVGFEAAGDGVETGRHAATFTAGSPGAFHGSFSYLLQDEDGQTIESHSISAGLDYPGVGPEHAWLKEAGRVDYRPITDSEAMDAFGLLCRMEGIIPAIESAHAVAGALKLGVELGRGAVIVVNLSGRGDKDVETAAKWFGLLGN 5tcj B 2.4 BS02 79V B 1 F188 Y200 F202 P208 H294 F180 Y192 F194 P200 H286 K101 E123 S390 K93 E115 S382 4.2.1.20 0000162,0004834,0005737,0006568,0016829 remove_due_to_license_issue P9WFX9 28671682 505 TSHDPDSGGHFGGPSGWGGRYVPEALMAVIEEVTAAYQKERVSQDFLDDLDRLQANYAGRPSPLYEATRLSQHAGSARIFLKREDLNHTGSHKINNVLGQALLARRMGKTRVIAETGAGQHGVATATACALLGLDCVIYMGGIDTARQALNVARMRLLGAEVVAVQTGSKTLKDAINEAFRDWVANADNTYYCFGTAAGPHPFPTMVRDFQRIIGMEARVQIQGQAGRLPDAVVACVGGGSNAIGIFHAFLDDPGVRLVGFEAAGDGVETGRHAATFTAGSPGAFHGSFSYLLQDEDGQTIESHSISAGLDYPGVGPEHAWLKEAGRVDYRPITDSEAMDAFGLLCRMEGIIPAIESAHAVAGALKLGVELGRGAVIVVNLSGRGDKDVETAAKWFGLL 5tco A 2.1 BS01 79Q A 1 K53 E71 T106 L108 M109 G110 A111 L167 D168 F169 K44 E62 T97 L99 M100 G101 A102 L158 D159 F160 D150 K152 N155 D168 T185 D141 K143 N146 D159 T163 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 Kd=3.14nM remove_due_to_license_issue IC50=38nM, Kd=3.9nM Q16539 28397331 401 PTFYRQELNKTIWEVPERYQNLSPVGSSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 5tcy A 1.9 BS01 5LC A 1 V97 Q98 R118 K121 R205 R249 Y288 V76 Q77 R97 K100 R184 R228 Y267 ? 0006826,0030288,0030313,0046872,1901678 Kd=22nM remove_due_to_license_issue Q0P8Q4 28383577 402 AMLPISMSDEGDSFLVKDSLGENKIPKNPSKVVILDLGILDTFDALKLNDKVVGVPAKNLPKYLQQFKNKPSVGGVQQVDFEAINALKPDLIIISGRQSKFYDKLKEIAPTLFVGLDNANFLSSFENNVLSVAKLYGLEKEALEKISDIKNEIEKAKSIVDEDKKALIILTNSNKISAFGPQSRFGIIHDVLGINAVDENIKVGTLGKSINSEFILEKNPDYIFVVDRNVILGNKERAQGILDNALVAKTKAAQNKKIIYLDPEYWYLASGNGLESLKTMILEIKNAVK 5td2 A 2.68 BS01 7AE A 1 E595 G596 A617 K619 M650 L671 F673 M674 K675 N728 M730 E19 G20 A41 K43 M58 L74 F76 M77 K78 N131 M133 D723 A725 R727 N728 D741 D126 A128 R130 N131 D144 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q12866 28082036 1000 LEDVVIDRNLLILGKILGEGEFGSVMEGNLKQEDGTSLKVAVKTMAACMKDFSHPNVMRLLGVCIEMSSPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFPVKWIAIESLYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESL 5td7 A 2.85 BS02 FKS A 1 D94 P134 H136 H137 G145 F146 D174 H176 W205 E274 E304 G305 F307 D94 P134 H136 H137 G145 F146 D174 H176 W205 E274 E304 G305 F307 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 28516954 711 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGFNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFDLTDQNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCLREGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETAAKTRLMRVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGPLRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 5tdi A 1.4 BS01 7AS A 1 G23 C25 E59 N60 D61 G64 G65 G66 Y67 A134 L160 N161 H162 A163 G23 C25 E59 N60 D61 G64 G65 G66 Y67 A134 L160 N161 H162 A163 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 28049758 301 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLAPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 5tef A 1.95 BS01 GTG A 1 Y474 T540 L580 N582 K641 Y660 Y440 T498 L538 N540 K599 Y618 ? Kd=4uM remove_due_to_license_issue Q8TEQ6 27881600 801 QEPRTLPPSPNWYCARCSDAVPGGLFGFAARTSVFLVRVGPGAGESPGTPPFRVIGELVGHTERVSGFTFSHHPGQYNLCATSSDDGTVKIWDVETKTVVTEHALHQHTISTLHWSPRVKDLIVSGDEKGVVFCYWFNRNDSQHLFIEPRTIFCLTCSPHHEDLVAIGYKDGIVVIIDISKKGEVIHRLRGHDDEIHSIAWCPLPGECYLATGSKDQTIRIWSCSRGRGVMILKLPFLKRRGGGIDPTVKERLWLTLHWPSNQPTQLVSSCFGGELLQWDLTQRRKYTLFSASSEGQNHSRIVFNLCPLQTEDDKQLLLSTSMDRDVKCWDIATLECSWTLPSLGGFAYSLAFSSVDIGSLAIGVGDGMIRVWNTLSIKNNYDVKNFWQGVKSKVTALCWHPTKEGCLAFGTDDGKVGLYDTYSNKPPQISSTYHKKTVYTLAWGPPVPPMSSLALYSCGGEGIVLQHNPWKLSGEAFDINKLIRDTNSIKYKLPVHTEISWKADGKIMALGNEDGSIEIFQIPNLKLICTIQQHHKLVNTISWHHEHGSQPELSYLMASGSNNAVIYVHNLKTVIESSPESPVTITEPYRTLSGHTAKITSVAWSPHHDGRLVSASYDGTAQVWDALREEPLCNFRGHQGRLLCVAWSPLDPDCIYSGADDFCVHKWLTSMQDHSRPPQ 5teh A 2.99 BS01 S56 A 1 C281 A293 E310 M314 Y340 D404 C26 A38 E55 M59 Y85 D149 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F152 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00523 600 AKDAWEIPRESLRLEVKLGQGCFGECWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 5tex A 2.149 BS01 7AU A 1 L44 F49 A65 V126 L174 L12 F17 A33 V94 L142 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=0.4uM remove_due_to_license_issue IC50=400nM P11309 28947155 402 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 5tf6 A 2.3 BS01 rna B 0 T35 R36 R38 W120 T122 N123 R148 P150 S151 R153 F154 R158 R159 F160 Y162 N194 P195 K198 R201 T202 D203 E211 M213 R215 N216 N241 Q246 F251 N252 N253 C255 F257 R274 S283 D288 K289 K290 P291 F292 R295 K299 R300 T3 R4 R6 W88 T90 N91 R116 P118 S119 R121 F122 R126 R127 F128 Y130 N162 P163 K166 R169 T170 D171 E179 M181 R183 N184 N209 Q214 F219 N220 N221 C223 F225 R242 S251 D256 K257 K258 P259 F260 R263 K267 R268 ? 0003676,0003723 remove_due_to_license_issue P49960 28045380 30 ~ 100 MLTRNRELTTVLVKNLPKSYNQNKVYKYFKHCGPIIHVDVADSLKKNFRFARIEFARYDGALAAITKTHKVVGQNEIIVSHLTECTLWMTNFPPSYTQRNIRDLLQDINVVALSIRLPSLRFNTSRRFAYIDVTSKEDARYCVEKLNGLKIEGYTLVTKVSNPLEKSKRTDSATLEGREIMIRNLSTELLDENLLRESFEGFGSIEKINIPAGQKEHSFNNCCAFMVFENKDSAERALQMNRSLLGNREISVSLADKKPFLERNEVKRLLASRNSKELETLICLFPLSDKVSPSLICQFLQEEIHINEKDIRKILLVSDFNGAIIIFRDSKFAAKMLMILNGSQFQGKVIRSGTINDMKRYYNNQQN 5tf6 C 2.3 BS01 rna B 0 K62 H63 Y90 K102 K30 H31 Y58 K70 ? 0003676,0003723 remove_due_to_license_issue P49960 28045380 30 ~ 100 MLTRNRELTTVLVKNLPKSYNQNKVYKYFKHCGPIIHVDVADSLKKNFRFARIEFARYDGALAAITKTHKVVGQNEIIVSHLTECTLWMTNFPPSYTQRNIRDLLQDINVVALSIRLPSLRFNTSRRFAYIDVTSKEDARYCVEKLNGLKIEGYTLVTKVSNPLEKSKRTDSATLEGREIMIRNLSTELLDENLLRESFEGFGSIEKINIPAGQKEHSFNNCCAFMVFENKDSAERALQMNRSLLGNREISVSLADKKPFLERNEVKRLLASRNSKELETLICLFPLSDKVSPSLICQFLQEEIHINEKDIRKILLVSDFNGAIIIFRDSKFAAKMLMILNGSQFQGKVIRSGTINDMKRYYNNQQ 5tf6 C 2.3 BS02 rna D 0 M33 T35 R36 R38 W120 T122 N123 R148 P150 S151 F154 R158 R159 F160 Y162 S193 N194 P195 K198 R201 T202 D203 T206 E211 M213 R215 N216 K239 N241 P243 Q246 F251 N252 N253 C255 F257 S283 D288 K289 K290 P291 F292 R295 K299 M1 T3 R4 R6 W88 T90 N91 R116 P118 S119 F122 R126 R127 F128 Y130 S161 N162 P163 K166 R169 T170 D171 T174 E179 M181 R183 N184 K207 N209 P211 Q214 F219 N220 N221 C223 F225 S251 D256 K257 K258 P259 F260 R263 K267 ? 0003676,0003723 remove_due_to_license_issue P49960 28045380 30 ~ 101 MLTRNRELTTVLVKNLPKSYNQNKVYKYFKHCGPIIHVDVADSLKKNFRFARIEFARYDGALAAITKTHKVVGQNEIIVSHLTECTLWMTNFPPSYTQRNIRDLLQDINVVALSIRLPSLRFNTSRRFAYIDVTSKEDARYCVEKLNGLKIEGYTLVTKVSNPLEKSKRTDSATLEGREIMIRNLSTELLDENLLRESFEGFGSIEKINIPAGQKEHSFNNCCAFMVFENKDSAERALQMNRSLLGNREISVSLADKKPFLERNEVKRLLASRNSKELETLICLFPLSDKVSPSLICQFLQEEIHINEKDIRKILLVSDFNGAIIIFRDSKFAAKMLMILNGSQFQGKVIRSGTINDMKRYYNNQQ 5tfx A 1.5 BS02 7B1 A 1 I91 Q92 H94 H96 H119 F131 L198 T199 T200 I89 Q90 H92 H94 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=60.9nM remove_due_to_license_issue P00918 27892589 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5tg1 A 1.4 BS01 V56 A 1 H30 I109 Q110 G133 T134 I135 P136 C139 A158 A159 A160 H27 I106 Q107 G128 T129 I130 P131 C134 A153 A154 A155 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 28038326 203 TLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLANAKGMDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSNTVVCAVQ 5tg2 A 1.75 BS01 V69 A 1 H30 I109 Q110 C139 A158 A159 A160 H29 I108 Q109 C130 A149 A150 A151 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 28038326 201 PPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGDCGAPYVHKRGNDWVVCGVHAAATGNTVVCAVQA 5tg4 A 1.44 BS01 JW1 A 1 S81 K84 W115 S128 V130 L168 W221 M223 S51 K54 W85 S98 V100 L138 W191 M193 S81 K84 S128 Y133 W167 W221 S51 K54 S98 Y103 W137 W191 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 27997706 301 MHISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPEWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 5tg5 A 1.75 BS01 JW8 A 1 S81 W115 S128 V130 L168 W221 M223 S51 W85 S98 V100 L138 W191 M193 S81 K84 S128 Y133 W167 W221 S51 K54 S98 Y103 W137 W191 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 27997706 301 MHISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 5tg5 A 1.75 BS02 JW8 A 2 Y112 L127 W221 G258 R261 Y82 L97 W191 G228 R231 S81 K84 S128 Y133 W167 W221 S51 K54 S98 Y103 W137 W191 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 27997706 302 MHISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 5tg6 A 1.78 BS01 J4W A 1 S81 W115 S128 V130 L168 W221 M223 G224 S51 W85 S98 V100 L138 W191 M193 G194 S81 K84 S128 Y133 W167 W221 S51 K54 S98 Y103 W137 W191 ? 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 27997706 301 MHISSQQHEKAIKSYFDPAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 5tg7 A 2.28 BS01 JW3 A 1 S81 S128 L168 W221 M223 S50 S97 L137 W190 M192 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 3.5.2.6 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 27997706 301 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPPWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 5tgc A 3.245 BS01 ATP A 1 S14 H15 R16 A161 G186 K232 S233 S397 K433 S15 H16 R17 A155 G180 K215 S216 S342 K378 ? 0000785,0003674,0003682,0005198,0005515,0005634,0006325,0006337,0006338,0006355,0006357,0006368,0016514,0016586,0035267,0043232,0045944 remove_due_to_license_issue Q12406 29809203 501 MMTLNRKCVVIHNGSHRTVAGFSNVELPQCIIPSSYIKREFIFGTYNMIDAAAEKRNGDEVYTLVDSQGLPYNWDALEMQWRYLYDTQLKVSPEELPLVITMPATNGKPDMAILERYYELAFDKLNVPVFQIVIEPLAIALSMGKSSAFVIDIGASGCNVTPIIDGIVVKNAVVRSKFGGDFLDFQVHERLAPLIKQKRSTDVWYEASTWIQQFKSTMLQVSEKDLFELERYYKEQADIYAKQQEQLKQMDQQLQYTANNPLVQKKNFLFKPLNKTLTLDLKECYQFAEYLFKPQLISDKFSPEDGLGPLMAKSVKKAGASINISPEQVYSLLLTNVIITGSTSLIEGMEQRIIKELSIRFPQYKLTTFANQVMMDRKIQGWLGALTMANLPSWSLGKWYSKEDYET 5tgy A -1.00 BS01 7BU A 1 L6 R7 H46 R47 F50 A56 G65 D66 W68 V69 L98 I101 R102 A105 L6 R7 H46 R47 F50 A56 G65 D66 W68 V69 L98 I101 R102 A105 0044780 remove_due_to_license_issue 29168496 201 SEFEKLRQTGDELVQAFQRLREIFDKGDDDSLEQVLEEIEELIQKHRQLFDNRQEAADTEAAKQGDQWVQLFQRFREAIDKGDKDSLEQLLEELEQALQKIRELAEKKN 5th4 A 1.47 BS02 BEW A 1 H94 H96 H119 T199 T200 W209 H91 H93 H116 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 28389830 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSGTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5th7 A 1.95 BS01 7BY A 1 Y286 C311 Y312 M313 Y314 R336 T348 Y375 Y51 C76 Y77 M78 Y79 R101 T113 Y140 2.1.1.-,2.1.1.361 0042799 remove_due_to_license_issue Q9NQR1 27804297 401 KAELQSEERKRIDELIESGKEEGMKIDLIDGKGRGVIATKQFSRGDFVVEYHGDLIEITDAKKREALYAQDPSTGCYMYYFQYLSKTYCVDATRETNRLGRLINHSKSGNCQTKLHDIDGVPHLILIASRDIAAGEELLYDYG 5th7 A 1.95 BS02 7BY B 1 E300 P307 C311 E65 P72 C76 2.1.1.-,2.1.1.361 0042799 remove_due_to_license_issue Q9NQR1 27804297 402 KAELQSEERKRIDELIESGKEEGMKIDLIDGKGRGVIATKQFSRGDFVVEYHGDLIEITDAKKREALYAQDPSTGCYMYYFQYLSKTYCVDATRETNRLGRLINHSKSGNCQTKLHDIDGVPHLILIASRDIAAGEELLYDYG 5th7 B 1.95 BS01 7BY A 1 E300 P307 C311 E65 P72 C76 2.1.1.-,2.1.1.361 0042799 remove_due_to_license_issue Q9NQR1 27804297 401 KAELQSEERKRIDELIESGKEEGMKIDLIDGKGRGVIATKQFSRGDFVVEYHGDLIEITDAKKREALYAQDPSTGCYMYYFQYLSKTYCVDATRETNRLGRLINHSKSGNCQTKLHDIDGVPHLILIASRDIAAGEELLYDYGDR 5th7 B 1.95 BS02 7BY B 1 Y286 C311 Y312 M313 Y314 R336 T348 Y375 Y51 C76 Y77 M78 Y79 R101 T113 Y140 2.1.1.-,2.1.1.361 0042799 remove_due_to_license_issue Q9NQR1 27804297 402 KAELQSEERKRIDELIESGKEEGMKIDLIDGKGRGVIATKQFSRGDFVVEYHGDLIEITDAKKREALYAQDPSTGCYMYYFQYLSKTYCVDATRETNRLGRLINHSKSGNCQTKLHDIDGVPHLILIASRDIAAGEELLYDYGDR 5tha A 1.8 BS01 GP3 A 1 Y474 T540 N582 Y660 Y442 T501 N543 Y621 ? Kd=140uM remove_due_to_license_issue Q8TEQ6 27881600 822 QEPRTLPPSPNWYCARCSDAVPGGLFGFAARTSVFLVRVGPGAGESPGTPPFRVIGELVGHTERVSGFTFSHHPGQYNLCATSSDDGTVKIWDVETKTVVTEHALHQHTISTLHWSPRVKDLIVSGDEKGVVFCYWFNRNDSQHLFIEPRTIFCLTCSPHHEDLVAIGYKDGIVVIIDISKKGEVIHRLRGHDDEIHSIAWCPLPGEGCYLATGSKDQTIRIWSCSRGRGVMILKLPFLKRRGGGIDPTVKERLWLTLHWPSNQPTQLVSSCFGGELLQWDLTQSRRKYTLFSASSEGQNHSRIVFNLCPLQTEDDKQLLLSTSMDRDVKCWDIATLECSWTLPSLGGFAYSLAFSSVDIGSLAIGVGDGMIRVWNTLSIKNNYDVKNFWQGVKSKVTALCWHPTKEGCLAFGTDDGKVGLYDTYSNKPPQISSTYHKKTVYTLAWGPPVPPMSLSLALYSCGGEGIVLQHNPWKLSGEAFDINKLIRDTNSIKYKLPVHTEISWKADGKIMALGNEDGSIEIFQIPNLKLICTIQQHHKLVNTISWHHEHGSQPELSYLMASGSNNAVIYVHNLKTVIESSPESPVTITEPYRTLSGHTAKITSVAWSPHHDGRLVSASYDGTAQVWDALREEPLCNFRGHQGRLLCVAWSPLDPDCIYSGADDFCVHKWLTSMQDHSRPPQG 5thi A 1.5 BS02 0TR A 1 H94 H96 H119 G198 T199 T200 H91 H93 H116 G194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=245uM remove_due_to_license_issue P00918 28389830 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSGTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5thn A 1.33 BS02 7CZ A 1 H94 H96 H119 V121 T199 T200 H91 H93 H116 V118 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=96uM remove_due_to_license_issue P00918 28389830 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5tho H 3.002 BS01 7C7 H 1 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue A5U4D6 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5tho H 3.002 BS02 7C7 N 1 L91 S122 F123 D124 A125 W129 L91 S122 F123 D124 A125 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue A5U4D6 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5tho I 3.002 BS01 7C7 H 1 D124 G128 W129 D124 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue A5U4D6 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5tho I 3.002 BS02 7C7 I 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue A5U4D6 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5tho Y 3.002 BS01 7C7 X 1 L91 F123 D124 A125 A126 W129 L91 F123 D124 A125 A126 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue A5U4D6 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5tho Y 3.002 BS02 7C7 Y 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue A5U4D6 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5ti0 A 1.42 BS02 7CZ A 1 H94 H96 H119 T199 T200 H91 H93 H116 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=61uM remove_due_to_license_issue P00918 28389830 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSGTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ti2 A 1.65 BS01 7CJ A 1 V87 L92 L94 N140 I146 V46 L51 L53 N99 I105 ? ic50=24uM remove_due_to_license_issue O60885 28884163 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ti3 A 1.703 BS01 7CG A 1 V87 L92 L94 N140 I146 M149 V46 L51 L53 N99 I105 M108 ? ic50=44uM remove_due_to_license_issue O60885 28884163 205 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ti4 A 1.62 BS01 7CM A 1 W81 P82 V87 L92 N140 D145 I146 M149 W40 P41 V46 L51 N99 D104 I105 M108 ? ic50=26uM remove_due_to_license_issue O60885 28884163 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ti5 A 1.83 BS01 7CN A 1 F83 V87 L92 L94 N140 I146 M149 F42 V46 L51 L53 N99 I105 M108 ? ic50=41uM remove_due_to_license_issue O60885 28884163 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ti6 A 1.704 BS01 7CO A 1 W81 P82 F83 L92 L94 N140 I146 W40 P41 F42 L51 L53 N99 I105 ? ic50=21uM remove_due_to_license_issue O60885 28884163 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5ti7 A 1.65 BS01 7CQ A 1 W81 L94 N140 I146 M149 W40 L53 N99 I105 M108 ? ic50=11uM remove_due_to_license_issue O60885 28884163 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5tig A 2.7 BS01 7DH B 1 F50 R61 F50 R61 P1 R39 F50 R61 P1 R39 F50 R61 5.3.2.6 0009056,0016853,0042184,0042203 remove_due_to_license_issue Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELASKVRR 5tig B 2.7 BS01 7DH B 1 P1 S37 P1 S37 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 remove_due_to_license_issue Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELAS 5tiu A 1.49 BS01 7CU A 1 L377 A400 M448 M450 A451 G454 P455 R498 L501 D512 L15 A33 M75 M77 A78 G81 P82 R125 L128 D139 D494 A496 R498 N499 D512 K533 D121 A123 R125 N126 D139 K160 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5nM remove_due_to_license_issue IC50=5.2nM P43405 27994755 701 VYLDRKLLTLEDKELGTVKKGYYQMKKVVKTVAVKILKALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH 5tjx A 1.408 BS01 GBT A 1 H434 S478 E479 G480 Y555 M561 A573 C574 S578 S597 W598 G599 G601 C602 H44 S88 E89 G90 Y160 M166 A178 C179 S183 S202 W203 G204 G206 C207 H434 D483 K575 G576 D577 S578 G579 H44 D93 K180 G181 D182 S183 G184 3.4.21.34 0004252,0006508 remove_due_to_license_issue IC50=4.8nM P03952 28197309 701 IVGGTESSWGEWPWQVSLQVKLTAQRHLCGGSLIGHQWVLTAAHCFDGLPLQDVWRIYSGILELSDITKDTPFSQIKEIIIHQNYKVSEGNHDIALIKLQAPLEYTEFQKPISLPSTIYTNCWVTGWGFSKEKGEIQNILQKVNIPLVTNEECQKRYQDYKITQRMVCAGYKEGGKDACKGDSGGPLVCKHNGMWRLVGITSWGEGCARREQPGVYTKVAEYMDWILEKTQ 5tkb A 2.16 BS02 7DJ A 1 M439 I502 M523 Q535 F538 M190 I250 M271 Q283 F286 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 30108788 807 VKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 5tkd A 1.92 BS01 7GL A 1 L595 G596 V603 V640 K642 Y689 V690 G693 P694 R738 L741 L15 G16 V23 V33 K35 Y82 V83 G86 P87 R131 L134 N734 R738 N739 D759 N127 R131 N132 D152 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue P29597 30108788 901 FHRVDQKEITQLSHLGQGTRTNVYEGRLRLRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLRSPSEKEHFYQRQHRLPEPSLATLTSQCLTYEPTQRPSFRTILRDL 5tks A 1.55 BS01 7DL A 1 R39 H40 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 V227 R26 H27 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=68nM remove_due_to_license_issue Ki=68nM P03951 28085275 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5tkt A 2.12 BS01 7DS A 1 R39 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=3.2nM remove_due_to_license_issue Ki=0.160000nM P03951 28085275 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5tku A 2.12 BS01 7DK A 1 R39 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.16nM remove_due_to_license_issue Ki=3.2nM P03951 28085275 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5tl9 A 1.2 BS01 7DN A 1 Y28 G35 F44 R52 H53 Y24 G31 F40 R48 H49 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=1nM remove_due_to_license_issue IC50=6.0nM O14684 28190634 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5tln A 2.3 BS06 BAN A 1 N112 F130 L133 V139 H142 E143 H146 E166 L202 R203 D226 H231 N112 F130 L133 V139 H142 E143 H146 E166 L202 R203 D226 H231 H142 E143 H146 Y157 E166 D226 H231 H142 E143 H146 Y157 E166 D226 H231 3.4.24.27 0004222,0006508 Ki=0.43uM remove_due_to_license_issue Ki=99999999999999nM P00800 7317361 322 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5tmn E 1.6 BS01 0PJ E 1 N112 A113 F114 F130 E143 H146 Y157 L202 R203 H231 N112 A113 F114 F130 E143 H146 Y157 L202 R203 H231 3.4.24.27 0004222,0006508 Ki=9.1nM remove_due_to_license_issue Ki=99999999999999nM P00800 3442675 317 ITGTSTVGVGRGVLGDQKNINTTYSTYYYLQDNTRGDGIFTYDAKYRTTLPGSLWADADNQFFASYDAPAVDAHYYAGVTYDYYKNVHNRLSYDGNNAAIRSSVHYSQGYNNAFWNGSEMVYGDGDGQTFIPLSGGIDVVAHELTHAVTDYTAGLIYQNESGAINEAISDIFGTLVEFYANKNPDWEIGEDVYTPGISGDSLRSMSDPAKYGDPDHYSKRYTGTQDNGGVHINSGIINKAAYLISQGGTHYGVSVVGIGRDKLGKIFYRALTQYLTPTSNFSQLRAAAVQSATDLYGSTSQEVASVKQAFDAVGVK 5tmp A 1.98 BS01 Z5A A 1 E12 G13 G15 K16 T17 E40 R51 F74 R100 S104 T105 Y108 Q109 R149 R153 I159 E11 G12 G14 K15 T16 E39 R50 F73 R99 S103 T104 Y107 Q108 R148 R152 I158 2.7.4.9 0004798,0005524,0005737,0005829,0006227,0006233,0006235,0009165,0015949,0016301,0042803,0046940 Kd=34nM remove_due_to_license_issue P0A720 9826650 214 RSKYIVIEGLEGAGKTTARNVVVETLEQLGIRDMVFTREPGGTQLAEKLRSLLLDIKSVGDEVITDKAEVLMFYAARVQLVETVIKPALANGTWVIGDRHDLSTQAYQGGGRGIDQHMLATLRDAVLGDFRPDLTLYLDVTPEVGLKRARARGELDRIEQESFDFFNRTRARYLELAAQDKSIHTIDATQPLEAVMDAIRTTVTHWVKEL 5tnt A 1.4 BS01 7GQ A 1 Y99 F174 D189 S190 C191 Q192 W215 G216 E217 C220 Y86 F162 D179 S180 C181 Q182 W205 G206 E207 C209 H57 D102 Q192 G193 D194 S195 G196 H41 D89 Q182 G183 D184 S185 G186 3.4.21.22 0004252,0006508 ic50=4.9nM remove_due_to_license_issue IC50=550nM P00740 28408226 301 VVGGEDAKPGQFPWQVVLNGKVDAFCGGSIVNEKWIVTAAHCVETGVKITVVAGEHNIEETEHTEQKRNVIRIIPHHNYNAAINKYNHDIALLELDEPLVLNSYVTPICIADKEYTNIFLKFGSGYVSGWGRVFHKGASALVLQYLRVPLVDRATCLRSTKFTIYNNMFCAGFHEGGRDSCQGDSGGPHVTEVEGTSFLTGIISWGEECAMKGKYGIYTKVSRYVNWIKEKTKLT 5to8 A 1.9849 BS01 7FM A 1 L431 G432 E433 M502 E503 L504 Y505 G508 E509 R553 L556 L12 G13 E14 M79 E80 L81 Y82 G85 E86 R128 L131 D549 A551 R553 N554 D567 D124 A126 R128 N129 D142 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3.1nM remove_due_to_license_issue IC50=3.1nM Q14289 27876318 701 IAREDVVLNRILGEGFFGEVYEGVYTNHKGEKINVAVKTCKKDCTNKEKFMSEAVIMKNLDHPHIVKLIGIIEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESCVHRDIAVRNILVASPECVKLGDFGLSRIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIAM 5tob A 2.117 BS01 YAM A 1 L431 G432 E433 M502 E503 L504 Y505 G508 E509 R553 L556 L12 G13 E14 M75 E76 L77 Y78 G81 E82 R126 L129 D549 A551 R553 N554 D567 D122 A124 R126 N127 D140 2.7.10.2 0004672,0004713,0005524,0006468 ic50=13nM remove_due_to_license_issue IC50=13nM Q14289 27876318 701 IAREDVVLNRILGEGFFGEVYEGVYTHKGEKINVAVKTCKDNKEKFMSEAVIMKNLDHPHIVKLIGIIEPTWIIMELYPYGELGHYLERNKNSLKVLTLVLYSLQICKAMAYLESINCVHRDIAVRNILVASPECVKLGDFGPIKWMSPESINFRRFTTASDVWMFAVCMWEILSFGKQPFFWLENKDVIGVLEKGDRLPKPDLCPPVLYTLMTRCWDYDPSDRPRFTELVCSLSDVYQMEKDIA 5toe A 2.301 BS01 7GK A 1 A65 L120 R122 D131 L174 A32 L86 R88 D97 L140 D167 K169 N172 D186 L193 T204 D133 K135 N138 D152 L159 T170 2.7.11.1 0004672,0004674,0005524,0006468,0043066 ic50=2.5uM remove_due_to_license_issue IC50=2500nM P11309 28947155 401 LESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 5tol A 2.51 BS01 7H3 A 1 G59 G61 L78 D80 Y119 F156 D276 S277 G278 T280 G15 G17 L34 D36 Y75 F112 D220 S221 G222 T224 D80 S83 N85 A87 Y119 D276 T279 D36 S39 N41 A43 Y75 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=33nM P56817 27816517 501 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGSVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQATTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5toz A 1.98 BS01 7H4 A 1 L828 A853 M902 Y904 L905 G908 C909 D912 L956 L14 A39 M84 Y86 L87 G90 C91 D94 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 27791347 1201 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 5tp0 A 1.25 BS02 BRN A 1 D189 S190 C191 W215 G216 G219 C220 D171 S172 C173 W193 G194 G196 C197 H57 D102 Q192 R193 D194 S195 G196 H40 D84 Q174 R175 D176 S177 G178 3.4.21.4 0004252,0006508 Ki=3.66uM remove_due_to_license_issue P35030 28463992 306 IVGGYTCEENSLPYQVSLNSGSHFCGGSLISEQWVVSAAHCYKTRIQVRLGEHNIKVLEGNEQFINAAKIIRHPKYNRDTLDNDIMLIKLSSPAVINARVSTISLPTAPPAAGTECLISGWGNTLSFGADYPDELKCLDAPVLTQAECKASYPGKITNSMFCVGFLEGGKDSCQRDSGGPVVCNGQLQGVVSWGHGCAWKNRPGVYTKVYNYVDWIKDTIAANS 5tpb B 2.6 BS02 SIA B 1 Y1267 G1279 Y382 G389 Q913 N979 Q37 N103 3.4.24.69 0005576 remove_due_to_license_issue P0DPI1 27958736 2301 SILNLRYESNHLIDLSRYASKINIGSKVNFDPIDKNQIQLFNLESSKIEVILKNAIVYNSMYENFSTSFWIRIPKYFNSISLNNEYTIINCMENNSGWKVSLNYGEIIWTLQDTQEIKQRVVFKYSQMINISDYINRWIFVTITNNRLNNSKIYINGRLIDQKPISNLGNIHASNNIMFKLDGCRDTHRYIWIKYFNLFDKELNEKEIKDLYDNQSNSGILKDFWGDYLQYDKPYYMLNLYDPNKYVDVNNVGIRGYMYLKGPRGSVMTTNIYLNSSLYRGTKFIIKKYASGNKDNIVRNNDRVYINVVVKNKEYRLATNASQAGVEKILSALEIPDVGNLSQVVVMKSCKMNLQDNNGNDIGFIGFHQFNNIAKLVASNWYNRQRTLGCSWEFIPVDDGWGERPLQ 5tpc A 2.0 BS01 GAL C 1 E1203 F1252 H1253 S1264 W1266 E331 F380 H381 S392 W394 Q913 N979 Q41 N107 3.4.24.69 0005576 remove_due_to_license_issue P0DPI1 27958736 2 HMDTSILNLRYESNHLIDLSRYASKINIGSKVNFDPIDKNQIQLFNLESSKIEVILKNAIVYNSMYENFSTSFWIRIPKYFNSISLNNEYTIINCMENNSGWKVSLNYGEIIWTLQDTQEIKQRVVFKYSQMINISDYINRWIFVTITNNRLNNSKIYINGRLIDQKPISNLGNIHASNNIMFKLDGCRDTHRYIWIKYFNLFDKELNEKEIKDLYDNQSNSGILKDFWGDYLQYDKPYYMLNLYDPNKYVDVNNVGIRGYMYLKGPRGSVMTTNIYLNSSLYRGTKFIIKKYASGNKDNIVRNNDRVYINVVVKNKEYRLATNASQAGVEKILSALEIPDVGNLSQVVVMKSKNDQGITNKCKMNLQDNNGNDIGFIGFHQFNNIAKLVASNWYNRQIERSSRTLGCSWEFIPVDDGWGERPLQ 5tpc A 2.0 BS02 SIA C 1 Y1117 F1252 Y245 F380 Q913 N979 Q41 N107 3.4.24.69 0005576 remove_due_to_license_issue P0DPI1 27958736 3 HMDTSILNLRYESNHLIDLSRYASKINIGSKVNFDPIDKNQIQLFNLESSKIEVILKNAIVYNSMYENFSTSFWIRIPKYFNSISLNNEYTIINCMENNSGWKVSLNYGEIIWTLQDTQEIKQRVVFKYSQMINISDYINRWIFVTITNNRLNNSKIYINGRLIDQKPISNLGNIHASNNIMFKLDGCRDTHRYIWIKYFNLFDKELNEKEIKDLYDNQSNSGILKDFWGDYLQYDKPYYMLNLYDPNKYVDVNNVGIRGYMYLKGPRGSVMTTNIYLNSSLYRGTKFIIKKYASGNKDNIVRNNDRVYINVVVKNKEYRLATNASQAGVEKILSALEIPDVGNLSQVVVMKSKNDQGITNKCKMNLQDNNGNDIGFIGFHQFNNIAKLVASNWYNRQIERSSRTLGCSWEFIPVDDGWGERPLQ 5tpg A 1.5 BS02 7H5 A 1 Y235 P238 F241 R257 Y264 T265 P266 E267 A309 Y312 E317 S336 S337 Y112 P115 F118 R134 Y141 T142 P143 E144 A186 Y189 E194 S213 S214 H272 H277 E317 S336 H149 H154 E194 S213 1.14.16.4 0004497,0005506,0009072,0016714 ic50=14nM remove_due_to_license_issue IC50=14nM P17752 28041831 505 TVPWFPKKISDLDHCNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFQELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTIK 5tpx A 2.1 BS01 7H7 A 1 W1379 P1380 K1383 P1384 V1385 E1389 N1436 Y1442 W25 P26 K29 P30 V31 E35 N82 Y88 2.3.1.48 0004402 Kd=280nM remove_due_to_license_issue Q8IB67 27966810 1505 GHKEVQLKDQILGVLDYLEKQQSAWPFLKPVSLSEAPDYYDIIKEPTDILTMRRKARHGDYKTKEDFGIELKRMFDNCRLYNAPTTIYFKYANELQTLIWPKYEAI 5tq3 A 2.69 BS01 7GZ A 1 L855 A880 K882 E898 L902 M929 E930 Y931 L932 G935 L983 G993 L13 A38 K40 E56 L60 M87 E88 Y89 L90 G93 L141 G151 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S172 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=2.2nM O60674 27983835 4000 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNQSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQVRDNMAG 5tq4 A 2.3 BS01 7GY A 1 L932 D994 L92 D154 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4.2nM remove_due_to_license_issue IC50=4.2nM O60674 27983835 4000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 5tq5 A 2.3 BS01 7GX A 1 L855 A880 E898 M929 E930 Y931 L932 P933 G935 L983 D994 F995 L15 A40 E58 M89 E90 Y91 L92 P93 G95 L143 D154 F155 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0004713,0005524,0006468 ic50=58.8nM remove_due_to_license_issue IC50=59nM O60674 27983835 4000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 5tq6 A 2.06 BS01 7GV A 1 L855 G856 G858 V863 A880 K882 M929 Y931 L932 L983 D994 L13 G14 G16 V21 A38 K40 M83 Y85 L86 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S167 2.7.10.2 0004672,0004713,0005524,0006468 ic50=123.6nM remove_due_to_license_issue IC50=124nM O60674 27983835 4000 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMISIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 5tq7 A 2.1 BS01 7GT A 1 L855 K857 G858 G861 S862 V863 A880 Y931 L932 L983 D994 L15 K17 G18 G21 S22 V23 A40 Y86 L87 L138 D149 D976 A978 R980 N981 D994 S1016 D131 A133 R135 N136 D149 S167 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue O60674 27983835 4000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQVRDNMAG 5tq8 A 1.59 BS01 7GS A 1 Q854 L855 K857 A880 K882 E898 M929 E930 Y931 L932 G935 L983 G993 D994 F995 Q14 L15 K17 A40 K42 E58 M89 E90 Y91 L92 G95 L143 G153 D154 F155 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0004713,0005524,0006468 ic50=23.1nM remove_due_to_license_issue O60674 27983835 4000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 5tqe H 1.9 BS01 7KQ H 1 L41 C42 H57 K60A G97 T98 T99 D189 S190 K192 S195 S214 W215 G216 Q217 G219 L25 C26 H41 K45 G85 T86 T87 D184 S185 K187 S190 S209 W210 G211 Q212 G213 3.4.21.21 0004252,0006508 Ki=190nM remove_due_to_license_issue Ki=190nM P08709 28105277 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5tqf H 1.85 BS01 7KR H 1 L41 C42 H57 K60A D189 S190 K192 S195 S214 W215 G216 Q217 G219 L25 C26 H41 K45 D182 S183 K185 S188 S207 W208 G209 Q210 G211 3.4.21.21 0004252,0006508 Ki<5nM remove_due_to_license_issue Ki=58nM P08709 28105277 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5tqg H 1.9 BS01 7KS H 1 L41 C42 H57 K60A P170I D189 S190 K192 S195 S214 W215 G216 Q217 G219 C220 L25 C26 H41 K45 P165 D182 S183 K185 S188 S207 W208 G209 Q210 G211 C212 3.4.21.21 0004252,0006508 Ki=0.24nM remove_due_to_license_issue Ki=0.240000nM P08709 28105277 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5tqu B 2.6 BS01 I53 B 1 I248 Y250 D287 H289 G290 Y472 V473 W474 Y481 F522 I17 Y19 D56 H58 G59 Y211 V212 W213 Y220 F261 H256 H259 S364 K554 K557 H25 H28 S133 K293 K296 6.1.1.10 0000166,0004812,0004825,0005524,0006418,0006431 remove_due_to_license_issue Q38C91 28110521 801 GPGSMKVEKVFFVTSPIYYVNAAPHIGHVYSTLITDVIGRYHRVKGERVFALTGTDEHGQKVAEAAKQKQVSPYDFTTAVAGEFKKCFEQMDYSIDYFIRTTNEQHKAVVKELWTKLEQKGDIYLGRYEGWYSISVTWVSEENYMFRLSAFRERLLEWYHANPGCIVPEFRRREVIRAVEKGLPDLSVSRARATLHNWAIPVPGNPDHCVYVWLDALTNYLTGSRLRVDESGKEVSLVDDFNELERFPADVHVIGKDILKFHAIYWPAFLLSAGLPLPKKIVAHGWWTKDRKKISKSLGNVFDPVEKAEEFGYDALKYFLLRESGFSDDGDYSDKNMIARLNGELADTLGNLVMRCTSAKINVNGEWPSPAAYTEEDESLIQLIKDLPGTADHYYLIPDIQKAIIAVFDVLRAINAYVTDMAPWKLVKTDPERLRTVLYITLEGVRVTTLLLSPILPRKSVVIFDMLGVPEVHRKGIENFEFGAVPPGTRLGPAVEGEVLFSKRST 5tr6 A 1.93 BS01 7KG A 1 A400 E449 M450 A451 G454 P455 R498 L501 S511 D512 A39 E82 M83 A84 G87 P88 R131 L134 S144 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3.2nM remove_due_to_license_issue IC50=2.0nM, EC50=9.8nM P43405 27839918 701 EVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHHH 5trf A 2.1 BS01 7HC A 1 V14 L54 L57 G58 I61 M62 Y67 F86 V93 H96 I99 Y100 V5 L45 L48 G49 I52 M53 Y58 F73 V80 H83 I86 Y87 2.3.2.27 0005634,0043066,0051726 Ki=0.88nM remove_due_to_license_issue Ki=0.880000nM, Kd=2.7nM Q00987 25145672 201 TDGAVTTSQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 5trg H 2.804 BS01 7HJ H 1 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trg H 2.804 BS02 7HJ N 1 D124 G128 W129 D124 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trg I 2.804 BS01 7HJ H 1 L91 M95 D124 A125 A126 G128 W129 L91 M95 D124 A125 A126 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trg I 2.804 BS02 7HJ I 1 S20 T21 Q22 S27 V31 K33 I45 A49 A52 S20 T21 Q22 S27 V31 K33 I45 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trg Y 2.804 BS01 7HJ X 1 L91 D124 G128 W129 L91 D124 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5trg Y 2.804 BS02 7HJ Y 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5trh A 2.7 BS02 7HL A 1 F193 C366 G410 M414 Y415 Y448 G449 F170 C343 G387 M391 Y392 Y425 G426 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 27908764 602 SMSYTWTGALITPCYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSLSRARPRWFM 5tri A 2.3 BS02 7HM A 1 F193 R200 C366 L384 G410 M414 Y415 Y448 F171 R178 C344 L362 G388 M392 Y393 Y426 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 27908764 602 SMSYTWTGALITPCVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSL 5trj A 2.57 BS02 7HO A 1 F193 P197 C316 C366 S368 L384 R386 G410 N411 M414 Y415 Q446 Y448 G449 F171 P175 C294 C344 S346 L362 R364 G388 N389 M392 Y393 Q424 Y426 G427 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 27908764 602 SMSYTWTGALITPCVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSLSRARPRWFM 5trk A 2.06 BS02 7HH A 1 F193 P197 S288 C316 C366 S368 L384 G410 M414 Y415 Q446 Y448 S556 F171 P175 S266 C294 C344 S346 L362 G388 M392 Y393 Q424 Y426 S534 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0003723,0003968,0039694 remove_due_to_license_issue Q9WMX2 27908764 602 SMSYTWTGALITPCVYATTSRSASLRQKKVTFDRLQVLDDHYRDVLKEMKAKASTVKAKLLSVEEACKLTPPHSARSKFGYGAKDVRNLSSKAVNHIRSVWKDLLEDTETPIDTTIMAKNEVFCVQPEKGGRKPARLIVFPDLGVRVCEKMALYDVVSTLPQAVMGSSYGFQYSPGQRVEFLVNAWKAKKCPMGFAYDTRCFDSTVTENDIRVEESIYQCCDLAPEARQAIRSLTERLYIGGPLTNSKGQNCGYRRCRASGVLTTSCGNTLTCYLKAAAACRAAKLQDCTMLVCGDDLVVICESAGTQEDEASLRAFTEAMTRYSAPPGDPPKPEYDLELITSCSSNVSVAHDASGKRVYYLTRDPTTPLARAAWETARHTPVNSWLGNIIMYAPTLWARMILMTHFFSILLAQEQLEKALDCQIYGACYSIEPLDLPQIIQRLHGLSAFSLHSYSPGEINRVASCLRKLGVPPLRVWRHRARSVRARLLSQGGRAATCGKYLFNWAVRTKLKLTPIPAASQLDLSSWFVAGYSGGDIYHSLSRARPRWFM 5trr H 3.103 BS01 7HY H 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trr H 3.103 BS02 7HY N 1 F123 D124 W129 F123 D124 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trr I 3.103 BS01 7HY H 1 L91 M95 D124 A126 G128 W129 L91 M95 D124 A126 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trr I 3.103 BS02 7HY I 1 S20 T21 Q22 S27 V31 K33 I45 A49 A52 L98 S20 T21 Q22 S27 V31 K33 I45 A49 A52 L98 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trr Y 3.103 BS01 7HY X 1 F123 D124 A126 W129 F123 D124 A126 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5trr Y 3.103 BS02 7HY Y 1 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 A52 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5trs H 3.08357 BS01 7HZ H 1 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trs H 3.08357 BS02 7HZ N 1 S122 D124 S122 D124 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trs I 3.08357 BS01 7HZ H 1 S122 D124 S122 D124 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trs I 3.08357 BS02 7HZ I 1 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 A52 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5trs Y 3.08357 BS01 7HZ X 1 S122 D124 W129 N130 S122 D124 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5trs Y 3.08357 BS02 7HZ Y 1 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5try H 3.00001 BS01 7J0 H 1 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5try H 3.00001 BS02 7J0 N 1 L91 S122 D124 A125 W129 N130 L91 S122 D124 A125 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5try I 3.00001 BS01 7J0 H 1 M95 S122 D124 W129 N130 M95 S122 D124 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5try I 3.00001 BS02 7J0 I 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 A52 L98 S20 T21 Q22 S27 V31 K33 I45 G47 A49 A52 L98 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5try Y 3.00001 BS01 7J0 X 1 L91 G128 W129 N130 L91 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5try Y 3.00001 BS02 7J0 Y 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5ts0 H 2.8468 BS01 7J1 H 1 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5ts0 H 2.8468 BS02 7J1 N 1 D124 W129 N130 D124 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5ts0 I 2.8468 BS01 7J1 H 1 L91 D124 G128 W129 L91 D124 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5ts0 I 2.8468 BS02 7J1 I 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 L98 S20 T21 Q22 S27 V31 K33 I45 G47 A49 L98 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 5ts0 Y 2.8468 BS01 7J1 X 1 D124 W129 D124 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5ts0 Y 2.8468 BS02 7J1 Y 1 S20 T21 S27 V31 K33 I45 G47 T48 A49 L98 S20 T21 S27 V31 K33 I45 G47 T48 A49 L98 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 27976853 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 5tt3 A 2.2 BS02 EZL A 1 H110 H112 H129 L190 T191 W201 H89 H91 H108 L166 T167 W177 H85 H110 H112 E116 H129 T191 H64 H89 H91 E95 H108 T167 ? 0004089,0008270,0046872 Ki=193nM remove_due_to_license_issue A0A0M3KL20 28002963 303 KWDYKNKENGPHRWDKLHKDFEVCKSGKSQSPINIEHYYHTQDKADLQFKYAASKPKAVFFTHHTLKASFEPTNHINYRGHDYVLDNVHFHAPMEFLINNKTRPLSAHFVHKDAKGRLLVLAIGFEEGKENPNLDPILEGIQNFKEVALDAFLPKSINYYHFNGSLTAPPCTEGVAWFVIEEPLEVSAKQLAEIKKRMKNSPNQRPVQPDYNTVIIKSSAETR 5tt7 A 1.77 BS01 7KF A 1 A400 M448 E449 M450 G454 P455 R498 L501 S511 D512 A40 M83 E84 M85 G89 P90 R133 L136 S146 D147 D494 A496 R498 N499 D512 K533 D129 A131 R133 N134 D147 K168 2.7.10.2 0004672,0004713,0005524,0006468 ic50=13nM remove_due_to_license_issue IC50=13nM, EC50=35nM P43405 27839918 901 IRPKEVYLDRKLLTLEDKELGSGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHHH 5tt8 A 2.4 BS02 D8W A 1 K88 D107 N108 H110 H112 H129 L190 T191 W201 K58 D77 N78 H80 H82 H99 L146 T147 W157 H85 H110 H112 E116 H129 T191 H55 H80 H82 E86 H99 T147 ? 0004089,0008270,0046872 Ki=315nM remove_due_to_license_issue A0A0M3KL20 28002963 303 ENGPHRWDKLHKDFEVCKSGKSQSPINIEHYYHTQDKADLQFKYAASKAVFFTHHTLKASFEPTNHINYRGHDYVLDNVHFHAPMEFLINNKTRPLSAHFVHLVLAIGFEEGKENPNLDPILNFKEVALDAFLPKSINYYHFNGSLTAPPCTEGVAWFVIEEPLEVSAKQLAEIKKRMKNSPNQRPVQPDYNTVIIKSSAE 5ttf A 1.72 BS06 7KZ A 1 D1083 L1086 D1088 F1158 D166 L169 D171 F237 Y1067 Y1154 Y150 Y233 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Kd=610nM, IC50=992nM Q96KQ7 28135087 1506 TEKIICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLDEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKSKYFTCQCGSEKCKHSAEAIALEQ 5ttg A 1.66 BS02 7KZ A 1 A1165 D1166 D1171 L1174 D1176 R1245 F1246 K1250 A160 D161 D166 L169 D171 R239 F240 K244 Y1155 Y1242 Y150 Y236 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 remove_due_to_license_issue Kd=46nM, IC50=7.0nM Q9H9B1 28135087 1302 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 5tts A 2.34 BS01 7KU A 1 A853 E903 L905 G908 C909 D912 L956 A40 E82 L84 G87 C88 D91 L135 D949 A951 R953 N954 D967 D128 A130 R132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 28139931 4000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 5ttu A 1.72 BS01 7KV A 1 L828 A853 M902 E903 L905 G908 C909 D912 L956 L14 A36 M79 E80 L82 G85 C86 D89 L133 D949 A951 R953 N954 D967 D126 A128 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 28139931 1201 TIFEERHLKYISQLGKGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 5ttv A 1.93 BS01 7KX A 1 L828 V836 A853 E903 Y904 L905 C909 D912 L956 L15 V23 A40 E87 Y88 L89 C93 D96 L140 D949 A951 R953 N954 D967 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 28139931 4000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 5tuo A 2.5 BS02 1SA A 1 H84 T86 H110 H112 L190 T191 A192 H61 T63 H87 H89 L167 T168 A169 H85 H110 H112 E116 H129 T191 H62 H87 H89 E93 H106 T168 4.2.1.1 0004089,0008270,0046872 Ki=323nM remove_due_to_license_issue A0A0M3KL20 28002963 303 TKWDYKNKENGPHRWDKLHKDFEVCKSGKSQSPINIEHYYHTQDLQFKYAASKPKAVFFTHHTLKASFEPTNHINYRGHDYVLDNVHFHAPMEFLINNKTRPLSAHFVHKDAKGRLLVLAIGFEEGKENPNLDPILEGIQKKQNFKEVALDAFLPKSINYYHFNGSLTAPPCTEGVAWFVIEEPLEVSAKQLAEIKKRMKNSPNQRPVQPDYNTVIIKSSAETR 5tuq A 2.705 BS01 J63 A 1 L100 K101 K103 V106 Y188 F227 W229 L234 H235 P236 Y318 L101 K102 K104 V107 Y189 F228 W230 L235 H236 P237 Y319 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28182989 601 VPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 5tur A 2.948 BS01 7LK A 1 F49 A65 I104 D131 L174 F16 A32 I68 D95 L138 D167 K169 N172 D186 L193 T204 D131 K133 N136 D150 L157 T168 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue IC50=900nM P11309 28947155 401 LESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNTRVPMEVVLLKKVSFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 5tuy A 2.6 BS06 7L6 A 1 D1074 A1077 D1078 R1080 D1083 L1086 D1088 R1157 F1158 D154 A157 D158 R160 D163 L166 D168 R237 F238 Y1067 Y1154 Y147 Y234 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue IC50=1.6nM, Kd=445nM Q96KQ7 28135087 1506 IICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLDNKDGEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKSKYFTCQCGSEKCKHSAEAIALEQS 5tuz A 1.95 BS06 7L6 A 1 A1165 D1166 R1168 D1171 L1174 D1176 R1245 F1246 I1249 A160 D161 R163 D166 L169 D171 R238 F239 I242 Y1155 Y1242 Y150 Y235 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 Kd=40nM remove_due_to_license_issue IC50=13nM, Kd=40nM Q9H9B1 28135087 3006 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 5tv1 A 2.4 BS01 IHP A 1 K227 R332 K220 R320 ? 0000822,0002029,0002031,0002092,0005547,0005634,0005737,0005886,0005905,0007165,0009968,0015031,0030139,0031410,0031623,0031701,0035091,0070374 Kd=90uM remove_due_to_license_issue P32120 29127291 401 RVFKKSSPNCKLTVYLGKRDFVDHLDKVDPVDGVVLVDPDYLKDRKVFVTLTCAFRYGREDLDVLGLSFRKDLFIANYQAFPPTPNPPRPPTRLQERLLRKLGQHAHPFFFTIPQNLPCSVTLQPGPEDTGKACGVDFEIRAFCAKSLEEKSHKRNSVRLVIRKVQFAPEKPGPQPSAETTRHFLMSDRSLHLEASLDKELYYHGEPLNVNVHVTNNSTKTVKKIKVSVRQYADICLFSTAQYKCPVAQVEQDDQVSPSSTFCKVYTITPLLSNNREKRGLALDGKLKHEDTNLASSTIVKEVLGILVSYRVKVKLVVSRGGDVSVELPFVLMHPKP 5tv1 A 2.4 BS02 IHP A 2 K233 R237 K251 K325 K327 K226 R230 K244 K313 K315 ? 0000822,0002029,0002031,0002092,0005547,0005634,0005737,0005886,0005905,0007165,0009968,0015031,0030139,0031410,0031623,0031701,0035091,0070374 Kd=90uM remove_due_to_license_issue P32120 29127291 402 RVFKKSSPNCKLTVYLGKRDFVDHLDKVDPVDGVVLVDPDYLKDRKVFVTLTCAFRYGREDLDVLGLSFRKDLFIANYQAFPPTPNPPRPPTRLQERLLRKLGQHAHPFFFTIPQNLPCSVTLQPGPEDTGKACGVDFEIRAFCAKSLEEKSHKRNSVRLVIRKVQFAPEKPGPQPSAETTRHFLMSDRSLHLEASLDKELYYHGEPLNVNVHVTNNSTKTVKKIKVSVRQYADICLFSTAQYKCPVAQVEQDDQVSPSSTFCKVYTITPLLSNNREKRGLALDGKLKHEDTNLASSTIVKEVLGILVSYRVKVKLVVSRGGDVSVELPFVLMHPKP 5tv3 A 2.9 BS02 7L3 A 1 K88 H110 H112 H129 L190 T191 K67 H89 H91 H108 L169 T170 H85 H110 H112 E116 H129 T191 H64 H89 H91 E95 H108 T170 4.2.1.1 0004089,0008270,0046872 remove_due_to_license_issue A0A0M3KL20 28002963 302 KWDYKNKENGPHRWDKLHKDFEVCKSGKSQSPINIEHYYHTQDKADLQFKYAASKPKAVFFTHHTLKASFEPTNHINYRGHDYVLDNVHFHAPMEFLINNKTRPLSAHFVHKDAKGRLLVLAIGFEEGKENPNLDPILEGIQKKQNFKEVALDAFLPKSINYYHFNGSLTAPPCTEGVAWFVIEEPLEVSAKQLAEIKKRMKNSPNQRPVQPDYNTVIIKSSAETR 5tvn A 2.9 BS01 7LD A 1 D135 F217 F340 D95 F174 F333 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41595 28129538 2001 EEMKQIVEEQGNKLHWAALLILMVIIPTIGGNTLVILAVSLEKKLQYATNYFLMSLAVADLLVGLFVMPIALLTIMFEAMWPLPLVLCPAWLFLDVLFSTASIWHLCAISVDRYIAIKKPIQANQYNSRATAFIKITVVWLISIGIAIPVPIKGIETNPNNITCVLTKERFGDFMLFGSLAAFFTPLAIMIVTYFLTIHALQKKAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLVQTISNEQRASKVLGIVFFLFLLMWCPFFITNITLVLCDSCNQTTLQMLLEIFVWIGYVSSGVNPLVYTLFNKTFRDAFGRYITCNYR 5tw2 A 1.75 BS02 7LP A 1 Y73 S76 F77 D80 L84 F120 W133 L150 D153 T156 Y67 S70 F71 D74 L78 F112 W125 L142 D145 T148 ? remove_due_to_license_issue P11609 28655912 305 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 5tw3 A 2.853 BS01 7N1 A 1 L100 K101 K102 K103 V106 V108 V179 Y181 Y188 G190 W229 L234 P236 Y318 L98 K99 K100 K101 V104 V106 V177 Y179 Y186 G188 W227 L232 P234 Y316 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28167742 601 SPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5tw5 A 1.85 BS01 7LM A 1 Y73 S76 D80 F120 W133 W142 L143 L150 D153 T156 Y67 S70 D74 F114 W127 W136 L137 L144 D147 T150 ? remove_due_to_license_issue P11609 28655912 306 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 5twj C 2.299 BS01 SAM C 1 L72 D73 I74 I102 G103 G107 L122 S123 L127 V132 L74 D75 I76 I104 G105 G109 L124 S125 L129 V134 2.1.1.177 0005515,0005737,0006364,0008168,0031167,0032259,0042803,0043022,0070038,0070475 Kd=5.58uM remove_due_to_license_issue P0A8I8 28428565 201 HHVKLQLVAVGTKMPDWVQTGFTEYLRRFPKDMPFELIEIPAGKRGKNADIKRILDKEGEQMLAAAGKNRIVTLDIPGKPWDTPQLAAELERWKLDGRDVSLLIGGPEGLSPACKAAAEQSWSLSALTLPHPLVRVLVAESLYRAWSITTNHPYHRE 5twj D 2.299 BS01 SAM D 1 L72 D73 I74 G103 G107 L122 L127 V132 L74 D75 I76 G105 G109 L124 L129 V134 2.1.1.177 0005515,0005737,0006364,0008168,0031167,0032259,0042803,0043022,0070038,0070475 Kd=5.58uM remove_due_to_license_issue P0A8I8 28428565 201 HHVKLQLVAVGTKMPDWVQTGFTEYLRRFPKDMPFELIEIPAGKRGKNADIKRILDKEGEQMLAAAGKNRIVTLDIPGKPWDTPQLAAELERWKLDGRDVSLLIGGPEGLSPACKAAAEQSWSLSALTLPHPLVRVLVAESLYRAWSITTNHPYHRE 5twl A 2.42 BS01 H91 A 1 I17 K40 E57 C70 L86 E87 C89 E93 E136 L139 I149 D150 I18 K41 E58 C71 L87 E88 C90 E94 E137 L140 I150 D151 D132 K134 E136 N137 D150 S171 D133 K135 E137 N138 D151 S157 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=10.5nM remove_due_to_license_issue Q14680 28926338 4000 GSKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 5two A 1.927 BS02 7MV A 1 F282 G284 C285 R288 S289 Y327 L330 I341 F363 M364 H449 L469 Y473 F76 G78 C79 R82 S83 Y121 L124 I135 F157 M158 H243 L263 Y267 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 28128331 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 5twx A 2.55 BS01 7P7 A 1 F160 F161 V165 I169 N216 R217 Y222 F24 F25 V29 I33 N80 R81 Y86 ? remove_due_to_license_issue Q9H8M2 28418626 4000 ESTPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKQAALLGNEDTA 5tx3 A 2.9 BS01 7MY A 1 V25 K40 Y88 C89 E93 L139 I149 V25 K40 Y80 C81 E85 L131 I141 D132 K134 E136 N137 D150 S171 D124 K126 E128 N129 D142 S147 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 28926338 1000 SGSMKDYDELLKYYELHETIGTAKVKLACHILTGEMVAIKIMDKNIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLGSLAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 5tx3 A 2.9 BS02 7MY B 1 E15 T16 E18 T19 D132 K134 E136 N137 D150 S171 D124 K126 E128 N129 D142 S147 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q14680 28926338 1001 SGSMKDYDELLKYYELHETIGTAKVKLACHILTGEMVAIKIMDKNIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLGSLAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 5tx5 A 2.56 BS01 7MJ A 1 V31 K45 M67 V76 L90 M92 H136 A155 D156 L157 L159 F162 V20 K34 M56 V65 L79 M81 H125 A144 D145 L146 L148 F151 D138 K140 E142 N143 D156 T189 D127 K129 E131 N132 D145 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13546 28151659 301 IKMKSSDFLESAELDSGGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 5txy A 1.206 BS02 7Q1 A 1 H94 H119 L197 T198 T199 W208 H90 H115 L193 T194 T195 W204 H64 H94 H96 E106 H119 T198 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.5uM remove_due_to_license_issue Kd=2600nM P00918 28817930 303 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ty1 A 1.6 BS02 7QV A 1 H94 H119 V121 F131 L198 T199 T200 W209 H92 H117 V119 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.5uM remove_due_to_license_issue Kd=3600nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ty8 A 1.45 BS02 7Q1 A 1 H94 H119 L198 T199 T200 W209 H92 H117 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.5uM remove_due_to_license_issue Kd=2600nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ty9 A 1.53 BS02 7QV A 1 H94 V121 F131 L198 T199 T200 W209 H92 V119 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=6.1uM remove_due_to_license_issue Kd=3600nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5tya A 1.5 BS02 7QS A 1 H94 H119 L198 T199 T200 W209 H92 H117 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=32.9uM remove_due_to_license_issue Kd=32900nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5tyh A 2.1 BS01 7O4 A 1 N118 S136 V137 F152 G154 I155 G173 N108 S126 V127 F142 G144 I145 G163 2.3.1.203 0006486,0016746,0016747,0018279 ic50=8.4mM remove_due_to_license_issue Q0P9D1 28182413 201 ARTEKIYIYGHGLVCEDVAKNMGYKECIFLDFESTLPKYDFFIAIGNNEIRKKIYQKISENGFKIVNLIHKSALISPSAIVEENAGILIMPYVVINAKAKIEKGVILNTSSVIEHECVIGEFSHVSVGAKCAGNVKIGKNCFLGINSCVLPNLSLADDSILGGGATLVKNQDEKGVFVGVPAKRM 5tyh A 2.1 BS02 7O4 A 2 I85 S86 N106 I75 S76 N96 2.3.1.203 0006486,0016746,0016747,0018279 ic50=8.4mM remove_due_to_license_issue Q0P9D1 28182413 202 ARTEKIYIYGHGLVCEDVAKNMGYKECIFLDFESTLPKYDFFIAIGNNEIRKKIYQKISENGFKIVNLIHKSALISPSAIVEENAGILIMPYVVINAKAKIEKGVILNTSSVIEHECVIGEFSHVSVGAKCAGNVKIGKNCFLGINSCVLPNLSLADDSILGGGATLVKNQDEKGVFVGVPAKRM 5tyj A 1.75 BS01 7ND A 1 G136 D137 S218 A219 W251 F354 Y420 G132 D133 S214 A215 W247 F350 Y416 G136 D137 S218 A219 E351 H471 G132 D133 S214 A215 E347 H467 3.1.1.- 0052689 remove_due_to_license_issue Q25252 31575743 601 VSLMEKLKWKIKCIENKFLNYRLTTNETVVAETEYGKVKGVKRLTVYDDSYYSFEGIPYAQPPVGELRFKAPQRPTPWAGVRDCCNHKDKSVQVDFITGKVCGSEDCLYLSVYTNNLNPETKRPVLVYIHGGDFIIGENHRDMYGPDYFIKKDVVLINIQYRLGALGFLSLNSEDLNVPGNAGLKDQVMALRWIKNNCANFGGNPDNITVFGESAGAASTHYMMLTEQTRGLFHRGILMSGNAICPWANTQCQHRAFTLAKLAGYKGEDNDKDVLEFLMKAKPQDLIKLEEKVLTLEERTNKVMFPFGPTVEPYQTADCVLPKHPREMVKTAWGNSIPTMMGNTSYEGLFFTSILKQMPLLVKELETCVNFVPSELADAERTAPETLEMGAKIKKAHVTGETPTADNFMDLCSHFYFWFPMHRLLQLRFNHTSGTPVYLYRFDFDSEDLINPYRIMRSGRGVKGVSHTDELTYFFWNQLAKRMPKESREYKTIERMTGIWTQFATTGNPYSNEIEGMENVSWDPIEKSDEVYKCLNISDELKMIDVPEMGKIKQWESMFEKHRDLF 5tyk A 1.65 BS01 7N4 A 1 G136 G137 S218 A219 M308 F309 F354 F355 M460 G132 G133 S214 A215 M304 F305 F350 F351 M456 G136 G137 G168 S218 A219 F309 F311 E351 H471 G132 G133 G164 S214 A215 F305 F307 E347 H467 3.1.1.- 0052689 remove_due_to_license_issue Q25252 31575743 601 VSLMEKLKWKIKCIENKFLNYRLTTNETVVAETEYGKVKGVKRLTVYDDSYYSFEGIPYAQPPVGELRFKAPQRPTPWAGVRDCCNHKDKSVQVDFITGKVCGSEDCLYLSVYTNNLNPETKRPVLVYIHGGGFIIGENHRDMYGPDYFIKKDVVLINIQYRLGALGFLSLNSEDLNVPGNAGLKDQVMALRWIKNNCANFGGNPDNITVFGESAGAASTHYMMLTEQTRGLFHRGILMSGNAICPWANTQCQHRAFTLAKLAGYKGEDNDKDVLEFLMKAKPQDLIKLEEKVLTLEERTNKVMFPFGPTVEPYQTADCVLPKHPREMVKTAWGNSIPTMMGNTSYEGLFFTSILKQMPLLVKELETCVNFVPSELADAERTAPETLEMGAKIKKAHVTGETPTADNFMDLCSHFYFWFPMHRLLQLRFNHTSGTPVYLYRFDFDSEDLINPYRIMRSGRGVKGVSHTDELTYFFWNQLAKRMPKESREYKTIERMTGIWTQFATTGNPYSNEIEGMENVSWDPIEKSDEVYKCLNISDELKMIDVPEMGKIKQWESMFEKHRDLF 5tyl A 1.75 BS01 7N7 A 1 G136 G137 S218 A219 W251 M308 F355 Y420 H471 G132 G133 S214 A215 W247 M304 F351 Y416 H467 G136 G137 G168 S218 A219 F309 F311 E351 H471 G132 G133 G164 S214 A215 F305 F307 E347 H467 3.1.1.- 0052689 remove_due_to_license_issue Q25252 31575743 601 VSLMEKLKWKIKCIENKFLNYRLTTNETVVAETEYGKVKGVKRLTVYDDSYYSFEGIPYAQPPVGELRFKAPQRPTPWAGVRDCCNHKDKSVQVDFITGKVCGSEDCLYLSVYTNNLNPETKRPVLVYIHGGGFIIGENHRDMYGPDYFIKKDVVLINIQYRLGALGFLSLNSEDLNVPGNAGLKDQVMALRWIKNNCANFGGNPDNITVFGESAGAASTHYMMLTEQTRGLFHRGILMSGNAICPWANTQCQHRAFTLAKLAGYKGEDNDKDVLEFLMKAKPQDLIKLEEKVLTLEERTNKVMFPFGPTVEPYQTADCVLPKHPREMVKTAWGNSIPTMMGNTSYEGLFFTSILKQMPLLVKELETCVNFVPSELADAERTAPETLEMGAKIKKAHVTGETPTADNFMDLCSHFYFWFPMHRLLQLRFNHTSGTPVYLYRFDFDSEDLINPYRIMRSGRGVKGVSHTDELTYFFWNQLAKRMPKESREYKTIERMTGIWTQFATTGNPYSNEIEGMENVSWDPIEKSDEVYKCLNISDELKMIDVPEMGKIKQWESMFEKHRDLF 5tyn A 1.531 BS01 7NS A 1 G135 G136 G137 S218 A219 W251 M308 F309 F354 G133 G134 G135 S216 A217 W249 M306 F307 F352 G136 G137 G168 S218 A219 F309 F311 E351 H471 G134 G135 G166 S216 A217 F307 F309 E349 H469 3.1.1.- 0052689 remove_due_to_license_issue Q25252 31575743 601 FNVSLMEKLKWKIKCIENKFLNYRLTTNETVVAETEYGKVKGVKRLTVYDDSYYSFEGIPYAQPPVGELRFKAPQRPTPWAGVRDCCNHKDKSVQVDFITGKVCGSEDCLYLSVYTNNLNPETKRPVLVYIHGGGFIIGENHRDMYGPDYFIKKDVVLINIQYRLGALGFLSLNSEDLNVPGNAGLKDQVMALRWIKNNCANFGGNPDNITVFGESAGAASTHYMMLTEQTRGLFHRGILMSGNAICPWANTQCQHRAFTLAKLAGYKGEDNDKDVLEFLMKAKPQDLIKLEEKVLTLEERTNKVMFPFGPTVEPYQTADCVLPKHPREMVKTAWGNSIPTMMGNTSYEGLFFTSILKQMPLLVKELETCVNFVPSELADAERTAPETLEMGAKIKKAHVTGETPTADNFMDLCSHFYFWFPMHRLLQLRFNHTSGTPVYLYRFDFDSEDLINPYRIMRSGRGVKGVSHTDELTYFFWNQLAKRMPKESREYKTIERMTGIWTQFATTGNPYSNEIEGMENVSWDPIEKSDEVYKCLNISDELKMIDVPEMGKIKQWESMFEKHRDLF 5tyo A 1.57 BS01 7NM A 1 G136 G137 I140 S218 A219 M308 F354 H471 G132 G133 I136 S214 A215 M304 F350 H467 G136 G137 G168 S218 A219 F309 F311 E351 H471 G132 G133 G164 S214 A215 F305 F307 E347 H467 3.1.1.- 0052689 remove_due_to_license_issue Q25252 31575743 601 VSLMEKLKWKIKCIENKFLNYRLTTNETVVAETEYGKVKGVKRLTVYDDSYYSFEGIPYAQPPVGELRFKAPQRPTPWAGVRDCCNHKDKSVQVDFITGKVCGSEDCLYLSVYTNNLNPETKRPVLVYIHGGGFIIGENHRDMYGPDYFIKKDVVLINIQYRLGALGFLSLNSEDLNVPGNAGLKDQVMALRWIKNNCANFGGNPDNITVFGESAGAASTHYMMLTEQTRGLFHRGILMSGNAICPWANTQCQHRAFTLAKLAGYKGEDNDKDVLEFLMKAKPQDLIKLEEKVLTLEERTNKVMFPFGPTVEPYQTADCVLPKHPREMVKTAWGNSIPTMMGNTSYEGLFFTSILKQMPLLVKELETCVNFVPSELADAERTAPETLEMGAKIKKAHVTGETPTADNFMDLCSHFYFWFPMHRLLQLRFNHTSGTPVYLYRFDFDSEDLINPYRIMRSGRGVKGVSHTDELTYFFWNQLAKRMPKESREYKTIERMTGIWTQFATTGNPYSNEIEGMENVSWDPIEKSDEVYKCLNISDELKMIDVPEMGKIKQWESMFEKHRDLF 5typ A 1.88 BS01 7NJ A 1 G137 S218 A219 W251 M308 Y420 F421 H471 G133 S214 A215 W247 M304 Y416 F417 H467 G136 G137 G168 S218 A219 F309 F311 E351 H471 G132 G133 G164 S214 A215 F305 F307 E347 H467 3.1.1.- 0052689 remove_due_to_license_issue Q25252 31575743 601 VSLMEKLKWKIKCIENKFLNYRLTTNETVVAETEYGKVKGVKRLTVYDDSYYSFEGIPYAQPPVGELRFKAPQRPTPWAGVRDCCNHKDKSVQVDFITGKVCGSEDCLYLSVYTNNLNPETKRPVLVYIHGGGFIIGENHRDMYGPDYFIKKDVVLINIQYRLGALGFLSLNSEDLNVPGNAGLKDQVMALRWIKNNCANFGGNPDNITVFGESAGAASTHYMMLTEQTRGLFHRGILMSGNAICPWANTQCQHRAFTLAKLAGYKGEDNDKDVLEFLMKAKPQDLIKLEEKVLTLEERTNKVMFPFGPTVEPYQTADCVLPKHPREMVKTAWGNSIPTMMGNTSYEGLFFTSILKQMPLLVKELETCVNFVPSELADAERTAPETLEMGAKIKKAHVTGETPTADNFMDLCSHFYFWFPMHRLLQLRFNHTSGTPVYLYRFDFDSEDLINPYRIMRSGRGVKGVSHTDELTYFFWNQLAKRMPKESREYKTIERMTGIWTQFATTGNPYSNEIEGMENVSWDPIEKSDEVYKCLNISDELKMIDVPEMGKIKQWESMFEKHRDLF 5tyr A 1.8 BS01 7O7 A 1 D25 G27 A28 D30 G48 P81 V82 D25 G27 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.26nM remove_due_to_license_issue G0X8E8 29039736 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5tyr B 1.8 BS01 7O7 A 1 D25 G27 D29 D30 I47 G48 G49 I50 I84 D25 G27 D29 D30 I47 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue G0X8E8 29039736 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5tys A 2.007 BS01 7OA A 1 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 G27 A28 D29 D30 G48 G49 I50 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 ic50=0.019nM remove_due_to_license_issue G0X8E8 29039736 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5tys B 2.007 BS01 7OA A 1 D25 G27 A28 D30 G48 P81 V82 D25 G27 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue G0X8E8 29039736 400 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 5tz3 A 1.72 BS01 7OM A 1 L809 I826 F830 M847 L858 Q859 F862 L234 I251 F255 M272 L283 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.14uM remove_due_to_license_issue O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5tza A 1.7 BS01 7OG A 1 L770 L809 Q812 I826 M847 L858 Q859 F862 L195 L234 Q237 I251 M272 L283 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.001uM remove_due_to_license_issue IC50=1nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5tzc A 2.36 BS01 7OJ A 1 H656 L809 I826 F830 M847 Q859 F862 H81 L234 I251 F255 M272 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.008uM remove_due_to_license_issue IC50=8.0nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLDE 5tzd J 1.749 BS01 C2E J 1 K84 R114 S123 R125 Q126 K1 R31 S40 R42 Q43 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 201 KLVLDLERMAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzd J 1.749 BS02 C2E J 2 I110 Q113 R114 R125 D128 I27 Q30 R31 R42 D45 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 202 KLVLDLERMAHVPQEKAGPLQRYAATIQSQRGDYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzf B 2.4 BS01 C2E B 1 I110 Q113 R114 R125 D128 I28 Q31 R32 R43 D46 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 201 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGAYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzf B 2.4 BS02 C2E B 2 R114 S123 R125 Q126 R32 S41 R43 Q44 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 202 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGAYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzg A 2.5 BS01 C2E C 1 R114 S123 R125 Q126 R31 S40 R42 Q43 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 203 KLVLDLERLAHVPQEKAGPLQRYAATIQSQRGAYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzg A 2.5 BS02 C2E C 2 I110 Q113 R114 R125 D128 I27 Q30 R31 R42 D45 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 204 KLVLDLERLAHVPQEKAGPLQRYAATIQSQRGAYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzg C 2.5 BS01 C2E C 1 I110 Q113 R114 R125 D128 I28 Q31 R32 R43 D46 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 203 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGAYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzg C 2.5 BS02 C2E C 2 R114 S123 R125 Q126 R32 S41 R43 Q44 ? 0045892 remove_due_to_license_issue F2RCL8 28449057 204 PKLVLDLERLAHVPQEKAGPLQRYAATIQSQRGAYNGKVLSIRQDDLRTLAVIYDQSPSVLTEQLISWGVLDADAR 5tzh A 1.6 BS01 7OP A 1 H656 L770 Q812 I826 F830 M847 Q859 F862 I866 H81 L195 Q237 I251 F255 M272 Q284 F287 I291 3.1.4.17 0004114,0007165,0008081 ic50=0.679uM remove_due_to_license_issue IC50=679nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5tzo A 1.67 BS01 7V7 A 1 W63 W90 T91 Q127 W129 W63 W90 T91 Q127 W129 S35 V69 A78 Y80 A172 S35 V69 A78 Y80 A172 3.2.1.8 0004553,0005975,0016798,0031176,0045493 Kd=5.9uM remove_due_to_license_issue P18429 28925919 201 MSTDYWLNFTDGGGIVNAVNGSGGNYSVNWSNTGSFVVGKGWTTGSPFRTINYNAGVWAPNGWGALALVGWTRSPLIAYYVVDSWGTARWTGTYKGTVKSDGGTYDIYTTTRYNAPSIDGDRTTFTQYWSVRQSKRPTGSNATITFSNHVNAWKSHGMNLGSNWAYQVMATAGYQSSGSSNVTVW 5tzo A 1.67 BS02 7V7 A 2 F9 S35 F36 V37 W63 A65 P116 S117 W129 Y166 A172 G173 Y174 F9 S35 F36 V37 W63 A65 P116 S117 W129 Y166 A172 G173 Y174 S35 V69 A78 Y80 A172 S35 V69 A78 Y80 A172 3.2.1.8 0004553,0005975,0016798,0031176,0045493 Kd=5.9uM remove_due_to_license_issue P18429 28925919 202 MSTDYWLNFTDGGGIVNAVNGSGGNYSVNWSNTGSFVVGKGWTTGSPFRTINYNAGVWAPNGWGALALVGWTRSPLIAYYVVDSWGTARWTGTYKGTVKSDGGTYDIYTTTRYNAPSIDGDRTTFTQYWSVRQSKRPTGSNATITFSNHVNAWKSHGMNLGSNWAYQVMATAGYQSSGSSNVTVW 5tzw A 1.59 BS01 7P4 A 1 H656 L770 Q812 I826 F830 M847 Q859 F862 I866 H81 L195 Q237 I251 F255 M272 Q284 F287 I291 3.1.4.17 0004114,0007165,0008081 ic50=0.987uM remove_due_to_license_issue IC50=987nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 5tzx A 1.9 BS01 7OY A 1 H656 L770 L809 Q812 I826 Y827 F830 M847 Q859 F862 H81 L195 L234 Q237 I251 Y252 F255 M272 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.052uM remove_due_to_license_issue IC50=52nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 5tzz A 1.6 BS01 7OJ A 1 H656 L770 L809 I826 Y827 F830 M847 Q859 F862 H81 L195 L234 I251 Y252 F255 M272 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.014uM remove_due_to_license_issue IC50=8.0nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 5u00 A 1.41 BS01 7OV A 1 H656 L770 L809 Q812 I826 Y827 F830 M847 Q859 F862 H81 L195 L234 Q237 I251 Y252 F255 M272 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.002uM remove_due_to_license_issue IC50=2nM O00408 28165743 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5u0d A 1.59 BS02 7R7 A 1 H94 H119 V121 F131 L198 T199 T200 W209 H92 H117 V119 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=28.6uM remove_due_to_license_issue Kd=28600nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5u0e A 1.27 BS02 7R4 A 1 H94 H96 H119 F131 L198 T199 T200 W209 H92 H94 H117 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=7.7uM remove_due_to_license_issue Kd=7700nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5u0f A 1.21 BS02 7R1 A 1 H94 H96 H119 F131 L198 T199 T200 W209 H92 H94 H117 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=3.4uM remove_due_to_license_issue Kd=2300nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5u0g A 1.54 BS02 7QY A 1 H94 H96 H119 F131 L198 T199 T200 W209 H92 H94 H117 F128 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Kd=16000nM P00918 28817930 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5u0w A 1.968 BS01 9MG A 1 D96 N115 M139 D185 F190 G217 K221 R255 D86 N105 M129 D175 F180 G207 K211 R245 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKERYE 5u0y A 1.88 BS01 7PJ A 1 T62 N115 M139 D185 F190 G217 K221 R255 T53 N106 M130 D176 F181 G208 K212 R246 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTPNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKENKRYE 5u0z A 2.29 BS01 7PM A 1 T62 N115 I117 M139 D185 F190 G217 K221 R255 T52 N105 I107 M129 D175 F180 G207 K211 R245 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKENKRYE 5u11 A 1.994 BS01 7PS A 1 N115 M139 D185 F190 G217 K221 R255 N106 M130 D176 F181 G208 K212 R246 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTPNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKENKRYE 5u12 A 1.839 BS01 5RU A 1 T62 N115 M139 D185 F190 G217 K221 R255 T53 N106 M130 D167 F172 G199 K203 R237 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue Kd=8500nM P0AC13 29171692 301 SMKLFAQGTSLDLSHPHVMGILNVTNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKENKRYE 5u13 A 1.951 BS01 YH5 A 1 N115 M139 D185 F190 G217 R220 K221 R255 N105 M129 D175 F180 G207 R210 K211 R245 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue Kd=3900nM P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKENKRYE 5u14 A 1.953 BS01 7PV A 1 T62 R63 P64 N115 I117 M139 D185 F190 G217 K221 S222 R255 T53 R54 P55 N106 I108 M130 D176 F181 G208 K212 S213 R246 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTPNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAKENKRYE 5u1j A 2.95 BS01 dna W 0 R52 K270 R51 K258 ? 0046872 remove_due_to_license_issue O93708 28373206 4 ~ 24 IAKVITIHNFKGGVGKTTTTAIIAMGLGAMGKRVLLIDFDAQMSLTQIFVREEDRLKILESSHDQDKSAFALLRTMEPARIKFFHEGKGVKFGIDVIPGSYMSIFKLMFEIQSEWNILRMLDLYRDQYDYILIDTAPSDTVTIKPILRASHYLLIPEDGTPEAFTAMRIFLNEALPKYILPRPEGGFYKYPRILGVILTRVRRNSTAILMKHNKILEEELSNSELKDHVIYPPYFGADKDNPEDYILSLSDLIWRDEKRAPISEVFDKLFSKVFTEIPKEVVRRVENDQ 5u1j B 2.95 BS01 dna W 0 K85 F87 K270 K81 F83 K257 ? 0046872 remove_due_to_license_issue O93708 28373206 4 ~ 24 IAKVITIHNFKGGVGKTTTTAIIAMGLGAMGKRVLLIDFDAQMSLTQIFVREEDRLKILESSHQDKSAFALLRTMEPARIKFFHEGKGVKFGIDVIPGSYMSIFKLMFEIQSEWNILRMLDLYRDQYDYILIDTAPSDTVTIKPILRASHYLLIPEDGTPEAFTAMRIFLNEALPKYILPRPEGGFYKYPRILGVILTRVRRNSTAILMKHNKILEEELSNSELKDHVIYPPYFGADKDNPEDYILSSSDLIWRDEKRAPISEVFDKLFAFFSKVFTEIPKEVVRRVENDQ 5u28 A 1.798 BS01 82V A 1 W81 P82 Q85 V87 L92 L94 N140 I146 W39 P40 Q43 V45 L50 L52 N98 I104 ? remove_due_to_license_issue O60885 28137841 201 ANPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEETEIMIVQA 5u2c A 3.3 BS01 82Y A 1 W374 P375 V380 L385 N433 H437 W36 P37 V42 L47 N95 H99 ? remove_due_to_license_issue O60885 28137841 501 GILPAPEKSSKVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMP 5u2e A 1.991 BS01 837 A 1 W81 P82 V87 N140 I146 W40 P41 V46 N99 I105 ? remove_due_to_license_issue O60885 28137841 201 STNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEETEIM 5u2f A 2.525 BS01 82Y A 1 P82 V87 L94 N140 I146 P40 V45 L52 N98 I104 ? remove_due_to_license_issue O60885 28137841 201 TNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEETEIMI 5u3b A 2.0 BS02 7TD A 1 E77 T190 F191 I197 G209 S210 V216 H237 D241 H264 E77 T188 F189 I195 G207 S208 V214 H235 D239 H262 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=1.5nM remove_due_to_license_issue IC50=0.001000nM P47205 28549219 502 MIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 5u48 A 1.5 BS01 S4B A 1 K15 L17 S117 K6 L8 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=470nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u48 B 1.5 BS01 S4B B 1 K15 L110 S117 K6 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=470nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4a A 1.9 BS01 7VG A 1 K15 L17 S117 K6 L8 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=440nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4a B 1.9 BS01 7VG B 1 K15 A108 L110 S117 K6 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=440nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4b A 1.448 BS01 XOS A 1 K15 L110 S117 K6 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=1800nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4b B 1.448 BS01 XOS B 1 K15 L110 S117 K6 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=1800nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4c A 1.7 BS01 XBS A 1 K15 L17 L110 K6 L8 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=990nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4c B 1.7 BS01 XBS B 1 L110 S117 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=990nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4d A 1.55 BS01 XLO A 1 K15 A108 L110 K6 A99 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=470nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4d B 1.55 BS01 XLO B 1 K15 L17 S117 K6 L8 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=470nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4e A 1.45 BS01 XLB A 1 K15 L17 L110 S117 K6 L8 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=450nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4e B 1.45 BS01 XLB B 1 K15 L110 S117 K6 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=450nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4f A 1.5 BS01 IWW A 1 L17 L110 S117 L8 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=470nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4f B 1.5 BS01 IWW B 1 K15 L17 L110 S117 K6 L8 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue Kd=470nM P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4g A 1.8 BS01 7UV A 1 L110 S117 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 5u4g B 1.8 BS01 7UV B 1 K15 L17 L110 S117 K6 L8 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 remove_due_to_license_issue P02766 28920684 200 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTN 5u4x A 1.88 BS02 7VM A 1 Y150 F153 Y154 M163 E258 M260 Y262 N266 E267 H415 Q447 K471 P473 F475 Y4 F7 Y8 M17 E112 M114 Y116 N120 E121 H269 Q301 K325 P327 F329 D166 E258 E267 H415 D20 E112 E121 H269 2.1.1.319 0016274,0018216 remove_due_to_license_issue Q86X55 29719619 502 AVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRY 5u51 A 2.8 BS01 G4P A 1 Y11 I52 R64 L65 N100 K101 Q105 Y14 I55 R67 L68 N103 K104 Q108 ? remove_due_to_license_issue Q5NFG1 28864445 301 SNAMLLYTKKDDIYSDIVRMILLIKGANAKIVDVSKEENSKHLEELNIITPNGNIPTLSTDDFAVYRLSVIIEAIEDLYPFPPMFPVFPKQRANARILLEYVNKTFLQNIIKLQSPDLDEKQANEIKMLMQRDIISTYKKIVSEREVNAESNPDAQNINVLTLIITFVFYYFIKLKISIPTKDKNIIKEIKELLSEPNFIKTI 5u5h A 1.8 BS01 7VV A 1 F97 Y148 N194 E238 L240 D310 Y365 R367 R414 F19 Y70 N116 E160 L162 D232 Y287 R289 R329 ? ic50=1.3uM remove_due_to_license_issue IC50=1300nM O75530 27992714 501 KYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5u5k A 2.33 BS01 7VY A 1 F97 Y148 Y365 R367 R414 F19 Y70 Y287 R289 R332 ? ic50=95uM remove_due_to_license_issue IC50=95000nM, Kd=32000nM O75530 27992714 502 KYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5u5l A 2.55 BS01 7VA A 1 I281 F282 C285 S289 H323 Y327 I341 M348 M364 Y473 I64 F65 C68 S72 H106 Y110 I124 M131 M147 Y256 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=43nM P37231 28499821 501 NPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 5u5t A 1.6 BS02 7W7 A 1 F97 Y148 N194 D310 Y365 R367 F19 Y70 N116 D224 Y279 R281 ? ic50=3.9uM remove_due_to_license_issue IC50=1600nM O75530 27992714 501 KYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVECTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5u62 A 1.9 BS02 7WD A 1 F97 Y148 D310 Y365 R367 F19 Y70 D226 Y281 R283 ? ic50=1.3uM remove_due_to_license_issue IC50=1300nM O75530 27992714 504 KYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRL 5u69 A 1.28 BS01 LQD A 1 F97 Y148 E238 L240 D310 Y365 R367 R414 F16 Y67 E157 L159 D229 Y284 R286 R333 ? Ki=600nM remove_due_to_license_issue Ki=600nM, Kd=38000nM O75530 28254486 501 FKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDR 5u6b A 2.84 BS01 7YS A 1 L542 V550 A565 M598 L620 P621 M623 G626 D627 N677 M679 A689 L22 V30 A45 M78 L93 P94 M96 G99 D100 N150 M152 A162 D672 A674 R676 N677 D690 D145 A147 R149 N150 D163 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P30530 28724631 9001 ELKEKLRDVMVDRHKVALGKTLGEGEFGAVMEGQLNQDDSILKVAVKTMKIAICTRSELEDFLSEAVCMKEFDHPNVMRLIGVCFQPAPVVILPFMKHGDLHSFLLYSRLGDQPVYLPTQMLVKFMADIASGMEYLSTKRFIHRDLAARNCMLNENMSVCVADFGLSKPVKWIAIESLADRVYTSKSDVWSFGVTMWEIATRGQTPYPGVENSEIYDYLRQGNRLKQPADCLDGLYALMSRCWELNPQDRPSFTELREDLENTLKALPPA 5u6c A 2.1 BS01 7YS A 1 L593 V601 A617 M650 L671 F673 M674 G677 D678 N728 M730 A740 L22 V30 A46 M79 L96 F98 M99 G102 D103 N153 M155 A165 D723 A725 R727 N728 D741 D148 A150 R152 N153 D166 2.7.10.1 0004672,0004713,0005524,0006468,0016627,0050660 Ki<0.05nM remove_due_to_license_issue Q12866 28724631 9001 ELQNKLEDVVIDRNLLILGKILGEGEFGSVMEGNLKQEDGTSLKVAVKTMKLDNSSQREIEEFLSEAACMKDFSHPNVMRLLGVCIEMIPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFGLSPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESLPDV 5u6c B 2.1 BS01 7YS B 1 L593 V601 A617 M650 F673 M674 D678 N728 M730 A740 L19 V24 A40 M64 F87 M88 D92 N142 M144 A154 D723 A725 R727 N728 D741 M762 D137 A139 R141 N142 D155 M157 2.7.10.1 0004672,0004713,0005524,0006468,0016627,0050660 Ki<0.05nM remove_due_to_license_issue Q12866 28724631 9001 NKLEDVVIDRNLLILGKILGEGSVMEGNLKQEDGTSLKVAVKTMIEEFLSEAACMKDFSHPNVMRLLGVCIEMSSQGIPKPMVILPFMKYGDLHTYLLYSRLETGPKHIPLQTLLKFMVDIALGMEYLSNRNFLHRDLAARNCMLRDDMTVCVADFMPVKWIAIESLADRVYTSKSDVWAFGVTMWEIATRGMTPYPGVQNHEMYDYLLHGHRLKQPEDCLDELYEIMYSCWRTDPLDRPTFSVLRLQLEKLLESLP 5u6d A 1.64 BS01 7XG A 1 P95 F97 Y148 E238 L240 D310 Y365 R367 P14 F16 Y67 E157 L159 D229 Y284 R286 ? Ki=2.6nM remove_due_to_license_issue Ki=2.6nM O75530 28254486 501 FKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDR 5u6j H 2.3 BS01 82J H 1 H57 G97 C191 K192 S195 S214 W215 G216 G219 H41 G85 C185 K186 S189 S208 W209 G210 G212 3.4.21.21 0004252,0006508 Ki=23nM remove_due_to_license_issue Ki=610nM P08709 28460818 301 IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP 5u6v A 1.775 BS01 7WY A 1 W370 P371 F372 V376 H433 V435 W24 P25 F26 V30 H87 V89 ? ic50=21nM remove_due_to_license_issue Kd=0.130000nM, IC50=21nM P25440 29259751 501 SEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 5u7d A 1.75 BS01 19F A 1 H656 T768 L770 H773 L809 I826 Y827 M847 L858 Q859 F862 I866 H78 T190 L192 H195 L231 I248 Y249 M269 L280 Q281 F284 I288 3.1.4.17 0004114,0007165,0008081 ic50=0.5nM remove_due_to_license_issue IC50=4.7nM O00408 28574706 1001 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5u7i A 2.0 BS01 7XS A 1 Y655 H656 Q812 I826 Q859 F862 I866 Y77 H78 Q234 I248 Q281 F284 I288 3.1.4.17 0004114,0007165,0008081 ic50=66.6nM remove_due_to_license_issue IC50=67nM O00408 28574706 1001 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5u7j A 1.9 BS01 7XV A 1 H656 L770 I826 F830 M847 Q859 F862 I866 H78 L192 I248 F252 M269 Q281 F284 I288 3.1.4.17 0004114,0007165,0008081 ic50=389.6nM remove_due_to_license_issue IC50=390nM O00408 28574706 1001 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5u7k A 2.06 BS02 7Y1 A 1 L770 T805 D808 L809 I826 F830 Q859 F862 L194 T229 D232 L233 I250 F254 Q283 F286 3.1.4.17 0004114,0007165,0008081 ic50=7.1nM remove_due_to_license_issue IC50=7.1nM O00408 28574706 1003 AMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5u7l A 2.38 BS01 7Y4 A 1 L770 D808 L809 Q812 I826 F830 M847 Q859 F862 L192 D230 L231 Q234 I248 F252 M269 Q281 F284 3.1.4.17 0004114,0007165,0008081 ic50=4.9nM remove_due_to_license_issue IC50=<5.84nM O00408 28574706 1001 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 5u7m G 3.025 BS02 83G G 1 W112 D113 L116 S375 F376 I424 N425 M426 W427 M475 W79 D80 L83 S324 F325 I361 N362 M363 W364 M412 ? 0019031 remove_due_to_license_issue Q2N0S5 28825711 657 AENLWVTVYYGVPVWKDAETTLFCASDAKAYKHNVWATHACVPTDPNPQEIHLENVTEEFNMWKNNMVEQMHTDIISLWDQSLKPCVKLTPLCVTLQCTNVTNNRGELKNCSFNMTTELRDKKQKVYSLFYRLDVVQINEYRLINCNTSAITQACPKVSFEPIPIHYCAPAGFAILKCKDKKFNGTGPCPSVSTVQCTHGIKPVVSTQLLLNGSLAEEEVMIRSENITNNAKNILVQFNTPVQINCTRPNNNTRKSIRIGPGQAFYATGDIIGDIRQAHCNVSKATWNETLGKVVKQLRKHFGNNTIIRFANSSGGDLEVTTHSFNCGGEFFYCNTSGLFNSTWISNNDSITLPCRIKQIINMWQRIGQAMYAPPIQGVIRCVSNITGLILTRDGGSTNSTTETFRPGGGDMRDNWRSELYKYKVVKIEPLGVAPTRCKRRV 5u7o G 3.031 BS01 83J G 1 I109 W112 D113 T202 V255 S375 I424 M426 W427 Q432 I78 W81 D82 T154 V207 S326 I363 M365 W366 Q371 ? 0019031 remove_due_to_license_issue Q2N0S5 28825711 659 AENLWVTVYYGVPVWKDAETTLFCASDAKAETEKHNVWATHACVPTDPNPQEIHLENVTEEFNMWKNNMVEQMHTDIISLWDQSLKPCVKLTPLCVTLQCTNVTNNRGELKNCSFNMTTELRDKKQKVYSLFYRLDVVQINEYRLINCNTSAITQACPKVSFEPIPIHYCAPAGFAILKCKDKKFNGTGPCPSVSTVQCTHGIKPVVSTQLLLNGSLAEEEVMIRSENITNNAKNILVQFNTPVQINCTRPNNNTRKSIRIGPGQAFYATGDIIGDIRQAHCNVSKATWNETLGKVVKQLRKHFGNNTIIRFANSSGGDLEVTTHSFNCGGEFFYCNTSGLFNSTWISNNDSITLPCRIKQIINMWQRIGQAMYAPPIQGVIRCVSNITGLILTRDGGSTNSTTETFRPGGGDMRDNWRSELYKYKVVKIEPLGVAPTRCKRRV 5u8a A 1.45 BS01 82D A 1 F97 Y148 E238 L240 D310 Y365 R367 R414 F16 Y67 E157 L159 D229 Y284 R286 R333 ? Ki=13nM remove_due_to_license_issue Kd=90nM, Ki=13nM, IC50=8300nM O75530 28254486 501 FKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDR 5u8c B 1.598 BS01 84J B 1 H88 S114 T116 R121 G172 S173 T174 Y214 D215 H85 S111 T113 R118 G169 S170 T171 Y211 D212 ? 0015276,0016020 Ki=29.58nM remove_due_to_license_issue Q00959 28468946 301 SDDNHLSIVTLEEAPFVIVEDIDPLTETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGICHN 5u8f A 1.343 BS01 82G A 1 F97 Y148 L240 D310 Y365 R367 R414 F16 Y67 L159 D229 Y284 R286 R333 ? Ki=11nM remove_due_to_license_issue Ki=11nM, Kd=10.0nM, IC50=290nM O75530 28254486 501 FKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDR 5u94 A 2.2 BS01 G93 A 1 V25 K40 E59 M92 E93 V95 M155 D156 V23 K38 E57 M90 E91 V93 M153 D154 D138 K140 N143 D156 T179 D136 K138 N141 D154 T164 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=3.2nM P9WI81 30285456 301 TPSHLSDRYELGEILGFGGMSEVHLARDLRLHRDVAVKVLRADLARDPSFYLRFRREAQNAAALNHPAIVAVYDTGEAETPAGPLPYIVMEYVDGVTLRDIVHTEGPMTPKRAIEVIADACQALNFSHQNGIIHRDVKPANIMISATNAVKVMDFGIARAIIGTAQYLSPEQARGDSVDARSDVYSLGCVLYEVLTGEPPFTGDSPVSVAYQHVREDPIPPSARHEGLSADLDAVVLKALAKNPENRYQTAAEMRADLVRVHN 5u9b A -1.00 BS01 rna B 0 V3 S4 V5 I8 R9 D10 W13 L14 Q44 I51 A52 F54 R63 K67 Y68 E80 G83 R84 N86 L87 Q89 V3 S4 V5 I8 R9 D10 W13 L14 Q44 I51 A52 F54 R63 K67 Y68 E80 G83 R84 N86 L87 Q89 ? 0046872 remove_due_to_license_issue Q9NR56 28718627 95 ~ 109 MAVSVTPIRDTKWLTLEVCREFQRGTCSRPDTECKFAHPSKSCQVENGRVIACFDSLKGRCSRENCKYLHPPPHLKTQLEINGRNNLIQQKN 5u9d A 1.33 BS01 83P A 1 L408 G409 G411 F413 G414 V416 A428 K430 M431 M477 L528 D539 L20 G21 G23 F25 G26 V28 A40 K42 M43 M89 L140 D151 D521 A523 R525 N526 D539 F559 D133 A135 R137 N138 D151 F171 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.00055uM remove_due_to_license_issue IC50=0.55nM Q06187 28056160 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 5u9i A 2.3 BS01 FAR A 1 F37 M59 W72 L100 F28 M50 W63 L91 ? 0003755 remove_due_to_license_issue Q9NZN9 28739921 201 EGVKKTILHGGTGELPNFITGSRVIFHFRTMKCDEERTVIDDSRQVGQPMHIIIGNMFKLEVWEILLTSMRVHEVAEFWCDTIHTGVYPILSRSLRQMAQGKDPTEWHVHTCGLANMFAYHTLGYEDLDELQKEPQPLVFVIELLQVDAP 5uac C 3.8 BS01 RFP C 1 Q510 Q513 F514 D516 R529 S531 R687 Q510 Q513 F514 D516 R529 S531 R687 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 28009073 3001 MVYSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 5uah C 4.1 BS01 RFP C 1 Q510 Q513 F514 V516 R529 S531 L533 R540 I572 Q508 Q511 F512 V514 R527 S529 L531 R538 I570 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 28009073 3001 YSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMVQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 5ual C 3.887 BS01 RFP C 1 Q510 Q513 F514 D516 R529 L531 R687 Q510 Q513 F514 D516 R529 L531 R677 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 28009073 3001 MVYSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRILAAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKGETQLTPEEKLLRAIFGEKASDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELEDE 5uan A 3.508 BS02 dna E 0 G144 K145 Y147 K156 K160 R164 Q206 R209 G12 K13 Y15 K24 K28 R32 Q63 R66 ? 0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P19793 29021580 1 ~ 17 HICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDCLIDKRQRNCQYCRYQKCLAMGMKREAVQEERANEDMPVERILEAELAVEPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEA 5uan A 3.508 BS03 dna F 0 E153 G154 F158 R161 R184 N185 E21 G22 F26 R29 R42 N43 ? 0003677,0003700,0003707,0005634,0006355,0008270,0043565 remove_due_to_license_issue P19793 29021580 1 ~ 17 HICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDCLIDKRQRNCQYCRYQKCLAMGMKREAVQEERANEDMPVERILEAELAVEPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEA 5uan B 3.508 BS02 dna E 0 G90 Y91 H92 Y93 K102 R106 V151 R152 G11 Y12 H13 Y14 K23 R27 V72 R73 ? 0003677,0003700,0004879,0005634,0006355,0008270,0043565,0048384 remove_due_to_license_issue P10826 29021580 1 ~ 17 PCFVCQDKSSGYHYGVSACEGCKGFFRRSIQKNMIYTCHRDKNCVINKVTRNRCQYCRLQKCFEVGMSKESVRTAELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALKIYIRKRRPSKPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLE 5uan B 3.508 BS03 dna F 0 E99 G100 F104 R107 R137 E20 G21 F25 R28 R58 ? 0003677,0003700,0004879,0005634,0006355,0008270,0043565,0048384 remove_due_to_license_issue P10826 29021580 1 ~ 17 PCFVCQDKSSGYHYGVSACEGCKGFFRRSIQKNMIYTCHRDKNCVINKVTRNRCQYCRLQKCFEVGMSKESVRTAELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALKIYIRKRRPSKPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLE 5ubg A 1.9 BS02 PRT A 1 Q12 G15 R16 R54 D55 N75 C104 L170 S172 S173 G174 A175 T176 Q9 G12 R13 R51 D52 N72 C101 L167 S169 S170 G171 A172 T173 2.4.2.17 0000105,0003879,0005737 remove_due_to_license_issue Q5HSJ4 29208762 302 NTRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQENKFQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARE 5ubg B 1.9 BS02 PRT B 1 Q12 G15 R16 R54 D55 N75 C104 L170 V171 S172 S173 G174 A175 T176 Q9 G12 R13 R51 D52 N72 C101 L167 V168 S169 S170 G171 A172 T173 2.4.2.17 0000105,0003879,0005737 remove_due_to_license_issue Q5HSJ4 29208762 303 NTRLRIAIQKSGRLSKESIELLSECGVKMHIHEQSLIAFSTNLPIDILRVRDDDIPGLIFDGVVDLGIIGENVLEENELERQSLGENPSYKLLKKLDFGYCRLSLALPQENKFQNLKDFEGLRIATSYPQLLKRFMKENGINYKNCTLTGSVEVAPRANLADAICDLVSSGATLQANNLKEVKVIYESRACLIQKENALSKEKQALVDKIMLRVAGVMQARE 5ubt A 2.83 BS01 85S A 1 M752 P758 W760 K779 Y813 I825 V828 T833 M900 I910 M659 P665 W667 K683 Y717 I729 V732 T737 M789 I799 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue IC50=4.0nM O00329 28108251 4000 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPLPNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKATLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEKADCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRTEEEQLQLREILEGELYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLLLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKT 5uc1 A 2.351 BS01 486 A 1 L559 N560 G563 G564 Q566 M600 R607 F619 M642 L40 N41 G44 G45 Q47 M81 R88 F98 M121 ? remove_due_to_license_issue G5AQS2,P04150 29437838 801 TLPQLTPTLVSLLEVIEPEVLYAGYDGTVPDTTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQGNVLCFAPDLIINEQRMGLPYMYDQCKQMLFVSSELKRLQVSYEEYLCMKTLLLFSSVPKEGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHENVT 5uc1 B 2.351 BS01 486 B 1 L559 N560 G563 G564 Q566 M600 F619 M642 L40 N41 G44 G45 Q47 M81 F98 M121 ? remove_due_to_license_issue G5AQS2,P04150 29437838 801 TLPQLTPTLVSLLEVIEPEVLYAGYDGTVPDTTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQGNVLCFAPDLIINEQRMGLPYMYDQCKQMLFVSSELKRLQVSYEEYLCMKTLLLFSSVPKEGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHENVT 5uc4 A 2.05 BS01 83S A 1 L43 N46 A50 D88 I91 G92 M93 F133 T179 L45 N48 A52 D90 I93 G94 M95 F135 T181 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.35uM remove_due_to_license_issue Kd=240nM P08238 29382832 301 GHMPEEVHHGEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYL 5uc6 A 2.1 BS01 dna B 0 M15 R16 K60 S61 K63 D64 D65 K67 I68 W113 M7 R8 K52 S53 K55 D56 D57 K59 I60 W105 ? 0005125,0005149,0005576,0005615,0006954,0006955 remove_due_to_license_issue P01583 28993621 1 ~ 22 NVKYNFMRIIKYEFILNDALNQSIIRANDQYLTAAALHNLDEAVKFDMGAYKSSKDDAKITVILRISKTQLYVTAQDEDQPVLLKEMPEIPKTITGSETNLLFFWETHGTKNYFTSVAHPNLFIATKQDYWVCLAGGPPSITDFQILENQA 5uch A 2.654 BS01 871 A 1 L43 N46 D49 A50 D88 I91 M93 F133 T179 L45 N48 D51 A52 D90 I93 M95 F135 T181 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Kd=970nM P08238 29382832 301 GHMPEEVHHGEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYL 5uci A 2.7 BS01 874 A 1 L43 N46 A47 D49 A50 K53 D88 I91 M93 F133 T179 L45 N48 A49 D51 A52 K55 D90 I93 M95 F135 T181 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Kd=4270nM P08238 29382832 301 GHMPEEVHHGEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYL 5ucj A 1.693 BS01 KU3 A 1 L43 N46 A50 K53 D88 I91 G92 M93 F133 T179 V181 L44 N47 A51 K54 D89 I92 G93 M94 F134 T180 V182 ? 0005524,0006457,0016887,0051082,0140662 Kd=0.44uM remove_due_to_license_issue P08238 29382832 301 HMPEEVHHGEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYL 5udz A 2.0 BS01 rna V 0 W46 F47 N48 V49 R50 M51 F53 F55 F73 H75 Q76 F84 R85 K102 G103 E105 K125 W14 F15 N16 V17 R18 M19 F21 F23 F41 H43 Q44 F52 R53 K70 G71 E73 K93 ? 0003676,0008270 remove_due_to_license_issue Q9H9Z2 28297670 1 ~ 24 DEPQLLHGAGICKWFNVRMGFGFLSMTARAGVALDPPVDVFVHQSKLHMEGFRSLKEGEAVEFTFKKSAKGLESIRVTGPGGVFCIGSERRPKGGDRCYNCGGLDHHAKECKLPPQPKKCHFCQSISHMVASCPLKAQQ 5udz A 2.0 BS02 rna W 0 G136 R138 C139 Y140 H148 A149 Q157 K159 K160 C161 H162 F163 M170 V171 K177 G95 R97 C98 Y99 H107 A108 Q116 K118 K119 C120 H121 F122 M129 V130 K136 ? 0003676,0008270 remove_due_to_license_issue Q9H9Z2 28297670 1 ~ 23 DEPQLLHGAGICKWFNVRMGFGFLSMTARAGVALDPPVDVFVHQSKLHMEGFRSLKEGEAVEFTFKKSAKGLESIRVTGPGGVFCIGSERRPKGGDRCYNCGGLDHHAKECKLPPQPKKCHFCQSISHMVASCPLKAQQ 5udz B 2.0 BS01 rna V 0 G136 R138 C139 Y140 H148 A149 Q157 K159 K160 C161 H162 F163 M170 V171 K177 G95 R97 C98 Y99 H107 A108 Q116 K118 K119 C120 H121 F122 M129 V130 K136 ? 0003676,0008270 remove_due_to_license_issue Q9H9Z2 28297670 1 ~ 24 DEPQLLHGAGICKWFNVRMGFGFLSMTARAGVALDPPVDVFVHQSKLHMEGFRSLKEGEAVEFTFKKSAKGLESIRVTGPGGVFCIGSERRPKGGDRCYNCGGLDHHAKECKLPPQPKKCHFCQSISHMVASCPLKAQQ 5udz B 2.0 BS02 rna W 0 K45 W46 F47 N48 V49 R50 M51 F53 F55 D71 F73 H75 F84 S100 K102 E105 R122 K13 W14 F15 N16 V17 R18 M19 F21 F23 D39 F41 H43 F52 S68 K70 E73 R90 ? 0003676,0008270 remove_due_to_license_issue Q9H9Z2 28297670 1 ~ 23 DEPQLLHGAGICKWFNVRMGFGFLSMTARAGVALDPPVDVFVHQSKLHMEGFRSLKEGEAVEFTFKKSAKGLESIRVTGPGGVFCIGSERRPKGGDRCYNCGGLDHHAKECKLPPQPKKCHFCQSISHMVASCPLKAQQ 5ue4 B 1.8 BS05 5XQ B 1 V101 P102 R106 F110 L114 Y179 H190 A191 F192 P193 H230 G233 L234 V55 P56 R60 F61 L65 Y130 H141 A142 F143 P144 H181 G184 L185 H226 E227 H230 H236 H177 E178 H181 H187 3.4.24.35 0004222,0006508,0008237,0008270,0031012 Kd=3.3uM remove_due_to_license_issue P14780 28860188 307 DRQLAEEYLYRYGYTRVAESLGPALLLLQKQLSLPETGELDSATLKAMRTPRCGVPDLGRFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5ueu A 2.26 BS01 0S6 A 1 W374 P375 F376 V380 L387 N433 V439 M442 W26 P27 F28 V32 L39 N85 V91 M94 ? remove_due_to_license_issue Ki=17nM, IC50=18.2nM O60885 28368119 501 SHMEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM 5uex A 2.29 BS01 89D A 1 W374 P375 F376 V380 L385 N433 H437 E438 V439 W26 P27 F28 V32 L37 N85 H89 E90 V91 ? Ki=1.5nM remove_due_to_license_issue O60885 28368119 501 SHMEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM 5uey A 2.41 BS01 88M A 1 W374 P375 V380 D381 L385 N433 E438 V439 W25 P26 V31 D32 L36 N84 E89 V90 ? Ki=5.1nM remove_due_to_license_issue O60885 28368119 501 HMEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM 5uez A 1.51 BS01 89G A 1 N433 H437 E438 V439 N85 H89 E90 V91 ? Ki=970nM remove_due_to_license_issue Ki=970nM, EC50=3000nM O60885 28368119 501 SHMEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM 5ufi A 2.58 BS01 8B1 A 1 F89 V102 A106 Q114 C115 E116 F117 F164 M177 Y181 F30 V43 A47 Q55 C56 E57 F58 F105 M118 Y122 ? remove_due_to_license_issue IC50=21nM Q96GG9 29074978 301 LDRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHKRSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQI 5ufi A 2.58 BS02 8B1 C 1 I83 Q87 P97 I24 Q28 P38 ? remove_due_to_license_issue IC50=21nM Q96GG9 29074978 301 LDRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHKRSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQI 5ufo A 2.802 BS01 87J A 1 L287 C320 H323 R364 M365 F377 F378 E379 F388 L396 H479 L23 C56 H59 R100 M101 F113 F114 E115 F124 L132 H215 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=240nM, Kd=37nM P51449 28318945 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHL 5ufp A 1.9 BS01 86D A 1 F244 H248 M252 A277 Y281 M289 S292 H293 L296 S304 Y307 M309 T321 I337 C339 N341 F6 H10 M14 A39 Y43 M51 S54 H55 L58 S66 Y69 M71 T83 I95 C97 N99 ? remove_due_to_license_issue IC50=10.0nM, EC50=6.0nM Q99814 27595393 401 LDSKTFLSEHSMDMKFTYCDDRITELIGYHPEELLGRSAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGGYVWLETQGTVIYNPPQCIMCVNYVLSE 5ufr A 2.068 BS01 88J A 1 Q286 L287 C320 H323 M365 F377 E379 F388 I400 Q22 L23 C56 H59 M101 F113 E115 F124 I136 ? 0003677,0004879,0005634,0006355 Kd=0.002uM remove_due_to_license_issue Kd=2.0nM, IC50=7.5nM P51449 28318945 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQ 5ufs A 2.118 BS02 1TA A 1 M29 L32 N33 Q39 M70 M73 F92 M108 Q111 F204 T208 M32 L35 N36 Q42 M73 M76 F95 M111 Q114 F207 T211 ? 0003677 Ki=3.2nM remove_due_to_license_issue A0A1X8XLE9 28396564 301 APTLISLLEVIEPEVLYSGYDSTLPDTSTRLMSTLNRLGGRQVVSAVKWAKALPGFRNLHLDDQMTLLQYSWMSLMAFSLGWRSYKQSNGNMLCFAPDLVINEERMQLPYMYDQCQQMLKISSEFVRLQVSYDEYLCMKVLLLLSTVPKDGLKSQAVFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEMVGGLLQFCFYTFVNKSLSVEFPEMLAEIISNQLPKFKAGSVKPLLFHQ 5ug8 A 1.46 BS01 8BP A 1 L718 G719 A743 C775 M790 M793 P794 G796 C797 D800 L844 F856 L17 G18 A42 C70 M85 M88 P89 G91 C92 D95 L139 F151 D837 A839 R841 N842 D855 G874 D132 A134 R136 N137 D150 G169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 28287730 9001 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 5ug9 A 1.33 BS01 8AM A 1 L718 G719 A743 C775 M790 M793 P794 G796 C797 D800 L844 L17 G18 A42 C70 M85 M88 P89 G91 C92 D95 L139 D837 A839 R841 N842 D855 G874 D132 A134 R136 N137 D150 G169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 28287730 9001 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 5uga A 1.82 BS01 8BM A 1 L718 V726 A743 M793 P794 G796 L844 L16 V24 A41 M91 P92 G94 L142 D837 A839 R841 N842 D855 G874 D135 A137 R139 N140 D153 G172 2.7.10.1 0004672,0004713,0005524,0006468 Ki=161nM remove_due_to_license_issue Ki=161nM P00533 28287730 9001 LLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 5ugb A 2.53 BS01 8BM A 1 L718 A743 T790 M793 P794 G796 L844 L24 A49 T94 M97 P98 G100 L148 D837 A839 R841 N842 D855 G874 D141 A143 R145 N146 D159 G178 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Ki=161nM P00533 28287730 9001 SGEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPDMDDVVDADEYLI 5ugc A 1.58 BS01 8BS A 1 L718 G719 A743 M790 M793 P794 G796 C797 D800 L844 L17 G18 A42 M85 M88 P89 G91 C92 D95 L139 D837 A839 R841 N842 D855 G874 D132 A134 R136 N137 D150 G169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 28287730 9001 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 5ugd A 1.38 BS01 89S A 1 F587 C588 H603 D735 S736 C737 Q738 G739 S741 T759 G762 F42 C43 H58 D190 S191 C192 Q193 G194 S196 T214 G217 H603 D646 Q738 G739 D740 S741 G742 H58 D101 Q193 G194 D195 S196 G197 3.4.21.7 0004252,0006508 remove_due_to_license_issue IC50=240nM P00747 29296720 801 PSFDCGKPQVEPKKCPVVGGCVAHPHSWPWQVSLRTRFGMHFCGGTLISPEWVLTAAHCLEKSPRPSSYKVILGAHQEVNLEPHVQEIEVSRLFLEPTRKDIALLKLSSPAVITDKVIPACLPSPNYVVADRTECFITGWGETQGTFGAGLLKEAQLPVIENKVCNRYEFLNGRVQSTELCAGHLAGGTDSCQGDSGGPLVCFEKDKYILQGVTSWGLGCARPNKPGVYVRVSRFVTWIEGVMRNN 5ugg A 1.2 BS01 89M A 1 F587 C588 H603 K607 D735 S736 C737 Q738 G739 S741 T759 G762 F42 C43 H58 K62 D190 S191 C192 Q193 G194 S196 T214 G217 H603 D646 Q738 G739 D740 S741 G742 H58 D101 Q193 G194 D195 S196 G197 3.4.21.7 0004252,0006508 remove_due_to_license_issue IC50=380nM P00747 29296720 801 PSFDCGKPQVEPKKCPVVGGCVAHPHSWPWQVSLRTRFGMHFCGGTLISPEWVLTAAHCLEKSPRPSSYKVILGAHQEVNLEPHVQEIEVSRLFLEPTRKDIALLKLSSPAVITDKVIPACLPSPNYVVADRTECFITGWGETQGTFGAGLLKEAQLPVIENKVCNRYEFLNGRVQSTELCAGHLAGGTDSCQGDSGGPLVCFEKDKYILQGVTSWGLGCARPNKPGVYVRVSRFVTWIEGVMRNN 5ugh A 2.062 BS01 8AJ A 1 L315 S331 I332 F333 E342 L289 S305 I306 F307 E316 H29 D31 K32 E57 E70 K181 F250 D258 A259 R264 K265 K285 K289 D291 H18 D20 K21 E46 E59 K157 F226 D232 A233 R238 K239 K259 K263 D265 2.5.1.6 0004478,0005515,0005524,0005829,0006556,0006730,0016740,0034214,0036094,0042802,0046872,0048269,0051291,0061431,1904263,1990830 Kd=170nM remove_due_to_license_issue P31153 28553945 401 FIEEGTFLFTSESVGEGHPDKICDQISDAVLDAHLQQDPDAKVACETVAKTGMILLAGEITSRAAVDYQKVVREAVKHIGYDDSSKGFDYKTCNVLVALEQQSEDIGAGDQGLMFGYATDETEECMPLTIVLAHKLNAKLAELRRNGTLPWLRPDSKTQVTVQYMQDRGAVLPIRVHTIVISVQHDEEVCLDEMRDALKEKVIKAVVPAKYLDEDTIYHLQPSGRFVIGGPDAGLTGRKIIVDTYGGWGAHGGGAFSGKDYTKVDRSAAYAARWVAKSLVKGGLCRRVLVQVSYAIGVSHPLSISIFHYGTSQKSERELLEIVKKNFDLRPGVIVRDLDLKKPIYQRTAAYGHFGRDSFPWEVPKKLKY 5ugh A 2.062 BS02 8AJ C 1 F18 F20 Q190 G273 W274 F7 F9 Q166 G247 W248 H29 D31 K32 E57 E70 K181 F250 D258 A259 R264 K265 K285 K289 D291 H18 D20 K21 E46 E59 K157 F226 D232 A233 R238 K239 K259 K263 D265 2.5.1.6 0004478,0005515,0005524,0005829,0006556,0006730,0016740,0034214,0036094,0042802,0046872,0048269,0051291,0061431,1904263,1990830 Kd=170nM remove_due_to_license_issue P31153 28553945 401 FIEEGTFLFTSESVGEGHPDKICDQISDAVLDAHLQQDPDAKVACETVAKTGMILLAGEITSRAAVDYQKVVREAVKHIGYDDSSKGFDYKTCNVLVALEQQSEDIGAGDQGLMFGYATDETEECMPLTIVLAHKLNAKLAELRRNGTLPWLRPDSKTQVTVQYMQDRGAVLPIRVHTIVISVQHDEEVCLDEMRDALKEKVIKAVVPAKYLDEDTIYHLQPSGRFVIGGPDAGLTGRKIIVDTYGGWGAHGGGAFSGKDYTKVDRSAAYAARWVAKSLVKGGLCRRVLVQVSYAIGVSHPLSISIFHYGTSQKSERELLEIVKKNFDLRPGVIVRDLDLKKPIYQRTAAYGHFGRDSFPWEVPKKLKY 5ugh C 2.062 BS01 8AJ A 1 G16 F18 F20 G273 W274 G3 F5 F7 G246 W247 H29 D31 K32 E57 E70 K181 F250 D258 A259 R264 K265 K285 K289 D291 H16 D18 K19 E44 E57 K156 F225 D231 A232 R237 K238 K258 K262 D264 2.5.1.6 0004478,0005515,0005524,0005829,0006556,0006730,0016740,0034214,0036094,0042802,0046872,0048269,0051291,0061431,1904263,1990830 Kd=170nM remove_due_to_license_issue P31153 28553945 401 EEGTFLFTSESVGEGHPDKICDQISDAVLDAHLQQDPDAKVACETVAKTGMILLAGEITSRAAVDYQKVVREAVKHIGYDDSSKGFDYKTCNVLVALEQQSEEDIGAGDQGLMFGYATDETEECMPLTIVLAHKLNAKLAELRRNGTLPWLRPDSKTQVTVQYMQDRGAVLPIRVHTIVISVQHDEEVCLDEMRDALKEKVIKAVVPAKYLDEDTIYHLQPSGRFVIGGPDAGLTGRKIIVDTYGGWGAHGGGAFSGKDYTKVDRSAAYAARWVAKSLVKGGLCRRVLVQVSYAIGVSHPLSISIFHYGTSQKSERELLEIVKKNFDLRPGVIVRDLDLKKPIYQRTAAYGHFGRDSFPWEVPKKLKY 5ugh C 2.062 BS02 8AJ C 1 L315 S331 I332 F333 E342 L288 S304 I305 F306 E315 H29 D31 K32 E57 E70 K181 F250 D258 A259 R264 K265 K285 K289 D291 H16 D18 K19 E44 E57 K156 F225 D231 A232 R237 K238 K258 K262 D264 2.5.1.6 0004478,0005515,0005524,0005829,0006556,0006730,0016740,0034214,0036094,0042802,0046872,0048269,0051291,0061431,1904263,1990830 Kd=170nM remove_due_to_license_issue P31153 28553945 401 EEGTFLFTSESVGEGHPDKICDQISDAVLDAHLQQDPDAKVACETVAKTGMILLAGEITSRAAVDYQKVVREAVKHIGYDDSSKGFDYKTCNVLVALEQQSEEDIGAGDQGLMFGYATDETEECMPLTIVLAHKLNAKLAELRRNGTLPWLRPDSKTQVTVQYMQDRGAVLPIRVHTIVISVQHDEEVCLDEMRDALKEKVIKAVVPAKYLDEDTIYHLQPSGRFVIGGPDAGLTGRKIIVDTYGGWGAHGGGAFSGKDYTKVDRSAAYAARWVAKSLVKGGLCRRVLVQVSYAIGVSHPLSISIFHYGTSQKSERELLEIVKKNFDLRPGVIVRDLDLKKPIYQRTAAYGHFGRDSFPWEVPKKLKY 5uhi A 3.198 BS01 8A4 A 1 Q286 L287 H323 M365 F377 F378 F388 I400 V480 Q22 L23 H59 M101 F113 F114 F124 I136 V216 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=9.2nM, IC50=73nM P51449 28318945 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQ 5ui5 I 3.4 BS01 dna A 0 L294 R295 S309 R310 R327 S361 D362 R378 R379 R385 R394 L216 R217 S231 R232 R249 S279 D280 R296 R297 R303 R312 ? 0001216,0003677,0006352,0016987 remove_due_to_license_issue O66858 28223493 1 ~ 31 ELEELQQNIKLELEGKEQELALELLNYLNEKGFLSKSVEEISDVLRCSVEELEKVRQKVLRLEPLGVCSKDVWEFLELQIEEIYPEEEEILKKALRDLKRGKKLKPEIKGKLSRLRLFPSAEKVYTFAKVDAIIEEENGEFFIYLYEDFIDIDLNEEYWELYKNLQKELKEAFERYESIRKVLDIRRRNLRKVLEKIVERQKDFLTGKGSLKPLTLREVSSEIGIHESTLSRIVNSKYVKTPVGTYSLRTFFVRESAEGLTQGELMKLIKEIVERKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERRI 5ui5 I 3.4 BS02 dna B 0 H304 S306 A377 R379 T380 Y384 H226 S228 A295 R297 T298 Y302 ? 0001216,0003677,0006352,0016987 remove_due_to_license_issue O66858 28223493 34 ~ 63 ELEELQQNIKLELEGKEQELALELLNYLNEKGFLSKSVEEISDVLRCSVEELEKVRQKVLRLEPLGVCSKDVWEFLELQIEEIYPEEEEILKKALRDLKRGKKLKPEIKGKLSRLRLFPSAEKVYTFAKVDAIIEEENGEFFIYLYEDFIDIDLNEEYWELYKNLQKELKEAFERYESIRKVLDIRRRNLRKVLEKIVERQKDFLTGKGSLKPLTLREVSSEIGIHESTLSRIVNSKYVKTPVGTYSLRTFFVRESAEGLTQGELMKLIKEIVERKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERRI 5ui5 V 3.4 BS01 dna N 0 T293 L294 R295 S309 R327 R332 D362 Q363 R378 R385 R394 T219 L220 R221 S235 R253 R258 D288 Q289 R304 R311 R320 ? 0001216,0003677,0006352,0016987 remove_due_to_license_issue O66858 28223493 1 ~ 31 ELEELQQNIKLELEGKEQELALELLNYLNEKGFLSKSVEEISDVLRCSVEELEKVRQKVLRLEPLGVCSKDVWEFLELQIEEIYPEEEEILKKALRDLKRGKKLKPEIKGKLSRLRLFPLSAEKVYTFAKVDAIIEEENGEFFIYLYEDFIDIDLNEEYWELYKKSRNLQKELKEAFERYESIRKVLDIRRRNLRKVLEKIVERQKDFLTGKGSLKPLTLREVSSEIGIHESTLSRIVNSKYVKTPVGTYSLRTFFVRESAEGLTQGELMKLIKEIVENEDKRKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERR 5ui5 V 3.4 BS02 dna O 0 S306 S334 R379 T380 Y384 R394 S232 S260 R305 T306 Y310 R320 ? 0001216,0003677,0006352,0016987 remove_due_to_license_issue O66858 28223493 34 ~ 63 ELEELQQNIKLELEGKEQELALELLNYLNEKGFLSKSVEEISDVLRCSVEELEKVRQKVLRLEPLGVCSKDVWEFLELQIEEIYPEEEEILKKALRDLKRGKKLKPEIKGKLSRLRLFPLSAEKVYTFAKVDAIIEEENGEFFIYLYEDFIDIDLNEEYWELYKKSRNLQKELKEAFERYESIRKVLDIRRRNLRKVLEKIVERQKDFLTGKGSLKPLTLREVSSEIGIHESTLSRIVNSKYVKTPVGTYSLRTFFVRESAEGLTQGELMKLIKEIVENEDKRKPYSDQEIANILKEKGFKVARRTVAKYREMLGIPSSRERR 5uig A 3.5 BS02 8D1 A 1 A63 S67 V84 L85 F168 M177 L249 M270 Y271 I274 A60 S64 V81 L82 F155 M164 L325 M346 Y347 I350 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P29274 28167788 503 MGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLRQQ 5uiq A 2.64 BS01 8BV A 1 M192 V200 A211 Y262 M265 L318 M23 V31 A40 Y78 M81 L134 D311 K313 A315 N316 D329 T351 D127 K129 A131 N132 D145 T163 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=55000nM Q9NWZ3 28498658 501 RFHSFSFYELKNVTNNFDERPKMGEGGFGVVYKGYVTTVAVKKLAAKQQFDQEIKVMAKCQHENLVELLGFSSDCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5uir A 2.64 BS01 8BY A 1 E194 V200 A211 K213 Y262 Y264 M265 K313 A315 L318 E26 V32 A43 K45 Y87 Y89 M90 K138 A140 L143 D311 K313 A315 N316 D329 T351 D136 K138 A140 N141 D154 T168 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=72nM Q9NWZ3 28498658 800 FHSFSFYELKNVTNNFDERPGNKMGEGGFGVVYKGYVNNTTVAVKKLADITTEELKQQFDQEIKVMAKCQHENLVELLGFSDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5uis A 2.5 BS01 8C1 A 1 E194 V200 A211 Y262 Y264 M265 A315 N316 L318 E30 V34 A45 Y85 Y87 M88 A138 N139 L141 D311 K313 A315 N316 D329 T351 D134 K136 A138 N139 D152 T166 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=146nM remove_due_to_license_issue IC50=146nM Q9NWZ3 28498658 800 FHSFSFYELKNVTNNFDERPISVGGNKMGEGGVVYKGYVNNTTVAVKKLKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5uit A 1.84 BS01 8CD A 1 M192 E194 G195 A211 Y262 Y264 M265 A315 N316 L318 S328 M31 E33 G34 A50 Y95 Y97 M98 A148 N149 L151 S161 D311 K313 A315 N316 D329 T351 D144 K146 A148 N149 D162 T179 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=4.6nM remove_due_to_license_issue IC50=4.60nM Q9NWZ3 28498658 501 DTRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLTTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5uiu A 2.02 BS01 8CG A 1 E194 G198 V200 A211 Y262 Y264 M265 A315 N316 L318 S328 E30 G34 V36 A47 Y98 Y100 M101 A151 N152 L154 S164 D311 K313 A315 N316 D329 T351 D147 K149 A151 N152 D165 T182 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=0.2nM remove_due_to_license_issue IC50=0.200nM Q9NWZ3 28498658 4000 FHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5ujo A 1.35 BS02 LSI A 1 I108 A125 Y129 I82 A99 Y103 S70 K73 S130 A166 K234 S237 S44 K47 S104 A140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9L5C8 29051683 303 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTAPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 5ujv A 2.7 BS01 A8S A 1 K72 A106 F125 Y137 F178 K62 A96 F115 Y127 F168 ? 0004864,0005634,0005737,0009738,0010427,0038023 remove_due_to_license_issue A0A2D1UXN2 29070857 900 EVPAGLGLTAAEYAELQPTVEAYHRYAVGPGQCSSLVAQRIEAPAAAVWAIVRRFDCPQVYKHFIRSCALRPDPDAGDELRPGRLREVSVISGLPASTSTERLDLLDDARRAFGFTITGGEHRLANYRSVTTVSELAPAAPAKICTVVLESYVVDVPEGNSEEDTRLFADTVVRLNLQKLKSLAEANATSAA 5uk8 A 2.5 BS01 8DV A 1 M772 S774 P778 M800 K802 D810 Y836 I848 E849 W850 V851 M922 I932 D933 M731 S733 P737 M759 K761 D769 Y795 I807 E808 W809 V810 M873 I883 D884 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 Kd=0.4uM remove_due_to_license_issue P42336 28433539 1101 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRISTSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECEIMSSAKRPLKLNWENPDIMSELLFQNNIIMFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEWVRNSHTIMQIQCKFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLVHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTTKMDW 5ukj A 2.8 BS01 3K6 A 1 M800 K802 I848 E849 W850 V851 S854 Q859 M922 I932 D933 M763 K765 I811 E812 W813 V814 S817 Q822 M878 I888 D889 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue IC50=>10000nM P42336 28433539 1101 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRISTSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSRELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECEIMSSAKRPLKLNWENPDIMSELLFQNNIIMFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEWVRNSHTIMQIQCKQFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLVHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTT 5ukk A 2.6 BS02 8DJ A 1 I197 R199 G200 F202 G203 V205 A218 L222 L235 A236 E239 V255 M274 D278 A321 L324 D335 A480 I159 R161 G162 F164 G165 V167 A180 L184 L197 A198 E201 V217 M236 D240 A283 L286 D297 A442 D317 K319 N322 D335 K344 T353 D279 K281 N284 D297 K306 T315 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue P25098 28323425 702 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVNAADAFDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNK 5ukl A 2.15 BS02 SIX A 1 R199 G200 F202 G203 V205 A218 V255 M274 D278 A321 A482 R169 G170 F172 G173 V175 A188 V225 M244 D248 A291 A452 D317 K319 N322 D335 K344 T353 D287 K289 N292 D305 K314 T323 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 ic50=0.63uM remove_due_to_license_issue P25098 28323425 702 KILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVNAADAFDIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGHEEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKPRAP 5ukm A 3.03 BS01 T0E A 1 I197 R199 G200 F202 G203 E204 V205 A218 E239 V255 M274 A321 L324 S334 D335 I167 R169 G170 F172 G173 E174 V175 A188 E209 V225 M244 A291 L294 S304 D305 D317 K319 N322 D335 K344 T353 D287 K289 N292 D305 K314 T323 2.7.11.15 0001664,0002026,0002029,0002031,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0006468,0006886,0007165,0007186,0007213,0007217,0007507,0009966,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0042995,0045202,0045880,0045988,0046718,0047696,0060048,0098793,0098794,1901081,1903566 remove_due_to_license_issue IC50=30nM P21146 28323425 701 KILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLKHLEEAKPLVEFYEEIKKYEKLETEEERLVCSREIFDTYIMKELLACSHPFSKSAIEHVQGHLVKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVNAADAFDIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKTKNKQLGHEEDYALGKDCIMHGYMSKMWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFVLQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKPR 5ul1 A 3.0 BS01 8DY A 1 K802 W850 V851 S854 H855 T856 Q859 M922 I932 D933 K759 W807 V808 S811 H812 T813 Q816 M869 I879 D880 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue P42336 28433539 1101 PPRPSSGELWGIHLMPPRILVECLLPNGMIVTLECLREATLITIKHELFKEARKYPLHQLLQDESSYIFVSVTQEAEREEFFDETRRLCDLRLFQPFLKVIEPVGNREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRITKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECEIMSSAKRPLKLNWENPDIMSELLFQNNIIMFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEWVRNSHTIMQIQCNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLVHIDFGHFLDHKKKKFGYKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGWTT 5ul5 A 2.2 BS02 8D7 A 1 F61 F103 T147 E148 N175 G176 F264 F279 F61 F103 T130 E131 N158 G159 F242 F257 3.1.1.64,5.3.3.22 0001523,0001786,0001895,0003834,0004744,0005634,0005737,0005783,0005789,0005886,0006629,0007601,0016020,0016702,0016787,0016853,0031210,0042572,0042574,0042802,0046872,0050251,0050908,0052884,0052885,1901612,1901827 ic50=106nM remove_due_to_license_issue IC50=<1000nM Q28175 28476927 603 MSSQVEHPAGGYKKLFETVEELSSPLTAHVTGRIPLWLTGSLLRCGPGLFEVGSEPFYHLFDGQALLHKFDFKEGHVTYHRRFIRTDAYVRAMTEKRIVITEFGTCAFVEVTDNALVNIYPVGEDYYACTETNFITKVNPETLETIKQVDLCNYVSVNGATAHPHIENDGTVYNIGNCFIAYNIVKIPPLQADKEDPISKSEIVVQFPCSDRFKPSYVHSFGLTPNYIVFVETPVKINLFKFLSSWSLWGANYMDCFESNETMGVWLHIADKKRKKYINNKYRTSPFNLFHHINTYEDHEFLIVDLCCWKGFEFVYNYLYLANLRENWEEVKKNARKAPQPEVRRYVLPLNIDKADTGKNLVTLPNTTATAILCSDETIWLEPEVLFSGPRQAFEFPQINYQKYGGKPYTYAYGLGLNHFVPDRLCKLNVKTKETWVWQEPDSYPSEPIFVSHPDALEEDDGVVLSVVVSPGAGQKPAYLLILNAKDLSEVARAEVEINIPVTFHGLFKKS 5ula A 1.5 BS01 5MJ A 1 W81 P82 V87 L92 I146 W38 P39 V44 L49 I103 ? Ki=77nM remove_due_to_license_issue O60885 28265070 201 NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKIN 5ulg A 2.1 BS02 8E4 A 1 F61 F103 T147 E148 Y275 F279 Y338 F61 F103 T130 E131 Y248 F252 Y311 3.1.1.64,5.3.3.22 0001523,0001786,0001895,0003834,0004744,0005634,0005737,0005783,0005789,0005886,0006629,0007601,0016020,0016702,0016787,0016853,0031210,0042572,0042574,0042802,0046872,0050251,0050908,0052884,0052885,1901612,1901827 ic50=189nM remove_due_to_license_issue Q28175 28476927 603 MSSQVEHPAGGYKKLFETVEELSSPLTAHVTGRIPLWLTGSLLRCGPGLFEVGSEPFYHLFDGQALLHKFDFKEGHVTYHRRFIRTDAYVRAMTEKRIVITEFGTCAFPEVTDNALVNIYPVGEDYYACTETNFITKVNPETLETIKQVDLCNYVSVNGATAHPHIENDGTVYNIGNCFIAYNIVKIPPLQADKEDPISKSEIVVQFPCSDRFKPSYVHSFGLTPNYIVFVETPVKINLFKFLSGANYMDCFESNETMGVWLHIADKKRKKYINNKYRTSPFNLFHHINTYEDHEFLIVDLCCWKGFEFVYNYLYLANLRENWEEVKKNARKAPQPEVRRYVLPLNIDKADTGKNLVTLPNTTATAILCSDETIWLEPEVLFSGPRQAFEFPQINYQKYGGKPYTYAYGLGLNHFVPDRLCKLNVKTKETWVWQEPDSYPSEPIFVSHPDALEEDDGVVLSVVVSPGAGQKPAYLLILNAKDLSEVARAEVEINIPVTFHGLFKKS 5uln A 1.35 BS02 8JS A 1 H94 H119 F131 L198 T199 T200 P202 H93 H118 F129 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=14.2nM remove_due_to_license_issue Ki=14nM P00918 28947945 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5ulp A 1.55 BS01 KB1 A 1 S56 G81 G86 W87 T104 K105 H110 V130 D131 V132 F133 D146 S52 G77 G82 W83 T100 K101 H106 V126 D127 V128 F129 D142 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004482,0004483,0008168,0032259 Kd=24.3uM remove_due_to_license_issue A0A024B7W1 28487506 301 GETLGEKWKARLNQMSALEFYSYKKSGITEVCREEARRALKDGVATGGHAVSRGSAKLRWLVERGYLQPYGKVIDLGCGRGGWSYYAATIRKVQEVKGYTKGGPGHEEPMLVQSYGWNIVRLKSGVDVFHMAAEPCDTLLCDIGESSSSPEVEEARTLRVLSMVGDWLEKRPGAFCIKVLCPYTSTMMETLERLQRRYGGGLVRVPLSRNSTHEMYWVSGAKSNTIKSVSTTSQLLLGRMDGPRRPVKYEEDVNLGSGTRAV 5ult A 1.53 BS01 8FM B 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 28418652 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5ult B 1.53 BS01 8FM B 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.014nM remove_due_to_license_issue P03366 28418652 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5umw A 2.27 BS01 RBF F 1 M34 W41 M33 W40 ? 0004462,0046872,0051213 remove_due_to_license_issue A0A125SA26 29937405 201 SARLSHVTVPVLDQDSAKEFYTEKLGFEVRNDMTMGGLRWLTVGPKDQPDVEMVLRRVGAPEYDEETAEQLRDLVAKGVIGVGVLHVDDTRATYERYRAAGVIFIQEPVKRPYGTEAVFRDDSGNWFSLTDARG 5umx A 1.59 BS01 RBF B 1 Q35 W42 Q37 W44 ? 0046872,0051213 remove_due_to_license_issue A0A125SA29 29937405 201 SHMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQP 5umx B 1.59 BS01 RBF B 1 W100 Q103 W102 Q105 ? 0046872,0051213 Kd=1100nM remove_due_to_license_issue A0A125SA29 29937405 201 SHMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQP 5umx B 1.59 BS02 RBF B 2 Q7 Q35 H39 W42 Q9 Q37 H41 W44 ? 0046872,0051213 Kd=1100nM remove_due_to_license_issue A0A125SA29 29937405 202 SHMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQP 5umy A 1.78 BS01 TNN A 1 G70 W100 Q103 G71 W101 Q104 ? 0046872,0051213 Kd=108nM remove_due_to_license_issue A0A125SA29 29937405 201 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 5umy A 1.78 BS02 TNN A 2 L8 S10 V38 H39 W42 L9 S11 V39 H40 W43 ? 0046872,0051213 Kd=108nM remove_due_to_license_issue A0A125SA29 29937405 202 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 5umy B 1.78 BS01 TNN A 1 L8 S10 V38 H39 W42 L9 S11 V39 H40 W43 ? 0046872,0051213 remove_due_to_license_issue A0A125SA29 29937405 201 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 5umy B 1.78 BS02 TNN A 2 G70 W100 G71 W101 ? 0046872,0051213 remove_due_to_license_issue A0A125SA29 29937405 202 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 5un1 G 3.6 BS03 BMK G 1 V634 A635 V232 A233 ? 0005216,0006811,0015276,0016020,0038023 remove_due_to_license_issue A0A1L8F5J9 29670280 1005 MSTRLKIVTIHQEPFVYVRPTTSDGTCREEYTINGDPIKKVICNGPDETIPGRPTVPQCCYGFCVDLLIKLAREMDFTYEVHLVADGKFGTQERVNNSNAAAWNGMMGELLSGQADMIVAPLTINNERAQYIEFSKPFKYQGLTILVKKEIPRSTLDSFMQPFQSTLWLLVGLSVHVVAVMLYLLDRFSTLSSAMWFSWRVLLNSGLGEGAPRSFSARILGMVWAGFAMIIVASYTANLAAFLVLRRPEERITGINDPRLRNPSDKFIYATVKQSSVDIYFRRQVELSTMYRHMEKHNYESAAEAIQAVRDNKLHAFIWDSAVLEFEASQKCDLVTTGELFFRSGFGIGMRKDSPWKQEVSLNILKSHENGFMEELDKTWVRYQECDSRSNAPATLTFENMAGVFMLVAGGIVAGIFLIFIEIA 5un9 A 2.5 BS01 NHT A 1 G67 K98 D174 D175 C215 Y219 T250 V254 W278 N280 D285 G9 K40 D116 D117 C157 Y161 T192 V196 W220 N222 D227 3.2.1.169 Ki=21nM remove_due_to_license_issue Ki=21nM, EC50=13nM, IC50=0.410000nM O60502 28319083 801 HFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKYSPQMALKLALTEWLQEFGVPHQYSSVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGRGGLAGEFQRLLPIDGAND 5un9 B 2.5 BS01 NHT B 1 G67 K98 D174 D175 C215 Y219 T250 V254 W278 N280 D285 N313 G9 K40 D116 D117 C157 Y161 T192 V196 W220 N222 D227 N255 3.2.1.169 Ki=21nM remove_due_to_license_issue Ki=21nM, EC50=13nM, IC50=0.410000nM O60502 28319083 801 HFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKYSPQMALKLALTEWLQEFGSVTLEDLQLLADLFYLPYEHGPKGAQMLREFQWLRANSSVVKIEEWRSRAAKFEEMCGLVMGMFTRLSNCANRTILYDMYSYVWDIKSIMSMVKSFVQWLGCRSHSSAQFLIGDQEPWAFRGGLAGEFQRLL 5unf A 2.8 BS01 8ES A 1 Y51 W100 Y103 L124 M128 F129 T178 R182 M214 K215 F272 I304 F308 Y109 W158 Y161 L182 M186 F187 T230 R234 M266 K267 F324 I356 F360 ? 0004930,0004945,0005506,0006954,0007186,0009055,0016020,0020037,0022900,0042597,0042981,0046872,0097746 remove_due_to_license_issue P0ABE7,P50052 28379944 1501 ADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAHLDAIPILYYIIFVIGFLVNIVVVTLFCCQKGPKKVSSIYIFNLAVADLLLLATLPLWATYYSYRYDWLFGPVMCKVFGSFLTLNMFASIFFITCMSVDRYQSVIYPFPWQASYIVPLVWCMACLSSLPTFYFRDVRTIEYLGVNACIMAFPPEKYAQWSAGIALMKNILGFIIPLIFIATCYFGIRKHLLKTNSYGKNRITRDQVLKMAAAVVLAFIICWLPFHVLTFLDALAWMGVINSCEVIAVIDLALPFAILLGFTNSCVNPFLYCFVGNRFQQKLRSVFR 5ung B 2.8 BS01 8ES B 1 Y51 W100 Y103 Y104 L124 T125 M128 F129 T178 R182 K215 F272 I304 F308 Y127 W176 Y179 Y180 L200 T201 M204 F205 T254 R258 K291 F348 I380 F384 ? 0004930,0004945,0005506,0006954,0007186,0009055,0016020,0020037,0022900,0042597,0042981,0046872,0097746 remove_due_to_license_issue P0ABE7,P50052 28379944 1201 ADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLGSGSCSQKPSDKHLDAIPILYYIIFVIGFLVNIVVVTLFCCQKGPKKVSSIYIFNLAVADLLLLATLPLWATYYSYRYDWLFGPVMCKVFGSFLTLNMFASIFFITCMSVDRYQSVIYPFLSQRRNPWQASYIVPLVWCMACLSSLPTFYFRDVRTIEYLGVNACIMAFPPEKYAQWSAGIALMKNILGFIIPLIFIATCYFGIRKHLLKTNSYGKNRITRDQVLKMAAAVVLAFIICWLPFHVLTFLDALAWMGVINSCEVIAVIDLALPFAILLGFTNSCVNPFLYCFVGNRFQQKLRSVFR 5unh A 2.9 BS01 8EM A 1 W100 Y103 L124 T125 M128 F129 T178 R182 M214 K215 W269 F272 I304 F308 W165 Y168 L189 T190 M193 F194 T232 R236 M268 K269 W321 F324 I356 F360 ? 0004930,0004945,0005506,0006954,0007186,0009055,0016020,0020037,0022900,0042597,0042981,0046872,0097746 remove_due_to_license_issue P0ABE7,P50052 28379944 1501 ADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLPSDKHLDAIPILYYIIFVIGFLVNIVVVTLFCCQKKVSSIYIFNLAVADLLLLATLPLWATYYSYRYDWLFGPVMCKVFGSFLTLNMFASIFFITCMSVDRYQSVIYASYIVPLVWCMACLSSLPTFYFRDVRTIEYLGVNACIMAFPPEKYAQWSAGIALMKNILGFIIPLIFIATCYFGIRKHLLKTYGKNRITRDQVLKMAAAVVLAFIICWLPFHVLTFLDALAWMGVINSCEVIAVIDLALPFAILLGFTNSCVNPFLYCFVGNRFQQKLRSVF 5unp A 2.92 BS01 8FY A 1 L169 G170 E171 V177 K193 F243 L246 G247 L297 V326 D327 L33 G34 E35 V41 K57 F107 L110 G111 L161 V190 D191 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P49760 2501 SRRAKSVEDDAEGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGARVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPIPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEEHHQLFDLIESMLEYEPAKRLTLGEALQHPFFARLR 5uoo A 1.69 BS01 8FV A 1 W374 P375 F376 L385 C429 N433 H437 V439 M442 W27 P28 F29 L38 C82 N86 H90 V92 M95 ? Ki=1.4nM remove_due_to_license_issue IC50=28nM, Ki=8.2nM, Kd=8.4nM O60885 28463487 501 SKVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMPDE 5uor A 2.75 BS01 8GV A 1 L686 V694 A707 K709 M754 E755 Q756 V757 G760 L810 D822 L16 V24 A37 K39 M84 E85 Q86 V87 G90 L140 D152 D803 K805 D807 N808 D822 T842 D133 K135 D137 N138 D152 T163 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue EC50=6.3nM, IC50=6.3nM Q99683 28337323 1002 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLFTGTLQYMAPEIIDYGKAADIWSLGCTIIEMATGKPPFYEAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 5uov A 1.33 BS01 8FP A 1 R8 D25 A28 D30 P81 V82 R8 D25 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.025nM remove_due_to_license_issue P03366 28434781 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5uov B 1.33 BS01 8FP A 1 D25 G27 D29 G48 I50 D25 G27 D29 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 28434781 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5uox A 2.5 BS01 8GY A 1 L686 V694 A707 K709 M754 E755 Q756 V757 G759 G760 D807 L810 S821 D822 L17 V25 A38 K40 M85 E86 Q87 V88 G90 G91 D138 L141 S152 D153 D803 K805 D807 N808 D822 T842 D134 K136 D138 N139 D153 T165 2.7.11.25 0004672,0005524,0006468 ic50=5.012nM remove_due_to_license_issue EC50=6.3nM, IC50=5.0nM Q99683 28337323 1000 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 5uoy A 1.82 BS02 8HM A 1 H373 L388 M389 F392 P408 L409 S420 Q421 F424 H224 L239 M240 F243 P259 L260 S271 Q272 F275 3.1.4.17 0004114,0007165,0008081 ic50=0.027uM remove_due_to_license_issue EC50=<100nM, IC50=<100.0nM Q01064 28406621 603 YSTAVLNCLKNLDLWCFDVFSLNQAADDHALRTIVFELLTRHNLISRFKIPTVFLMSFLDALETGYGKYKNPYHNQIHAADVTQTVHCFLLRTGMVHCLSEIELLAIIFAAAIHDYEHTGTTNSFHIQTKSECAIVYNDRSVLENHHISSVFRLMQDDEMNIFINLTKDEFVELRALVIEMVLATDMSCHFQQVKTMKTALQQLERIDKPKALSLLLHAADISHPTKQWLVHSRWTKALMEEFFRQGDKEAELGLPFSPLCDRTSTLVAQSQIGFIDFIVEPTFSVLTDVAEKSVPDVVSFRSTWVKRIQENKQKWKERAA 5uoy A 1.82 BS03 8HM A 2 Y150 R181 T182 F185 T201 M205 Y1 R32 T33 F36 T52 M56 3.1.4.17 0004114,0007165,0008081 ic50=0.027uM remove_due_to_license_issue EC50=<100nM, IC50=<100.0nM Q01064 28406621 604 YSTAVLNCLKNLDLWCFDVFSLNQAADDHALRTIVFELLTRHNLISRFKIPTVFLMSFLDALETGYGKYKNPYHNQIHAADVTQTVHCFLLRTGMVHCLSEIELLAIIFAAAIHDYEHTGTTNSFHIQTKSECAIVYNDRSVLENHHISSVFRLMQDDEMNIFINLTKDEFVELRALVIEMVLATDMSCHFQQVKTMKTALQQLERIDKPKALSLLLHAADISHPTKQWLVHSRWTKALMEEFFRQGDKEAELGLPFSPLCDRTSTLVAQSQIGFIDFIVEPTFSVLTDVAEKSVPDVVSFRSTWVKRIQENKQKWKERAA 5up0 A 2.04 BS02 8HP A 1 H373 L388 M389 L409 Q421 F424 H224 L239 M240 L260 Q272 F275 3.1.4.17 0004114,0007165,0008081 ic50=0.46uM remove_due_to_license_issue IC50=550nM Q01064 28406621 603 YSTAVLNCLKNLDLWCFDVFSLNQAADDHALRTIVFELLTRHNLISRFKIPTVFLMSFLDALETGYGKYKNPYHNQIHAADVTQTVHCFLLRTGMVHCLSEIELLAIIFAAAIHDYEHTGTTNSFHIQTKSECAIVYNDRSVLENHHISSVFRLMQDDEMNIFINLTKDEFVELRALVIEMVLATDMSCHFQQVKTMKTALQQLERIDKPKALSLLLHAADISHPTKQWLVHSRWTKALMEEFFRQGDKEAELGLPFSPLCDRTSTLVAQSQIGFIDFIVEPTFSVLTDVAEKSVPDVVSFRSTWVKRIQENKQKWKERAA 5up3 A 2.95 BS01 8GS A 1 L686 G687 K709 M754 E755 Q756 V757 G760 L810 S821 D822 L17 G18 K40 M80 E81 Q82 V83 G86 L136 S147 D148 D803 K805 D807 N808 D822 T842 D129 K131 D133 N134 D148 T160 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=13nM Q99683 28337323 1000 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 5upe A 1.93 BS01 8HY A 1 H191 F193 R196 D219 V242 A244 P273 S275 P307 R311 I351 H171 F173 R176 D199 V222 A224 P253 S255 P287 R291 I331 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Ki=9nM remove_due_to_license_issue P43490 28610984 901 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5upe B 1.93 BS01 8HY B 1 H191 F193 R196 D219 V242 A244 P273 S275 P307 I309 R311 I351 A379 H171 F173 R176 D199 V222 A224 P253 S255 P287 I289 R291 I331 A359 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Ki=9nM remove_due_to_license_issue P43490 28610984 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5upf A 1.69 BS01 8HV A 1 Y188 K189 H191 F193 R196 D219 V242 A244 S275 R311 R349 I351 A379 Y168 K169 H171 F173 R176 D199 V222 A224 S255 R291 R329 I331 A359 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Ki=2.5nM remove_due_to_license_issue P43490 28610984 901 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5upf B 1.69 BS01 8HV B 1 K189 H191 F193 R196 D219 V242 A244 S275 R311 R349 I351 A379 K169 H171 F173 R176 D199 V222 A224 S255 R291 R329 I331 A359 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 Ki=2.5nM remove_due_to_license_issue P43490 28610984 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5upj A 2.3 BS01 UIN B 1 D25 G27 A28 I50 I82 D25 G27 A28 I50 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 7783120 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTLEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 5upj B 2.3 BS01 UIN B 1 D25 G48 I50 D25 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=75nM remove_due_to_license_issue P04584 7783120 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTLEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 5upz A 1.27 BS01 8HD A 1 R8 D25 G27 A28 D30 V82 R8 D25 G27 A28 D30 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.63nM remove_due_to_license_issue P03366 28434781 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5upz B 1.27 BS01 8HD A 1 D25 G27 A28 D29 G48 G49 I50 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 28434781 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5uqv A 2.84 BS01 8JM A 1 Q297 C300 L304 D305 E308 I320 Y348 D349 H403 Q88 C91 L95 D96 E99 I111 Y139 D140 H194 N218 C223 H464 D481 N9 C14 H247 D264 3.4.19.12 0004843,0016579 remove_due_to_license_issue IC50=750nM, EC50=300nM Q93009 29045385 601 HTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQ 5uqx A 2.23 BS01 8JP A 1 Q297 C300 R301 D305 E308 Y348 D349 H403 Q89 C92 R93 D97 E100 Y140 D141 H195 N218 C223 H464 D481 N10 C15 H256 D273 3.4.19.12 0004843,0016579 Kd=246uM remove_due_to_license_issue IC50=1340nM, EC50=2580nM Q93009 29045385 601 KHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHDDDLSVRHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQK 5ur1 A 2.2 BS01 YY9 A 1 L484 V492 K514 E531 M535 V561 A564 G567 L630 A640 D641 L21 V28 K50 E67 M71 V97 A100 G103 L161 A171 D172 D623 A625 R627 N628 D641 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=1.06nM remove_due_to_license_issue IC50=1.1nM P11362 28521156 801 ELPEDPRWELPRDRLVLGKPLGEGFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 5ur5 A 1.93 BS01 8KP A 1 I62 A89 S92 E94 F108 H115 L117 Y120 F159 I58 A85 S88 E90 F104 H111 L113 Y116 F152 ? 0004864,0005515,0005634,0005737,0005773,0005829,0005886,0009705,0009738,0010427,0038023,0042802,0042803,0044389,0062049,0080163,1902584 remove_due_to_license_issue O49686 28949512 207 LTPEERSELKNSIAEFHTYQLDPGSCSSLHAQRIHAPPELVWSIVRRFDKPQTYKHFIKSCSVEQNFEMRVGCTRDVIVISGLPANTSTERLDILDDERRVTGFSIIGGEHRLTNYKSVTTVHRFEKENRIWTVVLESYVVDMPSEDDTRMFADTVVKLNLQKLATVAEAMARN 5ur6 A 1.631 BS01 8KM A 1 F61 A89 S92 E94 F108 I110 L117 Y120 V163 F60 A88 S91 E93 F107 I109 L116 Y119 V155 ? 0004864,0005515,0005634,0005737,0005773,0005829,0005886,0009705,0009738,0010427,0038023,0042802,0042803,0044389,0062049,0080163,1902584 ic50=87nM remove_due_to_license_issue O49686 28949512 207 PSELTPEERSELKNSIAEFHTYQLDPGSCSSLHAQRIHAPPELVWSIVRRFDKPQTYKHFIKSCSVEQNFEMRVGCTRDVIVISGLPANTSTERLDILDDERRVTGFSIIGGEHRLTNYKSVTTVHRFEKENRIWTVVLESYVVDMDTRMFADTVVKLNLQKLATVAEAMARN 5ur9 A 2.198 BS01 8KS A 1 L32 K61 T63 A78 L31 K60 T62 A77 ? 0001972,0005324,0005504,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0005886,0006006,0006629,0006656,0006869,0008289,0008544,0010829,0014069,0015908,0015909,0030667,0031392,0035360,0035578,0042593,0042802,0045202,0051930,0070062,0098921,0098978,0099092,0099178,0099524,0120162,1990379 Ki=0.9uM remove_due_to_license_issue Ki=810nM Q01469 28632393 201 ATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTLKTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVECVMNNVTCTRIYEKVE 5ura A 1.85002 BS01 8KS A 1 F17 M21 V26 T37 P39 S56 A76 D77 F105 M116 L118 Y129 F19 M23 V28 T39 P41 S58 A78 D79 F107 M118 L120 Y131 ? 0005504,0005515,0005634,0005737,0005829,0007399,0008285,0008289,0015908,0050673 Ki=0.4uM remove_due_to_license_issue Ki=450nM O15540 28632393 201 SHMVEAFCATWKLTNSQNFDEYMKALGVGFATRQVGNVTKPTVIISQEGDKVVIRTLSTFKNTEISFQLGEEFDETTADDRNCKSVVSLDGDKLVHIQKWDGKETNFVREIKDGKMVMTLTFGDVVAVRHYEKA 5urj A 2.75 BS01 8LS A 1 H1235 F1255 V1256 P1257 D1678 P1680 I1681 S1709 K1710 D1712 F1713 K1716 P1723 H826 F846 V847 P848 D1269 P1271 I1272 S1300 K1301 D1303 F1304 K1307 P1314 3.6.4.13 0003676,0005524 remove_due_to_license_issue O75643 28586220 2202 LAPRQVLDLEDLVFTQGSHFMANKRCQLPDGSFRRQRKGYEEVHVPALKPKPFGSEEQLLPVEKLPKYAQAGFEGFKTLNRIQSKLYRAALETDENLLLCAPTGAGKTNVALMCMLREIGKHINMDGTINVDDFKIIYIAPMRSLVQEMVGSFGKRLATYGITVAELTGEISATQIIVCTPEKWDIITRKGGERTYTQLVRLIILDEIHLLHDDRGPVLEALVARAIRNIEMTQEDVRLIGLSATLPNYEDVATFLRVDPAKGLFYFDNSFRPVPLEQTYVGITEKKAIKRFQIMNEIVYEKIMEHAGKNQVLVFVHSRKETGKTARAIRDMCLEKDTLGLFLREGSASTEVLRTEAEQCKNLELKDLLPYGFAIHHAGMTRVDRTLVEDLFADKHIQVLVSTATLAWGVNLPAHTVIIKGTQVYSPEKGRWTELGALDILQMLGRAGRPQYDTKGEGILITSHGELQYYLSLLNQQLPIESQMVSKLPDMLNAEIVLGNVQNAKDAVNWLGYAYLYIRMLRSPTLYGISHDDLKGDPLLDQRRLDLVHTAALMLDKNNLVKYDKKTGNFQVTELGRIASHYYITNDTVQTYNQLLKPTLSEIELFRVFSLSSEFKNITVREEEKLELQKLLERVPIPVKESIEEPSAKINVLLQAFISQLKLEGFALMADMVYVTQSAGRLMRAIFEIVLNRGWAQLTDKTLNLCKMIDKRMWQSMCPLRQFRKLPEEVVKKIEKKNFPFERLYDLNHNEIGELIRMPKMGKTIHKYVHLFPKLELSVHLQPITRSTLKVELTITPDFQWDEKVHGSSEAFWILVEDVDSEVILHHEYFLLKAKYAQDEHLITFFVPVFEPLPPQYFIRVVSDRWLSCETQLPVSFRHLILPEKYPPPTELLDLQPLPVSALRNSAFESLYQDKFPFFNPIQTQVFNTVYNSDDNVFVGAPTGSGKTICAEFAILRMLLQSSEGRCVYITPMEALAEQVYMDWYEKFQDRLNKKVVLLTGETSTDLKLLGKGNIIISTPEKWDILSRRWKQRKNVQNINLFVVDEVHLIGGENGPVLEVICSRMRYISSQIERPIRIVALSSSLSNAKDVAHWLGCSATSTFNFHPNVRPVPLELHIQGFNISHTQTRLLSMAKPVYHAITKHSPKKPVIVFVPSRKQTRLTAIDILTTCAADIQRQRFLHCTEKDLIPYLEKLSDSTLKETLLNGVGYLHEGLSPMERRLVEQLFSSGAIQVVVASRSLCWGMNVAAHLVIIMDTQYYNGKIHAYVDYPIYDVLQMVGHANRPLQDDEGRCVIMCQGSKKDFFKKFLYEPLPVESHLDHCMHDHFNAEIVTKTIENKQDAVDYLTWTFLYRRMTQNPNYYNLQGISHRHLSDHLSELVEQTLSDLEQSKCISIEDEMDVAPLNLGMIAAYYYINYTTIELFSMSLNAKTKVRGLIEIISNAAEYENIPIRHHEDNLLRQLAQKVPHKLNNPKFNDPHVKTNLLLQAHLSRMQLSAELQSDTEEILSKAIRLIQACVDVLSSNGWLSPALAAMELAQMVTQAMWSKDSYLKQLPHFTSEHIKRCTDESVFDIDEERNALLQLTDSQIADVARFCNRYPNIELSYEVVDKDSIRSGGPVVVLVQLEREEEVTGPVIAPLFPQKREEGWWVVIGDAKSNSLISIKRLTLQQKAKVKLDFVAPATGAHNYTLYFMSDAYMGCDQEYKFS 5urk A 2.95 BS01 8LP A 1 F1254 F1255 P1257 D1678 P1680 I1681 K1710 F1713 P1723 F847 F848 P850 D1271 P1273 I1274 K1303 F1306 P1316 3.6.4.13 0003676,0005524 remove_due_to_license_issue IC50=790nM O75643 28586220 2202 LAPRQVLDLEDLVFTQGSHFMANKRCQLPDGSFRRQRKGYEEVHVPALKPKPFGSEEQLLPVEKLPKYAQAGFEGFKTLNRIQSKLYRAALETDENLLLCAPTGAGKTNVALMCMLREIGKHINMDGTINVDDFKIIYIAPMRSLVQEMVGSFGKRLATYGITVAELTGKEEISATQIIVCTPEKWDIITRKGGERTYTQLVRLIILDEIHLLHDDRGPVLEALVARAIRNIEMTQEDVRLIGLSATLPNYEDVATFLRVDPAKGLFYFDNSFRPVPLEQTYVGITEKKAIKRFQIMNEIVYEKIMEHAGKNQVLVFVHSRKETGKTARAIRDMCLEKDTLGLFLREGSASTEVLRTEAEQCKNLELKDLLPYGFAIHHAGMTRVDRTLVEDLFADKHIQVLVSTATLAWGVNLPAHTVIIKGTQVYSPEKGRWTELGALDILQMLGRAGRPQYDTKGEGILITSHGELQYYLSLLNQQLPIESQMVSKLPDMLNAEIVLGNVQNAKDAVNWLGYAYLYIRMLRSPTLYGISHDDLKGDPLLDQRRLDLVHTAALMLDKNNLVKYDKKTGNFQVTELGRIASHYYITNDTVQTYNQLLKPTLSEIELFRVFSLSSEFKNITVREEEKLELQKLLERVPIPVKESIEEPSAKINVLLQAFISQLKLEGFALMADMVYVTQSAGRLMRAIFEIVLNRGWAQLTDKTLNLCKMIDKRMWQSMCPLRQFRKLPEEVVKKIEKKNFPFERLYDLNHNEIGELIRMPKMGKTIHKYVHLFPKLELSVHLQPITRSTLKVELTITPDFQWDEKVHGSSEAFWILVEDVDSEVILHHEYFLLKAKYAQDEHLITFFVPVFEPLPPQYFIRVVSDRWLSCETQLPVSFRHLILPEKYPPPTELLDLQPLPVSALRNSAFESLYQDKFPFFNPIQTQVFNTVYNSDDNVFVGAPTGSGKTICAEFAILRMLLQSSEGRCVYITPMEALAEQVYMDWYEKFQDRLNKKVVLLTGETSTDLKLLGKGNIIISTPEKWDILSRRWKQRKNVQNINLFVVDEVHLIGGENGPVLEVICSRMRYISSQIERPIRIVALSSSLSNAKDVAHWLGCSATSTFNFHPNVRPVPLELHIQGFNISHTQTRLLSMAKPVYHAITKHSPKKPVIVFVPSRKQTRLTAIDILTTCAADIQRQRFLHCTEKDLIPYLEKLSDSTLKETLLNGVGYLHEGLSPMERRLVEQLFSSGAIQVVVASRSLCWGMNVAAHLVIIMDTQYYNGKIHAYVDYPIYDVLQMVGHANRPLQDDEGRCVIMCQGSKKDFFKKFLYEPLPVESHLDHCMHDHFNAEIVTKTIENKQDAVDYLTWTFLYRRMTQNPNYYNLQGISHRHLSDHLSELVEQTLSDLEQSKCISIEDEMDVAPLNLGMIAAYYYINYTTIELFSMSLNAKTKVRGLIEIISNAAEYENIPIRHHEDNLLRQLAQKVPHKLNNPKFNDPHVKTNLLLQAHLSRMQLSAELQSDTEEILSKAIRLIQACVDVLSSNGWLSPALAAMELAQMVTQAMWSKDSYLKQLPHFTSEHIKRCTESVFDIERNALLQLTDSQIADVARFCNRYPNIELSYEVVDKDSIRSGGPVVVLVQLEREEEVTGPVIAPLFPQKREEGWWVVIGDAKSNSLISIKRLTLQQKAKVKLDFVAPATGAHNYTLYFMSDAYMGCDQEYKFS 5urm A 2.8 BS01 8LV A 1 M544 R545 S546 T589 E591 K592 I595 T814 M141 R142 S143 T186 E188 K189 I192 T411 3.6.4.13 0003676,0005524 remove_due_to_license_issue O75643 28586220 2501 APRQVLDLEDLVFTQGSHFMANKRCQLPDGSFRRQRKGYEEVHVPALKPKPFGSEEQLLPVEKLPKYAQAGFEGFKTLNRIQSKLYRAALETDENLLLCAPTGAGKTNVALMCMLREIGKHINMDGTINVDDFKIIYIAPMRSLVQEMVGSFGKRLATYGITVAELTGDHQLCKEEISATQIIVCTPEKWDIITRKGGERTYTQLVRLIILDEIHLLHDDRGPVLEALVARAIRNIEMTQEDVRLIGLSATLPNYEDVATFLRVDPAKGLFYFDNSFRPVPLEQTYVGITEKKAIKRFQIMNEIVYEKIMEHAGKNQVLVFVHSRKETGKTARAIRDMCLEKDTLGLFLREGSASTEVLRTEAEQCKNLELKDLLPYGFAIHHAGMTRVDRTLVEDLFADKHIQVLVSTATLAWGVNLPAHTVIIKGTQVYSPEKGRWTELGALDILQMLGRAGRPQYDTKGEGILITSHGELQYYLSLLNQQLPIESQMVSKLPDMLNAEIVLGNVQNAKDAVNWLGYAYLYIRMLRSPTLYGISHDDLKGDPLLDQRRLDLVHTAALMLDKNNLVKYDKKTGNFQVTELGRIASHYYITNDTVQTYNQLLKPTLSEIELFRVFSLSSEFKNITVREEEKLELQKLLERVPIPVKESIEEPSAKINVLLQAFISQLKLEGFALMADMVYVTQSAGRLMRAIFEIVLNRGWAQLTDKTLNLCKMIDKRMWQSMCPLRQFRKLPEEVVKKIEKKNFPFERLYDLNHNEIGELIRMPKMGKTIHKYVHLFPKLELSVHLQPITRSTLKVELTITPDFQWDEKVHGSSEAFWILVEDVDSEVILHHEYFLLKAKYAQDEHLITFFVPVFEPLPPQYFIRVVSDRWLSCETQLPVSFRHLILPEKYPPPTELLDLQPLPVSALRNSAFESLYQDKFPFFNPIQTQVFNTVYNSDDNVFVGAPTGSGKTICAEFAILRMLLQSSEGRCVYITPMEALAEQVYMDWYEKFQDRLNKKVVLLTGETSTDLKLLGKGNIIISTPEKWDILSRRWKQRKNVQNINLFVVDEVHLIGGENGPVLEVICSRMRYISSQIERPIRIVALSSSLSNAKDVAHWLGCSATSTFNFHPNVRPVPLELHIQGFNISHTQTRLLSMAKPVYHAITKHSPKKPVIVFVPSRKQTRLTAIDILTTCAADIQRQRFLHCTEKDLIPYLEKLSDSTLKETLLNGVGYLHEGLSPMERRLVEQLFSSGAIQVVVASRSLCWGMNVAAHLVIIMDTQYYNGKIHAYVDYPIYDVLQMVGHANRPLQDDEGRCVIMCQGSKKDFFKKFLYEPLPVESHLDHCMHDHFNAEIVTKTIENKQDAVDYLTWTFLYRRMTQNPNYYNLQGISHRHLSDHLSELVEQTLSDLEQSKCISIEDEMDVAPLNLGMIAAYYYINYTTIELFSMSLNAKTKVRGLIEIISNAAEYENIPIRHHEDNLLRQLAQKVPHKLNNPKFNDPHVKTNLLLQAHLSRMQLSAELQSDTEEILSKAIRLIQACVDVLSSNGWLSPALAAMELAQMVTQAMWSKDSYLKQLPHFTSEHIKRCTESVFDIMEMEDEERNALLQLTDSQIADVARFCNRYPNIELSYEVVDKDSIRSGGPVVVLVQLEREEEVTGPVIAPLFPQKREEGWWVVIGDAKSNSLISIKRLTLQQKAKVKLDFVAPATGAHNYTLYFMSDAYMGCDQEYKFSVD 5usf A 2.75 BS01 YSA A 1 Y36 D37 G38 E40 A48 Q49 W70 F75 Y163 Q167 D170 L181 G182 Q185 H210 M212 L213 Y38 D39 G40 E42 A50 Q51 W72 F77 Y165 Q169 D172 L183 G184 Q187 H212 M214 L215 6.1.1.1 0000166,0004812,0004831,0005524,0005737,0006412,0006418,0006437 remove_due_to_license_issue A0A3Q8ID88 28427904 701 GSMNTDERYKLLRSVGEECIQESELRNLIEKKPLIRCYDGFEPSGRMHIAQGIFKAVNVNKCTAAGCEFVFWVADWFALMNDKVGGELEKIRIVGRYLIEVWKAAGMDTDKVLFLWSSEEITSHADTYWRMVLDIGRQNTIARIKKCCTIMGKTEGTLTAAQVLYPLMQCCDIFFLKADICQLGLDQRKVNMLAREYCDLIGRKLKPVILSHHMLAGLRRGQAKMSKSDPDSAIFMEDTEEDVARKIRQAYCPRVKQSASAITDDGAPVATDDRNPVLDYFQCVVYARPGAVAAIDGTTYATYEDLEQAFVSDEVSEDALKSCLIDEVNALLAPVRQHFASNEEAHELLEAVKSYRKGGATLPLAETALPAAPEKPHACMWMPALLKVPLDVAEGMIKATEDFIAAHPGGTVTVVLPDWSAVASDEITGVEKDISAALQVNCALLKAYGLPNSVKIVTENEVILGNRNDFWVSVIGIARKNLLSHIEELYGGELRNAGQVIAALMRVATALMLSVSHVISTSLDGHINAFAREYTKERIECVQTLEGRIPALHRPGAAPAVLGADDVLYLDDNDMDIRRKIKKAYSAPNEEANPVISVAQHLLAQHGALNIERGEANGGNVSYNTPEALVADCGSGALHPADLKAAVLQLLLDRSAQARALLNGELKKNMTALRNAEKKMAK 5usq A 2.55 BS01 8LY A 1 I211 A230 K232 Y249 L278 V279 S280 Y282 H283 D290 L340 D351 I12 A31 K33 Y50 L79 V80 S81 Y83 H84 D91 L141 D152 D333 K335 N338 D351 T375 D134 K136 N139 D152 T176 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue EC50=1000nM, IC50=100nM P36897 28359790 500 TIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQ 5usy A 2.0 BS01 SKE A 1 L855 V863 M929 Y931 L932 G935 L983 L16 V24 M90 Y92 L93 G96 L144 D976 A978 R980 N981 D994 S1016 D137 A139 R141 N142 D155 S174 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Kd=220nM, IC50=2960nM, Ki=220000nM O60674 28626521 1201 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 5usz A 2.103 BS01 SKE A 1 I559 L579 K581 Q626 F628 V629 K630 G632 S633 K677 L680 S698 I23 L43 K45 Q90 F92 V93 K94 G96 S97 K141 L144 S162 N673 K677 N678 D699 N137 K141 N142 D163 2.7.10.2 0004672,0005524,0006468 Kd=106nM remove_due_to_license_issue Kd=220nM, IC50=2960nM, Ki=220000nM O60674 28626521 901 FHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSL 5ut0 A 2.102 BS01 35R A 1 L551 L579 F628 V629 K630 F631 G632 L680 L15 L43 F92 V93 K94 F95 G96 L144 N673 K677 N678 D699 N137 K141 N142 D163 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue Kd=11nM O60674 28626521 903 FHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSL 5ut4 A 2.0 BS01 DQX A 1 L551 I559 L579 F628 V629 K630 F631 G632 S633 T636 L680 S698 L15 I23 L43 F92 V93 K94 F95 G96 S97 T100 L144 S162 N673 K677 N678 D699 N137 K141 N142 D163 2.7.10.2 0004672,0005524,0006468 Kd=42uM remove_due_to_license_issue Kd=42000nM, IC50=7.3nM O60674 28626520 901 FHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSLF 5ut6 A 1.645 BS01 8MY A 1 L551 L579 Q626 F628 V629 K630 G632 S633 K677 L680 L15 L43 Q90 F92 V93 K94 G96 S97 K141 L144 N673 K677 N678 D699 N137 K141 N142 D163 2.7.10.2 0004672,0005524,0006468 Kd=57.3uM remove_due_to_license_issue Kd=57300nM O60674 28626520 901 FHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSL 5uuu A 2.7 BS01 QRW A 1 R199 G200 F202 G203 V205 A218 K220 L222 L235 A236 E239 M274 L324 G337 R88 G89 F91 G92 V94 A107 K109 L111 L124 A125 E128 M163 L213 G226 D317 K319 N322 D335 K344 T353 D206 K208 N211 D224 K233 T242 2.7.11.15 0004672,0004674,0004703,0005524,0006468,0007165 remove_due_to_license_issue EC50=10000nM, IC50=18nM P25098 28699740 601 KILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVEDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEA 5uv1 A 2.4 BS03 0FV A 1 W315 I336 D343 T446 F484 R485 D488 W248 I269 D276 T379 F417 R418 D421 R306 W315 I336 D343 D347 S444 I445 T446 R485 D488 T492 Y565 R239 W248 I269 D276 D280 S377 I378 T379 R418 D421 T425 Y492 4.2.3.20 0000287,0006720,0009507,0010333,0016102,0016114,0016829,0034002,0046872 Ki=2.4uM remove_due_to_license_issue A0A1C9J6A7 28272876 704 SIWDHDFLQSLNSNYTDETYKRRAEELKGKVKTAIKDVTEPLDQLELIDNLQRLGLAYHFEPEIRNILRNIHNHNKDYNWRKENLYATSLEFRLLRQHGYPVSQEVFSGFKDDKVGFICDDFKGILSLHEASYYSLEGESIMEEAWQFTSKHLKEMMIDVFVAEQAKRALELPLHWKAPMLEARWFIHVYEKREDKNHLLLELAKLEFNTLQAIYQEELKDISGWWKDTGLGEKLSFARNRLVASFLWSMGIAFEPQFAYCRRVLTISIALITVIDDIYDVYGTLDELEIFTDAVARWDINYALKHLPGYMKMCFLALYNFVNEFAYYVLKQQDFDMLLSIKHAWLGLIQAYLVEAKWYHSKYTPKLEEYLENGLVSITGPLIITISYLSGTNPIIKKELEFLESNPDIVHWSSKIFRLQDDLGTSSDVPKSIQCYMHETGASEEVAREHIKDMMRQMWKKVNAYTADKDSPLTRTTAEFLLNLVRMSHFMYLHGDVGFTLLFQPIPL 5uv2 A 2.2 BS03 LA6 A 1 W315 I336 T340 D343 I445 F484 R485 D488 K504 W248 I269 T273 D276 I378 F417 R418 D421 K437 R306 W315 I336 D343 D347 S444 I445 T446 R485 D488 T492 E496 Y565 R239 W248 I269 D276 D280 S377 I378 T379 R418 D421 T425 E429 Y498 4.2.3.20 0000287,0006720,0009507,0010333,0016102,0016114,0016829,0034002,0046872 Ki=39.5uM remove_due_to_license_issue A0A1C9J6A7 28272876 704 SIWDHDFLQSLNSNYTDETYKRRAEELKGKVKTAIKDVTEPLDQLELIDNLQRLGLAYHFEPEIRNILRNIHNHNKDYNWRKENLYATSLEFRLLRQHGYPVSQEVFSGFKDDKVGFICDDFKGILSLHEASYYSLEGESIMEEAWQFTSKHLKEMMIDVFVAEQAKRALELPLHWKAPMLEARWFIHVYEKREDKNHLLLELAKLEFNTLQAIYQEELKDISGWWKDTGLGEKLSFARNRLVASFLWSMGIAFEPQFAYCRRVLTISIALITVIDDIYDVYGTLDELEIFTDAVARWDINYALKHLPGYMKMCFLALYNFVNEFAYYVLKQQDFDMLLSIKHAWLGLIQAYLVEAKWYHSKYTPKLEEYLENGLVSITGPLIITISYLSGTNPIIKKELEFLESNPDIVHWSSKIFRLQDDLGTSSDEIQRGDVPKSIQCYMHETGASEEVAREHIKDMMRQMWKKVNAYTADKDSPLTRTTAEFLLNLVRMSHFMYLHGDVGFTLLFQPIPL 5uv5 A 3.0 BS03 Y55 A 1 D498 Q500 H539 D479 Q481 H520 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28760905 603 PIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFARKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFKKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVS 5uvc A 2.65 BS01 8PV A 1 G200 V205 A218 K220 M274 L324 D335 G144 V149 A162 K164 M218 L268 D279 D317 K319 N322 D335 K344 T353 D261 K263 N266 D279 K288 T297 2.7.11.15 0004672,0004674,0004703,0005524,0006468,0007165 remove_due_to_license_issue P25098 28699740 600 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLEVARSREIFDSYIMKELLAPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRL 5uwf C 1.87 BS01 8Q7 C 1 Y524 H525 L675 V678 I692 Y693 F696 I711 M713 Q726 F729 Y79 H80 L230 V233 I247 Y248 F251 I266 M268 Q281 F284 3.1.4.17 0004114,0007165,0008081 ic50=0.059uM remove_due_to_license_issue IC50=59nM Q9Y233 28406621 801 SMASICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRG 5uwk A 1.6 BS06 8OM A 1 L184 L185 A186 H222 E223 H226 H232 L239 F241 I243 Y244 T245 T247 P255 L78 L79 A80 H116 E117 H120 H126 L133 F135 I137 Y138 T139 T141 P146 H222 E223 H226 H232 H116 E117 H120 H126 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=2.3nM remove_due_to_license_issue IC50=2.2nM, Ki=2.3nM P45452 28653849 306 FPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGFMLPDDDVQGIQSLYGPG 5uwl A 2.55 BS06 8OJ A 1 G183 L184 L185 Y214 L218 H222 E223 L239 F241 P242 I243 Y244 T245 T247 P255 G74 L75 L76 Y105 L109 H113 E114 L130 F132 P133 I134 Y135 T136 T138 P146 H222 E223 H226 H232 H113 E114 H117 H123 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=9.4nM P45452 28653849 306 TLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 5uwm A 1.62 BS07 8OA A 1 G183 L184 L185 H222 E223 L239 F241 P242 I243 Y244 T245 T247 F252 P255 G73 L74 L75 H112 E113 L129 F131 P132 I133 Y134 T135 T137 F139 P142 H222 E223 H226 H232 H112 E113 H116 H122 3.4.24.- 0004222,0006508,0008237,0008270,0031012 ic50=356nM remove_due_to_license_issue IC50=356nM P45452 28653849 306 LKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTHFMLPDDDVQGIQSLYGP 5uwn A 3.2 BS05 8O7 A 1 L184 L185 L218 H222 E223 F241 P242 I243 Y244 T245 T247 P255 L76 L77 L110 H114 E115 F133 P134 I135 Y136 T137 T139 P147 H222 E223 H226 H232 H114 E115 H118 H124 3.4.24.- 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue Ki=14nM, IC50=8.3nM P45452 28653849 305 RTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTGKSHFMLPDDDVQGIQSLYGPG 5ux4 A 2.805 BS01 3UT A 1 D33 I76 Y78 I129 D226 G228 D33 I76 Y78 I126 D223 G225 3.4.23.5 0000045,0004175,0004190,0005576,0005615,0005764,0005765,0006508,0008233,0010008,0016787,0030163,0031667,0031904,0038020,0042159,0042277,0042470,0043065,0045121,0060441,0070001,0070201,0098830,0098982,0099003,0099532,1901143 remove_due_to_license_issue P24268 30108829 404 EPVSELLKNYLDAQYYGEIGIGTPPQCFTVVFDTGSSNLWVPSIHCKLLDIACWVHHKYNSDKSSTYVKNGTSFDIHYGSGSLSGYLSQDTVSVPCKGGIKVEKQIFGEATKQPGVVFIAAKFDGILGMGYPFISVNNVLPVFDNLMKQKLVEKNIFSFYLNRDPTGQPGGELMLGGTDSRYYHGELSYLNVTRKAYWQVHMDQLEVGSELTLCKGGCEAIVDTGTSLLVGPVDEVKELQKAIGAVPLIQGEYMIPCEKVSSLPIITFKLGGQNYELHPEKYILKVSKTICLSGFMGMDIPPPSGPLWILGDVFIGCYYTVFDREYNRVGFAKAATL 5uxf A 1.501 BS01 2BA A 1 Y24 G217 L219 T221 A253 Q270 S271 E276 N280 L306 Y27 G220 L222 T224 A246 Q263 S264 E269 N273 L299 D50 Y55 K84 H117 D53 Y58 K87 H120 1.1.1.- 0004033,0006805,0016491 Kd=87nM remove_due_to_license_issue Q8VC28 28329705 401 FQGMSSKQHCVKLNDGHLIPALGFGTYKPKEVPKSKSLEAACLALDVGYRHVDTAYAYQVEEEIGQAIQSAIAAGVVKREDLFVTTKLWCTCFRPELVKPALEKSLKKLQLDYVDLYIMHYPVPMKSGDNDFPVNEQGKSLLDTVDFCDTWERLEECKDAGLVKSIGVSNFNHRQLERILNKPGLKYKPVCNQVECHLYLNQRKLLDYCESKDIVLVAYGALGTSPVLLNDPVLCDVAKKNKRSPALIALRYLIQRGIVPLAQSFKENEMRENLQVFGFQLSPEDMKTLDGLNKNFRYLPAEFLVDHPEYPFVEEY 5uxm A 1.54 BS02 TRP A 1 V93 K105 A177 L179 Q223 E226 V90 K102 A174 L176 Q220 E223 2.5.1.54 0003849,0009073,0016740 Kd=3.6uM remove_due_to_license_issue Q9I000 29608284 502 SWSPESWRAKPIQQQPEYPDAAHLARVEQTLAGYPPLVFAGEARELRRQFAEVTAGRAFLLQGGDCAESFAEFSAAKIRDTFKVLLQMAVVMTFAAGCPVVKVGRMAGQFAKPRSSGDETQNGVTLPAYRGDIVNGIGFDEKSRVPDPERLLQAYHQSTASLNLLRAFAQGGFADLHQVHRWNLDFIANSALAERYQQLADRIDETLAFMRACGLDSAPQLRETSFFTAHEALLLNYEEALTRRDSLTGEWYDCSAHMLWIGDRTRQIDGAHVEMLRGVGNPIGVKVGPSMDSEELIRLIDILNPDNDPGRLNLIVRMGADKVGDHLPRLIQAIQREGRQVLWSSDPMHGNTIKASSGYKTRDFARVLAEVRQFFEVHQAEGSYAGGIHIEMTGQNVTECIGGSRPITEDGLSDRYHTHCDPRLNADQSLELAFLIAETLKQVRR 5uxn A 2.2 BS05 TYR A 1 A177 L179 Q223 E226 T227 A174 L176 Q220 E223 T224 2.5.1.54 0003849,0009073,0016740 Kd=23uM remove_due_to_license_issue Q9I000 29608284 505 SWSPESWRAKPIQQQPEYPDAAHLARVEQTLAGYPPLVFAGEARELRRQFAEVTAGRAFLLQGGDCAESFAEFSAAKIRDTFKVLLQMAVVMTFAAGCPVVKVGRMAGQFAKPRSSGDETQNGVTLPAYRGDIVNGIGFDEKSRVPDPERLLQAYHQSTASLNLLRAFAQGGFADLHQVHRWNLDFIANSALAERYQQLADRIDETLAFMRACGLDSAPQLRETSFFTAHEALLLNYEEALTRRDSLTGEWYDCSAHMLWIGDRTRQIDGAHVEMLRGVGNPIGVKVGPSMDSEELIRLIDILNPDNDPGRLNLIVRMGADKVGDHLPRLIQAIQREGRQVLWSSDPMHGNTIKASSGYKTRDFARVLAEVRQFFEVHQAEGSYAGGIHIEMTGQNVTECIGGSRPITEDGLSDRYHTHCDPRLNADQSLELAFLIAETLKQVRR 5uy8 A 2.39 BS01 8UM A 1 K266 M312 S313 F315 D339 K358 N489 K263 M309 S310 F312 D336 K355 N486 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 ic50<5nM remove_due_to_license_issue EC50=4.0nM, IC50=<5.0nM P31939 29072452 601 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uy8 A 2.39 BS05 8UM B 1 N431 S450 R451 I452 P543 F544 D546 N547 N428 S447 R448 I449 P540 F541 D543 N544 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 ic50<5nM remove_due_to_license_issue EC50=4.0nM, IC50=<5.0nM P31939 29072452 601 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uy8 B 2.39 BS01 8UM A 1 N431 S450 R451 I452 P543 F544 D546 N547 N428 S447 R448 I449 P540 F541 D543 N544 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 ic50<5nM remove_due_to_license_issue EC50=4.0nM, IC50=<5.0nM P31939 29072452 601 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uy8 B 2.39 BS03 8UM B 1 K266 M312 S313 F315 D339 K358 N489 K263 M309 S310 F312 D336 K355 N486 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 ic50<5nM remove_due_to_license_issue EC50=4.0nM, IC50=<5.0nM P31939 29072452 601 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uyu A 1.9 BS01 8QV A 1 G11 Q12 G13 L30 D32 G34 S35 Y71 F108 I110 W115 I118 R128 D228 S229 G230 T231 T232 G13 Q14 G15 L32 D34 G36 S37 Y73 F110 I112 W117 I120 R130 D220 S221 G222 T223 T224 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D220 T223 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 30108829 406 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5uz0 A 1.79 BS04 8US B 1 S450 R451 I452 P543 F544 D546 S447 R448 I449 P540 F541 D543 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue EC50=7.6nM, IC50=16nM P31939 29072452 601 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uz0 A 1.79 BS05 8US B 2 K266 M312 S313 F315 D339 K263 M309 S310 F312 D336 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 remove_due_to_license_issue EC50=7.6nM, IC50=16nM P31939 29072452 602 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uz0 B 1.79 BS02 8US B 1 K266 M312 S313 F315 D339 N489 K263 M309 S310 F312 D336 N486 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 ic50=16nM remove_due_to_license_issue EC50=7.6nM, IC50=16nM P31939 29072452 601 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uz0 B 1.79 BS03 8US B 2 N431 S450 R451 I452 P543 F544 D546 N547 N428 S447 R448 I449 P540 F541 D543 N544 2.1.2.3,3.5.4.10 0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761 ic50=16nM remove_due_to_license_issue EC50=7.6nM, IC50=16nM P31939 29072452 602 GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH 5uzj A 3.3 BS01 8UV A 1 G85 F87 G88 E89 V90 A103 K105 L107 Y155 M156 L205 D216 G80 F82 G83 E84 V85 A98 K100 L102 Y146 M147 L196 D207 D198 K200 N203 D216 T237 D189 K191 N194 D207 T228 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Ki=170nM Q13464 30082069 501 SFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEETFPIPKAFVGNQLPFVGFTYYSNRRY 5uzk A 2.3 BS02 504 A 1 L49 G52 S53 F54 G55 R56 V57 A70 K72 V104 M120 Y122 V123 D166 L173 T183 D184 G186 F187 F327 L36 G39 S40 F41 G42 R43 V44 A57 K59 V91 M107 Y109 V110 D153 L160 T170 D171 G173 F174 F314 D166 K168 N171 D184 T201 D153 K155 N158 D171 T188 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 Ki=180nM remove_due_to_license_issue P17612 30082069 401 SVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 5v0l A 4.0 BS01 dna C 0 R91 H94 R102 K128 R11 H14 R22 K48 ? 0003700,0005634,0005667,0005737,0006355,0046983 remove_due_to_license_issue P27540 28396409 4 ~ 20 QSSADKERLARENHSEIERRRRNKMTAYITELSDMVPTCSALARKPDKLTILRMAVSHMKSLKPSFLTDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPQPQSEWFGSTLYDQVHPDDVDKLREQLSGSRRSFICRMRCEPHFVVVHCTGYDDDPEAGQGSKFCLVAIGRLQ 5v0l B 4.0 BS01 dna C 0 R37 H38 R39 R1 H2 R3 ? 0003700,0005634,0005667,0005737,0006355,0006805,0009410,0046983 remove_due_to_license_issue P30561 28396409 4 ~ 20 RHRDRLNTELDRLASLLPFPQDVINKLDKLSVLRLSVSYLRAKSFFDVALKSTQEGEFLLQALVLVVTADALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQLHWALDQLPPENASFMERCFRCDNSSGFLAMNFQGRLKYLHLPPQLALFAIATPL 5v0l B 4.0 BS02 dna D 0 R39 K65 R3 K29 ? 0003700,0005634,0005667,0005737,0006355,0006805,0009410,0046983 remove_due_to_license_issue P30561 28396409 4 ~ 17 RHRDRLNTELDRLASLLPFPQDVINKLDKLSVLRLSVSYLRAKSFFDVALKSTQEGEFLLQALVLVVTADALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQLHWALDQLPPENASFMERCFRCDNSSGFLAMNFQGRLKYLHLPPQLALFAIATPL 5v0n A 2.155 BS01 8W4 A 1 G11 L30 D32 G34 S35 Y71 T72 Q73 F108 I118 Y198 D228 G230 T231 T232 N233 G13 L32 D34 G36 S37 Y73 T74 Q75 F110 I120 Y191 D221 G223 T224 T225 N226 D32 S35 N37 A39 Y71 D228 T231 D34 S37 N39 A41 Y73 D221 T224 3.4.23.46 0004190,0006508,0016020 Ki=67.1nM remove_due_to_license_issue Ki=67nM, EC50=19nM P56817 28427814 404 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 5v0q A 2.4 BS01 dna B 0 R32 R42 R44 T70 N72 H80 R83 F84 H122 L123 G177 E178 G179 H180 E184 K187 E201 A203 Q204 H205 R232 W234 R236 K262 N298 K299 R26 R32 R34 T60 N62 H70 R73 F74 H112 L113 G167 E168 G169 H170 E174 K177 E191 A193 Q194 H195 R222 W224 R226 K252 N288 K289 0004519 remove_due_to_license_issue 28873986 -1 ~ 24 RESINPWILTGFADAEGSFGLYIYNRNRYTTRLRFTITLHNKDKSILENIQSTWKVGIITNNGDNAVSLHVSRFEDLKVIIDHFEKYPLITQKLGDYKLFKQAFSVMENKEHLKENGIKELVRIKAKMNWGLTDELKKAFPGNISRERPLINKNIPNFKWLAGFTSGEGHFGVELIKNSRNSRVHVRLRFEIAQHVRDKNLMNSLITYLGCGYIYEQNYSERSWLRFSVSKFSDINDKIIPVFQENTLIGVKLEDFEDWCKVAKLIEEKKHLTESGLDEIKKIKLNMNKGR 5v0q A 2.4 BS02 dna C 0 A21 E22 S24 Y28 Y30 T48 L49 H50 N139 W140 T143 R190 H195 R197 R199 Y223 Y225 Q227 Y229 W234 R236 F242 H281 A15 E16 S18 Y22 Y24 T38 L39 H40 N129 W130 T133 R180 H185 R187 R189 Y213 Y215 Q217 Y219 W224 R226 F232 H271 0004519 remove_due_to_license_issue 28873986 1 ~ 26 RESINPWILTGFADAEGSFGLYIYNRNRYTTRLRFTITLHNKDKSILENIQSTWKVGIITNNGDNAVSLHVSRFEDLKVIIDHFEKYPLITQKLGDYKLFKQAFSVMENKEHLKENGIKELVRIKAKMNWGLTDELKKAFPGNISRERPLINKNIPNFKWLAGFTSGEGHFGVELIKNSRNSRVHVRLRFEIAQHVRDKNLMNSLITYLGCGYIYEQNYSERSWLRFSVSKFSDINDKIIPVFQENTLIGVKLEDFEDWCKVAKLIEEKKHLTESGLDEIKKIKLNMNKGR 5v13 B 1.84 BS01 JH3 B 1 Y33 V51 W53 Y64 Y129 F269 Y14 V32 W34 Y45 Y110 F248 ? 0005549,0005576,0005615,0007608 Kd=23.3nM remove_due_to_license_issue Q16Y94 28751377 301 EWQPRTPEQTLYAYVRCLNDSSASIEQKINWVKWHPDTTYESQCYVKCVSEELRLYDPKEKRFRPERFVLQAESFFHADPEQLQALKNNAEPMLAGVLADNSCESVFNKYATFYATHHSTILRMFHGDYRDIGNTYAKLGNGVKQIGQMFVDFCEKRTDFKWNEDNSCPPEAFLDCVFRGFRWITEEGEVNVNEIRRDYEAAGKGAADMADYCGSVGARQLYNCLRDKGADSLVAVIRDRNQKTAFYFDLSSKEEPWKSAVDFANNL 5v19 A 3.1 BS01 8V4 A 1 M754 Q756 V757 G760 L810 M78 Q80 V81 G84 L134 D803 K805 D807 N808 D822 T842 D127 K129 D131 N132 D146 T158 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue Q99683 28291695 1000 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYEAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 5v1b A 2.49 BS02 8UY A 1 Y287 Y294 H297 I311 Y313 H358 V360 R367 A369 Y110 Y117 H120 I134 Y136 H181 V183 R190 A192 1.14.11.-,1.14.11.29 0005506,0016705,0031418 ic50=0.034uM remove_due_to_license_issue IC50=34.0nM Q96KS0 28594552 504 PSAPERLALDYIVPCMRYYGICVVDSFLGAALGGRVLAEVEALKRGGRLRQLVSPRSIRGDQIAWVEGHEPGCRSIGALMAHVDAVIRHCAGRLGSYKINGRTKAMVACYPGNGLGYVRHVDNPHGDGRCITCIYYLNQNWDVKVHGGLLQIFPEGRPVVANIEPLFDRLLIFWSDRRNPHEVKPAYATRYAITVWYFDADERARAKDKYQLASGQKGVQVPVSQP 5v24 A 2.5 BS01 8V7 A 1 L686 G687 K688 V694 K709 M754 Q756 V757 L810 D822 L16 G17 K18 V24 K39 M80 Q82 V83 L136 D148 D803 K805 D807 N808 D822 T842 D129 K131 D133 N134 D148 T159 2.7.11.25 0004672,0005524,0006468 ic50=400nM remove_due_to_license_issue IC50=400nM Q99683 28291695 1000 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLFTGTLQYMAPEIIDYGKAADIWSLGCTIIEMATGKPPFYEEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 5v2l A 2.1 BS01 ATP A 1 F57 V72 S93 N95 A104 G109 F58 V73 S94 N96 A105 G110 4.1.1.33 0004163,0005524,0005829,0006629,0008299,0016301,0016829,0016831,0019287 remove_due_to_license_issue Q837E0 29025876 401 AMLSGKARAHTNIALIKYWGKANEEYILPMNSSLSLTLDAFYTETTVTFDAHYSEDVFILNGILQNEKQTKKVKEFLNLVRQQADCTWFAKVESQNFVPTAAGLASSASGLAALAGACNVALGLNLSAKDLSRLARRGSGSACRSIFGGFAQWNKGHSDETSFAENIPANNWENELAMLFILINSSRDGMKRTVETSSFYQGWLDNVEKDLSQVHEAIKTKDFPRLGEIIEANGLRMHGTTLGAVPPFTYWSPGSLQAMALVRQARAKGIPCYFTMDAGPNVKVLVEKKNLEALKTFLSEHFSKEQLVPAFAGPGIELFET 5v35 A 2.5 BS01 FAR A 1 F37 M59 I61 L100 F149 F30 M52 I54 L93 F142 ? 0003755 remove_due_to_license_issue Q9NZN9 28739921 201 NVEGVKKTILHGGTGELPNFITGSRVIFHFRTMKCDEERTVIDDSRQVGQPMHIIIGNMFKLEFWEILLTSMRVHEVAEFWCDTIHTGVYPILSRSLRQMAQGKDPTEWHVHTCGLANMFAYHTLGYEDLDELQKEPQPLVFVIELLQVDAP 5v3o C 3.2 BS01 8W7 C 1 N351 P352 E377 H378 S379 W380 W386 W400 F402 N286 P287 E312 H313 S314 W315 W321 W335 F337 ? 0005515,0005634,0005737,0005829,0016020,0016567,0030177,0031333,0031334,0031464,0034766,0035641,0043161,0044325,0046872,0048471 remove_due_to_license_issue Q96SW2 28425720 501 INFDTSLPTSHTYLGADMEEFHGRTLHDDDSCQVIPVLPQVMMILIPGQTLPLQLFHPQEVSMVRNLIQKDRTFAVLAYSAQFGTTAEIYAYREEQDFGIEIVKVKAIGRQRFKVLELRTQSDGIQQAKVQILPECVLPSTMSAVQLESLNKCQIFPSSYKWWQKYQKRKFHCANLTSWPRWLYSLYDAETLMDRIKKQLREWDDDSLPSNPIDFSYRVAACLPIDDVLRIQLLKIGSAIQRLRCELDIMNKCTSLCCKQCQETEITTKNEIFSLSLCGPMAAYVNPHGYVHETLTVYKACNLNLIGRPSTEHSWFPGYAWTVAQCKICASHIGWKFTATKKDMSPQKFWGLTRSALLPTIPD 5v3x A 1.936 BS01 I28 A 1 Q1633 S1636 Y1637 N1640 I1643 D1644 Y1663 D1666 F1670 Y1674 Q176 S179 Y180 N183 I186 D187 Y206 D209 F213 Y217 2.3.1.- 0009058 ic50=0.26uM remove_due_to_license_issue IC50=260nM I6X8D2 28669536 1801 DGFVRTLRARPEAGGKVPVFVFHPAGGSTVVYEPLLGRLPADTPMYGFERVEGSIEERAQQYVPKLIEMQGDGPYVLVGWSLGGVLAYACAIGLRRLGKDVRFVGLIDAVRAGEEIPQTKEEIRKRWDRYAAFAEKTFNVTIPAIPYEQLEELDDEGQVRFVLDAVSIPAGIIEHQRTSYLDNRAIDTAQIQPYDGHVTLYMADRYHDDAIMFEPRYAVRQPDGGWGEYVSDLEVVPIGGEHIQAIDEPIIAKVGEHMSRALGQIEADRT 5v3y A 1.98 BS01 5V8 A 1 Q1633 S1636 Y1637 N1640 D1644 Y1663 D1666 A1667 F1670 Y1674 Q175 S178 Y179 N182 D186 Y205 D208 A209 F212 Y216 2.3.1.- 0009058 ic50=0.19uM remove_due_to_license_issue IC50=0.190000nM I6X8D2 28669536 1801 DGFVRTLRARPEAGGKVPVFVFHPAGGSTVVYEPLLGRLPADTPMYGFERVEGSIEERAQQYVPKLIEMQGDGPYVLVGWSLGGVLAYACAIGLRRLGKDVRFVGLIDAVRAGEEIPQTKEEIRKRWDRYAAFAEKTFNVTIPAIPYEQLEELDDEGQVRFVLDAVIPAGIIEHQRTSYLDNRAIDTAQIQPYDGHVTLYMADRYHDDAIMFEPRYAVRQPDGGWGEYVSDLEVVPIGGEHIQAIDEPIIAKVGEHMSRALGQIEADRT 5v40 A 1.991 BS01 JS1 A 1 Q1633 S1636 Y1637 N1640 D1644 A1667 F1670 Y1674 Q179 S182 Y183 N186 D190 A213 F216 Y220 2.3.1.- 0009058 ic50=1.57uM remove_due_to_license_issue I6X8D2 28669536 1801 IDGFVRTLRARPEAGGKVPVFVFHPAGGSTVVYEPLLGRLPADTPMYGFERVEGSIEERAQQYVPKLIEMQGDGPYVLVGWSLGGVLAYACAIGLRRLGKDVRFVGLIDAVRAGEEIPQTKEEIRKRWDRYAAFAEKTFVTIPAIPYEQLEELDDEGQVRFVLDAVSQVQIPAGIIEHQRTSYLDNRAIDTAQIQPYDGHVTLYMADRYHDDAIMFEPRYAVRQPDGGWGEYVSDLEVVPIGGEHIQAIDEPIIAKVGEHMSRALGQIEADRT 5v41 A 2.051 BS01 J24 A 1 Y1582 S1636 Y1637 N1640 I1643 D1644 A1667 F1670 Y1674 Y130 S181 Y182 N185 I188 D189 A212 F215 Y219 2.3.1.- 0009058 ic50=0.71uM remove_due_to_license_issue I6X8D2 28669536 1801 DGFVRTLRARPEAGGKVPVFVFHPAGGSTVVYEPLLGRLPADTPMYGFERVEGSIEERAQQYVPKLIEMQGDGPYVLVGWSLGGVLAYACAIGLRRLGKDVRFVGLIDAVRAGEEIPQTKEEIRKRWDRYAAFAEKTFNVPAIPYEQLEELDDEGQVRFVLDAVSQSVQIPAGIIEHQRTSYLDNRAIDTAQIQPYDGHVTLYMADRYHDDAIMFEPRYAVRQPDGGWGEYVSDLEVVPIGGEHIQAIDEPIIAKVGEHMSRALGQIEADRT 5v42 A 1.987 BS01 I66 A 1 S1636 Y1637 N1640 D1644 F1670 Y1674 S177 Y178 N181 D185 F211 Y215 2.3.1.- 0009058 ic50=0.24uM remove_due_to_license_issue I6X8D2 28669536 1801 GFVRTLRARPEAGGKVPVFVFHPAGGSTVVYEPLLGRLPADTPMYGFERVEGSIEERAQQYVPKLIEMQGDGPYVLVGWSLGGVLAYACAIGLRRLGKDVRFVGLIDAVRAGEEIPQTKEEIRKRWDRYAAFAEKTFNVPAIPYEQLEELDDEGQVRFVLDAVSQIPAGIIEHQRTSYLDNRAIDTAQIQPYDGHVTLYMADRYHDDAIMFEPRYAVRQPDGGWGEYVSDLEVVPIGGEHIQAIDEPIIAKVGEHMSRALGQIEADRT 5v4q B 2.2 BS01 8WY B 1 T381 T399 N401 D423 S451 S452 G473 G474 T1 T19 N21 D43 S71 S72 G93 G94 2.3.2.2,3.4.19.13,3.4.19.14 0006751,0036374 remove_due_to_license_issue P19440 28378915 1102 TAHLSVVAEDGSAVSATSTINLYFGSKVRSPVSGILFNNEMDDFSSPSITNEFGVPPSPANFIQPGKQPLSSMCPTIMVGQDGQVRMVVGAAGGTQITTATALAIIYNLWFGYDVKRAVEEPRLHNQLLPNVTTVERNIDQAVTAALETRHHHTQIASTFIAVVQAIVRTAGGWAAASDSRKGGEPAGY 5v5d A 2.104 BS01 8OY A 1 W109 L110 W106 L107 H46 S114 S116 H134 R142 R143 H43 S111 S113 H131 R139 R140 3.4.21.97 0004252,0006508 remove_due_to_license_issue O40922 28759216 201 GLYVGGFVDVVSCPKLEQELYLDPDQVTDYLPVTEPLPITIEHLPETEVGWTLGLFQVSHGIFCTGAITSPAFLELASRLADTSHVARAPVKNLPKEPLLEILHTWLPGLSLSSIHPRELSQTPSGPVFQHVSLCALGRRRGTVAVYGHDAEWVVSRFSSVSKSERAHILQHVSSCRLEDLSTPNFVSPLE 5v5e A 2.299 BS01 8N4 A 1 I44 L79 L83 P192 I39 L74 L78 P187 H46 S114 S116 H134 R142 R143 H41 S109 S111 H129 R137 R138 3.4.21.97 0004252,0006508 remove_due_to_license_issue O40922 28759216 201 GLYVGGFVDVVSCPKLELYLDPDQVTDYLPVTEPLPITIEHLPETEVGWTLGLFQVSHGIFCTGAITSPAFLELASRLADTSHVARAPVKNLPKEPLLEILHTWLPGLSLSSIHPRELSQTPSGPVFQHVSLCALGRRRGTVAVYGHDAEWVVSRFSSVSKSERAHILQHVSSCRLEDLSTPNFVSPL 5v5n A 2.006 BS01 EDH A 1 K63 M104 E105 Y106 A107 L163 C174 K37 M78 E79 Y80 A81 L137 C148 D156 K158 P160 N161 I173 D175 D130 K132 P134 N135 I147 D149 2.7.11.25 0004672,0005524,0006468 ic50=9.5nM remove_due_to_license_issue O43318,Q15750 28820959 501 SLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIESESERKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPPGEDGRVEPYVDFAEFYRLWSVDHG 5v5y A 1.9 BS01 8X7 A 1 I305 V313 A326 K328 N376 Y378 C379 G382 D386 F433 I13 V21 A34 K36 N84 Y86 C87 G90 D94 F141 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 Kd=13.4nM remove_due_to_license_issue IC50=5.2nM, Kd=3.2nM P30291 28792760 601 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISRTKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVL 5v6u B 2.8 BS01 8YM B 1 K160 T163 A164 R167 E216 F219 F221 Y223 M294 K109 T112 A113 R116 E141 F144 F146 Y148 M204 G85 V86 H144 G145 C186 G34 V35 H93 G94 C135 3.4.22.60 0003723,0004190,0004197,0005515,0005576,0005615,0005634,0005654,0005737,0005829,0006508,0006915,0007507,0008233,0008234,0009411,0016485,0030163,0042742,0043525,0044346,0051146,0051402,0051604,0070227,0071222,0071887,0072734,0097153,0097194,1905686 remove_due_to_license_issue P55210 28940929 401 TTRDRTYQYNMNFEKLGKCIIINNKNFDKVTGMGVRNGTDKDAEALFKCFRSLGFDVIVYNDCSCAKMQDLLKKASEEDHTNAACFACILLSHGEENVIYGKDGVTPIKDLTAHFRGDRCKTLLEKPKLFFIQACRKIPVEADFLFAYSTVPSWRSPGRGSWFVQALCSILEEHGKDLEIMQILTRVNDRVARHFKQIPCVVSMLTKELYFSQ 5v79 A 2.25 BS01 8Y4 A 1 T62 D96 N115 M139 D185 F190 G217 R220 K221 R255 H257 T52 D86 N105 M129 D175 F180 G207 R210 K211 R245 H247 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAK 5v7a A 2.35 BS01 8Y7 A 1 T62 D96 N115 M139 D185 F190 G217 K221 R255 T52 D86 N105 M129 D175 F180 G207 K211 R245 2.5.1.15 0004156,0005737,0005829,0009396,0009410,0016740,0042558,0044237,0046654,0046656,0046872 remove_due_to_license_issue P0AC13 29171692 301 MKLFAQGTSLDLSHPHVMGILNVTNSLIDAVKHANLMINAGATIIDVGGESTRPGAAEVSVEEELQRVIPVVEAIAQRFEVWISVDTSKPEVIRESAKVGAHIINDIRSLSEPGALEAAAETGLPVCLMHMQGNPKTMQEAPKYDDVFAEVNRYFIEQIARCEQAGIAKEKLLLDPGFGFGKNLSHNYSLLARLAEFHHFNLPLLVGMSRKSMIGQLLNVGPSERLSGSLACAVIAAMQGAHIIRVHDVKETVEAMRVVEATLSAK 5v7i A 2.47 BS01 8Z1 A 1 L166 G170 H171 L172 L124 G128 H129 L130 Y96 E98 D251 T277 K280 R286 Y54 E56 D209 T235 K238 R244 2.1.2.1 0002082,0003682,0004372,0005515,0005634,0005737,0005739,0005743,0005759,0006544,0006545,0006563,0006564,0006730,0008284,0008732,0015630,0016597,0016740,0019264,0030170,0034340,0035999,0042645,0042802,0046653,0051262,0051289,0070062,0070129,0070536,0070552,1903715 remove_due_to_license_issue IC50=13.0nM P34897 29073064 601 WTGQESLSDSDPEMWELLQREKDRQCRGLELIASENFCSRAALEALGSCLNNKYSEGYPGKRYYGGAEVVDEIELLCQRRALEAFDLDPAQWGVNVQPYSGSPANLAVYTALLQPHDRIMGLDLPDGGHLTHGYMSDVKRISATSIFFESMPYKLNPKTGLIDYNQLALTARLFRPRLIIAGTSAYARLIDYARMREVCDEVKAHLLADMAHISGLVAAKVIPSPFKHADIVTTTTHKTLRGARSGLIFYRKGVKAVDPKTGREIPYTFEDRINFAVFPSLQGGPHNHAIAAVAVALKQACTPMFREYSLQVLKNARAMADALLERGYSLVSGGTDNHLVLVDLRPKGLDGARAERVLELVSITANKNTCPGDRSAITPGGLRLGAPALTSRQFREDDFRRVVDFIDEGVNIGLEVKSKTAKLQDFKSFLLKDSETSQRLANLRQRVEQFARAFPMPGFDEH 5v7i A 2.47 BS02 8Z1 B 1 E98 Y105 Y106 E56 Y63 Y64 Y96 E98 D251 T277 K280 R286 Y54 E56 D209 T235 K238 R244 2.1.2.1 0002082,0003682,0004372,0005515,0005634,0005737,0005739,0005743,0005759,0006544,0006545,0006563,0006564,0006730,0008284,0008732,0015630,0016597,0016740,0019264,0030170,0034340,0035999,0042645,0042802,0046653,0051262,0051289,0070062,0070129,0070536,0070552,1903715 remove_due_to_license_issue IC50=13.0nM P34897 29073064 601 WTGQESLSDSDPEMWELLQREKDRQCRGLELIASENFCSRAALEALGSCLNNKYSEGYPGKRYYGGAEVVDEIELLCQRRALEAFDLDPAQWGVNVQPYSGSPANLAVYTALLQPHDRIMGLDLPDGGHLTHGYMSDVKRISATSIFFESMPYKLNPKTGLIDYNQLALTARLFRPRLIIAGTSAYARLIDYARMREVCDEVKAHLLADMAHISGLVAAKVIPSPFKHADIVTTTTHKTLRGARSGLIFYRKGVKAVDPKTGREIPYTFEDRINFAVFPSLQGGPHNHAIAAVAVALKQACTPMFREYSLQVLKNARAMADALLERGYSLVSGGTDNHLVLVDLRPKGLDGARAERVLELVSITANKNTCPGDRSAITPGGLRLGAPALTSRQFREDDFRRVVDFIDEGVNIGLEVKSKTAKLQDFKSFLLKDSETSQRLANLRQRVEQFARAFPMPGFDEH 5v7i B 2.47 BS01 8Z1 A 1 Y105 Y106 Y63 Y64 Y96 E98 D251 T277 K280 R286 Y54 E56 D209 T235 K238 R244 2.1.2.1 0002082,0003682,0004372,0005515,0005634,0005737,0005739,0005743,0005759,0006544,0006545,0006563,0006564,0006730,0008284,0008732,0015630,0016597,0016740,0019264,0030170,0034340,0035999,0042645,0042802,0046653,0051262,0051289,0070062,0070129,0070536,0070552,1903715 remove_due_to_license_issue IC50=13.0nM P34897 29073064 601 WTGQESLSDSDPEMWELLQREKDRQCRGLELIASENFCSRAALEALGSCLNNKYSEGYPGKRYYGGAEVVDEIELLCQRRALEAFDLDPAQWGVNVQPYSGSPANLAVYTALLQPHDRIMGLDLPDGGHLTHGYMSDVKRISATSIFFESMPYKLNPKTGLIDYNQLALTARLFRPRLIIAGTSAYARLIDYARMREVCDEVKAHLLADMAHISGLVAAKVIPSPFKHADIVTTTTHKTLRGARSGLIFYRKGVKAVDPKTGREIPYTFEDRINFAVFPSLQGGPHNHAIAAVAVALKQACTPMFREYSLQVLKNARAMADALLERGYSLVSGGTDNHLVLVDLRPKGLDGARAERVLELVSITANKNTCPGDRSAITPGGLRLGAPALTSRQFREDDFRRVVDFIDEGVNIGLEVKSKTAKLQDFKSFLLKDSETSQRLANLRQRVEQFARAFPMPGFDEH 5v7i B 2.47 BS02 8Z1 B 1 L166 G170 H171 S226 K409 L124 G128 H129 S184 K367 Y96 E98 D251 T277 K280 R286 Y54 E56 D209 T235 K238 R244 2.1.2.1 0002082,0003682,0004372,0005515,0005634,0005737,0005739,0005743,0005759,0006544,0006545,0006563,0006564,0006730,0008284,0008732,0015630,0016597,0016740,0019264,0030170,0034340,0035999,0042645,0042802,0046653,0051262,0051289,0070062,0070129,0070536,0070552,1903715 remove_due_to_license_issue IC50=13.0nM P34897 29073064 601 WTGQESLSDSDPEMWELLQREKDRQCRGLELIASENFCSRAALEALGSCLNNKYSEGYPGKRYYGGAEVVDEIELLCQRRALEAFDLDPAQWGVNVQPYSGSPANLAVYTALLQPHDRIMGLDLPDGGHLTHGYMSDVKRISATSIFFESMPYKLNPKTGLIDYNQLALTARLFRPRLIIAGTSAYARLIDYARMREVCDEVKAHLLADMAHISGLVAAKVIPSPFKHADIVTTTTHKTLRGARSGLIFYRKGVKAVDPKTGREIPYTFEDRINFAVFPSLQGGPHNHAIAAVAVALKQACTPMFREYSLQVLKNARAMADALLERGYSLVSGGTDNHLVLVDLRPKGLDGARAERVLELVSITANKNTCPGDRSAITPGGLRLGAPALTSRQFREDDFRRVVDFIDEGVNIGLEVKSKTAKLQDFKSFLLKDSETSQRLANLRQRVEQFARAFPMPGFDEH 5v7t A 2.3 BS01 91V A 1 H1601 G1602 K1630 Y1633 S1641 Y1646 H1672 H70 G71 K87 Y90 S98 Y103 H129 2.4.2.- 0003950 ic50=610nM remove_due_to_license_issue Q460N5 28315326 1801 KQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 5v7w A 2.65 BS01 91J A 1 H1682 G1683 D1685 Y1714 A1716 S1722 Y1727 H69 G70 D72 Y89 A91 S97 Y102 2.4.2.- 0003950 remove_due_to_license_issue Q460N5 28315326 1901 QQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 5v82 A 1.888 BS01 96Y A 1 L44 F49 A65 K67 L120 D128 L174 I185 D186 L11 F16 A32 K34 L87 D95 L141 I152 D153 D167 K169 N172 D186 L193 T204 D134 K136 N139 D153 L160 T171 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 Ki=0.07nM remove_due_to_license_issue Ki=0.067nM P11309 28445037 401 LESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS 5v83 A 2.002 BS01 8Z7 A 1 I1086 F1089 P1097 A1098 V1102 I1105 A1106 A1111 Q1114 E1116 F1117 F1164 A1180 Y1181 L1184 I201 F204 P212 A213 V217 I220 A221 A226 Q229 E231 F232 F279 A292 Y293 L296 E11 D20 E23 D32 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 ic50=7uM remove_due_to_license_issue P00720,Q96GG9 28581483 401 SQDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRTKRVITTFRTGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHKRSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQIA 5v84 A 2.7 BS01 96V A 1 W457 P458 F459 V463 Y467 N514 Y520 W21 P22 F23 V27 Y31 N78 Y84 ? 0006338,0090537 remove_due_to_license_issue IC50=190nM Q9BXF3 28740608 602 DDDFTAMYKVLDVVKAHKDSWPFLEPVDESYAPNYYQIIKAPMDISSMEKKLNGGLYCTKEEFVNDMKTMFRNCRKYNGESSEYTKMSDNLERCFHRAMMKH 5v84 D 2.7 BS01 96V A 1 M503 K504 F531 H532 M66 K67 F94 H95 ? 0006338,0090537 remove_due_to_license_issue IC50=190nM Q9BXF3 28740608 602 DDFTAMYKVLDVVKAHKDSWPFLEPVDESYAPNYYQIIKAPMDISSMEKKLNGGLYCTKEEFVNDMKTMFRNCRKYNGESSEYTKMSDNLERCFHRAMMKH 5v84 D 2.7 BS02 96V D 1 P458 F459 V463 Y467 N514 Y520 P21 F22 V26 Y30 N77 Y83 ? 0006338,0090537 remove_due_to_license_issue IC50=190nM Q9BXF3 28740608 602 DDFTAMYKVLDVVKAHKDSWPFLEPVDESYAPNYYQIIKAPMDISSMEKKLNGGLYCTKEEFVNDMKTMFRNCRKYNGESSEYTKMSDNLERCFHRAMMKH 5v86 A 1.374 BS01 8ZA A 1 I1083 I1086 P1097 I1105 A1106 Q1114 E1116 F1117 F1164 A1180 Y1181 I197 I200 P211 I219 A220 Q228 E230 F231 F278 A294 Y295 E11 D20 E22 D31 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 ic50=80nM remove_due_to_license_issue P00720,Q96GG9 28581483 2001 QDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWAEAAVNLAKSRWYNQTPNRTKRVITTFATGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLESIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQ 5v88 A 1.601 BS01 8ZD A 1 I1086 F1089 P1097 V1102 A1106 Q1114 C1115 E1116 F1117 F1164 A1180 Y1181 L1184 I201 F204 P212 V217 A221 Q229 C230 E231 F232 F279 A295 Y296 L299 E11 D20 E23 D32 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,Q96GG9 28581483 401 SQDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWAEAAVNLAKSRWYNQTPNRTKRVITTFATGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLESIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQIA 5v8o A 3.1 BS02 8ZM A 1 R376 Y436 N482 F488 L490 R205 Y265 N311 F317 L319 2.7.7.86 remove_due_to_license_issue Kd=170000nM, IC50=78000nM Q8N884 28934246 602 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDEF 5v8p A 2.501 BS02 90G A 1 V70 I161 Q162 F163 F194 H223 E224 H227 E262 Y366 V70 I161 Q162 F163 F194 H210 E211 H214 E236 Y338 H223 E224 H227 E262 R363 H210 E211 H214 E236 R335 3.4.24.69 0004222,0006508,0008270 Ki=10.2uM remove_due_to_license_issue P0DPI1 28698055 502 SSGLVPRGSHMQFVNKQFNYKDPVNGVDIAYIKIPQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVTASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKL 5v8q A 1.44 BS01 97A A 1 L704 N705 M745 V746 M749 F764 L873 T877 M895 L34 N35 M75 V76 M79 F94 L203 T207 M225 ? ic50=3.6nM remove_due_to_license_issue EC50=4.7nM, IC50=3.6nM P10275 28454849 1004 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACARKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 5v8v A 2.6 BS01 90D A 1 T84 A295 S296 Y297 F319 D320 H367 T15 A226 S227 Y228 F250 D251 H298 D104 S107 N109 W111 Y149 D292 A295 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 28985999 502 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5v8v A 2.6 BS02 90D A 2 Q85 Y86 V102 D104 G106 P184 F185 L187 A188 F190 V193 D292 T293 G294 A295 S296 Q16 Y17 V33 D35 G37 P115 F116 L118 A119 F121 V124 D223 T224 G225 A226 S227 D104 S107 N109 W111 Y149 D292 A295 D35 S38 N40 W42 Y80 D223 A226 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 28985999 503 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSENSQSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5v9p A 3.0 BS03 90S A 1 W470 Y472 F480 H483 E485 N493 W503 H571 V584 N585 W282 Y284 F292 H295 E297 N305 W315 H383 V396 N397 G465 Y472 H483 E485 H571 A583 G277 Y284 H295 E297 H383 A395 1.14.11.67 0003677 remove_due_to_license_issue IC50=0.740nM P29375 28512031 904 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRVRLDFLDQLAKFWELQGSTLKIPVVERKILDLYALSKIVASKGGFEMVTKEKKWSKVGSRLGYLPGKGTGSLLKSHYERILYPYELFQSGVSLMGVQMYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINVDISGMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCTADWLPIGRQCVNHYRRLRRHCVFSHEELIFKMAADPECLDVGLAAMVCKELTLMTEEETRLRESVVQMGVLMSEEEVFELVPDDERQCSACRTTCFLSALTCSCNPERLVCLYHPTDLCPCPMQKKCLRYRYPLEDLPSLLYGVKVRAQSYDTWVSVMLEDAEDRKYPENDLFRKLR 5v9t A 3.05 BS03 90V A 1 Y472 F480 H483 E485 N493 K501 H571 N575 A583 V584 N585 Y284 F292 H295 E297 N305 K313 H383 N387 A395 V396 N397 G465 Y472 H483 E485 H571 A583 G277 Y284 H295 E297 H383 A395 1.14.11.67 0003677 remove_due_to_license_issue IC50=570nM, Kd=2400nM, EC50=960nM P29375 28512031 904 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRVRLDFLDQLAKFWELQGSTLKIPVVERKILDLYALSKIVASKGGFEMVTKEKKWSKVGSRLGYLPGKGTGSLLKSHYERILYPYELFQSGVSLMGVQMYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINVDISGMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCTADWLPIGRQCVNHYRRLRRHCVFSHEELIFKMAADPECLDVGLAAMVCKELTLMTEEETRLRESVVQMGVLMSEEEVFELVPDDERQCSACRTTCFLSALTCSCNPERLVCLYHPTDLCPCPMQKKCLRYRYPLEDLPSLLYGVKVRAQSYDTWVSVMLEDAEDRKYPENDLFRKLR 5va0 A 2.295 BS01 dna C 0 C431 H432 Y433 K446 C13 H14 Y15 K28 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 28591827 517 ~ 532 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNL 5va0 A 2.295 BS02 dna D 0 S440 F444 R447 R470 K471 R477 S22 F26 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 28591827 501 ~ 516 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNL 5va0 B 2.295 BS01 dna D 0 C431 H432 Y433 C13 H14 Y15 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 28591827 501 ~ 516 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEA 5va7 A 2.153 BS01 dna C 0 C431 H432 Y433 K442 K446 C13 H14 Y15 K24 K28 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 28591827 859 ~ 874 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNL 5va7 A 2.153 BS02 dna D 0 S440 F444 R447 R470 K471 R477 S22 F26 R29 R52 K53 R59 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 28591827 840 ~ 855 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNL 5va7 B 2.153 BS01 dna D 0 G430 C431 H432 Y433 G12 C13 H14 Y15 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P04150 28591827 840 ~ 855 KLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNL 5vad A 2.36 BS01 91Y A 1 R1152 E1154 F1161 L1162 R1163 T1164 F1167 W1169 T1240 T1276 R1278 R137 E139 F146 L147 R148 T149 F152 W154 T225 T261 R263 6.1.1.15,6.1.1.17 0000166,0004812,0004827,0005524,0005737,0006418,0006433 Kd=0.76nM remove_due_to_license_issue P07814 28501621 1601 LEAKKEENLADWYSQVITKSEMIEYHDISGCYILRPWAYAIWEAIKDFFDAEIKKLGVENCYFPMFVSQSALEKEKTHVADFAPEVAWVTRSGKTELAEPIAIRPTSETVMYPAYAKWVQSHRDLPIKLNQWCNVVRWEFKHPQPFLRTREFLWQEGHSAFATMEEAAEEVLQILDLYAQVYEELLAIPVVKGRKTEKEKFAGGDYTTTIEAFISASGRAIQGGTSHHLGQNFSKMFEIVFEDPKIPGEKQFAYQNSWGLTTRTIGVMTMVHGDNMGLVLPPRVACVQVVIIPCGILSEEDKEALIAKCNDYRRRLLSVNIRVRADLRDNYSPGWKFNHWELKGVPIRLEVGPRDMKSCQFVAVRRDTGEKLTVAENEAETKLQAILEDIQVTLFTRASEDLKTHMVVANTMEDFQKILDSGKIVQIPFCGEIDCEDWIKKTTAMGAKSLCIPFKPLCELQPGAKCVCNPAKYYTLFGRSY 5var A 1.83 BS01 92Y A 1 F932 D934 S936 W967 Y973 F36 D38 S40 W71 Y77 1.14.11.66,1.14.11.69 Kd=81.7uM remove_due_to_license_issue Kd=80000nM O75164 29691138 1101 QSITAGQKVISKHKNGRFYQCEVVRLTTETFYEVNFDDGSFSDNLYPEDIVSQDCLQFGPPAEGEVVQVRWTDGQVYGAKFVASHPIQMYQVEFEDGSQLVVKRDDVY 5vb5 A 2.226 BS01 92A A 1 Q286 W317 C320 L324 R364 M365 F378 F388 H479 Y502 F506 Q22 W53 C56 L60 R100 M101 F114 F124 H215 Y238 F242 ? 0003677,0004879,0005634,0006355 Kd=0.35uM remove_due_to_license_issue P51449,Q15596 28546429 602 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGGGEKHKILHRLLQDS 5vb6 A 2.041 BS01 927 A 1 L287 W317 C320 H323 L324 M365 R367 F388 H479 Y502 L23 W53 C56 H59 L60 M101 R103 F124 H215 Y238 ? 0003677,0004879,0005634,0006355 Kd=0.43uM remove_due_to_license_issue P51449,Q15596 28546429 602 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGGGEKHKILHRLLQDS 5vb7 A 2.335 BS01 921 A 1 Q286 L287 W317 C320 H323 L324 M365 R367 F388 I400 H479 Q22 L23 W53 C56 H59 L60 M101 R103 F124 I136 H215 ? 0003677,0004879,0005634,0006355 Kd=0.19uM remove_due_to_license_issue P51449,Q15596 28546429 602 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGGGEKHKILHRLLQDS 5vc3 A 1.97 BS01 DB8 A 1 E303 I305 A326 K328 V360 N376 Y378 C379 G382 F433 D463 E11 I13 A34 K36 V68 N84 Y86 C87 G90 F141 D153 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 Kd=77.5nM remove_due_to_license_issue Kd=510nM P30291 28792760 601 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISRTKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVLL 5vc4 A 2.1 BS01 XZN A 1 E303 I305 K328 I374 N376 Y378 C379 G382 F433 D463 E11 I13 K36 I82 N84 Y86 C87 G90 F141 D153 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 Kd=43.7nM remove_due_to_license_issue Kd=44nM P30291 28792760 601 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISRTKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVLLS 5vc5 A 1.93 BS01 96M A 1 I305 A326 K328 E346 I374 N376 Y378 C379 G382 F433 D463 I13 A34 K36 E54 I82 N84 Y86 C87 G90 F141 D153 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 Kd=11nM remove_due_to_license_issue IC50=165nM, Kd=11nM P30291 28792760 601 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISRTKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVLLS 5vc6 A 2.0 BS01 P48 A 1 I305 F310 V313 A326 K328 N376 C379 G382 F433 D463 I13 F18 V21 A34 K36 N84 C87 G90 F141 D151 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 Kd=13.6nM remove_due_to_license_issue Kd=14nM P30291 28792760 601 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISRVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVLLS 5vc9 C 2.1 BS01 dna A 0 R136 H164 R170 K171 R3 H31 R37 K38 ? 0003677,0008270 remove_due_to_license_issue Q9H2H0 29276034 1 ~ 12 KKRKRCGVCVPCKRLINCGVCSSCRNRKTGHQICKFRKCEELKKKP 5vc9 F 2.1 BS01 dna D 0 R136 H164 Q165 R170 K171 L175 R3 H31 Q32 R37 K38 L42 ? 0003677,0008270 remove_due_to_license_issue Q9H2H0 29276034 1 ~ 12 KKRKRCGVCVPCKRLINCGVCSSCRNRKTGHQICKFRKCEELKK 5vc9 F 2.1 BS02 dna E 0 G163 H164 G30 H31 ? 0003677,0008270 remove_due_to_license_issue Q9H2H0 29276034 1 ~ 12 KKRKRCGVCVPCKRLINCGVCSSCRNRKTGHQICKFRKCEELKK 5vcv A 1.92 BS01 1N1 A 1 L116 A137 K139 L185 T187 C190 G191 P192 Q196 F240 D251 L43 A64 K66 L112 T114 C117 G118 P119 Q123 F167 D178 D233 K235 N238 D251 D270 D160 K162 N165 D178 D197 2.7.11.1 0004672,0005524,0006468 Kd=150nM remove_due_to_license_issue Kd=130nM, IC50=6.0nM, Ki=73nM Q99640 28792760 404 MHQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ 5vcw A 2.25 BS01 93J A 1 L116 K139 V171 T187 C190 G191 P192 Q196 F240 L40 K63 V95 T111 C114 G115 P116 Q120 F164 D233 K235 N238 D251 D270 D157 K159 N162 D175 D194 2.7.11.1 0004672,0005524,0006468 Kd=1105nM remove_due_to_license_issue Kd=2900nM Q99640 28792760 401 LQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ 5vcx A 2.7 BS01 H8H A 1 L116 A137 K139 T187 C190 F240 D251 L42 A63 K65 T113 C116 F166 D177 D233 K235 N238 D251 D270 D159 K161 N164 D177 D196 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=418nM, Ki=40nM, Kd=2817nM Q99640 28792760 401 HQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ 5vcy A 1.56 BS01 DB8 A 1 L116 A137 V138 K139 V171 L185 T187 C190 G191 P192 F240 L50 A71 V72 K73 V105 L119 T121 C124 G125 P126 F174 D233 K235 N238 D251 D270 D167 K169 N172 D185 D204 2.7.11.1 0004672,0005524,0006468 Kd=270nM remove_due_to_license_issue Ki=13nM, IC50=704nM, Kd=350nM Q99640 28792760 401 DLGTENLYFQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQP 5vcz A 1.5 BS01 XZN A 1 L116 A137 K139 L185 T187 C190 G191 P192 Q196 F240 D251 L49 A70 K72 L118 T120 C123 G124 P125 Q129 F173 D184 D233 K235 N238 D251 D270 D166 K168 N171 D184 D203 2.7.11.1 0004672,0005524,0006468 Kd=444nM remove_due_to_license_issue Kd=444nM Q99640 28792760 401 LGTENLYFQSQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ 5vd0 A 2.13 BS01 8X7 A 1 L116 Y121 V124 K139 T187 C190 G191 P192 F240 L48 Y53 V56 K71 T119 C122 G123 P124 F172 D233 K235 N238 D251 D270 D165 K167 N170 D183 D202 2.7.11.1 0004672,0005524,0006468 Kd=324nM remove_due_to_license_issue IC50=4940nM, Ki=470nM, Kd=324nM Q99640 28792760 401 LGTENLYFLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ 5vd1 A 1.7 BS01 P48 A 1 L116 Y121 V124 A137 K139 C190 G191 P192 Q196 F240 D251 L50 Y55 V58 A71 K73 C124 G125 P126 Q130 F174 D185 D233 K235 N238 D251 D270 D167 K169 N172 D185 D204 2.7.11.1 0004672,0005524,0006468 Kd=990nM remove_due_to_license_issue Kd=990nM Q99640 28792760 401 LGTENLYFQSLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQ 5vd2 A 2.05 BS01 34W A 1 E303 I305 F310 A326 E377 Y378 C379 G382 F433 E11 I13 F18 A34 E85 Y86 C87 G90 F141 D426 K428 D134 K136 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue P30291 28792760 601 SRYTTEFHELEKIGSGEFGSVFKCVKRLDGCIYAIKRSKKPLAGSVDEQNALREVYAHAVLGQHSHVVRYFSAWAEDDHMLIQNEYCNGGSLADAISENYRIMSYFKEAELKDLLLQVGRGLRYIHSMSLVHMDIKPSNIFISRKVMFKIGDLGHVTRISSPQVEEGDSRFLANEVLQENYTHLPKADIFALALTVVCAAGAEPLPRNGDQWHEIRQGRLPRIPQVLSQEFTELLKVMIHPDPERRPSAMALVKHSVL 5vd3 A 1.8 BS01 H8H A 1 L116 A137 K139 L185 T187 C190 G191 P192 F240 L49 A70 K72 L118 T120 C123 G124 P125 F173 D233 K235 N238 D251 D270 D166 K168 N171 D184 D203 2.7.11.1 0004672,0005524,0006468 Kd=2817nM remove_due_to_license_issue IC50=418nM, Ki=40nM, Kd=2817nM Q99640 28792760 401 DLGTENLYFQQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLR 5vdk A 2.7 BS01 8X7 A 1 V220 G221 E222 V226 A239 N289 E290 Y291 C292 G295 F346 V17 G18 E19 V23 A36 N86 E87 Y88 C89 G92 F143 D339 K341 D136 K138 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue Kd=3.9nM P0C1S8 28792760 501 MASRYEKEFLEVEKIGVGEFGTVYKCIKRLDGCVYAIKRSMKTFTELSNENSALHEVYAHAVLGHHPHVVRYYSSWAEDDHMIIQNEYCNGGSLQAAISENTKSGNHFEEPKLKDILLQISLGLNYIHNSSMVHLDIKPSNIFICHKVMYKIGDLGHATSINKPKVEEGDSRFLANEILQEDYRHLPKADIFALGLTIAVAAGAESLPTNGAAWHHIRKGNFPDVPQELSESFSSLLKNMIQPDAEQRPSAAALARNTVL 5vdo A 3.218 BS02 1YC A 1 S305 A307 D319 K362 R376 S434 Y436 S144 A146 D158 K201 R215 S273 Y275 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vdp A 2.3 BS02 1SY A 1 G303 G304 S305 P306 D319 K362 R376 S434 Y436 G142 G143 S144 P145 D158 K201 R215 S273 Y275 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 605 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vdq A 3.246 BS02 9BG A 1 E216 S305 R376 S434 S435 Y436 E57 S143 R214 S272 S273 Y274 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vdr A 3.042 BS02 9B7 A 1 M229 T321 R376 S378 S380 S434 Y436 M68 T160 R212 S214 S216 S270 Y272 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vds A 2.766 BS02 9BJ A 1 T321 R376 S434 Y436 T148 R197 S255 Y257 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKKENPLSQFLEGEILSASKMLSKFRKIIKEEINDDVIMKRPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vdt A 2.576 BS02 4BW A 1 D227 M229 P306 A307 T321 K362 R376 S378 S380 S434 Y436 D66 M68 P145 A146 T160 K201 R215 S217 S219 S273 Y275 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vdu A 2.729 BS02 9BS A 1 R376 Y436 R217 Y277 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 MGASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFD 5vdv A 2.998 BS02 9BV A 1 R376 Y436 H437 R212 Y272 H273 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 5vdw A 2.711 BS02 9BY A 1 R376 L377 S434 Y436 N482 F488 R216 L217 S274 Y276 N322 F328 2.7.7.86 remove_due_to_license_issue Q8N884 28940468 602 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRGGSPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFD 5vee A 2.5 BS01 981 A 1 V335 A348 V349 K350 E366 M395 L398 G401 L447 V36 A49 V50 K51 E67 M96 L99 G102 L148 D440 K442 D444 S445 D458 K467 T478 D141 K143 D145 S146 D159 K168 T179 2.7.11.1 0004672,0005524,0006468 ic50=779nM remove_due_to_license_issue IC50=779nM O96013 28993291 601 SHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNR 5vew A 2.7 BS01 97Y A 1 F347 R348 K351 S352 T355 L401 V405 N406 F355 R356 K359 S360 T363 L402 V406 N407 E1011 D1020 E118 D127 3.2.1.17 0003796,0004888,0004930,0007166,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P43220 28514449 1201 SPEEQLLFLYIIYTVGYALSFSALVIASAILLGFRHLHCTRNYIHLNLFASFILRALCVFFKDAALKWLSYQDSLACRLVFLLDQYCVAANYYWLLVEGVYLYTLLAFNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYSEQWIFRLYVAIGWGVPLLFVVPWGIVKYLYEDEGCWTRNSNMNYWLIIRLPILFACIVNFLIFVRVICIVVSKLKANLMCKTDIAFRLAKSTLTLIPLLCTHEVIFAFVMDRFIKLFTELSFTSFQGLMVAILYCFVNNEVQLEFRKSWERWRL 5vex A 3.0 BS01 97V A 1 R348 K351 S352 T355 M397 V405 N406 R356 K359 S360 T363 M398 V406 N407 E1011 D1020 E118 D127 3.2.1.17 0003796,0004888,0004930,0007166,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P43220 28514449 1201 SPEEQLLFLYIIYTVGYALSFSALVIASAILLGFRHLHCTRNYIHLNLFASFILRALCVFFKDAALKWLSYQDSLACRLVFLLDQYCVAANYYWLLVEGVYLYTLLAFNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYSEQWIFRLYVAIGWGVPLLFVVPWGIVKYLYEDEGCWTRNSNMNYWLIIRLPILFACIVNFLIFVRVICIVVSKLKANLMCKTDIAFRLAKSTLTLIPLLCTHEVIFAFVMDRFIKLFTELSFTSFQGLMVAILYCFVNNEVQLEFRKSWERWRL 5vfc A 1.64 BS01 9BA A 1 A47 S49 A65 I90 S91 D107 F133 Y260 C261 F263 A17 S19 A35 I60 S61 D77 F103 Y230 C231 F233 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 ic50=0.9nM remove_due_to_license_issue P61964 28603984 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 5vfd A 1.93 BS02 9CM A 1 Y112 P113 M114 W115 L127 Y81 P82 M83 W84 L96 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 ? 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 28665414 307 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 5vfj A 2.084 BS01 DHC A 1 K16 K20 K115 R118 K15 K19 K105 R108 N28 G30 L32 H48 K49 Y52 Y73 D99 N27 G29 L31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0035821,0042130,0042742,0047498,0050482,0090729 Kd=20uM remove_due_to_license_issue Q9IAT9 28751219 203 SLFELGKMILQETGKNPAKSYGAYGCNCGVLGRGQPKDATDRCCYVHKCCYKKLTGCDPKKDRYSYSWKDKTIVCGENNPCLKELCECDKAVAICLRENLGTYNKKYRYHLKPFCKKADPC 5vfn A 2.389 BS01 HCI A 1 K16 K20 K115 R118 K15 K19 K105 R108 N28 G30 L32 H48 K49 Y52 Y73 D99 N27 G29 L31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0035821,0042130,0042742,0047498,0050482,0090729 remove_due_to_license_issue Q9IAT9 28751219 201 SLFELGKMILQETGKNPAKSYGAYGCNCGVLGRGQPKDATDRCCYVHKCCYKKLTGCDPKKDRYSYSWKDKTIVCGENNPCLKELCECDKAVAICLRENLGTYNKKYRYHLKPFCKKADPC 5vfx A 2.81 BS01 dna I 0 K41 R60 D70 R71 F72 N73 R75 N82 Y84 K40 R59 D69 R70 F71 N72 R74 N81 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx A 2.81 BS02 dna J 0 S27 R28 Y34 K74 R75 K77 I78 D79 G80 N82 S26 R27 Y33 K73 R74 K76 I77 D78 G79 N81 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx B 2.81 BS01 dna K 0 R28 R75 N82 Y84 R27 R74 N81 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx B 2.81 BS02 dna L 0 S27 R28 Y34 K74 R75 K77 D79 G80 N82 S26 R27 Y33 K73 R74 K76 D78 G79 N81 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx C 2.81 BS01 dna K 0 K41 R60 D70 R71 F72 N73 R75 Y84 K40 R59 D69 R70 F71 N72 R74 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx C 2.81 BS02 dna L 0 S27 R28 Y34 K74 R75 K77 D79 G80 N82 S26 R27 Y33 K73 R74 K76 D78 G79 N81 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx D 2.81 BS01 dna I 0 R28 R71 R75 N82 Y84 R27 R70 R74 N81 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLY 5vfx D 2.81 BS02 dna J 0 S27 R28 Y34 K74 R75 K77 D79 G80 N82 S26 R27 Y33 K73 R74 K76 D78 G79 N81 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLY 5vfx E 2.81 BS01 dna M 0 S27 R28 Y34 D79 G80 N82 S26 R27 Y33 D78 G79 N81 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx E 2.81 BS02 dna N 0 R28 K41 R60 D70 R71 F72 N73 R75 Y84 R27 K40 R59 D69 R70 F71 N72 R74 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx F 2.81 BS01 dna O 0 R28 N29 R71 R75 Y84 R27 N28 R70 R74 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYLE 5vfx F 2.81 BS02 dna P 0 S27 R28 Y34 K74 R75 K77 D79 G80 S26 R27 Y33 K73 R74 K76 D78 G79 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYLE 5vfx G 2.81 BS01 dna O 0 R28 K41 R60 D70 R71 F72 N73 R75 Y84 R27 K40 R59 D69 R70 F71 N72 R74 Y83 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx G 2.81 BS02 dna P 0 S27 R28 Y34 K74 R75 K77 D79 G80 N82 S26 R27 Y33 K73 R74 K76 D78 G79 N81 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 KDLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx H 2.81 BS01 dna M 0 S27 R28 Y34 K74 R75 D79 G80 N82 S25 R26 Y32 K72 R73 D77 G78 N80 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 DLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vfx H 2.81 BS02 dna N 0 N29 R75 Y84 N27 R73 Y82 ? remove_due_to_license_issue Q1PLI2 30213934 1 ~ 23 DLNLYAKELVDVVNYLMKKNQLVFSRNNKFIYVNTETIKSMLEKRNYDTVDGKLYLWRELEWIECAEDRFNKRIKIDGENMYAVVIKYSSYSILKRLYL 5vgi A 2.07 BS02 9DJ A 1 Q73 N86 Y132 Y177 F185 H188 K206 W208 K241 H276 R309 Q65 N78 Y124 Y169 F177 H180 K198 W200 K233 H268 R301 G170 Y177 H188 E190 H276 S288 G162 Y169 H180 E182 H268 S280 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=104nM O75164 28835804 503 NPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEF 5vgo A 1.621 BS01 9B1 A 1 L408 G411 F413 V416 K430 M477 A478 G480 N526 L528 D539 Y551 L15 G18 F20 V23 K37 M84 A85 G87 N133 L135 D146 Y158 D521 A523 R525 N526 D539 F559 D128 A130 R132 N133 D146 F166 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.28nM remove_due_to_license_issue Ki=1.3nM, EC50=33nM, IC50=87nM Q06187 28626519 707 SWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 5vgy A 1.39 BS02 9AA A 1 H94 H96 H119 V121 F131 V143 L198 T199 T200 W209 H92 H94 H117 V119 F128 V140 L195 T196 T197 W206 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=65.5uM remove_due_to_license_issue Kd=43600nM P00918 28817930 304 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5vih B 2.4 BS01 5DZ B 1 H88 T116 R121 T134 G135 G172 S173 T174 Y214 D215 H81 T109 R114 T127 G128 G165 S166 T167 Y207 D208 ? 0015276,0016020 Ki=32.2nM remove_due_to_license_issue Q00959 28760974 301 DNHLSIVTLEEAPFVIVEDIDPLTCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGICH 5vii B 1.951 BS01 5DY B 1 H88 T116 R121 G135 G172 S173 T174 Y214 D215 A241 H81 T109 R114 G128 G165 S166 T167 Y207 D208 A234 ? 0015276,0016020 Ki=51.8nM remove_due_to_license_issue Q00959 28760974 301 DNHLSIVTLEEAPFVIVEDIDTETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGIC 5vij B 2.105 BS01 5DX B 1 H88 T116 R121 I136 S173 T174 Y214 D215 A241 H83 T111 R116 I131 S168 T169 Y209 D210 A236 ? 0015276,0016020 Ki=24.3nM remove_due_to_license_issue Q00959 28760974 301 DNHLSIVTLEEAPFVIVEDIDPLTETCVRNTVPCRKFVKINNSTNEGMNVKKCCKGFCIDILKKLSRTVKFTYDLYLVTNGKHGKKVNNVWNGMIGEVVYQRAVMAVGSLTINEERSEVVDFSVPFVETGISVMVSRGTQVTGLSDKKFQRPHDYSPPFRFGTVPNGSTERNIRNNYPYMHQYMTRFNQRGVEDALVSLKTGKLDAFIYDAAVLNYKAGRDEGCKLVTIGSGYIFATTGYGIALQKGSPWKRQIDLALLQFVGDGEMEELETLWLTGICH 5vil A 2.64 BS01 9E1 A 1 L686 V694 K709 E755 Q756 V757 P758 G759 G760 L810 D822 L17 V25 K40 E86 Q87 V88 P89 G90 G91 L141 D153 D803 K805 D807 N808 D822 T842 D134 K136 D138 N139 D153 T173 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=736nM Q99683 29348070 1001 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGINPCTETFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 5vio A 2.84 BS01 9E4 A 1 L686 G687 V694 K709 M754 E755 Q756 V757 G759 L810 D822 L17 G18 V25 K40 M85 E86 Q87 V88 G90 L141 D153 D803 K805 D807 N808 D822 T842 D134 K136 D138 N139 D153 T173 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=272nM Q99683 29348070 4000 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGINPCTETFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 5vja A 2.46 BS01 DUK A 1 L19 G20 V27 K42 V96 M146 I160 D161 L13 G14 V21 K36 V85 M135 I149 D150 D139 K141 E143 N144 D161 T180 D128 K130 E132 N133 D150 T169 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43293 30033129 1002 SMVEDHYEMGEELGSGQFAIVRKCRQKGTGKEYAAKFIKKRRRGVSREEIEREVNILREIRHPNIITLHDIFENKTDVVLILELVSGGELFDFLAEKESLTEDEATQFLKQILDGVHYLHSKRIAHFDLKPENIMLLDKNVPNPRIKLIDFGIAHKIEAGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGETKQETLTNISAVNYDFDEEYFSNTSELAKDFIRRLLVKDPKRRMTIAQSLEHSWIKA 5vjn A 1.78 BS01 IR8 A 1 R69 D129 D130 A133 T134 G135 S137 R67 D127 D128 A131 T132 G133 S135 R69 R67 2.4.2.7 0002055,0003999,0005515,0005634,0005737,0006166,0006168,0009058,0016208,0016757,0044209,0046872 Ki=8.7uM remove_due_to_license_issue P49435 29178779 201 IASYAQELKLALHQYPNFPSEGILFEDFLPIFRNPGLFQKLIDAFKLHLEEAFPEVKIDYIVGLESRGFLFGPTLALALGVGFVPVRKAGKLPGECFKATYEKEYGSDLFEIQKNAIPAGSNVIIVDDIIATGGSAAAAGELVEQLEANLLEYNFVMELDFLKGRSKLNAPVFTLL 5vjn B 1.78 BS01 IR8 B 1 D129 D130 I131 A133 T134 G135 S137 D120 D121 I122 A124 T125 G126 S128 R69 R67 2.4.2.7 0002055,0003999,0005515,0005634,0005737,0006166,0006168,0009058,0016208,0016757,0044209,0046872 Ki=8.7uM remove_due_to_license_issue P49435 29178779 201 IASYAQELKLALHQYPNFPSEGILFEDFLPIFRNPGLFQKLIDAFKLHLEEAFPEVKIDYIVGLESRGFLFGPTLALALGVGFVPVRKAGKLPGECFKATYLFEIQKNAIPAGSNVIIVDDIIATGGSAAAAGELVEQLEANLLEYNFVMELDFLKGRSKLNAPVFTLL 5vjp A 1.98 BS01 IR9 A 1 D129 D130 I131 A133 T134 G135 S137 D122 D123 I124 A126 T127 G128 S130 R69 R69 2.4.2.7 0002055,0003999,0005515,0005634,0005737,0006166,0006168,0009058,0016208,0016757,0044209,0046872 Ki=14.9uM remove_due_to_license_issue P49435 29178779 201 MPIASYAQELKLALHQYPNFPSEGILFEDFLPIFRNPGLFQKLIDAFKLHLEEAFPEVKIDYIVGLESRGFLFGPTLALALGVGFVPVRKAGKLPGECFKATYLFEIQKNAIPAGSNVIIVDDIIATGGSAAAAGELVEQLEANLLEYNFVMELDFLKGRSKLNAPVFTLLN 5vjp B 1.98 BS01 IR9 B 1 D129 D130 I131 A133 T134 G135 G136 S137 D129 D130 I131 A133 T134 G135 G136 S137 R69 E106 R69 E106 2.4.2.7 0002055,0003999,0005515,0005634,0005737,0006166,0006168,0009058,0016208,0016757,0044209,0046872 Ki=14.9uM remove_due_to_license_issue P49435 29178779 201 MPIASYAQELKLALHQYPNFPSEGILFEDFLPIFRNPGLFQKLIDAFKLHLEEAFPEVKIDYIVGLESRGFLFGPTLALALGVGFVPVRKAGKLPGECFKATYEKEYGSDLFEIQKNAIPAGSNVIIVDDIIATGGSAAAAGELVEQLEANLLEYNFVMELDFLKGRSKLNAPVFTLLN 5vkc A 2.31 BS01 9EA A 1 V220 H224 A227 F228 M231 M250 V253 G262 R263 T266 L267 F270 V42 H46 A49 F50 M53 M72 V75 G84 R85 T88 L89 F92 ? 0042981 remove_due_to_license_issue Ki=98nM Q07820 25679114 401 MDLYRQSLEIISRYLREQATGAKSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 5vkm A 2.2 BS01 GAL C 1 Y64 F71 Y42 F49 ? remove_due_to_license_issue P20273 28970495 1 KWVFEHPETLYAWEGACVWIPCTYRALDGDLESFILFHNPEYNKATSKFDGTRLYESTKDGPSEQKRVQFLGDKNKNCTLSIHPVHLADSGQLGLRMESKTEKWMERIHLAVSERPFPPHIQLPPEIQESQEVTLTCLLAFSCYGYPIQLQWLLEGVPMRQAAVTSTSLTIKSVFTRSELKFSPQWSHHGKIVTCQLQDADGKFLSADTVQLNVKHTPKLEIKVTPSDAIVREGDSVTMTCEVSSSNPEYTTVSWLKDGTSLKKQNTFTLNLREVTKDQSGKYCCQVSNDVGPGRSEEVFLQVQYA 5vkm A 2.2 BS02 SIA C 1 R120 E126 W128 M129 R96 E102 W104 M105 ? remove_due_to_license_issue P20273 28970495 2 KWVFEHPETLYAWEGACVWIPCTYRALDGDLESFILFHNPEYNKATSKFDGTRLYESTKDGPSEQKRVQFLGDKNKNCTLSIHPVHLADSGQLGLRMESKTEKWMERIHLAVSERPFPPHIQLPPEIQESQEVTLTCLLAFSCYGYPIQLQWLLEGVPMRQAAVTSTSLTIKSVFTRSELKFSPQWSHHGKIVTCQLQDADGKFLSADTVQLNVKHTPKLEIKVTPSDAIVREGDSVTMTCEVSSSNPEYTTVSWLKDGTSLKKQNTFTLNLREVTKDQSGKYCCQVSNDVGPGRSEEVFLQVQYA 5vl2 A 1.9 BS01 9EG A 1 Q3 V4 A26 R29 T30 H31 T32 Y34 A79 T80 V81 T100 R101 A102 I115 Q2 V3 A25 R28 T29 H30 T31 Y33 A78 T79 V80 T99 R100 A101 I114 Kd=3.77nM remove_due_to_license_issue 30033524 201 AQVQLQQSGGGLVQAGGSLRLSCAASGRTHTPYAMGWFRQAPGKEREFVGGIGGVAATTTYADSVRGRFTISRDDAKATVYLQMNSLKPEDTAVYYCATRASMAVSTSPRVYPIWGQGTQVTVSS 5vl2 C 1.9 BS01 9EG C 1 Q3 V4 R29 T30 H31 T32 Y34 A79 V81 T100 R101 I115 Q3 V4 R29 T30 H31 T32 Y34 A79 V81 T100 R101 I115 Kd=3.77nM remove_due_to_license_issue 30033524 201 MAQVQLQQSGGGLVQAGGSLRLSCAASGRTHTPYAMGWFRQAPGKEREFVGGIGGVAATTTYADSVRGRFTISRDDAKATVYLQMNSLKPEDTAVYYCATRASMAVSTSPRVYPIWGQGTQVTVSS 5vlr A 2.8 BS01 9EM A 1 T750 M752 W760 I777 K779 Y813 I825 E826 V828 T833 M900 I910 D911 T665 M667 W675 I688 K690 Y724 I736 E737 V739 T744 M802 I812 D813 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue IC50=3.00nM O00329 28541707 4001 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPSLPNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKATEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEKAKADCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHTEEEQLQLREILEGELYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEASVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLNFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFINRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKT 5vm0 B 1.79 BS01 9EG B 1 V4 A26 R29 T30 Y31 T32 Y34 M36 K79 T80 T100 R101 A102 V3 A25 R28 T29 Y30 T31 Y33 M35 K78 T79 T99 R100 A101 Kd=1.6nM remove_due_to_license_issue 30033524 203 AEVQLVESGGGLVQTGDSLRLSCAASGRTYTPYAMAWFRQAPGKEREFVAGIGGIDGTAAYADSVRGRATISRDSAKKTVYLQMNSLKPEDTAVYSCATRASMQVLTSPRVYPIWGRGTQVTVSSPG 5vm6 A 1.5 BS01 9EG A 1 V4 G26 R28 R29 A30 T34 V36 N79 S100 Y120 V1 G23 R25 R26 A27 T31 V33 N76 S97 Y117 ic50=78nM remove_due_to_license_issue 30033524 203 VKLQQSGGGMVQTGDSLRLSCVGSRRALSSTIVGWFRQIPGKEREFVGGIAWSSSDTWYADSVKGRFTISKDDAANGVHLQMSSLKPEDTAVYYCASALRRPGSDASDYTRIPDYPYWGQGTQVTVSSH 5vmu A 2.346 BS01 dna D 0 Y503 V504 S508 R511 E535 Y536 Q563 F564 Y597 A598 Y23 V24 S28 R31 E55 Y56 Q83 F84 Y117 A118 ? remove_due_to_license_issue Q86T24 29546986 1 ~ 18 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAEYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQYAYLS 5vmu A 2.346 BS02 dna E 0 R511 Y522 E535 T538 R549 Y550 Y562 G579 Y584 L586 R595 Y597 Y599 R31 Y42 E55 T58 R69 Y70 Y82 G99 Y104 L106 R115 Y117 Y119 ? remove_due_to_license_issue Q86T24 29546986 19 ~ 36 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAEYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQYAYLS 5vmv A 2.313 BS01 dna D 0 R501 Y503 V504 C505 S508 R511 E535 Q563 R595 R21 Y23 V24 C25 S28 R31 E55 Q83 R115 ? remove_due_to_license_issue Q86T24 29546986 1 ~ 18 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAEYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQ 5vmv A 2.313 BS02 dna E 0 R511 Y522 A534 E535 T538 R549 Y550 Y562 S578 G579 Y584 R595 R31 Y42 A54 E55 T58 R69 Y70 Y82 S98 G99 Y104 R115 ? remove_due_to_license_issue Q86T24 29546986 19 ~ 36 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAEYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQ 5vmz A 2.319 BS01 dna D 0 R501 Y503 V504 C505 S508 R511 Q535 Y536 Q563 F564 R595 Y597 A598 R21 Y23 V24 C25 S28 R31 Q55 Y56 Q83 F84 R115 Y117 A118 ? remove_due_to_license_issue Q86T24 29546986 1 ~ 18 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAQYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQYAYLSD 5vmz A 2.319 BS02 dna E 0 R511 K520 Y522 A534 Q535 T538 R549 Y550 Y562 S578 G579 Y584 L586 R595 Y597 R31 K40 Y42 A54 Q55 T58 R69 Y70 Y82 S98 G99 Y104 L106 R115 Y117 ? remove_due_to_license_issue Q86T24 29546986 19 ~ 36 DDHYELIVDGRVYYICIVCKRSYVCLTSLRRHFNIHSWEKKYPCRYCEKVFPLAQYRTKHEIHHTGERRYQCLACGKSFINYQFMSSHIKSVHSQDPSGDSKLYRLHPCRSLQIRQYAYLSD 5vnd A 2.2 BS01 9ES A 1 V492 L494 A512 K514 E531 I545 V561 C563 A564 G567 E571 L630 A640 D641 V30 L32 A50 K52 E69 I83 V99 C101 A102 G105 E109 L168 A178 D179 D623 A625 R627 N628 D641 D161 A163 R165 N166 D179 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 29247039 801 YELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVECASKGNLREYLQARRPPGLEYSYNPSHNPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 5vo1 A 2.45 BS01 9FS A 1 G132 Q136 V139 A150 M190 F192 C193 G196 Q197 L243 G16 Q20 V23 A34 M74 F76 C77 G80 Q81 L127 D236 K238 P240 N241 D254 T273 D120 K122 P124 N125 D138 T144 2.7.11.25 0004672,0005524,0006468 Ki=0.007uM remove_due_to_license_issue Q12852 28929759 501 LWEVPFEEILDLQWVGSGAQGAVFLGRFHGEEVAVKKVRDLKETDIKHLRKLKHPNIITFKGVCTQAPCYCILMEFCAQGQLYEVLRAGRPVTPSLLVDWSMGIAGGMNYLHLHKIIHRDLKSPNMLITYDDVVKISDFGFAGTVAWMAPEVIRNEPVSEKVDIWSFGVVLWELLTGEIPYKDVDSSAIIWGVGSNSLHLPVPSSCPDGFKILLRQCWNSKPRNRPSFRQILLHLDIASADVLSTPQETYFKSQAEWREEVKLHFEKIK 5vo2 A 2.96 BS01 9FV A 1 V131 Q136 V139 A150 M190 E191 F192 C193 G196 Q197 L243 V15 Q20 V23 A34 M74 E75 F76 C77 G80 Q81 L127 D236 K238 P240 N241 D254 T273 D120 K122 P124 N125 D138 T144 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue Ki=154nM, IC50=1900nM Q12852 28929759 501 LWEVPFEEILDLQWVGSGAQGAVFLGRFHGEEVAVKKVRDLKETDIKHLRKLKHPNIITFKGVCTQAPCYCILMEFCAQGQLYEVLRAGRPVTPSLLVDWSMGIAGGMNYLHLHKIIHRDLKSPNMLITYDDVVKISDFGFAGTVAWMAPEVIRNEPVSEKVDIWSFGVVLWELLTGEIPYKDVDSSAIIWGVGSNSLHLPVPSSCPDGFKILLRQCWNSKPRNRPSFRQILLHLDIASADVLSTPQETYFKSQAEWREEVKLHFEKIK 5vo6 A 2.65 BS01 9J4 A 1 V836 A853 M902 E903 Y904 L905 G908 L956 V18 A35 M84 E85 Y86 L87 G90 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=0.900000nM P52333 28539220 4000 TIFEERHLKYISQLGGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 5voj A 1.799 BS01 9H4 A 1 Q1041 F1043 Y1056 H1057 V1078 D1081 L1135 K1136 G1137 S1139 F1154 R1155 A1156 A1157 Q59 F61 Y74 H75 V96 D99 L153 K154 G155 S157 F172 R173 A174 A175 H1057 D1081 G1137 S1139 H75 D99 G155 S157 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=3.6nM remove_due_to_license_issue P26664 28594175 1201 MASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVDFIPVESLETTMR 5vom A 1.67 BS01 9GY A 1 W81 P82 Q85 N140 D145 I146 W40 P41 Q44 N99 D104 I105 ? ic50=0.79uM remove_due_to_license_issue IC50=790nM O60885 28835800 201 NANPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5vp0 A 2.2 BS02 9GJ A 1 L770 H773 T805 L809 Q812 I826 M847 Q859 F862 L188 H191 T223 L227 Q230 I244 M265 Q277 F280 3.1.4.17 0004114,0007165,0008081 ic50=0.61nM remove_due_to_license_issue IC50=0.610000nM O00408 28796496 1003 TKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5vp1 A 1.86 BS02 9GA A 1 L770 H773 T805 D808 L809 I826 F830 M847 L858 F862 L192 H195 T227 D230 L231 I248 F252 M269 L280 F284 3.1.4.17 0004114,0007165,0008081 ic50=0.51nM remove_due_to_license_issue O00408 29093293 1004 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 5vp9 A 1.859 BS01 9H7 A 1 Q1041 F1043 Y1056 H1057 V1078 D1081 L1135 K1136 G1137 S1139 F1154 R1155 A1156 A1157 Q59 F61 Y74 H75 V96 D99 L153 K154 G155 S157 F172 R173 A174 A175 H1057 D1081 G1137 S1139 H75 D99 G155 S157 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 Ki=1.03nM remove_due_to_license_issue P26664 28594175 1201 MASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVDFIPVESLETTMR 5vpm A 2.9 BS01 9G7 A 1 T15 Q16 Y17 V33 Y80 T82 P115 F116 A119 F121 D223 T224 G225 A226 S227 T15 Q16 Y17 V33 Y80 T82 P115 F116 A119 F121 D220 T221 G222 A223 S224 D35 S38 N40 W42 Y80 D223 A226 D35 S38 N40 W42 Y80 D220 A223 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 28985999 402 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSESLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5vqe A 1.889 BS01 G2F A 1 M63 N92 Y145 K193 H194 M239 D288 A289 M63 N92 Y145 K193 H194 M239 D288 A289 ? 0004553,0005975,0009254,0016798 remove_due_to_license_issue A0A2R2JFS5 29317495 601 MYESILSIKPYNLSKEQITWVNQTLVSLSDDEKLGQLICEIIWDKPGCDPLDVMKHFLPGAVMYRPFKAKRMREFTQRLQKASKIPLLIACNLERGGSGGNGGMEDGTYVASPMGVAATDDESSAEHLGEVCASEGSAVGVNWTYEPIIDIDMNPENPITNVRTYGSDPERIIRMAKAYCRGCRKWGVLTTIKHFPGDGVDYRDQHLMSSVNNLSADEWMDTYGRIYQALIEDGAETLMSAHIRQPNVTRMVNPLIKDEEIMPGSLSKELMQGILRGRFHFNGLICTDATQMVGYTCSMPRHEALPTSIQNGADMLTFTLNPTEDFKALQEGLSCGLLTHERLDEAVARILGMKAKLRLPERKDVVPPLHAMERIQSKKHKKWALEIADESITLVKDKQKGLLPLSPQKTKRIILVQATNEKPEGGYLSEARLFKGLLEKEGFIVHWFEEVPRPGTGYSIEDLKRDTDLFIYYANFKVSSNQTTIRLVWSGDSSPKFVCDVPTLFLSFSNPYHLVDVPMVKTYINAYTSNEATVRMMIEKLMGRSSFKGKSPVDPFAGL 5vqq A 2.55 BS01 9JP A 1 L100 K101 K102 Y181 Y183 Y188 F227 W229 L234 H235 P236 Y318 L95 K96 K97 Y176 Y178 Y183 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqr A 2.55 BS01 9KG A 1 K101 K102 K103 Y181 Q182 Y188 G190 F227 W229 H235 P236 Y318 K96 K97 K98 Y176 Q177 Y183 G185 F222 W224 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqs A 2.504 BS01 9KD A 1 P95 L100 K103 V106 V108 Y181 Y188 G190 F227 W229 L234 H235 P236 Y318 P92 L97 K100 V103 V105 Y178 Y185 G187 F224 W226 L231 H232 P233 Y315 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=1.2uM remove_due_to_license_issue P03366 28827354 601 ISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 5vqt A 2.556 BS01 9K7 A 1 L100 K101 K102 K103 Y181 Y188 G190 F227 W229 L234 H235 P236 Y318 L95 K96 K97 K98 Y176 Y183 G185 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqu A 2.6 BS01 9JP A 1 P95 L100 K101 K102 K103 C181 Q182 Y183 Y188 F227 W229 L234 H235 P236 Y318 P90 L95 K96 K97 K98 C176 Q177 Y178 Y183 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqv A 2.58 BS01 9J1 A 1 L100 K101 K102 K103 C181 Q182 Y183 Y188 F227 W229 L234 H235 P236 Y318 L95 K96 K97 K98 C176 Q177 Y178 Y183 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqw A 2.5 BS01 9KD A 1 P95 L100 K101 K102 K103 V106 V179 C181 Y188 V189 G190 F227 W229 L234 H235 P236 Y318 P90 L95 K96 K97 K98 V101 V174 C176 Y183 V184 G185 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=0.4uM remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqx A 2.4 BS01 9HY A 1 P95 L100 K101 K102 K103 C181 Y188 F227 W229 L234 H235 P236 Y318 P90 L95 K96 K97 K98 C176 Y183 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqy A 2.35 BS01 9J1 A 1 K101 K102 N103 C181 Q182 Y183 Y188 F227 W229 L234 H235 P236 Y318 K96 K97 N98 C176 Q177 Y178 Y183 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vqz A 2.23 BS01 9HY A 1 K101 K102 N103 C181 Y188 F227 W229 L234 H235 P236 Y318 K96 K97 N98 C176 Y183 F222 W224 L229 H230 P231 Y313 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 28827354 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 5vr8 A 1.999 BS01 UDX A 1 G13 Y14 V15 D36 V37 R41 V89 N90 T91 Y108 S130 T131 R346 G13 Y14 V15 D36 V37 R41 V89 N90 T91 Y108 S130 T131 R346 T131 E165 K220 N224 C276 D280 T131 E165 K220 N224 C276 D280 1.1.1.22 0001702,0003979,0005634,0005654,0005829,0006024,0006065,0015012,0016491,0016616,0030206,0034214,0042802,0048666,0051287,0070062 remove_due_to_license_issue O60701 30420606 501 MFEIKKICCIGAGYVGGPTCSVIAHMCPEIRVTVVDVNESRINAWNSPTLPIYEPGLKEVVESCRGKNLFFSTNIDDAIKEADLVFISVNTPTKTYGMGKGRAADLKYIEACARRIVQNSNGYKIVTEKSTVPVRAAESIRRIFDANTKPNLNLQVLSNPEFLAEGTAIKDLKNPDRVLIGGDETPEGQRAVQALCAVYEHWVPREKILTTNTWSSELSKLAANAFLAQRISSINSISALCEATGADVEEVATAIGMDQRIGNKFLKASVGFGGSCFQKDVLNLVYLCEALNLPEVARYWQQVIDMNDYQRRRFASRIIDSLFNTVTDKKIAILGFAFKKDTGDTRESSSIYISKYLMDEGAHLHIYDPKVPREQIVVDLSHDDQVSRLVTISKDPYEACDGAHAVVICTEWDMFKELDYERIHKKMLKPAFIFDGRRVLDGLHNELQTIGFQIETIGKK 5vr8 A 1.999 BS02 UDX A 2 F162 L163 A164 E165 K220 I231 F265 K267 S269 F272 G273 C276 F277 F338 K339 R442 F162 L163 A164 E165 K220 I231 F265 K267 S269 F272 G273 C276 F277 F338 K339 R437 T131 E165 K220 N224 C276 D280 T131 E165 K220 N224 C276 D280 1.1.1.22 0001702,0003979,0005634,0005654,0005829,0006024,0006065,0015012,0016491,0016616,0030206,0034214,0042802,0048666,0051287,0070062 remove_due_to_license_issue O60701 30420606 502 MFEIKKICCIGAGYVGGPTCSVIAHMCPEIRVTVVDVNESRINAWNSPTLPIYEPGLKEVVESCRGKNLFFSTNIDDAIKEADLVFISVNTPTKTYGMGKGRAADLKYIEACARRIVQNSNGYKIVTEKSTVPVRAAESIRRIFDANTKPNLNLQVLSNPEFLAEGTAIKDLKNPDRVLIGGDETPEGQRAVQALCAVYEHWVPREKILTTNTWSSELSKLAANAFLAQRISSINSISALCEATGADVEEVATAIGMDQRIGNKFLKASVGFGGSCFQKDVLNLVYLCEALNLPEVARYWQQVIDMNDYQRRRFASRIIDSLFNTVTDKKIAILGFAFKKDTGDTRESSSIYISKYLMDEGAHLHIYDPKVPREQIVVDLSHDDQVSRLVTISKDPYEACDGAHAVVICTEWDMFKELDYERIHKKMLKPAFIFDGRRVLDGLHNELQTIGFQIETIGKK 5vrl A 2.65 BS01 9JA A 1 G99 D151 F152 Y161 K168 P196 I197 R198 M202 E222 G95 D147 F148 Y157 K164 P192 I193 R194 M198 E214 Y161 K168 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 remove_due_to_license_issue P9WGR1 30456352 300 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 5vrp A 3.22 BS01 9JD A 1 T84 Q85 Y86 V102 D104 P184 F190 V193 Y228 D292 T293 G294 A295 S296 T15 Q16 Y17 V33 D35 P115 F121 V124 Y159 D219 T220 G221 A222 S223 D104 S107 N109 W111 Y149 D292 A295 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 28985999 503 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5vrp A 3.22 BS02 9JD A 2 T84 A295 Y297 F319 D320 H367 T15 A222 Y224 F246 D247 H294 D104 S107 N109 W111 Y149 D292 A295 D35 S38 N40 W42 Y80 D219 A222 3.4.23.15 0004190,0006508 remove_due_to_license_issue P00797 28985999 504 GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRDSSLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR 5vs6 A 2.27 BS01 9QD A 1 Y224 D295 Q297 M407 F409 K420 H456 N460 H461 Y465 Y514 Y17 D88 Q90 M200 F202 K213 H249 N253 H254 Y258 Y299 N218 C223 H464 D481 N11 C16 H257 D274 3.4.19.12 0004843,0016579 Kd=104nM remove_due_to_license_issue IC50=90nM Q93009 29056421 601 KKHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQK 5vsb A 1.85 BS01 9QA A 1 Y224 D295 Q297 L406 M407 R408 F409 K420 H456 H461 Y465 Y514 Y14 D85 Q87 L196 M197 R198 F199 K210 H246 H251 Y255 Y295 N218 C223 H464 D481 N8 C13 H254 D271 3.4.19.12 0004843,0016579 Kd=7.614uM remove_due_to_license_issue Q93009 29056421 4000 TGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQK 5vsb B 1.85 BS01 9QA B 1 Y224 D295 Q297 M407 F409 M410 K420 H456 Y465 Y514 Y17 D88 Q90 M200 F202 M203 K213 H249 Y258 Y300 N218 C223 H464 D481 N11 C16 H257 D274 3.4.19.12 0004843,0016579 Kd=7.614uM remove_due_to_license_issue Q93009 29056421 4000 KKHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEK 5vsc A 1.4 BS06 9HJ A 1 A1077 D1078 R1080 D1083 L1086 D1088 R1157 F1158 I1161 K1162 A160 D161 R163 D166 L169 D171 R236 F237 I240 K241 Y1067 Y1154 Y150 Y233 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 Kd=510nM remove_due_to_license_issue Kd=510nM, IC50=295nM Q96KQ7 28662962 1506 TEKIICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLDEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKSKYFTCQCGSEKCKHSAEAIALEQSRLA 5vsd A 1.85 BS06 9HJ A 1 D1162 A1165 D1171 L1174 D1176 C1186 R1245 F1246 I1249 K1250 D157 A160 D166 L169 D171 C177 R236 F237 I240 K241 Y1155 Y1242 Y150 Y233 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 Kd=57nM remove_due_to_license_issue Kd=57nM, IC50=5.0nM Q9H9B1 28662962 3006 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 5vse A 1.6 BS06 9HG A 1 D1074 A1077 D1078 R1080 D1083 L1086 D1088 C1098 R1157 F1158 I1161 D156 A159 D160 R162 D165 L168 D170 C177 R236 F237 I240 Y1067 Y1154 Y149 Y233 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 Kd=1070nM remove_due_to_license_issue IC50=259nM, Kd=1070nM Q96KQ7 28662962 1506 EKIICRDVARGYENVPIPCVNGVDGEPCPEDYKYISENCETSTMNIDRNITHLQHCTCVDDCSSSNCLCGQLSIRCWYDKDGRLLQEFNKIEPPLIFECNQACSCWRNCKNRVVQSGIKVRLQLYRTAKMGWGVRALQTIPQGTFICEYVGELISDAEADVREDDSYLFDLDNEVYCIDARYYGNISRFINHLCDPNIIPVRVFMLHQDLRFPRIAFFSSRDIRTGEELGFDYGDRFWDIKSKYFTCQCGSEKCKHSAEAIALEQSRLA 5vsf A 1.7 BS06 9HG A 1 D1162 A1165 D1166 R1168 D1171 L1174 D1176 C1186 R1245 F1246 I1249 K1250 D157 A160 D161 R163 D166 L169 D171 C181 R240 F241 I244 K245 Y1155 Y1242 Y150 Y237 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 Kd=94nM remove_due_to_license_issue IC50=4.0nM, Kd=94nM Q9H9B1 28662962 3006 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 5vsj A 2.456 BS01 9HV A 1 K264 N268 S279 W281 K355 Y357 D359 I360 R392 D394 N395 E423 D480 K534 Y535 K250 N254 S265 W267 K341 Y343 D345 I346 R378 D380 N381 E409 D466 K520 Y521 2.4.99.16 0004553,0004556,0005975,0009313,0016757,0016758,0030979 remove_due_to_license_issue Q9L1K2 28422240 701 PTVVGRIPVLDVRPVVQRGRRPAKAVTGESFEVSATVFREGHDAVGANVVLRDPRGRPGPWTPMRELAPGTDRWGATVTAGETGTWSYTVEAWGDPVTTWRHHARIKIPAGLDTDLVLEEGARLYERAAADVPGREDRRELLAAVDALRDESRPAASRLAAALTPQVDAVLARHPLRDLVTSSDPLPLLVERERALYGAWYEFFPRSEGTPHTPHGTFRTAARRLPAIAAMGFDVVYLPPIHPIGTTHRKGRNNTLSATGDDVGSPWAIGSPEGGHDSIHPALGTLDDFDHFVTEAGKLGLEIALDFALQCSPDHPWVHKHPEWFHHRPDGTIAHAENPPKKYQDIYPIAFDADPDGLATETVRILRHWMDHGVRIFRVDNPHTKPVAFWERVIADINGTDPDVIFLAEAFTRPAMMATLAQIGFQQSYTYFTWRNTKQELTEYLTELSGEAASYMRPNFFANTPDILHAYLQHGGRPAFEVRAVLAATLSPTWGIYSGYELCENTPLREGSEEYLDSEKYQLKPRDWTRAAREGTTIAPLVTRLNTIRRENPALRQLRDLHFHPTDKEEVIAYSKRQGSNTVLVVVNLDPRHTQEATVSLDMPQLGLDWHESVPVRDELTGETYHWGRANYVRLEPGRTPAHVCTVLR 5vsk A 3.33 BS01 9HS A 1 Y224 D295 V296 M407 R408 F409 K420 H456 Y465 Y17 D88 V89 M200 R201 F202 K206 H242 Y251 N218 C223 H464 D481 N11 C16 H250 D267 3.4.19.12 0004843,0016579 remove_due_to_license_issue Q93009 29056421 601 KKHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEA 5vt1 A 1.9 BS01 9JS A 1 I171 A192 K194 L269 V270 Q272 I12 A33 K35 L89 V90 Q92 D312 K314 N317 D330 T350 D132 K134 N137 D150 T170 2.7.11.17 0004672,0005524,0006468 remove_due_to_license_issue Q96RR4 29783765 501 MQLNQYTLKDEIGKGSYGVVKLAYNENDNTYYAMKVLSKKKLIRQARGPIEQVYQEIAILKKLDHPNVVKLVEVLDDPNEDHLYMVFELVNQGPVMEVPTLKPLSEDQARFYFQDLIKGIEYLHYQKIIHRDIKPSNLLVGEDGHIKIADFGVSNEFKGSDALLSNTVGTPAFMAPESLSKIFSGKALDVWAMGVTLYCFVFGQCPFMDERIMCLHSKIKSQALEFPDQPDIAEDLKDLITRMLDKNPESRIVVPEIKLHPWVTR 5vt4 A 3.205 BS01 9KJ A 1 K264 N268 S279 W281 Q324 K355 Y357 D359 R392 D394 N395 E423 D480 K534 Y535 K250 N254 S265 W267 Q310 K341 Y343 D345 R378 D380 N381 E409 D466 K520 Y521 2.4.99.16 0004553,0004556,0005975,0009313,0016757,0016758,0030979 remove_due_to_license_issue Q9L1K2 28422240 701 PTVVGRIPVLDVRPVVQRGRRPAKAVTGESFEVSATVFREGHDAVGANVVLRDPRGRPGPWTPMRELAPGTDRWGATVTAGETGTWSYTVEAWGDPVTTWRHHARIKIPAGLDTDLVLEEGARLYERAAADVPGREDRRELLAAVDALRDESRPAASRLAAALTPQVDAVLARHPLRDLVTSSDPLPLLVERERALYGAWYEFFPRSEGTPHTPHGTFRTAARRLPAIAAMGFDVVYLPPIHPIGTTHRKGRNNTLSATGDDVGSPWAIGSPEGGHDSIHPALGTLDDFDHFVTEAGKLGLEIALDFALQCSPDHPWVHKHPEWFHHRPDGTIAHAENPPKKYQDIYPIAFDADPDGLATETVRILRHWMDHGVRIFRVDNPHTKPVAFWERVIADINGTDPDVIFLAEAFTRPAMMATLAQIGFQQSYTYFTWRNTKQELTEYLTELSGEAASYMRPNFFANTPDILHAYLQHGGRPAFEVRAVLAATLSPTWGIYSGYELCENTPLREGSEEYLDSEKYQLKPRDWTRAAREGTTIAPLVTRLNTIRRENPALRQLRDLHFHPTDKEEVIAYSKRQGSNTVLVVVNLDPRHTQEATVSLDMPQLGLDWHESVPVRDELTGETYHWGRANYVRLEPGRTPAHVCTVL 5vyy A 1.792 BS01 9QY A 1 N51 D93 M98 N106 L107 F138 W162 T184 N36 D78 M83 N91 L92 F123 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.62uM remove_due_to_license_issue Kd=620nM, IC50=13200nM, Ki=1800nM P07900 29528635 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 5w0e A 1.41 BS01 9U4 A 1 L1109 P1110 F1111 V1115 L1120 I1122 N1168 R1173 V1174 F1177 L27 P28 F29 V33 L38 I40 N86 R91 V92 F95 2.3.1.-,2.3.1.48 ic50=0.94nM remove_due_to_license_issue EC50=6.6nM, IC50=17nM Q92793 29155580 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5w0f A 1.6 BS01 9U7 A 1 L1109 P1110 F1111 V1115 L1120 I1122 N1168 R1173 V1174 L27 P28 F29 V33 L38 I40 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=16nM remove_due_to_license_issue IC50=16nM Q92793 28892380 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5w0i A 1.43 BS01 9UA A 1 L1109 P1110 V1115 L1120 I1122 N1168 R1173 V1174 F1177 L26 P27 V32 L37 I39 N85 R90 V91 F94 2.3.1.-,2.3.1.48 ic50=1.4nM remove_due_to_license_issue P45481 28892380 1201 IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5w0l A 1.549 BS01 9UD A 1 L1109 P1110 V1115 I1122 N1168 R1173 V1174 L27 P28 V33 I40 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=1.1nM remove_due_to_license_issue EC50=14nM, IC50=12nM Q92793 28892380 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 5w0q A 1.7 BS01 9UG A 1 P1110 F1111 L1120 N1168 V1174 P29 F30 L39 N87 V93 2.3.1.-,2.3.1.48 ic50=18uM remove_due_to_license_issue IC50=18000nM Q92793 28892380 1204 KKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 5w10 A 2.15 BS01 CMP A 1 N46 W47 S48 I67 G82 I83 A84 F105 V109 F115 T117 E136 N44 W45 S46 I65 G80 I81 A82 F103 V107 F113 T115 E134 ? Kd=0.24uM remove_due_to_license_issue Q72MQ6 28601495 201 LKDSKPELIKLYSSLGKIITSSLEQQEVLSAVMEEVRLFFSPKNWSLMRYDENSEELFFLIAEGIQFNHIRSIRLKSGEGIAGSVVQTKSPIFVENVKNDPRFSKKVDEKTGFETKTIIAVPMIFRGEVHGVIELVNRFDGSSFSPEDLVILQTIADFTAISLAHSDQYEKTK 5w12 A 1.88 BS01 9TG A 1 S64 Y150 S315 T316 R340 N343 S59 Y145 S310 T311 R335 N338 S64 K67 Y150 E272 K312 S315 S59 K62 Y145 E267 K307 S310 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144725 401 QEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5w13 A 1.95 BS01 SM2 A 1 S64 L119 Y150 G314 S315 T316 R340 S60 L115 Y146 G310 S311 T312 R336 S64 K67 Y150 E272 K312 S315 S60 K63 Y146 E268 K308 S311 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144725 401 DQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5w14 A 1.88 BS01 9TJ A 1 S64 Y150 Y222 G314 S315 S317 R340 S61 Y147 Y219 G311 S312 S314 R337 S64 K67 Y150 E272 K312 S315 S61 K64 Y147 E269 K309 S312 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144725 401 KDQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIKK 5w19 A 2.1 BS01 9TD A 1 F37 T50 Q99 G100 R101 F132 D133 T134 N194 D223 R226 S263 K266 R414 F459 F36 T49 Q98 G99 R100 F131 D132 T133 N193 D222 R225 S262 K265 R413 F458 Y72 F132 D133 D223 A225 K266 I391 H458 Y71 F131 D132 D222 A224 K265 I390 H457 4.1.99.1 0006520,0006568,0006569,0009034,0009072,0016829,0016830 Ki~5uM remove_due_to_license_issue P28796 30082510 502 AKRIVEPFRIKMVEKIRVPSREEREAALKEAGYNPFLLPSSAVYIDLLTDSGTNAMSDHQWAAMITGDEAYAGSRNYYDLKDKAKELFNYDYIIPAHQGRGAENILFPVLLKYKQKEGKAKNPVFISNFHFDTTAAHVELNGCKAINIVTEKAFDSETYDDWKGDFDIKKLKENIAQHGADNIVAIVSTVTCNSAGGQPVSMSNLKEVYEIAKQHGIFVVMDSARFCENAYFIKARDPKYKNATIKEVIFDMYKYADALTMSAKKDPLLNIGGLVAIRDNEEIFTLARQRCVPMEGFVTYGGLAGRDMAAMVQGLEEGTEEEYLHYRIGQVKYLGDRLREAGIPIQYPTGGHAVFVDCKKLVPQIPGDQFPAQAVINALYLESGVRAVEIGSFLLGRDPATGEQKHADMEFMRLTIARRVYTNDHMDYIADALIGLKEKFATLKGLEFEYEPPVLRHFTARLKPIE 5w19 B 2.1 BS01 9TD B 1 F37 T50 Q99 G100 R101 F132 D133 T134 N194 D223 R226 S263 K266 R414 F459 F36 T49 Q98 G99 R100 F131 D132 T133 N193 D222 R225 S262 K265 R413 F458 Y72 F132 D133 D223 A225 K266 I391 H458 Y71 F131 D132 D222 A224 K265 I390 H457 4.1.99.1 0006520,0006568,0006569,0009034,0009072,0016829,0016830 Ki~5uM remove_due_to_license_issue P28796 30082510 501 AKRIVEPFRIKMVEKIRVPSREEREAALKEAGYNPFLLPSSAVYIDLLTDSGTNAMSDHQWAAMITGDEAYAGSRNYYDLKDKAKELFNYDYIIPAHQGRGAENILFPVLLKYKQKEGKAKNPVFISNFHFDTTAAHVELNGCKAINIVTEKAFDSETYDDWKGDFDIKKLKENIAQHGADNIVAIVSTVTCNSAGGQPVSMSNLKEVYEIAKQHGIFVVMDSARFCENAYFIKARDPKYKNATIKEVIFDMYKYADALTMSAKKDPLLNIGGLVAIRDNEEIFTLARQRCVPMEGFVTYGGLAGRDMAAMVQGLEEGTEEEYLHYRIGQVKYLGDRLREAGIPIQYPTGGHAVFVDCKKLVPQIPGDQFPAQAVINALYLESGVRAVEIGSFLLGRDPATGEQKHADMEFMRLTIARRVYTNDHMDYIADALIGLKEKFATLKGLEFEYEPPVLRHFTARLKPIE 5w2m A 3.7 BS01 dna E 0 Y333 P350 P353 G356 L357 K358 Y359 Y144 P161 P164 G167 L168 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m B 3.7 BS01 dna E 0 Y333 K337 F351 K352 P353 K355 G356 L357 K358 Y359 Y144 K148 F162 K163 P164 K166 G167 L168 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m C 3.7 BS01 dna E 0 Y333 P353 W354 K355 G356 K358 Y359 Y144 P164 W165 K166 G167 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m D 3.7 BS01 dna E 0 Y333 W354 G356 K358 Y359 Y144 W165 G167 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m D 3.7 BS02 dna N 0 K352 K355 K163 K166 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m J 3.7 BS01 dna N 0 Y333 P350 P353 G356 L357 K358 Y359 Y144 P161 P164 G167 L168 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m K 3.7 BS01 dna N 0 Y333 K337 F351 K352 P353 K355 G356 L357 K358 Y359 Y144 K148 F162 K163 P164 K166 G167 L168 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m L 3.7 BS01 dna N 0 Y333 P353 W354 K355 G356 K358 Y359 Y144 P164 W165 K166 G167 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m M 3.7 BS01 dna E 0 K352 K355 K163 K166 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2m M 3.7 BS02 dna N 0 Y333 P353 W354 G356 K358 Y359 Y144 P164 W165 G167 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4 29191651 901 ~ 910 NPMEAMYPHIFYFHFKNLRKAYGRNESWLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5w2s A 2.399 BS01 KMG A 1 E120 E199 G200 P201 P206 E118 E197 G198 P199 P204 C171 H311 K340 H345 F402 F404 C169 H309 K338 H343 F400 F402 2.3.1.293 0004315,0005515,0005737,0005829,0005886,0006633,0009274,0016746,0016747,0019367,0030497,0042802 remove_due_to_license_issue P9WQD9 30563908 505 QPSTANGGFPSVVVTAVTATTSISPDIESTWKGLLAGESGIHALEDEFVTKWDLAVKIGGHLKDPVDSHMGRLDMRRMSYVQRMGKLLGGQLWESAGSPEVDPDRFAVVVGTGLGGAERIVESYDLMNAGGPRKVSPLAVQMIMPNGAAAVIGLQLGARAGVMTPVSACSSGSEAIAHAWRQIVMGDADVAVCGGVEGPIEALPIAAFSMMRAMSTRNDEPERASRPFDKDRDGFVFGEAGALMLIETEEHAKARGAKPLARLLGAGITSDAFHMVAPAADGVRAGRAMTRSLELAGLSPADIDHVNAHGTATPIGDAAEANAIRVAGCDQAAVYAPKSALGHSIGAVGALESVLTVLTLRDGVIPPTLNYETPDPEIDLDVVAGEPRYGDYRYAVNNSFGFGGHNVALAFGRY 5w34 A 2.95 BS01 dna D 0 G192 R193 G82 R83 2.7.7.101 0016779 remove_due_to_license_issue P9WNW1 29558114 3 ~ 9 MGSRSRLLAANAAAAAFYAQALQSDEAAPARQYLTERSFDAAAARKFGCGFAPSGWDSLTKHLQRKGFEFEELEAAGLSRQGRHGPMDRFHRRLLWPIRTSAGEVVGFGARRLFDDDAMEAKYVNTPETLLYKKSSVMFGIDLAKRDIAKGHQAVVVEGYTDVMAMHLAGVTTAVASCGTAFGGEHLAMLRRLMMDFFRGELIYVFDGDEAGRAAALKAFDGEQKLAGQSFVAVAPDGMDPCDLRLKCGDAALRDLVARRTPLFEFAIRAAIAEMDLDSAEGRVAALRRCVPMVGQIKDPTLRDEYARQLAGWVGWA 5w3i A 1.95 BS03 GY5 A 1 H41 E80 D108 E119 K134 H41 E61 D89 E100 K115 3.1.-.- 0003723,0039694 Ki=1.6uM remove_due_to_license_issue C3W5S0 29215062 304 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERAAAEL 5w44 A 2.1 BS02 GY6 A 1 Y24 E26 K34 H41 E61 D89 E100 K115 Y24 E26 K34 H41 E61 D89 E100 K115 3.1.-.- 0003723,0039694 Ki=0.36uM remove_due_to_license_issue C3W5S0 29215062 302 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERA 5w4r A 3.002 BS01 9WD A 1 C320 H323 M358 M365 V376 F377 F378 E379 I400 F401 C56 H59 M94 M101 V112 F113 F114 E115 I136 F137 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=33nM, IC50=46nM P51449 29079472 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQ 5w4v A 2.65 BS01 9WA A 1 L287 C320 L324 M365 F377 F378 E379 F388 I400 L21 C54 L58 M99 F111 F112 E113 F122 I134 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=5.0nM, IC50=89nM P51449 29079472 501 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSL 5w4v A 2.65 BS02 9WA B 1 M313 W317 M47 W51 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=5.0nM, IC50=89nM P51449 29079472 501 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSL 5w4v B 2.65 BS01 9WA A 1 M313 W317 M47 W51 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=5.0nM, IC50=89nM P51449 29079472 501 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSL 5w4v B 2.65 BS02 9WA B 1 C320 L324 M365 F377 F378 E379 F388 I400 C54 L58 M99 F111 F112 E113 F122 I134 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=5.0nM, IC50=89nM P51449 29079472 501 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSL 5w4w A 1.99 BS01 9WG A 1 I23 A36 K38 M80 M82 L85 I148 I21 A34 K36 M78 M80 L83 I146 D128 K130 D126 K128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=8nM remove_due_to_license_issue IC50=13nM P48730 28609096 4001 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 5w5j A 2.85 BS01 9WS A 1 V32 A45 V46 K47 L79 I93 T95 M98 L153 V24 A37 V38 K39 L51 I64 T66 M69 L124 D146 K148 Q150 N151 D164 T189 D117 K119 Q121 N122 D135 T137 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1500nM O43353 29057049 401 ALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHILHKARFSYILPILGICNEPFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFTIIYMPPENYEPIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5w5k A 2.7 BS02 K70 A 1 P464 H574 G582 F583 H614 F643 D705 L712 Y745 P28 H138 G146 F147 H178 F207 D269 L276 Y309 ? remove_due_to_license_issue F8W4B7 30645113 804 AGGSSPITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 5w5o A 2.89 BS01 9XA A 1 S25 V32 L79 T95 Y97 M98 G101 E105 L153 S21 V28 L66 T82 Y84 M85 G88 E92 L140 D146 K148 Q150 N151 D164 T189 D133 K135 Q137 N138 D151 T161 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=8.0nM O43353 29057049 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRMGTIIYMPPENYEPIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 5w5v A 3.645 BS01 ANW A 1 E87 F88 C89 G92 T96 M142 E75 F76 C77 G80 T84 M130 D135 K137 N140 D157 D123 K125 N128 D145 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=851nM Q9UHD2 30082428 701 MQSTSNHLWLLSDILTANVFRGRHKKTGDLFAIKVFVDVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFGEEYLHPDMYERATVDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILDQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVKVEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 5w6e A 1.9 BS02 0NY A 1 H223 H373 L388 F392 Q421 F424 H74 H224 L239 F243 Q272 F275 3.1.4.17 0004114,0007165,0008081 ic50=9.1nM remove_due_to_license_issue Q01064 29718668 1003 YSTAVLNCLKNLDLWCFDVFSLNQAADDHALRTIVFELLTRHNLISRFKIPTVFLMSFLDALETGYGKYKNPYHNQIHAADVTQTVHCFLLRTGMVHCLSEIELLAIIFAAAIHDYEHTGTTNSFHIQTKSECAIVYNDRSVLENHHISSVFRLMQDDEMNIFINLTKDEFVELRALVIEMVLATDMSCHFQQVKTMKTALQQLERIDKPKALSLLLHAADISHPTKQWLVHSRWTKALMEEFFRQGDKEAELGLPFSPLCDRTSTLVAQSQIGFIDFIVEPTFSVLTDVAEKSVQVVSFRSTWVKRIQENKQKWKERAAS 5w6o A 2.35 BS01 9X1 A 1 Y148 A176 M177 F200 P201 T252 Y256 E332 Y333 F341 L419 W420 Y68 A71 M72 F95 P96 T147 Y151 E227 Y228 F236 L314 W315 2.7.1.32,2.7.1.82 ic50=520nM remove_due_to_license_issue P35790 29389115 501 EQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5w6o B 2.35 BS01 9X1 B 1 Y148 M177 E180 F200 P201 Y256 Y333 F341 L419 W420 Y69 M73 E76 F96 P97 Y152 Y229 F237 L315 W316 2.7.1.32,2.7.1.82 ic50=520nM remove_due_to_license_issue P35790 29389115 501 DEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV 5w73 A 2.202 BS03 GY9 A 1 Y24 K34 I38 H41 E80 D108 E119 K134 K137 Y27 K37 I41 H44 E64 D92 E103 K118 K121 3.1.-.- 0003723,0039694 Ki=0.5uM remove_due_to_license_issue C3W5S0 29215062 205 GSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5w7u A 2.2 BS03 GY8 A 1 Y24 K34 A37 I38 H41 E80 D108 E119 K134 Y28 K38 A41 I42 H45 E65 D93 E104 K119 3.1.-.- 0003723,0039694 Ki=0.009uM remove_due_to_license_issue C3W5S0 29215062 203 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5w84 A 2.9 BS01 9YY A 1 M192 G193 V200 A211 K213 V246 Y262 V263 Y264 M265 G268 L318 D329 M28 G29 V36 A47 K49 V74 Y90 V91 Y92 M93 G96 L146 D157 D311 K313 A315 N316 D329 T351 D139 K141 A143 N144 D157 T174 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=360nM Q9NWZ3 28947151 4000 FHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLITTKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 5w85 A 2.25 BS01 9YS A 1 G193 V200 A211 K213 V246 Y262 V263 Y264 M265 P266 G268 D272 L318 G30 V36 A47 K49 V74 Y90 V91 Y92 M93 P94 G96 D100 L146 D311 K313 A315 N316 D329 T351 D139 K141 A143 N144 D157 T174 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=10nM remove_due_to_license_issue IC50=10.0nM Q9NWZ3 28947151 4000 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGFGVVYKGYVNNTTVAVKKLEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 5w86 A 2.61 BS01 9YV A 1 L828 A853 M902 E903 L905 G908 L956 L15 A37 M80 E81 L83 G86 L134 D949 A951 R953 N954 D967 D127 A129 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=2.0nM P52333 28947151 4000 PTIFEERHLKYISQLGKGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 5w88 A -1.00 BS01 9XG A 1 F27 L41 M45 M60 V72 F77 M80 I148 M153 F27 L41 M45 M60 V72 F77 M80 I103 M108 ? 0005509,0005861 remove_due_to_license_issue P19429,P63316 27825981 201 MDDIYKAAVEQLTEEQKNEFKAAFDIFVLGAEDGSISTKELGKVMRMLGQNPTPEELQEMIDEVDEDGSGTVDFDEFLVMMVRSMKDDSKGKFKRPTLRRVRISADAMMQALLGARAKGH 5w8h A 1.8 BS01 9Y1 A 1 L108 N137 R168 H192 G193 Y238 T247 L108 N137 R168 H192 G193 Y238 T247 R105 D165 R168 H192 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 ic50=23.4uM remove_due_to_license_issue IC50=23400nM P00338 29120638 501 ATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8h A 1.8 BS02 9Y1 A 2 G26 D51 V52 A95 I115 I119 G26 D51 V52 A95 I115 I119 R105 D165 R168 H192 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 ic50=23.4uM remove_due_to_license_issue IC50=23400nM P00338 29120638 502 ATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8h B 1.8 BS01 9Y1 B 1 S309 E310 R314 S309 E310 R314 R105 D165 R168 H192 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 ic50=23.4uM remove_due_to_license_issue IC50=23400nM P00338 29120638 402 ATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8i A 1.95 BS01 9YD A 1 Q99 R105 L108 N137 R168 H192 A237 T247 Q97 R103 L106 N135 R166 H190 A235 T245 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 ic50=0.15uM remove_due_to_license_issue IC50=>57000nM P00338 29120638 403 ATLKDQLIYNLLKQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8j A 1.55 BS01 9Y7 A 1 Q99 L108 N137 P138 D140 I141 R168 E191 H192 T247 L322 Q97 L106 N135 P136 D138 I139 R166 E189 H190 T245 L320 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 Kd=370nM remove_due_to_license_issue IC50=>57000nM, EC50=3530nM, Kd=370nM P00338 29120638 501 ATLKDQLIYNLLKQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8j A 1.55 BS02 9Y7 A 2 V25 G26 D51 V52 K80 Y82 A95 G96 I115 F118 I119 V23 G24 D49 V50 K78 Y80 A93 G94 I113 F116 I117 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 Kd=370nM remove_due_to_license_issue IC50=>57000nM, EC50=3530nM, Kd=370nM P00338 29120638 502 ATLKDQLIYNLLKQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8j B 1.55 BS01 9Y7 B 1 G26 D51 V52 K80 Y82 A95 G96 R98 I115 I119 G26 D51 V52 K80 Y82 A95 G96 R98 I115 I119 R105 D165 R168 H192 R105 D165 R168 H192 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 Kd=370nM remove_due_to_license_issue IC50=>57000nM, EC50=3530nM, Kd=370nM P00338 29120638 402 ATLKDQLIYNLLKEEQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8v A 2.346 BS01 9YP A 1 I135 D137 T138 G139 T141 K165 F186 V187 D193 I125 D127 T128 G129 T131 K155 F176 V177 D183 E133 D134 D137 F186 R199 E123 D124 D127 F176 R189 2.4.2.8 0000166,0000287,0001913,0001975,0004422,0005515,0005737,0005829,0006164,0006166,0006178,0007625,0007626,0016757,0021756,0021895,0021954,0032263,0032264,0042417,0042802,0043103,0044209,0045964,0046038,0046040,0046083,0046100,0046651,0046872,0048813,0051289,0052657,0070062,0071542 Ki=0.006uM remove_due_to_license_issue P00492 28813147 301 ASPGVVISDDEPGYDLDLFCIPNHYAEDLERVFIPHGLIMDRTERLARDVMKEMGGHHIVALCVLKGGYKFFADLLDYIKALNRNSDRSIPMTVDFIRLKSYIKVIGGDDLSTLTGKNVLIVEDIIDTGKTMQTLLSLVRQYNPKMVKVASLLVKRTPRSVGYKPDFVGFEIPDKFVVGYALDYNEYFRDLNHVCVISETGKAKYK 5w92 A 2.3 BS03 KU0 A 1 Y24 K34 I38 H41 E80 F105 L106 D108 E119 K134 K137 Y28 K38 I42 H45 E65 F90 L91 D93 E104 K119 K122 3.1.-.- 0003723,0039694 Ki=0.02uM remove_due_to_license_issue C3W5S0 29215062 203 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5w99 A 1.59 BS01 A1V A 1 E169 G174 V177 S178 S181 H182 L266 N269 T271 W272 V276 F282 R286 I328 G331 E168 G173 V176 S177 S180 H181 L254 N257 T259 W260 V264 F270 R274 I316 G319 ? remove_due_to_license_issue U5Q3T2 29158402 401 TWRRFDVAYHDPDLDRLILAARPLLSESPGRSWFQRHWVRGPHLELWFDHPEPSWERVREVLGTHLRAHPSRTRIDPDRLLPQHRRLALAEQIDEPLLPFYDDNTLHRAVPRSRVHVLGSAAAEDLFHDFHAAASTAAFDQLDAVVAGESRLGLAFELMIAAAHAHAEGGITGGFVSFRSHAEAFLAGAAGLRERWEAEYRTRAEALRAQVAAVVTGTPRGRAWTGLLDGFAGRGDELIASGALTPDTEFHRALRANRTWHDEVLRSPSFRRYRLLLNLTYLQMSRLGVTAVQRSLLCHFAASAVEEEYGVSAIEIAVG 5w9g A 2.1 BS03 KU2 A 1 Y24 I38 H41 E80 D108 E119 Y130 Y28 I42 H45 E65 D93 E104 Y115 3.1.-.- 0003723,0039694 Ki=0.15uM remove_due_to_license_issue C3W5S0 29215062 204 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5w9q A 1.8 BS01 dna C 0 R333 Q334 R336 K359 R369 Q370 R1 Q2 R4 K27 R37 Q38 ? 0003677,0008270 remove_due_to_license_issue Q9UIS9 29276034 1 ~ 12 RQNRKCGACAACLRRMDCGRCDFCCDKPKFGGSNQKRQKCRWRQCLQFAMKRLLPS 5w9q A 1.8 BS02 dna D 0 R333 R369 R384 R1 R37 R52 ? 0003677,0008270 remove_due_to_license_issue Q9UIS9 29276034 1 ~ 12 RQNRKCGACAACLRRMDCGRCDFCCDKPKFGGSNQKRQKCRWRQCLQFAMKRLLPS 5w9q B 1.8 BS01 dna E 0 Q334 R336 K359 R369 Q370 K371 R384 Q1 R3 K25 R35 Q36 K37 R50 ? 0003677,0008270 remove_due_to_license_issue Q9UIS9 29276034 1 ~ 12 QNRKCGCAACLRRMDCGRCDFCCDKPKFGGSNQKRQKCRWRQCLQFAMKRLLPS 5w9q B 1.8 BS02 dna F 0 R369 R384 R35 R50 ? 0003677,0008270 remove_due_to_license_issue Q9UIS9 29276034 1 ~ 12 QNRKCGCAACLRRMDCGRCDFCCDKPKFGGSNQKRQKCRWRQCLQFAMKRLLPS 5w9s C 2.1 BS01 dna A 0 K259 R260 H288 Q289 K295 L299 K2 R3 H31 Q32 K38 L42 ? 0003677,0008270 remove_due_to_license_issue Q7LFL8 29276034 1 ~ 12 KKRKRCGMCAPCRRRINCEQCSSCRNRKTGHQICKFRKCEELKK 5w9s C 2.1 BS02 dna B 0 S279 T286 G287 H288 S22 T29 G30 H31 ? 0003677,0008270 remove_due_to_license_issue Q7LFL8 29276034 1 ~ 12 KKRKRCGMCAPCRRRINCEQCSSCRNRKTGHQICKFRKCEELKK 5wa6 A 2.25 BS03 KU7 A 1 Y24 K34 I38 H41 E80 D108 E119 Y28 K38 I42 H45 E65 D93 E104 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 29215062 203 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wa7 A 2.204 BS03 KU4 A 1 A20 Y24 E26 K34 I38 H41 E119 A24 Y28 E30 K38 I42 H45 E104 3.1.-.- 0003723,0039694 Ki=0.4uM remove_due_to_license_issue C3W5S0 29215062 204 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wa8 A 1.3 BS01 9ZA A 1 I18 D43 I44 N99 G105 S107 N112 H114 I7 D32 I33 N88 G94 S96 N101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=0.587uM remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVNLHVLGGRQMHWPPG 5wa9 A 1.15 BS01 9ZD A 1 I18 D43 I44 N99 G105 Q106 S107 N112 H114 I7 D32 I33 N88 G94 Q95 S96 N101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=0.175uM remove_due_to_license_issue P49773 28968488 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVNLHVLGGRQMHWPPG 5wac A 2.061 BS01 A1M A 1 S64 Q120 Y150 V212 N213 T313 G314 S315 S317 S61 Q117 Y147 V209 N210 T310 G311 S312 S314 S64 K67 Y150 E272 K312 S315 S61 K64 Y147 E269 K309 S312 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144724 401 KDQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5wad A 2.09 BS01 QQZ A 1 S64 L119 Q120 Y150 V212 N213 Y222 T313 G314 S315 T316 S317 S58 L113 Q114 Y144 V206 N207 Y216 T307 G308 S309 T310 S311 S64 K67 Y150 E272 K312 S315 S58 K61 Y144 E266 K306 S309 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144724 401 EIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5wae A 1.804 BS01 A1J A 1 S64 Y150 V212 Y222 T313 G314 S315 S317 S61 Y147 V209 Y219 T310 G311 S312 S314 S64 K67 Y150 E272 K312 S315 S61 K64 Y147 E269 K309 S312 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144724 401 KDQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5waf A 2.03 BS01 A0Y A 1 S64 Q120 Y150 V212 N213 T313 G314 S315 T316 S317 R340 S59 Q115 Y145 V207 N208 T308 G309 S310 T311 S312 R335 S64 K67 Y150 E272 K312 S315 S59 K62 Y145 E267 K307 S310 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144724 401 QEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5wag B 1.931 BS01 A0V B 1 S64 K67 Q120 Y150 T313 S315 R340 S64 K67 Q120 Y150 T313 S315 R340 S64 K67 Y150 E272 K312 S315 S64 K67 Y150 E272 K312 S315 3.5.2.6 0008800,0016787,0017001,0030288,0046677 remove_due_to_license_issue Q6DRA1 29144724 401 NTPKDQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEMYYGLQSVQDKKAVNSNTIFELGSVSKLFTATAGGYAKNKGKISFDDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPALGLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLSFIHANLNPQKYPTDIQRAINETHQGRYQVNTMYQALGWEEFSYPATLQTLLDSNSEQIVMKPNKVTAISKEPSVKMYHKTGSTSGFGTYVVFIPKENIGLVMLTNKRIPNEERIKAAYVVLNAIK 5wal A 2.45 BS01 9ZS A 1 L903 G904 E905 V911 A928 I960 Y980 V981 P982 G984 L1030 L14 G15 E16 V22 A39 I71 Y91 V92 P93 G95 L141 N1023 A1025 R1027 N1028 D1041 P1064 N134 A136 R138 N139 D152 P173 2.7.10.2 0004672,0005524,0006468 Ki=0.0017uM remove_due_to_license_issue P29597 28830649 1201 TVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYR 5wap A 2.201 BS03 KU9 A 1 Y24 I38 H41 E80 D108 E119 Y28 I42 H45 E65 D93 E104 3.1.-.- 0003723,0039694 Ki=0.3uM remove_due_to_license_issue C3W5S0 29215062 204 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wb3 A 2.203 BS03 GYA A 1 A20 Y24 K34 I38 H41 E80 D108 E119 A24 Y28 K38 I42 H45 E65 D93 E104 3.1.-.- 0003723,0039694 Ki=0.06uM remove_due_to_license_issue C3W5S0 29215062 205 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wb6 A 2.35 BS01 9ZM A 1 R39 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=0.02nM remove_due_to_license_issue Ki=0.020000nM P03951 28780160 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 5wbm A 2.16 BS01 A4G A 1 A226 G229 A230 C282 C289 A224 G227 A228 C280 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 Kd=20uM remove_due_to_license_issue IC50=120226nM, Kd=20000nM P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbm B 2.16 BS01 A4G B 1 R77 W88 R81 W92 G255 A256 G257 D258 G259 A260 G261 D262 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 Kd=20uM remove_due_to_license_issue IC50=120226nM, Kd=20000nM P50053 28853885 301 SGLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbm B 2.16 BS02 A4G B 2 A226 A256 C282 C289 A230 A260 C286 C293 G255 A256 G257 D258 G259 A260 G261 D262 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 Kd=20uM remove_due_to_license_issue IC50=120226nM, Kd=20000nM P50053 28853885 302 SGLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbo A 2.25 BS01 A1Y A 1 A226 F260 A224 F258 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 Kd=62uM remove_due_to_license_issue Kd=62000nM, IC50=319000nM P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbo B 2.25 BS01 A1Y B 1 A226 F260 C289 A229 F263 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 Kd=62uM remove_due_to_license_issue Kd=62000nM, IC50=319000nM P50053 28853885 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbp A 2.74 BS01 A2J A 1 A226 A285 C289 A224 A283 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbq A 2.4 BS01 A3J A 1 A224 A226 P246 G257 F260 A285 G286 C289 A222 A224 P244 G255 F258 A283 G284 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=1.48uM remove_due_to_license_issue IC50=1480nM P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbq B 2.4 BS01 A3J B 1 A224 A226 E227 P246 P247 A256 C289 A227 A229 E230 P249 P250 A259 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=1.48uM remove_due_to_license_issue IC50=1480nM P50053 28853885 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbr A 2.58 BS01 A3Y A 1 N107 A224 A226 E227 T253 A256 G257 C289 N105 A222 A224 E225 T251 A254 G255 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=16790nM P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbr B 2.58 BS01 A3Y B 1 A224 A226 T253 G257 C289 A227 A229 T256 G260 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 remove_due_to_license_issue IC50=16790nM P50053 28853885 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbz A 2.4 BS01 A4J A 1 N107 A224 A226 E227 P246 A256 G257 F260 G286 C289 N105 A222 A224 E225 P244 A254 G255 F258 G284 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=0.39uM remove_due_to_license_issue IC50=450nM P50053 28853885 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wbz B 2.4 BS01 A4J B 1 A224 A226 E227 T253 G257 C289 A227 A229 E230 T256 G260 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=0.39uM remove_due_to_license_issue IC50=450nM P50053 28853885 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 5wcl A -1.00 BS01 9XG A 1 L41 M60 F77 M80 R83 T142 L41 M60 F77 M80 R83 T97 ? 0005509,0005861 remove_due_to_license_issue P19429,P63316 27825981 201 MDDIYKAAVEQLTEEQKNEFKAAFDIFVLGAEDGSISTKELGKVMRMLGQNPTPEELQEMIDEVDEDGSGTVDFDEFLVMMVRSMKDDSKGKFKRPTLRRVRISADAMMQALLGARAKGH 5wcm A 1.2 BS06 4NZ A 1 W34 L104 D105 L145 H177 L207 H242 W3 L73 D74 L114 H146 L176 H211 H101 H103 D105 H106 H177 N208 H242 H70 H72 D74 H75 H146 N177 H211 ? 0046872 remove_due_to_license_issue Q89GW5 20696874 307 KKWTAPFEPFQLIDNIYYVGTDGIAVYVIKTSQGLILMDTAMPQSTGMIKDNIAKLGFKVADIKLILNTHAHLDHTGGFAEIKKETGAQLVAGERDKPLLEGGYYPGDEKNEDLAFPAVKVDRAVKEGDRVTLGDTTLTAHATPGHSPGCTSWEMTVKDGKEDREVLFFCSGTVALNRLVGQPTYAGIVDDYRATFAKAKAMKIDVLLGPHPEVYGMQAKRAEMKDGAPNPFIKPGELVTYATSLSEDFDKQLAKQTAALEKK 5wdc A 2.1 BS03 G2K A 1 A20 Y24 K34 H41 E80 D108 E119 A24 Y28 K38 H45 E65 D93 E104 3.1.-.- 0003723,0039694 Ki=0.4uM remove_due_to_license_issue C3W5S0 29215062 205 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKISEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wdj B 2.4 BS01 AEY A 1 T238 R239 E242 F366 T126 R127 E130 F254 1.11.2.2 0004601,0006979,0020037 remove_due_to_license_issue IC50=110nM P05164 30108726 201 VNCETSCVQQPPCFPLKIPPNDPRIKNQADCIPFFRSCPACPGSNITIRNQINALTSFVDASMVYGSEEPLARNLRNMSNQLGLLAVNQRFQDNGRALLPFDNLHDDPCLLTNRSARIPCFLAGDTRSSEMPELTSMHTLLLREHNRLATELKSLNPRWDGERLYQEARKIVGAMVQIITYRDYLPLVLGPTAMRKYLPTYRSYNDSVDPRIANVFTNAFRYGHTLIQPFMFRLDNRYQPMEPNPRVPLSRVFFASWRVVLEGGIDPILRGLMATPAKLNRQNQIAVDEIRERLFEQVMRIGLDLPALNMQRSRDHGLPGYNAWRRFCGLPQPETVGQLGTVLRNLKLARKLMEQYGTPNNIDIWMGGVSEPLKRKGRVGPLLACIIGTQFRKLRDGDRFWWENEGVFSMQQRQALAQISLPRIICDNTGITTVSKNNIFMSNSYPRDFVNCSTLPALNLASWREA 5wdl A 2.625 BS01 R33 A 1 G54 C56 G108 G109 D237 D338 D339 H340 G22 C24 G76 G77 D205 D305 D306 H307 ? 0004177,0005737,0006508,0008234,0009401,0009636,0016020,0043418,0046872,0070005 remove_due_to_license_issue A6LE66 30085657 501 GFVFTTVKENPITSVKNQNRAGTCWCYSSYSFLESELLRMGKGEYDLSEMFTVYNTYLDRADAAVRTHGDVSFSQGGSFYDALYGMETFGLVPEEEMRPGMMYADTLSNHTELSALTDAMVAAIAKGKLRKLQSDENNAMLWKKAVAAVHQIYLGVPPEKFTYKGKEYTPKSFFESTGLKASDYVSLTSYTHHPFYTQFPLEIQDNWRHGMSYNLPLDEFMEVFDNAINTGYTIAWGSDVSESGFTRDGVAVMPDDEKVQELSSDMAHWLKLKPEEKKLNTKPQPQKWCTQAERQLAYDNYETTDDHGMQIYGIAKDQEGNEYYMVKNSWGTNSKYNGIWYASKAFVRYKTMNIVVHKDALPKAIKAKLGIK 5wdw A 2.3 BS03 8KU A 1 Y24 K34 A37 I38 H41 E80 D108 Y28 K38 A41 I42 H45 E65 D93 3.1.-.- 0003723,0039694 Ki=0.29uM remove_due_to_license_issue C3W5S0 29215062 203 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5we9 A 1.804 BS03 GY7 A 1 Y24 H41 E80 D108 E119 K134 Y24 H41 E61 D89 E100 K115 3.1.-.- 0003723,0039694 Ki=0.06uM remove_due_to_license_issue C3W5S0 29215062 303 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERA 5web A 2.254 BS03 KU5 A 1 Y24 E26 K34 H41 E80 L106 E119 Y28 E30 K38 H45 E65 L91 E104 3.1.-.- 0003723,0039694 Ki=0.01uM remove_due_to_license_issue C3W5S0 29215062 203 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wef A 2.0 BS03 GY6 A 1 A20 Y24 H41 E80 D108 E119 K134 A20 Y24 H41 E61 D89 E100 K115 3.1.-.- 0003723,0039694 Ki=0.36uM remove_due_to_license_issue C3W5S0 29215062 303 MEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKSLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERA 5wei A 2.25 BS03 GY6 A 1 Y24 K34 H41 D108 Y28 K38 H45 D93 3.1.-.- 0003723,0039694 Ki=2uM remove_due_to_license_issue C3W5S0 29215062 206 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIDIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wej A 1.95 BS01 V45 A 1 H30 I109 T134 C139 H157 A158 A159 A160 H30 I109 T133 C138 H156 A157 A158 A159 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 29227928 201 APPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQRLVHGQSGMLLTGANAKGMDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 5wep A 3.502 BS01 A81 A 1 H7 T9 W34 Y39 W46 C48 H7 T9 W34 Y39 W46 C48 ? 0016740,0046872 remove_due_to_license_issue D7UQM0 30642934 201 MLQGLNHLTLAVSDLASSLAFYQQLPGMRLHASWDSGAYLSCGALWLCLSLDEQRRKTPPQESDYTHYAFSVAEEEFAGVVALLAQAGAEVWKDNRSEGASYYFLDPDGHKLELHVGNLAQRLAACRERPYKGMVFFD 5wep A 3.502 BS03 A81 B 1 Y65 H67 Y131 Y65 H67 Y131 ? 0016740,0046872 remove_due_to_license_issue D7UQM0 30642934 201 MLQGLNHLTLAVSDLASSLAFYQQLPGMRLHASWDSGAYLSCGALWLCLSLDEQRRKTPPQESDYTHYAFSVAEEEFAGVVALLAQAGAEVWKDNRSEGASYYFLDPDGHKLELHVGNLAQRLAACRERPYKGMVFFD 5wep B 3.502 BS01 A81 A 1 Y65 H67 Y131 Y65 H67 Y127 ? 0016740,0046872 remove_due_to_license_issue D7UQM0 30642934 201 MLQGLNHLTLAVSDLASSLAFYQQLPGMRLHASWDSGAYLSCGALWLCLSLDEQRRKTPPQESDYTHYAFSVAEEEFAGVVALLAQAGAEVWKDNASYYFLDPDGHKLELHVGNLAQRLAACRERPYKGMVFF 5wep B 3.502 BS02 A81 B 1 H7 T9 Y39 W46 C48 H7 T9 Y39 W46 C48 ? 0016740,0046872 remove_due_to_license_issue D7UQM0 30642934 201 MLQGLNHLTLAVSDLASSLAFYQQLPGMRLHASWDSGAYLSCGALWLCLSLDEQRRKTPPQESDYTHYAFSVAEEEFAGVVALLAQAGAEVWKDNASYYFLDPDGHKLELHVGNLAQRLAACRERPYKGMVFF 5wev A 1.854 BS01 9ZS A 1 L855 Y931 L932 G935 L983 L23 Y96 L97 G100 L148 D976 A978 R980 N981 D994 S1016 D141 A143 R145 N146 D159 S181 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.15uM remove_due_to_license_issue O60674 28830649 1201 SGAFEDRDPTQFEERHLKFLQQLGKGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 5wew A 3.178 BS02 A81 A 1 Y65 H67 R122 Y131 Y65 H67 R122 Y131 ? 0046872 remove_due_to_license_issue W8UNW6 30642934 202 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFEQH 5wew A 3.178 BS03 A81 B 1 H7 T9 Y39 W46 C48 H7 T9 Y39 W46 C48 ? 0046872 remove_due_to_license_issue W8UNW6 30642934 202 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFEQH 5wew B 3.178 BS01 A81 A 1 H7 T9 Y39 W46 H7 T9 Y39 W46 ? 0046872 remove_due_to_license_issue W8UNW6 30642934 202 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFEQHH 5wew B 3.178 BS03 A81 B 1 Y65 H67 Y131 Y65 H67 Y131 ? 0046872 remove_due_to_license_issue W8UNW6 30642934 202 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFEQHH 5wex A 1.26 BS02 8JS A 1 H94 H119 F131 L198 T199 T200 P202 H92 H117 F128 L195 T196 T197 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=66.3nM remove_due_to_license_issue Ki=14nM P00918 28947945 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wf3 A 2.251 BS03 KU2 A 1 Y24 I38 H41 D108 Y28 I42 H45 D93 3.1.-.- 0003723,0039694 Ki=1.4uM remove_due_to_license_issue C3W5S0 29215062 205 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIDIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wf5 A 2.6 BS01 UKA A 1 S67 T88 Q89 F168 E169 W246 L249 H250 N253 T256 H264 M270 Y271 I274 S277 H278 S65 T86 Q87 F158 E159 W383 L386 H387 N390 T393 H401 M407 Y408 I411 S414 H415 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P29274 29395784 1201 IMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAANIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYRSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHV 5wf6 A 2.9 BS01 UKA A 1 L85 T88 L167 F168 E169 W246 L249 H250 N253 T256 H264 M270 Y271 I274 S277 H278 L83 T86 L154 F155 E156 W380 L383 H384 N387 T390 H398 M404 Y405 I408 S411 H412 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P29274 29395784 1201 IMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSAIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYRSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHV 5wf7 B 2.5 BS09 A9G B 1 Y303 R304 G808 Y809 R843 V853 Y878 Y103 R104 G511 Y512 R546 V552 Y577 ? 0006338,0042054 ic50=98.5uM remove_due_to_license_issue G0RYC6,G0SDW4 29904056 8009 WTVDKIASALSVLAEEVPQNHSRLVNFLLEETEKRAPQPRHLSKTDPFAHMKSKAIDAPEGVPTMDVKFKQHSGEYGKSRNSGRRFQYPVVCIKPDREPVPPYRFHHAEIRKNILALNSQLNFVPPRSQKIAKRAQAEYAATLAPYLEPWLRKLNIEGCTKSNLIRFMASDMSPQAVRNASMFTEAWDRVFNDQSKLRRVALRDILMLDKNVEPIFDNKRAKALMQKVIDALGSYTTLGCLICFSHDCEHGEIERDNQKRCFSLEEIGGLMPSLRRKWAAQIEQHPPCRNECYRIHGPPWSENEVGTLEWMFATIGYSQTLRPECFVGAILGRPCWDVHRKLQELDLPPVEIPKQKSLPWYDRRKKQLMSDWADATITHEHAVRELFAPCHHDGPCTAANGCPCASAGTHPVLCERFCLCTAEECPLKFTGCACHSSGKTCLQRQGRPCICVQLNRECDPTLCKGCGARERADPENAYDEVLHSTGCQNVALQRGAAKAVVLGKSQLEACGYGLFAAEDIEEGEFVIEYTGELISHDEGVRREHRRGDVNKVSYLFTLLEQEGIWVDAAIYGNLSRYINHATDGNIMPKIMYVNHEWRIKFTAIKDIKAGEELFFNYGDNFPNLTKKLVEPLLVPKTTQPLFDPLSKVQLLPGQPLPQHPIDDSWLLLKHRDNLQDFIDLRPEEKEFLQEWDAFILRRHISSEQYLPRYFLRFVREKADWLVSKRSRGEEFSKLVATLLARRVLPERVVIEATQVLNDARGRLRE 5wfc B 2.282 BS09 A97 B 1 I302 Y303 Y304 H307 G808 Y809 R843 R877 Y878 I100 Y101 Y102 H105 G522 Y523 R557 R582 Y583 ? 0006338,0042054 ic50=12.5uM remove_due_to_license_issue G0RYC6,G0SDW4 29904056 8009 EWTVDKIASALSVLAEEVPQNHSRLVNFLLEETEKRAPQPRHLSKTDPFAHMKSKAIDGVPTMDVKFKQHSGEYGKSRNSGRRFQYPVVCIKPDREPVPIYYFHHAEIRKNILALNSQLNPRSQKIAKRAQAEYAATLAPYLEPWLRKLNIEGCTKSNLIRFMASQPESDDSMTPQQKSNLLDTYSDDMGSPQAVRNASMFTEAWDRVFNDQSKLRRVALRDILMLDKNVEPIFDNKRAKLMQKVIDALGSYTTLGCLICFSHDCEHGEIERDNQKRCFSLEEIGGLMPSLRRKWAAQIEQHPPCRNECYRIHGVPPWSENEVGTLEWMFATIGYSQTLRPECFVGAILGRPCWDVHRKLQEIPKQKSLPWYDRRKKQLMSDWADATITHEHAVRELFAPCHHDGPCTAANGCPCASAGTHPVLCERFCLCTAEECPLKFTGCACHSSGKTCLQRQGRPCICVQLNRECDPTLCKGCGARERADPENAYDEVLHSTGCQNVALQRGAAKAVVLGKSQLEACGYGLFAAEDIEEGEFVIEYTGELISHDEGVRREHRRGSFLFTLLEQEGIWVDAAIYGNLSRYINHATDGNIMPKIMYVNHEWRIKFTAIKDIKAGEELFFNYGDNFPNLTKKLPLLVPKTTQPLFDPLSKVQLLPGQPLPQHPIDDSWLLLKHRDNLQDFIDLRPEEKEFLQEWDAFILRRHISSEQYLPRYFLRFVREKADWLVSKRSRGEEFSKLVATLLARRVLPERVVIEATQVLNDARGRLRE 5wfd B 2.654 BS09 A9G B 1 I302 Y303 Y304 H307 G808 Y809 R843 Y878 I99 Y100 Y101 H104 G530 Y531 R565 Y590 ? 0006338,0042054 remove_due_to_license_issue G0RYC6,G0SDW4 29904056 8009 EWTVDKIASALSVLAEEVPQNHSRLVNFLLEETEKRAPQPRHLSKTDPFAHMKSKAIGVPTMDVKFKQHSGEYGKSRNSGRRFQYPVVCIKPDREPVPIYYFHHAEIRKNILALNSQLNPRSQKIAKRAQAEYAATLAPYLEPWLRKLNIEGCTKSNLIRFMASQPESDDSMTPQQKSNLLDTYSDDMGSPQAVRNASMFTEAWDRVFNDQSKLRRVALRDILMLDKNVEPIFDNKRAKLMQKVIDALGSYTTLGCLICFSHDCEHGEIERDNQKRCFSLEEIGGLMPSLRRKWAAQIEQHPPCRNECYRIHGNQQVPPWSENEVGTLEWMFATIGYSQTLRPECFVGAILGRPCWDVHRKLQELPPVEPTIPKQKSLPWYDRRKKQLMSDWADATITHEHAVRELFAPCHHDGPCTAANGCPCASAGTHPVLCERFCLCTAEECPLKFTGCACHSSGKTCLQRQGRPCICVQLNRECDPTLCKGCGARERADPENAYDEVLHSTGQNVALQRGAAKAVVLGKSQLEACGYGLFAAEDIEEGEFVIEYTGELISHDEGVRREHRRGFLFTLLEQEGIWVDAAIYGNLSRYINHATDGNIMPKIMYVNHEWRIKFTAIKDIKAGEELFFNYGDNFPNLTRPLLVPKTTQPLFDPLSKVQLLPGQPLPQHPIDDSWLLLKHRDNLQDFIDLRPEEKEFLQEWDAFILRRHISSEQYLPRYFLRFVREKADWLVSKRSRGEEFSKLVATLLARRVLPERVVIEATQVLNDARGRLRE 5wfj A 2.48 BS01 9Z4 A 1 V836 A853 M902 E903 Y904 L905 C909 R953 L956 V16 A33 M75 E76 Y77 L78 C82 R126 L129 D949 A951 R953 N954 D967 D122 A124 R126 N127 D140 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 28927786 4000 FEERHLKYISQLGGSVELCRYDPLGDNTGALVAVKQLQPDQQRDFQREIQILKALHSDFIVKYRGVSYGPLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 5wfm A 2.251 BS03 KU5 A 1 Y24 I38 H41 E80 F105 L106 D108 D119 Y27 I41 H44 E64 F89 L90 D92 D103 3.1.-.- 0003723,0039694 Ki=0.3uM remove_due_to_license_issue C3W5S0 29215062 205 GSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIDIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wfw A 2.292 BS03 GYA A 1 A20 Y24 E26 I38 H41 D108 K134 A24 Y28 E30 I42 H45 D93 K119 3.1.-.- 0003723,0039694 Ki=0.8uM remove_due_to_license_issue C3W5S0 29215062 205 RGSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIDIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wfz A 2.35 BS03 KU0 A 1 K34 I38 H41 F105 L106 D108 D119 K134 K37 I41 H44 F89 L90 D92 D103 K118 3.1.-.- 0003723,0039694 Ki<0.01uM remove_due_to_license_issue C3W5S0 29215062 205 GSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIDIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wg3 A 2.896 BS01 AFM A 1 R199 G200 F202 G203 V205 K220 E239 M274 D278 A321 L324 D335 R170 G171 F173 G174 V176 K191 E210 M245 D249 A292 L295 D306 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue P25098 29070696 701 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRTKDKHEIDRMTLTVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVNAADAEDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 5wg4 A 2.31 BS01 AFV A 1 R199 G200 F202 G203 V205 A218 L222 E239 M274 A321 L324 D335 A480 R169 G170 F172 G173 V175 A188 L192 E209 M244 A291 L294 D305 A448 D317 K319 N322 D335 K344 T353 D287 K289 N292 D305 K314 T323 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue P25098 29070696 701 KILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRGEVNAADATKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 5wg5 A 3.1 BS01 ZSO A 1 I197 R199 G200 A218 K220 M274 A321 L324 I164 R166 G167 A185 K187 M241 A288 L291 D317 K319 N322 D335 K344 T353 D284 K286 N289 D302 K311 T320 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue P25098 29070696 701 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPVNAADAFDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 5wg6 A 3.901 BS08 A9G A 1 I109 W624 Y658 Y661 F665 T678 R685 F686 N688 I73 W285 Y319 Y322 F326 T339 R346 F347 N349 2.1.1.356,2.1.1.43 0000082,0000122,0000781,0000785,0000976,0000978,0000979,0001222,0003677,0003682,0003714,0003723,0005515,0005634,0005654,0005677,0005694,0005721,0006325,0006338,0006346,0006355,0006357,0008168,0008284,0009913,0010468,0010629,0010718,0014013,0014834,0014898,0016279,0021695,0021766,0030097,0030183,0030216,0030335,0031048,0031490,0031491,0031507,0031509,0032259,0032355,0034244,0035098,0035984,0036211,0036333,0042054,0042127,0042393,0042752,0043021,0043406,0043547,0043565,0045120,0045202,0045605,0045617,0045814,0045892,0046976,0048387,0048511,0048863,0050767,0051154,0051932,0070301,0070314,0070878,0071168,0071902,0090183,0097421,0106222,0140718,0140938,0140951,1900006,1900016,1902808,1904772,1990841,2000134,2000737 remove_due_to_license_issue Q15022,Q15910 29904056 9009 RFRRADEVKSMFSSNRQKILERTEILNQEWKQRRIQPVHILTSVRECSVTSDLDFPTQVIPLKTLNAVASVPIMYSWSPLQQNFMVEDTPNIDGPNAKSVQREQSLHSFHTLFCRRCFKYDCFLHPFHATPNTYKRWSGAEASMFRVLIGTYYDNFCAIARLIGTKTCRQVYEFRVKVYNYQPCDHPRQPCDSSCPCVIAQNFCEKFCQCSSECQNRFPGCRCKAQCNTKQCPCYLAVRECDPDLCLTCGAADHRDSKNVSCKNCSIQRGSKKHLLLAPSDVAGWGIFIKDPVQKNEFISEYCGEIISQDEADRRGKVYDKYMCSFLFNLNNDFVVDATRKGNKIRFANHSVNPNCYAKVMMVNGDHRIGIFAKRAIQTGEELFFDYRYSQNRLYFHSDTCLPLRPQEMEVDSEDEKDPEWLREKTITQIEEFSDVNEGEKEVMKLWNLHVMKHGFIADNQMNHACMLFVENYGQKIIKKNLCRNFMLHLVSMHDFNLISIMSIDKAVTKLREMQQK 5wg7 A 1.45 BS01 AUD A 1 H94 L198 T199 T200 H91 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wg7 A 1.45 BS02 AUD A 2 L164 D165 K228 L229 L160 D161 K224 L225 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wg7 A 1.45 BS03 AUD A 3 K111 K113 K108 K110 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wg7 A 1.45 BS04 AUD A 4 G6 Y7 G8 F231 E239 G3 Y4 G5 F227 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wg8 A 1.65 BS03 LB1 A 1 D242 H244 D271 H304 H427 E428 F446 Y451 D71 H73 D100 H133 H256 E257 F275 Y280 D242 H244 D271 D274 R275 N303 H304 H352 R400 H427 D71 H73 D100 D103 R104 N132 H133 H181 R229 H256 3.1.3.16 0016787 remove_due_to_license_issue P53041 30679389 503 IEDEYSGPKLEDGKVTISFMKELMQWYKDQKKLHRKCAYQILVQVKEVLSKLSTLVETTLKETEKITVCGDTHGQFYDLLNIFELNGLPSETNPYIFNGDFVDRGSFSVEVILTLFGFKLLYPDHFHLLRGNHETDNMNQIYGFEGEVKAKYTAQMYELFSEVFEWLPLAQCINGKVLIMHGGLFSEDGVTLDDIRKIERNRQPPDSGPMCDLLWSDPQPQNGRSISKRGVSCQFGPDVTKAFLEENNLDYIIRSHEVKAEGYEVAHGGRCVTVFSAPNYCDQMGNKASYIHLQGSDLRPQFHQFTAVPHPNVKPMAYAN 5wg9 A 2.3 BS03 KU4 A 1 A20 Y24 I38 H41 D108 D119 K134 A23 Y27 I41 H44 D92 D103 K118 3.1.-.- 0003723,0039694 Ki=2.6uM remove_due_to_license_issue C3W5S0 29215062 205 GSHMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDGGSKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIDIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 5wgp A 1.53 BS02 AUD A 1 H94 H96 H119 V143 L198 T199 T200 H91 H93 H116 V139 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wgp A 1.53 BS03 AUD A 2 G6 Y7 G8 F231 E239 G3 Y4 G5 F227 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wgp A 1.53 BS04 AUD A 3 L164 D165 K228 L229 L160 D161 K224 L225 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=>20000nM P00918 29266943 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wh5 A 1.8 BS01 R91 A 1 Y159 N321 Y329 W332 T333 I336 M357 S368 Q369 F372 Y74 N236 Y244 W247 T248 I251 M272 S283 Q284 F287 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 29975048 501 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 5wh6 A 1.6 BS01 AKJ A 1 N321 Y329 W332 T333 I336 F340 M357 S368 Q369 F372 N236 Y244 W247 T248 I251 F255 M272 S283 Q284 F287 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=18nM Q08499 29975048 601 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 5whc A 2.548 BS01 AJJ A 1 C300 R301 D305 Y348 D349 H403 C92 R93 D97 Y140 D141 H195 3.4.19.12 0004843,0016579 remove_due_to_license_issue IC50=79200nM, Kd=12000nM Q93009 29166018 601 KHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQK 5wi0 A 2.05 BS01 AQ1 A 1 H191 F193 R196 D219 S241 V242 A244 S275 R311 H171 F173 R176 D199 S221 V222 A224 S255 R291 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=360uM remove_due_to_license_issue IC50=360000nM P43490 29287958 901 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5wi0 A 2.05 BS02 AQ1 B 1 D16 Y18 D8 Y10 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=360uM remove_due_to_license_issue IC50=360000nM P43490 29287958 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5wi1 A 1.99 BS01 AOY A 1 F193 R196 D219 V242 A244 S275 R311 F173 R176 D199 V222 A224 S255 R291 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=10uM remove_due_to_license_issue IC50=10000nM P43490 29287958 901 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5wi1 A 1.99 BS02 AOY B 1 D16 Y18 D8 Y10 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=10uM remove_due_to_license_issue IC50=10000nM P43490 29287958 501 FNILLATDSYKVTHYKQYPPNTSKVYSYFECREYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 5wic B 2.55 BS01 FOA B 1 Q119 D148 Q31 D60 ? 0016020 remove_due_to_license_issue Q17U16 29097752 301 RDQTSYGDEIDKFWLTQYVIHRESYDFYSVQVDYTAVGLMSTPNVAESYQSKFKGRNGLDKVLGDSETTRVKINSVILDKPHGVATIRFTTVRRVRSNPVDDQPQRWIAIMGYEYKSLAMNAEQRYVNPLGFRVTSYRVNPE 5wic B 2.55 BS02 FOA B 2 R110 S112 Y137 K140 R22 S24 Y49 K52 ? 0016020 remove_due_to_license_issue Q17U16 29097752 302 RDQTSYGDEIDKFWLTQYVIHRESYDFYSVQVDYTAVGLMSTPNVAESYQSKFKGRNGLDKVLGDSETTRVKINSVILDKPHGVATIRFTTVRRVRSNPVDDQPQRWIAIMGYEYKSLAMNAEQRYVNPLGFRVTSYRVNPE 5wii A 2.79 BS01 AO4 A 1 R110 E111 S112 R21 E22 S23 ? 0016020 remove_due_to_license_issue Q17U16 29097752 301 DQTSYGDEIDKFWLTQYVIHRESYDFYSVQVDYTAVGLMSTPNVAESYQSKFKGRNGLDKVLGDSETTRVKINSVILDKPHGVATIRFTTVRRVRSNPVDDQPQRWIAIMGYEYKSLAMNAEQRYVNPLGFRVTSYRVNPE 5wij A 2.04 BS01 AQG A 1 L551 I559 L579 E627 F628 V629 K630 F631 G632 L680 L16 I24 L44 E92 F93 V94 K95 F96 G97 L145 N673 K677 N678 D699 N138 K142 N143 D164 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue O60674 30763067 901 VFHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSLF 5win A 2.38 BS01 SKE A 1 L551 I559 L579 F628 V629 K630 G632 L680 L16 I24 L44 F93 V94 K95 G97 L145 N673 K677 N678 D699 N138 K142 N143 D164 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue Kd=220nM, IC50=2960nM, Ki=220000nM O60674 30763067 901 VFHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSLF 5wio A 2.52 BS01 XXE A 1 I108 Y113 D114 D121 T156 T157 R158 I21 Y26 D27 D34 T69 T70 R71 ? 0016020 remove_due_to_license_issue Q17U16 29097752 301 TRDQTSYGDEIDKFWLTQYVIHRESYDFYSVQVDYTAVGLMSTPNVAESYQSKFKGRNGLDKVLGDSETTRVKINSVILDKPHGVATIRFTTVRRVRSNPVDDQPQRWIAIMGYEYKSLAMNAEQRYVNPLGFRVTSYRVNPE 5wip A 2.62 BS01 XXO A 1 H109 R110 S112 Y113 D121 Y137 K140 H22 R23 S25 Y26 D34 Y50 K53 ? 0016020 remove_due_to_license_issue Q17U16 29097752 301 TRDQTSYGDEIDKFWLTQYVIHRESYDFYSVQVDYTAVGLMSTPNVAESYQSKFKGRNGLDKVLGDSETTRVKINSVILDKPHGVATIRFTTVRRVRSNPVDDQPQRWIAIMGYEYKSLAMNAEQRYVNPLGFRVTSYRVNPE 5wj6 A 2.445 BS01 B4A A 1 R317 K320 L321 F322 L323 N324 E325 Y394 R181 K184 L185 F186 L187 N188 E189 Y258 S286 K289 Y414 Y466 V484 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 Kd=27nM remove_due_to_license_issue IC50=29nM O94925 29317493 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTADGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5wj6 C 2.445 BS01 B4A C 1 K320 L321 F322 L323 N324 E325 Y394 K184 L185 F186 L187 N188 E189 Y258 S286 K289 Y414 Y466 V484 S150 K153 Y278 Y330 V348 3.5.1.2 0004359,0006541 Kd=27nM remove_due_to_license_issue IC50=29nM O94925 29317493 601 PSLEDLLFYTIAEGQEKIPVHKFITALKSTGLRTSDPRLKECMDMLRLTLQTTSDGVMLDKDLFKKCVQSNIVLLTQAFRRKFVIPDFMSFTSHIDELYESAKKQSGGKVADYIPQLAKFSPDLWGVSVCTADGQRHSTGDTKVPFCLQSCVKPLKYAIAVNDLGTEYVHRYVGKEPSGLRFNKLFLNEDDKPHNPMVNAGAIVVTSLIKQGVNNAEKFDYVMQFLNKMAGNEYVGFSNATFQSERESGDRNFAIGYYLKEKKCFPEGTDMVGILDFYFQLCSIEVTCESASVMAATLANGGFCPITGERVLSPEAVRNTLSLMHSCGMYDFSGQFAFHVGLPAKSGVAGGILLVVPNVMGMMCWSPPLDKMGNSVKGIHFCHDLVSLCNFHNYDNLRHFAKKLDPRREG 5wjj A 1.6 BS01 AQY A 1 V30 Y35 V38 A51 K53 L75 L104 V105 T106 M109 F169 G170 L171 A172 H174 V26 Y31 V34 A47 K49 L71 L100 V101 T102 M105 F165 G166 L167 A168 H170 D150 K152 N155 D168 T185 D146 K148 N151 D164 T175 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=5.4nM remove_due_to_license_issue IC50=5.4nM Q16539 29291937 501 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARHTDDATRWYRAPEIMLNWHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 5wkl A 1.85 BS01 AVY A 1 H41 F143 C145 C148 H166 Q167 M168 E169 D190 Q192 H43 F142 C144 C147 H165 Q166 M167 E168 D189 Q191 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0008233,0019082 remove_due_to_license_issue K9N638 29544147 401 HHSGLVKMSHPSGDVEACMVQVTCGSMTLNGLWLDNTVWCPRHVMCPADQLSDPNYDALLISMTNHSFSVQKHIANLRVVGHAMQGTLLKLTVDVANPSTPAYTFTTVKPGAAFSVLACYNGRPTGTFTVVMRPNYTIKGSFLCGSCGSVGYTKEGSVINFCYMHQMELANGTHTGSAFDGTMYGAFMDKQVHQVQLTDKYCSVNVVAWLYAAILNGCAWFVKPNRTSVVSFNEWALANQFTEFVGTQSVDMLAVKTGVAIEQLLYAIQQLYTGFQGKQILGSTMLEDEFTPEDVNMQIMGVV 5wkm A 2.25 BS01 N02 A 1 F143 C148 H166 Q167 M168 E169 D190 F140 C145 H163 Q164 M165 E166 D187 2.7.7.50,3.4.19.12,3.4.22.-,3.4.22.69 0008233,0019082 remove_due_to_license_issue K9N638 29544147 401 HHSGLVKMSHPSGDVEACMVQVTCGSMTLNGLWLDNTVWCPRHVMCPQLSDPNYDALLISMTNHSFSVQKHIANLRVVGHAMQGTLLKLTVDVANPSTPAYTFTTVKPGAAFSVLACYNGRPTGTFTVVMRPNYTIKGSFLCGSCGSVGYTKEGSVINFCYMHQMELANGTHTGSAFDGTMYGAFMDKQVHQVQLTDKYCSVNVVAWLYAAILNGCAWFVKPNRTSVVSFNEWALANQFTEFVGTQSVDMLAVKTGVAIEQLLYAIQQLYTGFQGKQILGSTMLEDEFTPEDVNMQIMGVV 5wl0 A 2.4 BS01 21G A 1 F323 F325 S337 H357 E361 K376 F404 Q406 M431 N510 V511 F72 F74 S86 H106 E110 K125 F153 Q155 M180 N255 V256 ? 0003723,0006351 Kd=0.67nM remove_due_to_license_issue Q67296 28839261 801 NDDIDQSLIIAARNIVRRASVSADPLASLLEMCHSTQIGGTRMVDILRQNPTEEQAVDICKAAMGLRISSSFSFGGFTFKRTSGSSIKREEEVLTGNLQTLKIRVHEGYEEFTMVGKRATAILRKATRRLVQLIVSGRDEQSIAEAIIVAMVFSQEDCMIKAVRGDLNFVNRANQRLNPMHQLLRHFQKDAKVLFQNWGIEHIDNVMGMVGVLPDMTPSTEMSMRGIRVSKMGVSTERVVVSIDRFLRVRDQRGNVLLSPEEVSETHGTERLTITYSSSMMWEINGPESVLVNTYQWIIRNWETVKIQWSQNPTMLYNKMEFEPFQSLVPKAIRGQYSGFVRTLFQQMRDVLGTFDTTQIIKLLPFAAAPPKQSRMQFSSLTVNVRGSGMRILVRGNSPVFNYNKTTKRLTILGKDAGTLIEDPDESTSGVESAVLRGFLILGKEDRRYGPALSINELSNLAKGEKANVLIGQGDVVLVMKR 5wlo A 1.27 BS01 GR7 B 1 D25 A28 D30 G48 P81 V82 I84 D25 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 3.1.13.2,3.1.26.13 0004190,0006508 remove_due_to_license_issue Q72498 28958624 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5wlo B 1.27 BS01 GR7 B 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.1.13.2,3.1.26.13 0004190,0006508 Ki=0.015nM remove_due_to_license_issue Q72498 28958624 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 5wlt A 1.57 BS02 86B A 1 H94 H119 T199 T200 H91 H116 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=155.5nM remove_due_to_license_issue P00918 29851481 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wlt A 1.57 BS03 86B A 2 N67 E69 D71 D72 S73 I91 Q92 N64 E66 D68 D69 S70 I88 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=155.5nM remove_due_to_license_issue P00918 29851481 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wlt A 1.57 BS04 86B A 3 W5 H15 D19 W2 H12 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=155.5nM remove_due_to_license_issue P00918 29851481 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wlt A 1.57 BS05 86B A 4 D72 W123 G129 D130 F131 G132 D69 W120 G125 D126 F127 G128 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=155.5nM remove_due_to_license_issue P00918 29851481 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wlv A 1.4 BS02 42G A 1 Q92 H94 H96 H119 F131 L198 T199 T200 Q89 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3nM remove_due_to_license_issue P00918 29851481 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wlv A 1.4 BS03 42G A 2 D72 D130 F131 G132 D69 D126 F127 G128 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3nM remove_due_to_license_issue P00918 29851481 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 5wmt A 2.748 BS01 9QY A 1 N107 D149 M154 N162 F195 T245 I247 N34 D76 M81 N89 F109 T159 I161 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Ki=440nM, IC50=1100nM, Kd=1380nM P41148 29528635 405 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 5wo4 A 1.84 BS01 B7V A 1 L881 G882 V889 A906 F958 L959 G962 E966 R1007 N1008 L1010 G1020 L28 G29 V36 A53 F98 L99 G102 E106 R147 N148 L150 G160 D1003 A1005 R1007 N1008 D1021 D1040 D143 A145 R147 N148 D161 D180 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.1nM remove_due_to_license_issue IC50=0.100000nM P23458 29156136 2001 DIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 5wp5 A 1.5 BS01 SAH A 1 V263 S264 G290 G292 D312 L313 M317 D338 C339 R355 T357 H360 V235 S236 G262 G264 D284 L285 M289 D310 C311 R327 T329 H332 2.1.1.103 0000234,0003729,0005737,0006656,0008168,0008654,0009058,0032259,0052667 Kd=4.6uM remove_due_to_license_issue Q944H0 29084845 501 EERDIQKSYWMEHRPEVLSLIPPYEGKSVLELGAGIGRFTGELAQKAGEVIALDFIESAIQKNESVNGHYKNIKFMCADVTSPDLKIKDGSIDLIFSNWLLMYLSDKEVELMAERMIGWVKPGGYIFFRESCFHQSGDSKRKSNPTHYREPRFYTKVFQECQTRDASGNSFELSMVGCKCIGAYVKNKKNQNQICWIWQKVSVENDKDFQRFLDNVQYKSSGILRYERVFGEGYVSTGGFETTKEFVAKMDLKPGQKVLDVGCGIGGGDFYMAENFDVHVVGIDLSVNMISFALERAIGLKCSVEFEVADCTTKTYPDNSFDVIYSRDTILHIQDKPALFRTFFKWLKPGGKVLITDYCRSAETPSPEFAEYIKQRGYDLHDVQAYGQMLKDAGFDDVIAEDRTDQFVQVLRRELEKVEKEKEEFISDFSEEDYNDIVGGWSAKLERTASGEQKWGLFIADKK 5wp5 A 1.5 BS02 SAH A 2 W16 G61 R66 F67 D82 F83 D107 V108 N126 W127 W10 G33 R38 F39 D54 F55 D79 V80 N98 W99 2.1.1.103 0000234,0003729,0005737,0006656,0008168,0008654,0009058,0032259,0052667 Kd=4.6uM remove_due_to_license_issue Q944H0 29084845 502 EERDIQKSYWMEHRPEVLSLIPPYEGKSVLELGAGIGRFTGELAQKAGEVIALDFIESAIQKNESVNGHYKNIKFMCADVTSPDLKIKDGSIDLIFSNWLLMYLSDKEVELMAERMIGWVKPGGYIFFRESCFHQSGDSKRKSNPTHYREPRFYTKVFQECQTRDASGNSFELSMVGCKCIGAYVKNKKNQNQICWIWQKVSVENDKDFQRFLDNVQYKSSGILRYERVFGEGYVSTGGFETTKEFVAKMDLKPGQKVLDVGCGIGGGDFYMAENFDVHVVGIDLSVNMISFALERAIGLKCSVEFEVADCTTKTYPDNSFDVIYSRDTILHIQDKPALFRTFFKWLKPGGKVLITDYCRSAETPSPEFAEYIKQRGYDLHDVQAYGQMLKDAGFDDVIAEDRTDQFVQVLRRELEKVEKEKEEFISDFSEEDYNDIVGGWSAKLERTASGEQKWGLFIADKK 5wpb A 1.55 BS04 B8P A 1 W1143 G1154 R1155 S1175 D1178 W1182 Y1184 Y1189 W37 G48 R49 S69 D72 W76 Y78 Y83 3.5.1.-,3.5.1.98 0008270 remove_due_to_license_issue IC50=270000nM Q9UBN7 29019676 1304 GSPLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKF 5wqa A 2.3 BS01 J20 A 1 H160 S208 M273 H276 F340 Q343 P356 M357 Q369 F372 I376 H82 S130 M195 H198 F262 Q265 P278 M279 Q291 F294 I298 3.1.4.53 0004114,0007165,0008081 ic50=0.011uM remove_due_to_license_issue IC50=10.0nM Q08499 28159622 501 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 5wqc A 1.96 BS01 7MA A 1 P131 Q134 F227 I320 N324 H350 V353 Y354 P93 Q96 F186 I436 N440 H466 V469 Y470 ? 0004930,0007186,0007631,0016020,0016499 remove_due_to_license_issue O43614,Q9V2J8 29225076 2001 FLRYLWREYLHPKEYEWVLIAGYIIVFVVALIGNVLVCVAVWKNHHMRTVTNYFIVNLSLADVLVTITCLPATLVVDITETWFFGQSLCKVIPYLQTVSVSVSVLTLSCIALDRWYAICHPLMFKSTAKRARNSIVIIWIVSCIIMIPQAIVMECSTVFPNKTTLFTVCDERWGGEIYPKMYHICFFLVTYMAPLCLMVLAYLQIFRKLWCRQGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKQIRARRKTARMLMVVLLVFAICYLPISILNVLKRVFGMFAHTEDRETVYAWFTFSHWLVYANSAANPIIYNFLSGKFREEFKAAFSCCC 5wqj A 1.2 BS01 7N3 A 1 W36 L38 P39 D73 H74 Y108 R188 P196 R197 C248 G249 S250 V252 V277 W28 L30 P31 D65 H66 Y100 R180 P188 R189 C240 G241 S242 V244 V269 D63 H74 R188 C248 G249 S250 G251 V252 T253 A254 S275 D55 H66 R180 C240 G241 S242 G243 V244 T245 A246 S267 2.8.1.2 0001822,0001889,0004792,0005737,0005739,0005743,0016740,0016783,0016784,0019346,0021510,0042802,0043005,0045202,0070814 Kd=3uM remove_due_to_license_issue Q99J99 28079151 301 QLFRALVSAQWVAEALKAQPLKLLDASWYLPKLGRDARREFEERHIPGAAFFDIDRSSDHTSPYDHMLPNATHFADYAGSLGVSAATHVVIYDGSDQGLYSAPRVWWMFRAFGHHSVSLLDGGFRHWLNQNLPISSGKSHSEPAEFSAQLDPSFIKTHEDILENLDARRFQVVDARAAGRFQGTQPEPRDGIEPGHIPGSVNIPFTEFLTNEGLEKSPEEIKRLFKEKKVDLSKPLVATCGSGVTASHVVLGAFLSGKSDVPVYDGSWVEWYMRAQPEHIISEGRGKT 5wqk A 1.7 BS01 7NC A 1 W36 P39 D73 H74 R188 P196 R197 C248 G249 S250 V252 W32 P35 D69 H70 R184 P192 R193 C244 G245 S246 V248 D63 H74 R188 C248 G249 S250 G251 V252 T253 A254 S275 D59 H70 R184 C244 G245 S246 G247 V248 T249 A250 S271 2.8.1.2 0001822,0001889,0004792,0005737,0005739,0005743,0016740,0016783,0016784,0019346,0021510,0042802,0043005,0045202,0070814 Kd=0.5uM remove_due_to_license_issue Q99J99 28079151 301 QLFRALVSAQWVAEALKAPRSSQPLKLLDASWYLPKLGRDARREFEERHIPGAAFFDIDRSSDHTSPYDHMLPNATHFADYAGSLGVSAATHVVIYDGSDQGLYSAPRVWWMFRAFGHHSVSLLDGGFRHWLNQNLPISSGKSHSEPAEFSAQLDPSFIKTHEDILENLDARRFQVVDARAAGRFQGTQPEPRDGIEPGHIPGSVNIPFTEFLTNEGLEKSPEEIKRLFKEKKVDLSKPLVATCGSGVTASHVVLGAFLSGKSDVPVYDGSWVEWYMRAQPEHIISEGRGKTQ 5wr7 A 2.76 BS01 RCH A 1 L516 V524 A542 K544 E560 L564 I572 V573 F589 M592 G595 L657 G667 D668 F669 L28 V36 A54 K56 E72 L76 I84 V85 F101 M104 G107 L169 G179 D180 F181 D650 R654 N655 D668 D162 R166 N167 D180 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=1.5nM P04629 30242093 801 HIIENPQYFSDACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYL 5wre A 1.946 BS01 7TL A 1 F23 P25 D29 T33 W102 I105 F110 Y118 I139 L140 S141 F23 P25 D29 T33 W102 I105 F110 Y118 I139 L140 S141 ? 0005198 ic50=0.39uM remove_due_to_license_issue L7R9I1 28205569 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHCSPHHTALRQAILCWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISCLTFGRETVLEYLVSFGVWIRTPPAARPPNAPILST 5wre A 1.946 BS02 7TL F 1 V124 W125 T128 A132 R133 P134 V124 W125 T128 A132 R133 P134 ? 0005198 ic50=0.39uM remove_due_to_license_issue L7R9I1 28205569 201 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHCSPHHTALRQAILCWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISCLTFGRETVLEYLVSFGVWIRTPPAARPPNAPILST 5wrs A 2.75 BS01 ATP A 1 Y125 K129 K233 P279 S341 A342 F343 L344 S346 L347 R352 Y37 K41 K139 P185 S247 A248 F249 L250 S252 L253 R258 ? remove_due_to_license_issue Q96MK3 28432788 604 SSKLQALFAHPLYNVPEEPPLLGAEDSLLASQEALRYYRRKVARWNRRHKMYREQMDPPLQLRLEASWVQFHLGINRHGLYSRSSPVVSKLLQDMRHFPTISADYSQDEKALLGACDCTQIVKSGVHLKLVLRFSDFGKAMFKPMRQQRDEETPVDFFYFIDFQRHNAEIAAFHLDRILDFRRVPPTVGRIVNVTKEILEVTKNEILQSVFFVSPASNVCFFAKCPYMCKTEYAVCGKPHLLEGSLSAFLPSLNLAPRLSVPNPWIRSYTLAGKEEWEVNPLYCDTVKQIYPYNNSQRLLNVIDMAIFDFLIGNMDRHHYEMFTKFGDDGFLIHLDNARGFGRHSHDEISILSPLSQCCMIKKKTLLHLQLLAQADYRLSDVMRESLLEDQLSPVLTEPHLLALDRRLQTILRTVEGCIVAHGQQSVIVDG 5wrs B 2.75 BS01 ATP B 1 Y125 K129 K233 P279 A342 F343 S346 L347 R352 Y37 K41 K142 P188 A251 F252 S255 L256 R261 ? remove_due_to_license_issue Q96MK3 28432788 604 SSKLQALFAHPLYNVPEEPPLLGAEDSLLASQEALRYYRRKVARWNRRHKMYREQMNLDPPLQLRLEASWVQFHLGINRHGLYSRSSPVVSKLLQDMRHFPTISADYSQDEKALLGACDCTQIVKPSGVHLKLVLRFSDFGKAMFKPMRQQRDEETPVDFFYFIDFQRHNAEIAAFHLDRILDFRRVPPTVGRIVNVTKEILEVTKNEILQSVFFVSPASNVCFFAKCPYMCKTEYAVCGKPHLLEGSLSAFLPSLNLAPRLSVPNPWIRSYTLAGKEEWEVNPLYCDTVKQIYPYNNSQRLLNVIDMAIFDFLIGNMDRHHYEMFTKFGDDGFLIHLDNARGFGRHSHDEISILSPLSQCCMIKKKTLLHLQLLAQADYRLSDVMRESLLEDQLSPVLTEPHLLALDRRLQTILRTVEGCIVAHGQQSVIVDGP 5ws3 A 2.3 BS01 7MA A 1 P131 Q134 Q187 F227 I320 N324 H350 V353 Y354 P97 Q100 Q153 F193 I443 N447 H473 V476 Y477 ? 0004930,0007186,0007631,0016020,0016499 remove_due_to_license_issue O43614,Q9V2J8 29225076 2001 DDEEFLRYLWREYLHPKEYEWVLIAGYIIVFVVALIGNVLVCVAVWKNHHMRTVTNYFIVNLSLADVLVTITCLPATLVVDITETWFFGQSLCKVIPYLQTVSVSVSVLTLSCIALDRWYAICHPLMFKSTAKRARNSIVIIWIVSCIIMIPQAIVMECSTVFPGLANKTTLFTVCDERWGGEIYPKMYHICFFLVTYMAPLCLMVLAYLQIFRKLWCRQGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKQIRARRKTARMLMVVLLVFAICYLPISILNVLKRVFGMFAHTEDRETVYAWFTFSHWLVYANSAANPIIYNFLSGKFREEFKAAFSCCC 5wuk A 2.03 BS02 73K A 1 F97 Y148 N194 K211 L240 D310 Y365 R367 R414 F22 Y73 N119 K136 L165 D235 Y290 R292 R339 ? Kd=14nM remove_due_to_license_issue Kd=82nM, IC50=53.5nM O75530 28111304 502 KKCKYSFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCDMDHSLKLWRINSKRMMNAIKESYDYNPNKTNRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLEVEDPHKAKCTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDRLR 5wuu A 1.724 BS01 7UU A 1 W81 P82 L92 L94 N140 D145 I146 W39 P40 L50 L52 N98 D103 I104 ? ic50=0.81uM remove_due_to_license_issue IC50=810nM O60885 28347667 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5wvd A 3.0 BS01 7UX A 1 E53 L55 L108 K126 L127 Q128 G129 L177 D191 F192 E13 L15 L68 K86 L87 Q88 G89 L137 D151 F152 D170 K172 N175 D191 D130 K132 N135 D151 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9BUB5 29497019 402 PGKFEDMYKLTSELLGEGAYAKVQGAVSLQNGKEYAVKIIEKQAGHSRSRVFREVETLYQCQGNKNILELIEFFEDDTRFYLVFEKLQGGSILAHIQKQKHFNEREASRVVRDVAAALDFLHTKGIAHRDLKPENILCESPEKVSPVKICDFDLGSGYMAPEVVEVFTDQATFYDKRCDLWSLGVVLYIMLSGYPPFKYEFPDKDWAHISSEAKDLISKLLVRDAKQRLSAAQVLQHPWVQ 5wvd B 3.0 BS01 7UX B 1 L55 V63 L108 L127 G129 L177 D191 F192 L15 V23 L68 L87 G89 L128 D140 F141 D170 K172 N175 D191 D121 K123 N126 D140 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9BUB5 29497019 401 PGKFEDMYKLTSELLGEGAYAKVQGAVSLQNGKEYAVKIIEKQAGHSRSRVFREVETLYQCQGNKNILELIEFFEDDTRFYLVFEKLQGGSILAHIQASRVVRDVAAALDFLHTKGIAHRDLKPENILCESPVSPVKICDFDLGSGMEYMAPEVVEVFTDQATFYDKRCDLWSLGVVLYIMLSGYPDLISKLLVRDAKQRLSAAQVLQHPWV 5wwe A 2.4 BS01 rna B 0 E18 Q19 K22 F24 D49 V51 M53 R62 F64 F66 A96 V97 R99 S102 H108 E4 Q5 K8 F10 D35 V37 M39 R48 F50 F52 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P22626 29379020 1 ~ 10 REKEQFRKLFIGGLSFETTEESLRNYYEQWGKLTDCVVMRDPASKRSRGFGFVTFSSMAEVDAAMAARPHSIDGRVVEPKRAVAREESGKPGAHVTVKKLFVGGIKEDTEEHHLRDYFEEYGKIDTIEIITDRKKRGFGFVTFDDHDPVDKIVLQKYHTINGHNAEVRKALSRQ 5wwf A 2.15 BS01 rna B 0 E18 K22 F24 D49 V51 M53 F64 F66 K94 A96 V97 R99 H108 E3 K7 F9 D34 V36 M38 F49 F51 K79 A81 V82 R84 H93 ? 0003676,0003723 remove_due_to_license_issue P22626 29379020 1 ~ 10 EKEQFRKLFIGGLSFETTEESLRNYYEQWGKLTDCVVMRDPASKRSRGFGFVTFSSMAEVDAAMAARPHSIDGRVVEPKRAVAREESGKPGAHVTVKKLFVGGIKEDTEEHHLRDYFEEYGKIDTIEIITDRQSGKKRGFGFVTFDDHDPVDKIVLQKYHTINGHNAEVRKALSRQEM 5wwf C 2.15 BS01 rna D 0 E18 K22 F24 D49 V51 M53 F64 F66 A96 V97 R99 H108 E2 K6 F8 D33 V35 M37 F48 F50 A80 V81 R83 H92 ? 0003676,0003723 remove_due_to_license_issue P22626 29379020 1 ~ 10 KEQFRKLFIGGLSFETTEESLRNYYEQWGKLTDCVVMRDPASKRSRGFGFVTFSSMAEVDAAMAARPHSIDGRVVEPKRAVAREESGKPGAHVTVKKLFVGGIKEDTEEHHLRDYFEEYGKIDTIEIITDRQSGKKRGFGFVTFDDHDPVDKIVLQKYHTINGHNAEVRKALSRQE 5wwg A 2.03 BS01 rna B 0 Q19 K22 F24 D49 V51 M53 R62 F64 F66 E92 A96 V97 R99 H108 Q8 K11 F13 D38 V40 M42 R51 F53 F55 E81 A85 V86 R88 H97 ? 0003676,0003723 remove_due_to_license_issue P22626 29379020 1 ~ 8 RKKREKEQFRKLFIGGLSFETTEESLRNYYEQWGKLTDCVVMRDPASKRSRGFGFVTFSSMAEVDAAMAARPHSIDGRVVEPKRAVAREESGKPGAHVTVKKLFVGGIKEDTEEHHLRDYFEEYGKIDTIEIITDRQSGKKRGFGFVTFDDHDPVDKIVLQKYHTINGHNAEVRKALSRQEMQE 5wyq A 2.16 BS01 SAM A 1 Y91 L92 S93 P94 Q95 G118 Y120 E121 S137 Y141 L143 G145 G146 P149 Y89 L90 S91 P92 Q93 G116 Y118 E119 S135 Y139 L141 G143 G144 P147 P94 E121 R159 P92 E119 R157 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 401 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyq A 2.16 BS02 SAM B 1 D182 H185 D170 H173 P94 E121 R159 P92 E119 R157 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 301 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyq B 2.16 BS01 SAM A 1 D182 H185 D172 H175 P94 E121 R159 D174 P92 E119 R157 D164 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 401 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyq B 2.16 BS02 SAM B 1 Y91 L92 S93 P94 Q95 G118 Y120 E121 I138 L143 G145 G146 P149 Y89 L90 S91 P92 Q93 G116 Y118 E119 I136 L141 G143 G144 P147 P94 E121 R159 D174 P92 E119 R157 D164 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 301 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyr A 2.45 BS01 SFG A 1 Y91 L92 S93 P94 Q95 G118 Y120 E121 S137 I138 L143 G145 G146 P149 Y89 L90 S91 P92 Q93 G116 Y118 E119 S135 I136 L141 G143 G144 P147 P94 E121 R159 D174 P92 E119 R157 D166 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 400 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALGEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyr A 2.45 BS02 SFG B 1 S175 D182 S167 D174 P94 E121 R159 D174 P92 E119 R157 D166 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 400 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALGEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyr B 2.45 BS01 SFG A 1 D174 S175 D182 D172 S173 D180 P94 E121 R159 D174 P92 E119 R157 D172 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 400 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALGHADSAEEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wyr B 2.45 BS02 SFG B 1 Y91 L92 S93 P94 G118 Y120 E121 I138 V142 L143 S144 G145 G146 P149 Y89 L90 S91 P92 G116 Y118 E119 I136 V140 L141 S142 G143 G144 P147 P94 E121 R159 D174 P92 E119 R157 D172 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q02RL6 31399541 400 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALGHADSAEEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 5wys A 2.999 BS01 7V6 A 1 R218 F247 E311 A313 G315 G316 R337 T346 S347 A348 R214 F243 E307 A309 G311 G312 R333 T342 S343 A344 S198 R218 H245 T343 E344 K443 Q448 K529 S196 R214 H241 T339 E340 K439 Q444 K525 1.13.12.7 0004497,0005524,0005777,0008218,0016405,0046872,0047077,0051087 remove_due_to_license_issue P08659 28492074 601 DAKNIKKGPAPFYPLEDGTAGEQLHKAMKRYALVPGTIAFTDAHIEVNITYAEYFEMSVRLAEAMKRYGLNTNHRIVVCSENSLQFFMPVLGALFIGVAVAPANDIYNERELLNSMNISQPTVVFVSKKGLQKILNVQKKLPIIQKIIIMDSKTDYQGFQSMYTFVTSHLPPGFNEYDFVPESFDRDKTIALIMNSSTGLPKGVALPHRTACVRFSHARDPIFGNQIIPDTAILSVVPFHHGFGMFTTLGYLICGFRVVLMYRFEEELFLRSLQDYKIQSALLVPTLFSFFAKSTLIDKYDLSNLHEIASGGAPLSKEVGEAVAKRFHLPGIRQGYGLTETTSAILITPEGDDKPGAVGKVVPFFEAKVVDLDTGKTLGVNQRGELCVRGPMIMSGYVNNPEATNALIDKDGWLHSGDIAYWDEDEHFFIVDRLKSLIKYKGYQVAPAELESILLQHPNIFDAGVAGLPDDDAGELPAAVVVLEHGKTMTEKEIVDYVASQVTTAKKLRGGVVFVDEVPKGLTGKLDARKIREILIKAK 5wyx A 2.4 BS02 CU8 A 1 F495 A518 Q519 F427 A450 Q451 ? 0002224,0004888,0006955,0016020 Kd=0.22uM remove_due_to_license_issue Q9NR97 29155428 916 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSALETKTTTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 5wyx A 2.4 BS03 CU8 B 1 F261 Y348 G351 F405 F219 Y306 G309 F363 ? 0002224,0004888,0006955,0016020 Kd=0.22uM remove_due_to_license_issue Q9NR97 29155428 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSALETKTTTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 5wyx B 2.4 BS01 CU8 A 1 F261 Y348 G351 F405 F218 Y305 G308 F362 ? 0002224,0004888,0006955,0016020 Kd=0.22uM remove_due_to_license_issue Q9NR97 29155428 916 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVKFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLEL 5wyx B 2.4 BS02 CU8 B 1 F495 A518 Q519 F427 A450 Q451 ? 0002224,0004888,0006955,0016020 Kd=0.22uM remove_due_to_license_issue Q9NR97 29155428 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVKFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLEL 5wyz A 2.3 BS01 7VF A 1 F494 F495 A518 Q519 V520 Y567 F426 F427 A450 Q451 V452 Y499 ? 0002224,0004888,0006955,0016020 Kd=21nM remove_due_to_license_issue Q9NR97 29155428 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSALETKTTTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 5wyz A 2.3 BS02 7VF B 1 F261 Y348 G351 F405 F219 Y306 G309 F363 ? 0002224,0004888,0006955,0016020 Kd=21nM remove_due_to_license_issue Q9NR97 29155428 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKSALETKTTTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 5wyz B 2.3 BS01 7VF A 1 F261 Y348 K350 G351 F405 F219 Y306 K308 G309 F363 ? 0002224,0004888,0006955,0016020 Kd=21nM remove_due_to_license_issue Q9NR97 29155428 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVKDTFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 5wyz B 2.3 BS02 7VF B 1 F494 F495 A518 Q519 Y567 F429 F430 A453 Q454 Y502 ? 0002224,0004888,0006955,0016020 Kd=21nM remove_due_to_license_issue Q9NR97 29155428 901 RSYPCDEKKQNDSVIAECSNRRLQEVPQTVGKYVTELDLSDNFITHITNESFQGLQNLTKINLNHNPNVNGLNITDGAFLNLKNLRELLLEDNQLPQIPSGLPESLTELSLIQNNIYNITKEGISRLINLKNLYLAWNCYFNKVCEKTNIEDGVFETLTNLELLSLSFNSLSHVPPKLPSSLRKLFLSNTQIKYISEEDFKGLINLTLLDLSGNCPRCFNAPFPCVPCDGGASINIDRFAFQNLTQLRYLNLSSTSLRKINAAWFKNMPHLKVLDLEFNYLVGEIASGAFLTMLPRLEILDLSFNYIKGSYPQHINISRNFSKLLSLRALHLRGYVFQELREDDFQPLMQLPNLSTINLGINFIKQIDFKLFQNFSNLEIIYLSENRISPLVKDTFDPHSNFYHFTRPLIKPQCAAYGKALDLSLNSIFFIGPNQFENLPDIACLNLSANSNAQVLSGTEFSAIPHVKYLDLTNNRLDFDNASALTELSDLEVLDLSYNSHYFRIAGVTHHLEFIQNFTNLKVLNLSHNNIYTLTDKYNLESKSLVELVFSGNRLDILWNDDDNRYISIFKGLKNLTRLDLSLNRLKHIPNEAFLNLPASLTELHINDNMLKFFNWTLLQQFPRLELLDLRGNKLLFLTDSLSDFTSSLRTLLLSHNRISHLPSGFLSEVSSLKHLDLSSNLLKTINKTKLSMLELHGNPFECTCDIGDFRRWMDEHLNVKIPRLVDVICASPGDQRGKSIVSLE 5wzg A 2.55 BS01 rna B 0 S138 H139 Q142 R171 S174 H175 E178 Y220 H223 R226 G244 S248 L251 R254 Q300 Y301 L304 Q307 N357 S360 H361 E364 R394 C395 N397 F398 Q401 G431 K432 G434 V500 M501 L504 Q507 S539 S540 R543 E546 T576 S577 F580 S51 H52 Q55 R84 S87 H88 E91 Y133 H136 R139 G157 S161 L164 R167 Q201 Y202 L205 Q208 N251 S254 H255 E258 R288 C289 N291 F292 Q295 G325 K326 G328 V394 M395 L398 Q401 S433 S434 R437 E440 T470 S471 F474 ? 0003723 remove_due_to_license_issue Q9C552 29036323 1 ~ 10 IDPETSKYFSEIANLFDSNEVELEERSVICGNALEETRGREYEIATDYIISHVLQTLLEGCELDQLCSFIRNSASVFPAIAMDRSGSHVAESALKSLATHLENPDAYSVIEEALHSICKVIVDNPLDMMCNCYGSHVLRRLLCLCKGVSLDSPELYGAKSSKALAKRLNLPHQGFPGMLTYLLSGLLSCSREDMKYLQVDQYSSLVLQTALRLMLKQDEQLLEIIPLILRCNGFHIETNVAKEILESMKDNSFSHLVEVILEVAPESLYNEMFNKVFKNSLFELSVDRCANFVIQALISHARDQEQMGIMWEELAPRFKDLLEQGKSGVVASLIAVSQRLQSHENKCCEALVGAVCSTNESRISILPRLLFLDYYFGCRDKSTWEWAPGAKMHVMGCLILQGIFKFSSDHIQPYITSLTSMKAEYITETAKDSSGARVIEAFLASDAATKQKRRLIIKLRGHFGELSLHTSGSFTVEKCFDACNLTLREAIASELLDVKVDLSKTKQGPYLLRKLDIDGYASRPDQWKSRQEAK 5wzh A 2.509 BS01 rna B 0 S138 H139 Q142 R171 S174 H175 E178 Y220 H223 R226 Y243 G244 S248 L251 R254 Q300 Y301 L304 Q307 N357 S360 H361 E364 R394 N397 F398 Q401 G431 K432 G434 M501 L504 Q507 S539 S540 R543 E546 S577 S579 F580 E583 Y616 S51 H52 Q55 R84 S87 H88 E91 Y133 H136 R139 Y156 G157 S161 L164 R167 Q200 Y201 L204 Q207 N250 S253 H254 E257 R287 N290 F291 Q294 G324 K325 G327 M394 L397 Q400 S432 S433 R436 E439 S470 S472 F473 E476 Y509 ? 0003723 remove_due_to_license_issue Q9C552 29036323 0 ~ 10 IDPETSKYFSEIANLFDSNEVELEERSVICGNALEETRGREYEIATDYIISHVLQTLLEGCELDQLCSFIRNSASVFPAIAMDRSGSHVAESALKSLATHLENPDAYSVIEEALHSICKVIVDNPLDMMCNCYGSHVLRRLLCLCKGVSLDSPELYGAKSSKALAKRLNLHQGFPGMLTYLLSGLLSCSREDMKYLQVDQYSSLVLQTALRLMLKQDEQLLEIIPLILRCNGFHIETNVAKEILESMKDNSFSHLVEVILEVAPESLYNEMFNKVFKNSLFELSVDRCANFVIQALISHARDQEQMGIMWEELAPRFKDLLEQGKSGVVASLIAVSQRLQSHENKCCEALVGAVCSTNESRISILPRLLFLDYYFGCRDKSTWEWAPGAKMHVMGCLILQGIFKFSSDHIQPYITSLTSMKAEYITETAKDSSGARVIEAFLASDAATKQKRRLIIKLRGHFGELSLHTSGSFTVEKCFDACNLTLREAIASELLDVKVDLSKTKQGPYLLRKLDIDGYASRPDQWKSRQEAK 5wzj A 2.101 BS01 rna B 0 S138 H139 Q142 R171 S174 H175 E178 Y220 H223 R226 Y243 G244 K246 S248 L251 R254 Q300 L304 Q307 N357 S360 H361 E364 R394 C395 N397 F398 Q401 G431 K432 G434 M501 Q507 S539 S540 R543 E546 S577 S579 F580 E583 Q613 Y616 S51 H52 Q55 R84 S87 H88 E91 Y133 H136 R139 Y156 G157 K159 S161 L164 R167 Q201 L205 Q208 N251 S254 H255 E258 R288 C289 N291 F292 Q295 G325 K326 G328 M395 Q401 S433 S434 R437 E440 S471 S473 F474 E477 Q507 Y510 ? 0003723 remove_due_to_license_issue Q9C552 29036323 0 ~ 10 IDPETSKYFSEIANLFDSNEVELEERSVICGNALEETRGREYEIATDYIISHVLQTLLEGCELDQLCSFIRNSASVFPAIAMDRSGSHVAESALKSLATHLENPDAYSVIEEALHSICKVIVDNPLDMMCNCYGSHVLRRLLCLCKGVSLDSPELYGAKSSKALAKRLNLPHQGFPGMLTYLLSGLLSCSREDMKYLQVDQYSSLVLQTALRLMLKQDEQLLEIIPLILRCNGFHIETNVAKEILESMKDNSFSHLVEVILEVAPESLYNEMFNKVFKNSLFELSVDRCANFVIQALISHARDQEQMGIMWEELAPRFKDLLEQGKSGVVASLIAVSQRLQSHENKCCEALVGAVCSTNESRISILPRLLFLDYYFGCRDKSTWEWAPGAKMHVMGCLILQGIFKFSSDHIQPYITSLTSMKAEYITETAKDSSGARVIEAFLASDAATKQKRRLIIKLRGHFGELSLHTSGSFTVEKCFDACNLTLREAIASELLDVKVDLSKTKQGPYLLRKLDIDGYASRPDQWKSRQEAK 5wzk A 2.8 BS01 rna B 0 S138 H139 Q142 R171 S174 H175 E178 Y220 H223 R226 Q266 Y267 L270 Q273 N323 S326 H327 E330 R360 N363 F364 Q367 G397 K398 G400 V466 M467 Q473 S505 S506 R509 E512 S543 F546 S51 H52 Q55 R84 S87 H88 E91 Y133 H136 R139 Q179 Y180 L183 Q186 N229 S232 H233 E236 R266 N269 F270 Q273 G303 K304 G306 V372 M373 Q379 S411 S412 R415 E418 S449 F452 ? 0003723 remove_due_to_license_issue Q9C552 29036323 0 ~ 10 IDPETSKYFSEIANLFDSNEVELEERSVICGNALEETRGREYEIATDYIISHVLQTLLEGCELDQLCSFIRNSASVFPAIAMDRSGSHVAESALKSLATHLENPDAYSVIEEALHSICKVIVDNPLDMMCNCYGSHVLRRLLCLCKGVPHQGFPGMLTYLLSGLLSCSREDMKYLQVDQYSSLVLQTALRLMLKQDEQLLEIIPLILRCNGFHIETNVAKEILESMKDNSFSHLVEVILEVAPESLYNEMFNKVFKNSLFELSVDRCANFVIQALISHARDQEQMGIMWEELAPRFKDLLEQGKSGVVASLIAVSQRLQSHENKCCEALVGAVCSTNESRISILPRLLFLDYYFGCRDKSTWEWAPGAKMHVMGCLILQGIFKFSSDHIQPYITSLTSMKAEYITETAKDSSGARVIEAFLASDAATKQKRRLIIKLRGHFGELSLHTSGSFTVEKCFDACNLTLREAIASELLDVKVDLSKTKQGPYLLRKLDIDGYASRPDQWKSRQEAKQ 5wzr A 2.79 BS02 DJN A 1 Y329 D330 D371 W398 D435 V436 E478 H492 D561 Y329 D330 D371 W398 D435 V436 E478 H492 D561 3.2.1.- 0016798,0033926,0046872 remove_due_to_license_issue G5ELM1 28546425 702 MMQFTMSGTMLRFDETTLRFSFSRDGATWSGCDGIEPQLTREDRSFSFAGAATVTHERIETGTGVGVRSVFAGFAGADYAFETYIWIERSSGDVLCEWVPLRECGAEPRIDRVLWPAPLSFDRADAHDVTLITHEQGVMIPNSWPTEVGTDAVSFGGRFETAGGYMPWFAQLRSDGHAYIAICETPWNAGYDIDHPAGGPYTHVGMWFEPSLGRMDYRRVVRYRLLDHADHTAICKTYRAYVNERGRLRTLAEKAARNPSVRDLLGRSWVHVGIKTNVQPDSSFYDPAQPGKNDSLVTFAQRERQMRTLHEMGAGRLYLHLDGWAQPGYDNGHPDYLPACREAGGWKGMKSLIDACHEQGDLFGTHDQYRDYYFAARTFDPRNAIRLADGTMPEHAMWAGGRQTYLCAELAPDYVRRNFSEIATHGIVLDCAYLDVFTCNEGDECSHPEHRMTRRECYERRAECFEYLLAHGILTSSEEVSDWAVPSLVFCHYAPYDFQMRSPDAPRHGIPVPLYNLVYHDCVIQPWMMDRVAGGDDYMLYALLNGGAPYLIRDAAYAGMDGDMNAALRTENDIERCAVVAGLHRRVGMQELVRHDLVGGDPLVQRSVFADGTAVTCDFHAQTYEVAANG 5wzs A 2.3 BS01 7W9 A 1 L2 F5 G6 I9 A17 Y20 N21 C27 G28 C43 H46 D47 L2 F5 G6 I9 A17 Y20 N21 C27 G28 C43 H46 D47 Y26 G28 G30 H46 D47 Y50 Y65 D90 Y26 G28 G30 H46 D47 Y50 Y65 D90 3.1.1.4 0004623,0005509,0005515,0005543,0005576,0005737,0006629,0006644,0006954,0016042,0016787,0034374,0046470,0046471,0046872,0047498,0047499,0050482 ic50=0.28uM remove_due_to_license_issue Q9NZK7 28883454 201 NLVQFGVMIEKMTGKSALQYNDYGCYCGIGGSHWPVDQTDWCCHAHDCCYGRLEKLGCEPKLEKYLFSVSERGIFCAGRTTCQRLTCECDKRAALCFRRNLGTYNRKYAHYPNKLCTGPTPPC 5wzt A 2.4 BS02 7W6 A 1 L2 F5 G6 I9 A17 Y20 N21 C27 G28 I29 C43 H46 D47 F97 L2 F5 G6 I9 A17 Y20 N21 C27 G28 I29 C43 H46 D47 F97 Y26 G28 G30 H46 D47 Y50 Y65 D90 Y26 G28 G30 H46 D47 Y50 Y65 D90 3.1.1.4 0004623,0005509,0005515,0005543,0005576,0005737,0006629,0006644,0006954,0016042,0016787,0034374,0046470,0046471,0046872,0047498,0047499,0050482 ic50=0.22uM remove_due_to_license_issue Q9NZK7 28883454 204 NLVQFGVMIEKMTGKSALQYNDYGCYCGIGGSHWPVDQTDWCCHAHDCCYGRLEKLGCEPKLEKYLFSVSERGIFCAGRTTCQRLTCECDKRAALCFRRNLGTYNRKYAHYPNKLCTGPTPPC 5wzu A 2.2 BS02 7W3 A 1 L2 F5 G6 I9 A17 Y20 N21 Y26 C27 G28 C43 H46 D47 L2 F5 G6 I9 A17 Y20 N21 Y26 C27 G28 C43 H46 D47 Y26 G28 G30 H46 D47 Y50 Y65 D90 Y26 G28 G30 H46 D47 Y50 Y65 D90 3.1.1.4 0004623,0005509,0005515,0005543,0005576,0005737,0006629,0006644,0006954,0016042,0016787,0034374,0046470,0046471,0046872,0047498,0047499,0050482 ic50=0.1uM remove_due_to_license_issue Q9NZK7 28883454 202 NLVQFGVMIEKMTGKSALQYNDYGCYCGIGGSHWPVDQTDWCCHAHDCCYGRLEKLGCEPKLEKYLFSVSERGIFCAGRTTCQRLTCECDKRAALCFRRNLGTYNRKYAHYPNKLCTGPTPPC 5wzv A 2.2 BS02 7W0 A 1 L2 F5 G6 L18 N21 C27 G28 C43 H46 D47 L2 F5 G6 L18 N21 C27 G28 C43 H46 D47 Y26 G28 G30 H46 D47 Y50 Y65 D90 Y26 G28 G30 H46 D47 Y50 Y65 D90 3.1.1.4 0004623,0005509,0005515,0005543,0005576,0005737,0006629,0006644,0006954,0016042,0016787,0034374,0046470,0046471,0046872,0047498,0047499,0050482 ic50=0.21uM remove_due_to_license_issue Q9NZK7 28883454 202 NLVQFGVMIEKMTGKSALQYNDYGCYCGIGGSHWPVDQTDWCCHAHDCCYGRLEKLGCEPKLEKYLFSVSERGIFCAGRTTCQRLTCECDKRAALCFRRNLGTYNRKYAHYPNKLCTGPTPPC 5wzw A 1.95 BS02 U8D A 1 L2 F5 G6 Y20 N21 Y26 C27 G28 G30 C43 H46 D47 K61 F97 L2 F5 G6 Y20 N21 Y26 C27 G28 G30 C43 H46 D47 K61 F97 Y26 G28 G30 H46 D47 Y50 Y65 D90 Y26 G28 G30 H46 D47 Y50 Y65 D90 3.1.1.4 0004623,0005509,0005515,0005543,0005576,0005737,0006629,0006644,0006954,0016042,0016787,0034374,0046470,0046471,0046872,0047498,0047499,0050482 ic50=1.23uM remove_due_to_license_issue Q9NZK7 28883454 209 NLVQFGVMIEKMTGKSALQYNDYGCYCGIGGSHWPVDQTDWCCHAHDCCYGRLEKLGCEPKLEKYLFSVSERGIFCAGRTTCQRLTCECDKRAALCFRRNLGTYNRKYAHYPNKLCTGPTPPC 5x02 A 2.401 BS01 F6M A 1 L616 V624 A642 K644 V675 F691 E692 Y693 C694 C695 Y696 L818 C828 F830 L44 V52 A70 K72 V103 F119 E120 Y121 C122 C123 Y124 L176 C186 F188 D811 R815 N816 D829 D169 R173 N174 D187 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue P36888 29187377 1001 ESQLQMVQVTGSSDNEYFYVDFREYEYDLKWEFPRENLEFGKVLGSGAFGKVMNATAYGISKTGVSIQVAVKMLKEKADSSEREALMSELKMMTQLGSHENIVNLLGACTLSGPIYLIFEYCCYGDLLNYLRSKREKFSVLTFEDLLCFAYQVAKGMEFLEFKSCVHRDLAARNVLVTHGKVVKICDFGLARDIMSDSNYVVRGNARLPVKWMAPESLFEGIYTIKSDVWSYGILLWEIFSLGVNPYPGIPVDANFYKLIQNGFKMDQPFYATEEIYIIMQSCWAFDSRKRPSFPNLTSFLGCQL 5x07 C 2.796 BS01 dna D 0 G155 A158 G1 A4 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 C 2.796 BS02 dna E 0 P156 Q198 N199 P2 Q44 N45 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 C 2.796 BS03 dna A 0 L182 R208 H209 S212 K219 K229 G230 S231 L28 R54 H55 S58 K65 K75 G76 S77 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 C 2.796 BS04 dna B 0 S163 Y164 I165 R202 N205 S206 H209 S9 Y10 I11 R48 N51 S52 H55 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 F 2.796 BS01 dna D 0 L182 S183 R208 H209 S212 K219 G230 S231 W233 L28 S29 R54 H55 S58 K65 G76 S77 W79 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 F 2.796 BS02 dna E 0 S163 Y164 I165 R202 N205 S206 H209 S9 Y10 I11 R48 N51 S52 H55 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 F 2.796 BS03 dna G 0 G155 A158 G1 A4 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 F 2.796 BS04 dna H 0 G155 P156 Q198 G1 P2 Q44 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 I 2.796 BS01 dna G 0 L182 R208 H209 S212 K219 K229 G230 S231 W233 L26 R52 H53 S56 K63 K73 G74 S75 W77 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 HAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 I 2.796 BS02 dna H 0 S163 Y164 I165 R202 N205 S206 H209 S7 Y8 I9 R46 N49 S50 H53 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 HAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 I 2.796 BS03 dna J 0 H157 F195 H1 F39 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 HAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPD 5x07 L 2.796 BS01 dna A 0 G155 A158 G1 A4 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 L 2.796 BS02 dna B 0 G155 P156 Q198 G1 P2 Q44 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 L 2.796 BS03 dna J 0 L182 R208 H209 S212 K219 K229 G230 S231 W233 L28 R54 H55 S58 K65 K75 G76 S77 W79 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x07 L 2.796 BS04 dna K 0 S163 Y164 I165 R202 N205 S206 H209 G228 S9 Y10 I11 R48 N51 S52 H55 G74 ? 0003700,0006355,0043565 remove_due_to_license_issue Q9Y261 28644006 1 ~ 16 GPHAKPPYSYISLITMAIQQSPNKMLTLSEIYQWIMDLFPFYRQNQQRWQNSIRHSLSFNDCFLKVPRSPDKPGKGSFWTLHPDS 5x11 A 2.65 BS01 dna I 0 Y20 H38 S39 Y42 K67 K68 K95 Y23 H41 S42 Y45 K70 K71 K98 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 KDPMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMI 5x11 A 2.65 BS02 dna J 0 P0 R2 K37 S39 Q40 G62 T63 K64 L65 P3 R5 K40 S42 Q43 G65 T66 K67 L68 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 KDPMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMI 5x11 B 2.65 BS01 dna I 0 R2 K37 S39 Q40 T63 R4 K39 S41 Q42 T65 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 DPMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 B 2.65 BS02 dna J 0 Y20 H38 Y42 Q61 K67 K68 K95 Y22 H40 Y44 Q63 K69 K70 K97 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 DPMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 C 2.65 BS01 dna M 0 Y20 H38 S39 Y42 K67 K68 Y19 H37 S38 Y41 K66 K67 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 RVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMAPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 C 2.65 BS02 dna N 0 S39 Q40 Q61 G62 T63 K64 L65 S38 Q39 Q60 G61 T62 K63 L64 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 RVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMAPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 D 2.65 BS01 dna I 0 Y20 H38 S39 Y42 K67 K68 Y19 H37 S38 Y41 K66 K67 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 RVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 D 2.65 BS02 dna J 0 S39 Q40 Q61 G62 T63 K64 L65 S38 Q39 Q60 G61 T62 K63 L64 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 RVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 E 2.65 BS01 dna M 0 Y20 H38 S39 Y42 K67 K95 Y22 H40 S41 Y44 K69 K97 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 DPMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASAEPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMI 5x11 E 2.65 BS02 dna N 0 R2 K37 S39 Q40 G62 T63 L65 R4 K39 S41 Q42 G64 T65 L67 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 DPMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMASAEPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMI 5x11 F 2.65 BS01 dna M 0 R2 S39 Q40 G62 T63 K64 L65 R3 S40 Q41 G63 T64 K65 L66 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 PMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMAPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 F 2.65 BS02 dna N 0 Y20 H38 Y42 K67 K68 K95 Y21 H39 Y43 K68 K69 K96 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 PMRVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMAPMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 H 2.65 BS01 dna M 0 S39 Q40 Q61 T63 L65 S38 Q39 Q60 T62 L64 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 RVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x11 H 2.65 BS02 dna N 0 Y20 H38 Y42 Q61 K67 K68 Y19 H37 Y41 Q60 K66 K67 ? remove_due_to_license_issue E0TW95 29136175 1 ~ 28 RVLKYAILGLLRKGELSGYDITSYFKEELGQFWSAKHSQIYPELKKLTDEGFITFRTTIQGTKLEKKMYTLTDSGKQELHDWLIRHQPIPETVKDEFMLKAYFISSLSRQEASDLFTDQLLKRKAKLSDLQGSYEKLMSFSSPDFGHYLVLTKALEREKNYVSWLESILAMID 5x26 A 2.951 BS01 7XO A 1 L718 A743 K745 M766 T790 M793 P794 G796 L844 L22 A47 K49 M70 T94 M97 P98 G100 L148 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=5nM P00533 29568384 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPEEDMDDVVDADEYLIPQ 5x27 A 2.952 BS01 7XR A 1 A743 K745 M766 M793 P794 G796 L844 A47 K49 M70 M97 P98 G100 L148 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1nM P00533 29568384 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPEEDMDDVVDADEYLIPQ 5x28 A 2.952 BS01 7XU A 1 L718 A743 K745 M766 T790 M793 P794 G796 L844 L22 A47 K49 M70 T94 M97 P98 G100 L148 D837 A839 R841 N842 D855 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 29568384 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGAEEVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPYRALMDEEDMDDVVDADEYLIPQ 5x33 A 3.7 BS01 7Y9 A 1 D66 V69 F76 L80 H96 C99 S102 S106 W236 K267 I270 A273 F274 S276 S277 D52 V55 F62 L66 H82 C85 S88 S92 W390 K419 I422 A425 F426 S428 S429 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue A0A097J792,Q9WTK1 29309055 2001 SNTFIPLLAMILLSVSMVVGLPGNTFVVWSILKRMRKRSVTALMVLNLALADLAVLLTAPFFLHFLTWGTWSFGLAGCRLCHYICGVSMYASVLLITAMSLDRSLAVASPFLSQKVRTKTAARWLLVGIWGASFLLATPVLAFRKVVKLTNETDLCLAVYPSDRHKAFHLLFEAFTGFVVPFLIVVASYADISRRLRARGSGSNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYGSGSRFHRRRRTGRLVVIIILAFAAFWLPYHVVDLVEGSRVLAGDQSKQQLRNARKVCIALAFLSSSVNPLLYACA 5x4m A 1.65 BS01 7ZF A 1 N21 R24 L25 N23 R26 L27 ? Kd=1200uM remove_due_to_license_issue Kd=1200000nM P41182 28471657 801 NLYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5x4n A 1.94 BS01 7ZL A 1 N21 L25 N22 L26 ? Kd=68uM remove_due_to_license_issue Kd=68000nM P41182 28471657 801 LYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5x4o A 2.05 BS01 YAM A 1 N21 R24 L25 N22 R25 L26 ? Kd=88uM remove_due_to_license_issue Kd=88000nM P41182 28471657 801 LYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5x4p A 2.06 BS01 7ZO A 1 N21 L25 R28 N22 L26 R29 ? Kd=9.3uM remove_due_to_license_issue Kd=9300nM P41182 28471657 801 LYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5x4q A 2.0 BS01 7Z6 A 1 N21 R24 L25 R28 N22 R25 L26 R29 ? Kd=0.078uM remove_due_to_license_issue IC50=2699nM, Kd=1190nM P41182 28471657 801 LYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5x5g A 2.0 BS04 OP0 A 1 S56 W93 S120 N122 H160 T206 T225 G226 S227 D229 S45 W82 S109 N111 H149 T195 T214 G215 S216 D218 S56 K59 S120 E156 K224 S227 S45 K48 S109 E145 K213 S216 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue A0A0B6VPP7 28739781 305 GTDSLKNSIEKYLKDKKAKVGVAVLGIEDNFKLNVNEKHHYPMQSTYKFHLALAVLDKLDKENISVDKKLFVKKSDLQPNTWSPLKDKYPNGNLELSFSEIIKSTVSHSDNNGCDILFRFVGGTNKVHNFISKLGVKNISIKATEEEMHKAWNVQYTNWTTPDATVQLLKKFYKNEILSKNSYDFLLNTMIETTTGPKRLKGLLPDGTVVAHKTGSSDTNNKGITAATNDIGIITLPNGKHFAIAVYVSDSSEKSDVNEKIIAEICKSVWDYLVK 5x5l A 2.75 BS01 dna F 0 R189 R205 S212 R215 K216 N229 R231 G232 Y235 R45 R60 S67 R70 K71 N84 R86 G87 Y90 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 1 ~ 24 KLYKNIEIDTDTHSVYIHKILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMNSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDNP 5x5l A 2.75 BS02 dna G 0 T169 T171 A202 L203 T206 S209 H210 K213 R231 T25 T27 A57 L58 T61 S64 H65 K68 R86 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 0 ~ 24 KLYKNIEIDTDTHSVYIHKILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMNSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDNP 5x5l B 2.75 BS01 dna C 0 R189 R205 S212 K213 R215 K216 N229 R231 G232 Y235 R41 R57 S64 K65 R67 K68 N81 R83 G84 Y87 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 1 ~ 24 NKLYKNIETDTHSVYILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMNDSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDNPLAV 5x5l B 2.75 BS02 dna D 0 T169 T171 N198 A202 T206 S209 H210 R231 T21 T23 N50 A54 T58 S61 H62 R83 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 0 ~ 24 NKLYKNIETDTHSVYILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMNDSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDNPLAV 5x5l E 2.75 BS01 dna F 0 R189 R205 S212 K213 R215 N229 R231 G232 Y235 R49 R64 S71 K72 R74 N88 R90 G91 Y94 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 1 ~ 24 NKLYKNIEIDTDTHSVYIHENKKILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMNSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDN 5x5l E 2.75 BS02 dna G 0 T169 T171 M197 S200 A202 L203 T206 S209 H210 K213 R231 T29 T31 M57 S59 A61 L62 T65 S68 H69 K72 R90 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 0 ~ 24 NKLYKNIEIDTDTHSVYIHENKKILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMNSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDN 5x5l H 2.75 BS01 dna C 0 R189 R205 S212 K213 R215 K216 N229 R231 G232 Y235 R46 R60 S67 K68 R70 K71 N84 R86 G87 Y90 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 1 ~ 24 NKLYKNIEIDTDTHSVYIHSILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDNP 5x5l H 2.75 BS02 dna D 0 T169 T171 A202 L203 T206 S209 H210 K213 R231 T26 T28 A57 L58 T61 S64 H65 K68 R86 ? 0000160,0003677,0006355 remove_due_to_license_issue E1A0Z5 28934482 0 ~ 24 NKLYKNIEIDTDTHSVYIHSILLNLTLTEYKIISFMIDQPHKVFTRGELMNHCMSDALERTVDSHVSKLRKKLEEQGIFQMLINVRGVGYRLDNP 5x5o A 1.868 BS01 7Z0 A 1 A43 K45 F68 I80 T82 Y84 A85 V140 C150 D151 F152 G153 H158 A36 K38 F61 I73 T75 Y77 A78 V133 C143 D144 F145 G146 H151 D133 R137 N138 D151 D126 R130 N131 D144 2.7.11.25 0004672,0005524,0006468 ic50=5nM remove_due_to_license_issue IC50=5.0nM Q9NYL2 28586211 401 FVQIKFDDLQFFENCGGGSFGSVYRAKWISQDKEVAVKKLLKIEKEAEILSVLSHRNIIQFYGVILEPPNYGIVTEYASLGSLYDYINSNRSEEMDMDHIMTWATDVAKGMHYLHMEAPVKVIHRDLKSRNVVIAADGVLKICDFGASRFHNHTTHSLVGTFPWMAPEVIQSLPVSETCDTYSYGVVLWEMLTREVPFKGLEGLQVAWLVVEKNERLTIPSSCPRSFAELLHQCWEADAKKRPSFKQIISILESMSNDTSLPDKCNSFLHNKAEWRCEIEATLERLKKLER 5x62 A 2.204 BS01 SAH A 1 R111 G146 E167 F168 M172 S234 F235 N274 F275 F276 T279 Y371 R104 G139 E160 F161 M165 S222 F223 N262 F263 F264 T267 Y352 2.1.1.22 0005575,0008168,0008757,0030735,0032259,0035498 remove_due_to_license_issue P53934 28654751 501 NQRENKAVARVIISFLKYEEYALKEIYNLRVKKWASISDRQKDMVPNYTKYLANLKAAIIENGKFFRSVAEYALQSISFEPGEIVQPNDLDMSKTCSLLTQVYREWSAEAISERNCLNSRLVPFLKTLSPPKADILIPGCGTGRLLVDLSRMGYNCEGNEFSYHMLLVSQYMLNAGLLQNQIIIYPFIHCFSHWKKIEDQLSPIKVPDIEAWMGSMSICAGSFVDCYGRNQGTKISSHYTFSRRMQLSRAKAENSKDVVVTNFFIDTGSNILDYLDTIGHVLKPGGIWCNFGPLLYHFENDHGVETTYEVNPINDYTPLMGLELSSDDIISIATNHLDFELIRRESGILCGYGRYAGPESCAMPGYMCHYWILKSN 5x6b F 2.596 BS01 rna P 0 N117 K118 K119 K125 E137 K161 N168 N84 K85 K86 K92 E104 K128 N135 ? remove_due_to_license_issue Q58876 29142195 1 ~ 75 ISYKDAKPGKIDVNEFKKAIYLLIEADDFLYKKAPKHELNEEEAKEFCKLIIKCQEHLNKILANFGFEFEEKEIDEGALYIVSNKKLFKKLKNKNPNLKVVCTEGMLDIEDMRAIGVPEKALEGLKKKVEIARKNVERFIEKYKPEKIFVVVEDDKDELLYLRAKNLYNAEKLDADE 5x6b I 2.596 BS01 rna P 0 N19 D21 Y127 R345 G346 F347 Y350 K354 R362 G364 V365 T366 K367 K370 N4 D6 Y98 R316 G317 F318 Y321 K325 R333 G335 V336 T337 K338 K341 2.5.1.73 0005515,0006412,0016740,0043766,0071952 remove_due_to_license_issue Q59072 29142195 1 ~ 75 LDINLDKYKNLTRSLTREFINLNPIQRGGILPKEAKKAVYEYWDGYCPPIKDFLEDIAKFLNMDCARPTHGAREGKFIVMHAICKEGDYVVLDKNAHYTSYVAAERAKLNVAEVGYEEEYPTYKINLEGYKEVIDNLEDKGKNVGLILLTHVDGEYGNLNDAKKVGKIAKEKGIPFLLNCAYTVGRMPVNGKEVKADFIVASGHKSMAASAPCGILAFSEEFSDKITKTSEKFPVKEIEMLGCTSRGLPIVTLMASFPHVVERVKKWDEELKKTRYVVDELEKIGFKQLGIKPKEHDLIKFETPVLDEIAKKDKRRGFFFYDELKKRGIGGIRAGVTKEIKMSVYGLEWEQVEYVVNAIKEIVESCK 5x6b J 2.596 BS01 rna P 0 F262 K265 F243 K246 2.5.1.73 0005515,0006412,0016740,0043766,0071952 remove_due_to_license_issue Q59072 29142195 1 ~ 75 VITLDINLDKYKNLTRSLTREFINLNPIQRGGILPKEAKKAVYEYWDGYSVCDEVTCPPIKDFLEDIAKFLNMDCARPTHGAREGKFIVMHAICKEGDYVVLDKNAHYTSYVAAERAKLNVAEVGYEEEYPTYKINLEGYKEVIDNLEDKGKNVGLILLTHVDGEYGNLNDAKKVGKIAKEKGIPFLLNCAYTVGRMPVNGKEVKADFIVASGHKSMAASAPCGILAFSEEFSDKITKTSEKFPVKEIEMLGCTSRGLPIVTLMASFPHVVERVKKWDEELKKTRYVVDELEKIGFKQLGIKPKEHDLIKFETPVLDEIAKKDKRRGFFFYDELKKRGIGGIRAGVTKEIKMSVYGLEWEQVEYVVNAIKEIVESCK 5x72 A 1.95 BS01 P59 A 1 M20 W32 R61 Q78 I109 V145 M20 W32 R61 Q78 I109 V144 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=467nM remove_due_to_license_issue O43924 28929751 201 MSAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAAPSQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5x73 A 2.5 BS01 P59 A 1 M20 W32 R61 Q78 I109 V145 M20 W32 R61 Q78 I109 V143 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=184nM remove_due_to_license_issue O43924 28929751 201 MSAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAASQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5x73 A 2.5 BS02 P59 A 2 I53 V80 W90 A111 M117 Y149 I53 V80 W90 A111 M115 Y147 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=184nM remove_due_to_license_issue O43924 28929751 202 MSAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLIEAASQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5x74 A 2.25 BS01 JAY A 1 M20 L22 W32 L38 I53 R61 Q78 E88 W90 A111 M117 V145 Y149 M20 L22 W32 L38 I53 R61 Q78 E88 W90 A111 M117 V145 Y149 ? 0005095,0005515,0005737,0005829,0005856,0005929,0007601,0016020,0030659,0031267,0031410,0042995,0050953 Kd=2.3nM remove_due_to_license_issue Kd=12nM O43924 28929751 201 MSAKDERAREILRGFKLNWMNLRDAETGKILWQGTEDLSVPGVEHEARVPKKILKCKAVSRELNFSSTEQMEKFRLEQKVYFKGQCLEEWFFEFGFVIPNSTNTWQSLISAAPESQMMPASVLTGNVIIETKFFDDDLLVSTSRVRLFYV 5x79 A 1.9 BS01 GF5 A 1 Y8 F9 R14 W39 K45 Q52 L53 Q65 S66 Y109 Y8 F9 R14 W39 K45 Q52 L53 Q65 S66 Y109 Y8 R14 Y8 R14 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 28848941 301 MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 5x79 B 1.9 BS01 GF5 B 1 F9 R14 W39 K45 Q52 L53 Q65 S66 Y109 N205 F9 R14 W39 K45 Q52 L53 Q65 S66 Y109 N205 Y8 R14 Y8 R14 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 remove_due_to_license_issue P09211 28848941 301 MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 5x8i B 1.902 BS01 SQZ B 1 L167 G168 F172 V175 A189 K191 F241 L244 N293 L295 D325 L13 G14 F18 V21 A35 K37 F87 L90 N139 L141 D171 D288 K290 N293 D325 T342 D134 K136 N139 D171 T188 2.7.12.1 0004672,0005524,0006468 ic50=2nM remove_due_to_license_issue IC50=2.0nM P49759 28692292 501 DVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLK 5x9h A 3.598 BS01 ATP A 1 Y170 V183 S185 R187 V206 V207 F227 P231 Y148 V161 S163 R165 V184 V185 F205 P209 ? 0000287,0005886,0006812,0008324,0015095,0015693,0016020,0042802,0042803,0046872,1903830 remove_due_to_license_issue Q5SMG8 28747715 501 EVLEEIHPQDLLALWDELKGEHRYVVLTLLPKAKAAEVLSHLSPEEQAEYLKTLPPWRLREILEELSLDDLADALQAVRKEDPAYFQRLKDLLDPRTRAEVEALARYEEDEAGGLMTPEYVAVREGMTVEEVLRFLRRAAPDAETIYYIYVVDEKGRLKGVLSLRDLIVADPRTRVAEIMNPKVVYVRTDTDQEEVARLMADYDFTVLPVVDEEGRLVGIVTVDDVLDVLEAEATEDIHKLGAVDVPDLVYSEAGPVALWLARVRWLVILILTGMVTSSILQGFESVLEAVTALAFYVPVLLGTGGNTGNQSATLIIRALATRDLDLRDWRRVFLKEMGVGLLLGLTLSFLLVGKVYWDGHPLLLPVVGVSLVLIVFFANLVGAMLPFLLRRLGVDPALVSNPLVATLSDVTGLLIYLSVARLLLEA 5x9h B 3.598 BS01 ATP B 1 Y170 V183 S185 R187 D188 V206 V207 F227 Y148 V161 S163 R165 D166 V184 V185 F205 ? 0000287,0005886,0006812,0008324,0015095,0015693,0016020,0042802,0042803,0046872,1903830 remove_due_to_license_issue Q5SMG8 28747715 501 EVLEEIHPQDLLALWDELKGEHRYVVLTLLPKAKAAEVLSHLSPEEQAEYLKTLPPWRLREILEELSLDDLADALQAVRKEDPAYFQRLKDLLDPRTRAEVEALARYEEDEAGGLMTPEYVAVREGMTVEEVLRFLRRAAPDAETIYYIYVVDEKGRLKGVLSLRDLIVADPRTRVAEIMNPKVVYVRTDTDQEEVARLMADYDFTVLPVVDEEGRLVGIVTVDDVLDVLEAEATEDIHKLGAVDVPDLVYSEAGPVALWLARVRWLVILILTGMVTSSILQGFESVLEAVTALAFYVPVLLGTGGNTGNQSATLIIRALATRDLDLRDWRRVFLKEMGVGLLLGLTLSFLLVGKVYWDGHPLLLPVVGVSLVLIVFFANLVGAMLPFLLRRLGVDPALVSNPLVATLSDVTGLLIYLSVARLLLE 5x9o A 1.58 BS01 80R A 1 N21 R24 L25 R28 N22 R25 L26 R29 ? Kd=5uM remove_due_to_license_issue Kd=5000nM P41182 28760529 801 LYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5x9p A 1.86 BS01 80L A 1 N21 R24 L25 R28 N23 R26 L27 R30 ? ic50=0.13uM remove_due_to_license_issue P41182 28760529 801 NLYFQGADSCIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKCNLSVINLDPEINPEGFCILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKASE 5xaf A 2.551 BS03 84F B 1 T179 A180 V181 T179 A180 V181 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 29306206 508 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVD 5xaf B 2.551 BS03 84F B 1 V238 C241 L242 L248 A250 D251 L255 N258 A316 A317 I318 K352 V236 C239 L240 L246 A248 D249 L253 N256 A308 A309 I310 K344 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Q6B856 29306206 508 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5xag A 2.56 BS04 93X B 1 T179 A180 V181 T179 A180 V181 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 29306206 508 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVDS 5xag B 2.56 BS04 93X B 1 C241 L242 L248 A250 D251 K254 L255 N258 M259 A317 I318 K352 C239 L240 L246 A248 D249 K252 L253 N256 M257 A311 I312 K346 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Q6B856 29306206 508 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5xbt A 2.495 BS01 C2E A 1 S0 M1 R31 D35 N36 Y40 S1 M2 R32 D36 N37 Y41 ? 0000166,0000976,0001216,0003677,0003700,0006355,0032993,0045892,0045893 remove_due_to_license_issue Q9HUT5 29967320 301 SMLTIGQLARIFEISTKTLRHYDAIGLFVPARTGSDNGYRYYQPEQIEQLSRILALRRLDVPLEAIDRLKRDGALDDPQRLRHFLQRHQHTLREEISARQRLLAELDRTLATLAHWRIRNMHARIVERPAFSVVGMEYFGSAPGDTIGQLWERFIPREHEIAGKHDPEVSYGICAQQPNGEFHYVAGFEVQEGWPVPEGMVRFQVPAQKYAVFTHKGTAPQIAESFQAIYSHLLAERGLEPKAGVDFEYYDQRFRGPLDPNSQVDLYIPIY 5xbt A 2.495 BS02 C2E A 2 E63 A64 R67 R86 E64 A65 R68 R87 ? 0000166,0000976,0001216,0003677,0003700,0006355,0032993,0045892,0045893 remove_due_to_license_issue Q9HUT5 29967320 302 SMLTIGQLARIFEISTKTLRHYDAIGLFVPARTGSDNGYRYYQPEQIEQLSRILALRRLDVPLEAIDRLKRDGALDDPQRLRHFLQRHQHTLREEISARQRLLAELDRTLATLAHWRIRNMHARIVERPAFSVVGMEYFGSAPGDTIGQLWERFIPREHEIAGKHDPEVSYGICAQQPNGEFHYVAGFEVQEGWPVPEGMVRFQVPAQKYAVFTHKGTAPQIAESFQAIYSHLLAERGLEPKAGVDFEYYDQRFRGPLDPNSQVDLYIPIY 5xbt B 2.495 BS01 C2E B 1 M1 R31 D35 N36 Y40 M2 R32 D36 N37 Y41 ? 0000166,0000976,0001216,0003677,0003700,0006355,0032993,0045892,0045893 remove_due_to_license_issue Q9HUT5 29967320 301 SMLTIGQLARIFEISTKTLRHYDAIGLFVPARTGSDNGYRYYQPEQIEQLSRILALRRLDVPLEAIDRLKRDGALDDPQRLRHFLQRHQHTLREEISARQRLLAELDRTLATLAHWRIRNMHARIVERPAFSVVGMEYFGSAPGDTIGQLWERFIPREHEIAGKHDPEVSYGICAQQPNGEFHYVAGFEVQEGWPVPEGMVRFQVPAQKYAVFTHKGTAPQIAESFQAIYSHLLAERGLEPKAGVDFEYYDQRFRGPLDPNSQVDLYIPIY 5xbt B 2.495 BS02 C2E B 2 E63 A64 R67 E64 A65 R68 ? 0000166,0000976,0001216,0003677,0003700,0006355,0032993,0045892,0045893 remove_due_to_license_issue Q9HUT5 29967320 302 SMLTIGQLARIFEISTKTLRHYDAIGLFVPARTGSDNGYRYYQPEQIEQLSRILALRRLDVPLEAIDRLKRDGALDDPQRLRHFLQRHQHTLREEISARQRLLAELDRTLATLAHWRIRNMHARIVERPAFSVVGMEYFGSAPGDTIGQLWERFIPREHEIAGKHDPEVSYGICAQQPNGEFHYVAGFEVQEGWPVPEGMVRFQVPAQKYAVFTHKGTAPQIAESFQAIYSHLLAERGLEPKAGVDFEYYDQRFRGPLDPNSQVDLYIPIY 5xfp B 2.3 BS01 dna C 0 K323 K324 R325 K326 K288 K289 R290 K291 ? remove_due_to_license_issue O43189 28869966 1 ~ 13 RLWEGQDVLARWTDGLLYLGTIKKVDSAREVCLVQFEDDSQFLVLWKDISPAALPGEELLCCVCRSETVVPGNRLVSCEKCRHAYHQDCHVPRAPAPSWVCRQCVFAIATKRGGALKKGPYARAMLGMKLSLPYGLKGLDWDAGHLSNRQQSYCYCGGPGEWNLKMLQCRSCLQWFHEACTQCLSKPLLYGDRFYEFECCVCRGGPEKVRRLQLRWVDVAHLVLYHLSVCCKKKYFDFDREILPFTSENWDSLLLGELSDTPKGERSSRLLSALNSHKDRFISGREIKKRKCLFGLHARMPPPVE 5xfp B 2.3 BS02 dna D 0 K268 K269 Y270 I322 K323 K324 K233 K234 Y235 I287 K288 K289 ? remove_due_to_license_issue O43189 28869966 1 ~ 13 RLWEGQDVLARWTDGLLYLGTIKKVDSAREVCLVQFEDDSQFLVLWKDISPAALPGEELLCCVCRSETVVPGNRLVSCEKCRHAYHQDCHVPRAPAPSWVCRQCVFAIATKRGGALKKGPYARAMLGMKLSLPYGLKGLDWDAGHLSNRQQSYCYCGGPGEWNLKMLQCRSCLQWFHEACTQCLSKPLLYGDRFYEFECCVCRGGPEKVRRLQLRWVDVAHLVLYHLSVCCKKKYFDFDREILPFTSENWDSLLLGELSDTPKGERSSRLLSALNSHKDRFISGREIKKRKCLFGLHARMPPPVE 5xg4 U 3.0 BS01 QUE U 1 H57 H99 S190 S195 S214 W215 G216 G219 H46 H94 S193 S198 S217 W218 G219 G221 3.4.21.73 0004252,0006508 remove_due_to_license_issue IC50=20000nM P00749 28644504 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 5xhr A 1.8 BS01 PXH A 1 S64 Y150 N152 Y221 L293 T316 G317 S318 S63 Y149 N151 Y220 L292 T315 G316 S317 S64 K67 Y112 V121 Y150 G156 E272 K315 S318 S63 K66 Y111 V120 Y149 G155 E271 K314 S317 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P05364 28971874 401 PVSEKQLAEVVANTITPLMKAQSVPGMAVAVIYQGKPHYYTFGKADIAANKPVTPQTLFELGSISKTFTGVLGGDAIARGEISLDDAVTRYWPQLTGKQWQGIRMLDLATYTAGGLPLQVPDEVTDNASLLRFYQNWQPQWKPGTTRLYANASIGLFGALAVKPSGMPYEQAMTTRVLKPLKLDHTWINVPKAEEAHYAWGYRDGKAVRVSPGMLDAQAYGVKTNVQDMANWVMANMAPENVADASLKQGIALAQSRYWRIGSMYQGLGWEMLNWPVEANTVVEGSDSKVALAPLPVAEVNPPAPPVKASWVHKTGSTGGFGSYVAFIPEKQIGIVMLANTSYPNPARVEAAYHILEAL 5xhs A 2.19 BS01 SLL A 1 Y102 R105 H158 V221 Y255 Y67 R70 H123 V186 Y220 P68 T69 F70 R71 N141 D143 H158 P33 T34 F35 R36 N106 D108 H123 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q9NXA8 402 PSSSMADFRKFFAKAKHIVIISGAGVSAESGVPTFRGAGGYWRKWQAQDLATPLAFAHNPSRVWEFYHYRREVMGSKEPNAGHRAIAECETRLGKQGRRVVVITQNIDELHRKAGTKNLLEIHGSLFKTRCTSCGVVAENYKSPICPALSGKGAPEPGTQDASIPVEKLPRCEEAGCGGLLRPHVVWFGENLDPAILEEVDRELAHCDLCLVVGTSSVVYPAAMFAPQVAARGVPVAEFNTETTFRFHFQGPCGTTLPEALA 5xhs A 2.19 BS02 MCM A 1 E225 N226 L227 L232 E190 N191 L192 L197 P68 T69 F70 R71 N141 D143 H158 P33 T34 F35 R36 N106 D108 H123 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q9NXA8 403 PSSSMADFRKFFAKAKHIVIISGAGVSAESGVPTFRGAGGYWRKWQAQDLATPLAFAHNPSRVWEFYHYRREVMGSKEPNAGHRAIAECETRLGKQGRRVVVITQNIDELHRKAGTKNLLEIHGSLFKTRCTSCGVVAENYKSPICPALSGKGAPEPGTQDASIPVEKLPRCEEAGCGGLLRPHVVWFGENLDPAILEEVDRELAHCDLCLVVGTSSVVYPAAMFAPQVAARGVPVAEFNTETTFRFHFQGPCGTTLPEALA 5xig A 2.41 BS02 87F A 1 F415 P438 T439 E441 R470 W487 F534 H560 W589 F79 P102 T103 E105 R134 W151 F198 H224 W253 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=350nM remove_due_to_license_issue S8G8I1 28867614 1004 AMVTAKKDENFSEWYTQAIVRSEMIEYYDISGCYIMRPWAFHIWEKVQRFFDDEIKKMGVENSYFPMFVSRHKLEKEGFSPEVAWVTHYGDSPLPEKIAIRPTSETIMYPAYAKWIRSHRDLPLKLNQWCSVVRWEFKQPTPFLRTREFLWQEGHTAHATEEEAWELVLDILELYRRWYEECLAVPVIKGEKSEGEKFAGGKKTTTVEAFIPENGRGIQAATSHLLGTNFAKMFEIEFEDEEGHKRLVHQTSWGCTTRSLGVMIMTHGDDKGLVIPPRVASVQVVIIPILFKDENTGEILGKCRELKTMLEKADIRVRIDDRSNYTPGWKYNHWEVKGVPLRLELGPKDLAKGTARVVRRDTGEAYQISWADLAPKLLELMEGIQRSLFEKAKARLHEGIEKISTFDEVMPALNRKHLVLAPWCEDPESEEQIKKETQKLSEIQAIETGAMKTLCIPFDQPPMPEGTKCFYTGKPAKRWTLWGRSY 5xih A 2.2 BS02 86U A 1 F415 E418 V419 P438 T439 E441 R470 W487 F534 H560 W589 F77 E80 V81 P100 T101 E103 R132 W149 F196 H222 W251 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=68nM remove_due_to_license_issue S8G8I1 28867614 1004 MVTAKKDENFSEWYTQAIVRSEMIEYYDISGCYIMRPWAFHIWEKVQRFFDDEIKKMGVENSYFPMFVSRHKLEKGFSPEVAWVTHYGDSPLPEKIAIRPTSETIMYPAYAKWIRSHRDLPLKLNQWCSVVRWEFKQPTPFLRTREFLWQEGHTAHATEEEAWELVLDILELYRRWYEECLAVPVIKGEKSEGEKFAGGKKTTTVEAFIPENGRGIQAATSHLLGTNFAKMFEIEFEDEEGHKRLVHQTSWGCTTRSLGVMIMTHGDDKGLVIPPRVASVQVVIIPILFNTGEILGKCRELKTMLEKADIRVRIDDRSNYTPGWKYNHWEVKGVPLRLELGPKDLAKGTARVVRRDTGEAYQISWADLAPKLLELMEGIQRSLFEKAKARLHEGIEKISTFDEVMPALNRKHLVLAPWCEDPESEEQIKKETQKLSEITGAMKTLCIPFDQPPMPEGTKCFYTGKPAKRWTLWGRSY 5xih B 2.2 BS02 86U B 1 F415 P438 T439 E441 R470 F534 H560 S588 F77 P100 T101 E103 R132 F196 H222 S250 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=68nM remove_due_to_license_issue S8G8I1 28867614 1004 MVTAKKDENFSEWYTQAIVRSEMIEYYDISGCYIMRPWAFHIWEKVQRFFDDEIKKMGVENSYFPMFVSRHKLEKGFSPEVAWVTHYGDSPLPEKIAIRPTSETIMYPAYAKWIRSHRDLPLKLNQWCSVVRWEFKQPTPFLRTREFLWQEGHTAHATEEEAWELVLDILELYRRWYEECLAVPVIKGEKSEGEKFAGGKKTTTVEAFIPENGRGIQAATSHLLGTNFAKMFEIEFEDEEGHKRLVHQTSWGCTTRSLGVMIMTHGDDKGLVIPPRVASVQVVIIPILFKDENTGEILGKCRELKTMLEKADIRVRIDDRSNYTPGWKYNHWEVKGVPLRLELGPKDLAKGTARVVRRDTGEAYQISWADLAPKLLELMEGIQRSLFEKAKARLHEGIEKISTFDEVMPALNRKHLVLAPWCEDPESEEQIKKETQKLSEIGAMKTLCIPFDQPPMPEGTKCFYTGKPAKRWTLWGRSY 5xii A 2.17 BS02 86X A 1 F415 V419 P438 T439 E441 R470 W487 F534 H560 F77 V81 P100 T101 E103 R132 W149 F196 H222 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=72nM remove_due_to_license_issue S8G8I1 28867614 1004 MVTAKKDENFSEWYTQAIVRSEMIEYYDISGCYIMRPWAFHIWEKVQRFFDDEIKKMGVENSYFPMFVSRHKLEKGFSPEVAWVTHYGDSPLPEKIAIRPTSETIMYPAYAKWIRSHRDLPLKLNQWCSVVRWEFKQPTPFLRTREFLWQEGHTAHATEEEAWELVLDILELYRRWYEECLAVPVIKGEKSEGEKFAGGKKTTTVEAFIPENGRGIQAATSHLLGTNFAKMFEIEFEDEEGHKRLVHQTSWGCTTRSLGVMIMTHGDDKGLVIPPRVASVQVVIIPILFTGEILGKCRELKTMLEKADIRVRIDDRSNYTPGWKYNHWEVKGVPLRLELGPKDLAKGTARVVRRDTGEAYQISWADLAPKLLELMEGIQRSLFEKAKARLHEGIEKISTFDEVMPALNRKHLVLAPWCEDPESEEQIKKETQKLSEITGAMKTLCIPFDQPPMPEGTKCFYTGKPAKRWTLWGRSY 5xii C 2.17 BS02 86X C 1 F415 V419 P438 T439 E441 R470 W487 F534 H560 F77 V81 P100 T101 E103 R132 W149 F196 H222 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=72nM remove_due_to_license_issue S8G8I1 28867614 1004 MVTAKKDENFSEWYTQAIVRSEMIEYYDISGCYIMRPWAFHIWEKVQRFFDDEIKKMGVENSYFPMFVSRHKLEKGFSPEVAWVTHYGDSPLPEKIAIRPTSETIMYPAYAKWIRSHRDLPLKLNQWCSVVRWEFKQPTPFLRTREFLWQEGHTAHATEEEAWELVLDILELYRRWYEECLAVPVIKGEKSEGEKFAGGKKTTTVEAFIPENGRGIQAATSHLLGTNFAKMFEIEFEDEEGHKRLVHQTSWGCTTRSLGVMIMTHGDDKGLVIPPRVASVQVVIIPILFKDENTGEILGKCRELKTMLEKADIRVRIDDRSNYTPGWKYNHWEVKGVPLRLELGPKDLAKGTARVVRRDTGEAYQISWADLAPKLLELMEGIQRSLFEKAKARLHEGIEKISTFDEVMPALNRKHLVLAPWCEDPESEEQIKKETQKLSEIGAMKTLCIPFDQPPMPEGTKCFYTGKPAKRWTLWGRSY 5xij A 2.5 BS02 873 A 1 F415 P438 T439 E441 R470 W487 F534 H560 F79 P102 T103 E105 R134 W151 F198 H224 6.1.1.15 0000166,0004812,0004827,0005524,0005737,0006418,0006433 ic50=67nM remove_due_to_license_issue S8G8I1 28867614 1004 GAMVTAKKDENFSEWYTQAIVRSEMIEYYDISGCYIMRPWAFHIWEKVQRFFDDEIKKMGVENSYFPMFVSRHKLEKEFSPEVAWVTHYGDSPLPEKIAIRPTSETIMYPAYAKWIRSHRDLPLKLNQWCSVVRWEFKQPTPFLRTREFLWQEGHTAHATEEEAWELVLDILELYRRWYEECLAVPVIKGEKSEGEKFAGGKKTTTVEAFIPENGRGIQAATSHLLGTNFAKMFEIEFEDEEGHKRLVHQTSWGCTTRSLGVMIMTHGDDKGLVIPPRVASVQVVIIPILFKDENTGEILGKCRELKTMLEKADIRVRIDDRSNYTPGWKYNHWEVKGVPLRLELGPKDLAKGTARVVRRDTGEAYQISWADLAPKLLELMEGIQRSLFEKAKARLHEGIEKISTFDEVMPALNRKHLVLAPWCEDPESEEQIKKETQKLSEIQGAMKTLCIPFDQPPMPEGTKCFYTGKPAKRWTLWGRSY 5xiw A 2.9 BS03 LOC B 1 S178 V181 S178 V181 3.6.5.- 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0015630,0016787,0046872 remove_due_to_license_issue Q2XVP4 29691282 504 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGV 5xiw B 2.9 BS02 LOC B 1 C239 L246 K252 L253 N256 I316 K350 C239 L246 K252 L253 N256 I316 K350 ? 0000226,0000278,0003924,0005200,0005515,0005525,0005737,0005856,0005874,0007017,0046872 remove_due_to_license_issue IC50=1400nM, Kd=3700nM, Ki=5750nM P02554 29691282 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5xkm A 2.16 BS02 87R A 1 L770 H773 T805 D808 L809 I826 Y827 F830 Q859 F862 L192 H195 T227 D230 L231 I248 Y249 F252 Q281 F284 3.1.4.17 0004114,0007165,0008081 ic50=24nM remove_due_to_license_issue IC50=53nM O00408 28759228 2004 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLDE 5xmp A 2.4 BS02 8A3 A 1 L124 G128 H129 V141 T183 K355 A364 L124 G128 H129 V141 T183 K355 A364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmp A 2.4 BS04 8A3 B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmp B 2.4 BS02 8A3 A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmp B 2.4 BS04 8A3 B 1 L124 G128 V141 T183 K355 N356 R371 L124 G128 V141 T183 K355 N356 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmr A 2.55 BS02 8AO A 1 L124 G128 L130 V141 T183 K355 N356 T357 A364 P367 L124 G128 L130 V141 T183 K355 N356 T357 A364 P367 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmr A 2.55 BS04 8AO B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmr B 2.55 BS02 8AO A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmr B 2.55 BS04 8AO B 1 L124 G128 H129 L130 V141 T183 K355 N356 A364 V365 P367 R371 L124 G128 H129 L130 V141 T183 K355 N356 A364 V365 P367 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDAVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xms A 2.45 BS02 8B3 A 1 L124 G128 H129 L130 T183 K355 T357 C364 L124 G128 H129 L130 T183 K355 T357 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xms A 2.45 BS04 8B3 B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xms B 2.45 BS01 8B3 A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xms B 2.45 BS03 8B3 B 1 L124 G128 H129 T183 N354 K355 N356 T357 C364 L124 G128 H129 T183 N354 K355 N356 T357 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmt A 2.55 BS02 8B0 A 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmt A 2.55 BS04 8B0 B 1 L124 G128 H129 L130 T183 C364 L124 G128 H129 L130 T183 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmt B 2.55 BS02 8B0 A 1 L124 G128 L130 T183 K355 C364 L124 G128 L130 T183 K355 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmt B 2.55 BS04 8B0 B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmu A 2.39 BS02 8A0 A 1 L124 G128 H129 T183 K355 P367 R371 L124 G128 H129 T183 K355 P367 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmu A 2.39 BS03 8A0 B 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmu B 2.39 BS01 8A0 A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmu B 2.39 BS03 8A0 B 1 L124 G128 H129 L130 T183 K355 C364 P367 L124 G128 H129 L130 T183 K355 C364 P367 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmv A 2.16 BS02 8AU A 1 L124 G128 L130 T183 K355 N356 C364 R371 L124 G128 L130 T183 K355 N356 C364 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmv A 2.16 BS04 8AU B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmv B 2.16 BS01 8AU A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmv B 2.16 BS03 8AU B 1 L124 G128 T183 K355 N356 C364 L124 G128 T183 K355 N356 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0016740,0019264,0030170,0035999,0046653 remove_due_to_license_issue A5K8L9 28967982 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5xmx A 2.0 BS01 89L A 1 F246 C249 T252 T253 H287 L294 L303 V305 V312 I328 H413 Y437 F65 C68 T71 T72 H106 L113 L122 V124 V131 I147 H232 Y256 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=37nM, Kd=57nM Q03181 29103972 900 VADLKAFSKHIYNAYLKNFNMTKKKARSILTGAPFVIHDIETLWQAEKGLVWGLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYK 5xo2 A 2.201 BS03 SIA C 1 Y33 R126 Q138 W139 Q140 I142 Y3 R96 Q108 W109 Q110 I112 ? remove_due_to_license_issue Q9UKJ1 29046357 2 MLYGVTQPKHLSASMGGSVEIPFSFYYPWELATAPDVRISWRRGHFHGQSFYSTRPPSIHKDYVNRLFLNWTEGQKSGFLRISNLQKQDQSVYFCRVELDTRSSGRQQWQSIEGTKLSIT 5xo7 A 1.88 BS01 36J A 1 G35 L36 A105 S106 P131 N134 L138 M153 S157 Y160 W185 P190 I193 P194 H243 G32 L33 A102 S103 P128 N131 L135 M150 S154 Y157 W182 P187 I190 P191 H240 ? remove_due_to_license_issue A0A0D2ILK1 301 TRTRGYVTTKDGIKWYYEQEGSGPDVVLIPDGLGECQMFDKPMSLIASNGFRVTTFDMPGMSRSSDAPPETYQDITGRKLAGYIITLLDTLDIKIASVWGCASGASTVLALCSDYPERVRNGMPHEVPTENPDILLHIHEVDPATISQEMAANSRAYSGNVEAWDALGPEVHARLHDNYPRWAYGYPRTIPPSAPVKTEDLHKVPIDWTVGASTPTKLFFENIVIAAREGINIGTLPGNHFPYVSHPEEFAKYVVETSRKYLK 5xof A 1.963 BS03 SIA E 1 Y33 R126 Q138 Q140 I142 Y3 R96 Q108 Q110 I112 ? remove_due_to_license_issue Q9UKJ1 29046357 2 MLYGVTQPKHLSASMGGSVEIPFSFYYPWELATAPDVRISWRRGHFHGQSFYSTRPPSIHKDYVNRLFLNWTEGQKSGFLRISNLQKQDQSVYFCRVELDTRSSGRQQWQSIEGTKLSI 5xpi A 2.2 BS01 8C3 A 1 D145 M148 F152 Y188 Y191 N194 F237 D19 M22 F26 Y45 Y48 N51 F94 2.3.2.27 Kd=5.2uM remove_due_to_license_issue Q96T88 29562800 301 WDETELGLYKVNEYVDARDTNMGAWFEAQVVRVTRKEDVIYHVKYDDYPENGVVQMNSRDVRARARTIIKWQDLEVGQVVMLNYNPDNPKERGFWYDAEISRKRETRTARELYANVVLGDDSLNDCRIIFVDEVFKIERP 5xpl A 2.05 BS02 8C9 A 1 Y143 S233 I264 R270 S271 S274 W282 C284 L305 H393 S394 F418 Y21 S53 I84 R90 S91 S94 W102 C104 L125 H213 S214 F236 ? 0003677,0004879,0006355 ic50=20nM remove_due_to_license_issue P13053 28954197 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSPENSMKLTPLVLEVFG 5xpm A 2.2 BS02 8C0 A 1 Y143 V230 S233 R270 S271 S274 W282 C284 A299 H301 L305 H393 L400 Y21 V49 S52 R89 S90 S93 W101 C103 A118 H120 L124 H212 L219 ? 0003677,0004879,0006355 ic50=23nM remove_due_to_license_issue P13053 28954197 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5xpn A 1.96 BS02 8BO A 1 Y143 L223 V230 S233 R270 S271 S274 W282 C284 A299 H301 L400 Y21 L43 V50 S53 R90 S91 S94 W102 C104 A119 H121 L220 ? 0003677,0004879,0006355 ic50=102nM remove_due_to_license_issue P13053 28954197 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 5xpo A 2.28 BS02 8BL A 1 Y143 L223 S233 R270 S271 S274 W282 C284 V296 H301 Y397 L400 L410 Y21 L43 S53 R90 S91 S94 W102 C104 V116 H121 Y217 L220 L230 ? 0003677,0004879,0006355 ic50=84nM remove_due_to_license_issue P13053 28954197 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 5xpp A 2.85 BS02 8BF A 1 Y143 L223 S233 R270 S271 S274 W282 C284 A299 H301 H393 Y21 L43 S53 R90 S91 S94 W102 C104 A119 H121 H213 ? 0003677,0004879,0006355 remove_due_to_license_issue P13053 28954197 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFG 5xqx A 2.3 BS01 8CC A 1 Y32 A50 K52 F97 A100 L158 D173 Y35 A53 K55 F100 A103 L153 D168 D151 K153 N156 D173 N181 T196 D146 K148 N151 D168 N176 T178 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=410nM P49336 28802632 402 MEFMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQESNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEE 5xs0 F 3.0 BS01 dna Y 0 L132 K133 S134 L137 L108 K109 S110 L113 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 10 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 G 3.0 BS01 dna Y 0 G58 K102 Y104 E130 G131 L132 K133 S134 L137 G34 K78 Y80 E106 G107 L108 K109 S110 L113 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 10 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 H 3.0 BS01 dna Y 0 G58 G59 G34 G35 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 10 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 I 3.0 BS01 dna Z 0 K102 L132 K133 S134 L137 K78 L108 K109 S110 L113 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 9 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 J 3.0 BS01 dna Z 0 G58 G59 G60 K102 G34 G35 G36 K78 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 9 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 N 3.0 BS01 dna Y 0 L132 K133 L108 K109 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 10 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 O 3.0 BS01 dna Y 0 K102 Y104 E130 G131 L132 K133 S134 K78 Y80 E106 G107 L108 K109 S110 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 10 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 P 3.0 BS01 dna Y 0 G58 G59 G34 G35 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 10 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 Q 3.0 BS01 dna W 0 L132 K133 S134 L137 L108 K109 S110 L113 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 6 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 R 3.0 BS01 dna W 0 G58 G59 K102 Y104 E130 G34 G35 K78 Y80 E106 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 6 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 T 3.0 BS01 dna X 0 L132 K133 S134 L137 L108 K109 S110 L113 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 8 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 U 3.0 BS01 dna X 0 G58 G59 K102 Y104 E130 G131 K133 S134 L137 G34 G35 K78 Y80 E106 G107 K109 S110 L113 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 8 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs0 V 3.0 BS01 dna X 0 G58 G59 G34 G35 ? 0000724,0000730,0005634,0006281,0006310,0045002 remove_due_to_license_issue P43351 30428330 1 ~ 8 CFGQCQYTAEEYQAIQKALRQRLGPEYISSRMAGGGQKVCYIEGHRVINLANEMFGYNGWAHSITQQNVDFVDLNNGKFYVGVCAFVRVQLKDGSYHEDVGYGVSEGLKSKALSLEKARKEAVTDGLKRALRSFGNALGNCILDKDYLRSLNKLPRQLPLEVDLTKAKRQDLEPSVEEARYNSC 5xs2 A 2.04 BS01 8D6 A 1 Y32 V35 A50 K52 F97 Y99 A100 L158 D173 Y35 V38 A53 K55 F100 Y102 A103 L161 D176 D151 K153 N156 D173 N181 T196 D154 K156 N159 D176 N184 T199 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=5nM P49336 28802632 402 MEFMDYDFKVKLSSERERVEDLFEYEGCKVGRGTYGHVYKAKRKDGKDDKDYALKQIEGTGISMSACREIALLRELKHPNVISLQKVFLSHADRKVWLLFDYAEHDLWHIIKFHRASKANKKPVQLPRGMVKSLLYQILDGIHYLHANWVLHRDLKPANILVMGEGPERGRVKIADMGFARLFNSPLKPLADLDPVVVTFWYRAPELLLGARHYTKAIDIWAIGCIFAELLTSEPIFHCRQEDIKTSNPYHHDQLDRIFNVMGFPADKDWEDIKKMPEHSTLMKDFRRNTYTNCSLIKYMEKHKVKPDSKAFHLLQKLLTMDPIKRITSEQAMQDPYFLEDPLPTSDVFAGCQIPYPKREFLTEEE 5xs8 A 1.952 BS01 8EX E 1 H36 L37 Y146 R204 K210 W284 L326 L389 R393 H10 L11 Y120 R178 K184 W258 L300 L363 R367 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 29208901 1 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5xs8 A 1.952 BS02 GCD E 1 W284 S287 L389 Q405 Y409 E410 W258 S261 L363 Q379 Y383 E384 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 29208901 2 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 5xsr A 2.3 BS01 8EC A 1 E102 H201 G202 Y228 Y235 F236 A237 S243 Y246 E102 H195 G196 Y222 Y229 F230 A231 S237 Y240 S243 Y246 E327 S237 Y240 E321 2.4.2.-,2.4.2.30 0003950 Kd=0.000000064M remove_due_to_license_issue Kd=2.0nM, IC50=17nM P09874 29335205 401 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHAAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 5xst A 2.3 BS01 8E6 A 1 E102 D105 H201 G202 G227 Y228 Y235 K242 S243 Y246 E103 D106 H202 G203 G228 Y229 Y236 K243 S244 Y247 S243 Y246 E327 S244 Y247 E328 2.4.2.-,2.4.2.30 0003950 ic50=27nM remove_due_to_license_issue IC50=27nM P09874 29335205 401 SKSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSDDSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 5xsu A 2.4 BS01 8E3 A 1 E102 H201 G202 G227 Y228 Y235 F236 A237 K242 S243 Y246 E102 H198 G199 G224 Y225 Y232 F233 A234 K239 S240 Y243 S243 Y246 E327 S240 Y243 E324 2.4.2.-,2.4.2.30 0003950 Kd=180nM remove_due_to_license_issue Kd=1.8nM, IC50=244nM P09874 29335205 407 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGGSSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 5xv7 A 2.32 BS01 EMH A 1 L86 V94 F165 L168 G169 H170 L220 Y227 L20 V28 F99 L102 G103 H104 L154 Y161 2.7.11.1 0004672,0005524,0006468 ic50=11nM remove_due_to_license_issue IC50=11.0nM Q96SB4 29478907 705 YHLVKIGDLFNGRYHVIRKLGWGHFSTVWLSWDIQGKKFVAMKVVKSAEHYTETALDEIRLLKSVRNSDPNDPNREMVVQLLDDFKISGVNGTHIVMVFEVLGHHLLKWIIKSNYQGLPLPCVKKIIQQVLQGLDYLHTKCRIIHTDIKPENILLSVNEQYIRRLAAEATENFLVNPLEPKNAEKLKVKIADLGNACWVHKHFTEDIQTRQYRSLEVLIGSGYNTPADIWSTACMAFELATGDYLFEPHSGEEYTRDEDHIALIIELLGKVPRKLIVAGKYSKEFFTKKGDLKHITKLKPWGLFEVLVEKYEWSQEEAAGFTDFLLPMLELIPEKRATAAECLRHPWLNS 5xva A 1.847 BS01 8FU A 1 I327 G328 E329 V335 A348 E396 F397 L398 E399 G401 D444 L447 D458 I29 G30 E31 V37 A50 E98 F99 L100 E101 G103 D146 L149 D160 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 Ki=0.051uM remove_due_to_license_issue Ki=51nM O96013 29190083 601 SSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNRTR 5xvf A 2.655 BS01 8FR A 1 I327 E329 A348 M395 F397 L398 E399 G401 L447 I29 E31 A50 M97 F99 L100 E101 G103 L149 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=156nM, Ki=710nM O96013 29190083 601 SSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQN 5xvg A 2.1 BS01 8FX A 1 I327 G328 A348 M395 E396 F397 L398 E399 G401 D444 L447 D458 I29 G30 A50 M97 E98 F99 L100 E101 G103 D146 L149 D160 D440 K442 D444 S445 D458 K467 T478 D142 K144 D146 S147 D160 K169 T180 2.7.11.1 0004672,0005524,0006468 Ki=0.009uM remove_due_to_license_issue IC50=11nM, Ki=9nM O96013 29190083 601 SSHEQFRAALQLVVDPGDPRSYLDNFIKIGEGSTGIVCIATVRSSGKLVAVKKMDLRKQQRRELLFNEVVIMRDYQHENVVEMYNSYLVGDELWVVMEFLEGGALTDIVTHTRMNEEQIAAVCLAVLQALSVLHAQGVIHRDIKSDSILLTHDGRVKLSDFGFCAQVSKEVPRRKSLVGTPYWMAPELISRLPYGPEVDIWSLGIMVIEMVDGEPPYFNEPPLKAMKMIRDNLPPRLKNLHKVSPSLKGFLDRLLVRDPAQRATAAELLKHPFLAKAGPPASIVPLMRQNRTR 5xvk A 1.88 BS02 8GC A 1 Y24 L164 A198 S201 Y204 S213 Y242 Y21 L161 A195 S198 Y201 S210 Y239 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0031100,0032259,0045722,0090312 ic50=9uM remove_due_to_license_issue O55239 28720493 302 GFTSKDTYLSHFNPRDYLEKYYSFGSRHCAENEILRHLLKNLFKIFCLGAVKGELLIDIGSGPTIYQLLSACESFTEIIVSDYTDQNLWELQKWLKKEPGAFDWSPVVTYVCDLEGNRMKGPEKEEKLRRAIKQVLKCDVTQSQPLGGVSLPPADCLLSTLCLDAACPDLPAYRTALRNLGSLLKPGGFLVMVDALKSSYYMIGEQKFSSLPLGWETVRDAVEEAGYTIEQFEVISQNYSSTTSNNEGLFSLVGRKPGRSE 5xvq A 2.29 BS02 8GC A 1 Y20 L164 A198 S201 Y204 S213 Y242 Y16 L155 A189 S192 Y195 S204 Y233 ? 0005829,0006769,0008112,0008168,0008757,0032259,0045722,0090312 ic50=9uM remove_due_to_license_issue F7ERX8 28720493 302 FTSKDTYLRHFNPRDYLEKYYKSAESQILKHLLENLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIIVTDYSDQNLQELEKWLKKEPEAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPLADCLLSTLCLDAACPDLPTYRRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVGRKLS 5xvu A 3.0 BS01 ATP A 1 G50 K53 Y54 S55 V57 A70 K72 I120 M167 I178 S179 G39 K42 Y43 S44 V46 A59 K61 I109 M156 I167 S168 D160 K162 N165 S179 S198 D149 K151 N154 S168 S187 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005737,0005829,0005956,0006338,0006468,0006974,0018105,0019901,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0046777,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 remove_due_to_license_issue Q8IIR9 29743645 403 IPKFYADVNIHKPKEYYDYDNLELQWNKPNRYEIMKKIGRGKYSEVFNGYDTECNRPCAIKVLKPVKKKKIKREIKILQNLNGGPNIIKLLDIVKDPVTKTPSLIFEYINNIDFKTLYPKFTDKDIRYYIYQILKALDYCHSQGIMHRDVKPHNIMIDHENRQIRLISWGLAEFYHPGQEYNVRVASRYYKGPELLIDLQLYDYSLDIWSLGCMLAGMIFKKEPFFCGHDNYDQLVKIAKVLGTEDLHAYLKKYNIKLKPHYLNILGEYERKPWSHFLTQSNIDIAKDEVIDLIDKMLIYDHAKRIAPKEAMEHPYFREVR 5xw6 B 3.1 BS01 128 C 1 T112 H131 K236 Y274 K298 Y300 T86 H105 K210 Y248 K272 Y274 0001614,0004931,0005886,0033198,0098655 remove_due_to_license_issue 29026074 502 SCVKWFIYGVIAVYICYTLIVHKRYQEKEELTSSVRVTLKGVAHVDRIWDAAEYTIPTQTRDSFFVMTNIIRTENQIQKTCPEYPTAKAICSSDKSCAKGIVDVHSNGVQTGKCVHYNITHKTCEIKAWCPVQGEERPPVPAVLRSSEDFTVFIKNNIHFPTFQYTVQNISPKLNTSCKFNKVTAPLCPIFRLGDILQEAKENFSEMAVKGGIIAIEIKWDCDLDSWSYYCSPEYSFRRLDDKTRTQYPGFSIRFARHYKLPDGTEQRTLFKAYGIRFDVLVFGMGGQFKLIELFTFIGSTIAYFGLAVTIIEMCFHLYN 5xw6 B 3.1 BS02 128 B 1 T64 K66 T177 V178 F179 K181 T202 T38 K40 T151 V152 F153 K155 T176 0001614,0004931,0005886,0033198,0098655 remove_due_to_license_issue 29026074 401 SCVKWFIYGVIAVYICYTLIVHKRYQEKEELTSSVRVTLKGVAHVDRIWDAAEYTIPTQTRDSFFVMTNIIRTENQIQKTCPEYPTAKAICSSDKSCAKGIVDVHSNGVQTGKCVHYNITHKTCEIKAWCPVQGEERPPVPAVLRSSEDFTVFIKNNIHFPTFQYTVQNISPKLNTSCKFNKVTAPLCPIFRLGDILQEAKENFSEMAVKGGIIAIEIKWDCDLDSWSYYCSPEYSFRRLDDKTRTQYPGFSIRFARHYKLPDGTEQRTLFKAYGIRFDVLVFGMGGQFKLIELFTFIGSTIAYFGLAVTIIEMCFHLYN 5xw6 C 3.1 BS01 128 C 1 T64 K66 T177 F179 T202 I216 T38 K40 T151 F153 T176 I190 0001614,0004931,0005886,0033198,0098655 remove_due_to_license_issue 29026074 502 SCVKWFIYGVIAVYICYTLIVHKRYQEKEELTSSVRVTLKGVAHVDRIWDAAEYTIPTQTRDSFFVMTNIIRTENQIQKTCPEYPTAKAICSSDKSCAKGIVDVHSNGVQTGKCVHYNITHKTCEIKAWCPVQGEERPPVPAVLRSSEDFTVFIKNNIHFPTFQYTVQNISPKLNTSCKFNKVTAPLCPIFRLGDILQEAKENFSEMAVKGGIIAIEIKWDCDLDSWSYYCSPEYSFRRLDDKTRTQYPGFSIRFARHYKLPDGTEQRTLFKAYGIRFDVLVFGMGGQFKLIELFTFIGSTIAYFGLAVTIIEMCFHLYN 5xw6 C 3.1 BS02 128 A 1 T112 A113 V130 K236 Y274 K298 Y300 T86 A87 V104 K210 Y248 K272 Y274 0001614,0004931,0005886,0033198,0098655 remove_due_to_license_issue 29026074 401 SCVKWFIYGVIAVYICYTLIVHKRYQEKEELTSSVRVTLKGVAHVDRIWDAAEYTIPTQTRDSFFVMTNIIRTENQIQKTCPEYPTAKAICSSDKSCAKGIVDVHSNGVQTGKCVHYNITHKTCEIKAWCPVQGEERPPVPAVLRSSEDFTVFIKNNIHFPTFQYTVQNISPKLNTSCKFNKVTAPLCPIFRLGDILQEAKENFSEMAVKGGIIAIEIKWDCDLDSWSYYCSPEYSFRRLDDKTRTQYPGFSIRFARHYKLPDGTEQRTLFKAYGIRFDVLVFGMGGQFKLIELFTFIGSTIAYFGLAVTIIEMCFHLYN 5xyx A 2.61 BS01 FTZ A 1 K53 T106 H107 L108 M109 D168 K44 T97 H98 L99 M100 D155 D150 K152 N155 D168 T185 D137 K139 N142 D155 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=14445nM Q16539 28945083 401 ERPTFYRQELNKTIWEVPERYQNLSPVSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 5xyy A 1.7 BS01 P0F A 1 A51 I84 T106 H107 M109 D112 D168 A48 I81 T103 H104 M106 D109 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T182 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=9.221uM remove_due_to_license_issue Q16539 28945083 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 5xyz A 2.64 BS01 GYL A 1 A428 T474 E475 Y476 M477 G480 C481 L528 S538 A28 T68 E69 Y70 M71 G74 C75 L119 S129 D521 R525 N526 D539 D112 R116 N117 D130 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 28945083 701 SWEIDPKDLTFLKELVKYGKWRGQYDVAIKMIKMSDEEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLRERFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRFPVRWSPPEVLMFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMD 5xzr A 2.8 BS01 8J6 A 1 E110 R111 F113 H114 N217 T218 E250 T253 P491 K492 E110 R111 F113 H114 N217 T218 E247 T250 P476 K477 V25 G49 L436 S502 V505 V25 G49 L421 S487 V490 3.1.3.48 0000077,0001784,0004721,0004725,0004726,0005158,0005515,0005634,0005654,0005737,0005739,0005829,0006338,0006470,0006629,0006641,0007165,0007173,0007229,0007409,0007420,0007507,0008543,0009755,0009967,0016311,0019221,0019901,0021697,0030159,0030220,0030946,0030971,0031295,0031666,0032331,0032480,0032528,0032728,0032760,0032991,0033628,0033629,0035264,0035265,0035335,0035855,0036302,0038127,0042445,0042593,0043254,0043408,0045296,0045778,0045931,0046326,0046628,0046676,0046825,0046887,0046888,0048008,0048011,0048013,0048806,0048839,0048873,0050731,0050839,0051428,0051463,0060020,0060090,0060125,0060325,0060338,0061582,0070374,0071364,0140793,1902564,1990782 remove_due_to_license_issue Q06124 29155585 601 MTSRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAALVQYYMEHHGQLKEKNGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQSHPGDFVLSVRTGDDKGESNDGKSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLAEKVKQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPNEPVSDYINANIIMPKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETLQRRIEEEQK 5y0f A 1.54 BS01 8JO A 1 F16 M20 T74 A75 D76 R78 I104 V115 C117 R126 Y128 F21 M25 T79 A80 D81 R83 I109 V120 C122 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.21uM remove_due_to_license_issue IC50=1690nM, Ki=210nM P15090 29775936 200 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5y0g A 1.542 BS01 8JL A 1 F16 Y19 M20 A33 T74 A75 D76 R78 C117 R126 Y128 F21 Y24 M25 A38 T79 A80 D81 R83 C122 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.2uM remove_due_to_license_issue IC50=1650nM, Kd=1.4nM, Ki=200nM P15090 29775936 200 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5y0x A 1.604 BS01 8JR A 1 F16 M20 D76 R78 C117 R126 Y128 F21 M25 D81 R83 C122 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=7.75uM remove_due_to_license_issue Kd=6.0nM, Ki=7750nM P15090 29775936 200 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5y0z A 2.0 BS02 8K9 A 1 F96 R97 F119 Y139 P140 I169 H187 F190 V233 F235 F41 R42 F64 Y84 P85 I114 H132 F135 V178 F180 P94 D95 F96 R97 N168 D170 H187 P39 D40 F41 R42 N113 D115 H132 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=0.46uM remove_due_to_license_issue Q8IXJ6 29685974 502 ERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPSTGLYDNLEKYHLPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5y12 A 1.75 BS01 8JX A 1 F16 M20 T74 A75 D76 R78 I104 C117 R126 Y128 F21 M25 T79 A80 D81 R83 I109 C122 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=0.59uM remove_due_to_license_issue Ki=590nM P15090 29775936 201 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5y13 A 1.75 BS01 8K0 A 1 F16 M20 A33 T74 D76 R78 R126 Y128 F21 M25 A38 T79 D81 R83 R131 Y133 ? 0005324,0005504,0005634,0005737,0005811,0005829,0008289,0009617,0015908,0015909,0036041,0042632,0045892,0050729,0050872,0050873,0051427,0070062,0071285,0071356,0120162 Ki=1.16uM remove_due_to_license_issue Ki=1160nM P15090 29775936 201 RGSHMCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA 5y1y A 1.912 BS01 HNQ A 1 V87 L92 L94 C136 N140 I146 V45 L50 L52 C94 N98 I104 ? ic50=0.98uM remove_due_to_license_issue IC50=980nM O60885 29087414 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5y2f A 2.53 BS03 8L9 A 1 N2 F80 T83 F84 E85 N2 F80 T83 F84 E85 P60 D61 F62 R63 N112 D114 H131 P60 D61 F62 R63 N112 D114 H131 2.3.1.-,2.3.1.286,2.4.2.- 0070403 remove_due_to_license_issue EC50=5700nM Q8N6T7 30374165 402 VNYAAGLSPYADKGKCGLPEIFDPPEELERKVWELARLVWQSSSVVFHTGAGISTASGIPDFRGPHGVWTMEERGLAPKFDTTFESARPTQTHMALVQLERVGLLRFLVSQNVDGLHVRSGFPRDKLAELHGNMFVEECAKCKTQYVRDTVVGTMGLKATGRLCTVAKARGLRACRGELRDTILDWEDSLPDRDLALADEASRNADLSITLGTSLQIRPSGNLPLATKRRGGRLVIVNLQPTKHDRHADLRIHGYVDEVMTRLMKHLGLEIPAWDGPRVLERALPPLPRPPTPKLEP 5y3n A 2.4 BS01 8MF A 1 A123 I161 G162 M163 F201 F205 W231 A54 I92 G93 M94 F104 F108 W134 ? 0005524,0006457,0016887,0051082,0140662 ic50=0.079uM remove_due_to_license_issue IC50=79nM Q12931 28816449 601 PLHSIISSTESVQGSTSKHEFQAETKKLLDIVARSLYSEKEVFIRELISNASDALEKLRHKLVSDGQALPEMEIHLQTNAEKGTITIQDTGIGMTQEELVSNQFGVGFYSAFMVADRVEVYSRSAAPGSLGYQWLSDGSGVFEIAEASGVRTGTKIIIHLKSDCKEFSSEARVRDVVTKYSNFVSFPLYLNGRRMNTLQAIWMMDPKDVREWQHEEFYRYVAQAHDKPRYTLHYKTDAPLNIRSIFYVPDMKPSVALYSRKVLIQTKATDILPKWLRFIRGVVDSEDIPLLQESALIRKLRDVLQQRLIKFFIDQSKKDAEKYAKFFEDYGLFMREGIVTATEQEVKEDIAKLLRYESSALPSGQLTSLSEYASRMRAGTRNIYYLCAPNRHLAEHSPYYEAMKKKDTEVLFCFEQFDELTLLHLREFDKKKLISVET 5y3o A 2.7 BS01 8M9 A 1 D158 I161 G162 M163 F201 F205 V217 W231 T251 D90 I93 G94 M95 F103 F107 V119 W133 T153 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=138nM Q12931 28816449 601 EPLHSIISSTESVQGSTSKHEFQAETKKLLDIVARSLYSEKEVFIRELISNASDALEKLRHKLVSDGQALPEMEIHLQTNAEKGTITIQDTGIGMTQEELVSFGVGFYSAFMVADRVEVYSRSAAPGSLGYQWLSDGSGVFEIAEASGVRTGTKIIIHLKSDCKEFSSEARVRDVVTKYSNFVSFPLYLNGRRMNTLQAIWMMDPKDVREWQHEEFYRYVAQAHDKPRYTLHYKTDAPLNIRSIFYVPDMKPSVALYSRKVLIQTKATDILPKWLRFIRGVVDSEDIPSALIRKLRDVLQQRLIKFFIDQSKKDAEKYAKFFEDYGLFMREGIVTATEQEVKEDIAKLLRYESSALPSGQLTSLSEYASRMRAGTRNIYYLCAPNRHLAEHSPYYEAMKKKDTEVLFCFEQFDELTLLHLREFDKKKLISVET 5y48 A 1.7 BS01 URA A 1 Y70 I71 E85 G109 N110 Y70 I71 E85 G109 N110 I71 E160 R163 I71 E160 R163 3.2.2.22 0000166,0006952,0016787,0017148,0030598,0035821,0090729 remove_due_to_license_issue D9J2T9 30007053 301 DVSFRLSGADPSSYGMFIKDLRNALPHTEKVYNIPLLLPSVSGAGRYLLMHLFNYDGNTITVAVDVTNVYIMGYLALTTSYFFNEPAADLASQYVFRSARRKITLPYSGNYERLQIAAGKPREKIPIGLPALDTAISTLLHYDSTAAAGALLVLIQTTAEAARFKYIEQQIQERAYRDEVPSSATISLENSWSGLSKQIQLAQGNNGVFRTPTVLVDSKGNRVQITNVTSNVVTSNIQLLLNTKNI 5y58 A 2.8 BS01 rna X 0 H292 E293 K294 V297 R298 Y299 R316 K333 N424 S425 H426 D453 R456 H256 E257 K258 V261 R262 Y263 R280 K297 N388 S389 H390 D417 R420 3.6.4.12 0000723,0000724,0000725,0000727,0000781,0003677,0003678,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005635,0005694,0006281,0006303,0006310,0006325,0009378,0016787,0016887,0030466,0031509,0032508,0036121,0042162,0043564,0061749,0061775,0070034,0097552,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P32807 29290466 286 ~ 315 IHEGILFCIELSETMFKESSDLEYKSPLLEILESLDELMSQLVITRPGTAIGCYFYYCNREDAKEGIYELFPLRDINATFMKKLNDLLEDLSSGRISLYDYFMFQQTGSEKQVRLSVLFTFMLDTFLEEIPGQKQLSNKRVFLFTDIDKPQEAQDIDERARLRRLTIDLFDNKVNFATFFIGYADKPFDNEFYSDILQLGDSEFDGPSTKPIDAKYIKSRILRKKEVKRIMFQCPLILDEKTNFIVGVKGYTMYTHEKAGVRYKLVYEHEDIRQEAYSKRKFLNPITGEDVTGKTVKVYPYGDLDINLSDSQDQIVMEAYTQKDAFLKIIGFRSSSKSIHYFNNIDKSSFIVPDEAKYEGSIRTLASLLKILRKKDKIAILWGKLKSNSHPSLYTLSPSSVKDYNEGFYLYRVPFLDEIRKFPSLLSYDDGSEHKLDYDNMKKVTQSIMGYFNLRDGYNPSDFKNPLLQKHYKVLHDYLLQIETTFDENETPNTKKDRMMREDDSLRKLYYIRNKILESEKSEDPIIQRLNKYVKIWNMFYKKFNDDN 5y58 A 2.8 BS02 rna Y 0 R122 R537 R95 R501 3.6.4.12 0000723,0000724,0000725,0000727,0000781,0003677,0003678,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005635,0005694,0006281,0006303,0006310,0006325,0009378,0016787,0016887,0030466,0031509,0032508,0036121,0042162,0043564,0061749,0061775,0070034,0097552,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P32807 29290466 286 ~ 315 IHEGILFCIELSETMFKESSDLEYKSPLLEILESLDELMSQLVITRPGTAIGCYFYYCNREDAKEGIYELFPLRDINATFMKKLNDLLEDLSSGRISLYDYFMFQQTGSEKQVRLSVLFTFMLDTFLEEIPGQKQLSNKRVFLFTDIDKPQEAQDIDERARLRRLTIDLFDNKVNFATFFIGYADKPFDNEFYSDILQLGDSEFDGPSTKPIDAKYIKSRILRKKEVKRIMFQCPLILDEKTNFIVGVKGYTMYTHEKAGVRYKLVYEHEDIRQEAYSKRKFLNPITGEDVTGKTVKVYPYGDLDINLSDSQDQIVMEAYTQKDAFLKIIGFRSSSKSIHYFNNIDKSSFIVPDEAKYEGSIRTLASLLKILRKKDKIAILWGKLKSNSHPSLYTLSPSSVKDYNEGFYLYRVPFLDEIRKFPSLLSYDDGSEHKLDYDNMKKVTQSIMGYFNLRDGYNPSDFKNPLLQKHYKVLHDYLLQIETTFDENETPNTKKDRMMREDDSLRKLYYIRNKILESEKSEDPIIQRLNKYVKIWNMFYKKFNDDN 5y58 B 2.8 BS01 rna X 0 K39 R41 K42 T43 S204 K251 L256 N257 R258 S278 R318 Y323 V531 Q535 K38 R40 K41 T42 S187 K234 L239 N240 R241 S261 R290 Y295 V503 Q507 3.6.4.12 0000723,0000724,0000725,0000781,0003677,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005694,0006281,0006303,0006310,0006325,0007535,0009378,0016787,0016887,0031509,0032508,0034502,0036121,0042162,0043564,0061749,0061775,0070034,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q04437 29290466 286 ~ 315 SSESTTFIVDVSPSMMKNNNVSKSMAYLEYTLLNKSKKSRKTDWISCYLANCPVSENSQEIPNVFQIQSFLAPVTTTATIGFIKRLKQYCDQHSHDSMIQCLLVVSLDIKQQFQARKILKQIVVFTDNLDDLDITDEEIDLLTEELSTRIILIDCGSNWLKLVEAIPNSRIYNMNELLVEITSPATSVVKPVRVFSGELRLGADILSTQTSNPSGSMQDENCLCIKVEAFPATKAVSGLNRKTAVEVEDSQKKERYVGVKSIIEYEIHNEGGSSYIPVTISKDSVTKAYRYGADYVVLPSVLVDQTVYESFPGLDLRGFLNREALPRYFLTSESSFITADTRLGCQSDLMAFSALVDVMLENRKIAVARYVSKKDSEVNMCALCPVLIEHSNINSEKKFVKSLTLCRLPFAEDERVTDFPKLLDRTTTSGVPLKKETDGHQIDELMEQFVDSMDTDELPEIPLGNYYQPIGEVTTDTTLPLPSLNKDQEENKKDPLRIPTVFVYRQQQVLLEWIHQLMINDSREFEIPELPDSLKNKISPYTHKKFDSTKLVEVLGIKKVKRGEQHSR 5y58 C 2.8 BS01 rna Y 0 H292 E293 K294 V297 R298 Y299 R316 K333 N424 S425 H426 D453 R456 H256 E257 K258 V261 R262 Y263 R280 K297 N388 S389 H390 D417 R420 3.6.4.12 0000723,0000724,0000725,0000727,0000781,0003677,0003678,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005635,0005694,0006281,0006303,0006310,0006325,0009378,0016787,0016887,0030466,0031509,0032508,0036121,0042162,0043564,0061749,0061775,0070034,0097552,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P32807 29290466 286 ~ 315 IHEGILFCIELSETMFKESSDLEYKSPLLEILESLDELMSQLVITRPGTAIGCYFYYCNREDAKEGIYELFPLRDINATFMKKLNDLLEDLSSGRISLYDYFMFQQTGSEKQVRLSVLFTFMLDTFLEEIPGQKQLSNKRVFLFTDIDKPQEAQDIDERARLRRLTIDLFDNKVNFATFFIGYADKPFDNEFYSDILQLGDSEFDGPSTKPIDAKYIKSRILRKKEVKRIMFQCPLILDEKTNFIVGVKGYTMYTHEKAGVRYKLVYEHEDIRQEAYSKRKFLNPITGEDVTGKTVKVYPYGDLDINLSDSQDQIVMEAYTQKDAFLKIIGFRSSSKSIHYFNNIDKSSFIVPDEAKYEGSIRTLASLLKILRKKDKIAILWGKLKSNSHPSLYTLSPSSVKDYNEGFYLYRVPFLDEIRKFPSLLSYDDGSEHKLDYDNMKKVTQSIMGYFNLRDGYNPSDFKNPLLQKHYKVLHDYLLQIETTFDENETPNTKKDRMMREDDSLRKLYYIRNKILESEKSEDPIIQRLNKYVKIWNMFYKKFNDDN 5y58 C 2.8 BS02 rna Z 0 R122 R537 R543 Y547 R95 R501 R507 Y511 3.6.4.12 0000723,0000724,0000725,0000727,0000781,0003677,0003678,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005635,0005694,0006281,0006303,0006310,0006325,0009378,0016787,0016887,0030466,0031509,0032508,0036121,0042162,0043564,0061749,0061775,0070034,0097552,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P32807 29290466 286 ~ 315 IHEGILFCIELSETMFKESSDLEYKSPLLEILESLDELMSQLVITRPGTAIGCYFYYCNREDAKEGIYELFPLRDINATFMKKLNDLLEDLSSGRISLYDYFMFQQTGSEKQVRLSVLFTFMLDTFLEEIPGQKQLSNKRVFLFTDIDKPQEAQDIDERARLRRLTIDLFDNKVNFATFFIGYADKPFDNEFYSDILQLGDSEFDGPSTKPIDAKYIKSRILRKKEVKRIMFQCPLILDEKTNFIVGVKGYTMYTHEKAGVRYKLVYEHEDIRQEAYSKRKFLNPITGEDVTGKTVKVYPYGDLDINLSDSQDQIVMEAYTQKDAFLKIIGFRSSSKSIHYFNNIDKSSFIVPDEAKYEGSIRTLASLLKILRKKDKIAILWGKLKSNSHPSLYTLSPSSVKDYNEGFYLYRVPFLDEIRKFPSLLSYDDGSEHKLDYDNMKKVTQSIMGYFNLRDGYNPSDFKNPLLQKHYKVLHDYLLQIETTFDENETPNTKKDRMMREDDSLRKLYYIRNKILESEKSEDPIIQRLNKYVKIWNMFYKKFNDDN 5y58 D 2.8 BS01 rna Y 0 K39 R41 K42 T43 S204 K251 L256 N257 R258 S278 R318 Y323 V531 Q535 K38 R40 K41 T42 S184 K231 L236 N237 R238 S258 R287 Y292 V495 Q499 3.6.4.12 0000723,0000724,0000725,0000781,0003677,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005694,0006281,0006303,0006310,0006325,0007535,0009378,0016787,0016887,0031509,0032508,0034502,0036121,0042162,0043564,0061749,0061775,0070034,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q04437 29290466 286 ~ 315 SSESTTFIVDVSPSMMKNNNVSKSMAYLEYTLLNKSKKSRKTDWISCYLANCPVSENSQEIPNVFQIQSFLAPVTTTATIGFIKRLKQYCDQHSMIQCLLVVSLDIKQQFQARKILKQIVVFTDNLDDLDITDEEIDLLTEELSTRIILIDCGSNWLKLVEAIPNSRIYNMNELLVEITSPATSVVKPVRVFSGELRLGADILSTQTSNPSGSMQDENCLCIKVEAFPATKAVSGLNRKTAVEVEDSQKKERYVGVKSIIEYEIHNEGGSSYIPVTISKDSVTKAYRYGADYVVLPSVLVDQTVYESFPGLDLRGFLNREALPRYFLTSESSFITADTRLGCQSDLMAFSALVDVMLENRKIAVARYVSKKDSEVNMCALCPVLIEHSNINSEKKFVKSLTLCRLPFAEDERVTDFPKLLDRTTTSGVPLKKETDGHQIDELMEQFVDSMDTDELPEIPLGNYYQPIGEVTTDTTLPLPSLENKKDPLRIPTVFVYRQQQVLLEWIHQLMINDSREFEIPELPDSLKNKISPYTHKKFDSTKLVEVLGIKKVKRGEQHSR 5y58 E 2.8 BS01 rna X 0 R122 R537 R543 Y547 R95 R501 R507 Y511 3.6.4.12 0000723,0000724,0000725,0000727,0000781,0003677,0003678,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005635,0005694,0006281,0006303,0006310,0006325,0009378,0016787,0016887,0030466,0031509,0032508,0036121,0042162,0043564,0061749,0061775,0070034,0097552,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P32807 29290466 286 ~ 315 IHEGILFCIELSETMFKESSDLEYKSPLLEILESLDELMSQLVITRPGTAIGCYFYYCNREDAKEGIYELFPLRDINATFMKKLNDLLEDLSSGRISLYDYFMFQQTGSEKQVRLSVLFTFMLDTFLEEIPGQKQLSNKRVFLFTDIDKPQEAQDIDERARLRRLTIDLFDNKVNFATFFIGYADKPFDNEFYSDILQLGDSEFDGPSTKPIDAKYIKSRILRKKEVKRIMFQCPLILDEKTNFIVGVKGYTMYTHEKAGVRYKLVYEHEDIRQEAYSKRKFLNPITGEDVTGKTVKVYPYGDLDINLSDSQDQIVMEAYTQKDAFLKIIGFRSSSKSIHYFNNIDKSSFIVPDEAKYEGSIRTLASLLKILRKKDKIAILWGKLKSNSHPSLYTLSPSSVKDYNEGFYLYRVPFLDEIRKFPSLLSYDDGSEHKLDYDNMKKVTQSIMGYFNLRDGYNPSDFKNPLLQKHYKVLHDYLLQIETTFDENETPNTKKDRMMREDDSLRKLYYIRNKILESEKSEDPIIQRLNKYVKIWNMFYKKFNDDN 5y58 E 2.8 BS02 rna Z 0 H292 E293 K294 V297 R298 Y299 R316 K333 N424 S425 H426 D453 R456 H256 E257 K258 V261 R262 Y263 R280 K297 N388 S389 H390 D417 R420 3.6.4.12 0000723,0000724,0000725,0000727,0000781,0003677,0003678,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005635,0005694,0006281,0006303,0006310,0006325,0009378,0016787,0016887,0030466,0031509,0032508,0036121,0042162,0043564,0061749,0061775,0070034,0097552,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P32807 29290466 286 ~ 315 IHEGILFCIELSETMFKESSDLEYKSPLLEILESLDELMSQLVITRPGTAIGCYFYYCNREDAKEGIYELFPLRDINATFMKKLNDLLEDLSSGRISLYDYFMFQQTGSEKQVRLSVLFTFMLDTFLEEIPGQKQLSNKRVFLFTDIDKPQEAQDIDERARLRRLTIDLFDNKVNFATFFIGYADKPFDNEFYSDILQLGDSEFDGPSTKPIDAKYIKSRILRKKEVKRIMFQCPLILDEKTNFIVGVKGYTMYTHEKAGVRYKLVYEHEDIRQEAYSKRKFLNPITGEDVTGKTVKVYPYGDLDINLSDSQDQIVMEAYTQKDAFLKIIGFRSSSKSIHYFNNIDKSSFIVPDEAKYEGSIRTLASLLKILRKKDKIAILWGKLKSNSHPSLYTLSPSSVKDYNEGFYLYRVPFLDEIRKFPSLLSYDDGSEHKLDYDNMKKVTQSIMGYFNLRDGYNPSDFKNPLLQKHYKVLHDYLLQIETTFDENETPNTKKDRMMREDDSLRKLYYIRNKILESEKSEDPIIQRLNKYVKIWNMFYKKFNDDN 5y58 F 2.8 BS01 rna Z 0 K39 R41 K42 T43 S204 K251 L256 N257 R258 S278 R318 Y323 V531 Q535 K38 R40 K41 T42 S187 K234 L239 N240 R241 S261 R287 Y292 V500 Q504 3.6.4.12 0000723,0000724,0000725,0000781,0003677,0003684,0003689,0003690,0004386,0005515,0005524,0005634,0005694,0006281,0006303,0006310,0006325,0007535,0009378,0016787,0016887,0031509,0032508,0034502,0036121,0042162,0043564,0061749,0061775,0070034,0097695,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue Q04437 29290466 286 ~ 315 SSESTTFIVDVSPSMMKNNNVSKSMAYLEYTLLNKSKKSRKTDWISCYLANCPVSENSQEIPNVFQIQSFLAPVTTTATIGFIKRLKQYCDQHSHDSMIQCLLVVSLDIKQQFQARKILKQIVVFTDNLDDLDITDEEIDLLTEELSTRIILIDCGSNWLKLVEAIPNSRIYNMNELLVEITSPATSVVKPVRVFSGELRLGADILSTQTSNPSGSMQDENCLCIKVEAFPATKAVSGLNRKTAVEVEDSQKKERYVGVKSIIEYEIHNEGYIPVTISKDSVTKAYRYGADYVVLPSVLVDQTVYESFPGLDLRGFLNREALPRYFLTSESSFITADTRLGCQSDLMAFSALVDVMLENRKIAVARYVSKKDSEVNMCALCPVLIEHSNINSEKKFVKSLTLCRLPFAEDERVTDFPKLLDRTTTSGVPLKKETDGHQIDELMEQFVDSMDTDELPEIPLGNYYQPIGEVTTDTTLPLPSLNKDQEENKKDPLRIPTVFVYRQQQVLLEWIHQLMINDSREFEIPELPDSLKNKISPYTHKKFDSTKLVEVLGIKKVKRGEQHSR 5y5n A 2.3 BS02 8NO A 1 F96 R97 F119 F131 A135 P140 F143 I169 F190 I232 V233 F63 R64 F75 F87 A91 P96 F99 I125 F146 I188 V189 P94 D95 F96 R97 N168 D170 H187 P61 D62 F63 R64 N124 D126 H143 2.3.1.-,2.3.1.286 0017136,0051287,0070403 remove_due_to_license_issue IC50=1000nM Q8IXJ6 28989670 1002 GEADMDFLRNLFSQTLSLGSQKERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPHLPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5y5t A 1.8 BS01 8OR A 1 A400 M448 E449 A451 G454 P455 L501 D512 A33 M76 E77 A79 G82 P83 L129 D140 D494 R498 N499 D512 D122 R126 N127 D140 2.7.10.2 0004672,0004713,0005524,0006468 ic50=211nM remove_due_to_license_issue P43405 29890824 701 VYLDRKLLTLEDKELGTVKKGYYQMKKVVKTVAVKILKNALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN 5y5u A 2.14 BS01 8OU A 1 L377 G378 V385 A400 M448 E449 M450 A451 E452 G454 P455 L501 L14 G15 V22 A37 M80 E81 M82 A83 E84 G86 P87 L133 D494 R498 N499 D512 D126 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 ic50=17.7nM remove_due_to_license_issue P43405 29890824 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV 5y62 B 3.0 BS01 5GP B 1 R60 R175 H177 R23 R138 H140 ? remove_due_to_license_issue Q9I4L4 28870806 600 RTSIEQRSNAVSQVLLGIFSYVRWPKEPAVLQLCVVGPTEYADGLLRGMVQANGRRVHAERRAVDNPDLGTLCNVIYLGVVDERERQQVFRSLAGHPVLSISERGTECSVGSMFCLNVGGPRITFEANLDSIARSGVRVHPSVLKLAR 5y6d A 2.1 BS03 8PL A 1 F62 Y67 W87 D118 H179 R205 N210 H240 F31 Y36 W56 D87 H148 R174 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=54.8nM remove_due_to_license_issue Q9K2N0 29353720 304 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTN 5y6e A 1.8 BS03 8PO A 1 Y67 W87 D118 H179 R205 G209 N210 H240 Y36 W56 D87 H148 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=13.7nM remove_due_to_license_issue Q9K2N0 29353720 304 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 5y6f A 2.3 BS01 C2E A 1 R113 R114 R115 R118 D145 L146 S147 G149 G150 M151 G152 I189 S210 F211 R212 R112 R113 R114 R117 D142 L143 S144 G146 G147 M148 G149 I181 S193 F194 R195 ? 0000166,0005515,0009288,0009425,0035438,0071945,0071973,1902201 remove_due_to_license_issue P76010 31836667 302 SHYHEQFLKQNPLAVLGVLRDLHKAAIPLRLSWNGGQLISKLLAITPDKLVLDFGSQAEDNIAVLKAQHITITAETQGAKVEFTVEQLQQSEYLQLPAFITVPPPTLWFVQRRRYFRISAPPPYFCQTKLADNSTLRFRLYDLSLGGMGALLAELQEGMRFAQIEVNMGQWGVFHFDAQLISISERITTPRLSFRFLNVSPTVERQLQRIIFSLEREAREKADKVR 5y6f A 2.3 BS02 C2E A 2 E76 G79 K81 V111 R113 R114 R118 I189 S190 R208 S210 E75 G78 K80 V110 R112 R113 R117 I181 S182 R191 S193 ? 0000166,0005515,0009288,0009425,0035438,0071945,0071973,1902201 remove_due_to_license_issue P76010 31836667 303 SHYHEQFLKQNPLAVLGVLRDLHKAAIPLRLSWNGGQLISKLLAITPDKLVLDFGSQAEDNIAVLKAQHITITAETQGAKVEFTVEQLQQSEYLQLPAFITVPPPTLWFVQRRRYFRISAPPPYFCQTKLADNSTLRFRLYDLSLGGMGALLAELQEGMRFAQIEVNMGQWGVFHFDAQLISISERITTPRLSFRFLNVSPTVERQLQRIIFSLEREAREKADKVR 5y6g A 2.3 BS01 C2E A 1 R113 R114 R118 S192 R208 S210 R2 R3 R7 S81 R97 S99 ? 0035438 remove_due_to_license_issue P76010 31836667 301 QRRRYFRISAPLHPPYFCQTKLADNSTLRFRLYDLSLGGMGALLETAKPAELQEGMRFAQIEVNMGQWGVFHFDAQLISISERKVIDGKNETITTPRLSFRFLNVSPTVERQLQRIIFSLEREAREKADKV 5y6g A 2.3 BS02 C2E A 2 R113 R114 R115 R118 D145 G149 G150 M151 G152 R208 S210 F211 R212 R2 R3 R4 R7 D34 G38 G39 M40 G41 R97 S99 F100 R101 ? 0035438 remove_due_to_license_issue P76010 31836667 302 QRRRYFRISAPLHPPYFCQTKLADNSTLRFRLYDLSLGGMGALLETAKPAELQEGMRFAQIEVNMGQWGVFHFDAQLISISERKVIDGKNETITTPRLSFRFLNVSPTVERQLQRIIFSLEREAREKADKV 5y6k A 2.86 BS02 8R6 A 1 D63 Y188 K206 K296 D61 Y186 K204 K294 ? 0005515,0005576,0005615,0005768,0005769,0005770,0005788,0005886,0005905,0006826,0006879,0007015,0008198,0008199,0009617,0009925,0009986,0010008,0016020,0016324,0019731,0019899,0030139,0030316,0030669,0031410,0031647,0031982,0032436,0034756,0034774,0034986,0042327,0044325,0045178,0045780,0045893,0046872,0048260,0048471,0055037,0060586,0070062,0070371,0071281,0072562,1990459,1990712,2000147 remove_due_to_license_issue P02787 29323384 704 DKTVRWCAVSEHEATKCQSFRDHMKSVIPSDGPSVACVKKASYLDCIRAIAANEADAVTLDAGLVYDAYLAPNNLKPVVAEFYGSKEDPQTFYYAVAVVKKDSGFQMNQLRGKKSCHTGLGRSAGWNIPIGLLYCDLPEPRKPLEKAVANFFSGSCAPCADGTDFPQLCQLCPGCGCSTLNQYFGYSGAFKCLKDGAGDVAFVKHSTIFENLANKADRDQYELLCLDNTRKPVDEYKDCHLAQVPSHTVVARSMGGKEDLIWELLNQAQEHFGKDKSKEFQLFSSPHGKDLLFKDSAHGFLKVPPRMDAKMYLGYEYVTAIRNLREGTCPCKPVKWCALSHHERLKCDEWSVNSVGKIECVSAETTEDCIAKIMNGEADAMSLDGGFVYIAGKCGLVPVLAENYNAGYFAIAVVKKSASDLTWDNLKGKKSCHTAVGRTAGWNIPMGLLYNKINHCRFDEFFSEGCAPGSKKDSSLCKLCMGSGLNLCEPNNKEGYYGYTGAFRCLVEKGDVAFVKHQTVPQNTGGKNPDPWAKNLNEKDYELLCLDGTRKPVEEYANCHLARAPNHAVVTRKDKEACVHKILRQQQHLFGSNSETKDLLFRDDTVCLAKLHDRNTYEKYLGEEYVKAVGNLRKCSTSSLLEACTFRRP 5y6k A 2.86 BS03 8R6 A 2 R602 Q603 R584 Q585 ? 0005515,0005576,0005615,0005768,0005769,0005770,0005788,0005886,0005905,0006826,0006879,0007015,0008198,0008199,0009617,0009925,0009986,0010008,0016020,0016324,0019731,0019899,0030139,0030316,0030669,0031410,0031647,0031982,0032436,0034756,0034774,0034986,0042327,0044325,0045178,0045780,0045893,0046872,0048260,0048471,0055037,0060586,0070062,0070371,0071281,0072562,1990459,1990712,2000147 remove_due_to_license_issue P02787 29323384 705 DKTVRWCAVSEHEATKCQSFRDHMKSVIPSDGPSVACVKKASYLDCIRAIAANEADAVTLDAGLVYDAYLAPNNLKPVVAEFYGSKEDPQTFYYAVAVVKKDSGFQMNQLRGKKSCHTGLGRSAGWNIPIGLLYCDLPEPRKPLEKAVANFFSGSCAPCADGTDFPQLCQLCPGCGCSTLNQYFGYSGAFKCLKDGAGDVAFVKHSTIFENLANKADRDQYELLCLDNTRKPVDEYKDCHLAQVPSHTVVARSMGGKEDLIWELLNQAQEHFGKDKSKEFQLFSSPHGKDLLFKDSAHGFLKVPPRMDAKMYLGYEYVTAIRNLREGTCPCKPVKWCALSHHERLKCDEWSVNSVGKIECVSAETTEDCIAKIMNGEADAMSLDGGFVYIAGKCGLVPVLAENYNAGYFAIAVVKKSASDLTWDNLKGKKSCHTAVGRTAGWNIPMGLLYNKINHCRFDEFFSEGCAPGSKKDSSLCKLCMGSGLNLCEPNNKEGYYGYTGAFRCLVEKGDVAFVKHQTVPQNTGGKNPDPWAKNLNEKDYELLCLDGTRKPVEEYANCHLARAPNHAVVTRKDKEACVHKILRQQQHLFGSNSETKDLLFRDDTVCLAKLHDRNTYEKYLGEEYVKAVGNLRKCSTSSLLEACTFRRP 5y7z A 2.804 BS01 IRE A 1 L46 K69 C126 K127 G128 E132 L180 C190 L23 K46 C103 K104 G105 E109 L157 C167 D173 K175 N178 D191 T223 D150 K152 N155 D168 T200 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O14976 30214852 401 SQSDFVGQTVELGELRLRVRRVLAEGGFAFVYEAQDVGSGREYALKRLLSNEEEKNRAIIQEVCFMKKLSGHPNIVQFCSAASIGKEESDTGQAEFLLLTELCKGQLVEFLKKMESRGPLSCDTVLKIFYQTCRAVQHMHRQKPPIIHRDLKVENLLLSNQGTIKLCDFGSATTISHYPDYSWSAQRRALVEEEITRNTTPMYRTPEIIDLYSNFPIGEKQDIWALGCILYLLCFRQHPFEDGAKLRIVNGKYSIPPHDTQYTVFHSLIRAMLQVNPEERLSIAEVVHQLQEIAAARNVNPKSPITELLEQN 5y80 A 2.5 BS01 IRE A 1 L46 K69 C126 G128 Q129 L180 L23 K46 C103 G105 Q106 L154 D173 K175 N178 D191 T223 D147 K149 N152 D165 T197 2.7.11.1 0004672,0005524,0006468 Kd=1.62nM remove_due_to_license_issue O14976 30214852 401 SQSDFVGQTVELGELRLRVRRVLAEGGFAFVYEAQDVGSGREYALKRLLSNEEEKNRAIIQEVCFMKKLSGHPNIVQFCSAASIGKEESDTGQAEFLLLTELCKGQLVEFLKKMGPLSCDTVLKIFYQTCRAVQHMHRQKPPIIHRDLKVENLLLSNQGTIKLCDFGSATTISHYPDYSWSAQRRALVEEEITRNTTPMYRTPEIIDLYSNFPIGEKQDIWALGCILYLLCFRQHPFEDGAKLRIVNGKYSIPPHDTQYTVFHSLIRAMLQVNPEERLSIAEVVHQLQEIAAARNVNPKSPITELL 5y80 A 2.5 BS02 IRE A 2 A81 R172 G193 S194 H200 V214 I218 N221 Q244 A58 R146 G167 S168 H174 V188 I192 N195 Q218 D173 K175 N178 D191 T223 D147 K149 N152 D165 T197 2.7.11.1 0004672,0005524,0006468 Kd=1.62nM remove_due_to_license_issue O14976 30214852 402 SQSDFVGQTVELGELRLRVRRVLAEGGFAFVYEAQDVGSGREYALKRLLSNEEEKNRAIIQEVCFMKKLSGHPNIVQFCSAASIGKEESDTGQAEFLLLTELCKGQLVEFLKKMGPLSCDTVLKIFYQTCRAVQHMHRQKPPIIHRDLKVENLLLSNQGTIKLCDFGSATTISHYPDYSWSAQRRALVEEEITRNTTPMYRTPEIIDLYSNFPIGEKQDIWALGCILYLLCFRQHPFEDGAKLRIVNGKYSIPPHDTQYTVFHSLIRAMLQVNPEERLSIAEVVHQLQEIAAARNVNPKSPITELL 5y86 A 1.9 BS01 HRM A 1 A236 K238 F288 L291 L342 I354 A99 K101 F151 L154 L205 I217 D335 K337 N340 D355 S372 D198 K200 N203 D218 S235 2.7.12.1 0000242,0000287,0004672,0004674,0004712,0004713,0005524,0005634,0005654,0005737,0005813,0005829,0005856,0006338,0006468,0010494,0016607,0030218,0035063,0035401,0035617,0043066,0043231,0043518,0046872,0051301,0080135,0106310,0140801,1902751,1903008,1903432 ic50=0.8uM remove_due_to_license_issue IC50=800nM O43781 29634919 601 VVPLTPEQALKQYKHHLTAYEKLEIINYPEIYFVGPNAKKRHGVIGGPNNGGYDDADGAYIHVPRDHLAYRYEVLKIIGKGSFGQVARVYDHKLRQYVALKMVRNEKRFHRQAAEEIRILEHLKKQDKTGSMNVIHMLESFTFRNHVCMAFELLSIDLYELIKKNKFQGFSVQLVRKFAQSILQSLDALHKNKIIHCDLKPENILLKHHGRSSTKVIDFGSSCFEYQKLYTYIQSRFYRAPEIILGSRYSTPIDIWSFGCILAELLTGQPLFPGEDEGDQLACMMELLGMPPPKLLEQSKRAKYFINSKGIPRYCSVTTQADGRVVLVGGRSRRGKKRGPPGSKDWGTALKGCDDYLFIEFLKRCLHWDPSARLTPAQALRHPWISKSVPRPLTT 5y8c A 1.42 BS01 8P9 A 1 W81 L94 N140 I146 M149 W49 L62 N108 I114 M117 ? ic50=0.16uM remove_due_to_license_issue O60885 29566488 203 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5y8w A 1.76 BS01 8PU A 1 W81 L94 I146 M149 W40 L53 I105 M108 ? ic50=0.23uM remove_due_to_license_issue O60885 29566488 201 GSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 5y8y A 1.87 BS01 8PX A 1 W81 L94 N140 I146 M149 W49 L62 N108 I114 M117 ? Kd=82nM remove_due_to_license_issue O60885 29566488 206 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 5y8z A 1.84 BS01 8Q3 A 1 W81 L92 L94 N140 I146 W40 L51 L53 N99 I105 ? ic50=0.62uM remove_due_to_license_issue O60885 29566488 201 GSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 5y93 A 1.62 BS01 8Q9 A 1 W81 L94 N140 I146 M149 W49 L62 N108 I114 M117 ? ic50=2.27uM remove_due_to_license_issue O60885 29566488 201 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 5y94 A 2.0 BS01 8QC A 1 W81 L94 N140 I146 W40 L53 N99 I105 ? Kd=164nM remove_due_to_license_issue O60885 29566488 201 GSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5y9l A 2.15 BS01 8R3 A 1 H57 H99 F151 A190 C191 N192 S195 S214 W215 G216 C220 H41 H80 F130 A171 C172 N173 S176 S191 W192 G193 C197 H57 D102 N192 G193 D194 S195 G196 H41 D83 N173 G174 D175 S176 G177 3.4.21.117 0001533,0002803,0004222,0004252,0005576,0005615,0006508,0008233,0008236,0008544,0016787,0022617,0030141,0051604,0097209 ic50=1.9uM remove_due_to_license_issue P49862 29102227 301 IIDGAPCARGSHPWQVALLSGNQLHCGGVLVNERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNSQARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVYKDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCKFTKWINDTMKKHR 5ya5 A 1.89 BS01 6TD A 1 A1108 Y1159 M1160 D1164 N1167 R1208 M1211 A1221 D1222 Y1230 A48 Y87 M88 D92 N95 R136 M139 A149 D150 Y158 D1204 A1206 R1208 N1209 D1222 D132 A134 R136 N137 D150 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.19uM remove_due_to_license_issue IC50=190nM P08581 29202410 1401 ALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKKIHCAVKSLNRSQFLTEGIIMKDFSHPNVLSLLGICSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFI 5yas A 2.2 BS01 FAC A 1 T11 I12 S80 W128 L148 L157 I209 T10 I11 S79 W127 L147 L156 I208 T11 S80 C81 D207 H235 K236 T10 S79 C80 D206 H234 K235 4.1.2.47 0009694,0009696,0016829,0047606,0052891,0052892,0080030,0080031,0080032 Ki=0.55mM remove_due_to_license_issue P52704 10548044 300 AFAHFVLIHTICHGAWIWHKLKPLLEALGHKVTALDLAASGVDPRQIEEIGSFDEYSEPLLTFLEALPPGEKVILVGESCGGLNIAIAADKYCEKIAAAVFHNSVLPDTEHCPSYVVDKLMEVFPDWKDTTYFTYTKDGKEITGLKLGFTLLRENLYTLCGPEEYELAKMLTRKGSLFQNILAKRPFFTKEGYGSIKKIYVWTDQDEIFLPEFQLWQIENYKPDKVYKVEGGDHKLQLTKTKEIAEILQEVADTYN 5ybi A 2.268 BS01 ANP A 1 G162 G164 K165 T166 F167 F339 Y412 G82 G84 K85 T86 F87 F258 Y319 K165 E188 R189 R350 K85 E108 R109 R269 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 remove_due_to_license_issue P0A1C1 30013545 505 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEDDDFDPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTISQDKIYNKISVVESFLKQDYRLGFTYEQTMELIGETIR 5yc8 A 2.5 BS01 3C0 A 1 D103 Y104 S107 N108 W155 A191 A194 W400 Y403 N404 Y426 C429 D88 Y89 S92 N93 W140 A176 A179 W326 Y329 N330 Y352 C355 ? 0004930,0005506,0005886,0007186,0009055,0016020,0016907,0020037,0022900,0042597,0046872 Kd=6.4nM remove_due_to_license_issue P08172,P0ABE7 30420692 501 SPYKTFEVVFIVLVAGSLSLVTIIGNILVMVSIKVNRHLQTVNNYFLFSLACADLIIGVFSMNLYTLYTVIGYWPLGPVVCDLWLALDYVVSNARVMNLLIISFDRYFCVTKPLTYPVKRTTKMAGMMIAAAWVLSFILWAPAILFWQFIVGVRTVEDGECYIQFFSNAAVTFGTAIAAFYLPVIIMTVLYWHISRASKADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLSREKKVTRTILAILLAFIITWAPYNVMVLINTFCAPCIPNTVWTIGYWLCYINSTINPACYALCNATFKKTFKHLLMCH 5ye7 A 2.312 BS01 8U0 A 1 L107 F110 L153 G154 H272 S273 Q352 F357 L371 L50 F53 L96 G97 H215 S216 Q295 F300 L314 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=3431nM remove_due_to_license_issue IC50=3431nM Q13093 29193967 501 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5ye8 A 1.851 BS01 8U3 A 1 L107 L153 G154 A155 L159 H272 S273 Q352 F357 L50 L94 G95 A96 L100 H213 S214 Q293 F298 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50~1mM remove_due_to_license_issue IC50=1000000nM Q13093 29193967 501 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQRLDTLWIPNKEYFWGLSKFLGTLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTT 5ye9 A 1.876 BS01 8U6 A 1 L107 F110 L153 G154 A155 H272 S273 Q352 A355 F357 L49 F52 L95 G96 A97 H214 S215 Q294 A297 F299 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=355nM remove_due_to_license_issue IC50=355nM Q13093 29193967 501 KIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINTTNQ 5yea A 1.805 BS01 8U9 A 1 L107 F110 L111 L121 L153 G154 A155 L159 H272 S273 Q352 A355 F357 L55 F58 L59 L69 L101 G102 A103 L107 H220 S221 Q300 A303 F305 3.1.1.47 0003847,0005515,0005543,0005576,0005615,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 ic50=5nM remove_due_to_license_issue IC50=5.0nM Q13093 29193967 503 QTKIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINT 5yej A 2.698 BS01 dna G 0 T25 M26 R27 G38 Y41 N46 K47 T24 M25 R26 G37 Y40 N45 K46 ? 0000976,0003677,0003700,0006355,0045892,0046677,0046872 remove_due_to_license_issue A0QX69 29852200 18 ~ 36 QLHKPDVVAAATKILDDHGIADLTMRRLARELDVTPGALYWHFANKQELLGAVADHILRTARTDTADLAWREQIHESCRALRDALLSHTDGAELVSASFASGQSVVITEIVEQLGRAARAAGVSDADVDAAARTVIYYVLGFTVDEQSRLQWRQFRFGLQLLVDGLAAH 5yej B 2.698 BS01 dna D 0 T25 M26 R27 Y41 N46 K47 T24 M25 R26 Y40 N45 K46 ? 0000976,0003677,0003700,0006355,0045892,0046677,0046872 remove_due_to_license_issue A0QX69 29852200 2 ~ 20 QLHKPDVVAAATKILDDHGIADLTMRRLARELDVTPGALYWHFANKQELLGAVADHILRTARTDTDLAWREQIHESCRALRDALLSHTDGAELVSASFASGQSVVITEIVEQLGRAARAAGVSDADVDAAARTVIYYVLGFTVDEQSRRQFRFGLQLLVDGLAAH 5yej B 2.698 BS02 dna F 0 L3 V35 T36 A39 W42 H43 L2 V34 T35 A38 W41 H42 ? 0000976,0003677,0003700,0006355,0045892,0046677,0046872 remove_due_to_license_issue A0QX69 29852200 18 ~ 36 QLHKPDVVAAATKILDDHGIADLTMRRLARELDVTPGALYWHFANKQELLGAVADHILRTARTDTDLAWREQIHESCRALRDALLSHTDGAELVSASFASGQSVVITEIVEQLGRAARAAGVSDADVDAAARTVIYYVLGFTVDEQSRRQFRFGLQLLVDGLAAH 5yej C 2.698 BS01 dna D 0 Q2 L3 V35 T36 W42 Q1 L2 V34 T35 W41 ? 0000976,0003677,0003700,0006355,0045892,0046677,0046872 remove_due_to_license_issue A0QX69 29852200 2 ~ 20 QLHKPDVVAAATKILDDHGIADLTMRRLARELDVTPGALYWHFANKQELLGAVADHILRTARTDTADLAWREQIHESCRALRDALLSHTDGAELVSASFASGQSVVITEIVEQLGRAARAAGVSDADVDAAARTVIYYVLGFTVDEQSRLQWRQFRFGLQLLVDGLAAH 5yej C 2.698 BS02 dna F 0 T25 M26 R27 Y41 N46 K47 T24 M25 R26 Y40 N45 K46 ? 0000976,0003677,0003700,0006355,0045892,0046677,0046872 remove_due_to_license_issue A0QX69 29852200 18 ~ 36 QLHKPDVVAAATKILDDHGIADLTMRRLARELDVTPGALYWHFANKQELLGAVADHILRTARTDTADLAWREQIHESCRALRDALLSHTDGAELVSASFASGQSVVITEIVEQLGRAARAAGVSDADVDAAARTVIYYVLGFTVDEQSRLQWRQFRFGLQLLVDGLAAH 5yf1 A 2.399 BS02 8V0 A 1 F313 D316 H347 Y386 Y396 Y398 F244 D247 H278 Y317 Y327 Y329 2.1.1.22 0008757 Kd=0.52mM remove_due_to_license_issue Q8N4J0 29463897 502 EEERLEREHFWKIINAFRYYGTSMHERVNRTERQFRSLPANQQKLLPQFLLHLDKIRKCIDHNQEILLTIVNDCIHKIMPASTFDMDKLKSTLKQFVRDWSETGKAERDACYQPIIKEILKNFPKERWDPSKVNILVPGAGLGRLAWEIAMLGYACQGNEWSFFMLFSSNFVLNRCSEINKYKLYPWIHQFSNNRRSADQIRPIFFPDVDPHSLPPGSNFSMTAGDFQEIYSECNTWDCIATCFFIDTAHNVIDYIDTIWKILKPGGIWINLGPLLYHFENLANELSIELSYEDIKNVVLQYGFKVEVEKESVLSTYTVNDLSMMKYYYECVLFVVRKPQ 5yf1 B 2.399 BS02 8V0 B 1 F313 D316 H347 Y386 Y398 F255 D258 H289 Y328 Y340 2.1.1.22 0008757 Kd=0.52mM remove_due_to_license_issue Q8N4J0 29463897 502 EEEERLEREHFWKIINAFRYYGTSMHERVNRTERQFRSLPANQQKLLPQFLLHLDKIRKCIDHNQEILLTIVNDCIHMFENKEYGEGKIMPASTFDMDKLKSTLKQFVRDWSETGKAERDACYQPIIKEILKNFPKERWDPSKVNILVPGAGLGRLAWEIAMLGYACQGNEWSFFMLFSSNFVLNRCSEINKYKLYPWIHQFSNNRRSADQIRPIFFPDVDPHSLPPGSNFSMTAGDFQEIYSECNTWDCIATCFFIDTAHNVIDYIDTIWKILKPGGIWINLGPLLYHFENLANELSIELSYEDIKNVVLQYGFKVEVEKESVLSTYTVNDLSMMKYYYECVLFVVRKPQ 5yfs A 2.3 BS01 RI2 A 1 M19 R22 G23 A24 R65 S137 K138 A139 D204 N214 K215 K240 F281 M17 R20 G21 A22 R63 S135 K136 A137 D202 N212 K213 K238 F279 5.3.1.29 0016853,0019323,0019509,0043917,0044237,0044249,0046523 Kd=13.8uM remove_due_to_license_issue O57947 29382938 401 AMIVKEVYETAEKIKSMEIRGAGRIARAAAQALMIQAEKSKAKEPEELWNELKVASKILYNTRPTAVSLPNALRYVMHRVKAAYLGGADLETLRFTAINSAKEFIYNSEKAIERIGEIGAKRIEDGDIIMTHSHSKAAISVMKKAFEQGKNIKVIVTETRPKWQGKITAKELASYGIPVIYIVDSAARHYMKMTDKVVMGADSITANGAVINKIGTSLIALTAKEHRVWVMIAAETYKFHPATMLGQLVEIEMRDPTEVIPEEELRTWPKNIEVWNPAFDVTPPEYIDVIITERGIIPPYAAIDILKEEFGWALKYKEPWED 5yft A 2.21 BS01 RI2 A 1 R22 G23 A24 G25 R65 S137 K138 A139 N204 N214 K215 K240 F281 R20 G21 A22 G23 R63 S135 K136 A137 N202 N212 K213 K238 F279 5.3.1.29 0016853,0019323,0019509,0043917,0044237,0044249,0046523 Kd=10uM remove_due_to_license_issue O57947 29382938 401 AMIVKEVYETAEKIKSMEIRGAGRIARAAAQALMIQAEKSKAKEPEELWNELKVASKILYNTRPTAVSLPNALRYVMHRVKAAYLGGADLETLRFTAINSAKEFIYNSEKAIERIGEIGAKRIEDGDIIMTHCHSKAAISVMKKAFEQGKNIKVIVTETRPKWQGKITAKELASYGIPVIYIVDSAARHYMKMTDKVVMGANSITANGAVINKIGTSLIALTAKEHRVWVMIAAETYKFHPATMLGQLVEIEMRDPTEVIPEEELRTWPKNIEVWNPAFDVTPPEYIDVIITERGIIPPYAAIDILKEEFGWALKYKEPWED 5yfz A 2.16 BS02 8UO A 1 L124 G128 T183 K355 N356 R371 L124 G128 T183 K355 N356 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yfz A 2.16 BS03 8UO B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yfz B 2.16 BS01 8UO A 1 E56 Y63 E56 Y63 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yfz B 2.16 BS03 8UO B 1 L124 G128 L130 T183 K355 N356 T357 C364 R371 L124 G128 L130 T183 K355 N356 T357 C364 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg2 A 2.2 BS02 N05 A 1 L124 G128 T183 K355 N356 T357 R371 L124 G128 T183 K355 N356 T357 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg2 A 2.2 BS03 N05 B 1 E56 Y63 Y64 P267 E56 Y63 Y64 P267 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg2 B 2.2 BS02 N05 A 1 E56 Y63 Y64 P267 E56 Y63 Y64 P267 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg2 B 2.2 BS04 N05 B 1 L124 G128 T183 K355 N356 T357 C364 R371 L124 G128 T183 K355 N356 T357 C364 R371 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg3 A 2.4 BS02 8UC A 1 L124 G128 H129 L130 T183 K355 L124 G128 H129 L130 T183 K355 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg3 A 2.4 BS04 8UC B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg3 B 2.4 BS02 8UC A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg3 B 2.4 BS04 8UC B 1 L124 G128 H129 L130 T183 K355 C364 L124 G128 H129 L130 T183 K355 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg4 A 2.3 BS02 8UF A 1 L124 G128 H129 L130 T183 K355 C364 L124 G128 H129 L130 T183 K355 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg4 A 2.3 BS04 8UF B 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg4 B 2.3 BS02 8UF A 1 E56 Y63 Y64 E56 Y63 Y64 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5yg4 B 2.3 BS04 8UF B 1 L124 G128 H129 L130 T183 K355 N356 C364 L124 G128 H129 L130 T183 K355 N356 C364 Y54 E56 D208 T234 K237 R243 Y54 E56 D208 T234 K237 R243 2.1.2.1 0004372,0005737,0005739,0006730,0008168,0019264,0030170,0032259,0035999,0046653 remove_due_to_license_issue A0A1G4H5I1 29655285 502 MFNNEPLEQIDKELHDILADEEKRQRETINLIASENLTNGAVRECLGNRVSNKYSEGYPKKRYYGGNDFIDKIEELCQKRALEAFNVSDEEWGVNVQPLSGSAANVQALYALVGVKGKIMGMHLCSGGHLTHGFFDEKKKVSITSDMFESKLYKCNSQGYVDLDAVREMALSFKPKVIICGYTSYPRDIDYQQFRQICDEVNAYLFADISHISSFVACNILNNPFLHADVVTTTTHKILRGPRSALIFFNKKRNPGIEQKINSAVFPSFQGGPHNNKIAAVACQLKEVHSPAFKEYTQQVLLNSKALAKALISKQIDLVTNGTDNHLIVVDLRKFSITGSKLQETCNAINVSLNKNTIPSDVDCVSPSGVRIGTPAMTTRGAKEKDMEFIADVLARAIKITVDLQEQYGKKLVDFKKGLPGNAQLQQLKQEVVTWAGALPFP 5ygi A 2.177 BS03 T93 A 1 F98 F99 D103 M106 R112 Q171 K200 D243 K257 F87 F88 D92 M95 R101 Q160 K189 D232 K246 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K46 F87 D92 D96 R101 D163 K189 F228 D232 D233 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue P14324 30270039 506 DVYAQEKQDFVQHFSQIVRVLTEHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIY 5yh8 A 2.12 BS01 8UX A 1 Y27 W103 R140 D224 R225 R393 W406 Y410 N423 Y497 Y30 W106 R143 D227 R228 R396 W409 Y413 N426 Y500 ? 0005886,0006824,0006829,0015675,0015833,0016151,0020037,0030288,0042597,0043190,0055085,1904680 Kd=167.8nM remove_due_to_license_issue Q2FVE7 29581261 602 PHMGLEEKKENKQLTYTTVKDIGDMNPHVYGGSMSAESMIYEPLVRNTKDGIKPLLAKKWDVSEDGKTYTFHLRDDVKFHDGTPFDADAVKKNIDAVQENKKLHSWLKISTLIDNVKVKDKYTVELNLKEAYQPALAELAMPRPYVFVSPKDFKNGTTKDGVKKFDGTGPFKLGEHKKDESADFNKNDQYWGEKSKLNKVQAKVMPAGETAFLSMKKGETNFAFTDDRGTDSLDKDSLKQLKDTGDYQVKRSQPMNTKMLVVNSGKKDNAVSDKTVRQAIGHMVNRDKIAKEILDGQEKPATQLFAKNVTDINFDMPTRKYDLKKAESLLDEAGWKKGKDSDVRQKDGKNLEMAMYYDKGSSSQKEQAEYLQAEFKKMGIKLNINGETSDKIAERRTSGDYDLMFNQTWGLLYDPQSTIAAFKAKNGYESATSGIENKDKIYNSIDDAFKIQNGKERSDAYKNILKQIDDEGIFIPISHGSMTVVAPKDLEKVSFTQSQYELPFNEMQYK 5yhe A 2.465 BS01 8UX A 1 Y27 W103 R140 D224 R225 R393 W406 N423 Y497 Y28 W104 R141 D225 R226 R392 W405 N422 Y496 ? 0005886,0006824,0006829,0015675,0015833,0016151,0020037,0030288,0042597,0043190,0055085,1904680 Kd=203.3nM remove_due_to_license_issue Q2FVE7 29581261 604 MGLEEKKENKQLTYTTVKDIGDMNPHVYGGSMSAESMIYEPLVRNTKDGIKPLLAKKWDVSEDGKTYTFHLRDDVKFHDGTPFDADAVKKNIDAVQENKKLHSWLKISTLIDNVKVKDKYTVELNLKEAYQPALAELAMPRPYVFVSPKDFKNGTTKDGVKKFDGTGPFKLGEHKKDESADFNKNDQYWGEKSKLNKVQAKVMPAGETAFLSMKKGETNFAFTDDRGTDSLDKDSLKQLKDTGDYQVKRSQPMNTKMLVVNSGKKDNAVSDKTVRQAIGHMVNRDKIAKEILDGQEKPATQLFAKNVTDINFDMPTRKYDLKKAESLLDEAGWKKGSDVRQKDGKNLEMAMYYDKGSSSQKEQAEYLQAEFKKMGIKLNINGETSDKIAERRTSGDYDLMFNQTWGLLYDPQSTIAAFKAKNGYESATSGIENKDKIYNSIDDAFKIQNGKERSDAYKNILKQIDDEGIFIPISHGSMTVVAPKDLEKVSFTQSQYELPFNEMQYK 5yhg A 2.03 BS01 8UX A 1 Y27 W103 R140 D224 R225 R393 W406 Y410 N423 Y497 Y27 W103 R140 D224 R225 R393 W406 Y410 N423 Y497 ? 0005886,0006824,0006829,0015675,0015833,0016151,0020037,0030288,0042597,0043190,0055085,1904680 Kd=952.3nM remove_due_to_license_issue Q2FVE7 29581261 608 GLEEKKENKQLTYTTVKDIGDMNPHVYGGSMSAESMIYEPLVRNTKDGIKPLLAKKWDVSEDGKTYTFHLRDDVKFHDGTPFDADAVKKNIDAVQENKKLHSWLKISTLIDNVKVKDKYTVELNLKEAYQPALAELAMPRPYVFVSPKDFKNGTTKDGVKKFDGTGPFKLGEHKKDESADFNKNDQYWGEKSKLNKVQAKVMPAGETAFLSMKKGETNFAFTDDRGTDSLDKDSLKQLKDTGDYQVKRSQPMNTKMLVVNSGKKDNAVSDKTVRQAIGHMVNRDKIAKEILDGQEKPATQLFAKNVTDINFDMPTRKYDLKKAESLLDEAGWKKGKDSDVRQKDGKNLEMAMYYDKGSSSQKEQAEYLQAEFKKMGIKLNINGETSDKIAERRTSGDYDLMFNQTWGLLYDPQSTIAAFKAKNGYESATSGIENKDKIYNSIDDAFKIQNGKERSDAYKNILKQIDDEGIFIPISHGSMTVVAPKDLEKVSFTQSQYELPFNEMQYK 5yhl A 4.2 BS01 8VL A 1 T76 Y80 W169 L312 I315 R316 S319 T59 Y63 W152 L246 I249 R250 S253 ? 0004930,0004955,0004957,0007186,0016020 remove_due_to_license_issue P35408 30510193 401 NSPVTIPAVMFIFGVVGNLVAIVVLCKSRKEQKETTFYTLVCGLLVTDLLGTLLVSPVTIATYMKGQWPGGQPLCEYSTFILLFFSLSRLSIICAMSVERYLAINHAYFYSHYVDKRLAGLTLFAVYASNVLFCALPNMGLGSSRLQYPDTWCFIDWTTQVTAHAAYSYMYAGFSSFLILATVLCNVLVCGALLRMHAGAEIQMVILLIATSLVVLICSIPLVVRVFVNQLYQPSLEREVSKNPDLQAIRIASVNPILDPWIYILLRKTVLSKAIEKIKC 5yi2 A 2.6 BS01 dna C 0 N21 H23 T37 S64 A67 K70 N21 H23 T37 S64 A67 K70 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 A 2.6 BS02 dna D 0 N54 A55 T69 K73 N54 A55 T69 K73 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 A 2.6 BS03 dna H 0 T53 V92 T53 V92 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 B 2.6 BS01 dna C 0 N54 A55 P65 A66 T69 N53 A54 P64 A65 T68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 B 2.6 BS02 dna D 0 T37 T39 I63 S64 A67 K70 T36 T38 I62 S63 A66 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 E 2.6 BS01 dna G 0 T37 S64 A67 K70 T37 S64 A67 K70 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 E 2.6 BS02 dna D 0 T53 A55 K56 V92 T53 A55 K56 V92 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 E 2.6 BS03 dna H 0 N54 A55 P65 T69 K73 N54 A55 P65 T69 K73 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 F 2.6 BS01 dna G 0 N54 A55 P65 A66 T69 K73 N53 A54 P64 A65 T68 K72 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 F 2.6 BS02 dna H 0 H23 T37 T39 I63 S64 K70 H22 T36 T38 I62 S63 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 I 2.6 BS01 dna K 0 H23 T37 T39 S64 K70 H22 T36 T38 S63 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 I 2.6 BS02 dna L 0 N54 A55 P65 A66 T69 N53 A54 P64 A65 T68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 J 2.6 BS01 dna K 0 N54 A55 T69 N53 A54 T68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 J 2.6 BS02 dna O 0 T53 V92 T52 V91 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 J 2.6 BS03 dna P 0 E90 V92 E89 V91 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 J 2.6 BS04 dna L 0 T37 T39 S64 A67 K70 T36 T38 S63 A66 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 M 2.6 BS01 dna O 0 N21 H23 T37 T39 I63 S64 A66 A67 N21 H23 T37 T39 I63 S64 A66 A67 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 M 2.6 BS02 dna P 0 N54 A55 P65 A66 T69 N54 A55 P65 A66 T69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 N 2.6 BS01 dna O 0 N54 A55 P65 A66 T69 K73 N53 A54 P64 A65 T68 K72 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi2 N 2.6 BS02 dna P 0 T37 T39 S64 A66 A67 K70 T36 T38 S63 A65 A66 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKCESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 A 2.9 BS01 dna C 0 T37 S64 K70 T37 S64 K70 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 A 2.9 BS02 dna H 0 T53 V92 T53 V92 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 A 2.9 BS03 dna D 0 N54 A55 P65 A66 T69 N54 A55 P65 A66 T69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 GMSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 B 2.9 BS01 dna C 0 N54 A55 T69 N52 A53 T67 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 B 2.9 BS02 dna D 0 H23 T37 T39 S64 A67 K70 H21 T35 T37 S62 A65 K68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 E 2.9 BS01 dna G 0 T37 T39 S64 A67 T36 T38 S63 A66 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 E 2.9 BS02 dna H 0 N54 A55 P65 A66 T69 N53 A54 P64 A65 T68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 E 2.9 BS03 dna D 0 T53 V92 T52 V91 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 F 2.9 BS01 dna G 0 N54 A55 P65 A66 T69 N53 A54 P64 A65 T68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 F 2.9 BS02 dna H 0 T37 T39 S64 A67 K70 T36 T38 S63 A66 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 I 2.9 BS01 dna K 0 T37 T39 S64 A67 K70 T36 T38 S63 A66 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 I 2.9 BS02 dna P 0 T53 V92 T52 V91 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 I 2.9 BS03 dna L 0 A55 P65 A66 T69 R85 A54 P64 A65 T68 R84 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 J 2.9 BS01 dna K 0 N54 A55 P65 A66 T69 N53 A54 P64 A65 T68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 J 2.9 BS02 dna L 0 H23 T37 T39 I63 S64 A67 K70 H22 T36 T38 I62 S63 A66 K69 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 MSLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 M 2.9 BS01 dna O 0 T37 T39 I63 S64 A67 K70 T35 T37 I61 S62 A65 K68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 M 2.9 BS02 dna P 0 N54 A55 P65 A66 T69 N52 A53 P63 A64 T67 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 M 2.9 BS03 dna L 0 T53 V92 T51 V90 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 N 2.9 BS01 dna O 0 N54 A55 T69 N52 A53 T67 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yi3 N 2.9 BS02 dna P 0 H23 T37 T39 S64 A67 K70 H21 T35 T37 S62 A65 K68 ? 0003677,0003700,0006355,0008270,0046872 remove_due_to_license_issue Q9CDU5 29229866 1 ~ 16 SLANQIDQFLGTIMQFAENKHEILLGKSESDVKLTSTQEHILMLLAEQISTNAKIAEKLKISPAAVTKALKKLQEQELIKSSRATNDERVVLWSLTEKAVPVAKEHATHHEKTLSTYQELGNKFTDEEQEVISKFLSALTEEFQ 5yia A 2.0 BS01 8V9 A 1 D36 G38 N78 Y79 V80 S81 L133 D216 G218 T219 S220 F296 I302 D33 G35 N75 Y76 V77 S78 L130 D213 G215 T216 S217 F293 I299 3.4.23.39 0004190,0006508 Ki=3nM remove_due_to_license_issue Q8I6V3 29943906 401 SNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNQSVGIALAKKNL 5yib A 2.15 BS01 8VC A 1 D36 G38 Y79 V80 S81 S134 D216 G218 T219 S220 I292 F296 I302 D33 G35 Y76 V77 S78 S131 D213 G215 T216 S217 I289 F293 I299 3.4.23.39 0004190,0006508 Ki=3.3nM remove_due_to_license_issue Q8I6V3 29943906 401 SNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNQSVGIALAKKNL 5yic A 1.9 BS01 8VO A 1 D36 G38 Y79 V80 S81 D216 G218 T219 S220 L294 F296 I302 D33 G35 Y76 V77 S78 D213 G215 T216 S217 L291 F293 I299 3.4.23.39 0004190,0006508 Ki=1.3nM remove_due_to_license_issue Q8I6V3 29943906 401 SNDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNQSVGIALAKKNL 5yid A 2.1 BS01 K95 A 1 D36 G38 Y79 V80 S81 I125 G218 T219 S220 L294 F296 I302 D32 G34 Y75 V76 S77 I121 G214 T215 S216 L290 F292 I298 3.4.23.39 0004190,0006508 Ki=4nM remove_due_to_license_issue Q8I6V3 29943906 401 NDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNQSVGIALAKKNL 5yie A 2.1 BS01 8VF A 1 D36 G38 Y79 V80 S81 I125 L133 I135 D216 G218 T219 S220 L294 F296 I302 D32 G34 Y75 V76 S77 I121 L129 I131 D212 G214 T215 S216 L290 F292 I298 3.4.23.39 0004190,0006508 Ki=5.6nM remove_due_to_license_issue Q8I6V3 29943906 403 NDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNQSVGIALAKKNL 5yij A 3.18 BS01 NAI A 1 Q713 F719 N723 Q727 R729 R766 G767 N769 S820 T822 W832 E862 Q480 F486 N490 Q494 R496 R533 G534 N536 S587 T589 W599 E629 ? 0106274 remove_due_to_license_issue Q6RCR0 29795342 1201 GFSLYTDDTVKAAAQYAYDNYLGKPYTGSVESAPANFGGRMVYRQHHGLSHTLRTMAYAELIVEEARKAKLRGETLGKFKDGRTIADVTPQELKKIMIAQAFFVAGRDDEASDAKNYQKYHEQSRDAFLKYVKDNESTLIPDVFKDQEDVNFYARVIEDKSHDWESTPAHVLINQGHMVDLVRVKQPPESFLQRYFSSMQRWIGSQATEAVFGIQRQFFHATYEVVAGFDSDNKEPHLVVSGLGRYVIGEDGQPIREAPKKGQKEGDLKVFPQTYKNERLMRVDEFLKLPEIQNTFPGSGKHLQGGMPGMNEMDYWNRLNSLNRARCENDVDFCLKQLQTAHDKAKIEPIKQAFQSSKGKERRQPNVDEIAAARIIQQILANPDCIHDDHVLINGQKLEQQFFRDLLAKCEMAVVGSLLNDTDIGNIDTLMRHEKDTEFHSTNPEAVPVKIGEYWINDQRINNSSGNITQKKHDLIFLMQNDAWYFSRVNAIAQNRDKGSTFKEVLITTLMTPLTSKALVDTSQAKPPTRLFRGLNLSEEFTKGLIDQANAMIANTTERLFTDHSPEAFKQIKLNDLSKMSGRTNASTTTEIKLVKETWDSNVIFEMLDPDGLLHSKQVGRHGEGTESEFSVYLPEDVALVPVKVTLDGKTQKGENRYVFTFVAVKSPDFTPRHESGYAVEPFLRMQAAKLAEVKSSIEKAQRAPDLETIFNLQNEVEAVQYSHLSTGYKNFLKNTVGPVLENSLSGLMESDTDTLSKALAAFPSDTQWSAFNFEEARQAKRQMDAIKQMVGNKVVLDALTQCQDALEKQNIAGALDALKKIPSEKEMGTIRRELREQIQSARQELESLQRAVVTPVVTDEKKVRERYDALIENTSKKITELETGKLPNLDAVKKGISNLSNLKQEVTVLRNEKIRMHVGTDKVDFSDVEKLEQQIQVIDTKLADAYLLEVTKQISALE 5yj3 C 2.845 BS01 dna A 0 R609 R614 R61 R66 ? remove_due_to_license_issue P10074 29134956 1 ~ 18 PHFCQICGKTFKAVEQLRVHVRRHKGVRKFECTECGYKFTRQAHLRRHMEIHDRVENYNPRQRKLRNLII 5yj3 C 2.845 BS02 dna B 0 R576 Y585 H592 R595 H596 I599 Y606 R611 L613 R614 R28 Y37 H44 R47 H48 I51 Y58 R63 L65 R66 ? remove_due_to_license_issue P10074 29134956 1 ~ 18 PHFCQICGKTFKAVEQLRVHVRRHKGVRKFECTECGYKFTRQAHLRRHMEIHDRVENYNPRQRKLRNLII 5yj3 D 2.845 BS01 dna A 0 R594 R611 K612 R614 R46 R63 K64 R66 ? remove_due_to_license_issue P10074 29134956 1 ~ 18 PHFCQICGKTFKAVEQLRVHVRRHKGVRKFECTECGYKFTRQAHLRRHMEIHDRVENYNPRQRKLR 5yj3 D 2.845 BS02 dna B 0 R576 Y585 F587 R589 H592 R595 H596 I599 R611 L613 R614 R28 Y37 F39 R41 H44 R47 H48 I51 R63 L65 R66 ? remove_due_to_license_issue P10074 29134956 1 ~ 18 PHFCQICGKTFKAVEQLRVHVRRHKGVRKFECTECGYKFTRQAHLRRHMEIHDRVENYNPRQRKLR 5yj8 A 1.762 BS01 8W9 A 1 Y566 Y573 F591 Y594 N596 Y18 Y25 F43 Y46 N48 ? Kd=0.104mM remove_due_to_license_issue Q9H7E2 29645362 701 HHHHHMMWKPGDECFALYWEDNKFYRAEVEALHSSGMTAVVKFIDYGNYEEVLLSNIKPI 5yjb A 2.96 BS02 8WC A 1 M332 F538 D555 L659 K661 W695 A809 M161 F367 D384 L488 K490 W524 A638 T335 D553 K661 T164 D382 K490 1.14.99.66 0005634,0006355,0016491,0050660 remove_due_to_license_issue Ki=29nM O60341 29949906 902 SGVEGAAFQSRLPHDRMTSQEAACFPDIISGPQQTQKVFLFIRNRTLQLWLDNPKIQLTFEATLQQLEAPYNSDTVLVHRVHSYLERHGLINFGIYKRIKPLPTKKTGKVIIIGSGVSGLAAARQLQSFGMDVTLLEARDRVGGRVATFRKGNYVADLGAMVVTGLGGNPMAVVSKQVNMELAKIKQKCPLYEANGQAVPKEKDEMVEQEFNRLLEATSYLSHQLDFNVLNNKPVSLGQALEVVIQLQEKHVKDEQIEHWKKIVKTQEELKELLNKMVNLKEKIKELHQQYKEASEVKPPRDITAEFLVKSKHRDLTALCKEYDELAETQGKLEEKLQELEANPPSDVYLSSRDRQILDWHFANLEFANATPLSTLSLKHWDQDDDFEFTGSHLTVRNGYSCVPVALAEGLDIKLNTAVRQVRYTASGCEVIAVNTRSTSQTFIYKCDAVLCTLPLGVLKQQPPAVQFVPPLPEWKTSAVQRMGFGNLNKVVLCFDRVFWDPSVNLFGHVGSTTASRGELFLFWNLYKAPILLALVAGEAAGIMENISDDVIVGRCLAILKGIFGSSAVPQPKETVVSRWRADPWARGSYSYVAAGSSGNDYDLMAQPITPGPSIPGAPQPIPRLFFAGEHTIRNYPATVHGALLSGLREAGRIADQFLGA 5yjf A 2.49 BS02 8WO A 1 Y20 Y24 L164 A198 S201 Y204 S213 Y242 Y16 Y20 L160 A194 S197 Y200 S209 Y238 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0030760,0031100,0032259,0034356,0045722,0090312 ic50=1.8uM remove_due_to_license_issue P40261 29483571 302 FTSKDTYLSHFNPRDYLEKYYKFGSRHSAESQILKHLLKNLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIVVTDYSDQNLQELEKWLKAAPAAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPPADCVLSTLCLDAACPDLPTYCRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVARKL 5yji A 1.99 BS02 8WO A 1 Y20 Y24 L164 A198 S201 Y204 S213 Y242 Y16 Y20 L160 A194 S197 Y200 S209 Y238 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0031100,0032259,0045722,0090312 ic50=5uM remove_due_to_license_issue O55239 29483571 302 FTSKDTYLSHFNPRDYLEKYYSFGSRHCAENEILRHLLKNLFKIFCLGAVKGELLIDIGSGPTIYQLLSACESFTEIIVSDYTDQNLWELQKWLKKEPGAFDWSPVVTYVCDLEGNRMKGPEKEEKLRRAIKQVLKCDVTQSQPLGGVSLPPADCLLSTLCLDAACPDLPAYRTALRNLGSLLKPGGFLVMVDALKSSYYMIGEQKFSSLPLGWETVRDAVEEAGYTIEQFEVISQNYSSTTSNNEGLFSLVGRKP 5yjk A 2.4 BS01 8VX A 1 H57 H99 F151 A190 C191 N192 G193 S195 S214 W215 G216 T217 F218 C220 H41 H80 F130 A171 C172 N173 G174 S176 S191 W192 G193 T194 F195 C197 H57 D102 N192 G193 D194 S195 G196 H41 D83 N173 G174 D175 S176 G177 3.4.21.117 0001533,0002803,0004222,0004252,0005576,0005615,0006508,0008233,0008236,0008544,0016787,0022617,0030141,0051604,0097209 ic50=0.82uM remove_due_to_license_issue IC50=820nM P49862 29102227 301 IIDGAPCARGSHPWQVALLSGNQLHCGGVLVNERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNSQARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVYKDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCKFTKWINDTMKKHR 5yjm A 1.9 BS02 8W3 A 1 F41 C42 H57 Y94 L99 D102 R143 A190 F191 K192 S195 S214 G216 R217 F29 C30 H45 Y81 L86 D89 R122 A169 F170 K171 S174 S189 G191 R192 H57 D102 K192 G193 D194 S195 H45 D89 K171 G172 D173 S174 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 Kd=0.000000064M remove_due_to_license_issue Kd=2.1nM, IC50=8.9nM P23946 29191554 304 IIGGTESKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGVAQGIVSYGRSDAKPPAVFTRISHYRPWINQILQAN 5yjp A 1.8 BS02 8W6 A 1 F41 C42 H57 R143 A190 F191 K192 S195 S214 G216 R217 F29 C30 H45 R124 A171 F172 K173 S176 S191 G193 R194 H57 D102 K192 G193 D194 S195 H45 D89 K173 G174 D175 S176 3.4.21.39 0002003,0004175,0004252,0005576,0005615,0005829,0006508,0006518,0008236,0016485,0016787,0022617,0030141,0030163,0030901,0034769,0036464,0042277,0045766,0050727,0051604,0062023,0071333,0140447 ic50=0.24uM remove_due_to_license_issue IC50=240nM P23946 29191554 304 IIGGTESKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGVAQGIVSYGRSDAKPPAVFTRISHYRPWINQILQAN 5yjy A 3.4 BS06 8WF A 1 Q394 H397 M485 Q349 H352 M435 1.6.5.9 0003954,0005739,0005743,0005759,0006116,0006120,0008137,0016491,0042802,0043065,0050136,1902600 remove_due_to_license_issue P32340 29402945 606 GVENSGAGPTSFKTMKVIDPQHSDKPNVLILGSGWGAISFLKHIDTKKYNVSIISPRSYFLFTPLLPSAPVGTVDEKSIIEPIVNFALKKKGNVTYYEAEATSINPDRNTVTIKSLSAPAEIKYDYLISAVGAEPNTFGIPGVTDYGHFLKEIPNSLEIRRTFAANLEKANLLPKGDPERRRLLSIVVVGGGPTGVEAAGELQDYVHQDLRKFLPALAEEVQIHLVEALPIVLNMFEKKLSSYAQSHLENTSIKVHLRTAVAKVEEKQLLAKTKHEDGKITEETIPYGTLIWATGNKARPVITDLFKKIPEQNSSKRGLAVNDFLQVKGSNNIFAIGDNAFAGLPPTAQVAHQEAEYLAKNFDKMAQIPNFQKNDKIDLLFEENNFKPFKYNDLGALAYLGSERAIATIRSGKRTFYTGGGLMTFYLWRILYLSMILSARSRLKVFFDWIKLAFFKRDFFKGL 5yki A 2.25 BS01 rna C 0 R37 Q40 N72 Y73 R109 Q112 N144 Y145 K177 N181 E184 Y221 N223 Y224 N259 Y260 Q263 K292 N296 E299 Y336 N338 Y339 H375 R37 Q40 N72 Y73 R109 Q112 N144 Y145 K177 N181 E184 Y221 N223 Y224 N259 Y260 Q263 K292 N296 E299 Y336 N338 Y339 H375 ? 0003723 remove_due_to_license_issue Q14671 29490074 1 ~ 9 GRSRLLEDFRNNRYPNLQLREIAGHIMEFSQDQHGSRFIQLKLERATPAERQLVFNEILQAAYQLMVDVFGNYVIQKFFEFGSLEQKLALAERIRGHVLSLALQMYGCRVIQKALEFIPSDQQNEMVRELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHELHQHTEQLVQDQYGNYVIQHVLEHGRPEDKSKIVAEIRGNVLVLSQHKFASNVVEKCVTHASRTERAVLIDEVCTMNDGPHSALYTMMKDQYANYVVQKMIDVAEPGQRKIVMHKIRPHIATLRKYTYGKHILAKLEKY 5ykp A 1.68 BS04 OVA A 1 P192 Y195 H212 Y300 C301 E336 P104 Y107 H124 Y212 C213 E248 3.4.11.18 0006508,0070006 remove_due_to_license_issue P53582 30837307 405 PYRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 5yl2 A 2.09 BS03 8WU B 1 T179 A180 V181 T179 A180 V181 3.6.5.- 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0015630,0016787,0046872 remove_due_to_license_issue Q2XVP4 29691282 504 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGV 5yl2 B 2.09 BS02 8WU B 1 V236 C239 L246 A248 D249 L253 N256 M257 N348 K350 A352 V236 C239 L246 A248 D249 L253 N256 M257 N348 K350 A352 ? 0000226,0000278,0003924,0005200,0005515,0005525,0005737,0005856,0005874,0007017,0046872 Kd=31.69uM remove_due_to_license_issue P02554 29691282 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5ylj B 2.7 BS02 8X0 B 1 V236 C239 L246 A248 L253 N256 N348 K350 A352 V236 C239 L246 A248 L253 N256 N348 K350 A352 ? 0000226,0000278,0003924,0005200,0005515,0005525,0005737,0005856,0005874,0007017,0046872 remove_due_to_license_issue P02554 29691282 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5yls A 3.0 BS03 Y50 B 1 A180 V181 A180 V181 3.6.5.- 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0015630,0016787,0046872 remove_due_to_license_issue Q2XVP4 29691282 504 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGV 5yls B 3.0 BS02 Y50 B 1 V236 C239 A248 D249 L253 N256 M257 T312 N348 K350 A352 V236 C239 A248 D249 L253 N256 M257 T312 N348 K350 A352 ? 0000226,0000278,0003924,0005200,0005515,0005525,0005737,0005856,0005874,0007017,0046872 remove_due_to_license_issue P02554 29691282 504 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 5ylt A 1.69 BS02 C7N A 1 N263 G264 T266 Y305 Y335 G336 D338 P341 Y353 N149 G150 T152 Y191 Y221 G222 D224 P227 Y236 Y245 H293 H297 Y305 Y335 Y131 H179 H183 Y191 Y221 2.1.1.364 0005694,0006355,0016279,0140945 ic50=0.41uM remove_due_to_license_issue Q8WTS6 29882380 402 RHGVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDERTALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCISTNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITHQEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPNCIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHSPPGKSAPEWYQVELKAFQATQ 5ylu A 2.79989 BS01 HKT A 1 L141 A335 A339 V341 E343 L796 Y799 C813 I816 L94 A288 A292 V294 E296 L749 Y752 C766 I769 7.2.2.19 0000166,0000287,0005215,0005391,0005515,0005524,0005886,0005889,0006813,0006883,0008556,0008900,0010248,0016020,0016324,0016887,0030007,0030955,0036376,0046872,0071805,1902600,1990573 remove_due_to_license_issue IC50=22.0nM P19156 29618813 1101 MEINDHQLSVAELEQKYQTSATKGLSASLAAELLLRDGPNALRPPRGTPEYVKFARQLAGGLQCLMWVAAAICLIAFAIQASEGDLTTDDNLYLALALIAVVVVTGCFGYYQEFKSTNIIASFKNLVPQQATVIRDGDKFQINADQLVVGDLVEMKGGDRVPADIRILQAQGCKVDNSSLTGESEPQTRSPECTHESPLETRNIAFFSTMCLEGTAQGLVVNTGDRTIIGRIASLASGVENEKTPIAIEIEHFVDIIAGLAILFGATFFIVAMCIGYTFLRAMVFFMAIVVAYVPEGLLATVTVCLSLTAKRLASKNCVVKNLEAVETLGSTSVICSDKTGTLTQNRMTVSHLWFDNHIHSADTTEDQSGQTFDQSSETWRALCRVLTLCNRAAFKSGQDAVPVPKRIVIGDASETALLKFSELTLGNAMGYRERFPKVCEIPFNSTNKFQLSIHTLEDPRDPRHVLVMKGAPERVLERCSSILIKGQELPLDEQWREAFQTAYLSLGGLGERVLGFCQLYLSEKDYPPGYAFDVEAMNFPTSGLCFAGLVSMIDPPRATVPDAVLKCRTAGIRVIMVTGDHPITAKAIAASVGIISEGSETVEDIAARLRVPVDQVNRKDARACVINGMQLKDMDPSELVEALRTHPEMVFARTSPQQKLVIVESCQRLGAIVAVTGDGVNDSPALKKADIGVAMGIAGSDAAKNAADMILLDDNFASIVTGVEQGRLIFDNLKKSIAYTLTKNIPELTPYLIYITVSVPLPLGCITILFIELCTDIFPSVSLAYEKAESDIMHLRPRNPKRDRLVNEPLAAYSYFQIGAIQSFAGFTDYFTAMAQEGWFPLLCVGLRPQWENHHLQDLQDSYGQEWTFGQRLYQQYTCYTVFFISIEMCQIADVLIRKTRRLSAFQQGFFRNRILVIAIVFQVCIGCFLCYCPGMPNIFNFMPIRFQWWLVPMPFSLLIFVYDEIRKLGVRCCPG 5ylv A 2.79978 BS01 8WX A 1 A123 N138 M334 A335 E795 Y799 L811 C813 A77 N92 M288 A289 E749 Y753 L765 C767 7.2.2.19 0000166,0000287,0005215,0005391,0005515,0005524,0005886,0005889,0006813,0006883,0008556,0008900,0010248,0016020,0016324,0016887,0030007,0030955,0036376,0046872,0071805,1902600,1990573 remove_due_to_license_issue IC50=101nM P19156 29618813 1101 EMEINDHQLSVAELEQKYQTSATKGLSASLAAELLLRDGPNALRPPRGTPEYVKFARQLAGGLQCLMWVAAAICLIAFAIQASEGDLTTDDNLYLALALIAVVVVTGCFGYYQEFKSTNIIASFKNLVPQQATVIRDGDKFQINADQLVVGDLVEMKGGDRVPADIRILQAQGCKVDNSSLTGESEPQTRSPECTHESPLETRNIAFFSTMCLEGTAQGLVVNTGDRTIIGRIASLASGVENEKTPIAIEIEHFVDIIAGLAILFGATFFIVAMCIGYTFLRAMVFFMAIVVAYVPEGLLATVTVCLSLTAKRLASKNCVVKNLEAVETLGSTSVICSDKTGTLTQNRMTVSHLWFDNHIHSADTTEDQSGQTFDQSSETWRALCRVLTLCNRAAFKSGQDAVPVPKRIVIGDASETALLKFSELTLGNAMGYRERFPKVCEIPFNSTNKFQLSIHTLEDPRDPRHVLVMKGAPERVLERCSSILIKGQELPLDEQWREAFQTAYLSLGGLGERVLGFCQLYLSEKDYPPGYAFDVEAMNFPTSGLCFAGLVSMIDPPRATVPDAVLKCRTAGIRVIMVTGDHPITAKAIAASVGIISEGSETVEDIAARLRVPVDQVNRKDARACVINGMQLKDMDPSELVEALRTHPEMVFARTSPQQKLVIVESCQRLGAIVAVTGDGVNDSPALKKADIGVAMGIAGSDAAKNAADMILLDDNFASIVTGVEQGRLIFDNLKKSIAYTLTKNIPELTPYLIYITVSVPLPLGCITILFIELCTDIFPSVSLAYEKAESDIMHLRPRNPKRDRLVNEPLAAYSYFQIGAIQSFAGFTDYFTAMAQEGWFPLLCVGLRPQWENHHLQDLQDSYGQEWTFGQRLYQQYTCYTVFFISIEMCQIADVLIRKTRRLSAFQQGFFRNRILVIAIVFQVCIGCFLCYCPGMPNIFNFMPIRFQWWLVPMPFSLLIFVYDEIRKLGVRCCPGSWWDQELYY 5ymx A 1.35 BS01 GDP A 1 L22 C23 G24 K25 T26 T27 G81 N141 K142 D144 L145 V169 P171 L21 C22 G23 K24 T25 T26 G80 N140 K141 D143 L144 V168 P170 3.6.5.2 0003924,0005515,0005525,0005737,0032880 remove_due_to_license_issue Q1DB04 31560685 301 SFINYSSREINCKIVYYGPGLCGKTTNLQYIYNKTAAETKGKLISLSTETDRTLFFDFLPLSLGEIRGFKTRFHLYTVPGQVFYDASRKLILKGVDGVVFVADSQIERMEANMESLENLRINLAEQGYDLNKIPYVIQYNKRDLPNAVTVEEMRKALNHRNIPEYQAVAPTGVGVFDTLKAVAKLVLTELKKGGGSHHHHHH 5yof A 1.51 BS01 7HS B 1 G82 D83 G33 D34 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0004252,0044423 remove_due_to_license_issue Q32ZE1 29526431 201 DMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVE 5yof B 1.51 BS01 7HS B 1 H51 D129 Y130 A132 S135 G151 N152 G153 Y161 H36 D114 Y115 A117 S120 G136 N137 G138 Y146 2.1.1.56,2.1.1.57,2.7.7.48,3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0005524 remove_due_to_license_issue Q32ZE1 29526431 201 GETTDGVYRVMTRRLLGSTQVGVGVMQEGVFHTMWHVTKGAALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGLSEVQLLAVPPGERAKNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKSGRVIGLYGNGVVIKNGSYVSAITQGKRE 5yp5 A 2.65 BS02 4CZ A 1 Q286 L287 C320 H323 L324 M358 R364 M365 R367 A368 F377 F378 F388 I397 I400 F401 Q22 L23 C56 H59 L60 M94 R100 M101 R103 A104 F113 F114 F124 I133 I136 F137 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=<25119nM, EC50=25nM P51449 29456799 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5yp6 A 2.2 BS02 4CX A 1 Q286 L287 W317 C320 H323 L324 R364 M365 R367 A368 V376 F377 F378 F388 L391 I397 I400 Q22 L23 W53 C56 H59 L60 R100 M101 R103 A104 V112 F113 F114 F124 L127 I133 I136 ? 0003677,0004879,0005634,0006355 ic50>0.0000316M remove_due_to_license_issue IC50=<25119nM, EC50=20nM P51449 29456799 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 5ypp A 1.9 BS01 VAL A 1 H20 G22 V23 M24 C43 H12 G14 V15 M16 C35 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypp A 1.9 BS02 VAL A 2 N37 V38 N29 V30 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 102 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypp B 1.9 BS01 VAL A 1 N37 V38 N29 V30 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypp B 1.9 BS02 VAL A 2 H20 G22 V23 M24 C43 H12 G14 V15 M16 C35 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 102 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypw A 2.3 BS01 VAL A 1 H20 G22 V23 M24 C43 H12 G14 V15 M16 C35 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypw A 2.3 BS02 VAL B 1 N37 V38 N29 V30 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypw B 2.3 BS01 VAL A 1 N37 V38 N29 V30 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypw B 2.3 BS02 VAL B 1 H20 M24 C43 H12 M16 C35 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypy A 1.966 BS01 VAL A 1 H20 G22 V23 M24 C43 H13 G15 V16 M17 C36 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 HDNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypy A 1.966 BS02 VAL B 1 N37 V38 N30 V31 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 HDNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypy B 1.966 BS01 VAL A 1 N37 V38 N29 V30 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5ypy B 1.966 BS02 VAL B 1 H20 V23 M24 C43 H12 V15 M16 C35 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 DNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5yql A 1.601 BS01 A2I A 1 F96 F119 F131 A135 L138 Y139 P140 F143 D170 F190 I232 F234 F46 F66 F78 A82 L85 Y86 P87 F90 D117 F137 I179 F181 P94 D95 F96 R97 N168 D170 H187 P44 D45 F46 R47 N115 D117 H134 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=25.9uM remove_due_to_license_issue IC50=26303nM Q8IXJ6 29957526 1001 GASGSERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPSTGLLEKYHLPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGQSDPFLGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5yqn A 1.6 BS02 L55 A 1 F96 R97 F119 L138 Y139 P140 F143 H187 F190 V233 F235 F46 R47 F58 L77 Y78 P79 F82 H126 F129 V172 F174 P94 D95 F96 R97 N168 D170 H187 P44 D45 F46 R47 N107 D109 H126 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=93.7uM remove_due_to_license_issue IC50=93700nM Q8IXJ6 29957526 402 GASGSERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPSTPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGQSDPFLGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5yqo A 1.483 BS02 L5C A 1 F96 R97 F119 A135 Y139 P140 F143 I169 D170 H187 F190 V233 F235 F46 R47 F58 A74 Y78 P79 F82 I108 D109 H126 F129 V172 F174 P94 D95 F96 R97 N168 D170 H187 P44 D45 F46 R47 N107 D109 H126 2.3.1.-,2.3.1.286 0017136,0051287,0070403 ic50=0.815uM remove_due_to_license_issue IC50=813nM Q8IXJ6 29957526 402 GASGSERLLDELTLEGVARYMQSERCRRVICLVGAGISTSAGIPDFRSPSTPYPEAIFEISYFKKHPEPFFALAKELYPGQFKPTICHYFMRLLKDKGLLLRCYTQNIDTLERIAGLEQEDLVEAHGTFYTSHCVSASCRHEYPLSWMKEKIFSEVTPKCEDCQSLVKPDIVFFGESLPARFFSCMQSDFLKVDLLLVMGTSLQVQPFASLISKAPLSTPRLLINKEKAGQSDPFLGGMDFDSKKAYRDVAWLGECDQGCLALAELLGWKKELEDLVRREHASIDAQS 5yqx A 1.82 BS01 E0K A 1 W81 P82 F83 L92 N140 I146 W40 P41 F42 L51 N99 I105 ? remove_due_to_license_issue Kd=110nM, IC50=100nM O60885 29758518 201 GSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5yr4 A 1.82 BS04 TN4 A 1 P192 Y195 H212 Y300 C301 M309 H310 E336 P103 Y106 H123 Y211 C212 M220 H221 E247 3.4.11.18 0006508,0070006 remove_due_to_license_issue P53582 30837307 410 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLMHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 5yr5 A 1.6 BS04 OVA A 1 Y195 H212 Y300 C301 E336 Y106 H123 Y211 C212 E247 3.4.11.18 0006508,0070006 remove_due_to_license_issue P53582 30837307 405 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLLHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 5yr6 A 1.75 BS03 TN4 A 1 P192 Y195 H212 Y300 C301 H310 E336 W353 P103 Y106 H123 Y211 C212 H221 E247 W264 3.4.11.18 0006508,0070006 remove_due_to_license_issue P53582 30837307 410 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLLHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS 5yto B 1.9 BS02 946 B 1 E21 P28 K30 W32 E100 E22 P29 K31 W33 E101 H46 H48 H63 H71 H80 D83 H120 R143 H47 H49 H64 H72 H81 D84 H121 R144 1.15.1.1 0000302,0000303,0001541,0001819,0001890,0001895,0002262,0004784,0005507,0005515,0005576,0005615,0005634,0005654,0005737,0005739,0005758,0005759,0005777,0005829,0005886,0006749,0006801,0006879,0006915,0006979,0007283,0007566,0007605,0007626,0008089,0008090,0008217,0008270,0008340,0009408,0009410,0010467,0016209,0016491,0019226,0019228,0019430,0030346,0031267,0031410,0032287,0032839,0032930,0032991,0033081,0035234,0040014,0042542,0042554,0042802,0042803,0043025,0043065,0043066,0043087,0043410,0043524,0045471,0046620,0046716,0046872,0048538,0048678,0050665,0050728,0050766,0051087,0051093,0051881,0060047,0060052,0060087,0060088,0070062,0072593,0099610,1902177,1904115,2000242 Kd=33uM remove_due_to_license_issue P00441 29679384 203 MATKAVCVLKGDGPVQGIINFEQKESNGPVKVWGSIKGLTEGLHGFHVHEFGDNTAGCTSAGPHFNPLSRKHGGPKDEERHVGDLGNVTADKDGVADVSIEDSVISLSGDHCIIGRTLVVHEKADDLGKGGNEESTKTGNAGSRLACGVIGIAQ 5yto B 1.9 BS04 946 H 1 K3 E21 K4 E22 H46 H48 H63 H71 H80 D83 H120 R143 H47 H49 H64 H72 H81 D84 H121 R144 1.15.1.1 0000302,0000303,0001541,0001819,0001890,0001895,0002262,0004784,0005507,0005515,0005576,0005615,0005634,0005654,0005737,0005739,0005758,0005759,0005777,0005829,0005886,0006749,0006801,0006879,0006915,0006979,0007283,0007566,0007605,0007626,0008089,0008090,0008217,0008270,0008340,0009408,0009410,0010467,0016209,0016491,0019226,0019228,0019430,0030346,0031267,0031410,0032287,0032839,0032930,0032991,0033081,0035234,0040014,0042542,0042554,0042802,0042803,0043025,0043065,0043066,0043087,0043410,0043524,0045471,0046620,0046716,0046872,0048538,0048678,0050665,0050728,0050766,0051087,0051093,0051881,0060047,0060052,0060087,0060088,0070062,0072593,0099610,1902177,1904115,2000242 Kd=33uM remove_due_to_license_issue P00441 29679384 202 MATKAVCVLKGDGPVQGIINFEQKESNGPVKVWGSIKGLTEGLHGFHVHEFGDNTAGCTSAGPHFNPLSRKHGGPKDEERHVGDLGNVTADKDGVADVSIEDSVISLSGDHCIIGRTLVVHEKADDLGKGGNEESTKTGNAGSRLACGVIGIAQ 5yts A 1.77 BS01 rna B 0 K64 W65 N67 N70 Y72 F74 D83 F85 H87 K118 K13 W14 N16 N19 Y21 F23 D32 F34 H36 K63 ? 0003676 remove_due_to_license_issue P67809 31160337 2 ~ 5 KKVIATKVLGTVKWFNVRNGYGFINRNDTKEDVFVHQTAIKKKYLRSVGDGETVEFDVVEGEKGAEAANVTGPG 5ytt A 1.6 BS01 rna B 0 W65 N67 N70 Y72 F74 D83 F85 H87 K118 G119 A120 W14 N16 N19 Y21 F23 D32 F34 H36 K64 G65 A66 ? 0003676 remove_due_to_license_issue P67809 31160337 1 ~ 7 KKVIATKVLGTVKWFNVRNGYGFINRNDTKEDVFVHQTAIKKNKYLRSVGDGETVEFDVVEGEKGAEAANVTGPG 5ytu A 1.9 BS01 5FW A 1 G12 P13 G13 P14 H46 H48 H63 H71 H80 D83 H120 R143 H47 H49 H64 H72 H81 D84 H121 R144 1.15.1.1 0000302,0000303,0001541,0001819,0001890,0001895,0002262,0004784,0005507,0005515,0005576,0005615,0005634,0005654,0005737,0005739,0005758,0005759,0005777,0005829,0005886,0006749,0006801,0006879,0006915,0006979,0007283,0007566,0007605,0007626,0008089,0008090,0008217,0008270,0008340,0009408,0009410,0010467,0016209,0016491,0019226,0019228,0019430,0030346,0031267,0031410,0032287,0032839,0032930,0032991,0033081,0035234,0040014,0042542,0042554,0042802,0042803,0043025,0043065,0043066,0043087,0043410,0043524,0045471,0046620,0046716,0046872,0048538,0048678,0050665,0050728,0050766,0051087,0051093,0051881,0060047,0060052,0060087,0060088,0070062,0072593,0099610,1902177,1904115,2000242 Kd=12uM remove_due_to_license_issue P00441 29679384 201 MATKAVCVLKGDGPVQGIINFEQKESNGPVKVWGSIKGLTEGLHGFHVHEFGDNTAGCTSAGPHFNPLSRKHGGPKDEERHVGDLGNVTADKDGVADVSIEDSVISLSGDHCIIGRTLVVHEKADDLGKGGNEESTKTGNAGSRLACGVIGIAQ 5ytv A 1.7 BS01 rna B 0 K64 W65 N67 N70 Y72 F74 D83 F85 H87 K118 K13 W14 N16 N19 Y21 F23 D32 F34 H36 K64 ? 0003676 remove_due_to_license_issue P67809 31160337 2 ~ 5 KKVIATKVLGTVKWFNVRNGYGFINRNDTKEDVFVHQTAIKKNKYLRSVGDGETVEFDVVEGEKGAEAANVTGPG 5ytx A 1.551 BS01 rna B 0 W65 N67 N70 Y72 F74 D83 F85 H87 K118 G119 A120 W14 N16 N19 Y21 F23 D32 F34 H36 K63 G64 A65 ? 0003676 remove_due_to_license_issue P67809 31160337 2 ~ 5 KKVIATKVLGTVKWFNVRNGYGFINRNDTKEDVFVHQTAIKKKYLRSVGDGETVEFDVVEGEKGAEAANVTGPG 5yu9 A 1.95 BS01 1E8 A 1 L718 G719 A743 K745 M766 M790 M793 C797 R841 L844 T854 D855 F856 L19 G20 A44 K46 M63 M87 M90 C94 R138 L141 T151 D152 F153 D837 A839 R841 N842 D855 D134 A136 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=0.5nM, Kd=6.9nM P00533 27626175 1101 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDADEYL 5yum A 2.432 BS01 ILE A 1 N19 H20 V23 M24 C43 N12 H13 V16 M17 C36 2.2.1.6 0003984,0005515,0005737,0005829,0005948,0008652,0009082,0009097,0009099,0016740,1990610 remove_due_to_license_issue P0ADF8 30887800 101 HDNVILELTVRNHPGVMTHVCGLFARRAFNVEGILCLPIQDSDKSHIWLLVNDDQRLEQMISQIDKLEDVVKVQRNQSDPTMFNKIAVFFQ 5yun B 2.67 BS01 MYC B 1 R62 I105 N106 G107 R51 I94 N95 G96 ? 0003697,0006260 remove_due_to_license_issue P40947 30213633 201 GVNKVILVGNVGGDPETRYMPNGNAVTNITLATSESWQERTEWHRVVFFGRLAEIAGEYLRKGSQVYVEGSLRTRKWQGQDGQDRYTTEIVVDINGNMQLLGG 5yun D 2.67 BS01 MYC D 1 I105 N106 I95 N96 ? 0003697,0006260 remove_due_to_license_issue P40947 30213633 201 ARGVNKVILVGNVGGDPETRYMPNGNAVTNITLATSESWERTEWHRVVFFGRLAEIAGEYLRKGSQVYVEGSLRTRKWQGQDGQDRYTTEIVVDINGNMQLL 5yve A 3.4 BS02 AF9 A 1 L265 D266 L245 D246 ? 0001614,0001666,0004931,0005216,0005524,0005886,0006811,0006812,0007165,0007268,0007274,0009266,0009408,0009409,0009612,0009743,0010524,0014832,0015267,0016020,0030424,0030432,0033198,0034220,0035590,0043005,0043235,0046872,0048167,0048266,0050804,0050850,0050909,0051649,0060079,0070207,0070588,0071318,0098655,0098662,0098685,0098686,0098794 remove_due_to_license_issue IC50=45nM P56373 29674445 405 WTIGIINRVVQLLIISYFVGWVFLHEKAYQVRDTAIESSVVTKVKGSGLYANRVMDVSDYVTPPQGTSVFVIITKMIVTENQMQGFCPESEEKYRCVSDSQCGPERLPGGGILTGRCVNYSSVLRTCEIQGWCPTEVDTVETPIMMEAENFTIFIKNSIRFPLFNFEKGNLLPNLTARDMKTCRFHPDKDPFCPILRVGDVVKFAGQDFAKLARTGGVLGIKIGWVCDLDKAWDQCIPKYSFTRLDSVSEKSSVSPGYNFRFAKYYKMENGSEYRTLLKAFGIRFDVLVYGNAGKFNIIPTIISSVAAFTSVGVGTVLCDIILLNFL 5yvt A 2.4 BS02 NAI A 1 L72 T74 N84 E260 V262 H263 G264 I269 N276 D317 L69 T71 N79 E255 V257 H258 G259 I264 N271 D312 Y126 K173 D206 D230 D234 Y121 K168 D201 D225 D229 1.1.1.41 0000287,0004449,0005515,0005634,0005739,0005759,0005975,0006099,0006102,0016491,0016616,0045242,0046872,0051287 Kd=109uM remove_due_to_license_issue P50213 29453450 402 VQTVTLIPGDGIGPEISAAVMKIFDAAKAPIQWEERNVTAIQGPGGKWMIPSEAKESMDKNKMGLKGPLKTPIAAPSMNLLLRKTFDLYANVRPCVSIEGYKTPYTDVNIVTIRENTEGEYSGIEHVIVDGVVQSIKLITEGASKRIAEFAFEYARNNHRSNVTAVHKANIMRMSDGLFLQKCREVAESCKDIKFNEMYLDTVCLNMVQDPSQFDVLVMPNLYGDILSDLCAGLIGGLGVTPSGNIGANGVAIFESVHGTAPDIAGKDMANPTALLLSAVMMLRHMGLFDHAARIEAACFATIKDGKSLTKDLGGNAKCSDFTEEICRRVKD 5yvt A 2.4 BS03 NAI B 1 N175 D206 N170 D201 Y126 K173 D206 D230 D234 Y121 K168 D201 D225 D229 1.1.1.41 0000287,0004449,0005515,0005634,0005739,0005759,0005975,0006099,0006102,0016491,0016616,0045242,0046872,0051287 Kd=109uM remove_due_to_license_issue P50213 29453450 401 VQTVTLIPGDGIGPEISAAVMKIFDAAKAPIQWEERNVTAIQGPGGKWMIPSEAKESMDKNKMGLKGPLKTPIAAPSMNLLLRKTFDLYANVRPCVSIEGYKTPYTDVNIVTIRENTEGEYSGIEHVIVDGVVQSIKLITEGASKRIAEFAFEYARNNHRSNVTAVHKANIMRMSDGLFLQKCREVAESCKDIKFNEMYLDTVCLNMVQDPSQFDVLVMPNLYGDILSDLCAGLIGGLGVTPSGNIGANGVAIFESVHGTAPDIAGKDMANPTALLLSAVMMLRHMGLFDHAARIEAACFATIKDGKSLTKDLGGNAKCSDFTEEICRRVKD 5yvt B 2.4 BS01 NAI B 1 I26 E80 T81 P252 G253 R272 N273 T274 G275 S277 I278 A284 N285 D326 I12 E66 T67 P238 G239 R258 N259 T260 G261 S263 I264 A270 N271 D312 Y135 K182 D215 N239 N243 Y121 K168 D201 N225 N229 ? 0000287,0004449,0005515,0005524,0005730,0005739,0005759,0005975,0006099,0006102,0016616,0045242,0046872,0051287 Kd=109uM remove_due_to_license_issue P51553 29453450 401 RHTVTMIPGDGIGPELMLHVKSVFRHACVPVDFEEVHVSSNADEEDIRNAIMAIRRNRVALKGNIETNHNLPPSHKSRNNILRTSLDLYANVIHCKSLPGVVTRHKDIDILIVRENTEGEYSSLEHESVAGVVESLKIITKAKSLRIAEYAFKLAQESGRKKVTAVHKANIMKLGDGLFLQCCREVAARYPQITFENMIVDNTTMQLVSRPQQFDVMVMPNLYGNIVNNVCAGLVGGPGLVAGANYGHVYAVFETATRNTGKSIANKNIANPTATLLASCMMLDHLKLHSYATSIRKAVLASMDNENMHTPDIGGQGTTSEAIQDVIRHIRVI 5ywx A 1.74 BS02 93C A 1 M11 G13 R14 Q36 M99 W104 Y152 M10 G12 R13 Q35 M98 W103 Y151 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.14nM remove_due_to_license_issue Kd=0.140000nM O60760 30121213 302 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 5ywy A 3.2 BS01 7UR A 1 T76 Y80 W169 L312 I315 R316 S319 V320 T59 Y63 W152 L246 I249 R250 S253 V254 ? 0004930,0004955,0004957,0007186,0016020 remove_due_to_license_issue P35408 30510193 501 NSPVTIPAVMFIFGVVGNLVAIVVLCKSRKEQKETTFYTLVCGLLVTDLLGTLLVSPVTIATYMKGQWPGGQPLCEYSTFILLFFSLSRLSIICAMSVERYLAINHAYFYSHYVDKRLAGLTLFAVYASNVLFCALPNMGLGSSRLQYPDTWCFIDWTTQVTAHAAYSYMYAGFSSFLILATVLCNVLVCGALLRMHAGAEIQMVILLIATSLVVLICSIPLVVRVFVNQLYQPSLEREVSKNPDLQAIRIASVNPILDPWIYILLRKTVLSKAIEKIKC 5yyb A 2.484 BS01 NGE A 1 S27 H333 S362 Y366 D383 P384 F387 W397 R408 S22 H328 S357 Y361 D378 P379 F382 W392 R403 ? 0015833,0030288,0043190,0055085,1904680 Kd=277nM remove_due_to_license_issue Q7VL18 30315109 501 GSTIEAGIAYPISTGFDPLTSSGASSMAANLHIFEGLVDLHPVTRQPYLALAAKEPEQKDDLTYYISLREGAMFHDGSPVTTEDVVYSFERVLDPAKASLFAQFIPFIASVTALDDNVVEFKLKYPFALFKERLTIIKIVPKHIVEAGQSAFDAKPIGSGPYKFVSATKDDRIVFEANTVYNGHYPAKVEKMTWFLLSDDAARVTAQESGRVQAIESVPYLDAERLKRKNNVESVQSFGLLFLMFNCEKAPFDNPKVRQALHYALDKQKLIDIVFLGNAKAATSYLQDTHPDYVKASSQYDYDKAKAEKLLAEAGITNLTFQLLATDHAWVKECAPLILESWNALSVVKVTLQHLQSGALYSAHVDKGAYEVVIAPGDPSVFGNDLDLLLSWWYRGDVWPKRRFRWANTAEYHEVQKLLDEAIKNPAGSKVAWQKAINIIAEQVPLYPIIHRKLPTAWNTKKLTDFQPLPTTGLSFLGVGRT 5yyf A 1.903 BS03 FOA B 1 F28 F59 S76 G77 Y78 F28 F59 S76 G77 Y78 ? remove_due_to_license_issue P42568 30374167 101 MASSCAVQVKLELGHRAQVRKKPTVEGFTHDWMVFVRGPEHSNIQHFVEKVVFHLHESFPRPKRVCKDPPYKVEESGYAGFILPIEVYFKNKEEPRKVRFDYDLFLHLEGHPPVNHLRCEKLTFNNPTEDFRRKLLKA 5yz2 A 1.75 BS01 AMP A 1 I80 H100 T180 D183 I18 H38 T118 D121 ? Kd=11.3uM remove_due_to_license_issue P0AE78 29453981 301 ELALQRVRDIMIPRSQMITLKRNQTLDECLDVIIESAHSRFPVISEDKDHIEGILMAKDLLPFMRSDAEAFSMDKVLRQAVVVPESKRVDRMLKEFRSQRYHMAIVIDEFGGVSGLVTIEDILELIVGEIE 5yz2 B 1.75 BS01 AMP B 1 I74 M79 I80 H100 S101 T180 D183 I12 M17 I18 H38 S39 T118 D121 ? Kd=11.3uM remove_due_to_license_issue P0AE78 29453981 301 ELALQRVRDIMIPRSQMITLKRNQTLDECLDVIIESAHSRFPVISEDKDHIEGILMAKDLLPFMRSDAEAFSMDKVLRQAVVVPESKRVDRMLKEFRSQRYHMAIVIDEFGGVSGLVTIEDILELIVGEIEKGQFL 5yz7 A 1.898 BS01 94X A 1 F78 S147 Y209 C241 V244 F245 F25 S94 Y156 C188 V191 F192 3.1.-.- remove_due_to_license_issue Q10QA5 29727000 500 AKLLQILNVRVVGSGERVVVLSHGFGTDQSAWSRVLPYLTRDHRVVLYDLVCAGSVNPDHFDFRRYDNLDAYVDDLLAILDALRIPRCAFVGHSVSAMIGILASIRRPDLFAKLVLIGASPRFLNDSDYHGGFELEEIQQVFDAMGANYSAWATGYAPLAVGADVPAAVQEFSRTLFNMRPDISLHVCQTVFKTDLRGVLGMVRAPCVVVQTTRDVSVPASVAAYLKAHLGGRTTVEFLQTEGHLPHLSAPSLLAQVLRRALARY 5yzc B 2.334 BS01 95C B 1 T369 L370 P451 I452 S453 N462 T255 L256 P337 I338 S339 N348 ? 0019064 remove_due_to_license_issue Q786F3 29463726 601 GVVLAGAALGVATAAQITAGIALHQSMLNSQAIDNLRASLETTNQAIEAIRQAGQEMILAVQGVQDYINNELIPSMNQLSCDLIGQKLGLKLLRYYTEILSLFGPSLRDPISAEISIQALSYALGGDINKVLEKLGYSGGDLLGILESRGIKARITHVDTESYFIVLSIAYPTLSEIKGVIVHRLEGVSYNIGSQEWYTTVPKYVATQGYLISNFDESSCTFMPEGTVCSQNALYPMSPLLQECLRGSTKSCARTLVSGSFGNRFILSQGNLIANCASILCKCYTTGTIINQDPDKILTYIAADHCPVVEVNGVTIQVGSRRYPDAVYLHRIDLGPPISLERLDVGTNLGNAIAKLEDAKELLESSD 5yzz C 2.58 BS01 dna A 0 R309 R347 W349 N351 R23 R61 W63 N65 ? 0003677 remove_due_to_license_issue Q8W4L5 29733847 1 ~ 13 LNLNIVPLFEKTLSASDAGRIGRLVLPKACAEAYFPPISQSEGIPLKIQDVRGREWTFQFRYWPNNNSRMYVLEGVTPCIQSMMLQAGDTVTFSRVDPGGKLIMGSRKAAN 5yzz C 2.58 BS02 dna B 0 K297 S300 A301 S302 V311 P313 K314 N351 M356 K11 S14 A15 S16 V25 P27 K28 N65 M70 ? 0003677 remove_due_to_license_issue Q8W4L5 29733847 1 ~ 13 LNLNIVPLFEKTLSASDAGRIGRLVLPKACAEAYFPPISQSEGIPLKIQDVRGREWTFQFRYWPNNNSRMYVLEGVTPCIQSMMLQAGDTVTFSRVDPGGKLIMGSRKAAN 5z1c U 1.45 BS01 ZXI U 1 D189 S190 S195 W215 G216 D192 S193 S198 W218 G219 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue P00749 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5z1r A 1.62 BS01 EFL A 1 W81 V87 L94 N140 I146 W49 V55 L62 N108 I114 ? remove_due_to_license_issue IC50=1990nM O60885 29541371 201 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 5z1s A 1.42 BS01 EFM A 1 W81 V87 N140 I146 W49 V55 N108 I114 ? remove_due_to_license_issue Kd=302nM, IC50=690nM O60885 29541371 201 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 5z1t A 1.42 BS01 EFN A 1 W81 V87 L94 N140 I146 W49 V55 L62 N108 I114 ? remove_due_to_license_issue Kd=498nM, IC50=630nM O60885 29541371 201 HHHHHLVPRGSNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 5z2t C 2.623 BS01 dna E 0 V12 R48 I51 N55 R59 V4 R40 I43 N47 R51 ? 0003677 remove_due_to_license_issue Q9UBX2 29572508 2 ~ 14 RTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARHP 5z2t C 2.623 BS02 dna F 0 F29 R57 F21 R49 ? 0003677 remove_due_to_license_issue Q9UBX2 29572508 14 ~ 26 RTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARHP 5z2t D 2.623 BS01 dna E 0 T10 R48 I51 W52 N55 R59 T2 R40 I43 W44 N47 R51 ? 0003677 remove_due_to_license_issue Q9UBX2 29572508 2 ~ 14 RTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARHPG 5z4h A 2.0 BS01 A8K A 1 N46 A47 Q72 D73 I78 A91 I94 M95 T165 V167 N31 A32 Q57 D58 I63 A76 I79 M80 T133 V135 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue P0AES6 30429968 303 LDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLHGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHY 5z4o A 1.73 BS01 HX8 A 1 V43 N46 A47 Q72 D73 I78 I94 M95 T165 V167 V28 N31 A32 Q57 D58 I63 I79 M80 T131 V133 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue P0AES6 30429968 301 LDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHY 5z5f A 2.1 BS02 FUB A 1 D14 F31 F73 A74 D121 E177 T197 H238 R269 D14 F31 F73 A74 D121 E177 T197 H238 R269 3.2.1.37 0004553,0005975,0009044,0016798,0046872 remove_due_to_license_issue Q2I2N4 29698436 602 MEYSNPVIKGFYPDPSICRVGSDYYLVTSSFQYFPGVPIFHSTNLINWNKIGYCLIRPSQLMLNNATNRSGIFAPTLRYHEGIFYLITTNVTLKKNFIVMSEDLQGEWSEPIWIDGWGGIDPSLFFDNDGKVYITGTNDNARGEELGIYQAEIDLKKGSIIGERKLIWKGTGGSYPEAPHLYKVNGWYYLLIAEGGTEYGHMVTVARSKYPFGPFESCPFNPILTHRSTNHPLQAIGHADIVQYHDGSWWAVFHGTRPISYPPKHHLGRETCLAPIKWTDDGWPIIGYNGRIDIKMDAGYLPVKEIIEDDFNSDIFSTDWNFIQNPRLEHYSLKGRPSWLKMRGTEKTLNDINSPTFIGRRQEHFVCNVSTLLEFKPNQDNEEAGLTVYMNEKHHYEIALTKKNGRINVVLKKTVGDIQVVVNSLEYFSNTIIFSIQANPEEYKFSFVDPNTGQTYLLGTGLTTLLSTEVAGGFTGVYFGLYATGNGKVCTAPAFFDWFKYIPE 5z66 A 1.8 BS01 VDM A 1 P150 F154 Y158 W160 D161 N197 Y203 Q208 R277 E279 G310 D312 W447 E511 Y512 F518 W520 P116 F120 Y124 W126 D127 N163 Y169 Q174 R243 E245 G276 D278 W413 E477 Y478 F484 W486 0004555,0005975,0005991,0005993,0042597,0071474 remove_due_to_license_issue 30657252 609 TQTTSPDILLGPLFNDVQSAKLFPDQKTFADAVPKSDPLMILADYRMQHTQSSFDLRHFVEMNFTLPAEGEKYVPPAGQSLREHIDDLWPVLTRTTDKASNKWDSLLPLPKPYVVPGGRFREVYYWDSYFTMLGLAESDHWDKISDMVDNFAYEIDTFGHIPNGNRSYYLSRSQPPFFSMMVELLATHDSDALKKYRPQMEKEYAYWMDGVDALQPGQANKRVVKLDDGAILNRYWDDRDTPRPESWLDDVNTAKSNPNRPATEIYRDLRSAAASGWDFSSRWMDDPQKLGTIRTTSIVPVDLNALMFKMEKLLARASQESGDAASASKYEALATARQKAIESHLWNDKEGWYADYDLKSKKVRNQLTAAALFPLYVKAAAQDRADKVAAATSSRLLKPGGIATTTVNSGQQWDAPNGWAPLQWVAAEGLQNYGQEKVSMDVTWRFLKNVQHTYDREKKLVEKYDVSTTGTGGGGGEYPLQDGFGWSNGVTLKMLDRVCPKAKPCDSVPENQ 5z68 A 3.0 BS01 ATP A 1 R12 N13 L31 N32 A33 G35 K36 S37 N38 V61 F63 R16 N17 L35 N36 A37 G39 K40 S41 N42 V65 F67 ? 0000731,0003677,0003697,0005524,0005737,0006260,0006281,0006302,0009432 remove_due_to_license_issue Q8RDL3 29391496 401 AYYSMYLKEIFVDNFRNLKKQKLEFCEGVNLIYGLNAQGKSNLLEAIRLLSMGRSFRGSKMSELVKFDEEYFYVRGLVRSADFYEKKIEFGYKVNGNKVIKVNGNKLKSTGEILGHFLTVIFSPEDIEIIKEGPSRRRKYLDACISVIDKNYFFDLLQYNKTLSNRNSLLKKIKEEGKGEDLLEIFDEKLAEYGARIIKVRNNYLEKLKNSMSKFLMEISNEKLEIIYLNSAGVKEVHEENLIREKLKNRLTKSLTLDLKYLSTQVGPHREDFKILINGYDSRVYSSQGQKRTAALCLKLSELEILEEETGEKPVLLLDDVMSELDDNRKKYILKKLEGFQSFITHTSKSDVEGDCCFKIYDGIVDKL 5z68 A 3.0 BS02 ATP B 1 Y281 S283 Q286 Y285 S287 Q290 ? 0000731,0003677,0003697,0005524,0005737,0006260,0006281,0006302,0009432 remove_due_to_license_issue Q8RDL3 29391496 401 AYYSMYLKEIFVDNFRNLKKQKLEFCEGVNLIYGLNAQGKSNLLEAIRLLSMGRSFRGSKMSELVKFDEEYFYVRGLVRSADFYEKKIEFGYKVNGNKVIKVNGNKLKSTGEILGHFLTVIFSPEDIEIIKEGPSRRRKYLDACISVIDKNYFFDLLQYNKTLSNRNSLLKKIKEEGKGEDLLEIFDEKLAEYGARIIKVRNNYLEKLKNSMSKFLMEISNEKLEIIYLNSAGVKEVHEENLIREKLKNRLTKSLTLDLKYLSTQVGPHREDFKILINGYDSRVYSSQGQKRTAALCLKLSELEILEEETGEKPVLLLDDVMSELDDNRKKYILKKLEGFQSFITHTSKSDVEGDCCFKIYDGIVDKL 5z68 B 3.0 BS01 ATP A 1 Y281 S283 Q286 Y284 S286 Q289 ? 0000731,0003677,0003697,0005524,0005737,0006260,0006281,0006302,0009432 remove_due_to_license_issue Q8RDL3 29391496 401 YYSMYLKEIFVDNFRNLKKQKLEFCEGVNLIYGLNAQGKSNLLEAIRLLSMGRSFRGSKMSELVKFDEEYFYVRGLVRSADFYEKKIEFGYKVNGNKVIKVNGNKLKSTGEILGHFLTVIFSPEDIEIIKEGPSRRRKYLDACISVIDKNYFFDLLQYNKTLSNRNSLLKKIKEEGKGEDLLEIFDEKLAEYGARIIKVRNNYLEKLKNSMSKFLMEISNEKLEIIYLNSAGVKEVHEENLIREKLKNRLTKSLTLDLKYLSTQVGPHREDFKILINGYDSRVYSSQGQKRTAALCLKLSELEILEEETGEKPVLLLDDVMSELDDNRKKYILKKLEGFQSFITHTSKSDVEGDCCFKIYDGIVDKLA 5z68 B 3.0 BS02 ATP B 1 R12 N13 N32 Q34 G35 K36 S37 N38 F63 R15 N16 N35 Q37 G38 K39 S40 N41 F66 ? 0000731,0003677,0003697,0005524,0005737,0006260,0006281,0006302,0009432 remove_due_to_license_issue Q8RDL3 29391496 401 YYSMYLKEIFVDNFRNLKKQKLEFCEGVNLIYGLNAQGKSNLLEAIRLLSMGRSFRGSKMSELVKFDEEYFYVRGLVRSADFYEKKIEFGYKVNGNKVIKVNGNKLKSTGEILGHFLTVIFSPEDIEIIKEGPSRRRKYLDACISVIDKNYFFDLLQYNKTLSNRNSLLKKIKEEGKGEDLLEIFDEKLAEYGARIIKVRNNYLEKLKNSMSKFLMEISNEKLEIIYLNSAGVKEVHEENLIREKLKNRLTKSLTLDLKYLSTQVGPHREDFKILINGYDSRVYSSQGQKRTAALCLKLSELEILEEETGEKPVLLLDDVMSELDDNRKKYILKKLEGFQSFITHTSKSDVEGDCCFKIYDGIVDKLA 5z6z A 2.301 BS01 dna D 0 R20 R21 R23 L24 W26 R62 N69 R73 R95 R124 Q139 Q143 R146 R2 R3 R5 L6 W8 R44 N51 R55 R68 R97 Q112 Q116 R119 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 GRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5z6z A 2.301 BS02 dna E 0 R20 R23 Y43 Q64 Q68 R71 R95 R96 R98 T99 R137 W141 N144 R148 R2 R5 Y25 Q46 Q50 R53 R68 R69 R71 T72 R110 W114 N117 R121 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 GRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5z7b A 2.1 BS01 VNL A 1 S28 V29 M133 H142 T144 L145 R148 Y168 S32 V33 M137 H146 T148 L149 R152 Y172 ? Kd=13uM remove_due_to_license_issue Q8NN31 30095229 201 AKDLMTLRSALLALLSSGPLTGYDASQRFGASVGFVWSGSDSQIYPELRKMEAEELLVGSDVPWGSKGATKTEYALSEKGWEALRKAWYEPVTYGPTRDPARLKAAYFEVGTNGDARRHLRAHIAHFEQQKIQSESMIDELKAKTHPTLARRLERSPKKEHERIVAFKVLAYEGQIARAQAEIEWAEKGLKLLDTL 5z7b B 2.1 BS01 VNL B 1 S28 M133 H142 T144 R148 Y168 S33 M138 H147 T149 R153 Y173 ? Kd=13uM remove_due_to_license_issue Q8NN31 30095229 201 SAKDLMTLRSALLALLSSGPLTGYDASQRFGASVGFVWSGSDSQIYPELRKMEAEELLVGSDVPWGSKGATKTEYALSEKGWEALRKAWYEPVTYGPTRDPARLKAAYFEVGTNGDARRHLRAHIAHFEQQKIQSESMIDELKAKTHPTLARRLERSPKKEHERIVAFKVLAYEGQIARAQAEIEWAEKGLKLLDTL 5z7j A 1.98 BS01 36J A 1 G35 L36 A105 S106 S157 W185 P190 I193 P194 H243 G32 L33 A102 S103 S154 W182 P187 I190 P191 H240 ? remove_due_to_license_issue A0A0D2ILK1 301 TRTRGYVTTKDGIKWYYEQEGSGPDVVLIPDGLGECQMFDKPMSLIASNGFRVTTFDMPGMSRSSDAPPETYQDITGRKLAGYIITLLDTLDIKIASVWGCASGASTVLALCSDYPERVRNGMPHEVPTENPDILLHIHEVDPATISQEMAANSRAASGNVEAWDALGPEVHARLHDNYPRWAYGYPRTIPPSAPVKTEDLHKVPIDWTVGASTPTKLFFENIVIAAREGINIGTLPGNHFPYVSHPEEFAKYVVETSRKYLK 5z89 A 1.42 BS01 EGC A 1 M139 T142 T190 M137 T140 T188 ? 0046872 remove_due_to_license_issue A0A0M3PNA2 30021834 304 SIGLAHNVTILGSGETTVVLGHGYGTDQSVWKLLVPYLVDDYKVLLYDHMGAGTTNPDYFDFDRYSSLEGYSYDLIAILEEFQVSKCIYVGHDMSSMAAAVASIFRPDLFHKLVMISPTPRLINTEEYYGGFEQKVMDETLRSLDENFKSLSLGTAPLLLACDLESAAMQEYCRTLFNMRPDIACCITRMICGLDLRPYLGHVTVPCHIIQSSNDIMVPVAVGEYLRKNLGGPSVVEVMPTEGHLPHLSMPEVTIPVVLRHIRQDITD 5z95 A 1.2 BS01 EGC A 1 F134 V138 M139 T142 T190 F132 V136 M137 T140 T188 ? 0046872 remove_due_to_license_issue A0A0M3PNA2 30021834 301 SIGLAHNVTILGSGETTVVLGHGYGTDQSVWKLLVPYLVDDYKVLLYDHMGAGTTNPDYFDFDRYSSLEGYSYDLIAILEEFQVSKCIYVGHSMSSMAAAVASIFRPDLFHKLVMISPTPRLINTEEYYGGFEQKVMDETLRSLDENFKSLSLGTAPLLLACDLESAAMQEYCRTLFNMRPDIACCITRMICGLDLRPYLGHVTVPCHIIQSSNDIMVPVAVGEYLRKNLGGPSVVEVMPTEGHLPHLSMPEVTIPVVLRHIRQDITD 5z99 A 1.494 BS01 SLB A 1 Y15 S27 H333 S362 Y366 D383 F387 W404 R408 Y13 S25 H331 S360 Y364 D381 F385 W402 R406 ? 0015833,0030288,0043190,0055085,1904680 Kd=133nM remove_due_to_license_issue Q7VL18 30315109 501 SPSGSTIEAGIAYPISTGFDPLTSSGASSMAANLHIFEGLVDLHPVTRQPYLALAAKEPEQKDDLTYYISLREGAMFHDGSPVTTEDVVYSFERVLDPAKASLFAQFIPFIASVTALDDNVVEFKLKYPFALFKERLTIIKIVPKHIVEAGQSAFDAKPIGSGPYKFVSATKDDRIVFEANTVYNGHYPAKVEKMTWFLLSDDAARVTAQESGRVQAIESVPYLDAERLKRKNNVESVQSFGLLFLMFNCEKAPFDNPKVRQALHYALDKQKLIDIVFLGNAKAATSYLQDTHPDYVKASSQYDYDKAKAEKLLAEAGITNLTFQLLATDHAWVKECAPLILESWNALSVVKVTLQHLQSGALYSAHVDKGAYEVVIAPGDPSVFGNDLDLLLSWWYRGDVWPKRRFRWANTAEYHEVQKLLDEAIKNPAGSKVAWQKAINIIAEQVPLYPIIHRKLPTAWNTKKLTDFQPLPTTGLSFLGVGRT 5z9e A 1.8 BS01 27K A 1 N46 I78 N31 I63 5.6.2.2 0003677,0003918,0005524,0006265 remove_due_to_license_issue P0AES6 30429968 304 LDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHY 5z9x A 2.8 BS01 rna R 0 D144 C145 E146 M147 R185 H223 S224 R227 R255 R256 P257 S258 L259 H278 D143 C144 E145 M146 R184 H222 S223 R226 R248 R249 P250 S251 L252 H266 3.1.-.- 0000175,0003676,0004527,0005515,0005634,0008408,0010587,0035198,0044747,0044748 remove_due_to_license_issue A3KPE8 30181559 2 ~ 10 ELKLATAEKQVLDELVKLLQSRDLRGENGNWKEFLHVYDKNADSPSDPSRRSHEDLVQFLTTFKKKEDLQLLKCHANHLLIENLKQESQDEDTPEQMLVRLTVEHPSYSLDYSFKPYSEDWFVSDVGMKMKKVMESTNMVAVDCEMVLCEDGTEGLVRVGVVDRDLKVILDEFVKPNKPVVDYRTDITGITAEDIENASLSVVDIQETLQPFLSTGTILVGHSLNRDLEVLKIDHPKVIDTALVFKLRRPSLNNLCKSILGYGVPHDCVHDASAAMKLALAVVEKRVD 5za1 A 2.52 BS01 9A0 A 1 Q286 L287 L324 M358 L362 M365 R367 A368 F377 F378 F388 H479 Q22 L23 L60 M94 L98 M101 R103 A104 F113 F114 F124 H215 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=14nM P51449 30301676 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVV 5za2 A 1.503 BS01 NXL A 1 S64 L119 Y150 T315 G316 S317 S57 L112 Y143 T308 G309 S310 S64 K67 Y150 E271 K314 S317 S57 K60 Y143 E264 K307 S310 3.5.2.6 0008800,0016787,0017001,0030288,0046677,0046872 Kd=1700nM remove_due_to_license_issue Q9L387 29439972 401 LTATVDGIIQPMLKAYRIPGMAVAVLKDGKAHYFNYGVANRESGQRVSEQTLFEIGSVSKTLTATLGAYAAVKGGFELDDKVSQHAPWLKGSAFDGVTMAELATYSAGGLPLQFPDEVDSNDKMQTYYRSWSPVYPAGTHRQYSNPSIGLFGHLAANSLGQPFEQLMSQTLLPKLGLHHTYIQVPESAMANYAYGYSKEDKPIRATPGVLAAEAYGIKTGSADLLKFVEANMGYQGDAALKSAIALTHTGFHSVGEMTQGLGWESYDYPVTEQVLLAGNSPAVSFQANPVTRFAVPKAMGEQRLYNKTGSTGGFGAYVAFVPARGIAIVMLANRNYPIEARVKAAHAILSQLAE 5za7 U 1.7 BS01 HMX U 1 D189 S190 Q192 G216 G219 D192 S193 Q195 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=1356nM remove_due_to_license_issue P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 5za8 U 1.9 BS01 27I U 1 D189 S190 Q192 S214 W215 G216 G219 C220 D192 S193 Q195 S217 W218 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=508nM remove_due_to_license_issue Ki=508nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5za9 U 1.62 BS01 50I U 1 S146 D189 S190 Q192 S214 W215 G216 G219 C220 G226 S145 D192 S193 Q195 S217 W218 G219 G221 C222 G229 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=183nM remove_due_to_license_issue Ki=183nM, IC50=530nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5zae U 1.73 BS01 EAU U 1 D189 S190 C191 Q192 S214 W215 G216 G219 C220 D192 S193 C194 Q195 S217 W218 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=156nM remove_due_to_license_issue Ki=156nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 5zaf U 1.65 BS01 28I U 1 D189 S190 C191 Q192 S214 G216 G219 C220 D192 S193 C194 Q195 S217 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=166nM remove_due_to_license_issue Ki=166nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5zag U 1.95 BS01 94I U 1 D189 S190 Q192 G216 G219 C220 D192 S193 Q195 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=108nM remove_due_to_license_issue Ki=108nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5zah U 2.98 BS01 30I U 1 D189 S190 Q192 S195 G216 G219 D192 S193 Q195 S198 G219 G221 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 remove_due_to_license_issue Ki=53nM, IC50=39nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5zaj U 1.65 BS01 32I U 1 D189 S190 C191 Q192 G216 G219 C220 D192 S193 C194 Q195 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=42nM remove_due_to_license_issue Ki=42nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5zbz A 1.3086 BS01 SAU A 1 G79 G81 Q115 G59 G61 Q95 3.6.4.13 0003676,0003724,0005524 Kd=12.5uM remove_due_to_license_issue P60842 31402318 301 GVIESNWNEIVDSFDDMNLSESLLRGIYAYGFEKPSAIQQRAILPCIKGYDVIAQAQSGTGKTATFAISILQQIELDLKATQALVLAPTRELAQQIQKVVMALGDYMGASCHACIGGTNVRAEVQKLQMEAPHIIVGTPGRVFDMLNRRYLSPKYIKMFVLDEADEMLSRGFKDQIYDIFQKLNSNTQVVLLSATMPSDVLEVTKKFMRDPIRILVKK 5zc5 U 1.9 BS01 09I U 1 S146 D189 S190 Q192 S214 W215 G216 G219 C220 S145 D192 S193 Q195 S217 W218 G219 G221 C222 H57 D102 Q192 G193 D194 S195 G196 H46 D97 Q195 G196 D197 S198 G199 3.4.21.73 0004252,0006508 Ki=88nM remove_due_to_license_issue Ki=88nM, IC50=430nM P00749 30130401 301 IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT 5zc9 A 2.0 BS01 rna B 0 P108 T109 R110 G136 G137 V140 T158 P159 G160 R161 D164 R168 R190 G191 F192 Q195 N280 T281 R282 H303 G304 R311 T329 D330 L331 P80 T81 R82 G108 G109 V112 T130 P131 G132 R133 D136 R140 R162 G163 F164 Q167 N252 T253 R254 H275 G276 R283 T301 D302 L303 3.6.4.13 0000339,0002183,0003676,0003689,0003723,0003724,0003725,0003729,0003743,0004386,0005515,0005524,0005634,0005737,0005829,0005886,0006338,0006412,0006413,0008135,0010494,0016020,0016281,0016787,0016887,0045944,0048471,0061775,0070062,0097165,0140584,0140588,0140665,0140849 remove_due_to_license_issue P60842 30595437 1 ~ 10 EIVDSFDDMNLSESLLRGIYAYGFEKPSAIQQRAILPCIKGYDVIAQAQSGTGKTATFAISILQQIELDLKATQALVLAPTRELAQQIQKVVMALGDYMGASCHACIGGTNVRAEVQKLQMEAPHIIVGTPGRVFDMLNRRYLSPKYIKMFVLDEADEMLSRGFKDQIYDIFQKLNSNTQVVLLSATMPSDVLEVTKKFMRDPIRILVKKEELTLEGIRQFYINVEREEWKLDTLCDLYETLTITQAVIFINTRRKVDWLTEKMHARDFTVSAMHGDMDQKERDVIMREFRSGSSRVLITTDLLARGIDVQQVSLVINYDLPTNRENYIHRIGRGGRFGRKGVAINMVTEEDKRTLRDIETFYNTSIEEMPLNVADLI 5zcu C 2.413 BS01 PYV C 1 K76 F78 S107 E109 F125 H130 L132 Y135 L178 N182 K43 F45 S74 E76 F92 H97 L99 Y102 L145 N149 ? ic50=2160nM remove_due_to_license_issue Q6EN42 30941543 301 VRRFHRHEPRDHQCSSAVAKHIKAPVHLVWSLVRRFDQPQLFKPFVSRCEMKGNIEIGSVREVNVKSGLPATRSTERLELLDDNEHILSVRFVGGDHRLKNYSSILTVHPEVIDGRPGTLVIESFVVDVPEGNTKDETCYFVEALLKCNLKSLAEVSERLVV 5zd4 A 2.17 BS01 dna E 0 R34 R38 R41 D64 N65 R382 R386 R389 D412 N413 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 A 2.17 BS02 dna F 0 E37 R40 K61 H62 E385 R388 K409 H410 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 B 2.17 BS01 dna E 0 E37 R40 K61 H62 E384 R387 K408 H409 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 IEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 B 2.17 BS02 dna F 0 R30 R34 R38 R41 D64 N65 R377 R381 R385 R388 D411 N412 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 IEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 C 2.17 BS01 dna G 0 R36 E37 R40 K61 H62 R384 E385 R388 K409 H410 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 C 2.17 BS02 dna H 0 R30 N33 R34 R41 D64 N65 R378 N381 R382 R389 D412 N413 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 D 2.17 BS01 dna G 0 R30 N33 R34 R41 D64 N65 R353 N356 R357 R364 D387 N388 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 VIWINGDKGYNGLAEVGKKFVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zd4 D 2.17 BS02 dna H 0 R36 E37 R40 K61 H62 R359 E360 R363 K384 H385 ? 0008643,0015144,0015768,0030288,0034219,0042597,0042956,0055052,0055085,1901982 remove_due_to_license_issue P0AEY0,Q8S307 30287951 -3 ~ 11 VIWINGDKGYNGLAEVGKKFVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDAALAAAQTNAARRKPSWRERENNRRRERRRRAVAAKIYTGLRAQGDYNLPKHCDNNEVLKALCVEAGWVVEEDGTTYR 5zdb A 1.972 BS01 AR6 A 1 T73 T74 F93 S95 G101 A109 Q110 E111 D113 A222 G224 G226 V227 F228 L259 T45 T46 F65 S67 G73 A81 Q82 E83 D85 A194 G196 G198 V199 F200 L231 ? remove_due_to_license_issue Q9RZM4 30940816 301 VRLPGLAAMRQGTRLFTPEQGEDLREALRRRRGSFQTTCEVTSETTFAAARRLREKASALAALNFASAKNPGGGFLGGAQAQEEDLCRGSGLYFSLTSPQAEPYYAVNRQSHSALYTDHLIYSPQVPIFRDDAGQLLPAPVPVNIITAPAPNAGAVAQSRPEQLPQVLPTLRERARRVLGVAAWMEQTHLVLGAWGCGVFRNDPAGVARTFRELLEGEAQGAFEHVTFAVLDNHPQHPTLGAFRRELESLCLP 5zdc C 1.979 BS01 AR6 C 1 T73 T74 F93 S95 A109 Q110 E111 D113 A222 G224 G226 V227 F228 L259 T45 T46 F65 S67 A81 Q82 E83 D85 A194 G196 G198 V199 F200 L231 ? remove_due_to_license_issue Q9RZM4 30940816 301 VRLPGLAAMRQGTRLFTPEQGEDLREALRRRRGSFQTTCEVTSETTFAAARRLREKASALAALNFASAKNPGGGFLGGAQAQEEDLCRGSGLYFSLTSPQAEPYYAVNRQSHSALYTDHLIYSPQVPIFRDDAGQLLPAPVPVNIITAPAPNAGAVAQSRPEQLPQVLPTLRERARRVLGVAAWMEQTHLVLGAWGCGVFRNDPAGVARTFRELLEGEAQGAFEHVTFAVLDNHPQHPTLGAFRRELESLCLP 5zdd A 2.725 BS01 AR6 A 1 T73 T74 F93 S95 A109 Q110 E111 D113 A222 G224 G226 V227 F228 L259 T45 T46 F65 S67 A77 Q78 E79 D81 A190 G192 G194 V195 F196 L227 ? remove_due_to_license_issue Q9RZM4 30940816 301 VRLPGLAAMRQGTRLFTPEQGEDLREALRRRRGSFQTTCEVTSETTFAAARRLREKASALAALNFASAKNPGGGFQAQEEDLCRGSGLYFSLTSPQAEPYYAVNRQSHSALYTDHLIYSPQVPIFRDDAGQLLPAPVPVNIITAPAPNAGAVAQSRPEQLPQVLPTLRERARRVLGVAAWMEQTHLVLGAWGCGVFRNDPAGVARTFRELLEGEAQGAFEHVTFAVLDNHPQHPTLGAFRRELESLCL 5zde C 2.8 BS01 AR6 C 1 T73 T74 F93 S95 A109 Q110 D113 A222 G224 G226 V227 F228 L259 T45 T46 F65 S67 A78 Q79 D82 A191 G193 G195 V196 F197 L228 ? remove_due_to_license_issue Q9RZM4 30940816 301 VRLPGLAAMRQGTRLFTPEQGEDLREALRRRRGSFQTTCEVTSETTFAAARRLREKASALAALNFASAKNPGGGFAQAQEEDLCRGSGLYFSLTSPQAEPYYAVNRQSHSALYTDHLIYSPQVPIFRDDAGQLLPAPVPVNIITAPAPNAGAVAQSRPEQLPQVLPTLRERARRVLGVAAWMEQTHLVLGAWGCGVFRNDPAGVARTFRELLEGEAQGAFEHVTFAVLDNHPQHPTLGAFRRELESLC 5zdf A 2.504 BS01 AR6 A 1 T73 T74 F93 S95 A109 Q110 E111 E112 D113 A222 G224 C225 G226 V227 F228 L259 K267 T45 T46 F65 S67 A78 Q79 E80 E81 D82 A191 G193 C194 G195 V196 F197 L228 K236 ? remove_due_to_license_issue Q9RZM4 30940816 301 VRLPGLAAMRQGTRLFTPEQGEDLREALRRRRGSFQTTCEVTSETTFAAARRLREKASALAALNFASAKNPGGGFAQAQEEDLCRGSGLYFSLTSPQAEPYYAVNRQSHSALYTDHLIYSPQVPIFRDDAGQLLPAPVPVNIITAPAPNAGAVAQSRPEQLPQVLPTLRERARRVLGVAAWMEQTHLVLGAWGCGVFRNDPAGVARTFRELLEGEAQGAFEHVTFAVLDNHPQHPKLGAFRRELESLC 5zdg C 2.594 BS01 AR6 C 1 T73 T74 F93 S95 A109 Q110 D113 A222 G224 C225 G226 V227 F228 L259 R267 T45 T46 F65 S67 A78 Q79 D82 A191 G193 C194 G195 V196 F197 L228 R236 ? remove_due_to_license_issue Q9RZM4 30940816 301 VRLPGLAAMRQGTRLFTPEQGEDLREALRRRRGSFQTTCEVTSETTFAAARRLREKASALAALNFASAKNPGGGFAQAQEEDLCRGSGLYFSLTSPQAEPYYAVNRQSHSALYTDHLIYSPQVPIFRDDAGQLLPAPVPVNIITAPAPNAGAVAQSRPEQLPQVLPTLRERARRVLGVAAWMEQTHLVLGAWGCGVFRNDPAGVARTFRELLEGEAQGAFEHVTFAVLDNHPQHPRLGAFRRELESLC 5ze6 A 2.5 BS01 HJX A 1 H77 T80 L81 D84 D113 Y116 E146 H77 T80 L81 D84 D113 Y116 E146 2.5.1.90 0004659,0005515,0005829,0006744,0008299,0016094,0016740,0042802,0042803,0046872,0106350 remove_due_to_license_issue P0AD57 30730737 401 MNLEKINELTAQDMAGVNAAILEQLNSDVQLINQLGYYIVSGGGKRIRPMIAVLAARAVGYEGNAHVTIAALIEFIHTATLLHDDVVDESDMRRGKATANAAFGNAASVLVGDFIYTRAFQMMTSLGSLKVLEVMSEAVNVIAEGEVLQLMNVNDPDITEENYMRVIYSKTARLFEAAAQCSGILAGCTPEEEKGLQDYGRYLGTAFQLIDDLLDYNADGNVGDDLNEGKPTLPLLHAMHHGTPEQAQMIRTAIEQGNGRHLLEPVLEAMNACGSLEWTRQRAEEEADKAIAALQVLPDTPWREALIGLAHIAVQ 5ze6 C 2.5 BS01 HJX A 1 D113 Y116 D101 Y104 2.5.1.90 0004659,0005515,0005829,0006744,0008299,0016094,0016740,0042802,0042803,0046872,0106350 remove_due_to_license_issue P0AD57 30730737 401 MNLEKINELTAQDMAGVNAAILEQLNSDVQLINQLGYYIVSGGGKRIRPMIAVLAARAVGYEGNAHVTIAALIEFIHTATLLHDDVVDESFGNAASVLVGDFIYTRAFQMMTSLGSLKVLEVMSEAVNVIAEGEVLQLMNVNDPDITEMRVIYSKTARLFEAAAQCSGILAGCTPEEEKGLQDYGRYLGTAFQLIDDLLDYNVGDDLNEGKPTLPLLHAMHHGTPEQAQMIRTAIEQGNGRHLLEPVLEAMNACGSLEWTRQRAEEEADKAIAALQVLPDTPWREALIGLAHIAVQR 5zee A 1.74 BS01 HAR A 1 D124 H126 D128 N130 S137 H141 G142 D225 D124 H126 D128 N130 S137 H141 G142 D225 3.5.3.1 0000050,0004053,0005737,0005829,0006525,0016787,0019547,0030145,0042802,0046872 remove_due_to_license_issue C4LSS0 31199070 301 MQFEKVTYIAVPQKYGQKKVGVEEGPKFLEKLGFMNVLEQVAKSVNKKTITEPKTPQELGVTNARNLNEVESVNIELRDTIAKEYDVNNLLINIGGDHSIGLGTIAGVVKAMKPNARVGVVWFDAHPDMNTPENSPSGNIHGMPLACAVGLGPQRLTSIMPHYITPKDIMYVGIRSIDVGEQFEIQDKHIDHFTAEDVKRVGMKEVIEAINKKFVDYDVIHLSFDIDGIDPEFILGTGTPVPKGISLEDSLYFMSEMGKMKKLHSVDIVEYNPKIEEEITGKNVLKCISSLFGIK 5zef A 2.01 BS01 NVA A 1 N130 S137 H141 D178 N130 S137 H141 D178 3.5.3.1 0000050,0004053,0005737,0005829,0006525,0016787,0019547,0030145,0042802,0046872 remove_due_to_license_issue C4LSS0 31199070 301 MQFEKVTYIAVPQKYGQKKVGVEEGPKFLEKLGFMNVLEQVAKSVNKKTITEPKTPQELGVTNARNLNEVESVNIELRDTIAKEYDVNNLLINIGGDHSIGLGTIAGVVKAMKPNARVGVVWFDAHPDMNTPENSPSGNIHGMPLACAVGLGPQRLTSIMPHYITPKDIMYVGIRSIDVGEQFEIQDKHIDHFTAEDVKRVGMKEVIEAINKKFVDYDVIHLSFDIDGIDPEFILGTGTPVPKGISLEDSLYFMSEMGKMKKLHSVDIVEYNPKIEEEITGKNVLKCISSLFGI 5zeq A 1.9 BS04 9B3 A 1 H69 E72 R127 N144 R145 S207 Y248 A250 G253 D255 E270 H64 E67 R122 N139 R140 S203 Y244 A246 G249 D251 E266 H69 E72 R127 H196 E270 H64 E67 R122 H192 E266 3.4.17.2 0004181,0006508,0008270 remove_due_to_license_issue P09955 29859906 406 GHSYEKYNNWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREWISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTNAGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAYLTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAGGSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL 5zfi A 1.8 BS01 9C9 A 1 H57 F151 T190 C191 N192 G193 S195 S214 W215 G216 T217 C220 H41 F130 T171 C172 N173 G174 S176 S191 W192 G193 T194 C197 H57 D102 N192 G193 D194 S195 H41 D83 N173 G174 D175 S176 3.4.21.117 0001533,0002803,0004252,0005576,0005615,0006508,0008233,0008236,0097209 ic50=1.2uM remove_due_to_license_issue Q91VE3 29884582 301 IIDGYKCKEGSHPWQVALLKGNQLHCGGVLVDKYWVLTAAHCKMGQYQVQLGSDKIGDQSAQKIKATKSFRHPGYSTKTHVNDIMLVRLDEPVKMSSKVEAVQLPEHCEPPGTSCTVSGWGTTTSPDVTFPSDLMCSDVKLISSRECKKVYKDLLGKTMLCAGIPDSKTNTCNGDSGGPLVCNDTLQGLVSWGTYPCGQPNDPGVYTQVCKYKRWVMETMKTHR 5zfw A 2.103 BS01 dna D 0 R20 R21 R23 L24 W26 R62 N69 R73 R95 F118 R124 Q139 R146 R2 R3 R5 L6 W8 R44 N51 R55 R68 F91 R97 Q112 R119 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 GRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5zfw A 2.103 BS02 dna E 0 R20 R23 Y43 R49 Q64 R71 R79 R95 R96 R98 T99 R137 W141 N144 R148 R2 R5 Y25 R31 Q46 R53 R61 R68 R69 R71 T72 R110 W114 N117 R121 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 GRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5zfy A 2.3 BS01 dna D 0 R20 R21 R23 L24 W26 R62 N69 R73 R95 F118 R124 R146 R3 R4 R6 L7 W9 R45 N52 R56 R69 F92 R98 R120 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 RGRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5zfy A 2.3 BS02 dna E 0 R20 R23 Y43 R71 R79 R95 R96 R98 T99 R137 W141 N144 R148 R3 R6 Y26 R54 R62 R69 R70 R72 T73 R111 W115 N118 R122 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 RGRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5zfz A 1.9 BS01 dna D 0 R20 R21 R23 W26 R62 N69 R73 R95 F118 R124 R146 R2 R3 R5 W8 R44 N51 R55 R68 F91 R97 R119 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 GRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5zfz A 1.9 BS02 dna E 0 R20 R23 Y43 R71 R95 R96 R98 T99 R137 W141 N144 R148 R2 R5 Y25 R53 R68 R69 R71 T72 R110 W114 N117 R121 ? 0003677 remove_due_to_license_issue Q9UBX2 30322619 1 ~ 19 GRRRRLVWTPSQSEALRACFERNPYPGIATRERLAQAIGIPEPRVQIWFQNERSRQLRQHRRESPEGRRKRTAVTGSQTALLLRAFEKDRFPGIAAREELARETGLPESRIQIWFQNRRARH 5zh2 A 2.66 BS02 9CU A 1 E332 H338 N339 F342 E500 V501 L502 L555 R559 E250 H256 N257 F260 E401 V402 L403 L438 R442 R330 E332 T337 H338 E500 N503 R559 R248 E250 T255 H256 E401 N404 R442 6.1.1.6 0000049,0000166,0003676,0004812,0004824,0005524,0005737,0005829,0006418,0006430 remove_due_to_license_issue W7JP72 29779382 602 EVDPRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAGGANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKNQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMIPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRP 5zh3 A 2.86 BS02 9CF A 1 H338 N339 F342 E500 V501 L555 R559 H246 N247 F250 E408 V409 L443 R447 R330 E332 T337 H338 E500 N503 R559 R238 E240 T245 H246 E408 N411 R447 6.1.1.6 0000049,0000166,0003676,0004812,0004824,0005524,0005737,0005829,0006418,0006430 remove_due_to_license_issue W7JP72 29779382 602 PRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKDSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRP 5zh4 A 2.6 BS02 9CC A 1 E332 H338 N339 F342 V501 L502 R559 E251 H257 N258 F261 V413 L414 R450 R330 E332 T337 H338 E500 N503 R559 R249 E251 T256 H257 E412 N415 R450 6.1.1.6 0000049,0000166,0003676,0004812,0004824,0005524,0005737,0005829,0006418,0006430 remove_due_to_license_issue W7JP72 29779382 602 EVDPRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAGGANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKEAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRP 5zh5 A 3.08 BS02 9CX A 1 T337 H338 N339 F342 V501 G556 R559 T254 H255 N256 F259 V418 G457 R460 R330 E332 T337 H338 E500 N503 R559 R247 E249 T254 H255 E417 N420 R460 6.1.1.6 0000049,0000166,0003676,0004812,0004824,0005524,0005737,0005829,0006418,0006430 remove_due_to_license_issue W7JP72 29779382 602 EVDPRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKYGLTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFLDSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRP 5zhj A 1.75 BS01 SAH A 1 P83 T84 P85 G109 E112 S132 I133 L138 G140 G141 P83 T84 P85 G109 E112 S132 I133 L138 G140 G141 P85 E112 R154 P85 E112 R154 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=10.1uM remove_due_to_license_issue Kd=10100nM P9WFY7 31442049 301 MRIDIVTIFPACLDPLRQSLPGKAIESGLVDLNVHDLRRWTHDVHHSVDDAPYGGGPGMVMKAPVWGEALDEICSSETLLIVPTPAGVLFTQATAQRWTTESHLVFACGRYEGIDQRVVQDAARRMRVEEVSIGDYVLPGGESAAVVMVEAVLRLLAGVLGPSYTRPASWRGLDVPEVLLSGDHARIAAWRREVSLQRTRERRPDL 5zk3 A 2.6 BS01 QNB A 1 D103 Y104 S107 N108 F181 A191 A194 W400 Y403 N404 Y426 D86 Y87 S90 N91 F164 A174 A177 W322 Y325 N326 Y348 ? 0004930,0005506,0005886,0007186,0009055,0016020,0016907,0020037,0022900,0042597,0046872 remove_due_to_license_issue P08172,P0ABE7 30420692 501 YKTFEVVFIVLVAGSLSLVTIIGNILVMVSIKVNRHLQTVNNYFLFSLACADLIIGVFSMNLYTLYTVIGYWPLGPVVCDLWLALDYVVSNARVMNLLIISFDRYFCVTKPLTYPVKRTTKMAGMMIAAAWVLSFILWAPAILFWQFIVGVRTVEDGECYIQFFSNAAVTFGTAIAAFYLPVIIMTVLYWHISRASKADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLEKKVTRTILAILLAFIITWAPYNVMVLINTFCAPCIPNTVWTIGYWLCYINSTINPACYALCNATFKKTFKHLLMCH 5zk8 A 3.0 BS01 3C0 A 1 D103 Y104 S107 N108 W155 A191 W400 Y403 N404 Y426 C429 D86 Y87 S90 N91 W138 A174 W311 Y314 N315 Y337 C340 ? 0004930,0005506,0005886,0007186,0009055,0016020,0016907,0020037,0022900,0042597,0046872 remove_due_to_license_issue P08172,P0ABE7 30420692 501 YKTFEVVFIVLVAGSLSLVTIIGNILVMVSIKVNRHLQTVNNYFLFSLACADLIIGVFSMNLYTLYTVIGYWPLGPVVCDLWLALDYVVSNASVMNLLIISFDRYFCVTKPLTYPVKRTTKMAGMMIAAAWVLSFILWAPAILFWQFIVGVRTVEDGECYIQFFSNAAVTFGTAIAAFYLPVIIMTVLYWHISRASKADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLKKVTRTILAILLAFIITWAPYNVMVLINTFCAPCIPNTVWTIGYWLCYINSTINPACYALCNATFKKTFKHLLMCH 5zkb A 2.95 BS01 82F A 1 W99 L100 D103 Y104 S107 N108 V111 A191 W400 Y403 N404 Y426 C429 Y430 W83 L84 D87 Y88 S91 N92 V95 A175 W325 Y328 N329 Y351 C354 Y355 ? 0004930,0005506,0005886,0007186,0009055,0016020,0016907,0020037,0022900,0042597,0046872 remove_due_to_license_issue P08172,P0ABE7 30420692 1201 PYKTFEVVFIVLVAGSLSLVTIIGNILVMVSIKVNRHLQTVNNYFLFSLACADLIIGVFSMNLYTLYTVIGYWPLGPVVCDLWLALDYVVSNARVMNLLIISFDRYFCVTKPLTYPVKRTTKMAGMMIAAAWVLSFILWAPAILFWQFIVGVRTVEDGECYIQFFSNAAVTFGTAIAAFYLPVIIMTVLYWHISRASKSRIADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLPPPSREKKVTRTILAILLAFIITWAPYNVMVLINTFCAPCIPNTVWTIGYWLCYINSTINPACYALCNATFKKTFKHLLM 5zkc A 2.3 BS01 3C0 A 1 D103 Y104 S107 N108 A191 A194 W400 Y403 N404 Y426 C429 D88 Y89 S92 N93 A176 A179 W326 Y329 N330 Y352 C355 ? 0004930,0005506,0005886,0007186,0009055,0016020,0016907,0020037,0022900,0042597,0046872 Kd=6.4nM remove_due_to_license_issue P08172,P0ABE7 30420692 501 SPYKTFEVVFIVLVAGSLSLVTIIGNILVMVSIKVNRHLQTVNNYFLFSLACADLIIGVFSMNLYTLYTVIGYWPLGPVVCDLWLALDYVVSNARVMNLLIISFDRYFCVTKPLTYPVKRTTKMAGMMIAAAWVLSFILWAPAILFWQFIVGVRTVEDGECYIQFFSNAAVTFGTAIAAFYLPVIIMTVLYWHISRASKADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLSREKKVTRTILAILLAFIITWAPYNVMVLINTFCAPCIPNTVWTIGYWLCYINSTINPACYALCNATFKKTFKHLLMCH 5zki A 2.321 BS01 dna C 0 R109 S137 R138 G139 A144 G145 F168 N171 S172 N176 Y310 R314 R52 S80 R81 G82 A87 G88 F111 N114 S115 N119 Y253 R257 C112 A140 N162 N171 E179 C55 A83 N105 N114 E122 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 EKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKAK 5zki A 2.321 BS02 dna D 0 S172 L311 K315 R320 R324 S115 L254 K258 R263 R267 C112 A140 N162 N171 E179 C55 A83 N105 N114 E122 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 EKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKAK 5zki B 2.321 BS01 dna E 0 R109 S137 R138 G139 A140 A144 G145 F168 N171 S172 N176 L311 R314 R53 S81 R82 G83 A84 A88 G89 F112 N115 S116 N120 L255 R258 C112 A140 N162 N171 E179 C56 A84 N106 N115 E123 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 AEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKAKEQS 5zki B 2.321 BS02 dna F 0 K113 S172 L311 K315 R320 R324 K57 S116 L255 K259 R264 R268 C112 A140 N162 N171 E179 C56 A84 N106 N115 E123 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 AEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKAKEQS 5zkj A 2.798 BS01 rna E 0 R109 K110 S137 R138 A144 G145 K148 F168 N171 S172 N176 R183 R314 R54 K55 S82 R83 A89 G90 K93 F113 N116 S117 N121 R128 R259 C112 A140 N162 N171 E179 C57 A85 N107 N116 E124 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 SAEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLE 5zkj A 2.798 BS02 dna F 0 K115 S172 L311 R320 R324 K327 K60 S117 L256 R265 R269 K272 C112 A140 N162 N171 E179 C57 A85 N107 N116 E124 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 SAEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLE 5zkj B 2.798 BS01 rna C 0 R109 K110 S137 R138 G139 A140 A144 G145 K148 F168 N171 S172 N176 L311 R314 R54 K55 S82 R83 G84 A85 A89 G90 K93 F113 N116 S117 N121 L256 R259 C112 A140 N162 N171 E179 C57 A85 N107 N116 E124 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 SAEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKAKE 5zkj B 2.798 BS02 dna D 0 K115 S172 L311 K315 R320 K60 S117 L256 K260 R265 C112 A140 N162 N171 E179 C57 A85 N107 N116 E124 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 12 SAEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEELKAKE 5zkl A 1.951 BS01 dna B 0 F12 W30 F39 M58 G59 K60 T63 F2 W20 F29 M48 G49 K50 T53 ? 0003677,0006355 remove_due_to_license_issue Q8DQG2 31713614 1 ~ 5 EFTFEIEEHLLTLSENEKGWTKEINRVSFNGAPAKFDIRAWSPDHTKMGKGITLSNEEFQTMVDAF 5zku A 2.32 BS01 9F3 A 1 S84 E210 F256 P257 R258 Q391 S83 E208 F254 P255 R256 Q389 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 PSNNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPAGGADSAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSCFEAQVDALLATEAADLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTVG 5zku A 2.32 BS02 9F3 C 1 D177 D199 D175 D197 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 PSNNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPAGGADSAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSCFEAQVDALLATEAADLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTVG 5zku B 2.32 BS01 9F3 A 1 D177 D199 D175 D197 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 SNNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPAGGAGDSAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSCFEAQVDALLATEAADLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTVG 5zku B 2.32 BS02 9F3 B 1 S84 E210 F256 P257 R258 F281 W309 Q391 S82 E208 F254 P255 R256 F279 W307 Q389 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 SNNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPAGGAGDSAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSCFEAQVDALLATEAADLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTVG 5zla A 1.7 BS01 9F3 A 1 S84 E210 F256 P257 R258 F281 W309 S83 E209 F255 P256 R257 F280 W308 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 PSNNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPAGGAGDSAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSAFEAQVDALLATDLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTV 5zla A 1.7 BS02 9F3 B 1 D177 D199 D176 D198 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 PSNNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPAGGAGDSAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSAFEAQVDALLATDLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTV 5zla D 1.7 BS01 9F3 A 1 D177 D199 D169 D191 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 NNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPASAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSAFEAQVDALLATEAADLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTVGF 5zla D 1.7 BS02 9F3 D 1 S84 E210 F256 P257 R258 F281 W309 Q391 S81 E202 F248 P249 R250 F273 W301 Q383 4.2.2.17 0016740,0016829,0033997 remove_due_to_license_issue B8HDZ1 501 NNRYDVTEWPAGNPAKDIGEVINSIIADIKARQGAADVDDGGKPGAVIYLPPGDYHLRTQVLIDISFLRIEGSGHGFTSSSIRFNVPEEEWPDLHELWPGGSRVIVDLPASAAGAAFLVAREGSPRISSVEFSNFCIDGLHFTADGSGRHPENTYANGKTGIHVASANDSFRVTDMGFVYLENALTIHKADALSIHHNFIAECGSCIELRGWGQASKITDNLVGAGPRGHSIYAENHGGLLVTANNVFPRGASSVHFKGVTRSSVTNNRLHAFYPGMVRLEENSSENLVATNHFLRDHEPWTPFFGVDNGLDDLTGLLSISGNNNSVIGNHFSEVVDANEIRPEGATPVIIRLTAGTGNFVSTNHVVAMDVDAASSDSAFEAQVDALLATEAADLAVTAVLVDPGSARNTILDSGSDTQVVADRAVNAIRATPTVGF 5zlf A 2.845 BS01 B29 A 1 T80 D84 R93 I142 A143 E146 T79 D83 R92 I141 A142 E145 2.5.1.90 0004659,0005515,0005829,0006744,0008299,0016094,0016740,0042802,0042803,0046872,0106350 remove_due_to_license_issue P0AD57 30730737 901 NLEKINELTAQDMAGVNAAILEQLNSDVQLINQLGYYIVSGGGKRIRPMIAVLAARAVGYEGNAHVTIAALIEFIHTATLLHDDVVDESDMRRGKATANAAFGNAASVLVGDFIYTRAFQMMTSLGSLKVLEVMSEAVNVIAEGEVLQLMNVNITEENYMRVIYSKTARLFEAAAQCSGILAGCTPEEEKGLQDYGRYLGTAFQLIDDLLDYNNVGDDLNEGKPTLPLLHQAQMIRTAIEQGNGRHLLEPVLEAMEWTRQRAEEEADKAIAALQVLPDTPWREALIGLAHIAV 5zlf B 2.845 BS01 B29 A 1 L110 D113 L94 D97 2.5.1.90 0004659,0005515,0005829,0006744,0008299,0016094,0016740,0042802,0042803,0046872,0106350 remove_due_to_license_issue P0AD57 30730737 901 MNLEKINELTAQDMAGVNAAILEQLNSDVQLINQLGYYIVSGGGKRIRPMIAVLAARAVGYEGNAHVTIAALIEFIHTATLLHDDVFGNAASVLVGDFIYTRAFQMMTSLGSLKVLEVMSEAVNVIAEGEVLQLMNVNDPDITEENYMRVIYSKTARLFEAAAQCSGILAGCTPEEEKGLQDYGRYLGTAFQLIDDLLLNEGKPTLPLRHLLEPVLEAMNACEWTRQRAEEEADKAIAALQVDTPWREALIGLAHIAVQ 5zmd A 3.3 BS01 dna B 0 I85 K86 K88 P93 R96 Y108 L109 N110 P213 Y214 K216 S229 W230 H231 E234 I49 K50 K52 P57 R60 Y72 L73 N74 P147 Y148 K150 S163 W164 H165 E168 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAAKEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQ 5zmd A 3.3 BS02 dna D 0 Y214 S277 W278 K306 Y148 S194 W195 K223 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAAKEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQ 5zmd C 3.3 BS01 dna B 0 K88 S277 W278 K306 K52 S192 W193 K221 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAADEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQ 5zmd C 3.3 BS02 dna D 0 I85 K86 K88 P93 R96 Y108 L109 K216 M226 V228 S229 W230 H231 E234 R459 T463 I49 K50 K52 P57 R60 Y72 L73 K149 M159 V161 S162 W163 H164 E167 R355 T359 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAADEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQ 5zmd E 3.3 BS01 dna F 0 I85 K86 K88 L90 P93 R96 Y108 L109 N110 K216 M226 V228 S229 H231 E234 R459 I460 I49 K50 K52 L54 P57 R60 Y72 L73 N74 K145 M155 V157 S158 H160 E163 R356 I357 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKKHTEAEIAAACETFLKLNDYLQIETIQALEELAAVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRG 5zmd E 3.3 BS02 dna H 0 S277 W278 K306 S189 W190 K218 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKKHTEAEIAAACETFLKLNDYLQIETIQALEELAAVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRG 5zmd G 3.3 BS01 dna F 0 Y214 W278 K306 Y150 W196 K224 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAAKDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQ 5zmd G 3.3 BS02 dna H 0 I85 K86 K88 L90 P93 R96 Y108 L109 N110 P213 Y214 L215 K216 V228 S229 W230 H231 E234 I49 K50 K52 L54 P57 R60 Y72 L73 N74 P149 Y150 L151 K152 V164 S165 W166 H167 E170 1.14.11.-,1.14.11.53 0001659,0005634,0005654,0005737,0005829,0005886,0006307,0008198,0010883,0016180,0016607,0016706,0016740,0035515,0035516,0040014,0042245,0043231,0044065,0046872,0051213,0060612,0061157,0070350,0090335,1990931,1990984 remove_due_to_license_issue Q9C0B1 30718435 2 ~ 10 EFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIKGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGSNIKHTEAEIAAACETFLKLNDYLQIETIQALEELAAKDEVDIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHKHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQ 5zmo A 1.69 BS01 dna B 0 H116 R117 Y164 P165 R190 R191 H23 R24 Y71 P72 R97 R98 ? remove_due_to_license_issue Q9L0M9 30409991 1 ~ 7 PKTFHRRVGDVRPARRAMGPALHRPVLLLWAIGQAVARAPRLQPWSTTRDAVAPLMEKYGQVEDGVDGVRYPFWALVRDDLWCVEQAEELTLTSRGRRPTLESLNAVDPSAGLREDDYNLLRSQPEAAASAAAGLIARYFHLLPAGLLEDFGLHELLA 5zmo A 1.69 BS02 dna C 0 A107 R108 T186 S187 R188 R190 R191 T193 L194 A14 R15 T93 S94 R95 R97 R98 T100 L101 ? remove_due_to_license_issue Q9L0M9 30409991 2 ~ 8 PKTFHRRVGDVRPARRAMGPALHRPVLLLWAIGQAVARAPRLQPWSTTRDAVAPLMEKYGQVEDGVDGVRYPFWALVRDDLWCVEQAEELTLTSRGRRPTLESLNAVDPSAGLREDDYNLLRSQPEAAASAAAGLIARYFHLLPAGLLEDFGLHELLA 5znc A 1.66 BS01 QI9 A 1 V66 S91 C92 G93 Y160 V181 E182 M183 D218 V63 S88 C89 G90 Y157 V178 E179 M180 D215 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006166,0006218,0009116,0016757,0047975 Kd=65nM remove_due_to_license_issue Q8T9Z7 30602534 301 LLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKWDEGDFDNNLVPHQLENMIKIALGACAKLATKYA 5zni A 2.3 BS01 YMZ A 1 C92 G93 Y160 V181 M183 D206 G207 C208 C90 G91 Y158 V179 M181 D204 G205 C206 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006166,0006218,0009116,0016757,0047975 Kd=11uM remove_due_to_license_issue Q8T9Z7 30602534 302 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVVEMELATLMVIGTLRKVKTGGILIVDGCPFKHQLENMIKIALGACAKLATKYA 5zo7 A 2.6 BS02 5C5 A 1 E116 G117 E118 R119 Y211 L214 E215 E97 G98 E99 R100 Y192 L195 E196 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=14nM P52732 31459302 602 MKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTDKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 5zo8 A 2.2 BS02 4C5 A 1 E116 G117 E118 R119 A133 P137 Y211 L214 E95 G96 E97 R98 A112 P116 Y190 L193 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=22nM, IC50=28.5nM, EC50=230nM P52732 31459302 602 MKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVNQ 5zo9 A 2.7 BS02 4C5 A 1 E116 G117 E118 I136 P137 Y211 L214 E95 G96 E97 I115 P116 Y190 L193 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue Ki=22nM, IC50=28.5nM, EC50=230nM P52732 31459302 602 MKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVNQ 5zt1 A 3.114 BS02 AGS A 1 G162 G164 K165 T166 F167 F339 Y412 G82 G84 K85 T86 F87 F255 Y313 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 remove_due_to_license_issue P0A1C1 30013545 502 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5ztm A 2.899 BS01 rna C 0 D2 K4 S5 Y8 E17 K28 N29 F33 T51 N52 K53 K54 K58 K171 E172 N175 E195 H196 R198 F200 S222 N223 K224 K225 D2 K4 S5 Y8 E17 K28 N29 F33 T51 N52 K53 K54 K58 K92 E93 N96 E116 H117 R119 F121 S143 N144 K145 K146 3.6.4.13 0003725 remove_due_to_license_issue P24785 30649456 114 ~ 168 MDIKSFLYQFCAKSQIEPKFDIRQTGPKNRQRFLCEVRVEPNTYIGVGNSTNKKDAEKNACRDFVNYLVRVGKLNTNDVPAIHGNWTIENAKERLNIYKQTNNIRDDYKYTPVGPEHARSFLAELSIYVPALNRTVTARESGSNKKSASKSCALSLVRQLFHLNVIEP 5ztm B 2.899 BS01 rna C 0 D2 K4 S5 Y8 F33 N52 K53 E168 E172 E195 H196 F200 S222 N223 K224 K229 D2 K4 S5 Y8 F33 N52 K53 E85 E89 E112 H113 F117 S139 N140 K141 K146 3.6.4.13 0003725 remove_due_to_license_issue P24785 30649456 114 ~ 168 MDIKSFLYQFCAKSQIEPKFDIRQTGPKNRQRFLCEVRVEPNTYIGVGNSTNKKDAEKNACRDFVNYLVRVGKLNTNDVPAWTIENAKERLNIYKQTNNIRDDYKYTPVGPEHARSFLAELSIYVPALNRTVTARESGSNKKSASKSCALSLVRQLFHLNVIEP 5ztn A 2.496 BS01 CUR A 1 K153 F160 A176 K178 E193 I212 F228 L230 L231 L282 I294 D295 K94 F101 A117 K119 E134 I153 F169 L171 L172 L223 I235 D236 D275 K277 N280 D295 S312 D216 K218 N221 D236 S253 2.7.12.1 0004672,0004712,0005524,0006468 ic50=5nM remove_due_to_license_issue Q92630 29987021 501 GVDLGTENLYFQSMGKVKATPMTPEQAMKQYMQKLTAFEHHEIFSYPEIYFLGLNAKKRQGMTGGPNNGGYDDDQGSYVQVPHDHVAYRYEVLKVIGKGSFGQVVKAYDHKVHQHVALKMVRNEKRFHRQAAEEIRILEHLRKQDKDNTMNVIHMLENFTFRNHICMTFELLSMNLYELIKKNKFQGFSLPLVRKFAHSILQCLDALHKNRIIHCDLKPENILLKQQGRSGIKVIDFGSSCYEHQRVYTYIQSRFYRAPEVILGARYGMPIDMWSLGCILAELLTGYPLLPGEDEGDQLACMIELLGMPSQKLLDASKRAKNFVSSKGYPRYCTVTVLNGGRSRRGKLRGPPESREWGNALKGCDDPLFLDFLKQCLEWDPAVRMTPGQALRHPWLR 5zu0 A 2.76 BS01 SAH A 1 T135 G170 G172 E200 A201 N205 Q257 E258 F259 T53 G88 G90 E118 A119 N123 Q175 E176 F177 2.1.1.320 remove_due_to_license_issue Q54S83 30134162 501 KYPITDFEKYLQDITKVRGPMSIDTFIKEVLTNPKYGYYMNKDVFGKGGDFITAPEVSQLFGEMIGIWCVATWEAMGKPKKLQIVEMGPGRGTLMKDILRSTKVFKEFYDSISVHLVEASPANKKTQKQNLLYFKDKAINFDHKTIGETPNGIKVTWVGKLEEVPTDIPTLFLAQEFFDALPIHVFRFSREKNDWCEVLVDEDITEHGEYYLRFVQSKGPTLMTTAVKHLLPEFGLDGYQVELGLAGLAISQQIANRIDKSGGAALIIDYGYDKIVKSSLQAIRDHEFVDILDKPGTADLSVWVDFQTIRKTVKLLKNKSTAIGPVDQGIFLKEMGIEHRLAQIGRKLDSNEKFEELVMGYKKLVDPKEMGTNYKVITICDKNITPIGFSTSKTYDDEDL 5zun A 1.35 BS01 9JX A 1 G50 A51 E53 R57 H121 S122 M123 I179 S181 S185 E190 V191 Y194 L205 L241 V270 K273 G44 A45 E47 R51 H115 S116 M117 I173 S175 S179 E184 V185 Y188 L199 L235 V264 K267 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 ic50=0.64nM remove_due_to_license_issue IC50=0.640000nM Q99685 30251836 401 PRRTPQSIPYQDLPHLVNADGQYLFCRYWAPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNSVLPNLSSGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTA 5zux A -1.00 BS01 dna B 0 R105 R108 T110 A111 R112 G114 S115 K116 I152 P153 N154 R174 R4 R7 T9 A10 R11 G13 S14 K15 I51 P52 N53 R73 ? remove_due_to_license_issue O34857 30252102 1 ~ 18 GTTRRRRGTARPGSKAAKLREAAIKTLKRHNAAIKSSELQKEIEKESGLEIPNMTTFMQSLIKMYPEVKKPYRGQYILEGEIESLEHHHHHH 5zux A -1.00 BS02 dna C 0 R106 R107 R108 G109 A111 T156 T157 Q160 K171 Y173 R174 R5 R6 R7 G8 A10 T55 T56 Q59 K70 Y72 R73 ? remove_due_to_license_issue O34857 30252102 19 ~ 36 GTTRRRRGTARPGSKAAKLREAAIKTLKRHNAAIKSSELQKEIEKESGLEIPNMTTFMQSLIKMYPEVKKPYRGQYILEGEIESLEHHHHHH 5zva A 2.3 BS01 dna C 0 Y333 K352 P353 W354 G356 K358 Y359 Y144 K163 P164 W165 G167 K169 Y170 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4,Q9HC16 1 ~ 10 ENLYFQGSAMDPPTFTFNFNNEPWVRGRHETYLCFTMEVVKHHSPVSWKRGVFRNQTHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5zva B 2.3 BS01 dna C 0 W-9 V-8 H-4 W277 Y307 Y308 W310 W21 V22 H26 W89 Y119 Y120 W122 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4,Q9HC16 1 ~ 10 YFQGSAMDPPTFTFNFNNEPWVRGRHETYLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5zvb A 2.0 BS01 dna C 0 Y333 P353 W354 G356 K358 Y359 Y140 P160 W161 G163 K165 Y166 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4,Q9HC16 1 ~ 9 YFQGSAMDPPTFTFNFNNEPWVRGRHETYLCFTMEVVKHHSPVSWKRGVFRNQHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5zvb B 2.0 BS01 dna C 0 W-9 V-8 H-4 N240 W277 Y307 Y308 W310 W21 V22 H26 N52 W89 Y119 Y120 W122 3.5.4.38 0003824,0008270,0016787 remove_due_to_license_issue Q8IUX4,Q9HC16 1 ~ 9 YFQGSAMDPPTFTFNFNNEPWVRGRHETYLCFTMEVVKHHSPVSWKRGVFRNQVDPETHCHAERCFLSWFCDDILSPNTNYEVTWYTSWSPCPECAGEVAEFLARHSNVNLTIFTARLYYFWDTDYQEGLRSLSQEGASVEIMGYKDFKYCWENFVYNDDEPFKPWKGLKYNFLFLDSKLQEILE 5zwe A 2.72 BS02 9K0 A 1 L226 V230 S233 R270 S271 S274 W282 H301 L309 L46 V50 S53 R90 S91 S94 W102 H121 L129 ? 0003677,0004879,0006355 remove_due_to_license_issue P13053 29936834 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5zwf A 2.1 BS02 9KR A 1 Y143 S233 R270 S271 S274 W282 V296 H301 H393 Y21 S50 R87 S88 S91 W99 V113 H118 H210 ? 0003677,0004879,0006355 remove_due_to_license_issue P13053 29936834 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5zwh A 2.38 BS03 9N9 A 1 Y143 V230 S233 R270 S271 S274 W282 H301 Y21 V47 S50 R87 S88 S91 W99 H118 ? 0003677,0004879,0006355 ic50=1.9nM remove_due_to_license_issue P13053 29936834 502 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5zwi A 2.4 BS02 9KX A 1 Y143 L223 A227 V230 S233 R270 S271 S274 W282 V296 Y21 L43 A47 V50 S53 R90 S91 S94 W102 V116 ? 0003677,0004879,0006355 ic50=2.3nM remove_due_to_license_issue P13053 29936834 501 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGN 5zxk A 1.96 BS01 H6P A 1 H351 Y352 R412 R418 R469 L471 H55 Y56 R116 R122 R173 L175 ? Kd=3.3uM remove_due_to_license_issue EC50=0.510000nM, IC50=16100nM, Kd=1540nM O00481 30902636 501 GAYNEWKKALFKPADVILDPKTANPILLVSEDQRSVQRAKEPQDLPDNPERFNWHYCVLGCESFISGRHYWEVEVGDRKEWHIGVCSKNVQRKGWVKMTPENGFWTMGLTDGNKYRTLTEPRTNLKLPKPPKKVGVFLDYETGDISFYNAVDGSHIHTFLDVSFSEALYPVFRILTLEPTALTICP 5zz2 A 2.6 BS02 9M0 A 1 L725 A767 I768 Q775 A783 F786 F787 Q817 F820 L181 A223 I224 Q231 A239 F242 F243 Q256 F259 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue IC50=1.4nM O76074 30148362 904 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQGEKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 5zz4 A 2.9 BS01 9M3 A 1 L408 G411 Q412 A428 K430 Y476 M477 N479 G480 D521 N526 L528 L542 S543 Y551 L14 G17 Q18 A34 K36 Y82 M83 N85 G86 D127 N132 L134 L148 S149 Y157 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=0.670000nM Q06187 30216722 701 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVM 5zzw B 2.6 BS01 SAH B 1 Y121 F133 T135 G170 P171 G172 E200 N205 Q257 F259 Y39 F51 T53 G88 P89 G90 E118 N123 Q175 F177 2.1.1.320 remove_due_to_license_issue Q54S83 30134162 501 KYPITDFEKYLQDITKVRGPMSIDTFIKEVLTNPKYGYYMNKDVFGKGGDFITAPEVSQLFGEMIGIWCVATWEAMGKPKKLQIVEMGPGRGTLMKDILRSTKVFKEFYDSISVHLVEASPANKKTQKQNLLYFKDKAINFDHKTIGETPNGIKVTWVGKLEEVPTDIPTLFLAQEFFDALPIHVFRFSREKNDWCEVLVDEDITEHGEYYLRFVQSKGPTLMTTAVKHLLPEFGLDGYQVELGLAGLAISQQIANRIDKSGGAALIIDYGYDKIVKSSLQAIRDHEFVDILDKPGTADLSVWVDFQTIRKTVKLLKNKSTAIGPVDQGIFLKEMGIEHRLAQIGRKLDSNEKFEELVMGYKKLVDPKEMGTNYKVITICDKNITPIGFSTSKTYDDEDL 6a04 A 1.9 BS01 C2E B 1 S162 Y167 I235 R238 Y240 T263 P264 S12 Y17 I85 R88 Y90 T113 P114 ? 0002218,0032481 remove_due_to_license_issue B8XX90 31167783 402 ANFNVAHGLAWSYYIGYLRLILPGLRARIQAYNQRHKNVLGGIGNHRLHILFPLDCGVPDDLSVADPNIRFLHELPQQSADRAGIKGRVYTNSIYELLENGQPAGVCVLEYATPLQTLFAMSQDGRAGFSREDRLEQAKLFCRTLEDILADAPEAQNNCRLIVYQEPTEGGSFSLSQEILRHLRQEE 6a04 B 1.9 BS01 C2E B 1 S162 Y163 Y167 R238 Y240 T263 S12 Y13 Y17 R80 Y82 T105 ? 0002218,0032481 Kd~6uM remove_due_to_license_issue B8XX90 31167783 402 ANFNVAHGLAWSYYIGYLRLILPGLRARIQAYNQRHKNVLGGIGNHRLHILFPLDCGVPDDLSVADPNIRFLHELPQQGRVYTNSIYELLENGQPAGVCVLEYATPLQTLFAMSQDGRAGFSREDRLEQAKLFCRTLEDILADAPEAQNNCRLIVYQEPTEGGSFSLSQEILRHLRQEEREV 6a2h A 2.3 BS01 dna B 0 K24 W26 L28 A29 P30 K31 R33 L40 K21 W23 L25 A26 P27 K28 R30 L37 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 30499242 106 ~ 111 GKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 6a2h A 2.3 BS02 dna C 0 V36 I38 R51 K53 V33 I35 R48 K50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 30499242 114 ~ 119 GKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 6a2i A 2.4 BS01 dna C 0 K24 W26 L28 A29 P30 K31 K48 Y49 R51 K20 W22 L24 A25 P26 K27 K44 Y45 R47 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 30499242 101 ~ 118 KKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 6a2i A 2.4 BS02 dna D 0 L28 V36 R51 H52 K53 L24 V32 R47 H48 K49 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 30499242 119 ~ 136 KKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 6a2i B 2.4 BS01 dna C 0 K24 W26 L28 A29 P30 Y49 K21 W23 L25 A26 P27 Y46 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 30499242 101 ~ 118 GKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 6a2i B 2.4 BS02 dna D 0 R33 V36 R51 H52 K53 R30 V33 R48 H49 K50 ? 0003677,0003690,0005737 remove_due_to_license_issue Q97ZE3 30499242 119 ~ 136 GKKPVKVKTPAGKEAELVPEKVWALAPKGRKGVKIGLFKDPETGKYFRHKLPDDYPI 6a6j A 2.255 BS01 rna B 0 W45 N47 F54 F65 H67 E97 K98 G99 A100 W13 N15 F22 F33 H35 E65 K66 G67 A68 ? 0003676 remove_due_to_license_issue P67809 31399345 2 ~ 6 KVIATKVLGTVKWFNVRNGYGFINRNDTKEDVFVHQTAIKKNNPRKYLRSVGDGETVEFDVVEGEKGAEAANVTGPGGVPVQGSKYAADR 6a6j C 2.255 BS01 rna D 0 W45 N47 Y52 F54 D63 F65 H67 G99 E101 W13 N15 Y20 F22 D31 F33 H35 G67 E69 ? 0003676 remove_due_to_license_issue P67809 31399345 2 ~ 6 KVIATKVLGTVKWFNVRNGYGFINRNDTKEDVFVHQTAIKKNNPRKYLRSVGDGETVEFDVVEGEKGAEAANVTGPGGVPVQGSKYAADR 6a73 A 2.447 BS01 IHP A 1 K43 K73 K77 S114 K11 K41 K45 S82 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P61201 32047038 401 ENQYYNSKALKEDDPKAALSSFQKVLELEGEKGEWGFKALKQMIKINFKLTNFPEMMNRYKQLLTYIRSAVTRNYSEKSINSILDYISTSKQMDLLQEFYETTLEALKDAKNDRLWFKTNTKLGKLYLERNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAY 6a80 A 1.56 BS01 CYS A 1 A77 R82 H95 A70 R75 H88 ? Kd=0.000000064M remove_due_to_license_issue C6XGT2 31063259 319 SALRVGTDGIYPPHSFHAQDGRGELTGFDIDLIKEVAHRLNLKVEFFETAVSGLITGLDTNRYDVLVNVAITPERQKKYDFSIPYIAHRVLLVVRSDQQDIRSFKDLTDKTVAQILGTDLSRFAKELKSHLVFSHNFEQSLQLLLSKRTDATMIPDIPFFNFLERRPHDGNLFKIADRMKDNSAVAFMMRKGNNKLTRSINEILCAIHLDGTYKKIFDRYFDKNIISSVPGCSS 6a80 A 1.56 BS02 CYS A 2 I62 R82 T125 I55 R75 T118 ? Kd=0.000000064M remove_due_to_license_issue C6XGT2 31063259 320 SALRVGTDGIYPPHSFHAQDGRGELTGFDIDLIKEVAHRLNLKVEFFETAVSGLITGLDTNRYDVLVNVAITPERQKKYDFSIPYIAHRVLLVVRSDQQDIRSFKDLTDKTVAQILGTDLSRFAKELKSHLVFSHNFEQSLQLLLSKRTDATMIPDIPFFNFLERRPHDGNLFKIADRMKDNSAVAFMMRKGNNKLTRSINEILCAIHLDGTYKKIFDRYFDKNIISSVPGCSS 6a80 B 1.56 BS01 CYS B 1 A77 R82 H95 A70 R75 H88 ? Kd=0.000000064M remove_due_to_license_issue C6XGT2 31063259 310 SALRVGTDGIYPPHSFHAQDGRGELTGFDIDLIKEVAHRLNLKVEFFETAVSGLITGLDTNRYDVLVNVAITPERQKKYDFSIPYIAHRVLLVVRSDQQDIRSFKDLTDKTVAQILGTDLSRFAKELKSHLVFSHNFEQSLQLLLSKRTDATMIPDIPFFNFLERRPHDGNLFKIADRMKDNSAVAFMMRKGNNKLTRSINEILCAIHLDGTYKKIFDRYFDKNIISSVPGCSS 6a80 B 1.56 BS02 CYS B 2 R82 T125 D126 R75 T118 D119 ? Kd=0.000000064M remove_due_to_license_issue C6XGT2 31063259 311 SALRVGTDGIYPPHSFHAQDGRGELTGFDIDLIKEVAHRLNLKVEFFETAVSGLITGLDTNRYDVLVNVAITPERQKKYDFSIPYIAHRVLLVVRSDQQDIRSFKDLTDKTVAQILGTDLSRFAKELKSHLVFSHNFEQSLQLLLSKRTDATMIPDIPFFNFLERRPHDGNLFKIADRMKDNSAVAFMMRKGNNKLTRSINEILCAIHLDGTYKKIFDRYFDKNIISSVPGCSS 6a94 A 2.9 BS01 ZOT A 1 W151 D155 S159 L229 V235 G238 S242 W336 F339 F340 W83 D87 S91 L161 V167 G170 S174 W307 F310 F311 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900 remove_due_to_license_issue P0ABE7,P28223 30723326 3001 THLQEKNWSALLTAVVIILTIAGNILVIMAVSLEKKLQNATNYFLMSLAIADMLLGFLVMPVSMLTILYGYRWPLPSKLCAVWIYLDVLFSTAKIWHLCAISLDRYVAIQNPIHHSRFNSRTKAFLKIIAVWTISVGISMPIPVFGLQDDSKVFKEGSCLLADDNFVLIGSFVSFFIPLTIMVITYFLTIKSLQKEAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAGSGSGDILVGQIDDALKLANEGKVKEAQAAAEQLKTTINAYIQKYGQSISNEQKACKVLGIVFFLFVVMWCPFFITNIMAVICKESCNEDVIGALLNVFVWIGYLSSAVNPLVYTLFNKTYRSAFSRYIQCQY 6aa4 A 1.9 BS03 MKS A 1 Y7 F27 F72 F74 M81 W117 D119 G141 Y5 F25 F70 F72 M79 W115 D117 G139 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=0.47uM remove_due_to_license_issue IC50=470nM P36639 30771603 203 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTVLEHHHHHH 6aa5 A 1.901 BS01 MKU A 1 Y7 F27 N33 F72 F74 M81 W117 D119 G141 Y5 F25 N31 F70 F72 M79 W115 D117 G139 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=0.052uM remove_due_to_license_issue P36639 30771603 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTVLEHHHHHH 6aah A 1.83 BS01 9T6 A 1 L881 A906 M956 F958 L959 G962 R1007 N1008 L1010 D1021 L17 A42 M87 F89 L90 G93 R138 N139 L141 D152 D1003 A1005 R1007 N1008 D1021 D134 A136 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=3.9nM P23458 30145050 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6aah B 1.83 BS01 9T6 B 1 L881 A906 M956 E957 F958 L959 G962 R1007 N1008 L1010 L17 A42 M88 E89 F90 L91 G94 R139 N140 L142 D1003 A1005 R1007 N1008 D1021 D135 A137 R139 N140 D153 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=3.9nM P23458 30145050 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6aaj A 2.37 BS01 9T6 A 1 G856 V863 Y931 L932 L983 G14 V21 Y84 L85 L136 D976 R980 N981 D994 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=5.0nM O60674 30145050 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQAHAERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 6aak A 2.67 BS01 9T6 A 1 L828 A853 M902 Y904 L905 L956 L14 A39 M84 Y86 L87 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=0.700000nM P52333 30145050 1201 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMRDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 6aam A 1.98 BS01 9T6 A 1 L903 A928 I960 E979 Y980 V981 G984 L1030 D1041 L16 A35 I65 E84 Y85 V86 G89 L135 D146 N1023 A1025 R1027 N1028 D1041 P1064 N128 A130 R132 N133 D146 P155 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=4.8nM P29597 30145050 1201 DPTVFHKRYLKKIRDLGGKVSLYCYDPTNTGEMVAVKALDAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGLAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYQG 6abk A 1.58 BS03 9VF A 1 A302 A306 N346 F384 S399 W417 A115 A119 N159 F197 S212 W230 6.1.1.26 0000049,0004812,0005524,0043039 Kd=11.3mM remove_due_to_license_issue Q8PWY1 31031143 505 PALTKSQTDRLEVLLNPKDEISLNSGKPFRELESELLSRRKKDLQQIYAEERENYLGKLEREITRFFVDRGFLEIKSPILIPLEYIERMGIDNDTELSKQIFRVDKNFCLRPMLAPNLANYLRKLDRALPDPIKIFEIGPCYRKESDGKEHLEEFTMLNFCQMGSGCTRENLESIITDFLNHLGIDFKIVGDSCMVFGDTLDVMHGDLELSSAVVGPIPLDREWGIDKPWIGAGFGLERLLKVKHDFKNIKRAARSGSYYNGISTNL 6abp A 1.67 BS01 ARA A 1 K10 E14 W16 D90 R151 N232 K9 E13 W15 D89 R150 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.44uM remove_due_to_license_issue P02924 2069949 307 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMLAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 6abp A 1.67 BS02 ARB A 1 K10 E14 W16 D90 R151 N232 K9 E13 W15 D89 R150 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.44uM remove_due_to_license_issue P02924 2069949 308 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMLAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 6abx A 1.7 BS01 FLC A 1 H179 N182 G215 G216 H253 R262 N305 R332 H179 N182 G215 G216 H253 R262 N305 R332 S184 H214 H253 R262 D307 S184 H214 H253 R262 D307 2.3.3.16 0004108,0005737,0005975,0006099,0016746,0036440,0046912 Ki=7.19mM remove_due_to_license_issue A4YGX6 30794680 401 MELRKGLEDIAIKETSITYIDGELGRLYYRGYSIFDLASFSNFEEVAYLLWYGKLPTRHELDDFKSRLAEERSISEDISTFVKRTAKFGNPMDILRTTVSMMGLEDRSEGDLIGKAIKMTAKIPTIISLIQRTRRNQEFVEPDPSLSHSENFLYMIRGERPSPSDTRVLDVSLMLHMDHEMNASTMACLVVASTLSDIYSSVVAGISALKGPLHGGANSEALKQFMEIETPDNVEKYVMNKLSSGQRLMGFGHRIYKTMDPRAKILKEYANQLSKNEEIKRLFEIANRVEEIGIKILGKRGIYPNVDFYSGLVFYAMGFDPDLFPTIFASARVIGWTAHVDEYLKDNKLIRPKAIYVGDLGKRYVPIEER 6abx B 1.7 BS01 FLC B 1 H179 N182 H214 H253 R262 D307 R332 H179 N182 H214 H253 R262 D307 R332 S184 H214 H253 R262 D307 S184 H214 H253 R262 D307 2.3.3.16 0004108,0005737,0005975,0006099,0016746,0036440,0046912 Ki=7.19mM remove_due_to_license_issue A4YGX6 30794680 401 MELRKGLEDIAIKETSITYIDGELGRLYYRGYSIFDLASFSNFEEVAYLLWYGKLPTRHELDDFKSRLAEERSISEDISTFVKRTAKFGNPMDILRTTVSMMGLEDRSEGDLIGKAIKMTAKIPTIISLIQRTRRNQEFVEPDPSLSHSENFLYMIRGERPSPSDTRVLDVSLMLHMDHEMNASTMACLVVASTLSDIYSSVVAGISALKGPLHGGANSEALKQFMEIETPDNVEKYVMNKLSSGQRLMGFGHRIYKTMDPRAKILKEYANQLSKNEEIKRLFEIANRVEEIGIKILGKRGIYPNVDFYSGLVFYAMGFDPDLFPTIFASARVIGWTAHVDEYLKDNKLIRPKAIYVGDLGKRYVPIEER 6acb A 2.8 BS02 9T9 A 1 V660 I768 A783 F786 F787 M816 Q817 F820 V126 I234 A249 F252 F253 M264 Q265 F268 3.1.4.35 0004114,0007165,0008081 remove_due_to_license_issue O76074 30148362 904 EETRELQSLAAAVVPSAQTLKITDFSFSDFELSDLETALCTIRMFTDLNLVQNFQMKHEVLCRWILSVKKNYRKNVAYHNWRHAFNTAQCMFAALKAGKIQNKLTDLEILALLIAALSHDLDHRGVNNSYIQRSEHPLAQLYCHSIMEHHHFDQCLMILNSPGNQILSGLSIEEYKTTLKIIKQAILATDLALYIKRRGEFFELIRKNQFNLEDPHQKELFLAMLMTACDLSAITKPWPIQQRIAELVATEFFDQEKKNKIPSMQVGFIDAICLQLYEALTHVSEDCFPLLDGCRKNRQKWQALAEQQ 6aec A 1.72 BS03 ATP A 1 G319 G320 R323 H329 D330 D332 F389 D418 W434 G183 G184 R187 H193 D194 D196 F237 D254 W270 D330 D332 D418 D194 D196 D254 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=0.71uM remove_due_to_license_issue Q9NP87 31067051 503 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6aeh A 1.64 BS03 UTP A 1 G319 G320 R323 H329 D330 D332 W434 G436 G182 G183 R186 H192 D193 D195 W269 G271 D330 D332 D418 D193 D195 D253 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=1.77uM remove_due_to_license_issue Q9NP87 31067051 503 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6af9 A 1.39 BS01 ISN A 1 E18 G74 G75 C106 A107 H126 E17 G73 G74 C105 A106 H125 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6af9 A 1.39 BS02 ISN A 2 L101 K148 A171 L100 K147 A170 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 202 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6af9 A 1.39 BS03 ISN A 3 L166 E170 K175 A178 K182 L165 E169 K174 A177 K181 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 203 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afa A 1.65 BS01 ISN A 1 E15 E18 G75 C106 A107 H126 E14 E17 G74 C105 A106 H125 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afc A 1.45 BS01 72R A 1 E15 E18 G75 C106 A107 H126 E14 E17 G74 C105 A106 H125 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afd A 1.48 BS01 72S A 1 E18 G74 G75 N76 C106 A107 H126 E17 G73 G74 N75 C105 A106 H125 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afd A 1.48 BS02 72S A 2 L101 K148 A171 L100 K147 A170 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 202 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afe A 1.5 BS01 72T A 1 E18 G75 N76 C106 A107 H126 L128 E17 G74 N75 C105 A106 H125 L127 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afe A 1.5 BS02 72T A 2 L101 K148 A171 L100 K147 A170 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 202 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6aff A 1.6 BS01 72U A 1 E18 G74 G75 N76 C106 A107 H126 L128 E17 G73 G74 N75 C105 A106 H125 L127 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6aff A 1.6 BS02 72U A 2 L101 K148 A171 L100 K147 A170 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 202 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afg A 1.5 BS01 72V A 1 E15 E18 G75 N76 C106 A107 H126 E14 E17 G74 N75 C105 A106 H125 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afg A 1.5 BS02 72V A 2 L101 K148 A171 L100 K147 A170 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 202 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afh A 1.65 BS01 73F A 1 E15 E18 G75 C106 A107 H126 L128 A129 E14 E17 G74 C105 A106 H125 L127 A128 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afi A 1.65 BS01 73D A 1 E15 E18 G75 N76 C106 A107 H126 E14 E17 G74 N75 C105 A106 H125 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afj A 1.48 BS01 73G A 1 E18 G75 N76 C106 A107 H126 L128 K132 E17 G74 N75 C105 A106 H125 L127 K131 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afl A 1.6 BS01 73H A 1 E15 E18 G75 C106 A107 H126 L128 A129 P158 E14 E17 G74 C105 A106 H125 L127 A128 P157 3.1.2.-,3.5.1.-,3.5.1.124 0000785,0001046,0001933,0001963,0002866,0003690,0003697,0003713,0003723,0003729,0005102,0005507,0005515,0005634,0005654,0005737,0005739,0005758,0005759,0005783,0005829,0005886,0005912,0006281,0006508,0006914,0006954,0006979,0007005,0007265,0007338,0008021,0008047,0008233,0008344,0009438,0010273,0010628,0010629,0016532,0016605,0016684,0019249,0019430,0019826,0019899,0019900,0019955,0030073,0030091,0030414,0030424,0030521,0030546,0031334,0031397,0032435,0032679,0032757,0033138,0033234,0034599,0034614,0036470,0036471,0036478,0036524,0042177,0042542,0042593,0042743,0042802,0042803,0043005,0043523,0043524,0044297,0044388,0044390,0045121,0045296,0045340,0045944,0046295,0046826,0048471,0050681,0050727,0050787,0050821,0051583,0051881,0051897,0051899,0051920,0055105,0060081,0060765,0061691,0061727,0070062,0070301,0070994,0097110,0106044,0106045,0106046,0110095,0140041,0140297,1900182,1900242,1901984,1902176,1902177,1902236,1902903,1902958,1903073,1903094,1903122,1903135,1903136,1903181,1903189,1903190,1903197,1903376,1903377,1903384,1903427,1903428,1903599,1903751,1905259,1990381,1990422,2000379,2001237 remove_due_to_license_issue Q99497 30063823 201 ASKRALVILAKGAEEMETVIPVDVMRRAGIKVTVAGLAGKDPVQCSRDVVICPDASLEDAKKEGPYDVVVLPGGNLGAQNLSESAAVKEILKEQENRKGLIAAICAGPTALLAHEIGFGSKVTTHPLAKDKMMNGGHYTYSENRVEKDGLILTSRGPGTSFEFALAIVEALNGKEVAAQVKAPLVLK 6afr A 1.998 BS01 9E3 A 1 W81 P82 L92 Y139 N140 W40 P41 L51 Y98 N99 ? ic50=70nM remove_due_to_license_issue IC50=70nM O60885 30529546 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6agg Z 2.706 BS02 AG2 Z 1 D193 N194 V203 C204 G215 R217 D193 N194 V203 C204 G215 R217 6.3.4.22 0002101,0003676,0005524,0005737,0008033,0016874,0016879 remove_due_to_license_issue O28025 30121296 503 MRVWVGIDDTDSSRGMCTTYLAVLAMERVERELGKVIGFPRLIRLNPTIPYKTRGNGAVSFLVEVDDVGELVDVVNEVIIEHAMLDDEKTNPGAVFVDEELAVKLKPFADKAIKDVLQIDEALFVIGKYFIPHLRHKKGRGLIGALAAVGAELEDFTLELIAYRYPERFGTEREYDEESFFDMDYELYPQTFDNVDWCNDVVVCIPNTPCPVLYGIRGESVEALYKAMESVKTEPVDRRMIFVTNHATDMHLIGEEEVHRLENYRSYRLRGRVTLEPYDIEGGHVFFEIDTKFGSVKCAAFEPTKQFRNVIRLLRKGDVVEVYGSMKKDTINLEKIQIVELAEIWVEKNPICPSCGRRMESAGRGQGFRCKKCRTKADEKLREKVERELQPGFYEVPPSARRHLSKPLIRMNVEGRHIFR 6agp A -1.00 BS01 GDP A 1 G12 A13 V14 G15 K16 T17 C18 K116 D118 L119 A159 C160 G12 A13 V14 G15 K16 T17 C18 K116 D118 L119 A159 C160 3.6.5.2 0001764,0001934,0003376,0003924,0003925,0005515,0005525,0005634,0005737,0005789,0005802,0005829,0005856,0005884,0005886,0005925,0005938,0006954,0007015,0007155,0007160,0007163,0007264,0008045,0008360,0008361,0009611,0009653,0010310,0010591,0010592,0010595,0010764,0010811,0016020,0016477,0016601,0016787,0019899,0019901,0030027,0030031,0030032,0030036,0030041,0030334,0030425,0030667,0030865,0031116,0031410,0031529,0031996,0032587,0032707,0032956,0034446,0035025,0035556,0036464,0042470,0042554,0042995,0043020,0043197,0044877,0045202,0045428,0045730,0048012,0048261,0048870,0051022,0051492,0051496,0051668,0051894,0055038,0060071,0060263,0060326,0070062,0071526,0090023,0097178,0098794,0098978,0101003,1900026,1902622,1903348,1990606 remove_due_to_license_issue P63000 30891502 201 MQAIKCVVVGDGAVGKTCLLISYTTNAFPGCYIPTVFDNYSANVMVDGKPVNLGLWDTAGQECYDRLRPLSYPCTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLRDDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSACTQRGLKTVFDEAIRAVLCPPP 6ahi B 1.9 BS01 MET B 1 X46 T73 A74 G75 N76 T77 K104 X46 T73 A74 G75 N76 T77 K104 K46 S267 K46 S267 2.5.1.47 0004122,0004124,0005737,0006535,0016740,0016765,0019344 remove_due_to_license_issue P56067 31132312 601 MMIITTMQDAIGRTPVFKFTNKDYPIPLNSAIYAKLEHLNPGGSVKDRLGQYLIGEGFKTGKITSKTTIIEPTAGNTGIALALVAIKHHLKTIFVVPEKFSTEKQQIMRALGALVINTPTSEGISGAIKKSKELAESIPDSYLPLQFENPDNPAAYYHTLAPEIVQELGTNLTSFVAGIGSGGTFAGTARYLKERIPAIRLIGVEPEGSILNGGEPGPHEIEGIGVEFIPPFFENLDIDGFETISDEEGFSYTRKLAKKNGLLVGSSSGAAFVAALKEAQRLPEGSQVLTIFPDVADRYLSKGIYL 6ai9 A 2.09 BS01 PAZ A 1 S99 A100 G101 T102 R103 A209 A210 A211 F280 L282 N308 R313 S62 A63 G64 T65 R66 A172 A173 A174 F230 L232 N258 R263 6.3.2.5 0003824,0004632,0005515,0005634,0005737,0015937,0016874,1990143 remove_due_to_license_issue P40506 30653991 401 TEEEQYFKTNPKPAYIDELIKDAKEFIDLQYSLKRNKIVLITSGGTTVPLENNTVRFIDNFSAGTRGASSAEQFLANGYSVIFLHREFSLTPYNRSFSHSINTLFLDYIDSEGKIKPEFAENVLKNKKLYDKYMEKEEKLLLLPFTTVNQYLWSLKSIAKLLNNSGCLFYLAAAVSDFFVPYSRLPQHKIQEGTTRTTPDGKLIVNLDPVPKFLRRLVESWATQAMIVSFKLETDESMLLYKCTQALDRYNHQLVIGNLLQTRNKQVIFVSPENRKGDWVRLDEKHASIEEMIIPEVIARHDKWVAHSKT 6ai9 B 2.09 BS01 PAZ B 1 S99 A100 G101 T102 R103 A209 A210 F280 L282 N308 R313 S63 A64 G65 T66 R67 A173 A174 F231 L233 N259 R264 6.3.2.5 0003824,0004632,0005515,0005634,0005737,0015937,0016874,1990143 remove_due_to_license_issue P40506 30653991 401 TTEEEQYFKTNPKPAYIDELIKDAKEFIDLQYSLKRNKIVLITSGGTTVPLENNTVRFIDNFSAGTRGASSAEQFLANGYSVIFLHREFSLTPYNRSFSHSINTLFLDYIDSEGKIKPEFAENVLKNKKLYDKYMEKEEKLLLLPFTTVNQYLWSLKSIAKLLNNSGCLFYLAAAVSDFFVPYSRLPQHKIQEGTTRTTPDGKLIVNLDPVPKFLRRLVESWATQAMIVSFKLETDESMLLYKCTQALDRYNHQLVIGNLLQTRNKQVIFVSPENRKGDWVRLDEKHASIEEMIIPEVIARHDKWVAHSKT 6aji A 2.9 BS01 AY6 A 1 L248 I253 V638 L642 D645 Y646 F649 V689 A690 L708 L251 I256 V590 L594 D597 Y598 F601 V641 A642 L660 3.2.1.17 0003796,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue A0QP27,D9IEF7 30682372 1001 SNAMFAWWGRTVYQFRYIVIGVMVALCLGGGVYGISLGNHVTQSGFYDEGSQSVAASLIGDEVYGRDRTSHVVAILTPPDDKKVTDKAWQKKVTEELDQVVKDHEDQIVGWVGWLKAPDTTDPTVSAMKTQDLRHTFISIPLQGDDDDEILKNYQVVEPELQQVNGGDIRLAGLNPLASELTGTIGEDQKRAEVAAIPLVAVVLFFVFGTVIAAALPAIIGGLAIAGALGIMRLVAEFTPVHFFAQPVVTLIGLGIAIDYGLFIVSRFREEIAEGYDTEAAVRRTVMTSGRTVVFSAVIIVASSVPLLLFPQGFLKSITYAIIASVMLAAILSITVLAAALAILGPRVDALGPIAFAAPILVVMVLLIIPLGQLSLGGISEKYLPPDNAVRQSQEQFDKLFPGFRTEPLTLVMKREDGEPITDAQIADMRAKALTVSGFTDPDNDPEKMWKERPANDSGSKDPSVRVIQNGLENRNDAAKKIDELRALQPPHGIEVFVGGTPALEQDSIHSLFDKLPLMALILIVTTTVLMFLAFGSVVLPIKAALMSALTLGSTMGILTWMFVDGHGSGLMNYTPQPLMAPMIGLIIAVIWGLSTDYEVFLVSRMVEARERGMSTAEAIRIGTATTGRLITGAALILAVVAGAFVFSDLVMMKYLAFGLLIALLLDATIIRMFLVPAVMKLLGDDCWWAPRKEFNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYEFHLGGIKAFHHHHHHHH 6ajj A 2.794 BS07 J9E A 1 I249 I253 F260 I297 V638 G641 L642 D645 Y646 F649 I254 I258 F265 I302 V611 G614 L615 D618 Y619 F622 3.2.1.17 0003796,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue A0QP27,D9IEF7 30682372 1008 FQSNAMFAWWGRTVYQFRYIVIGVMVALCLGGGVYGISLGNHVTQSGFYDEGSQSVAASLIGDEVYGRDRTSHVVAILTPPDDKKVTDKAWQKKVTEELDQVVKDHEDQIVGWVGWLKAPDTTDPTVSAMKTQDLRHTFISIPLQGDDDDEILKNYQVVEPELQQVNGGDIRLAGLNPLASELTGTIGEDQKRAEVAAIPLVAVVLFFVFGTVIAAALPAIIGGLAIAGALGIMRLVAEFTPVHFFAQPVVTLIGLGIAIDYGLFIVSRFREEIAEGYDTEAAVRRTVMTSGRTVVFSAVIIVASSVPLLLFPQGFLKSITYAIIASVMLAAILSITVLAAALAILGPRVDALGVTTLLKGFWGRLVNVVMKRPIAFAAPILVVMVLLIIPLGQLSLGGISEKYLPPDNAVRQSQEQFDKLFPGFRTEPLTLVMKREDGEPITDAQIADMRAKALTVSGFTDPDNDPEKMWKERPANDSGSKDPSVRVIQNGLENRNDAAKKIDELRALQPPHGIEVFVGGTPALEQDSIHSLFDKLPLMALILIVTTTVLMFLAFGSVVLPIKAALMSALTLGSTMGILTWMFVDGHGSGLMNYTPQPLMAPMIGLIIAVIWGLSTDYEVFLVSRMVEARERGMSTAEAIRIGTATTGRLITGAALILAVVAGAFVFSDLVMMKYLAFGLLIALLLDATIIRMFLVPAVMKLLGDDCWWAPRWMKRVQEKEFNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYEFHLGGIKAFHHHHHHHH 6ajr A 1.341 BS02 URA A 1 E52 Q53 E58 P64 F65 N91 H178 E51 Q52 E57 P63 F64 N90 H174 ? 0004844,0006281,0046872,0051539,0097506 remove_due_to_license_issue A0QP43 31101917 302 AGAQDFVPHTADLAELAAAAGECRGCGLYRDATQAVFGAGGRSARIMMIGEQPGDKEDLAGLPFVGPAGRLLDRALEAADIDRDALYVTNAVKHFKFTRAAGGKRRIHKTPSRTEVVACRPWLIAEMTSVEPDVVVLLGATAAKALLGNDFRVTQHRGEVLHVDVPPALVATVHPSSLLRGPKEERESAFAGLVDDLRVAADVR 6ajv A 1.45 BS01 HCC A 1 W81 Q85 V87 K91 L92 I146 W48 Q52 V54 K58 L59 I113 ? Kd=9.1uM remove_due_to_license_issue O60885 30565859 202 MHHHHHHMSTNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6ajx A 1.887 BS01 HCC A 1 V87 L92 L94 Y97 C136 I146 V51 L56 L58 Y61 C100 I110 ? Kd=9.1uM remove_due_to_license_issue O60885 30565859 201 HHHHMSTNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6ajy A 1.6 BS01 A0R A 1 W81 Q85 V87 K91 L92 I146 W48 Q52 V54 K58 L59 I113 ? Kd=5.3uM remove_due_to_license_issue O60885 30565859 201 MHHHHHHMSTNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6ajz A 1.301 BS01 LOC A 1 F83 L92 L94 N140 D144 I146 F50 L59 L61 N107 D111 I113 ? remove_due_to_license_issue O60885 30565859 200 MHHHHHHMSTNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6ak4 A 2.8 BS02 PD9 A 1 R96 Y108 N205 H231 D233 Y295 R316 T320 R322 R70 Y82 N140 H166 D168 Y217 R238 T242 R244 1.14.11.-,1.14.11.53 0006307,0035515,0035516,0040014,0042245 remove_due_to_license_issue Q9C0B1 30996080 602 RGSHMTPKDDEFYQQWQLKYPKLILREASSVSEELHKEVQEAFLTLHKHGCLFRDLVRIQGKDLLTPVSRILIGNPGCTYKYLNTRLFTVPWPVKGAEIAAACETFLKLNDYLQIETIQALEELAADIKSRAAYNVTLLNFMDPQKMPYLKEEPYFGMGKMAVSWHHDENLVDRSAVAVYSYSCEGRDPDIWHVGFKISWDIETPGLAIPLHQGDCYFMLDDLNATHQHCVLAGSQPRFSSTHRVAECSTGTLDYILQRCQLALQNVCDDVDNDDVSLKSFEPAVLKQGEEIHNEVEFEWLRQFWFQGNRYRKCTDWWCQPMAQLEALWKKMEGVTNAVLHEVKREGLPVEQRNEILTAILASLTARQNLRREWHARCQSRIARTLPADQKPECRPYWEKDDASMPLPFDLTDIVSELRGQLLEA 6ak5 A 1.7 BS03 GTP A 1 G319 G320 R323 H329 D330 D332 R387 W434 S458 G183 G184 R187 H193 D194 D196 R236 W271 S295 D330 D332 D418 D194 D196 D255 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=0.75uM remove_due_to_license_issue Q9NP87 31067051 503 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHDAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak6 A 1.75 BS03 CTP A 1 G319 G320 R323 K325 H329 D330 D332 W434 G183 G184 R187 K189 H193 D194 D196 W270 D330 D332 D418 D194 D196 D254 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=2.76uM remove_due_to_license_issue Q9NP87 31067051 503 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak8 A 1.74 BS01 dna T 0 L177 F385 E386 R387 R442 R445 R449 K450 L456 N457 H459 L40 F230 E231 R232 R275 R278 R282 K283 L289 N290 H292 D330 D332 D418 D193 D195 D251 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 remove_due_to_license_issue Q9NP87 31067051 1 ~ 9 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak8 A 1.74 BS02 dna P 0 G245 V246 G247 T250 F389 R416 D418 W434 G108 V109 G110 T113 F234 R249 D251 W267 D330 D332 D418 D193 D195 D251 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 remove_due_to_license_issue Q9NP87 31067051 1 ~ 4 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak8 A 1.74 BS03 dna D 0 G174 R175 T178 F179 H204 G206 H208 S209 G37 R38 T41 F42 H67 G69 H71 S72 D330 D332 D418 D193 D195 D251 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 remove_due_to_license_issue Q9NP87 31067051 1 ~ 4 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak9 A 1.91 BS01 dna T 0 L177 F385 E386 R387 R442 R445 R449 K450 L456 N457 H459 L40 F230 E231 R232 R275 R278 R282 K283 L289 N290 H292 D330 D332 D418 D193 D195 D251 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 remove_due_to_license_issue Q9NP87 31067051 1 ~ 9 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak9 A 1.91 BS02 dna P 0 G245 V246 G247 T250 F389 R416 D418 W434 G108 V109 G110 T113 F234 R249 D251 W267 D330 D332 D418 D193 D195 D251 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 remove_due_to_license_issue Q9NP87 31067051 1 ~ 4 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ak9 A 1.91 BS03 dna D 0 G174 R175 T178 F179 H204 G206 H208 S209 G37 R38 T41 F42 H67 G69 H71 S72 D330 D332 D418 D193 D195 D251 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 remove_due_to_license_issue Q9NP87 31067051 1 ~ 4 MPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ako C 2.396 BS01 dna A 0 K72 S76 Y77 I78 N118 S119 H122 R164 K3 S7 Y8 I9 N49 S50 H53 R95 ? 0003700,0006355,0043565 remove_due_to_license_issue Q99958 30722065 1 ~ 16 GPKPPYSYIALITMAIQNAPEKKITLNGIYQFIMDRFPFYRENKQGWQNSIRHNLSLNECFVKVPRDDKKPGKGSYWTLDPDSYNMFENGSFLRRRR 6ako C 2.396 BS02 dna B 0 L95 R121 H122 S125 K132 K142 S144 W146 R163 R166 L26 R52 H53 S56 K63 K73 S75 W77 R94 R97 ? 0003700,0006355,0043565 remove_due_to_license_issue Q99958 30722065 1 ~ 16 GPKPPYSYIALITMAIQNAPEKKITLNGIYQFIMDRFPFYRENKQGWQNSIRHNLSLNECFVKVPRDDKKPGKGSYWTLDPDSYNMFENGSFLRRRR 6alc B 1.391 BS01 BKD B 1 P1110 V1115 I1122 N1168 V1174 P28 V33 I40 N86 V92 2.3.1.-,2.3.1.48 remove_due_to_license_issue IC50=31nM Q92793 29169673 1201 AAFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQAL 6alg I 3.7 BS01 dna A 0 R151 K163 R175 W183 D199 R473 R542 V547 R150 K162 R174 W182 D198 R472 R541 V546 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 28318486 1 ~ 29 VYSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELED 6alg I 3.7 BS02 dna B 0 N139 T141 K496 G1261 K1262 R1269 M1273 N138 T140 K495 G1239 K1240 R1247 M1251 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 28318486 1 ~ 29 VYSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELED 6alg I 3.7 BS03 rna R 0 Q510 Q513 Q688 K1065 K1073 H1237 S1252 L1253 L1259 Q509 Q512 Q687 K1043 K1051 H1215 S1230 L1231 L1237 2.7.7.6 0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0009408,0016020,0016779,0031564,0032549,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8V2 28318486 11 ~ 20 VYSYTEKKRIRKDFGKRPQVLDVPYLLSIQLDSFQKFIEQDPEGQYGLEAAFRSVFPIQSYSGNSELQYVSYRLGEPVFDVQECQIRGVTYSAPLRVKLRLVIYEREAPEGTVKDIKEQEVYMGEIPLMTDNGTFVINGTERVIVSQLHRSPGVFFDSDKGKTHSSGKVLYNARIIPYRGSWLDFEFDPKDNLFVRIDRRRKLPATIILRALNYTTEQILDLFFEKVIFEIRDNKLQMELVPERLRGETASFDIEANGKVYVEKGRRITARHIRQLEKDDVKLIEVPVEYIAGKVVAKDYIDESTGELICAANMELSLDLLAKLSQSGHKRIETLFTNDLDHGPYISETLRVDPTNDRLSALVEIYRMMRPGEPPTREAAESLFENLFFSEDRYDLSAVGRMKFNRSLLREEIEGSGILSKDDIIDVMKKLIDIRNGKGEVDDIDHLGNRRIRSVGEMAENQFRVGLVRVERAVKERLSLGDLDTLMPQDMINAKPISAAVKEFFGSSQLSQFMDQNNPLSEITHKRRISALGPGGLTRERAGFEVRDVHPTHYGRVCPIETPEGPNIGLINSLSVYAQTNEYGFLETPYRKVTDGVVTDEIHYLSAIEEGNYVIAQANSNLDEEGHFVEDLVTCRSKGESSLFSRDQVDYMDVSTQQVVSVGASLIPFLEHDDANRALMGANMQRQAVPTLRADKPLVGTGMERAVAVDSGVTAVAKRGGVVQYVDASRIVIKVNEDEMYPGEAGIDIYNLTKYTRSNQNTCINQMPCVSLGEPVERGDVLADGPSTDLGELALGQNMRVAFMPWNGYNFEDSILVSERVVQEDRFTTIHIQELACVSRDTKLGPEEITADIPNVGEAALSKLDESGIVYIGAEVTGGDILVGKVTPKDVKDSSLRVPNGVSGTVIDVQVFTRDGVEKDKRALEIEEMQLKQAKKDLSEELQILEAGLFSRIRAVLVAGGVEAEKLDKLPRDRWLELGLTDEEKQNQLEQLAEQYDELKHEFEKKLEAKRRKITQGDDLAPGVLKIVKVYLAVKRRIQPGDKMAGRHGNKGVISKINPIEDMPYDENGTPVDIVLNPLGVPSRMNIGQILETHLGMAAKGIGDKINAMLKQQQEVAKLREFIQRAYDLGADVRQKVDLSTFSDEEVMRLAENLRKGMPIATPVFDGAKEAEIKELLKLGDLPTSGQIRLYDGRTGEQFERPVTVGYMYMLKLNHLVDDKMHARSTGSYSLVTQQPLGGKAQFGGQRFGEMEVWALEAYGAAYTLQEMLTVKSDDVNGRTKMYKNIVDGNHQMEPGMPESFNVLLKEIRSLGINIELED 6alg J 3.7 BS01 dna A 0 R270 N274 R275 M298 R1148 R255 N259 R260 M283 R1110 2.7.7.6 0000287,0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0008270,0009408,0016020,0016779,0031564,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0046872,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8T7 28318486 1 ~ 29 EFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTMSSIQVKNKGSIKLSNVKSVVNSSGKLVITSRNTELKLIDEFGRTKESYKVPYGAVLAKGDGEQVAGGETVANWDPHTMPVITEVSGFVRFTDMIDGQTITRQTDELTGLSSLVVLDSAERTAGGKDLRPALKIVDAQGNDVLIPGTDMPAQYFLPGKAIVQLEDGVQISSGDTLARIPQTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRR 6alg J 3.7 BS02 dna B 0 S210 K334 R339 R352 T790 A791 Y795 K1172 Q1326 E1327 S195 K319 R324 R337 T775 A776 Y780 K1134 Q1288 E1289 2.7.7.6 0000287,0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0008270,0009408,0016020,0016779,0031564,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0046872,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8T7 28318486 1 ~ 29 EFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTMSSIQVKNKGSIKLSNVKSVVNSSGKLVITSRNTELKLIDEFGRTKESYKVPYGAVLAKGDGEQVAGGETVANWDPHTMPVITEVSGFVRFTDMIDGQTITRQTDELTGLSSLVVLDSAERTAGGKDLRPALKIVDAQGNDVLIPGTDMPAQYFLPGKAIVQLEDGVQISSGDTLARIPQTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRR 6alg J 3.7 BS03 rna R 0 L255 R425 D464 L240 R410 D449 2.7.7.6 0000287,0000345,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005737,0005829,0006351,0006352,0006360,0006366,0006383,0006879,0008023,0008270,0009408,0016020,0016779,0031564,0032784,0034062,0036460,0042128,0042793,0044780,0046677,0046872,0048870,0071973,0090605,2000142 remove_due_to_license_issue P0A8T7 28318486 11 ~ 20 EFDAIKIALASPDMIRSWSFGEVKKPETINYRTFKPERDGLFCARIFGPVKDYECLCGKYKRLKHRGVICEKCGVEVTQTKVRRERMGHIELASPTAHIWFLKSLPSRIGLLLDMPLRDIERVLYFESYVVIEGGMTNLERQQILTEEQYLDALEEFGDEFDAKMGAEAIQALLKSMDLEQECEQLREELNETNSETKRKKLTKRIKLLEAFVQSGNKPEWMILTVLPVLPPDLRPLVPLDGGRFATSDLNDLYRRVINRNNRLKRLLDLAAPDIIVRNEKRMLQEAVDALLDNGRRGRAITGSNKRPLKSLADMIKGKQGRFRQNLLGKRVDYSGRSVITVGPYLRLHQCGLPKKMALELFKPFIYGKLELRGLATTIKAAKKMVEREEAVVWDILDEVIREHPVLLNRAPTLHRLGIQAFEPVLIEGKAIQLHPLVCAAYNADFDGDQMAVHVPLTLEAQLEARALMMSTNNILSPANGEPIIVPSQDVVLGLYYMTRDCVNAKGEGMVLTGPKEAERLYRSGLASLHARVKVRITEYEKDANGELVAKTSLKDTTVGRAILWMIVPKGLPYSIVNQALGKKAISKMLNTCYRILGLKPTVIFADQIMYTGFAYAARSGASVGIDDMVIPEKKHEIISEAEAEVAEIQEQFQSGLVTAGERYNKVIDIWAAANDRVSKAMMDNLQTETVINRDGQEEKQVSFNSIYMMADSGARGSAAQIRQLAGMRGLMAKPDGSIIETPITANFREGLNVLQYFISTHGARKGLADTALKTANSGYLTRRLVDVAQDLVVTEDDCGTHEGIMMTPVIEGGDVKEPLRDRVLGRVTAEDVLKPGTADILVPRNTLLHEQWCDLLEENSVDAVKVRSVVSCDTDFGVCAHCYGRDLARGHIINKGEAIGVIAAQSIGEPGTQLTMSSIQVKNKGSIKLSNVKSVVNSSGKLVITSRNTELKLIDEFGRTKESYKVPYGAVLAKGDGEQVAGGETVANWDPHTMPVITEVSGFVRFTDMIDGQTITRQTDELTGLSSLVVLDSAERTAGGKDLRPALKIVDAQGNDVLIPGTDMPAQYFLPGKAIVQLEDGVQISSGDTLARIPQTGGLPRVADLFEARRPKEPAILAEISGIVSFGKETKGKRRLVITPVDGSDPYEEMIPKWRQLNVFEGERVERGDVISDGPEAPHDILRLRGVHAVTRYIVNEVQDVYRLQGVKINDKHIEVIVRQMLRKATIVNAGSSDFLEGEQVEYSRVKIANRELEANGKVGATYSRDLLGITKASLATESFISAASFQETTRVLTEAAVAGKRDELRGLKENVIVGRLIPAGTGYAYHQDRMRRR 6alz A 2.208 BS03 BKM A 1 R96 C127 S129 Y134 V195 W206 R221 V223 V250 Y272 F276 R90 C121 S123 Y128 V189 W200 R215 V217 V244 Y266 F270 D64 H66 D92 D95 R96 N124 H125 H173 R221 H248 D58 H60 D86 D89 R90 N118 H119 H167 R215 H242 3.1.3.16 0016787 remove_due_to_license_issue P62136 29156132 403 LNLDSIIGRLLEVQGSRPGKNVQLTENEIRGLCLKSREIFLSQPILLELEAPLKICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFLLRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDLQSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVQGWGENDRGVSFTFGAEVVAKFLHKHDLDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYCGEFDNAGAMMSVDETLMCSFQILKPA 6am8 A 1.83 BS01 TRP A 1 X82 E104 T105 G106 A107 L161 S185 V187 G228 Y301 X82 E104 T105 G106 A107 L161 S185 V187 G228 Y301 K82 E104 S371 K82 E104 S371 4.2.1.20 0000162,0004834,0005737,0006568,0016829 remove_due_to_license_issue Q8U093 29712420 401 MWFGEFGGQYVPETLVGPLKELEKAYKRFKDDEEFNRQLNYYLKTWAGRPTPLYYAKRLTEKIGGAKVYLKREDLVHGGAHKTNNAIGQALLAKLMGKTRLIAETGAGQHGVATAMAGALLGMKVDIYMGAEDVERQKMNVFRMKLLGANVIPVNSGSRTLKDAINEALRDWVATFEYTHYLIGSVVGPHPYPTIVRDFQSVIGREAKAQILEAEGQLPDVIVACVGGGSNAMGIFYPFVNDKKVKLVGVEAGGKGLESGKHSASLNAGQVGVSHGMLSYFLQDEEGQIKPSHSIAPGLDYPGVGPEHAYLKKIQRAEYVAVTDEEALKAFHELSRTEGIIPALESAHAVAYAMKLAKEMSRDEIIIVNLSGRGDKDLDIVLKA 6ami A 1.97 BS01 TRP A 1 X82 E104 T105 A107 Q109 H110 L161 V187 Y301 X82 E104 T105 A107 Q109 H110 L161 V187 Y299 4.2.1.20 0000162,0004834,0005737,0006568,0016829 Kd=1400uM remove_due_to_license_issue Q8U093 29712420 401 MWFGEFGGQYVPETLIGPLKELEKAYKRFKDDEEFNRQLNYYLKTWAGRPTPLYYAKRLTEKIGGAKVYLKREDLVHGGAHKTNNAIGQALLAKFMGKTRLIAETGAGQHGVATAMAGALLGMKVDIYMGAEDVERQKMNVFRMKLLGANVIPVNSGSRTLKDAINEALRDWVATFEYTHYLIGSVVGPHPYPTIVRDFQSVIGREAKAQILEAEGQLPDVIVACVGGGSNAMGIFYPFVNDKKVKLVGVEAGGKGLESGKHSASLNAGQVGVSHGMLSYFLQDGQIKPSHSIAPGLDYPGVGPEHAYLKKIQRAEYVAVTDEEALKAFHELSRTEGIIPALESAHAVAYAMKLAKEMSRDEIIIVNLSGRGDKDLDIVLKVS 6amk A 3.288 BS01 dna R 0 P14 A15 K26 T29 H46 R47 P6 A7 K18 T21 H38 R39 ? 0003677,0006355 remove_due_to_license_issue F2REK9 29556010 7 ~ 28 PPLLTPAEVATMFRVDPKTVTRWAKAGKLTSIRTMGGHRRYREAEVRALMAG 6amk A 3.288 BS02 dna Z 0 D24 T27 R30 W31 T42 G44 H46 D16 T19 R22 W23 T34 G36 H38 ? 0003677,0006355 remove_due_to_license_issue F2REK9 29556010 5 ~ 26 PPLLTPAEVATMFRVDPKTVTRWAKAGKLTSIRTMGGHRRYREAEVRALMAG 6amk B 3.288 BS01 dna R 0 P14 A15 K26 H46 R47 P5 A6 K17 H37 R38 ? 0003677,0006355 remove_due_to_license_issue F2REK9 29556010 7 ~ 28 PLLTPAEVATMFRVDPKTVTRWAKAGKLTSIRTMGGHRRYREAEVRALMAG 6amk B 3.288 BS02 dna Z 0 V23 D24 T27 R30 W31 G44 H46 V14 D15 T18 R21 W22 G35 H37 ? 0003677,0006355 remove_due_to_license_issue F2REK9 29556010 5 ~ 26 PLLTPAEVATMFRVDPKTVTRWAKAGKLTSIRTMGGHRRYREAEVRALMAG 6an1 A 2.687 BS01 BKY A 1 L228 C285 R288 L330 I341 S342 E343 M348 M364 L25 C71 R74 L116 I127 S128 E129 M134 M150 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=1144nM P37231 29449830 501 LNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKD 6anl A 2.0 BS01 T75 A 1 Y35 A51 K53 L75 L104 T106 M109 F169 L171 A172 Y32 A48 K50 L72 L101 T103 M106 F166 L168 A169 D150 K152 N155 D168 T185 D147 K149 N152 D165 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=240nM remove_due_to_license_issue IC50=240nM Q16539 29291937 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLAATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 6aol A 2.764 BS01 VC1 A 1 N107 A111 D149 M154 N162 I166 F199 Y200 T245 I247 N34 A38 D76 M81 N89 I93 F120 Y121 T166 I168 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=540nM, Kd=540nM P41148 28857290 401 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTESTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 6aom A 2.87 BS01 VC5 A 1 N107 D110 A111 K114 D149 M154 N162 F199 T245 I247 N34 D37 A38 K41 D76 M81 N89 F118 T164 I166 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Kd=630nM P41148 28857290 409 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKTSEFLNKMTESTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTTVWDWELMN 6ap6 A 1.65 BS01 TLF A 1 F27 S96 F125 F135 F158 S190 V193 F194 S219 H246 F25 S94 F123 F133 F156 S188 V191 F192 S217 H244 3.1.-.- 0010223,0016787,0016788,1901601 Kd=4.3uM remove_due_to_license_issue J9U5U9 29523686 300 QTLLDALNVRVVGSGERVLVLAHGFGTDQSAWNRILPFFLRDYRVVLYDLVCAGSVNPDFFDFRRYTTLDPYVDDLLHILDALGIDQCAYVGHSVSAMIGILASIRRPELFSKLILIGASPRFLNDEDYHGGFEQGEIEKVFSAMEANYEAWVNGFAPLAVGADVPAAVREFSRTLFNMRPDITLFVSRTVFNSDMRGVLGLVKVPCHIFQTARDHSVPASVATYLKNHLGGKNTVHWLNIEGHLPHLSAPTLLAQELRRALSH 6ap7 A 1.51 BS01 BNY A 1 F27 S96 F125 F135 V143 F158 S190 V193 F194 H218 S219 H246 F25 S94 F123 F133 V141 F156 S188 V191 F192 H216 S217 H244 3.1.-.- 0010223,0016787,0016788,1901601 Kd=4.6uM remove_due_to_license_issue J9U5U9 29523686 300 QTLLDALNVRVVGSGERVLVLAHGFGTDQSAWNRILPFFLRDYRVVLYDLVCAGSVNPDFFDFRRYTTLDPYVDDLLHILDALGIDQCAYVGHSVSAMIGILASIRRPELFSKLILIGASPRFLNDEDYHGGFEQGEIEKVFSAMEANYEAWVNGFAPLAVGADVPAAVREFSRTLFNMRPDITLFVSRTVFNSDMRGVLGLVKVPCHIFQTARDHSVPASVATYLKNHLGGKNTVHWLNIEGHLPHLSAPTLLAQELRRALSH 6ap8 A 1.27 BS01 BNY A 1 F78 S147 F176 F186 V194 C241 V244 S270 H297 F26 S95 F124 F134 V142 C189 V192 S218 H245 3.1.-.- Kd=8uM remove_due_to_license_issue Q10QA5 29523686 401 GAKLLQILNVRVVGSGERVVVLSHGFGTDQSAWSRVLPYLTRDHRVVLYDLVCAGSVNPDHFDFRRYDNLDAYVDDLLAILDALRIPRCAFVGHSVSAMIGILASIRRPDLFAKLVLIGASPRFLNDSDYHGGFELEEIQQVFDAMGANYSAWATGYAPLAVGADVPAAVQEFSRTLFNMRPDISLHVCQTVFKTDLRGVLGMVRAPCVVVQTTRDVSVPASVAAYLKAHLGGRTTVEFLQTEGHLPHLSAPSLLAQVLRRALARY 6aps A 1.762 BS01 SV2 A 1 G55 D114 I115 D117 T118 A119 T121 K145 F166 V167 D173 R179 G58 D97 I98 D100 T101 A102 T104 K128 F149 V150 D156 R162 E113 D114 D117 F166 R179 E96 D97 D100 F149 R162 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=0.22uM remove_due_to_license_issue Q07010 29481567 301 HHHMEPACKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRLCDIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGKELERR 6apt A 1.795 BS01 45T A 1 L53 K54 G55 I115 D117 T118 A119 T121 K145 F166 V167 D173 R179 L49 K50 G51 I89 D91 T92 A93 T95 K119 F140 V141 D147 R153 E113 D114 D117 F166 R179 E87 D88 D91 F140 R153 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=0.89uM remove_due_to_license_issue Q07010 29481567 301 CKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRDIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETW 6apt B 1.795 BS01 45T B 1 K54 G55 I115 D117 T118 A119 T121 K145 F166 V167 D173 R179 K50 G51 I88 D90 T91 A92 T94 K118 F139 V140 D146 R152 E113 D114 D117 F166 R179 E86 D87 D90 F139 R152 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=0.89uM remove_due_to_license_issue Q07010 29481567 301 CKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGK 6apu B 1.842 BS01 3L6 B 1 I115 D117 T118 A119 T121 K145 F166 V167 D173 I90 D92 T93 A94 T96 K120 F141 V142 D148 E113 D114 D117 F166 R179 E88 D89 D92 F141 R154 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=13.46uM remove_due_to_license_issue Q07010 29481567 305 ACKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRDIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGKELERR 6apv A 1.993 BS01 3L4 A 1 K54 G55 I115 D117 T118 A119 T121 K145 F166 V167 D173 R179 K50 G51 I90 D92 T93 A94 T96 K120 F141 V142 D148 R154 E113 D114 D117 F166 R179 E88 D89 D92 F141 R154 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=0.11uM remove_due_to_license_issue Q07010 29481567 301 CKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRADIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGKELE 6apv B 1.993 BS01 3L4 B 1 K54 G55 I115 D117 T118 A119 T121 K145 F166 V167 D173 R179 K50 G51 I93 D95 T96 A97 T99 K123 F144 V145 D151 R157 E113 D114 D117 F166 R179 E91 D92 D95 F144 R157 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0020015,0031981,0032263,0032264,0046100,0046872,0052657,0097014 Ki=0.11uM remove_due_to_license_issue Q07010 29481567 301 CKYDFATSVLFTEAELHTRMRGVAQRIADDYSNCNLKPLENPLVIVSVLKGSFVFTADMVRILGDFGVPTRVEFLRASSYDIRGKHVLVLEDILDTALTLREVVDSLKKSEPASIKTLVAIDKPGGRKIPFTAEYVVADVPNVFVVGYGLDYDQSYREVRDVVILKPSVYETWGKELERRKAA 6apw A 2.614 BS01 BTV A 1 S93 T94 Q116 R120 G121 R122 R125 W127 K187 G190 F191 G208 I209 G210 S92 T93 Q115 R119 G120 R121 R124 W126 K186 G189 F190 G207 I208 G209 0004077,0006355,0036211 remove_due_to_license_issue 29131575 401 SKYSQDVLQLLYKNKPNYISGQSIAESLNISRTAVKKVIDQLKLEGCKIDSVNHKGHLLQQLPDIWYQGIIDQYTKSSALFDFSEVYDSIDSTQLAAKKSLVGNQSSFFILSDEQTKGRGRFNRHWSSSKGQGLWMSVVLRPNVAFSMISKFNLFIALGIRDAIQHFSQDEVKVKWPNDIYIDNGKVCGFLTEMVANNDGIEAIICGIGINLTQQLENFDESIRHRATSIQLHDKNKLDRYQFLERLLQEIEKRYNQFLTLPFSEIREEYNAASNIWNRTLLFTENDKQFKGQAIDLDYDGYLIVRDEAGESHRLISADIDF 6apz A 2.254 BS02 BQ4 A 1 R339 G459 L461 D462 M515 W541 M631 D633 R325 G442 L444 D445 M498 W524 M614 D616 D271 E273 R339 E434 D462 D633 D267 E269 R325 E417 D445 D616 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=0.15uM remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRREPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6aqf A 2.51 BS01 ZMA A 1 L85 F168 M177 L249 H250 N253 I274 L88 F171 M180 L333 H334 N337 I358 ? 0001609,0001973,0004930,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P29274 29290469 1201 DGAPPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKNHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLERARSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSH 6aqo A 2.64 BS01 45T A 1 K87 G88 I149 D151 T152 G153 T155 K180 Y201 V202 E208 R214 K79 G80 I126 D128 T129 G130 T132 K157 Y178 V179 E185 R191 E147 D148 D151 Y201 R214 E124 D125 D128 Y178 R191 ? 0000166,0000287,0000310,0004422,0005737,0005829,0006178,0016757,0020015,0032263,0032264,0042301,0046100,0046872,0052657 remove_due_to_license_issue Q38CA1 29481567 301 PNFVGRDADGNVTVDGRSYPMAESVVATESTIHRSMKEMAQTLANAYKTLKHRDTHNKGNSALAPITDENPLIIISVLKGSYIFTADMVRYLGDCGLPNVVDFIRILDNLRFTELTGKHVLIMEDIADTGRTMKLLVEKIRREYRPASLKVCVLVDKPGGRVVDFKPEFVCLTAPTRYVVGYGFEVNDRYRNYRHVFVLKPEYAKRYPSKL 6aqo E 2.64 BS01 45T E 1 I149 D151 T152 G153 T155 K180 Y201 V202 E208 R214 I125 D127 T128 G129 T131 K156 Y177 V178 E184 R190 E147 D148 D151 Y201 R214 E123 D124 D127 Y177 R190 ? 0000166,0000287,0000310,0004422,0005737,0005829,0006178,0016757,0020015,0032263,0032264,0042301,0046100,0046872,0052657 remove_due_to_license_issue Q38CA1 29481567 301 KPNFVGRDADGNVTVDGRSYPMAESVVATESTIHRSMKEMAQTLANAYKTLKHRDTHNKGNSALAPITDENPLIIISVLKGSYIFTADMVRYLGDCGLPNVVDFIRINLRFTELTGKHVLIMEDIADTGRTMKLLVEKIRREYRPASLKVCVLVDKPGGRVVDFKPEFVCLTAPTRYVVGYGFEVNDRYRNYRHVFVLKPEYAKRYPSKL 6aqq A 2.71 BS01 BVY A 1 S93 T94 Q95 Q116 G119 R120 R125 K187 G190 I209 G210 S92 T93 Q94 Q115 G118 R119 R124 K182 G185 I204 G205 0004077,0006355,0036211 remove_due_to_license_issue 29131575 401 SKYSQDVLQLLYKNKPNYISGQSIAESLNISRTAVKKVIDQLKLEGCKIDSVNHKGHLLQQLPDIWYQGIIDQYTKSSALFDFSEVYDSIDSTQLAAKKSLVGNQSSFFILSDEQTKGRGRFNRHKGQGLWMSVVLRPNVAFSMISKFNLFIALGIRDAIQHFSQDEVKVKWPNDIYIDNGKVCGFLTEMVANNDGIEAIICGIGINLTQQLENFDESIRHRATSIQLHDKNKLDRYQFLERLLQEIEKRYNQFLTLPFSEIREEYIAASNIWNRTLLFTENDKQFKGQAIDLDYDGYLIVRDEAGESHRLISADIDF 6aqs A 1.57 BS01 IM5 A 1 S91 C92 Y160 D181 E182 M183 E184 S89 C90 Y158 D179 E180 M181 E182 2.4.2.1,2.4.2.44 0003824,0004731,0004850,0005829,0006148,0006166,0006195,0006218,0009116,0016757,0017061,0047975 Ki=28nM remove_due_to_license_issue Q8I3X4 29440412 302 NLLRHLKISKEQITPVVLVVGDPGRVDKIKVVCDSYVDLAYNREYKSVECHYKGQKFLCVSHGVGSAGCAVCFEELCQNGAKVIIRAGSCGSLQPDLIKRGDICICNAAVREDRVSHLLIHGDFPAVGDFDVYDTLNKCAQELNVPVFNGISVSSDMYYPNKIIPSRLEDYSKANAAVDEMELATLMVIGTLRKVKTGGILIVDGCVPHQLENMIKIALGACAKLATKYA 6ar4 A 1.69 BS01 BQA A 1 L32 I33 G34 I35 F53 A87 L14 I15 G16 I17 F35 A69 ? ic50=0.573uM remove_due_to_license_issue Q9NRD5 30194389 201 VPGKVTLQKDAQNLIGISIGGGAQYCPCLYIVQVFDNTPAALDGTVAAGDEITGVNGRSIKGKTKVEVAKMIQEVKGEVTIHYNKL 6ar4 B 1.69 BS01 BQA B 1 L32 I33 G34 I35 I37 F53 K83 A87 L15 I16 G17 I18 I20 F36 K66 A70 ? ic50=0.573uM remove_due_to_license_issue Q9NRD5 30194389 201 TVPGKVTLQKDAQNLIGISIGGGAQYCPCLYIVQVFDNTPAALDGTVAAGDEITGVNGRSIKGKTKVEVAKMIQEVKGEVTIHYNKL 6ar9 A 2.28 BS01 3L4 A 1 G88 D148 D151 T152 G153 T155 K180 Y201 V202 E208 R214 G81 D128 D131 T132 G133 T135 K160 Y181 V182 E188 R194 E147 D148 D151 Y201 R214 E127 D128 D131 Y181 R194 ? 0000166,0000287,0000310,0004422,0005737,0005829,0006178,0016757,0020015,0032263,0032264,0042301,0046100,0046872,0052657 Ki=6.54uM remove_due_to_license_issue Q38CA1 29481567 301 KPNFVGRDADGNVTVDGRSYPMAESVVATESTIHRSMKEMAQTLANAYKTLKHRDTHNKGNSALAPITDENPLIIISVLKGSYIFTADMVRYLGDCGLPNVVDFIRITVLDNLRFTELTGKHVLIMEDIADTGRTMKLLVEKIRREYRPASLKVCVLVDKPGGRVVDFKPEFVCLTAPTRYVVGYGFEVNDRYRNYRHVFVLKPEYAKRYPSKL 6arj A 1.92 BS02 BW4 A 1 F152 Y153 M162 E257 P258 M259 Y261 N265 E266 H414 W415 K470 F474 T477 F19 Y20 M29 E124 P125 M126 Y128 N132 E133 H281 W282 K337 F341 T344 D165 E257 E266 H414 D32 E124 E133 H281 2.1.1.319 0016274,0018216 Ki=25nM remove_due_to_license_issue IC50=<100nM Q86X55 29269946 502 RSVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 6arj B 1.92 BS02 BW4 B 1 F152 Y153 M162 E257 P258 M259 Y261 N265 E266 H414 W415 K470 F474 F19 Y20 M29 E124 P125 M126 Y128 N132 E133 H281 W282 K337 F341 D165 E257 E266 H414 D32 E124 E133 H281 2.1.1.319 0016274,0018216 Ki=25nM remove_due_to_license_issue IC50=<100nM Q86X55 29269946 502 RSVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 6arn A 1.25 BS01 BQY A 1 F1 N44 D45 Y46 D51 D53 K132 A134 N140 F1 N44 D45 Y46 D51 D53 K126 A128 N134 ? 0007155,0009289 remove_due_to_license_issue Q1RBS0 29507247 201 FSCNVDGGSSIGAGTTSVYVNLDPVIQPGQNLVVDLSQHISCWNDYGGWYDTDHINLVQGSAFAGSLQSYKGSLYWNNVTYPFPLTTNTNVLDIGDKTPMPLPLKLYITGVVIKAGEVIARIHMYKIATLGSGNPRNFTWNIISNNSVVM 6aro A 1.2 BS01 BS7 A 1 F1 N44 D45 Y46 D51 D53 K132 N140 F1 N44 D45 Y46 D51 D53 K132 N140 ? 0007155,0009289 remove_due_to_license_issue Q1RBS0 29507247 201 FSCNVDGGSSIGAGTTSVYVNLDPVIQPGQNLVVDLSQHISCWNDYGGWYDTDHINLVQGSAFAGSLQSYKGSLYWNNVTYPFPLTTNTNVLDIGDKTPMPLPLKLYITPVGAAGGVVIKAGEVIARIHMYKIATLGSGNPRNFTWNIISNNSVVMP 6arv A 2.0 BS02 BW7 A 1 Y149 F152 Y153 M162 E257 M259 Y261 H414 W415 F474 Y16 F19 Y20 M29 E124 M126 Y128 H281 W282 F341 D165 E257 E266 H414 D32 E124 E133 H281 2.1.1.319 0016274,0018216 ic50=46nM remove_due_to_license_issue Q86X55 29269946 502 RSVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 6arv B 2.0 BS02 BW7 B 1 Y149 F152 Y153 M162 E257 M259 Y261 E266 H414 W415 F474 Y16 F19 Y20 M29 E124 M126 Y128 E133 H281 W282 F341 D165 E257 E266 H414 D32 E124 E133 H281 2.1.1.319 0016274,0018216 ic50=46nM remove_due_to_license_issue Q86X55 29269946 502 RSVFSERTEESSAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRYT 6ary A 2.257 BS01 BT7 A 1 W245 G278 G279 S280 S360 A361 W393 Y489 F490 F560 H600 W83 G116 G117 S118 S198 A199 W231 Y327 F328 F398 H438 G279 S280 S360 A361 E486 H600 G117 S118 S198 A199 E324 H438 3.1.1.7 0004104 remove_due_to_license_issue Q869C3 29276037 801 NDPLVVNTDKGRIRGITVDAPSGKKVDVWLGIPYAQPPVGPLRFRHPRPAEKWTGVLNTTTPPNSCVQIVDTVFGDFPGATMWNPNTPLSEDCLYINVVAPRPRPKNAAVMLWIFGGSFYSGTATLDVYDHRALASEENVIVVSLQYRVASLGFLFLGTPEAPGNAGLFDQNLALRWVRDNIHRFGGDPSRVTLFGESAGAVSVSLHLLSALSRDLFQRAILQSGSPTAPWALVSREEATLRALRLAEAVGCPHEPSKLSDAVECLRGKDPHVLVNNEWGTLGICEFPFVPVVDGAFLDETPQRSLASGRFKKTEILTGSNTEEGYYFIIYYLTELLRKEEGVTVTREEFLQAVRELNPYVNGAARQAIVFEYTDWTEPDNPNSNRDALDKMVGDYHFTCNVNEFAQRYAEEGNNVYMYLYTHRSKGNPWPRWTGVMHGDEINYVFGEPLNPTLGYTEDEKDFSRKIMRYWSNFAKTGNPNPNTASSEFPEWPKHTAHGRHYLELGLNTSFVGRGPRLRQCAFWKKYLPQLVAATSN 6as6 A 1.4 BS02 BSV A 1 R339 E434 G459 L461 D462 M515 W541 D633 R328 E421 G446 L448 D449 M502 W528 D620 D271 E273 R339 E434 D462 D633 D270 E272 R328 E421 D449 D620 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=15.2uM remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6as7 A 2.95 BS01 dna B 0 D1002 K1053 Y1055 K1075 G1076 R1081 R1082 T1140 D624 K675 Y677 K697 G698 R703 R704 T762 2.7.7.7 0000166,0003676,0003677,0003887,1902975 remove_due_to_license_issue P09884 29555682 1 ~ 11 EQVFHFYWLDAYEDQYNQPGVVFLFGKVWIESAETHVSCCVMVKNIERTLYFLPREMKIDLNTGKETGTPISMKDVYEEFDEKIATKYKIMKFKSKPVEKNYAFEIPDVPEKSEYLEVKYSAEMPQLPQDLKGETFSHVFGTNTSSLELFLMNRKIKGPCWLEVKSPQLLNQPVSWCKAEAMALKPDLVNVIKDVSPPPLVVMAFSMKTMQNAKNHQNEIIAMAALVHHSFALDKAAPKPPFQSHFCVVSKPKDCIFPYAFKEVIEKKNVKVEVAATERTLLGFFLAKVHKIDPDIIVGHNIYGFELEVLLQRINVCKAPHWSKIGRLKRSNMPKLGFGERNATCGRMICDVEISAKELIRCKSYHLSELVQQILKTERVVIPMENIQNMYSESSQLLYLLEHTWKDAKFILQIMCELNVLPLALQITNIAGNIMSRTLMGGRSERNEFLLLHAFYENNYIVPDKQIFRKKAAYAGGLVLDPKVGFYDKFILLLDFNSLYPSIIQEFNICFTTVQRVEQIPELPDPSLEMGILPREIRKLVERRKQVKQLMKQQDLNPDLILQYDIRQKALKLTANSMYGCLGFSYSRFYAKPLAALVTYKGREILMHTKEMVQKMNLEVIYGDTDSIMINTNSTNLEEVFKLGNKVKSEVNKLYKLLEIDIDGVFKSLLLLKKKKYAALVVEPTSDGNYVTKQELKGLDIVRRDWCDLAKDTGNFVIGQILSDQSRDTIVENIQKRLIEIGENVLNGSVPVSQFEINKALTKDPQDYPDKKSLPHVHVALWINSQGGRKVKAGDTVSYVICQDGSNLTASQRAYAPEQLQKQDNLTIDTQYYLAQQIHPVVARICEPIDGIDAVLIATWLGLDPTQFRV 6as7 A 2.95 BS02 dna C 0 S785 R834 A837 Y839 G841 G842 F962 K1051 R1222 S444 R469 A472 Y474 G476 G477 F584 K673 R844 2.7.7.7 0000166,0003676,0003677,0003887,1902975 remove_due_to_license_issue P09884 29555682 109 ~ 121 EQVFHFYWLDAYEDQYNQPGVVFLFGKVWIESAETHVSCCVMVKNIERTLYFLPREMKIDLNTGKETGTPISMKDVYEEFDEKIATKYKIMKFKSKPVEKNYAFEIPDVPEKSEYLEVKYSAEMPQLPQDLKGETFSHVFGTNTSSLELFLMNRKIKGPCWLEVKSPQLLNQPVSWCKAEAMALKPDLVNVIKDVSPPPLVVMAFSMKTMQNAKNHQNEIIAMAALVHHSFALDKAAPKPPFQSHFCVVSKPKDCIFPYAFKEVIEKKNVKVEVAATERTLLGFFLAKVHKIDPDIIVGHNIYGFELEVLLQRINVCKAPHWSKIGRLKRSNMPKLGFGERNATCGRMICDVEISAKELIRCKSYHLSELVQQILKTERVVIPMENIQNMYSESSQLLYLLEHTWKDAKFILQIMCELNVLPLALQITNIAGNIMSRTLMGGRSERNEFLLLHAFYENNYIVPDKQIFRKKAAYAGGLVLDPKVGFYDKFILLLDFNSLYPSIIQEFNICFTTVQRVEQIPELPDPSLEMGILPREIRKLVERRKQVKQLMKQQDLNPDLILQYDIRQKALKLTANSMYGCLGFSYSRFYAKPLAALVTYKGREILMHTKEMVQKMNLEVIYGDTDSIMINTNSTNLEEVFKLGNKVKSEVNKLYKLLEIDIDGVFKSLLLLKKKKYAALVVEPTSDGNYVTKQELKGLDIVRRDWCDLAKDTGNFVIGQILSDQSRDTIVENIQKRLIEIGENVLNGSVPVSQFEINKALTKDPQDYPDKKSLPHVHVALWINSQGGRKVKAGDTVSYVICQDGSNLTASQRAYAPEQLQKQDNLTIDTQYYLAQQIHPVVARICEPIDGIDAVLIATWLGLDPTQFRV 6as8 A 2.101 BS01 BTG A 1 F1 N44 D45 Y46 D51 D53 K132 A134 N140 R142 F1 N44 D45 Y46 D51 D53 K128 A130 N136 R138 ? 0007155,0009289 remove_due_to_license_issue Q1RBS0 29507247 201 FSCNVDGGSSIGAGTTSVYVNLDPVIQPGQNLVVDLSQHISCWNDYGGWYDTDHINLVQGSAFAGSLQSYKGSLYWNNVTYPFPLTTNTNVLDIGDKTPMPLPLKLYITPVGVVIKAGEVIARIHMYKIATLGSGNPRNFTWNIISNNSVVMP 6asb C 2.85 BS01 dna A 0 R35 R36 R38 K69 Q70 S71 R75 R1 R2 R4 K35 Q36 S37 R41 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCGEAGKEDTVEGEEEKFGLSLMECTICNEIVHPGCLKMGKAEGVINAEIPNCWECPRCTQEG 6asb C 2.85 BS02 dna B 0 R35 T37 H54 R67 M68 P83 H84 R1 T3 H20 R33 M34 P49 H50 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCGEAGKEDTVEGEEEKFGLSLMECTICNEIVHPGCLKMGKAEGVINAEIPNCWECPRCTQEG 6asb F 2.85 BS01 dna D 0 R35 R36 R38 K69 Q70 S71 R75 R1 R2 R4 K35 Q36 S37 R41 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCFGLSLMECTICNEIVHPGCIPNCWECRC 6asb F 2.85 BS02 dna E 0 R35 T37 R40 H54 R67 M68 K69 Q70 P83 H84 R1 T3 R6 H20 R33 M34 K35 Q36 P49 H50 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCFGLSLMECTICNEIVHPGCIPNCWECRC 6asb I 2.85 BS01 dna G 0 R35 R36 R38 K69 Q70 S71 R75 N118 R3 R4 R6 K37 Q38 S39 R43 N86 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRRRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCGEAGKEDTVEGEEEKFGLSLMECTICNEIVHPGCLKMGKAEGVINAEIPNCWECPRCTQEGR 6asb I 2.85 BS02 dna H 0 R33 R34 R35 T37 R67 M68 Q70 P83 H84 R1 R2 R3 T5 R35 M36 Q38 P51 H52 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRRRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCGEAGKEDTVEGEEEKFGLSLMECTICNEIVHPGCLKMGKAEGVINAEIPNCWECPRCTQEGR 6asb L 2.85 BS01 dna J 0 R36 R38 K69 Q70 S71 R4 R6 K37 Q38 S39 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRRRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCGEAGKEDTGEEEKFGLSLMECTICNEIVHPGCEGVINAEIPNCWECPRCTQ 6asb L 2.85 BS02 dna K 0 R33 R34 R40 R67 M68 K69 Q70 P83 H84 R1 R2 R8 R35 M36 K37 Q38 P51 H52 ? 0003677,0008270 remove_due_to_license_issue Q6PCT2 29276034 1 ~ 12 RRRRTRCRRCRACVRTECGDCHFCRDMKKFGGPGRMKQSCLLRQCTAPVLPHTAVCLLCGEAGKEDTGEEEKFGLSLMECTICNEIVHPGCEGVINAEIPNCWECPRCTQ 6asd C 1.85 BS01 dna A 0 K587 K589 T607 Y608 H616 Q617 K620 K2 K4 T22 Y23 H31 Q32 K35 1.14.11.80 0003677,0008270 remove_due_to_license_issue Q8NFU7 29276034 1 ~ 12 GKRKRCGVCEPCQQKTNCGECTYCKNRKNSHQICKKRKCEELKKK 6asd C 1.85 BS02 dna B 0 K587 R588 H616 K623 L627 K2 R3 H31 K38 L42 1.14.11.80 0003677,0008270 remove_due_to_license_issue Q8NFU7 29276034 1 ~ 12 GKRKRCGVCEPCQQKTNCGECTYCKNRKNSHQICKKRKCEELKKK 6asu A 2.316 BS02 BVS A 1 R339 E434 G459 L461 D462 W541 M631 D633 R328 E422 G447 L449 D450 W529 M619 D621 D271 E273 R339 E434 D462 D633 D267 E269 R328 E422 D450 D621 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=6.1uM remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAAVLRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKADVNGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAA 6au2 A 1.63 BS01 CGJ A 1 F296 F297 G300 C329 F332 I333 S392 F106 F107 G110 C139 F142 I143 S202 2.1.1.366 remove_due_to_license_issue Q15047 31327677 501 ENLYFQGDLIVSMRILGKKRTKTWHKGTLIAIQTVGPGKKYKVKFDNKGKSLLSGNHIAYDYHPPADKLYVGSRVVAKYKGNQVWLYAGIVAETPNVKNKLRFLIFFDDGYASYVTQSELYPICRPLKKTWEDIEDISCRDFIEEYVTAYPNRPMVLLKSGQLIKTEWEGTWWKSRVEEVDGSLVRILFLDDKRCEWIYRGSTRLEPMFS 6au9 A 2.1 BS02 BXS A 1 V118 R339 E434 G459 L461 D462 M515 W541 M631 D633 V117 R330 E422 G447 L449 D450 M503 W529 M619 D621 D271 E273 R339 E434 D462 D633 D270 E272 R330 E422 D450 D621 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=1.1uM remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAALRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6aud A 2.015 BS01 BWY A 1 W812 K833 I879 E880 V882 M953 I963 D964 W573 K594 I640 E641 V643 M714 I724 D725 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 remove_due_to_license_issue P48736 28947940 1201 MSEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKMAEQDFVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKEECDRKFRVKIRGIDIPVLPRNTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCLLYYVNLLLIDHRFLLRRGEYVLHMWQISGFNADKLTSATNPDKENSMSISILLDNHPIAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCTVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTGAFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPQLTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHLV 6aum A 2.95 BS02 BXV A 1 F267 D335 W336 M339 I375 Y383 L408 M419 Y466 F266 D334 W335 M338 I374 Y382 L407 M418 Y465 F267 D335 W336 N378 Y383 Y466 D496 H524 F266 D334 W335 N377 Y382 Y465 D495 H523 3.1.3.76,3.3.2.10 0000287,0001558,0003824,0004301,0005737,0005777,0005782,0005829,0006629,0009056,0009636,0010628,0015643,0016311,0016787,0016791,0033885,0042577,0042632,0042803,0046272,0046839,0046872,0052642,0070062,0090181,0097176 remove_due_to_license_issue Ki=156nM, IC50=0.400000nM P34913 29366648 603 TLRAAVFDLDGVLALPAVFGVLGRTEEALALPRGLLNDAFQKGGPEGATTRLMKGEITLSQWIPLMEENCRKCSETAKVCLPKNFSIKEIFDKAISARKINRPMLQAALMLRKKGFTTAILTNTWLDDRAERDGLAQLMCELKMHFDFLIESCQVGMVKPEPQIYKFLLDTLKASPSEVVFLDDIGANLKPARDLGMVTILVQDTDTALKELEKVTGIQLLNTPAPLPTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDARN 6avi A 2.29 BS02 KNA A 1 C285 R288 I341 S342 E343 C67 R70 I123 S124 E125 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 30575522 502 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 6awn A 3.62 BS01 8PR A 1 Y95 D98 A169 F335 T439 G442 V501 Y22 D25 A96 F262 T366 G369 V428 ? 0016020 remove_due_to_license_issue Ki=0.42nM, Kd=0.130000nM, IC50=0.200000nM P31645 29379174 705 GSQGERETWGKKVDFLLSVIGYAVDLGNVWRFPYICAQNGGGAFLLPYTIMAIFGGIPLFYMELALGQYHRNGCISIWRKICPIFKGIGYAICIIAFYIASYYNTIMAWALYYLISSFTDQLPWTSCKNSWNTGNCTNYFSEDNITWTLHSTSPAEEFYTRHVLQIHRSKGLQDLGGISWQLALCIMLIFTVIYFSIWKGVKTSGKVVWVTATFPYIALSVLLVRGATLPGAWRGVLFYLKPNWQKLLETGVWIDAAAQIFFSLGPGFGVLLAFASYNKFNNNCYQDALVTSVVNCMTSFVSGFVIFTVLGYMAEMRNEDVSEVAKDAGPSLLFITYAEAIANMPASTFFAIIFFLMLITLGLDSTFAGLEGVITAVLDEFPHVWAKRRERFVLAVVITCFFGSLVTLTFGGAYVVKLLEEYATGPAVLTVALIEAVAVSWFYGITQFCRDVKEMLGFSPGWFWRICWVAISPLFLLFIIASFLMSPPQLRLFQYNYPYWSIILGYAIGTSSFICIPTYIAYRLIITPGTFKERIIKSITPETP 6awo A 3.534 BS01 SRE A 1 Y95 D98 A169 I172 F335 F341 S438 G442 Y22 D25 A96 I99 F262 F268 S365 G369 ? 0016020 remove_due_to_license_issue IC50=3nM, Kd=0.290000nM, Ki=0.9nM P31645 29379174 701 GSQGERETWGKKVDFLLSVIGYAVDLGNVWRFPYICAQNGGGAFLLPYTIMAIFGGIPLFYMELALGQYHRNGCISIWRKICPIFKGIGYAICIIAFYIASYYNTIMAWALYYLISSFTDQLPWTSCKNSWNTGNCTNYFSEDNITWTLHSTSPAEEFYTRHVLQIHRSKGLQDLGGISWQLALCIMLIFTVIYFSIWKGVKTSGKVVWVTATFPYIALSVLLVRGATLPGAWRGVLFYLKPNWQKLLETGVWIDAAAQIFFSLGPGFGVLLAFASYNKFNNNCYQDALVTSVVNCMTSFVSGFVIFTVLGYMAEMRNEDVSEVAKDAGPSLLFITYAEAIANMPASTFFAIIFFLMLITLGLDSSFAGLEGVITAVLDEFPHVWAKRRERFVLAVVITCFFGSLVTLTFGGAYVVKLLEEYATGPAVLTVALIEAVAVSWFYGITQFCRDVKEMLGFSPGWFWRICWVAISPLFLLFIIASFLMSPPQLRLFQYNYPYWSIILGYAIGTSSFICIPTYIAYRLIITPGTFKERIIKSITPETP 6awp A 3.8 BS01 FVX A 1 Y95 A96 D98 I172 F335 S336 F341 S438 G442 Y22 A23 D25 I99 F262 S263 F268 S365 G369 ? 0016020 remove_due_to_license_issue Ki=14nM P31645 29379174 701 GSQGERETWGKKVDFLLSVIGYAVDLGNVWRFPYICAQNGGGAFLLPYTIMAIFGGIPLFYMELALGQYHRNGCISIWRKICPIFKGIGYAICIIAFYIASYYNTIMAWALYYLISSFTDQLPWTSCKNSWNTGNCTNYFSEDNITWTLHSTSPAEEFYTRHVLQIHRSKGLQDLGGISWQLALCIMLIFTVIYFSIWKGVKTSGKVVWVTATFPYIALSVLLVRGATLPGAWRGVLFYLKPNWQKLLETGVWIDAAAQIFFSLGPGFGVLLAFASYNKFNNNCYQDALVTSVVNCMTSFVSGFVIFTVLGYMAEMRNEDVSEVAKDAGPSLLFITYAEAIANMPASTFFAIIFFLMLITLGLDSSFAGLEGVITAVLDEFPHVWAKRRERFVLAVVITCFFGSLVTLTFGGAYVVKLLEEYATGPAVLTVALIEAVAVSWFYGITQFCRDVKEMLGFSPGWFWRICWVAISPLFLLFIIASFLMSPPQLRLFQYNYPYWSIILGYAIGTSSFICIPTYIAYRLIITPGTFKERIIKSITPETP 6ax1 A 2.26 BS01 C0S A 1 G50 A51 S122 M123 N152 G33 A34 S105 M106 N135 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 remove_due_to_license_issue IC50=0.380000nM Q99685 29148769 401 DLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTATA 6axb A 1.8 BS02 C0V A 1 V118 R339 E434 G459 L461 D462 M515 W541 M631 D633 V117 R330 E423 G448 L450 D451 M504 W530 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R330 E423 D451 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=0.5uM remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAALRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNADVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6axq A 1.3 BS01 C2Y A 1 V1115 L1120 N1168 V1174 V31 L36 N84 V90 2.3.1.-,2.3.1.48 ic50=99000nM remove_due_to_license_issue IC50=99000nM Q92793 29155580 1203 FKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL 6ay3 A 1.391 BS01 C3J A 1 L1109 P1110 F1111 V1115 N1168 R1173 V1174 L27 P28 F29 V33 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=9.5nM remove_due_to_license_issue EC50=2200nM, IC50=9.5nM Q92793 29155580 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 6ay5 A 1.44 BS01 C3V A 1 L1109 P1110 V1115 L1120 Y1167 N1168 R1173 V1174 L27 P28 V33 L38 Y85 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=69nM remove_due_to_license_issue IC50=64.0nM Q92793 29155580 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 6ayd A 3.0 BS01 C2J A 1 A65 K67 E89 L120 E121 L174 I185 D186 A32 K34 E56 L87 E88 L141 I152 D153 D167 K169 N172 D186 L193 T204 D134 K136 N139 D153 L160 T171 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005730,0005737,0005829,0005886,0006338,0006468,0006915,0007346,0008134,0022898,0030145,0035175,0035402,0035403,0035979,0043024,0043066,0043433,0044022,0044023,0044024,0044025,0045824,0045893,0046777,0046872,0050821,0060045,0070561,0071346,0072354,0072371,0072518,0090336,0106310,0140823,0140855,0140857,1902033,1904263,1905062,1990244,1990748 remove_due_to_license_issue P11309 29057057 401 LESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 6ayh A 2.05 BS01 C3G A 1 R71 A72 H75 F76 E99 K127 L161 T165 Y166 R66 A67 H70 F71 E94 K122 L156 T160 Y161 0003677 Kd=2.7uM remove_due_to_license_issue 29269393 302 NKLTEPLPTRMRILRAARQCFAENGFHSTSMKTICKASDMSPGTLYHHFPSKEALIEAIILEDQERALTHFREPLEGVGLVDYLVESTIAVTREDYAQRALVVEIMAEGMRNPQVAEMLTNKYHTIIASLVARFNDAQAKGEIGADVDKEMAARLLLATTYGVLSDSSSAENARHVSFATTLRTMLTGLLKC 6ayi A 2.09 BS01 C3G A 1 R69 A70 R73 E97 K125 T163 Y164 R59 A60 R63 E87 K115 T153 Y154 ? 0000976,0003677,0003700,0006351,0006355,0045892 Kd=0.21uM remove_due_to_license_issue P0ACT6 29269393 201 PTRTRILNAAREIFSENGFHSASMKAICKSCAISPGTLYHHFISKEALIQAIILQDQERALARFREPIEGIHFVDYMVESIVSLTHEAFGQRALVVEIMAEGMRNPQVAAMLKNKHMTITEFVAQRMRDAQQKGEISPDINTAMTSRLLLDLTYGVLADIEAEDLAREASFAQGLRAMIGGIL 6ayo A 1.67 BS01 C1Y A 1 M9 I50 V76 A77 G78 F151 I152 C170 M172 E173 D196 F206 M10 I51 V77 A78 G79 F152 I153 C171 M173 E174 D197 F207 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=5.1nM remove_due_to_license_issue Q0PC20 30339406 301 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ayo B 1.67 BS01 C1Y B 1 I50 V76 A77 G78 F151 I152 C170 M172 E173 D196 F206 I51 V77 A78 G79 F152 I153 C171 M173 E174 D197 F207 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=5.1nM remove_due_to_license_issue Q0PC20 30339406 301 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ayq A 1.42 BS01 TDI A 1 M9 I50 V76 A77 G78 F151 I152 C170 E171 M172 E173 D196 M10 I51 V77 A78 G79 F152 I153 C171 E172 M173 E174 D197 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=6.5nM remove_due_to_license_issue Q0PC20 30339406 301 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ayq B 1.42 BS01 TDI B 1 M9 I50 V76 A77 G78 F151 I152 C170 E171 M172 E173 D196 M9 I50 V76 A77 G78 F151 I152 C170 E171 M172 E173 D196 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=6.5nM remove_due_to_license_issue Q0PC20 30339406 301 MKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ayr A 1.95 BS01 BIG A 1 I50 V76 A77 G78 F151 I152 C170 E171 M172 E173 D196 F206 I51 V77 A78 G79 F152 I153 C171 E172 M173 E174 D197 F207 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=4.1nM remove_due_to_license_issue Q0PC20 30339406 301 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ayr A 1.95 BS02 BIG B 1 I102 F105 I103 F106 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=4.1nM remove_due_to_license_issue Q0PC20 30339406 301 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ayr B 1.95 BS01 BIG B 1 I50 V76 A77 G78 F151 I152 C170 M172 E173 D196 I51 V77 A78 G79 F152 I153 C171 M173 E174 D197 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Ki=4.1nM remove_due_to_license_issue Q0PC20 30339406 301 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ays A 1.7 BS01 HT6 A 1 I50 V76 A77 G78 F151 I152 C170 E171 M172 E173 D196 I51 V77 A78 G79 F152 I153 C171 E172 M173 E174 D197 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q0PC20 30339406 302 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ays A 1.7 BS02 HT6 B 1 I102 F105 I103 F106 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q0PC20 30339406 303 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ays B 1.7 BS01 HT6 A 1 F105 H107 F106 H108 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q0PC20 30339406 302 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6ays B 1.7 BS02 HT6 B 1 I50 V76 A77 G78 F151 I152 C170 E171 M172 E173 D196 F206 I51 V77 A78 G79 F152 I153 C171 E172 M173 E174 D197 F207 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 remove_due_to_license_issue Q0PC20 30339406 303 GMKIAILGAMSEEITPLLETLKDYTKIEHANNTYYFAKYKDHELVLAYSKIGKVNSTLSASVMIEKFGAQVLLFTGVAGAFNPELEIGDLLYATKLAQYDLDITAFGHPLGFVPGNEIFIKTDEKLNNLALEVAKELNIKLRAGIIATGDEFICDEAKKAKIREIFNADACEMEGASVALVCDALKVPCFILRAMSDKAGEKAEFDFDEFVINSAKISANFVLKMCEKL 6b0o A 1.552 BS01 dna B 0 R321 K332 Y334 H339 K346 F364 R366 Q369 R372 H373 R376 R390 S393 R394 H397 H401 T404 R424 E427 R430 R3 K14 Y16 H21 K28 F46 R48 Q51 R54 H55 R58 R72 S75 R76 H79 H83 T86 R106 E109 R112 ? remove_due_to_license_issue P19544 29294058 1 ~ 13 HMRPFMCAYPGCNKRYFKLSHLQMHSRKHTGEKPYQCDFKDCERRFSRSDQLKRHQRRHTGVKPFQCKTCQRKFSRSDHLKTHTRTHTGEKPFSCRWPSCQKKFARSDELVRHHNMHQR 6b0o A 1.552 BS02 dna C 0 Y353 S367 K371 D396 K399 S425 R430 Y35 S49 K53 D78 K81 S107 R112 ? remove_due_to_license_issue P19544 29294058 1 ~ 13 HMRPFMCAYPGCNKRYFKLSHLQMHSRKHTGEKPYQCDFKDCERRFSRSDQLKRHQRRHTGVKPFQCKTCQRKFSRSDHLKTHTRTHTGEKPFSCRWPSCQKKFARSDELVRHHNMHQR 6b0o D 1.552 BS01 dna E 0 R362 R366 Q369 R372 H373 R376 R390 S393 R394 H397 H401 T404 R424 E427 R430 R42 R46 Q49 R52 H53 R56 R70 S73 R74 H77 H81 T84 R104 E107 R110 ? remove_due_to_license_issue P19544 29294058 1 ~ 13 RPFMCAYPGCNKRYFKLSHLQMHSRKHTGEKPYQCDFKDCERRFSRSDQLKRHQRRHTGVKPFQCKTCQRKFSRSDHLKTHTRTHTGEKPFSCRWPSCQKKFARSDELVRHHNMHQ 6b0o D 1.552 BS02 dna F 0 S367 K399 S425 R430 S47 K79 S105 R110 ? remove_due_to_license_issue P19544 29294058 1 ~ 13 RPFMCAYPGCNKRYFKLSHLQMHSRKHTGEKPYQCDFKDCERRFSRSDQLKRHQRRHTGVKPFQCKTCQRKFSRSDHLKTHTRTHTGEKPFSCRWPSCQKKFARSDELVRHHNMHQ 6b0v A 1.29 BS01 C8G A 1 C12 K16 A59 G60 E63 Y64 R68 D69 M72 Q99 I100 V103 C12 K16 A59 G60 E63 Y64 R68 D69 M72 Q99 I100 V103 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 29760531 203 MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6b0y A 1.43 BS01 8ZG A 1 C12 K16 P34 T58 A59 G60 E62 R68 M72 H95 Y96 Q99 V103 C12 K16 P34 T58 A59 G60 E62 R68 M72 H95 Y96 Q99 V103 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 29760531 203 MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKE 6b14 H 1.64 BS01 rna R 0 Y34 P56 Y57 S58 S60 Q102 Y104 R105 R106 R110 Y31 P53 Y54 S55 S57 Q99 Y101 R102 R103 R107 remove_due_to_license_issue 29309709 2 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPYSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARQGYRRRSGRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 6b14 L 1.64 BS01 rna R 0 S92 F95 N97 S92 F95 N97 remove_due_to_license_issue 29309709 2 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSYSFPNTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 6b16 A 2.285 BS01 C7Y A 1 A297 E345 Y346 L347 D393 L396 T406 A47 E88 Y89 L90 D136 L139 T149 N389 K391 D393 N394 D407 P416 T427 N132 K134 D136 N137 D150 P159 T170 2.7.11.1 0004672,0005524,0006468 Ki=32nM remove_due_to_license_issue Ki=32nM Q13153 27346791 601 EEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQQPKKELIINEILVMRENKNPNIVNYLDSYLDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK 6b1c A 2.163 BS01 C9J A 1 P1 M2 K32 Y36 H62 S63 I64 M101 V106 P1 M2 K32 Y36 H62 S63 I64 M101 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.111uM remove_due_to_license_issue Kd=111nM, Ki=75nM P14174 29259749 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1c A 2.163 BS02 C9J B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.111uM remove_due_to_license_issue Kd=111nM, Ki=75nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1c C 2.163 BS01 C9J A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Kd=111nM, Ki=75nM P14174 29259749 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1e A 1.77 BS01 LF7 A 1 E205 E206 Y547 S630 Y631 Y662 Y666 V711 E167 E168 Y509 S592 Y593 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue IC50=3.5nM P27487 30815539 801 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 6b1f A 1.44 BS01 C8Y A 1 S69 W104 S129 T215 T234 T236 S48 W83 S108 T194 T213 T215 S69 K72 S129 E165 K233 T236 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 29627985 301 ATALTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6b1h A 1.8 BS01 C8Y A 1 S70 W105 S130 N170 T216 T235 G236 T237 S48 W83 S108 N148 T194 T213 G214 T215 S70 K73 S130 E166 K234 T237 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 29627985 301 ATALTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6b1j A 1.6 BS01 C8V A 1 S70 W105 S130 N170 T216 T235 G236 T237 C238 S48 W83 S108 N148 T194 T213 G214 T215 C216 S70 K73 S130 E166 K234 T237 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 29627985 301 ATALTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6b1k A 1.17 BS01 C9G A 1 P1 M2 K32 Y36 H62 I64 V106 F113 P1 M2 K32 Y36 H62 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.213uM remove_due_to_license_issue Ki=363nM, Kd=213nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1k A 1.17 BS02 C9G B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.213uM remove_due_to_license_issue Ki=363nM, Kd=213nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1k C 1.17 BS01 C9G A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.213uM remove_due_to_license_issue Ki=363nM, Kd=213nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1k C 1.17 BS02 C9G C 1 P1 M2 K32 P33 Y36 H62 S63 I64 V106 P1 M2 K32 P33 Y36 H62 S63 I64 V106 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.213uM remove_due_to_license_issue Ki=363nM, Kd=213nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b1o A 1.91 BS01 C8S A 1 E205 E206 F357 Y547 S630 Y631 Y662 Y666 V711 E167 E168 F319 Y509 S592 Y593 Y624 Y628 V673 Y547 S630 Y631 D708 H740 Y509 S592 Y593 D670 H702 3.4.14.5 0001618,0001662,0001666,0002020,0004177,0004252,0005102,0005515,0005576,0005765,0005886,0005925,0006508,0007155,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016486,0019065,0030027,0030139,0031258,0031295,0033632,0035641,0036343,0042110,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0046813,0050919,0061025,0070062,0070161,0090024,0120116 remove_due_to_license_issue P27487 30815539 811 TRKTYTLTDYLKNTYRLKLYSLRWISDHEYLYKQENNILVFNAEYGNSSVFLENSTFDEFGHSINDYSISPDGQFILLEYNYVKQWRHSYTASYDIYDLNKRQLITEERIPNNTQWVTWSPVGHKLAYVWNNDIYVKIEPNLPSYRITWTGKEDIIYNGITDWVYEEEVFSAYSALWWSPNGTFLAYAQFNDTEVPLIEYSFYSDESLQYPKTVRVPYPKAGAVNPTVKFFVVNTDSLSSVTNATSIQITAPASMLIGDHYLCDVTWATQERISLQWLRRIQNYSVMDICDYDESSGRWNCLVARQHIEMSTTGWVGRFRPSEPHFTLDGNSFYKIISNEEGYRHICYFQIDKKDCTFITKGTWEVIGIEALTSDYLYYISNEYKGMPGGRNLYKIQLSDYTKVTCLSCELNPERCQYYSVSFSKEAKYYQLRCSGPGLPLYTLHSSVNDKGLRVLEDNSALDKMLQNVQMPSKKLDFIILNETKFWYQMILPPHFDKSKKYPLLLDVYAGPCSQKADTVFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINRRLGTFEVEDQIEAARQFSKMGFVDNKRIAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDVGVDFQAMWYTDEDHGIASSTAHQHIYTHMSHFIKQCFSLP 6b1w A 1.73 BS02 C8V A 1 S70 W105 S130 N132 N170 T237 C238 S48 W83 S108 N110 N148 T215 C216 S70 K73 S130 E166 K234 T237 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 29627985 304 ATALTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6b1x A 1.45 BS01 C9D A 1 S70 W105 S130 L167 N170 T216 T235 G236 T237 S48 W83 S108 L145 N148 T194 T213 G214 T215 S70 K73 S130 E166 K234 T237 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 29627985 301 ATALTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6b1y A 1.8 BS01 CD7 A 1 S70 W105 S130 N132 N170 T237 C238 S48 W83 S108 N110 N148 T215 C216 S70 K73 S130 E166 K234 T237 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 29627985 301 ATALTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6b22 A 1.93 BS01 C8Y A 1 S81 S128 S219 G220 W221 R261 S50 S97 S188 G189 W190 R230 S81 K84 S128 Y133 W167 W221 S50 K53 S97 Y102 W136 W190 ? 0008658,0008800,0016787 remove_due_to_license_issue Q8RLA6 29627985 301 HISSQQHEKAIKSYFDEAQTQGVIIIKEGKNLSTYGNALARANKEYVPASTFKMLNALIGLENHKATTNEIFKWDGKKRTYPMWEKDMTLGEAMALSAVPVYQELARRTGLELMQKEVKRVNFGNTNIGTQVDNFWLVGPLKITPVQEVNFADDLAHNRLPFKLETQEEVKKMLLIKEVNGSKIYAKSGWGMGVTPQVGWLTGWVEQANGKKIPFSLNLEMKEGMSGSIRNEITYKSLENLGII 6b2c A 2.0 BS01 C9Y B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Ki=90nM, Kd=94nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b2c B 2.0 BS01 C9Y B 1 P1 K32 Y36 H62 I64 M101 V106 F113 P1 K32 Y36 H62 I64 M101 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Kd=0.094uM remove_due_to_license_issue Ki=90nM, Kd=94nM P14174 29259749 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6b2p A 3.01 BS01 CJJ A 1 G18 V25 A38 M92 E93 Y94 V95 G97 M145 M155 G15 V22 A35 M89 E90 Y91 V92 G94 M142 M152 D138 K140 N143 D156 T179 D135 K137 N140 D153 T156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=<1.3nM P9WI81 29259738 301 PSHLSDRYELGEILGFGGMSEVHLARDLRLHRDVAVKVLRADLARDPSFYLRFRREAQNAAALNHPAIVAVYDTGEAETPAGPLPYIVMEYVDGVTLRDIVHTEGPMTPKRAIEVIADACQALNFSHQNGIIHRDVKPANIMISATNAVKVMDFGTAQYLSPEQARGDSVDARSDVYSLGCVLYEVLTGEPPFTGDSPVSVAYQHVREDPIPPSARHEGLSADLDAVVLKALAKNPENRYQTAAEMRADLVRVHN 6b2q A 2.88 BS01 CJJ A 1 I19 A20 V27 A40 M95 E96 V98 G100 L148 T158 I17 A18 V25 A38 M86 E87 V89 G91 L139 T149 D141 K143 N146 D159 T180 D132 K134 N137 D150 T158 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=9.0nM P9WI83 29259738 301 PRVGVTLSGRYRLQRLIATGGMGQVWEAVDNRLGRRVAVKVLKSEFSSDPEFIERFRAEARTTAMLNHPGIASVHDYGESTAYLVMELVNGEPLNSVLKRTGRLSLRHALDMLEQTGRALQIAHAAGLVHRDVKPGNILITPTGQVKITDFGIAKAGTAQYIAPEQALGHDASPASDVYSLGVVGYEAVSGKRPFAGDGALTVAMKHIKEPPPPLPPDLPPNVRELIEITLVKNPAMRYRSGGPFADAVAAVRAGRRPPRPS 6b2q D 2.88 BS01 CJJ D 1 I19 A20 V27 A40 K42 V98 G100 L148 T158 I17 A18 V25 A38 K40 V90 G92 L140 T150 D141 K143 N146 D159 T180 D133 K135 N138 D151 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=9.0nM P9WI83 29259738 300 PRVGVTLSGRYRLQRLIATGGMGQVWEAVDNRLGRRVAVKVLKSEFSSDPEFIERFRAEARTTAMLNHPGIASVHDYGESRTAYLVMELVNGEPLNSVLKRTGRLSLRHALDMLEQTGRALQIAHAAGLVHRDVKPGNILITPTGQVKITDFGIAKVMGTAQYIAPEQALGSPASDVYSLGVVGYEAVSGKRPFAGDGALTVAMKHIKEPPPPLPPDLPPNVRELIEITLVKNPAMRYRSGGPFADAVAAVRAGRRPPRP 6b30 A 2.69 BS01 CFG A 1 Q286 L287 H323 M365 F377 E379 F388 Q22 L23 H59 M101 F113 E115 F124 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P51449 29262987 600 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQH 6b31 A 3.18 BS01 CFJ A 1 C320 H323 M365 A368 F377 F378 F388 C56 H59 M101 A104 F113 F114 F124 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=47nM P51449 29342416 600 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPI 6b33 A 2.48 BS01 CF7 A 1 Q286 C320 L324 V361 M365 A368 F377 F388 H479 Q22 C56 L60 V97 M101 A104 F113 F124 H215 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P51449 31659845 1000 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVER 6b3e A 3.06 BS01 CJM A 1 I733 A754 Y815 M816 H818 D819 L866 I17 A38 Y89 M90 H92 D93 L140 D859 K861 N864 D877 S889 T898 D133 K135 N138 D151 S163 T172 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue Q9NYV4 29266803 1102 SDWGKRCVDKFDIIGIIGEGTYGQVYKAKDKDTGELVALKKVRLDNEKEGFPITAIREIKILRQLIHRSVVNMKEIVTDKGAFYLVFEYMDHDLMGLLESGLVHFSEDHIKSFMKQLMEGLEYCHKKNFLHRDIKCSNILLNNSGQIKLADFGLARLYNSEESRPYTNKVITLWYRPPELLLGEERYTPAIDVWSCGCILGELFTKKPIFQANLELAQLELISRLCGSPCPAVWPDVIKLPYFNTMKPKKQYRRRLREEFSFIPSAALDLLDHMLTLDPSKRCTAEQTLQSDFLKDVELSKMAPPDLPHW 6b3k H 2.09 BS01 rna R 0 Y34 S55 P56 Y57 S58 S60 Q102 Y104 R105 R110 Y31 S52 P53 Y54 S55 S57 Q99 Y101 R102 R107 remove_due_to_license_issue 29309709 2 ~ 84 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPYSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARQGYRRRSGRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 6b3k L 2.09 BS01 rna R 0 S92 F95 S92 F95 remove_due_to_license_issue 29309709 2 ~ 84 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSYSFPSTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 6b3v A 1.601 BS02 7DQ A 1 R207 G210 R190 G193 2.7.1.33 0004594,0005524,0005634,0005737,0005829,0005975,0015937,0016301,0016310,0019842,0042803,1905502 Kd=203pM remove_due_to_license_issue Q9H999 30352999 505 SPWFGMDIGGTLVKLSYFEPIDITAEEEQEEVESLKSIRKYLTSNVAYGSTGIRDVHLELKDLTLFGRRGNLHFIRFPTQDLPTFIQMGRDTVLCATGGGAYKFEKDFRTIGNLHLHKLDELDCLVKGLLYIDSVSFNGQAECYYFANASEPERCQKMPFNLDDPYPLLVVNIGSGVSILAVHSKDNYKRVTGTSLGGGTFLGLCSLLTGCESFEEALEMASKGDSTQADKLVRDIYGGDYERFGLPGWAVASSFGNMIYKEKRESVSKEDLARATLVTITNNIGSVARMCAVNEKINRVVFVGNFLRVNTLSMKLLAYALDYWSKGQLKALFLEHEGYFGAVGALLGLPNF 6b41 A 2.61 BS01 CJV A 1 S178 E179 D180 H181 F238 C241 A242 Y276 M278 Y319 M322 Y323 G326 C329 E363 V371 S174 E175 D176 H177 F234 C237 A238 Y272 M274 Y315 M318 Y319 G322 C325 E359 V367 ? 0000122,0000165,0000400,0000403,0000781,0000785,0000976,0001933,0002076,0003677,0003682,0003690,0005515,0005634,0005654,0005737,0005788,0005829,0006281,0006325,0006357,0006974,0008285,0009411,0010332,0016363,0017053,0030511,0030674,0032154,0032991,0035097,0043433,0044665,0045064,0045668,0045736,0045786,0045815,0045892,0045944,0046329,0051219,0070412,0071339 remove_due_to_license_issue O00255 29284071 701 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVIPTNVPELTFQPSPAPDGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEASALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSGTVAGTARGPVLTFQSEKMKGMKELLVATKINSSAIKLQLTA 6b4d A 1.196 BS02 53X A 1 V121 F131 L198 T200 P202 V118 F127 L194 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.78uM remove_due_to_license_issue Ki=780nM P00918 28947941 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6b4h C 2.17 BS01 IHP C 1 H221 K225 R228 K327 K374 W401 H10 K14 R17 K116 K163 W190 ? 0005643,0016973 remove_due_to_license_issue G0S7F3 29899397 601 GPHMRYVEIHRNLKGLRKYMAEQAKTNLKLKQRMGDMRREIRKSVGQLTTGGMAANKDKQQKIKSILTEALSNQVESALVDPNNFVVEPRKPVEGATNNDPLLPSIFVYLINIFAKAAISQFINEAGARPETADPVGICVAAILSEPDFLWRGASLIDILIAKFRIVCPVLFGYRGSEKTEQGRQRLGWWKESGQWISEQQHMDRMTGLGAGFAAISLRKFALSKKQNPYPPRFYWMAMAKIVNTPPAEISNTQCVVLKAMVQNYEAKFIEFYGSAAIAALRTALIDFPARAPHKSAAVNSLEVLAQMLKRDTGLDLG 6b4h C 2.17 BS02 IHP C 2 S435 K436 K437 S224 K225 K226 ? 0005643,0016973 remove_due_to_license_issue G0S7F3 29899397 603 GPHMRYVEIHRNLKGLRKYMAEQAKTNLKLKQRMGDMRREIRKSVGQLTTGGMAANKDKQQKIKSILTEALSNQVESALVDPNNFVVEPRKPVEGATNNDPLLPSIFVYLINIFAKAAISQFINEAGARPETADPVGICVAAILSEPDFLWRGASLIDILIAKFRIVCPVLFGYRGSEKTEQGRQRLGWWKESGQWISEQQHMDRMTGLGAGFAAISLRKFALSKKQNPYPPRFYWMAMAKIVNTPPAEISNTQCVVLKAMVQNYEAKFIEFYGSAAIAALRTALIDFPARAPHKSAAVNSLEVLAQMLKRDTGLDLG 6b4l A 2.25 BS01 CJY A 1 M231 V253 R263 L267 F270 M61 V83 R93 L97 F100 ? 0042981 Ki=0.34uM remove_due_to_license_issue Ki=7300nM Q07820 25679114 401 SMDLYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6b4n A 1.3 BS01 G53 A 1 D25 A28 D29 D30 K45 I47 G48 P81 V82 D25 A28 D29 D30 K45 I47 G48 P81 V82 D25 T26 G27 D25 T26 G27 3.1.13.2,3.1.26.13 0004190,0006508 Ki=27.9pM remove_due_to_license_issue Q72498 29110408 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6b4n B 1.3 BS01 G53 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 3.1.13.2,3.1.26.13 0004190,0006508 remove_due_to_license_issue Q72498 29110408 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6b4u A 1.95 BS01 CN7 A 1 A227 F228 M250 V253 R263 T266 L267 F270 G271 A57 F58 M80 V83 R93 T96 L97 F100 G101 ? 0042981 Ki=21nM remove_due_to_license_issue Ki=1230nM Q07820 25679114 401 SMDLYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLE 6b4w A 2.9 BS01 CQ7 A 1 I531 Q541 A551 M602 E603 G605 N606 D608 L654 I663 I17 Q27 A37 M88 E89 G91 N92 D94 L140 I149 F540 D647 K649 N652 D664 T686 F26 D133 K135 N138 D150 T163 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=57nM P33981 28991472 801 NECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDVGTVNYMPPEAIKDMKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQI 6b59 A 1.638 BS02 CQS A 1 H94 G132 L198 T199 T200 P202 H91 G128 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=8.2nM remove_due_to_license_issue Ki=8.2nM P00918 29259754 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6b5a A 1.622 BS02 CQS A 1 L91 H94 V131 L198 T199 T200 L88 H91 V127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=8.2nM P00918 29259754 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6b5i A 2.6 BS01 CU4 A 1 V138 G142 F188 W195 Q310 F314 C320 T321 N475 L477 N478 F483 V112 G116 F162 W169 Q284 F288 C294 T295 N449 L451 N452 F457 N187 E286 C320 E494 N161 E260 C294 E468 1.2.1.36 0001568,0001758,0001822,0001889,0002138,0003007,0004028,0004029,0005737,0005829,0006629,0006776,0007494,0008283,0008284,0008285,0009855,0009952,0009954,0010628,0014032,0016331,0016491,0016620,0016918,0021915,0021983,0030182,0030324,0030326,0030900,0030902,0031016,0031076,0032355,0032526,0033189,0034097,0035115,0035799,0042572,0042573,0042574,0042904,0043010,0043065,0048384,0048471,0048566,0048738,0051289,0060324,0071300,1905562 remove_due_to_license_issue O94788 29240402 601 PSPTPNLEIKYTKIFINNEWQNSESGRVFPVYNPATGEQVCEVQEADKADIDKAVQAARLAFSLGSVWRRMDASERGRLLDKLADLVERDRAVLATMESLNGGKPFLQAFYVDLQGVIKTFRYYAGWADKIHGMTIPVDGDYFTFTRHEPIGVCGQIIPWNFPLLMFAWKIAPALCCGNTVVIKPAEQTPLSALYMGALIKEAGFPPGVINILPGYGPTAGAAIASHIGIDKIAFTGSTEVGKLIQEAAGRSNLKRVTLELGGKSPNIIFADADLDYAVEQAHQGVFFNQGQCCTAGSRIFVEESIYEEFVRRSVERAKRRVVGSPFDPTTEQGPQIDKKQYNKILELIQSGVAEGAKLECGGKGLGRKGFFIEPTVFSNVTDDMRIAKEEIFGPVQEILRFKTMDEVIERANNSDFGLVAAVFTNDINKALTVSSAMQAGTVWINCYNALNAQSPFGGFKMSGNGREMGEFGLREYSEVKTVTVKIPQKNS 6b5i C 2.6 BS01 CU4 C 1 V138 G142 F188 W195 Q310 F314 C320 T321 N475 L477 N478 F483 V112 G116 F162 W169 Q284 F288 C294 T295 N449 L451 N452 F457 N187 E286 C320 E494 N161 E260 C294 E468 1.2.1.36 0001568,0001758,0001822,0001889,0002138,0003007,0004028,0004029,0005737,0005829,0006629,0006776,0007494,0008283,0008284,0008285,0009855,0009952,0009954,0010628,0014032,0016331,0016491,0016620,0016918,0021915,0021983,0030182,0030324,0030326,0030900,0030902,0031016,0031076,0032355,0032526,0033189,0034097,0035115,0035799,0042572,0042573,0042574,0042904,0043010,0043065,0048384,0048471,0048566,0048738,0051289,0060324,0071300,1905562 remove_due_to_license_issue O94788 29240402 601 PSPTPNLEIKYTKIFINNEWQNSESGRVFPVYNPATGEQVCEVQEADKADIDKAVQAARLAFSLGSVWRRMDASERGRLLDKLADLVERDRAVLATMESLNGGKPFLQAFYVDLQGVIKTFRYYAGWADKIHGMTIPVDGDYFTFTRHEPIGVCGQIIPWNFPLLMFAWKIAPALCCGNTVVIKPAEQTPLSALYMGALIKEAGFPPGVINILPGYGPTAGAAIASHIGIDKIAFTGSTEVGKLIQEAAGRSNLKRVTLELGGKSPNIIFADADLDYAVEQAHQGVFFNQGQCCTAGSRIFVEESIYEEFVRRSVERAKRRVVGSPFDPTTEQGPQIDKKQYNKILELIQSGVAEGAKLECGGKGLGRKGFFIEPTVFSNVTDDMRIAKEEIFGPVQEILRFKTMDEVIERANNSDFGLVAAVFTNDINKALTVSSAMQAGTVWINCYNALNAQSPFGGFKMSGNGREMGEFGLREYSEVKTVTVKIPQKNS 6b5j A 2.97 BS01 CV4 A 1 I469 A488 K490 T539 Y541 I542 G545 L595 D606 I25 A42 K44 T86 Y88 I89 G92 L142 D153 D588 N590 H592 N593 D606 D135 N137 H139 N140 D153 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=79nM Q59H18 29561151 801 ILLLRAGLPSHFHLQLSEIEFHEIIGSFGKVYKGRCRNKIVAIKRYRSDVDMFCREVSILCQLNHPCVIQFVGACLNDPSQFAIVTQYISGGSLFSLLHEQKRILDLQSKLIIAVDVAKGMEYLHNLTQPIIHRDLNSHNILLYEDGHAVVADFGESRFLQSGNLRWMAPEVFTQCTRYTIKADVFSYALCLWEILTGEIPFAHLKPAAAAADMAYHHIRPPIGYSIPKPISSLLIRGWNACPEGRPEFSEVVMKLEECLCNI 6b7a A 1.991 BS01 CWM A 1 L73 M74 N106 L72 M73 N105 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=32uM remove_due_to_license_issue P0A6I6 29190085 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6b7a B 1.991 BS01 CWM B 1 L73 M74 A75 N106 L72 M73 A74 N105 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=32uM remove_due_to_license_issue P0A6I6 29190085 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6b7b A 1.981 BS01 CWJ A 1 G9 M74 R88 L102 N106 G9 M71 R85 L99 N103 H18 R91 S129 H18 R88 S126 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=1280uM remove_due_to_license_issue P0A6I6 29190085 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6b7c A 1.564 BS01 CWP A 1 G9 A37 L73 M74 L102 G8 A36 L72 M73 L101 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=7.2uM remove_due_to_license_issue P0A6I6 29190085 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6b7d A 1.8 BS01 CWG A 1 A37 F70 S71 D72 L73 M74 L102 A37 F67 S68 D69 L70 M71 L99 H18 R91 S129 H18 R88 S126 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=52uM remove_due_to_license_issue P0A6I6 29190085 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6b7e B 2.104 BS01 CWA B 1 F70 M74 Y98 L102 F69 M73 Y97 L101 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=28uM remove_due_to_license_issue P0A6I6 29190085 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6b7f B 2.562 BS01 CW4 B 1 F70 L73 M74 L102 F68 L71 M72 L100 H18 K42 R91 S129 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 remove_due_to_license_issue P0A6I6 29190085 203 KRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6b7h A 2.82 BS01 CWY A 1 R64 R68 Y150 S151 A172 S173 T174 Y222 R277 S278 D279 D301 K389 R30 R34 Y95 S96 A117 S118 T119 Y167 R222 S223 D224 D246 K327 ? 0004930,0007186,0016020 remove_due_to_license_issue EC50=12nM, Ki=0.927000nM Q14832 29350927 806 RREIKIGDLVLGGLFPINEKEECGRINEDRGIQRLEAMLFAIDEINKDDYLLPGVKLGVHILDTCSRDTYALEQSLEFVRASLPLLIAGVIGGSYSSVSIQVANLLRLFQIPQISYASTSAKLSDKSRYDYFARTVPPDFYQAKAMAEILRFFNWTYVSTVASEGDYGETGIEAFEQEARLRNISIATAEKVGRSNIRKSYDSVIRELLQKPNARVVVLFMRSDDSRELIAAASRANASFTWVASDGWGAQESIIKGSEHVAYGAITLELASQPVRQFDRYFQSLNPYNNHRNPWFRDFWEQKFQCSLRVCDKHLAIDSSNYEQESKIMFVVNAVYAMAHALHKMQRTLCPNTTKLCDAMKILDGKKLYKDYLLKINFTAPDADSIVKFDTFGDGMGRYNVFNFQNVGGKYSYLKVGHWAETLSLDVNSIHWSRNSVPTSE 6b8j A 2.595 BS02 65C A 1 G63 F67 V70 A83 Y134 V135 T138 L188 D200 G27 F31 V34 A47 Y95 V96 T99 L149 D161 D181 K183 N186 D200 S219 D142 K144 N147 D161 S180 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue IC50=30nM, EC50=1500nM P49841 29016121 502 VTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 6b8u A 2.68 BS01 8EN A 1 V471 A481 K483 E501 L505 L514 I527 T529 W531 C532 F583 G593 D594 F595 V23 A33 K35 E53 L57 L66 I79 T81 W83 C84 F135 G145 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.200000nM, EC50=230nM P15056 29107542 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLAGSILWMAPEVIRMNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS 6b8y A 1.65 BS01 D0A A 1 A230 K232 E245 Y249 F262 L278 S280 Y282 H283 K337 L340 D351 I501 A33 K35 E48 Y52 F65 L81 S83 Y85 H86 K140 L143 D154 I304 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 remove_due_to_license_issue IC50=0.550000nM, Ki=0.220000nM P36897 29422332 601 HMTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEGI 6b95 A 1.95 BS01 D0P A 1 R105 V155 Q157 E170 C197 S201 R105 V155 Q157 E170 C197 S201 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P18031 29877794 402 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPSRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTVGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFCVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDS 6b96 A 1.88 BS02 CZV A 1 H656 T805 D808 L809 Q859 F862 H83 T232 D235 L236 Q286 F289 3.1.4.17 0004114,0007165,0008081 Ki=14.3nM remove_due_to_license_issue Ki=14nM O00408 29113762 1003 SLYKKAGFYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6b97 A 1.76 BS02 CZY A 1 T768 L770 T805 D808 Q812 F830 F862 T195 L197 T232 D235 Q239 F257 F289 3.1.4.17 0004114,0007165,0008081 Ki=0.237uM remove_due_to_license_issue Ki=237nM O00408 29113762 1003 SLYKKAGFYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6b98 A 1.97 BS02 D07 A 1 L809 I826 F862 L237 I254 F290 3.1.4.17 0004114,0007165,0008081 Ki=22.4uM remove_due_to_license_issue Ki=22400nM O00408 29113762 1003 TSLYKKAGFYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6ba7 A 2.496 BS02 D1Y A 1 V118 R339 G459 L461 D462 M515 W541 D633 V115 R329 G444 L446 D447 M500 W526 D618 D271 E273 R339 E434 D462 D633 D268 E270 R329 E419 D447 D618 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=0.007uM remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAAFLRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGCSKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6bau A 3.8 BS01 CYS A 1 S278 M311 T314 A353 G354 V355 G359 D394 C397 T398 N401 S270 M303 T306 A345 G346 V347 G351 D386 C389 T390 N393 ? 0005283,0005886,0006865,0015108,0015183,0015293,0015501,0016020,0035725,0042802,0046872,0046942,0070207,0070778,0140009,1902476 remove_due_to_license_issue O59010 29295993 503 EYPVLQKILIGLILGAIVGLILGHYGYADAVKTYVKPFGDLFVRLLKMLVMPIVFASLVVGAASISPARLGRVGVKIVVYYLLTSAFAVTLGIIMARLFNPGAGIHLAVGGQQFQPKQAPPLVKILLDIVPTNPFGALANGQVLPTIFFAIILGIAITYLMNSENEKVRKSAETLLDAINGLAEAMYKIVNGVMQYAPIGVFALIAYVMAEQGVKVVGELAKVTAAVYVGLTLQILLVYFVLLKIYGIDPISFIKKAKDAMLTAFVTRSSSGTLPVTMRVAKEMGISEGIYSFTLPLGATINMDGTALYQGVCTFFIANALGSHLTVGQQLTIVLTAVLASIGTAGVPGAGAIMLAMVLESVGLPLTDPNVAAAYAMILGIDAILDMGCTMVNVTGDLTGTAIVAKTE 6baw B 2.703 BS01 D57 B 1 A111 D149 M154 N162 L163 F195 W223 T245 I247 A36 D74 M79 N87 L88 F108 W136 T158 I160 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue IC50=17400nM, Ki=4100nM P41148 29528635 401 FAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTTVWDWELMN 6bbs A 2.0 BS02 BZ1 A 1 Q92 L198 T199 T200 Q89 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=3nM, IC50=3.2nM, Kd=0.13nM P00918 29429876 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6bbu A 2.08 BS01 D7D A 1 G882 E883 A906 E957 F958 L959 N1008 L1010 G16 E17 A40 E84 F85 L86 N135 L137 D1003 A1005 R1007 N1008 D1021 D1040 D130 A132 R134 N135 D148 D167 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.029uM remove_due_to_license_issue IC50=29nM P23458 29298069 4000 PTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6bbv A 1.8 BS01 D7D A 1 G856 K857 A880 Y931 L932 R980 N981 L983 D994 G14 K15 A38 Y89 L90 R138 N139 L141 D152 D976 A978 R980 N981 D994 S1016 D134 A136 R138 N139 D152 S174 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.803uM remove_due_to_license_issue IC50=803nM O60674 29298069 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 6bbx A 2.2 BS01 D77 A 1 L8 S10 G37 V38 H39 W42 L9 S11 G38 V39 H40 W43 ? 0046872,0051213 Kd=215nM remove_due_to_license_issue A0A125SA29 29937405 201 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 6bbx A 2.2 BS02 D77 A 2 G70 W100 Q103 M105 G71 W101 Q104 M106 ? 0046872,0051213 Kd=215nM remove_due_to_license_issue A0A125SA29 29937405 202 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 6bbx B 2.2 BS01 D77 A 1 G70 W100 Q103 M105 G71 W101 Q104 M106 ? 0046872,0051213 remove_due_to_license_issue A0A125SA29 29937405 201 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 6bbx B 2.2 BS02 D77 A 2 S10 G37 V38 H39 W42 F60 S11 G38 V39 H40 W43 F61 ? 0046872,0051213 remove_due_to_license_issue A0A125SA29 29937405 202 HMAISHVQLFSVPVSDQEKAKDFYVETVGFDLLADQPGVHGRWLQVAPKGADTSLVLVDWFPTMPPGSLRGLLLRTDDVDADCARLQERGVAVDGPKNTPWGRQAMFSDPDGNVIGLNQPS 6bc9 A 1.8 BS02 ETS A 1 Q92 H94 H119 V121 F131 L198 T199 T200 W209 Q89 H91 H116 V118 F127 L194 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=9nM, IC50=26.61nM, Kd=0.043000nM P00918 29429876 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6bdy A 1.512 BS01 SFG A 1 D946 R1134 P1135 A1136 Y1139 P1140 A1141 Y1189 D46 R234 P235 A236 Y239 P240 A241 Y289 2.1.1.13 0008705,0009086 Kd=2.04uM remove_due_to_license_issue P13009 29733595 1301 TPPVTLEAARDNDFAFDWQAYTPPVAHRLGVQEVEASIETLRNYIDWTPFFMTWSLAGKYPRILEDEVVGVEAQRLFKDANDMLDKLSAEKTLNPRGVVGLFPANRVGDDIEIYRDETRTHVINVSHHLRQQTEKTGFANYCLADFVAPKLSGKADYIGAFAVTGGLEEDALADAFEAQHDDYNKIMVKALADRLAEAFAEYLHERVRKVYWGYAPNENLSNEELIRENYQGIRPAPGYPACPEHTEKATIWELLEVEKHTGMKLTESFAMWPGASVSGWYFSHPDSKYYAVAQIQRDQVEDYARRKGMSVTEVERWLAPNLGYDA 6beb A 2.55 BS01 RFV A 1 F486 F487 F470 F471 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 MNIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMGVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bec A 2.91 BS01 RBT C 1 P483 F486 P476 F479 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 AMNNTIINSLSIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bec B 2.91 BS01 RBT C 1 V24 F168 F486 V21 F162 F480 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 MNNTIINSLIDSIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bec C 2.91 BS01 RBT C 1 Q27 F486 Q24 F480 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 IPTTENLYFQGAIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bed A 2.75 BS01 RFP C 1 P483 F486 F487 P478 F481 F482 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 GAMNNTIINSLISIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bed C 2.75 BS01 RFP C 1 Q27 F168 F486 Q12 F151 F469 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 IKRSNVFAVDSQIPTLYMPQYISLSGVMTNDDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bee A 3.11 BS01 RXM B 1 F168 F486 F163 F481 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 GAMNNTIINSLISIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bee C 3.11 BS01 RXM B 1 Q27 F168 F486 Q12 F150 F468 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 IKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bef A 3.21 BS01 3YI A 1 Q27 P483 F486 Q24 P476 F479 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 AMNNTIINSLISIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bef C 3.21 BS01 3YI A 1 F168 F486 F150 F468 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 IKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6beh A 3.0 BS01 RPT A 1 P483 F486 P477 F480 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 AMNNTIINSLISIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6beh B 3.0 BS01 RPT A 1 S19 F486 S19 F483 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 GAMNNTIINSLIGDSIKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6beh C 3.0 BS01 RPT A 1 Q27 F168 F486 Q12 F150 F468 ? 0016020,0042802,0046677 remove_due_to_license_issue P68440 30068608 601 IKRSNVFAVDSQIPTLYMPQYISLSGVMTNDNQAIASFEIRDQYITALNHLVLSLELPEVKGMGRFGYVPYVGYKCINHVSISSCNGVIWEIEGEELYNNCINNTIALKHSGYSSELNDISIGLTPNDTIKEPSTVYVYIKTPFDVEDTFSSLKLSDSKITVTVTFNPVSDIVIRDSSFDFETFNKEFVYVPELSFIGYMVKNVQIKPSFIEKPRRVIGQINQPTATVTEVHAATSLSVYTKPYYGNTDNKFISYPGYSQDEKDYIDAYVSRLLDDLVIVSDGPPTGYPESAEIVEVPEDGIVSIQDADVYVKIDNVPDNMSVYLHTNLLMFGTRKNSFIYNISKKFSAITGTYSDATKRTIFAHISHSINIIDTSIPVSLWTSQRNVYNGDNRSAESKAKDLFINDPFIKGIDFKNKTDIISRLEVRFGNDVLYSENGPISRIYNELLTKSNNGTRTLTFNFTPKIFFRPTTITANVSRGKDKLSVRVVYSTMDVNHPIYYVQKQLVVVCNDLYKVSYDQGVSITKIM 6bfa A 2.8 BS01 UW5 A 1 L57 G58 V65 A78 K80 M112 L126 Y131 L181 I194 D195 L14 G15 V22 A35 K37 M69 L83 Y88 L138 I151 D152 D174 K176 E178 N179 D195 T214 D131 K133 E135 N136 D152 T171 2.7.11.17 0004672,0004674,0005509,0005524,0006468,0016020,0046872 remove_due_to_license_issue IC50=1.000nM A0A0F7UUA6 27309760 601 TAIFSDRYKGQRVLGKGSFGEVILCKDKITGQECAVKVISKRQVKQKTDKESLLREVQLLKQLDHPNIMKLYEFFEDKGYFYLVGEVYTGGELFDEIISRKRFSEVDAARIIRQVLSGITYMHKNKIVHRDLKPENLLLESKSKDANIRIIDFGLSTHFEASKKMKDKIGTAYYIAPEVLHGTYDEKCDVWSTGVILYILLSGCPPFNGANEYDILKKVEKGKYTFELPQWKKVSESAKDLIRKMLTYVPSMRISARDALDHEWIQTYTKEQISVDVPSLDNAILNIRQFQGTQKLAQAALLYMGSKLTSQDETKELTAIFHKMDKNGDGQLDRAELIEGYKELMRMKGQDASMLDASAVEHEVDQVLDAVDFDKNGYIEYSEFVTVAMDRKTLLSRERLERAFRMFDSDNSGKISSTELATIFGVSDVDSETWKSVLSEVDKNNDGEVDFDEFQQMLLKLCGN 6bfd A 1.62 BS01 DJS A 1 S10 G13 D32 G34 Y71 T72 Q73 F108 I118 D228 G230 T231 T232 N233 R235 S18 G21 D40 G42 Y79 T80 Q81 F116 I126 D236 G238 T239 T240 N241 R243 D32 S35 N37 A39 Y71 D228 T231 D40 S43 N45 A47 Y79 D236 T239 3.4.23.46 0004190,0006508,0016020 ic50=0.005uM remove_due_to_license_issue P56817 29088532 401 PGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6bfe A 1.51 BS01 DJV A 1 D32 G34 S35 Y71 T72 Q73 G74 F108 W115 I126 D228 G230 D40 G42 S43 Y79 T80 Q81 G82 F116 W123 I134 D236 G238 D32 S35 N37 A39 Y71 D228 T231 D40 S43 N45 A47 Y79 D236 T239 3.4.23.46 0004190,0006508,0016020 ic50=1.4uM remove_due_to_license_issue P56817 29088532 401 PGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6bfn A 2.26 BS01 DL1 A 1 I218 A237 Y288 F290 L291 G294 L347 D358 I26 A45 Y91 F93 L94 G97 L150 D161 2.7.11.1 0004672,0005524,0006468 ic50=9.3nM remove_due_to_license_issue P51617 29208712 601 SRPFPFCWPLCEISRGTHNFSEELKIGEGGFGCVYRAVMRNTVYAVKRLKEWTAVKQSFLTEVEQLSRFRHPNIVDFAGYCAQNGFYCLVYGFLPNGSLEDRLHCQTQACPPLSWPQRLDILLGTARAIQFLHQDSPSLIHGDIKSSNVLLDERLTPKLGDFGLARFSRTVRGTLAYLPEEYIKTGRLAVDTDTFSFGVVVLETLAGQRAVKTHGARTKYLKDLVEEEAEEAGVAAADAWAAPIAMQIYKKHLDPRPGPCPPELGLGLGQLACCCLHRRAKRRPPMTQVYERLEKLQAVVA 6bfp A 1.292 BS02 DJY A 1 H63 L104 Y154 D194 S195 Q197 S200 V214 S215 W216 G217 G219 H40 L81 Y129 D169 S170 Q172 S175 V189 S190 W191 G192 G194 H63 D107 Q197 G198 D199 S200 G201 H40 D84 Q172 G173 D174 S175 G176 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 remove_due_to_license_issue P00760 30876891 302 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN 6bfw A 1.84 BS01 DK7 A 1 D32 G34 S35 Y71 T72 F108 Y198 D228 G230 D40 G42 S43 Y79 T80 F116 Y206 D236 G238 D32 S35 N37 A39 Y71 D228 T231 D40 S43 N45 A47 Y79 D236 T239 3.4.23.46 0004190,0006508,0016020 ic50=0.22uM remove_due_to_license_issue P56817 29088532 401 PGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6bfx A 1.99 BS01 DKJ A 1 D32 G34 S35 Y71 T72 F108 Y198 D228 G230 D36 G38 S39 Y75 T76 F112 Y202 D232 G234 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=0.079uM remove_due_to_license_issue P56817 29088532 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6bg3 A 1.05 BS01 DOJ A 1 I1083 I1086 F1089 P1097 V1102 I1105 A1106 A1111 Q1114 E1116 F1117 F1164 A1180 Y1181 I199 I202 F205 P213 V218 I221 A222 A227 Q230 E232 F233 F280 A296 Y297 E11 D20 E24 D33 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 ic50=12uM remove_due_to_license_issue P00720,Q96GG9 29547696 1301 HSQDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRTKRVITTFRTGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHKRSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQ 6bg5 A 1.1 BS01 DQD A 1 I1083 I1086 F1089 P1097 A1106 Q1114 E1116 F1117 F1164 Y1181 I199 I202 F205 P213 A222 Q230 E232 F233 F280 Y297 E11 D20 E24 D33 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 ic50=1uM remove_due_to_license_issue P00720,Q96GG9 29547696 1301 HSQDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRTKRVITTFRTGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHKRSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQ 6bgu A 1.684 BS01 DKP A 1 R73 Y409 A411 Y472 F480 H483 N493 K501 W503 Q535 H571 R63 Y136 A138 Y193 F201 H204 N214 K222 W224 Q256 H292 Y472 H483 E485 H571 A583 Y193 H204 E206 H292 A304 1.14.11.67 Kd=0.53uM remove_due_to_license_issue IC50=<100nM, Kd=530nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bgv A 1.592 BS01 DQG A 1 Y409 D412 W470 Y472 F480 C481 H483 K501 W503 H571 Y136 D139 W191 Y193 F201 C202 H204 K222 W224 H292 Y472 H483 E485 H571 A583 Y193 H204 E206 H292 A304 1.14.11.67 Kd=0.18uM remove_due_to_license_issue Kd=60nM, IC50=590nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bgw A 1.644 BS01 DKS A 1 Y409 D412 W470 Y472 F480 C481 H483 N493 K501 W503 H571 Y136 D139 W191 Y193 F201 C202 H204 N214 K222 W224 H292 Y472 H483 E485 H571 A583 Y193 H204 E206 H292 A304 1.14.11.67 Kd=0.21uM remove_due_to_license_issue IC50=4500nM, Kd=210nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bgx A 1.882 BS01 DKV A 1 Y409 Y472 F480 C481 H483 D486 K501 W503 H571 Y135 Y192 F200 C201 H203 D206 K221 W223 H291 Y472 H483 E485 H571 A583 Y192 H203 E205 H291 A303 1.14.11.67 Kd=0.47uM remove_due_to_license_issue Kd=470nM, IC50=22000nM P29375 29537847 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMRPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bgy A 1.22 BS01 DLJ A 1 Y409 Y472 F480 C481 H483 K501 W503 H571 Y124 Y181 F189 C190 H192 K210 W212 H280 Y472 H483 E485 H571 A583 Y181 H192 E194 H280 A292 1.14.11.67 Kd=0.15uM remove_due_to_license_issue Kd=150nM, IC50=290nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bgz A 1.688 BS01 DNV A 1 Y409 Y472 F480 C481 H483 K501 W503 Q535 L536 H571 Y126 Y177 F185 C186 H188 K206 W208 Q240 L241 H276 Y472 H483 E485 H571 A583 Y177 H188 E190 H276 A288 1.14.11.67 Kd=0.41uM remove_due_to_license_issue Kd=410nM, IC50=1400nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bh0 A 1.985 BS01 DO1 A 1 R73 Y409 A411 W470 Y472 S479 F480 H483 K501 W503 H571 R63 Y131 A133 W173 Y175 S182 F183 H186 K204 W206 H274 Y472 H483 E485 H571 A583 Y175 H186 E188 H274 A286 1.14.11.67 Kd=0.22uM remove_due_to_license_issue IC50=670nM, Kd=180nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKILPEEEEYALSGWNLNNMPVLEKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bh1 A 1.932 BS01 DQG A 1 Y409 D412 W470 Y472 F480 C481 H483 N493 K501 W503 H571 Y128 D131 W179 Y181 F189 C190 H192 N202 K210 W212 H280 Y472 H483 E485 H571 A583 Y181 H192 E194 H280 A292 1.14.11.67 Kd=0.06uM remove_due_to_license_issue Kd=60nM, IC50=590nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bh2 A 1.447 BS02 90V A 1 Y472 S479 F480 H483 E485 K501 H571 N575 V584 N585 Y179 S186 F187 H190 E192 K208 H278 N282 V291 N292 Y472 H483 E485 H571 A583 Y179 H190 E192 H278 A290 1.14.11.67 Kd=2.4uM remove_due_to_license_issue IC50=570nM, Kd=2400nM, EC50=960nM P29375 29537847 604 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMFGFEREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bh3 A 1.701 BS01 DQJ A 1 Y472 S479 F480 H483 E485 K501 H571 A583 V584 Y186 S193 F194 H197 E199 K215 H285 A297 V298 Y472 H483 E485 H571 A583 Y186 H197 E199 H285 A297 1.14.11.67 remove_due_to_license_issue EC50=1600nM, IC50=90nM P29375 29537847 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bh5 A 1.651 BS01 DNY A 1 Y409 Y472 F480 C481 H483 I484 D486 K501 W503 H571 Y124 Y176 F184 C185 H187 I188 D190 K205 W207 H275 Y472 H483 E485 H571 A583 Y176 H187 E189 H275 A287 1.14.11.67 Kd=0.25uM remove_due_to_license_issue IC50=430nM, Kd=250nM P29375 29537847 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6bh8 A 3.85 BS02 RDF A 1 S264 N265 V332 H335 E336 H339 E415 N442 H459 R465 S210 N211 V233 H236 E237 H240 E316 N343 H360 R366 3.4.24.84 0001889,0001942,0003007,0003229,0003231,0003417,0003690,0004175,0004222,0005515,0005634,0005635,0005637,0005768,0005783,0005789,0006281,0006325,0006355,0006508,0006925,0006974,0006997,0006998,0007346,0007628,0008016,0008233,0008235,0008237,0008340,0008360,0008544,0010506,0010628,0010629,0010906,0016020,0016485,0019216,0030282,0030327,0030500,0031901,0031902,0032006,0032350,0032991,0035264,0040014,0040029,0043007,0043516,0044029,0044255,0046872,0048145,0048538,0050688,0050905,0051276,0051604,0055013,0060307,0060993,0061337,0061762,0070062,0070302,0071480,0071586,0072423,1903463,1903522,1903799,1990036,2000730,2000772 remove_due_to_license_issue O75844 30082509 502 EKRIFGAVLLFSWTVYLWETFLAQRQRRIYKTTTHVPPELGQIMDYLWRLSGRFCGYAGFGPEYEITQSLVFLLLATLFSALAGLPWSLYNTFVIEEKHGFNQQTLGFFMKDAIKKFVVTQCILLPVSSLLLYIIKIGGDYFFIYAWLFTLVVSLVLVTIYADYIAPLFDKFTPLPEGKLKEEIEVMAKSIDFPLTKVYVVEGSKRSSHSNAYFKRIVLFDTLGCKNEEVLAVLGHELGHWKLGHTVKNIIISQMNSFLCFFLFAVLIGRKELFAAFGFYDSQPTLIGLLIIFQFIFSPYNEVLSFCLTVLSRRFEFQADAFAKKLGKAKDLYSALIKLNKDNLGFPVSDWLFSMWHYSHPPLLERLQALK 6bhv A 2.3 BS01 DQV A 1 H862 G863 S864 N868 G871 I872 L877 R878 Y889 M890 Y896 F897 S904 Y907 E988 H90 G91 S92 N96 G99 I100 L105 R106 Y117 M118 Y124 F125 S132 Y135 E216 S904 Y907 E988 S132 Y135 E216 2.4.2.-,2.4.2.30 0003950 Kd=5.87uM remove_due_to_license_issue P09874 29487285 1101 SKLPKPVQDLIKMIFGPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 6bib A 1.95 BS01 DW7 A 1 H30 E54 I109 Q110 R112 T134 I135 P136 C139 A158 A159 A160 K162 H31 E55 I110 Q111 R113 T126 I127 P128 C131 A150 A151 A152 K154 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 30883881 201 HAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 6bid A 1.15 BS01 DW4 A 1 H30 E54 Q110 G133 T134 I135 P136 C139 A158 A159 A160 T161 H31 E55 Q111 G133 T134 I135 P136 C139 A158 A159 A160 T161 2.7.7.48,3.4.22.66,3.6.1.15 0004197,0006508 remove_due_to_license_issue Q83883 30883881 201 HAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQA 6bik A 1.901 BS01 DTJ A 1 L408 G411 F413 V416 A428 K430 Y476 M477 A478 G480 L528 D539 Y551 L14 G17 F19 V22 A34 K36 Y82 M83 A84 G86 L134 D145 Y157 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30756207 703 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 6bjo A 1.75 BS01 DUY A 1 L32 I33 G34 I35 S36 F53 A87 I90 L14 I15 G16 I17 S18 F35 A69 I72 ? ic50=513nM remove_due_to_license_issue Q9NRD5 29280296 201 VPGKVTLQKDAQNLIGISIGGGAQYCPCLYIVQVFDNTPAALDGTVAAGDEITGVNGRSIKGKTKVEVAKMIQEVKGEVTIHYNKL 6bjo B 1.75 BS01 DUY B 1 L32 I33 G34 I35 F53 K83 A87 L14 I15 G16 I17 F34 K64 A68 ? ic50=513nM remove_due_to_license_issue Q9NRD5 29280296 201 VPGKVTLQKDAQNLIGISIGGGAYCPCLYIVQVFDNTPAALDGTVAAGDEITGVNGRSIKGKTKVEVAKMIQEVKGEVTIHYNKL 6bjv A 2.198 BS01 rna C 0 R11 W39 V69 S113 R115 S120 R10 W38 V68 S112 R114 S119 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 31021526 1 ~ 21 ERAIQGNDTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDETNSNQDNPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLTP 6bjv A 2.198 BS02 rna D 0 R18 W19 P37 W42 K60 Q107 V108 G109 S124 G126 R17 W18 P36 W41 K59 Q106 V107 G108 S123 G125 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 31021526 1 ~ 21 ERAIQGNDTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDETNSNQDNPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLTP 6bjv B 2.198 BS01 rna C 0 R18 W19 W42 K60 V108 S124 G125 R16 W17 W40 K58 V106 S122 G123 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 31021526 1 ~ 21 RAIQGNDTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDETNSNQDNPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLT 6bjv B 2.198 BS02 rna D 0 R11 W39 K71 S113 R115 S120 R9 W37 K69 S111 R113 S118 ? 0003723,0019049,0044423,0052170 remove_due_to_license_issue Q66104 31021526 1 ~ 21 RAIQGNDTREQANGERWDGGSGGITSPFKLPDESPSWTEWRLYNDETNSNQDNPLGFKESWGFGKVVFKRYLRYDRTEASLHRVLGSWTGDSVNYAASRFLGANQVGCTYSIRFRGVSVTISGGSRTLQHLCEMAIRSKQELLQLT 6bke A 1.95 BS01 DVJ A 1 L408 F413 V416 K430 Y476 M477 A478 G480 N526 L528 D539 L14 F19 V22 K36 Y82 M83 A84 G86 N132 L134 D145 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30756207 704 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 6bkh A 1.792 BS01 DVD A 1 L408 Q412 F413 V416 K430 Y476 M477 G480 L528 D539 L542 S543 L13 Q17 F18 V21 K35 Y81 M82 G85 L133 D144 L147 S148 D521 R525 N526 D539 D126 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30756207 705 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 6bkw A 1.499 BS01 DXM A 1 L408 T410 G411 F413 V416 K430 Y476 M477 G480 N526 L528 D539 Y551 L16 T18 G19 F21 V24 K38 Y84 M85 G88 N134 L136 D147 Y159 D521 R525 N526 D539 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30756207 704 GSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 6bkx A 1.65 BS02 DWP A 1 H309 V312 R314 H315 S326 K374 D375 H307 V310 R312 H313 S324 K372 D373 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 remove_due_to_license_issue O75874 30004704 501 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSL 6bkx C 1.65 BS02 DWP C 1 H309 V312 R314 H315 S326 K374 D375 H307 V310 R312 H313 S324 K372 D373 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 remove_due_to_license_issue O75874 30004704 503 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSLEHH 6bky C 2.17 BS01 K32 D 1 V255 M259 Q277 S280 V253 M257 Q275 S278 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 remove_due_to_license_issue IC50=270nM O75874 30004704 503 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSL 6bky D 2.17 BS02 K32 D 1 V255 M259 Q277 S280 V253 M257 Q275 S278 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 ic50=270nM remove_due_to_license_issue IC50=270nM O75874 30004704 503 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSLEH 6bl1 A 2.02 BS02 DWG A 1 H309 V312 R314 H315 M318 K374 L383 H307 V310 R312 H313 M316 K372 L381 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 ic50=110nM remove_due_to_license_issue IC50=1770nM O75874 30004704 501 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSLEH 6bl1 B 2.02 BS01 DWG B 1 H309 V312 R314 H315 M318 T325 N328 K374 L383 H307 V310 R312 H313 M316 T323 N326 K372 L381 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 ic50=110nM remove_due_to_license_issue IC50=1770nM O75874 30004704 502 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSLEH 6bl2 A 1.92 BS01 DWS A 1 H309 V312 R314 H315 T325 K374 D375 A378 L383 H307 V310 R312 H313 T323 K372 D373 A376 L381 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 remove_due_to_license_issue O75874 30004704 504 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSLEH 6bl2 C 1.92 BS02 DWS C 1 H309 V312 R314 H315 M318 T325 K374 D375 H307 V310 R312 H313 M316 T323 K372 D373 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 remove_due_to_license_issue O75874 30004704 501 KKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGRHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNYDGDVQSDSVAQGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKLSLEH 6bln A 1.3 BS01 DY4 A 1 L408 T410 G411 F413 V416 K430 Y476 M477 G480 N526 L528 D539 Y551 L14 T16 G17 F19 V22 K36 Y82 M83 G86 N132 L134 D145 Y157 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30756207 704 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEN 6blw A 1.835 BS01 dna B 0 K332 Y334 F335 K336 H339 R342 K346 R362 F364 R366 R372 H373 R376 R390 F392 R394 H397 H401 T404 K16 Y18 F19 K20 H23 R26 K30 R46 F48 R50 R56 H57 R60 R74 F76 R78 H81 H85 T88 ? remove_due_to_license_issue P19544 29294058 2 ~ 17 HMEKRPFMCAYPGCNKRYFKLSHLQRHSRKHTGEKPYQCDFKDCERRFSRSDQLKRHQRRHTGVKPFQCKTCQRKFSRSDHLKTHTRTHTGKSCRWPSCQLVRHHNMHQ 6blw A 1.835 BS02 dna C 0 S338 K371 F383 S395 S420 S22 K55 F67 S79 S98 ? remove_due_to_license_issue P19544 29294058 2 ~ 18 HMEKRPFMCAYPGCNKRYFKLSHLQRHSRKHTGEKPYQCDFKDCERRFSRSDQLKRHQRRHTGVKPFQCKTCQRKFSRSDHLKTHTRTHTGKSCRWPSCQLVRHHNMHQ 6bm5 A 1.5 BS01 SAM A 1 D946 R1134 P1135 A1136 Y1139 P1140 A1141 Y1189 D46 R234 P235 A236 Y239 P240 A241 Y289 2.1.1.13 0008705,0009086 Kd=1.43uM remove_due_to_license_issue P13009 29733595 1301 TPPVTLEAARDNDFAFDWQAYTPPVAHRLGVQEVEASIETLRNYIDWTPFFMTWSLAGKYPRILEDEVVGVEAQRLFKDANDMLDKLSAEKTLNPRGVVGLFPANRVGDDIEIYRDETRTHVINVSHHLRQQTEKTGFANYCLADFVAPKLSGKADYIGAFAVTGGLEEDALADAFEAQHDDYNKIMVKALADRLAEAFAEYLHERVRKVYWGYAPNENLSNEELIRENYQGIRPAPGYPACPEHTEKATIWELLEVEKHTGMKLTESFAMWPGASVSGWYFSHPDSKYYAVAQIQRDQVEDYARRKGMSVTEVERWLAPNLGYD 6bm6 A 1.504 BS01 SAH A 1 D946 R1134 P1135 A1136 Y1139 P1140 A1141 Y1189 D46 R234 P235 A236 Y239 P240 A241 Y289 2.1.1.13 0008705,0009086 Kd=20.8uM remove_due_to_license_issue P13009 29733595 1301 TPPVTLEAARDNDFAFDWQAYTPPVAHRLGVQEVEASIETLRNYIDWTPFFMTWSLAGKYPRILEDEVVGVEAQRLFKDANDMLDKLSAEKTLNPRGVVGLFPANRVGDDIEIYRDETRTHVINVSHHLRQQTEKTGFANYCLADFVAPKLSGKADYIGAFAVTGGLEEDALADAFEAQHDDYNKIMVKALADRLAEAFAEYLHERVRKVYWGYAPNENLSNEELIRENYQGIRPAPGYPACPEHTEKATIWELLEVEKHTGMKLTESFAMWPGASVSGWYFSHPDSKYYAVAQIQRDQVEDYARRKGMSVTEVERWLAPNLGYD 6bmi A 3.9 BS01 SER A 1 R276 S278 T314 D394 T398 N401 R268 S270 T306 D374 T378 N381 ? 0005283,0005886,0006865,0015108,0015183,0015293,0015501,0016020,0035725,0042802,0046872,0046942,0070207,0070778,0140009,1902476 remove_due_to_license_issue O59010 29295993 502 EYPVLQKILIGLILGAIVGLILGHYGYADAVKTYVKPFGDLFVRLLKMLVMPIVFASLVVGAASISPARLGRVGVKIVVYYLLTSAFAVTLGIIMARLFNPGAGIHLAVGGQQFQPKQAPPLVKILLDIVPTNPFGALANGQVLPTIFFAIILGIAITYLMNSENEKVRKSAETLLDAINGLAEAMYKIVNGVMQYAPIGVFALIAYVMAEQGVKVVGELAKVTAAVYVGLTLQILLVYFVLLKIYGIDPISFIKKAKDAMLTAFVTRSSSGTLPVTMRVAKEMGISEGIYSFTLPLGATINMDGTALYQGVCTFFIANALGSHLTVGQQLTIVLTAVLAIMLAMVLESVGLPLTDPNVAAAYAMILGIDAILDMGCTMVNVTGDLTGTAIVAKTE 6bmr A 2.205 BS01 DZV A 1 Q79 Y80 E83 H84 L262 Y263 S264 R265 Q269 N281 Q77 Y78 E81 H82 L239 Y240 S241 R242 Q246 N258 D425 C459 R465 T466 Q506 D389 C423 R429 T430 Q470 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Q06124 29304282 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHHGQLKENGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQPGDFVLSVRTGSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPPVSDYINANIIMPEKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6bmv A 2.053 BS01 DZS A 1 Q79 Y80 E83 H84 L262 Y263 S264 R265 K266 Q269 N281 Q77 Y78 E81 H82 L237 Y238 S239 R240 K241 Q244 N256 D425 C459 R465 T466 Q506 D383 C417 R423 T424 Q464 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Q06124 29304282 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHHGQLKNGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQPGDFVLSVRTGSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHPVSDYINANIIMPEKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6bmx A 2.424 BS01 DYV A 1 Q79 Y80 E83 H84 L262 Y263 S264 R265 K266 Q269 K280 N281 Q77 Y78 E81 H82 L238 Y239 S240 R241 K242 Q245 K256 N257 D425 C459 R465 T466 Q506 D388 C422 R428 T429 Q469 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue Q06124 29304282 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHHGQLKENGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESPGDFVLSVRTGSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPPVSDYINANIIMPEKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6bnk A 3.2 BS01 AGH A 1 S28 L66 F70 Y73 S76 F77 D80 W133 W142 L150 D153 T156 F171 S21 L59 F63 Y66 S69 F70 D73 W126 W135 L143 D146 T149 F164 ? remove_due_to_license_issue P11609 29576533 405 YTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6bnk C 3.2 BS01 AGH A 1 P28 R95 P28 R94 remove_due_to_license_issue 29576533 405 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKSDFACANAFNNSIIPEDTFFPS 6bnl A 2.6 BS01 QWV A 1 S28 M69 F70 Y73 S76 F77 D80 W133 D153 G155 T156 T159 F171 S23 M64 F65 Y68 S71 F72 D75 W128 D148 G150 T151 T154 F166 ? remove_due_to_license_issue P11609 29576533 405 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLLACRVKHSSLGGQDIILY 6bnl C 2.6 BS01 QWV A 1 P28 R95 P28 R94 remove_due_to_license_issue 29576533 405 TQVEQSPQSLVVRQGENSVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKSDFACANAFNNSIIPEDTFFP 6bny A 3.341 BS01 E0M A 1 L15 A36 M86 E87 F88 C89 G92 M142 T156 L15 A36 M83 E84 F85 C86 G89 M139 T153 D135 K137 N140 D157 T176 D132 K134 N137 D154 T157 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=180nM Q9UHD2 30082428 801 MQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFNNISFLDVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFGTEEYLHPDMYEVDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVELGEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 6bo6 A 2.801 BS01 E0V A 1 M149 D172 H343 F374 E425 Y481 Y485 F486 E516 W561 R574 N578 K580 M127 D136 H228 F259 E310 Y366 Y370 F371 E401 W446 R459 N463 K465 3.2.1.31 0004553,0004565,0004566,0005975,0016798,0030246 remove_due_to_license_issue C4Z6Z2 30062115 701 SDLSGVWDFKLDNGKGFEEKWYEKPLKDADTMPVPASYNDLKEGTDFRDHYGWVFYQRNISVLRCAAVTHYAMIYLNGKLICEHKGGFLPFEVELNDDLQDGDNLLTIAVNNVIDYTTLPVGGKANMMPQNNPNFDFFNYCGITRPVKIYLWQPLNAYLYKIYTLPYGVRSVRVDGTKFLINEKPFYFKGYGKHEDTFPNGRGINLPMNTKDISIMKWQHANSFRTSHYPYSEEMMRLCDEEGIVVIDETTAVGVNLQFGGGANFGGERIGTFDKEHGVQTQEHHKDVIRDLISRDKNHACVVMWSIANEPDSAAEGAYDYFKPLYDLARELDPQKRPCTLVSVQGTTADTDCSSQLSDVICLNRYYGWYFGGPDLEVSEIGLRKELSDWGKLGKPVMFTEYGADTVSGLHDTTSVMYTEEYQVEYYEMNNKVFDEFDFVVGEQAWNFADFATSQSLLRVQGNKKGLFTRDRKPKMVAHYFRNRWSTIPEFGY 6bod A 3.197 BS01 E0P A 1 L15 C89 M142 T156 D157 L16 C81 M134 T148 D149 D135 K137 N140 D157 T176 D127 K129 N132 D149 T156 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=123000nM Q9UHD2 30082428 801 AMQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFNVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFGAARETEEYLHPDMYERATVDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVKVEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 6boe A 3.598 BS01 E0S A 1 L15 A36 E87 F88 C89 P90 M142 L16 A33 E74 F75 C76 P77 M129 D135 K137 N140 D157 T176 D122 K124 N127 D144 T147 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=180nM Q9UHD2 30082428 701 AMQSTSNHLWLLSDILGQNVFRGRHKKTGDLFAIKVFVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFGTEEYLHPDMYEDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVKVELGEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 6boy B 3.33 BS02 RN6 B 1 N351 P352 H353 H378 S379 W380 W386 W400 F402 N299 P300 H301 H326 S327 W328 W334 W348 F350 ? 0005515,0005634,0005737,0005829,0016020,0016567,0030177,0031333,0031334,0031464,0034766,0035641,0043161,0044325,0046872,0048471 remove_due_to_license_issue Q96SW2 29892083 502 PNIINFDTSLPTSHTYLGADMEEFHGRTLHDDDSCQVIPVLPQVMMILIPGQTLPLQLFHPQEVSMVRNLIQKDRTFAVLAYSNVQEREAQFGTTAEIYAYREEQDFGIEIVKVKAIGRQRFKVLELRTQSDGIQQAKVQILPECVLPSTMSAVQLESLNKCQIFPCSYKWWQKYQKRKFHCANLTSWPRWLYSLYDAETLMDRIKKQLREWDENLKDDSLPSNPIDFSYRVAACLPIDDVLRIQLLKIGSAIQRLRCELDIMNKCTSLCCKQCQETEITTKNEIFSLSLCGPMAAYVNPHGYVHETLTVYKACNLNLIGRPSTEHSWFPGYAWTVAQCKICASHIGWKFTATKKDMSPQKFWGLTRSALLPTIP 6boy C 3.33 BS01 RN6 B 1 W81 P82 L94 N140 I146 M149 W40 P41 L53 N99 I105 M108 ? remove_due_to_license_issue O60885 29892083 502 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6bq0 A 2.0 BS01 E3A A 1 A51 S122 M123 L176 G177 L241 A34 S105 M106 L159 G160 L224 3.1.1.23 0004622,0005515,0005737,0005789,0005829,0005886,0006629,0006633,0006639,0006954,0009966,0016020,0016042,0019369,0019433,0042803,0046464,0047372,0050727,0051930,0052651,0052689,2000124 remove_due_to_license_issue Q99685 29498843 401 DLPHLVNADGQYLFCRYWKPTGTPKALIFVSHGAGEHSGRYEELARMLMGLDLLVFAHDHVGHGQSEGERMVVSDFHVFVRDVLQHVDSMQKDYPGLPVFLLGHSMGGAIAILTAAERPGHFAGMVLISPLVLANPESATTFKVLAAKVLNLVLPNLSLGPIDSSVLSRNKTEVDIYNSDPLICRAGLKVCFGIQLLNAVSRVERALPKLTVPFLLLQGSADRLCDSKGAYLLMELAKSQDKTLKIYEGAYHVLHKELPEVTNSVFHEINMWVSQRTATA 6bqg A 3.0 BS01 ERM A 1 D134 V135 S138 T139 V208 L209 G218 F327 S334 V335 E347 L350 D92 V93 S96 T97 V163 L164 G173 F319 S326 V327 E339 L342 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P28335 29398112 1201 GGRFKFPDGVQNWPALSIVIIIIMTIGGNILVIMAVSMEKKLHNATNYFLMSLAIADMLVGLLVMPLSLLAILYDYVWPLPRYLCPVWISLDVLFSTASIMHLCAISLDRYVAIRNPIEHNSRTKAIMKIAIVWAISIGVSVPIPVIGLRDEEKVFVNNTTCVLNDPNFVLIGSFVAFFIPLTIMVITYCLTIYVLRRQAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKAMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLQAINNERKASKVLGIVFFVFLIMWCPFFITNILSVLCEKSCNQKLMEKLLNVFVWIGYVNSGINPLVYTLFNKIYRRAFSNYLRCN 6bqh A 2.7 BS01 E2J A 1 W130 D134 V135 S138 T139 I142 G218 S219 F223 W324 F327 F328 N351 V354 W85 D89 V90 S93 T94 I97 G173 S174 F178 W288 F291 F292 N315 V318 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P28335 29398112 1201 FKFPDGVQNWPALSIVIIIIMTIGGNILVIMAVSMEKKLHNATNYFLMSLAIADMLVGLLVMPLSLLAILYDYVWPLPRYLCPVWISLDVLFSTASIMHLCAISLDRYVAIRNPIEHSRFNSRTKAIMKIAIVWAISIGVSVPIPVIGLRDEEKVFVNNTTCVLNDPNFVLIGSFVAFFIPLTIMVITYCLTIYVLRRQAADLEDNWETLNDNLKVIEKAVKDALTKMRAAALDAQKATMKDFRHGFDILQLKTTRNAYIQKYLQAINNERKASKVLGIVFFVFLIMWCPFFITNILSVLCEKSCNQKLMEKLLNVFVWIGYVNSGINPLVYTLFNKIYRRAFSNYLRCNY 6bqj A 1.69 BS01 Z1B A 1 Q41 T42 Y56 H57 V78 D81 I132 L135 G137 S139 F154 R155 A156 A157 Q53 T54 Y68 H69 V90 D93 I144 L147 G149 S151 F166 R167 A168 A169 H57 D81 G137 S139 H69 D93 G149 S151 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue P27958 29456803 301 KGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTMRSP 6bqk A 1.97 BS01 Z1E A 1 Q41 H57 V78 D81 L135 K136 G137 S139 F154 R155 A156 A157 Q52 H68 V89 D92 L146 K147 G148 S150 F165 R166 A167 A168 H57 D81 G137 S139 H68 D92 G148 S150 2.7.7.48,3.4.21.98,3.4.22.-,3.6.1.15,3.6.4.13 0006508,0008236,0019087 ic50=1nM remove_due_to_license_issue P27958 29456803 301 GSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTMRSP 6br2 A 3.18 BS01 E3S A 1 L287 H323 M365 F377 F378 E379 F388 L23 H59 M101 F113 F114 E115 F124 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P51449 29510038 502 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQH 6br3 A 3.0 BS01 E3V A 1 C320 H323 L324 V361 M365 A368 F377 F378 E379 F388 C56 H59 L60 V97 M101 A104 F113 F114 E115 F124 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P51449 29510038 502 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHV 6bs3 A 2.3 BS01 ADP A 1 G31 G33 K34 S35 T36 N240 R241 V318 V322 G21 G23 K24 S25 T26 N230 R231 V308 V312 ? 0005524,0005886,0016887 Kd=1.5uM remove_due_to_license_issue P9WKX5 31036728 401 SVGWPSRLSGVRLHLVTGKGGTGKSTIAAALALTLAAGGRKVLLVEVEGRQGIAQLFDVPPLPYQELKIATAERGGQVNALAIDIEAAFLEYLDMFYNLGIAGRAMRRIGAVEFATTIAPGLRDVLLTGKIKETVVRLDKNKLPVYDAIVVDAPPTGRIARFLDVTKAVSDLAKGGPVHAQSEGVVKLLHSNQTAIHLVTLLEALPVQETLEAIEELAQMELPIGSVIVNRNIPAHLEPQDLAKAAEGEVDADSVRAGLLTAGVKLPDADFAGLLTETIQHATRITARAEIAQQLDALQVPRLELPTVSDGVDLGSLYELSESLAQQGVR 6bs3 B 2.3 BS01 ADP B 1 G29 G31 K32 T33 T34 N283 R284 S355 L356 D359 V360 G25 G27 K28 T29 T30 N269 R270 S335 L336 D339 V340 0005524,0016887 Kd=1.5uM remove_due_to_license_issue 31036728 401 PKTLDMGAILADTSNRVVVCCGAGGVGKTTTAAALALRAAEYGRTVVVLTIDPAKRLAQALGINDLGNTPQRVPLAPEVPGELHAMMLDMRRTFDEMVMQYSGPERAQSILDNQFYQTVATSLAGTQEYMAMEKLGQLLSQDRWDLIVVDTPPSRNALDFLDAPKRLGSFMDSRLWRLLLAITGVMGLAMKALSTVLGSQMLADAAAFVQSLDAGGFREKADRTYALLKRRGTQFVVVSAAEPDALREASFFVDRLSQESMPLAGLVFNRTHPMLCALPIERAIDAAETLDAETSLAAAVLRIHAERGQTAKREIRLLSRFTGANPTVPVVGVPSLPFDVSDLEALRALADQLTT 6bs4 A 2.5 BS01 AGS A 1 G31 G33 K34 S35 T36 R60 N240 R241 T317 V318 V322 G21 G23 K24 S25 T26 R50 N230 R231 T307 V308 V312 ? 0005524,0005886,0016887 Kd=2.8uM remove_due_to_license_issue P9WKX5 31036728 401 SVGWPSRLSGVRLHLVTGKGGTGKSTIAAALALTLAAGGRKVLLVEVEGRQGIAQLFDVPPLPYQELKIATAERGGQVNALAIDIEAAFLEYLDMFYNLGIAGRAMRRIGAVEFATTIAPGLRDVLLTGKIKETVVRLDKNKLPVYDAIVVDAPPTGRIARFLDVTKAVSDLAKGGPVHAQSEGVVKLLHSNQTAIHLVTLLEALPVQETLEAIEELAQMELPIGSVIVNRNIPAHLEPQDLAKAAEGEVDADSVRAGLLTAGVKLPDADFAGLLTETIQHATRITARAEIAQQLDALQVPRLELPTVSDGVDLGSLYELSESLAQQGVR 6bs5 A 3.1 BS01 ANP A 1 G31 G33 K34 S35 T36 R60 N240 R241 T317 V318 V322 G21 G23 K24 S25 T26 R50 N230 R231 T307 V308 V312 ? 0005524,0005886,0016887 remove_due_to_license_issue P9WKX5 31036728 401 SVGWPSRLSGVRLHLVTGKGGTGKSTIAAALALTLAAGGRKVLLVEVEGRQGIAQLFDVPPLPYQELKIATAERGGQVNALAIDIEAAFLEYLDMFYNLGIAGRAMRRIGAVEFATTIAPGLRDVLLTGKIKETVVRLDKNKLPVYDAIVVDAPPTGRIARFLDVTKAVSDLAKGGPVHAQSEGVVKLLHSNQTAIHLVTLLEALPVQETLEAIEELAQMELPIGSVIVNRNIPAHLEPQDLAKAAEGEVDADSVRAGLLTAGVKLPDADFAGLLTETIQHATRITARAEIAQQLDALQVPRLELPTVSDGVDLGSLYELSESLAQQGVR 6bsk A 2.573 BS01 MVG A 1 L44 F49 A65 K67 R122 V126 D128 L174 I185 D186 L12 F17 A33 K35 R90 V94 D96 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 remove_due_to_license_issue P11309 29559278 405 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 6bsl A 1.45 BS03 EVV A 1 R61 G64 C66 S67 Y68 R72 Q77 A78 H93 E94 H97 H103 R61 G64 C66 S67 Y68 R72 Q77 A78 H93 E94 H97 H103 3.4.24.19 0004222,0006508,0008237,0008270 Ki=6.8pM remove_due_to_license_issue Ki=6.8nM, IC50=<1.000000nM P13497 30034610 304 AATSRPERVWPDGVIPFVIGGNFTGSQRAVFRQAMRHWEKHTCVTFLERTDEDSYIVFTYRPCGCCSYVGRRGGGPQAISIGKNCDKFGIVVHELGHVVGFWHEHTRPDRDRHVSIVRENIQPGQEYNFLKMEPQEVESLGETYDFDSIMHYARNTFSRGIFLDTIVPKYEVNGVKPPIGQRTRLSKGDIAQARKLYKCPA 6bsm A 2.33 BS03 E7D A 1 C66 S67 Y68 V69 H93 E94 H97 W102 H103 C66 S67 Y68 V69 H93 E94 H97 W102 H103 3.4.24.19 0004222,0006508,0008237,0008270 ic50=160nM remove_due_to_license_issue P13497 30034610 303 AATSRPERVWPDGVIPFVIGGNFTGSQRAVFRQAMRHWEKHTCVTFLERTDEDSYIVFTYRPCGCCSYVGRRGGGPQAISIGKNCDKFGIVVHELGHVVGFWHEHTRPDRDRHVSIVRENIQPGQEYNFLKMEPQEVESLGETYDFDSIMHYARNTFSRGIFLDTIVPKYEVNGVKPPIGQRTRLSKGDIAQARKLYKCP 6bsx A 1.65 BS02 E7S A 1 E40 T61 G63 Q64 Y74 E39 T60 G62 Q63 Y73 3.6.5.- 0000139,0000287,0003924,0005515,0005525,0005681,0005737,0005764,0005765,0005783,0005789,0005794,0005829,0005886,0007165,0007264,0012505,0014069,0016020,0016241,0016787,0019003,0019901,0030295,0031669,0032006,0032008,0043539,0045202,0046872,0048709,0048714,0051726,0070062,0120163,1904263,2000074 remove_due_to_license_issue Q15382 29416044 204 PQSKSRKIAILGYRSVGKSSLTIQFVEGQFVDSYDPTIENTFTKLITVNGQEYHLQLVDTAGQDEYSIFPQTYSIDINGYILVYSVTSIKSFEVIKVIHGKLLDMVGKVQIPIMLVGNKKDLHMERVISYEEGKALAESWNAAFLESSAKENQTAVDVFRRIILEAEKLE 6bt0 B 2.6 BS02 E7V B 1 E40 A62 G63 F70 Y74 E38 A60 G61 F68 Y72 3.6.5.- 0000139,0000287,0003924,0005515,0005525,0005681,0005737,0005764,0005765,0005783,0005789,0005794,0005829,0005886,0007165,0007264,0012505,0014069,0016020,0016241,0016787,0019003,0019901,0030295,0031669,0032006,0032008,0043539,0045202,0046872,0048709,0048714,0051726,0070062,0120163,1904263,2000074 remove_due_to_license_issue Q15382 29416044 203 QSKSRKIAILGYRSVGKSSLTIQFVEGQFVDSYDPTIENTFTKLITVNGQEYHLQLVDTAGQDEYSIFPQTYSIDINGYILVYSVTSIKSFEVIKVIHGKLLDMVGKVQIPIMLVGNKKDLHMERVISYEEGKALAESWNAAFLESSAKENQTAVDVFRRIILEAEKL 6bt6 A 1.05 BS01 3GK A 1 N104 Y105 S130 N132 P167 N170 T171 T235 G236 A237 G238 D240 N79 Y80 S105 N107 P142 N145 T146 T210 G211 A212 G213 D214 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677,0046872 Ki=1.23uM remove_due_to_license_issue Q9L5C7 29844038 301 PTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGAGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 6bt6 A 1.05 BS02 3GK A 2 N104 Y105 A237 N79 Y80 A212 S70 K73 S130 E166 K234 A237 S45 K48 S105 E141 K209 A212 3.5.2.6 0008800,0016787,0017001,0030655,0046677,0046872 Ki=1.23uM remove_due_to_license_issue Q9L5C7 29844038 302 PTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGAGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 6bto A 2.05 BS03 E8P A 1 R8 C66 S67 Y68 V69 H93 E94 H97 W102 H103 Y127 R8 C66 S67 Y68 V69 H93 E94 H97 W102 H103 Y127 H93 E94 H97 H103 Y152 H93 E94 H97 H103 Y152 3.4.24.19 0004222,0006508,0008237,0008270 remove_due_to_license_issue P13497 30034610 304 AATSRPERVWPDGVIPFVIGGNFTGSQRAVFRQAMRHWEKHTCVTFLERTDEDSYIVFTYRPCGCCSYVGRRGGGPQAISIGKNCDKFGIVVHELGHVVGFWHEHTRPDRDRHVSIVRENIQPGQEYNFLKMEPQEVESLGETYDFDSIMHYARNTFSRGIFLDTIVPKYEVNGVKPPIGQRTRLSKGDIAQARKLYKCPA 6bu0 B 2.427 BS01 IHP B 1 Y1595 K1597 Y1599 K1609 K1611 N1655 Y38 K40 Y42 K52 K54 N98 2.7.1.137,2.7.1.153,2.7.1.154 remove_due_to_license_issue O00443 30293811 1701 AIGGAVKLSISYRNGTLFIMVMHIKDLVTEDGADPNPYVKTYLLPDNHKTSKRKTKISRKTRNPTFNEMLVYSGYSKETLRQRELQLSVLSAESLRGNFFLGGVTLPLKDFNLSKETVKWYQLTAA 6bu0 B 2.427 BS02 IHP B 2 K1564 W1677 K7 W120 2.7.1.137,2.7.1.153,2.7.1.154 remove_due_to_license_issue O00443 30293811 1702 AIGGAVKLSISYRNGTLFIMVMHIKDLVTEDGADPNPYVKTYLLPDNHKTSKRKTKISRKTRNPTFNEMLVYSGYSKETLRQRELQLSVLSAESLRGNFFLGGVTLPLKDFNLSKETVKWYQLTAA 6bu1 A 1.584 BS03 E9S A 1 V118 R339 E434 G459 L461 D462 M515 W541 M631 D633 V116 R327 E419 G444 L446 D447 M500 W526 M616 D618 D271 E273 R339 E434 D462 D633 D269 E271 R327 E419 D447 D618 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=0.06uM remove_due_to_license_issue P9WK17 30137983 805 DRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6bu3 A 1.15 BS01 3GK A 1 N104 Y105 S130 N132 P167 N170 T171 T235 G236 S237 G238 N78 Y79 S104 N106 P141 N144 T145 T209 G210 S211 G212 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.28uM remove_due_to_license_issue B5LY47 29844038 301 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKHADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGSGGYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 6bu3 A 1.15 BS02 3GK A 2 N104 Y105 S237 N78 Y79 S211 S70 K73 S130 E166 K234 S237 S44 K47 S104 E140 K208 S211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.28uM remove_due_to_license_issue B5LY47 29844038 302 TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKHADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGSGGYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 6buv B 1.86 BS01 E9A B 1 A108 D109 A112 M115 S116 A105 D106 A109 M112 S113 2.7.7.18 0000309,0003824,0004515,0005524,0009058,0009165,0009435,0016779,0019363,0070566 remove_due_to_license_issue P9WJJ5 30969758 301 RRLGVMGGTFDPIHYGHLVAASEVADLFDLDEVVFVPSGQPWQKGRQVSAAEHRYLMTVIATASNPRFSVSRVDIDRGGPTYTKDTLADLHALHPDSELYFTTGADALASIMSWQGWEELFELARFVGVSRPGHITSLLGQLAKDALTLVEIPALAISSTDCRQRAEQSRPLWYLMPDGVVQYVSKRRLYT 6bux A 1.856 BS01 dna B 0 W211 R213 H216 T218 N244 A246 K247 H257 W285 S286 Y315 D316 D317 K318 W18 R20 H23 T25 N51 A53 K54 H64 W92 S93 Y122 D123 D124 K125 3.5.4.38 0003824 remove_due_to_license_issue Q9HC16 29941968 -5 ~ 3 RHSMDPATFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLAQRRGFLANQAKHKHGFLEGRHAALCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDKGRAAEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQNQE 6buz A 3.92 BS01 dna I 0 Q45 R63 R72 N85 W86 Q87 R118 V119 T120 Q1 R19 R28 N41 W42 Q43 R74 V75 T76 ? 0000132,0000281,0000775,0000779,0000786,0003677,0003682,0005515,0005634,0005654,0005694,0005721,0005829,0030527,0034080,0043505,0046982,0051301,0051382,0061638,0061644,0071459 remove_due_to_license_issue P49450 29269420 -72 ~ 72 QGWLKEIRKLQKSTHLLIRKLPFSRLAREICVKFTRGVDFNWQAQALLALQEAAEAFLVHLFEDAYLLTLHAGRVTLFPKDVQLARRIRGL 6buz A 3.92 BS02 dna J 0 R63 K64 L65 P66 R69 R19 K20 L21 P22 R25 ? 0000132,0000281,0000775,0000779,0000786,0003677,0003682,0005515,0005634,0005654,0005694,0005721,0005829,0030527,0034080,0043505,0046982,0051301,0051382,0061638,0061644,0071459 remove_due_to_license_issue P49450 29269420 -72 ~ 72 QGWLKEIRKLQKSTHLLIRKLPFSRLAREICVKFTRGVDFNWQAQALLALQEAAEAFLVHLFEDAYLLTLHAGRVTLFPKDVQLARRIRGL 6buz B 3.92 BS01 dna I 0 R37 K45 R46 R14 K22 R23 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 remove_due_to_license_issue P62805 29269420 -72 ~ 72 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 6buz B 3.92 BS02 dna J 0 R46 I47 S48 G49 R79 K80 T81 R23 I24 S25 G26 R56 K57 T58 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 remove_due_to_license_issue P62805 29269420 -72 ~ 72 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 6buz C 3.92 BS01 dna I 0 R12 A13 K16 R18 R21 G29 R33 R78 R1 A2 K5 R7 R10 G18 R22 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031507,0043505,0046982,0061644,0070062 remove_due_to_license_issue P04908 29269420 -72 ~ 72 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLP 6buz C 3.92 BS02 dna J 0 R30 R43 V44 A46 K76 T77 R78 R19 R32 V33 A35 K65 T66 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031507,0043505,0046982,0061644,0070062 remove_due_to_license_issue P04908 29269420 -72 ~ 72 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLP 6buz D 3.92 BS01 dna I 0 R34 Y43 I55 S56 S57 R87 S88 T89 R3 Y12 I24 S25 S26 R56 S57 T58 ? 0000786,0001530,0002227,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0005886,0006325,0006334,0010804,0019731,0030527,0031640,0042742,0043505,0046982,0050829,0050830,0061644,0061844 remove_due_to_license_issue P06899 29269420 -72 ~ 72 RSRKESYSIYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 6buz D 3.92 BS02 dna J 0 R34 K35 Y41 R3 K4 Y10 ? 0000786,0001530,0002227,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0005886,0006325,0006334,0010804,0019731,0030527,0031640,0042742,0043505,0046982,0050829,0050830,0061644,0061844 remove_due_to_license_issue P06899 29269420 -72 ~ 72 RSRKESYSIYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 6buz E 3.92 BS01 dna I 0 K49 R63 K64 L65 P66 R69 K5 R19 K20 L21 P22 R25 ? 0000132,0000281,0000775,0000779,0000786,0003677,0003682,0005515,0005634,0005654,0005694,0005721,0005829,0030527,0034080,0043505,0046982,0051301,0051382,0061638,0061644,0071459 remove_due_to_license_issue P49450 29269420 -72 ~ 72 QGWLKEIRKLQKSTHLLIRKLPFSRLAREICVKFTRGVDFNWQAQALLALQEAAEAFLVHLFEDAYLLTLHAGRVTLFPKDVQLARRIRGL 6buz E 3.92 BS02 dna J 0 R63 R72 N85 W86 Q87 R118 V119 R19 R28 N41 W42 Q43 R74 V75 ? 0000132,0000281,0000775,0000779,0000786,0003677,0003682,0005515,0005634,0005654,0005694,0005721,0005829,0030527,0034080,0043505,0046982,0051301,0051382,0061638,0061644,0071459 remove_due_to_license_issue P49450 29269420 -72 ~ 72 QGWLKEIRKLQKSTHLLIRKLPFSRLAREICVKFTRGVDFNWQAQALLALQEAAEAFLVHLFEDAYLLTLHAGRVTLFPKDVQLARRIRGL 6buz F 3.92 BS01 dna I 0 R46 I47 R79 K80 T81 R23 I24 R56 K57 T58 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 remove_due_to_license_issue P62805 29269420 -72 ~ 72 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 6buz F 3.92 BS02 dna J 0 T31 R37 K45 T8 R14 K22 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 remove_due_to_license_issue P62805 29269420 -72 ~ 72 RDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 6buz G 3.92 BS01 dna I 0 R30 R43 V44 G45 A46 K76 T77 R78 R19 R32 V33 G34 A35 K65 T66 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031507,0043505,0046982,0061644,0070062 remove_due_to_license_issue P04908 29269420 -72 ~ 72 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLP 6buz G 3.92 BS02 dna J 0 R12 A13 K16 R18 R33 R78 R1 A2 K5 R7 R22 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031507,0043505,0046982,0061644,0070062 remove_due_to_license_issue P04908 29269420 -72 ~ 72 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLP 6buz H 3.92 BS01 dna I 0 R34 K35 E36 S37 I40 Y41 R3 K4 E5 S6 I9 Y10 ? 0000786,0001530,0002227,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0005886,0006325,0006334,0010804,0019731,0030527,0031640,0042742,0043505,0046982,0050829,0050830,0061644,0061844 remove_due_to_license_issue P06899 29269420 -72 ~ 72 RSRKESYSIYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 6buz H 3.92 BS02 dna J 0 R34 Y43 S56 S57 R87 S88 T89 R3 Y12 S25 S26 R56 S57 T58 ? 0000786,0001530,0002227,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0005886,0006325,0006334,0010804,0019731,0030527,0031640,0042742,0043505,0046982,0050829,0050830,0061644,0061844 remove_due_to_license_issue P06899 29269420 -72 ~ 72 RSRKESYSIYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 6buz N 3.92 BS01 dna I 0 M18 K45 R169 R170 M18 K41 R118 R119 ? 0007059,0008643,0015144,0034080,0055085 remove_due_to_license_issue P0AEX9,Q96H22 29269420 -72 ~ 72 MDETVAEFIKRTILKIPMNELTTILKAWDFLSENQLQRQRKESVVQHLIHLCEEKRSDAALLDIIYMQFHQHQKMKQFKNSFKKVTVSFRETAVWIRIAWGTKPNQYKPTYVVYYSQRRNTPLLGQALTIASKH 6bw2 A 2.75 BS01 ECY A 1 A227 F228 L246 M250 R263 T266 L267 F270 G271 A56 F57 L75 M79 R92 T95 L96 F99 G100 ? 0042981 remove_due_to_license_issue Ki=21nM Q07820 29323899 400 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6bw5 A 3.1 BS01 TUM A 1 L46 N119 W122 K125 L126 F179 N182 N185 A188 G189 I190 N191 F249 D252 H302 R303 L39 N105 W108 K111 L112 F153 N156 N159 A162 G163 I164 N165 F223 D226 H276 R277 2.7.8.15 0003975,0003976,0005515,0005783,0005789,0006047,0006486,0006487,0006488,0016020,0016757,0016780,0019348,0042802,0043231,0046872 remove_due_to_license_issue Q9H3H5 29459785 501 PMPLLINLIVSLLGFVATVTLIPAFRGHFIAARLCGQDLNKTSRQQIPESQGVISGAVFLIILFCFIPFPFLNCAFPHHEFVALIGALLAICCMIFLGFADDVLNLRWRHKLLLPTAASLPLLMVYFTNFGNTTIHLDLGILYYVYMGLLAVFCTNAINILAGINGLEAGQSLVISASIIVFNLVELEGDCRDDHVFSLYFMIPFFFTTLGLLYHNWYPSRVFVGDTFCYFAGMTFAVVGILGHFSKTMLLFFMPQVFNFLYSLPQLLHIIPCPRHRIPRLNIKTGKLEMSYSKFKTKSLSFLGTFILKVAESLQLVTVHQSETEDGEFTECNNMTLINLLLKVLGPIHERNLTLLLLLLQILGSAITFSIRYQLVRL 6bw8 A 2.9 BS01 ECM A 1 A227 F228 M231 M250 V253 N260 R263 T266 L267 F270 G271 I294 A56 F57 M60 M79 V82 N89 R92 T95 L96 F99 G100 I123 ? 0042981 remove_due_to_license_issue Ki=<1.000000nM Q07820 29323899 400 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6bwy A 2.9 BS01 dna I 0 S78 L79 H80 G81 T82 K83 D84 H106 F108 T131 R133 Y135 Q140 L142 S143 K144 D145 S49 L50 H51 G52 T53 K54 D55 H77 F79 T102 R104 Y106 Q111 L113 S114 K115 D116 3.5.4.-,3.5.4.38 0000723,0000781,0003677,0003824,0008270,0016787 remove_due_to_license_issue O13988,Q9HC16 29596531 1 ~ 7 QLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTNHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQN 6bwy B 2.9 BS01 dna C 0 Q318 Q322 R326 Q283 Q287 R291 3.5.4.-,3.5.4.38 0000723,0000781,0003677,0003824,0008270,0016787 remove_due_to_license_issue O13988,Q9HC16 29596531 1 ~ 7 QLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTNHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQN 6bwy B 2.9 BS02 dna D 0 R76 S78 G81 T82 D84 Q104 H106 F108 T131 Y135 Q140 L142 S143 K144 D145 R47 S49 G52 T53 D55 Q75 H77 F79 T102 Y106 Q111 L113 S114 K115 D116 3.5.4.-,3.5.4.38 0000723,0000781,0003677,0003824,0008270,0016787 remove_due_to_license_issue O13988,Q9HC16 29596531 1 ~ 7 QLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTNHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQN 6bwy E 2.9 BS01 dna F 0 R76 S78 L79 H80 G81 T82 D84 H106 F108 T131 Y135 Q140 L142 S143 K144 D145 R47 S49 L50 H51 G52 T53 D55 H77 F79 T102 Y106 Q111 L113 S114 K115 D116 3.5.4.-,3.5.4.38 0000723,0000781,0003677,0003824,0008270,0016787 remove_due_to_license_issue O13988,Q9HC16 29596531 1 ~ 7 QLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTNHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQN 6bwy G 2.9 BS01 dna C 0 S78 L79 H80 G81 T82 D84 H106 F108 T131 R133 Y135 Q140 L142 S143 K144 D145 S49 L50 H51 G52 T53 D55 H77 F79 T102 R104 Y106 Q111 L113 S114 K115 D116 3.5.4.-,3.5.4.38 0000723,0000781,0003677,0003824,0008270,0016787 remove_due_to_license_issue O13988,Q9HC16 29596531 1 ~ 7 QLNELLNAGEYKIGELTFQSIRSSQELQKKNTIVNLFGIVKDFTPSRQSLHGTKDWVTTVYLWDPTCDTSSIGLQIHLFSKQGNDLPVIKQVGQPLLLHQITLRSYRDRTQGLSKDQFRYALWPDFSSNSKDTLCPQPMPRLMKTGDKEEQFALLLNKIWDEQTNHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQN 6bx6 A 2.9 BS01 EDJ A 1 L22 G23 A43 V96 G99 A156 L10 G11 A31 V84 G87 A144 D139 K141 E143 N144 D157 D127 K129 E131 N132 D145 2.7.11.1,2.7.11.31 0004672,0005524,0006468 remove_due_to_license_issue P54646 29695504 301 IGHYVLGDTLGVGTFGKVKIGEHQLTGHKVAVKILNRQKIRSLDVVGKIKREIQNLKLFRHPHIIKLYQVISTPTDFFMVMEYVSGGELFDYICKHGRVEEMEARRLFQQILSAVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNYAAPEYAGPEVDIWSCGVILYALLCGTLPFDDEHVPTLFKKIRGGVFYIPEYLNRSVATLLMHMLQVDPLKRATIKDIREHEWFKQDLPSYLF 6bxy A 1.82 BS01 EEV A 1 S155 S178 H181 F238 C241 Y276 M278 Y319 M322 Y323 W341 E363 E366 S134 S157 H160 F217 C220 Y255 M257 Y298 M301 Y302 W320 E342 E345 ? 0005634 remove_due_to_license_issue IC50=7.5nM, Kd=10.0nM O00255 29738674 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 6by8 A 1.9 BS01 FNV A 1 S155 S178 H181 F238 Y276 M278 M322 Y323 W341 E363 E366 S134 S157 H160 F217 Y255 M257 M301 Y302 W320 E342 E345 ? 0005634 remove_due_to_license_issue IC50=123nM O00255 29738674 601 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEAGSQGSALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSVPPVLTFQSEKMKGMKELLVATKINSSAIKLQLTAQSQVQMK 6byz A 2.95625 BS02 J18 A 1 A198 L201 F202 E205 Y302 Y314 T316 V360 G361 Q363 K364 I374 A479 A156 L159 F160 E163 Y260 Y272 T274 V318 G319 Q321 K322 I332 A437 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 31086331 1101 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNPINLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 6c0n A 2.001 BS01 K5C A 1 L100 K101 K103 V106 V179 Y181 Y188 F227 W229 H235 P236 Y318 L102 K103 K105 V108 V181 Y183 Y190 F229 W231 H237 P238 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=4.3nM remove_due_to_license_issue P03366 30044217 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 6c0r A 2.049 BS01 K5C A 1 L100 K101 N103 K104 V179 C181 Y188 F227 W229 H235 P236 Y318 L102 K103 N105 K106 V181 C183 Y190 F229 W231 H237 P238 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=31nM remove_due_to_license_issue P03366 30044217 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKNKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 6c0s A 2.35 BS01 EEJ A 1 R39 H40 L41 H57 L147 I151 D189 A190 C191 K192 G193 S195 T213 W215 G216 G218 C219 G226 V227 R26 H27 L28 H44 L137 I141 D182 A183 C184 K185 G186 S188 T206 W208 G209 G211 C212 G219 V220 H57 D102 K192 G193 D194 S195 G196 H44 D93 K185 G186 D187 S188 G189 3.4.21.27 0004252,0006508 Ki=89nM remove_due_to_license_issue P03951 29501396 301 IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAV 6c0t A 1.98 BS01 EE4 A 1 V368 G369 G370 F371 G372 V374 A388 I406 M438 E439 A440 C441 E445 V501 D502 G504 V32 G33 G34 F35 G36 V38 A52 I70 M102 E103 A104 C105 E109 V165 D166 G168 D484 K486 N489 D502 T521 D148 K150 N153 D166 T185 2.7.11.12 0004672,0004674,0004692,0005524,0006468 ic50=43.1nM remove_due_to_license_issue Q13976 29769318 701 EDAEAKAKYEAEAAFFANLKLSDFNIIDTLGVGGFGRVELVQLKSEESKTFAMKILKKRHIVDTRQQEHIRSEKQIMQGAHSDFIVRLYRTFKDSKYLYMLMEACLGGELWTILRDRGSFEDSTTRFYTACVVEAFAYLHSKGIIYRDLKPENLILDHRGYAKLVDFGFAKKIGFGKKTWTFCGTPEYVAPEIILNKGHDISADYWSLGILMYELLTGSPPFSGPDPMKTYNIILRGIDMIEFPKKIAKNAANLIKKLCRDNPSERLGNLKNGVKDIQKHKWFEGFNWEGLRKGTLTPPIIPSVASPTDTSNFDSFPEDNDEPPPDDNSGWDIDF 6c0u A 2.65 BS01 EE4 A 1 G50 T51 G52 S53 F54 G55 V57 A70 L74 T88 M120 E121 Y122 V123 E127 E170 L173 T183 G40 T41 G42 S43 F44 G45 V47 A60 L64 T78 M110 E111 Y112 V113 E117 E160 L163 T173 D166 K168 N171 D184 T201 D156 K158 N161 D174 T191 2.7.11.11 0000287,0001669,0001707,0001843,0002027,0003091,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0010881,0016241,0016607,0018105,0019221,0019901,0019904,0030145,0031410,0031514,0031594,0031625,0032024,0032703,0034237,0034380,0034605,0034704,0035694,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0050850,0051726,0055117,0061136,0070062,0070417,0070613,0071333,0071374,0071377,0071872,0086064,0097546,0098794,0098978,0099103,0099170,0106310,1903779,1904262,1904539,1990044,2000810 remove_due_to_license_issue P17612 29769318 400 EQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 6c1a A 2.05 BS01 dna C 0 R166 S168 D176 K186 R20 S22 D30 K40 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 GKRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1a A 2.05 BS02 dna D 0 R188 S189 P191 R209 R42 S43 P45 R63 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 GKRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1a B 2.05 BS01 dna C 0 R166 S168 G169 L170 S171 M214 R19 S21 G22 L23 S24 M67 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1a B 2.05 BS02 dna D 0 R188 S189 P191 R209 R41 S42 P44 R62 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1a E 2.05 BS01 dna G 0 R166 S168 G169 D176 K186 R188 R19 S21 G22 D29 K39 R41 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1a E 2.05 BS02 dna H 0 R188 S189 P191 R41 S42 P44 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1a F 2.05 BS01 dna G 0 R166 S168 G169 L170 S171 R19 S21 G22 L23 S24 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1a F 2.05 BS02 dna H 0 R188 S189 R209 R41 S42 R62 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1s A 2.31 BS01 EFV A 1 W812 I831 K833 D841 Y867 I879 I881 V882 A885 M953 I963 D964 W563 I582 K584 D592 Y618 I630 I632 V633 A636 M702 I712 D713 2.7.11.1,2.7.1.137,2.7.1.153,2.7.1.154 0016301,0046854 Ki=0.004uM remove_due_to_license_issue Ki=3.0nM P48736 29847724 1201 SEESQAFQRQLTALIGYDVTDVSNVHDDELEFTRRGLVTPRMAEVASRDPKLYAMHPWVTSKPLPEYLWKKIANNCIFIVIHRSTTSQTIKVSPDDTPGAILQSFFTKVLRVCGRDEYLVGETPIKNFQWVRHCLKNGEEIHVVLDTPPDPALDEVRKECDRKFRVKIRGIDIPVLTDLTVFVEANIQHGQQVLCQRRTSPKPFTEEVLWNVWLEFSIKIKDLPKGALLNLQIYCVQLLYYVNLLLIDHRFLLRRGEYVLHMWQISGSFNADKLTSATNPDKENSMSISILLDNRAEMPNQLRKQLEAIIATDPLNPLTAEDKELLWHFRYESLKHPKAYPKLFSSVKWGQQEIVAKTYQLLARREVWDQSALDVGLTMQLLDCNFSDENVRAIAVQKLESLEDDDVLHYLLQLVQAVKFEPYHDSALARFLLKRGLRNKRIGHFLFWFLRSEIAQSRHYQQRFAVILEAYLRGCGTAMLHDFTQQVQVIEMLQKVTLDIKSLSAEKYDVSSQVISQLKQKLENLQNSQLPESFRVPYDPGLKAGALAIEKCKVMASKKKPLWLEFKCADPTALSNETIGIIFKHGDDLRQDMLILQILRIMESIWETESLDLCLLPYGCISTGDKIGMIEIVKDATTIAKIQQSTVGNTFKDEVLNHWLKEKSPTEEKFQAAVERFVYSCAGYCVATFVLGIGDRHNDNIMITETGNLFHIDFGHIKERVPFVLTPDFLFVMGTSGKKTSPHFQKFQDICVKAYLALRHHTNLLIILFSMMLMTGMPTSKEDIEYIRDALTVGKNEEDAKKYFLDQIEVCRDKGWTVQFNWFLHL 6c1t A 1.84 BS01 dna B 0 R188 S189 P191 R209 M214 R41 S42 P44 R62 M67 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1t A 1.84 BS02 dna C 0 R166 K167 S168 G169 L170 D176 K186 R188 R19 K20 S21 G22 L23 D29 K39 R41 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1t D 1.84 BS01 dna B 0 R188 S189 P191 R209 R40 S41 P43 R61 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 RMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1t D 1.84 BS02 dna C 0 R166 S168 G169 L170 S171 R18 S20 G21 L22 S23 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 RMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1v A 2.3 BS01 dna C 0 R166 K167 S168 G169 D176 K186 R188 R19 K20 S21 G22 D29 K39 R41 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1v A 2.3 BS02 dna D 0 S189 P191 S42 P44 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1v B 2.3 BS01 dna C 0 R166 S168 G169 L170 S171 R20 S22 G23 L24 S25 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 GKRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1v B 2.3 BS02 dna D 0 R188 S189 P191 R209 R42 S43 P45 R63 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 GKRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMM 6c1v E 2.3 BS01 dna G 0 R166 K167 S168 G169 D176 K186 R188 R19 K20 S21 G22 D29 K39 R41 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1v E 2.3 BS02 dna H 0 S189 K190 P191 S42 K43 P44 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1v F 2.3 BS01 dna G 0 R166 S168 G169 L170 S171 R19 S21 G22 L23 S24 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c1v F 2.3 BS02 dna H 0 R188 S189 P191 R209 R41 S42 P44 R62 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6c28 C 2.09 BS01 WCA C 1 F63 F66 T76 P77 S81 L101 N107 F23 F26 T36 P37 S41 L61 N67 ? 0003700,0006355,0006950 Kd=68uM remove_due_to_license_issue Q6N8V9 29794028 201 ELKMGELSELLGYALKRAQLRVFEDFLHCVAPVQLTPAQFSVLLLLDANPGRNQTEIATTLGILRPNFVAMLDALEGRGLCVRTRILMLTDKGRATLARAKKLVATRHEDRLTELLGRDNRDALLSMLATIAREF 6c2r A 1.96 BS01 EG7 A 1 L139 E211 Y212 A213 G216 T217 R220 L263 A273 L12 E84 Y85 A86 G89 T90 R93 L136 A146 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T153 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Ki=0.8nM remove_due_to_license_issue O14965 30373917 404 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK 6c2t A 1.73 BS01 EGJ A 1 L139 Y212 A213 G216 T217 N261 L263 A273 L12 Y85 A86 G89 T90 N134 L136 A146 D256 K258 E260 N261 D274 T292 D129 K131 E133 N134 D147 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 30373917 401 WALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS 6c2x A 2.6 BS02 EHV A 1 V118 R339 E434 G459 L461 D462 M515 W541 M631 D633 V115 R328 E418 G443 L445 D446 M499 W525 M615 D617 D271 E273 R339 E434 D462 D633 D268 E270 R328 E418 D446 D617 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 30137983 802 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAFLRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6c2y A 2.74 BS01 EJS A 1 I197 R199 G200 G201 F202 G203 V205 A218 L222 A236 E239 M274 A321 L324 S334 D335 I168 R170 G171 G172 F173 G174 V176 A189 L193 A207 E210 M245 A292 L295 S305 D306 D317 K319 N322 D335 K344 T353 D288 K290 N293 D306 K315 T324 2.7.11.15 0001664,0002026,0002029,0003108,0004672,0004674,0004703,0005515,0005524,0005737,0005829,0005886,0005929,0006468,0007165,0007186,0007213,0007217,0007507,0016020,0018105,0019079,0031623,0031694,0031755,0032473,0033605,0042995,0045202,0045988,0046718,0047696,0060048,0098793,0098794,1901081 remove_due_to_license_issue P25098 29627263 701 KKILLPEPSIRSVMQKYLEDRGEVTFEKIFSQKLGYLLFRDFCLNHLEEARPLVEFYEEIKKYEKLETEEERVARSREIFDSYIMKELLACSHPFSKSATEHVQGHLGKKQVPPDLFQPYIEEICQNLRGDVFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEADMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLAVELPDSFSPELRSLLEGLLQRDVNRRLGCLGRGAQEVKESPFFRSLDWQMVFLQKYPPPLIPPRTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDTINAETDRLEARKKAKNKQLGEDYALGKDCIMHGYMSKMGNPFLTQWQRRYFYLFPNRLEWRGEGEAPQSLLTMEEIQSVEETQIKERKCLLLKIRGGKQFILQCDSDPELVQWKKELRDAYREAQQLVQRVPKMKNKP 6c31 A 3.0 BS01 dna K 0 R6 T37 R48 Y52 D57 K58 R1 T32 R43 Y47 D52 K53 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 A 3.0 BS02 dna L 0 Q8 R11 S12 T15 T47 G49 A50 H53 Q3 R6 S7 T10 T42 G44 A45 H48 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 B 3.0 BS01 dna K 0 Q8 S12 T47 A50 H53 Q3 S7 T42 A45 H48 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 B 3.0 BS02 dna L 0 T7 Q8 T37 P38 R48 Y52 D57 T2 Q3 T32 P33 R43 Y47 D52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 C 3.0 BS01 dna K 0 G36 T37 R48 Y52 D57 K58 G30 T31 R42 Y46 D51 K52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 C 3.0 BS02 dna L 0 T47 G49 A50 T41 G43 A44 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 D 3.0 BS01 dna K 0 Q8 T15 T47 H53 Q2 T9 T41 H47 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 D 3.0 BS02 dna L 0 T37 R48 Y52 D57 K58 T31 R42 Y46 D51 K52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 E 3.0 BS01 dna I 0 T37 R48 Y52 D57 T32 R43 Y47 D52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 E 3.0 BS02 dna J 0 Q8 S12 T47 A50 H53 Q3 S7 T42 A45 H48 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 F 3.0 BS01 dna I 0 Q8 S12 T47 H53 Q3 S7 T42 H48 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 F 3.0 BS02 dna J 0 R6 T7 Q8 T37 P38 R48 Y52 D57 R1 T2 Q3 T32 P33 R43 Y47 D52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 G 3.0 BS01 dna I 0 T37 R48 Y52 D57 T32 R43 Y47 D52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 G 3.0 BS02 dna J 0 T47 G49 T42 G44 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 RTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 H 3.0 BS01 dna I 0 Q8 S12 T47 H53 Q54 Q2 S6 T41 H47 Q48 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 4 ~ 23 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c31 H 3.0 BS02 dna J 0 G36 T37 R48 Y52 D57 K58 G30 T31 R42 Y46 D51 K52 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 29921668 1 ~ 23 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6c3e A 2.6 BS01 EJY A 1 K45 L78 M92 L129 H136 A155 D156 S161 F162 K37 L66 M80 L117 H124 A143 D144 S149 F150 D138 K140 E142 N143 D156 T189 D126 K128 E130 N131 D144 T160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Ki=63nM Q13546 29485864 301 VIKMKSSDFLESAELDSGGFGKVSLAFHRTQGLMIMKTVYKIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNGTLYYMAPEHLPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDLTEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQL 6c3l A 1.46092 BS01 EGP A 1 M51 A52 C53 G55 Y58 E115 M47 A48 C49 G51 Y54 E111 ? Kd=44uM remove_due_to_license_issue Kd=36000nM, IC50=27000nM P41182 29969259 201 ADSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6c3l A 1.46092 BS02 EGP B 1 D17 N21 R28 D13 N17 R24 ? Kd=44uM remove_due_to_license_issue Kd=36000nM, IC50=27000nM P41182 29969259 201 ADSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6c3n A 2.53171 BS01 EHY A 1 M51 Y58 M45 Y52 ? remove_due_to_license_issue Kd=3200000nM P41182 29969259 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKASE 6c3n A 2.53171 BS02 EHY B 1 N21 R24 N15 R18 ? remove_due_to_license_issue Kd=3200000nM P41182 29969259 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKASE 6c3n B 2.53171 BS01 EHY A 1 N21 L25 N15 L19 ? remove_due_to_license_issue Kd=3200000nM P41182 29969259 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6c3n B 2.53171 BS02 EHY B 1 M51 G55 Y58 M45 G49 Y52 ? remove_due_to_license_issue Kd=3200000nM P41182 29969259 201 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6c3u A 1.85 BS02 NY2 A 1 Y65 H67 S97 R122 Y131 Y65 H67 S97 R122 Y131 ? 0046872 remove_due_to_license_issue A0A0H3GM04 30642934 202 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFE 6c3u A 1.85 BS03 NY2 A 2 H7 T9 W34 Y39 C48 H7 T9 W34 Y39 C48 ? 0046872 remove_due_to_license_issue A0A0H3GM04 30642934 203 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFE 6c3u B 1.85 BS01 NY2 A 1 H7 T9 W34 Y39 W46 C48 H7 T9 W34 Y39 W46 C48 ? 0046872 remove_due_to_license_issue A0A0H3GM04 30642934 202 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFE 6c3u B 1.85 BS02 NY2 A 2 Y65 H67 Y131 Y65 H67 Y131 ? 0046872 remove_due_to_license_issue A0A0H3GM04 30642934 203 MLSGLNHLTLAVSQLAPSVAFYQQLLGMTLHARWDSGAYLSCGDLWLCLSLDPQRRVTPPEESDYTHYAFSISEADFASFAARLEAAGVAVWKLNRSEGASHYFLDPDGHKLELHVGSLAQRLAACREQPYKGMVFFE 6c4d A 2.52 BS01 EJP A 1 K45 L70 V76 L78 L90 M92 V134 A155 D156 L157 L159 S161 F162 K31 L56 V62 L64 L76 M78 V120 A141 D142 L143 L145 S147 F148 D138 K140 E142 N143 D156 T189 D124 K126 E128 N129 D142 T162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.3nM, Ki=0.912011nM Q13546 29485864 1100 NVIKMKSSDFLEGFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 6c4g A 2.39 BS01 EQG A 1 D80 G82 Y139 C140 E141 L179 F180 Q183 D313 G315 S316 T317 H320 D36 G38 Y95 C96 E97 L135 F136 Q139 D237 G239 S240 T241 H244 3.4.23.- 0004190,0006508 ic50=0.005uM remove_due_to_license_issue A5K302 29800827 504 DLLYKYKLYGDIDEYAYYFLDIDIGTPEQRISLILDTGSSSLSFPCAGCKNCGVHMENPFNLNNSKTSSILYCENEECPFKLNCVKGKCEYMQSYCEGSQISGFYFSDVVSVVSYNNERVTFRKLMGCHMHEESLFLYQQATGVLGMSLSKPQGIPTFVNLLFDNAPQLKQVFTICISENGGELIAGGYDPAYIVRAEKVVWENVTRKYYYYIKVRGLDMFGTNMMSSSKGLEMLVDSGSTFTHIPEDLYNKLNYFFDILCIQDMNNAYDVNKRLKMTNESFNNPLVQFDDFRKSLKSIIAKENMCVKIVDGVQCWKYLEGLPDLFVTLSNNYKMKWQPHSYLYKKESFWCKGIEKQVNNKPILGLTFFKNRQVIFDIQKNRIGFVDANCPSHP 6c5f B 1.4 BS01 7L9 B 1 P1 R36 S63 I64 S104 I107 K109 P1 R36 S63 I64 S104 I107 K109 4.1.1.84 0004167,0005126,0005615,0005737,0010760,0016829,0032760,0033981,0042438,0050178,0050729,0070062,0070374 Ki=33uM remove_due_to_license_issue P30046 29847104 201 PFLELDTNLPANRVPAGLEKRLCAAAASILGKPADRVNVTVRPGLAMALSGSTEPCAQLSISSIGVVGTAEDNRSHSAHFFEFLTKELALGQDRILIRFFPLESWQIGKIGTV 6c5q A 2.404 BS01 EKS A 1 G284 C285 F287 R288 M329 L330 L333 I341 S342 Y473 G85 C86 F88 R89 M130 L131 L134 I142 S143 Y274 ? 0003677,0004879,0005634,0006355 ic50=220nM remove_due_to_license_issue IC50=321nM P37231 30123887 501 HHHGSHMESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 6c5q A 2.404 BS02 EKS A 2 G258 I262 F264 K265 H266 R280 Q283 L465 Y473 G59 I63 F65 K66 H67 R81 Q84 L266 Y274 ? 0003677,0004879,0005634,0006355 ic50=220nM remove_due_to_license_issue IC50=321nM P37231 30123887 502 HHHGSHMESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 6c5t A 2.75 BS01 EKP A 1 I281 G284 C285 F287 R288 A292 I326 L330 L333 I341 S342 I75 G78 C79 F81 R82 A86 I120 L124 L127 I135 S136 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 30123887 501 HGSHMESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHIQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDSLHPLLQEIYKDLY 6c6k A 2.54 BS01 rna E 0 R40 Q44 L48 T50 W149 K153 G156 Y159 R189 F193 L195 N218 Y220 Y254 Y258 K261 R265 L288 H291 Q292 K298 I302 K305 K338 F341 R388 F392 K419 K426 R430 R433 R30 Q34 L38 T40 W132 K136 G139 Y142 R172 F176 L178 N201 Y203 Y237 Y241 K244 R248 L271 H274 Q275 K281 I285 K288 K321 F324 R371 F375 K402 K409 R413 R416 ? 0003723,0005515,0005737,0005829,0009615,0019060,0032091,0043657,0045070,0045071,0045087,0051097,0051607,0051707,0071357,0071360,0140374 remove_due_to_license_issue P09914 29525521 1 ~ 11 QVKDSLEQLRCHFTWELSIDDDEMPDLENRVLDQIEFLDTKYSVGIHNLLAYVKHLKGQNEEALKSLKEAENLMANVRSLVTWGNFAWMYYHMGRLAEAQTYLDKVENICKKLSNPFRYRMECPEIDCEEGWALLKCGGKNYERAKACFEKVLEVDPENPESSAGYAISAYRLDGFKLATKNHKPFSLLPLRQAVRLNPDNGYIKVLLALKLQDEGQEAEGEKYIEEALANMSSQTYVFRYAAKFYRRKGSVDKALELLKKALQETPTSVLLHHQIGLCYKAQMIQIKEATKGQPRGQNREKLDKMIRSAIFHFESAVEKKPTFEVAHLDLARMYIEAGNHRKAEENFQKLLCMKPVVEETMQDIHFHYGRFQEFQKKSDVNAIIHYLKAIKIEQASLTRDKSINSLKKLVLRKLRRKALDLESLSLLGFVYKLEGNMNEALEYYERALRLAADFE 6c6k B 2.54 BS01 rna F 0 R40 Q44 L48 T50 W149 L152 K153 G156 Y159 I185 R189 F193 N218 Y220 Y254 R257 Y258 K261 R265 L288 H291 Q292 I302 K338 F341 E354 R388 F392 K426 R32 Q36 L40 T42 W132 L135 K136 G139 Y142 I168 R172 F176 N201 Y203 Y237 R240 Y241 K244 R248 L271 H274 Q275 I285 K321 F324 E337 R371 F375 K409 ? 0003723,0005515,0005737,0005829,0009615,0019060,0032091,0043657,0045070,0045071,0045087,0051097,0051607,0051707,0071357,0071360,0140374 remove_due_to_license_issue P09914 29525521 1 ~ 11 DHQVKDSLEQLRCHFTWELSIDDDEMPDLENRVLDQIEFLDTKYSVGIHNLLAYVKHLKGQNEEALKSLKEAENLMQNVRSLVTWGNFAWMYYHMGRLAEAQTYLDKVENICKSNPFRYRMECPEIDCEEGWALLKCGGKNYERAKACFEKVLEVDPENPESSAGYAISAYRLDGFKLATKNHKPFSLLPLRQAVRLNPDNGYIKVLLALKLQDEGQEAEGEKYIEEALANMSSQTYVFRYAAKFYRRKGSVDKALELLKKALQETPTSVLLHHQIGLCYKAQMIQIKEATKGQPRGQNREKLDKMIRSAIFHFESAVEKKPTFEVAHLDLARMYIEAGNHRKAEENFQKLLCMKPVVEETMQDIHFHYGRFQEFQKKSDVNAIIHYLKAIKIEQASLTRDKSINSLKKLVLRKLRRKALDLESLSLLGFVYKLEGNMNEALEYYERALRLAAD 6c6o A 2.3 BS02 ENG A 1 R339 G459 L461 D462 W541 M631 D633 R320 G437 L439 D440 W519 M606 D608 D271 E273 R339 E434 D462 D633 D265 E267 R320 E412 D440 D608 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=0.005uM remove_due_to_license_issue P9WK17 30137983 803 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6c7b A 2.133 BS01 ENY A 1 S275 R339 G459 L461 D462 M515 M631 D633 S274 R328 G444 L446 D447 M500 M616 D618 D271 E273 R339 E434 D462 D633 D270 E272 R328 E419 D447 D618 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=1.5uM remove_due_to_license_issue P9WK17 30137983 801 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6c7d A 1.79 BS01 EOJ A 1 L770 I826 F830 Q859 F862 L195 I251 F255 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.17nM remove_due_to_license_issue O00408 30070482 2001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 6c7e A 1.43 BS01 EOG A 1 L770 L809 I826 F830 M847 Q859 F862 L195 L234 I251 F255 M272 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.24nM remove_due_to_license_issue O00408 30070482 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 6c7f A 1.82 BS01 EOS A 1 T768 L770 T805 I826 F830 M847 F862 T190 L192 T227 I248 F252 M269 F284 3.1.4.17 0004114,0007165,0008081 ic50=0.00000001M remove_due_to_license_issue O00408 30070482 1001 DDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 6c7g A 1.68 BS01 EOY A 1 H656 T768 L770 D808 L809 F830 M845 M847 Q859 F862 H81 T193 L195 D233 L234 F255 M270 M272 Q284 F287 3.1.4.17 0004114,0007165,0008081 ic50=18.2nM remove_due_to_license_issue O00408 30070482 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6c7i A 1.713 BS01 EP7 A 1 H656 T768 L770 D808 L809 I826 F830 F862 H81 T193 L195 D233 L234 I251 F255 F287 3.1.4.17 0004114,0007165,0008081 ic50=0.38nM remove_due_to_license_issue O00408 30070482 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 6c7j A 1.85 BS01 EPV A 1 H656 T768 L770 L809 I826 M845 M847 F862 I866 H81 T193 L195 L234 I251 M270 M272 F287 I291 3.1.4.17 0004114,0007165,0008081 ic50=1.32nM remove_due_to_license_issue O00408 30070482 1001 SAMDDEYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFLD 6c7q A 1.51 BS01 EO1 A 1 W374 P375 F376 L385 C429 Y432 N433 H437 V439 M442 W26 P27 F28 L37 C81 Y84 N85 H89 V91 M94 ? remove_due_to_license_issue Ki=0.700000nM, IC50=9.1nM O60885 30015487 501 KVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMPDE 6c7r A 1.5 BS01 EO4 A 1 W81 P82 F83 V87 L92 D145 I146 M149 W24 P25 F26 V30 L35 D88 I89 M92 ? Kd=2.2nM remove_due_to_license_issue Kd=0.800000nM, Ki=<1.000000nM, IC50=2.0nM O60885 30015487 201 RQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 6c7w A 1.28 BS02 LMS A 1 Q92 H94 H96 F131 L198 T199 T200 P202 Q91 H93 H95 F129 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3410nM remove_due_to_license_issue Ki=3410nM P00918 29685656 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6c7x A 1.5 BS02 EO7 A 1 Q92 H94 H96 F131 V135 L198 T199 T200 P202 Q91 H93 H95 F129 V133 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=65.2nM remove_due_to_license_issue Ki=65nM P00918 29685656 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6c85 A 2.4 BS01 PLQ A 1 R114 N153 C154 R108 N147 C148 0004073,0006520,0008652,0016620,0046983,0050661,0051287 remove_due_to_license_issue A0A179UL48 30107909 401 SKKRCGVLGATGAVGTRFILLLEQSPLLELVAVGASERSAGKKYRDAVRWKQASPMPASVADLTVRRCAPSEFSDCDIIFSGLDPAGDIEMAFLKANFAVFSNAKNYRLDPIVPLVVPLVNAGHIDVIPAQRKHYGLDKGLIVCNSNCAVVGLVIPAKALIQKFGPIESVSMVTMQAVSGAGGVSSMDIFDNIVPFIPGEEGKIATESRKILGNLNPDLAGFSDQQPLQVSVACNRVPVLDGHTVCASLRFVNRPAPTASQVRDALREYKSEVQLLGCPSAPRQAIHVLDDVDRPQPRLDRDTEAGYACSVGRIREDDSGVFDIQFVALSHNTVLGASGSSILNAESAILKGYI 6c8c A 1.5 BS01 EQ7 B 1 L71 L101 Q105 L108 L116 L71 L101 Q105 L108 L116 2.7.7.-,2.7.7.7 remove_due_to_license_issue Q920Q2,Q9QUG2 31178121 201 SHMKSFFDKKRSERISNGGFRPAAPNLAGAVEFSDVKTLLKEWITTISDPMEEDILQVVRYCTDLIEEKDLEKLDLVIKYMKRLMQQSVESVWNMAFDFILDNVQVVLQQTYGSTLKVT 6c8c B 1.5 BS01 EQ7 B 1 K69 L71 L108 Y112 S114 K67 L69 L103 Y107 S109 2.7.7.-,2.7.7.7 ic50=0.78uM remove_due_to_license_issue Q920Q2,Q9QUG2 31178121 201 MKSFFDKKRSERISNGGFRPAAPNLAGAVEFSDVKTLLKEWITTISDPMEEDILQVVRYCTDLIEEKDLEKLDLVIKYMKRLMQQSVWNMAFDFILDNVQVVLQQTYGSTLKVT 6c8p A 1.635 BS02 EQA A 1 R339 E434 G459 L461 D462 M515 W541 M631 D633 R329 E423 G448 L450 D451 M504 W530 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R329 E423 D451 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=0.2uM remove_due_to_license_issue P9WK17 30137983 804 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDVGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6c8x A 1.613 BS01 BVR A 1 D25 G27 A28 D30 I47 G48 V82 D25 G27 A28 D30 I47 G48 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.5pM remove_due_to_license_issue P03366 30346745 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6c8x B 1.613 BS01 BVR A 1 D125 G127 D129 G148 G149 I150 D25 G27 D29 G48 G49 I50 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03366 30346745 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6c91 C 2.895 BS01 EQD C 1 N107 D149 M154 N162 F195 I247 N34 D76 M81 N89 F109 I161 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue Ki=440nM, IC50=1200nM P41148 29528635 403 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTGGGGKTVWDWELMN 6c98 A 1.85 BS02 ER7 B 1 W29 Q34 S230 G232 W26 Q31 S225 G227 ? remove_due_to_license_issue P55899 29782488 101 HLSLLYHLTAVSSPAPGTPAFWVSGWLGPQQYLSYNSLRGEAEPCGAWVWENQVSWYWEKETTDLRIKEKLFLEAFKALGGPYTLQGLLGCELGPDNTSVPTAKFALNGEEFMNFDLKQGTWGGDWPEALAISQRWQQQDKAANKELTFLLFSCPHRLREHLERGRGNLEWKEPPSMRLKARPSSPGFSVLTCSAFSFYPPELQLRFLRNGLAAGTGQGDFGPNSDGSFHASSSLTVKSGDEHHYCCIVQHAGLAQPLRVEL 6c98 B 1.85 BS01 ER7 B 1 S52 Y63 L64 L65 S52 Y63 L64 L65 ? 0000139,0001913,0001916,0002237,0002474,0002481,0002502,0002503,0002726,0005198,0005515,0005576,0005615,0005765,0005783,0005788,0005794,0005829,0005886,0005925,0006826,0006879,0006955,0007608,0007611,0009897,0009986,0010977,0012507,0016020,0019885,0019886,0023026,0030670,0031901,0031902,0031905,0032092,0033077,0034756,0035580,0042026,0042605,0042612,0042613,0042802,0042803,0042824,0045646,0048260,0050680,0050768,0050778,0050870,0051289,0055038,0060586,0070062,0071281,0071283,0071316,1900121,1900122,1904434,1904437,1904724,1990000,1990712,2000774,2000978 Kd~80uM remove_due_to_license_issue P61769 29782488 101 IQRTPKIQVYSRHPAENGKSNFLNCYVSGFHPSDIEVDLLKNGERIEKVEHSDLSFSKDWSFYLLYYTEFTPTEKDEYACRVNHVTLSQPKIVKWDRDM 6c99 A 2.0 BS01 EQY A 1 W29 Q34 G49 S230 G232 W26 Q31 G46 S227 G229 ? Kd=2.4uM remove_due_to_license_issue P55899 29782488 301 HLSLLYHLTAVSSPAPGTPAFWVSGWLGPQQYLSYNSLRGEAEPCGAWVWENQVSWYWEKETTDLRIKEKLFLEAFKALGGKGPYTLQGLLGCELGPDNTSVPTAKFALNGEEFMNFDLKQGTWGGDWPEALAISQRWQQQDKAANKELTFLLFSCPHRLREHLERGRGNLEWKEPPSMRLKARPSSPGFSVLTCSAFSFYPPELQLRFLRNGLAAGTGQGDFGPNSDGSFHASSSLTVKSGDEHHYCCIVQHAGLAQPLRVELE 6c99 B 2.0 BS01 EQY A 1 S52 D53 Y63 L65 Y67 S52 D53 Y63 L65 Y67 ? 0000139,0001913,0001916,0002237,0002474,0002481,0002502,0002503,0002726,0005198,0005515,0005576,0005615,0005765,0005783,0005788,0005794,0005829,0005886,0005925,0006826,0006879,0006955,0007608,0007611,0009897,0009986,0010977,0012507,0016020,0019885,0019886,0023026,0030670,0031901,0031902,0031905,0032092,0033077,0034756,0035580,0042026,0042605,0042612,0042613,0042802,0042803,0042824,0045646,0048260,0050680,0050768,0050778,0050870,0051289,0055038,0060586,0070062,0071281,0071283,0071316,1900121,1900122,1904434,1904437,1904724,1990000,1990712,2000774,2000978 remove_due_to_license_issue P61769 29782488 301 IQRTPKIQVYSRHPAENGKSNFLNCYVSGFHPSDIEVDLLKNGERIEKVEHSDLSFSKDWSFYLLYYTEFTPTEKDEYACRVNHVTLSQPKIVKWDRDM 6c9n A 2.1 BS01 SGV A 1 S8 D12 G48 N52 F102 F116 Q172 D257 S7 D11 G36 N40 F90 F104 Q160 D245 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=16500nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9n A 2.1 BS02 SGV A 2 G225 V243 E246 Q249 L288 G213 V231 E234 Q237 L276 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=16500nM P9WID5 31002508 402 TIAVTGSIATDHLMRFPGRFVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9n B 2.1 BS01 SGV B 1 S8 D12 G48 V49 N52 F102 F116 Q172 D257 S7 D11 G39 V40 N43 F93 F107 Q163 D248 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=16500nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEQVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9n B 2.1 BS02 SGV B 2 G225 V243 E246 Q249 V255 L288 G216 V234 E237 Q240 V246 L279 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=16500nM P9WID5 31002508 402 TIAVTGSIATDHLMRFPGRFSEQVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9p A 2.0 BS01 MTP A 1 S8 D12 G48 V49 N52 F102 F116 Q172 R176 D257 S7 D11 G38 V39 N42 F92 F106 Q162 R166 D247 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=2300nM P9WID5 31002508 403 TIAVTGSIATDHLMRFPGRFSEVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9p A 2.0 BS02 MTP A 2 G225 P226 V243 E246 V285 L288 G215 P216 V233 E236 V275 L278 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=2300nM P9WID5 31002508 404 TIAVTGSIATDHLMRFPGRFSEVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9p B 2.0 BS01 MTP B 1 S8 D12 G48 V49 N52 F102 F116 Q172 Q173 R176 D257 S7 D11 G39 V40 N43 F93 F107 Q163 Q164 R167 D248 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=2300nM P9WID5 31002508 404 TIAVTGSIATDHLMRFPGRFSEKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9p B 2.0 BS02 MTP B 2 G225 P226 V243 E246 Q249 V255 L288 G216 P217 V234 E237 Q240 V246 L279 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=2300nM P9WID5 31002508 405 TIAVTGSIATDHLMRFPGRFSEKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9r A 2.1 BS01 ERJ A 1 S8 D12 G47 G48 N52 F102 F116 Q172 R176 G254 D257 S21 D25 G60 G61 N65 F115 F129 Q185 R189 G267 D270 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=197nM P9WID5 31002508 401 GLQGTENLYFQSHMTIAVTGSIATDHLMRFPGRFSEQLLPEHLHKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 6c9r A 2.1 BS02 ERJ A 2 G225 V243 G238 V256 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=197nM P9WID5 31002508 402 GLQGTENLYFQSHMTIAVTGSIATDHLMRFPGRFSEQLLPEHLHKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 6c9r B 2.1 BS01 ERJ B 1 S8 D12 G48 N52 F102 F116 R176 D257 S21 D25 G61 N65 F115 F129 R189 D270 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=197nM P9WID5 31002508 401 GLQGTENLYFQSHMTIAVTGSIATDHLMRFPGRFSEQLLPEHLHKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 6c9r B 2.1 BS02 ERJ B 2 P226 V243 E246 Q249 P239 V256 E259 Q262 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue IC50=197nM P9WID5 31002508 402 GLQGTENLYFQSHMTIAVTGSIATDHLMRFPGRFSEQLLPEHLHKVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 6c9s A 2.23 BS01 ERP A 1 S8 D12 G48 V49 F102 F116 Q172 Q173 D257 S7 D11 G39 V40 F93 F107 Q163 Q164 D248 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue Ki=48nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEQVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9s A 2.23 BS02 ERP B 1 F17 S36 L38 F16 S27 L29 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue Ki=48nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEQVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9s B 2.23 BS01 ERP A 1 F17 S36 L38 F16 S26 L28 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue Ki=48nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9s B 2.23 BS02 ERP B 1 S8 D12 G48 V49 N52 F102 F116 Q172 Q173 D257 S7 D11 G38 V39 N42 F92 F106 Q162 Q163 D247 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 remove_due_to_license_issue Ki=48nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVL 6c9v A 1.7 BS01 ERS A 1 S8 D12 G48 V49 N52 F102 F116 Q172 Q173 A175 R176 D257 S7 D11 G39 V40 N43 F93 F107 Q163 Q164 A166 R167 D248 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 Ki=120.2nM remove_due_to_license_issue Ki=120nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEQVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 6c9v B 1.7 BS01 ERS B 1 S8 D12 G48 V49 N52 F102 F116 Q172 Q173 A175 R176 D257 S7 D11 G39 V40 N43 F93 F107 Q163 Q164 A166 R167 D248 2.7.1.20 0000287,0004001,0005515,0005524,0005525,0005886,0006166,0016301,0016772,0032567,0044209 Ki=120.2nM remove_due_to_license_issue Ki=120nM P9WID5 31002508 401 TIAVTGSIATDHLMRFPGRFSEQVSLSFLVDDLVMHRGGVAGNMAFAIGVLGGEVALVGAAGADFADYRDWLKARGVNCDHVLISETAHTARFTCTTDVDMAQIASFYPGAMSEARNIKLADVVSAIGKPELVIIGANDPEAMFLHTEECRKLGLAFAADPSQQLARLSGEEIRRLVNGAAYLFTNDYEWDLLLSKTGWSEADVMAQIDLRVTTLGPKGVDLVEPDGTTIHVGVVPETSQTDPTGVGDAFRAGFLTGRSAGLGLERSAQLGSLVAVLVLESTGTQEWQWDYEAAASRLAGAYGEHAAAEIVAVLA 6cb5 A 1.78 BS01 EV7 A 1 P1 K32 Y36 H62 S63 I64 F113 P1 K32 Y36 H62 S63 I64 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=4.3uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cb5 A 1.78 BS02 EV7 B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=4.3uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cb5 C 1.78 BS01 EV7 A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=4.3uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cb5 C 1.78 BS02 EV7 C 1 P1 K32 H62 S63 I64 P1 K32 H62 S63 I64 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=4.3uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbf A 2.3 BS01 EWD A 1 P1 M2 K32 Y36 I64 F113 P1 M2 K32 Y36 I64 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=6.8uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbf C 2.3 BS01 EWD A 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=6.8uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbf C 2.3 BS02 EWD C 1 P1 K32 Y36 H62 I64 V106 F113 P1 K32 Y36 H62 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=6.8uM remove_due_to_license_issue P14174 29575754 201 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbg A 2.0 BS01 EWG B 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Ki=113000nM P14174 29575754 204 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbg B 2.0 BS01 EWG B 1 P1 K32 H62 I64 V106 F113 P1 K32 H62 I64 V105 F112 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=113uM remove_due_to_license_issue Ki=113000nM P14174 29575754 204 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbg B 2.0 BS02 EWG C 1 Y95 N97 Y94 N96 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=113uM remove_due_to_license_issue Ki=113000nM P14174 29575754 204 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbh B 2.0 BS01 EWJ C 1 Y95 N97 Y95 N97 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 remove_due_to_license_issue Ki=510nM P14174 29575754 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cbh C 2.0 BS01 EWJ C 1 P1 K32 Y36 H62 S63 I64 V106 F113 P1 K32 Y36 H62 S63 I64 V106 F113 5.3.2.1,5.3.3.12 0001516,0001819,0002020,0002906,0004167,0005125,0005126,0005515,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0007166,0008284,0009986,0010629,0010760,0016853,0019752,0030330,0030336,0030890,0031666,0031982,0032760,0033033,0034774,0042056,0042127,0042327,0042802,0043030,0043066,0043518,0045087,0048146,0050178,0050918,0051248,0061078,0061081,0070062,0070207,0070374,0090238,0090398,0141163,1902166,1904813,2000343,2000773 Ki=0.51uM remove_due_to_license_issue Ki=510nM P14174 29575754 202 PMFIVNTNVPRASVPDGFLSELTQQLAQATGKPPQYIAVHVVPDQLMAFGGSSEPCALCSLHSIGKIGGAQNRSYSKLLCGLLAERLRISPDRVYINYYDMNAANVGWNNSTFA 6cc8 A 1.95 BS01 dna C 0 R22 R23 S24 L26 S27 K42 R22 R23 S24 L26 S27 K42 ? 0003677 remove_due_to_license_issue O95983 30980593 1 ~ 12 MERKRWECPALPQGWEREEVPRRSGLSAGHRDVFYYSPSGKKFRSKPQLARYLGGSMDLSTFDFRTGKMLM 6cc8 A 1.95 BS02 dna D 0 R44 S45 R44 S45 ? 0003677 remove_due_to_license_issue O95983 30980593 1 ~ 12 MERKRWECPALPQGWEREEVPRRSGLSAGHRDVFYYSPSGKKFRSKPQLARYLGGSMDLSTFDFRTGKMLM 6cc8 B 1.95 BS01 dna E 0 R22 R23 S24 L26 S27 K42 R22 R23 S24 L26 S27 K42 ? 0003677 remove_due_to_license_issue O95983 30980593 1 ~ 12 MERKRWECPALPQGWEREEVPRRSGLSAGHRDVFYYSPSGKKFRSKPQLARYLGGSMDLSTFDFRTGKMLM 6cc8 B 1.95 BS02 dna F 0 R44 S45 R65 R44 S45 R65 ? 0003677 remove_due_to_license_issue O95983 30980593 1 ~ 12 MERKRWECPALPQGWEREEVPRRSGLSAGHRDVFYYSPSGKKFRSKPQLARYLGGSMDLSTFDFRTGKMLM 6cc9 B -1.00 BS05 EWS B 1 K5 L6 V7 I55 L56 Y71 M72 T74 K5 L6 V7 I55 L56 Y71 M72 T74 3.6.5.2 0000139,0000165,0001934,0003924,0003925,0005515,0005525,0005737,0005741,0005789,0005829,0005886,0005925,0007165,0007265,0008283,0008542,0009898,0010467,0010628,0012505,0014009,0016020,0016601,0016787,0019003,0021897,0030036,0030857,0032228,0035022,0035914,0043495,0043524,0044877,0048169,0048873,0051146,0051402,0060252,0060441,0060509 remove_due_to_license_issue P01116 30122370 239 MTEYKLVVVGAVGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEKMSKDGKKKKKKSKTKC 6cck A 1.61 BS01 EXJ A 1 P8 G9 A37 S39 F70 S71 D72 L73 M74 L102 P8 G9 A37 S39 F70 S71 D72 L73 M74 L102 H18 K42 R91 S129 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=0.037uM remove_due_to_license_issue P0A6I6 29498517 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6ccl A 1.77 BS01 EXG A 1 A37 L73 M74 L102 A36 L72 M73 L101 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=273uM remove_due_to_license_issue P0A6I6 29498517 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6ccm A 1.79 BS01 EXP A 1 P8 G9 T10 A37 L73 M74 L102 P8 G9 T10 A37 L73 M74 L102 H18 K42 R91 S129 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=5.6uM remove_due_to_license_issue P0A6I6 29498517 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6ccn A 1.87 BS01 EXS A 1 G9 L73 M74 R88 L102 M105 N106 G7 L71 M72 R86 L100 M103 N104 H18 K42 R91 S129 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=30uM remove_due_to_license_issue P0A6I6 29498517 201 KRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6cco A 1.82 BS01 EXV A 1 G9 F70 L73 M74 A75 R88 L102 N106 G9 F70 L73 M74 A75 R88 L102 N106 H18 K42 R91 S129 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=0.051uM remove_due_to_license_issue P0A6I6 29498517 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6ccq A 1.92 BS01 EX7 A 1 P8 G9 A37 L73 M74 A75 L102 M105 N106 P6 G7 A35 L71 M72 A73 L100 M103 N104 H18 K42 R91 S129 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=0.25uM remove_due_to_license_issue P0A6I6 29498517 201 KRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKL 6ccs A 2.06 BS01 EXD A 1 L73 M74 L102 M105 N106 L72 M73 L101 M104 N105 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=230uM remove_due_to_license_issue P0A6I6 29498517 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6ccx B -1.00 BS05 EWS B 1 K5 V7 D54 L56 Q70 Y71 T74 K5 V7 D54 L56 Q70 Y71 T74 3.6.5.2 0000139,0000165,0001934,0003924,0003925,0005515,0005525,0005737,0005741,0005789,0005829,0005886,0005925,0007165,0007265,0008283,0008542,0009898,0010467,0010628,0012505,0014009,0016020,0016601,0016787,0019003,0021897,0030036,0030857,0032228,0035022,0035914,0043495,0043524,0044877,0048169,0048873,0051146,0051402,0060252,0060441,0060509 remove_due_to_license_issue P01116 30122370 237 MTEYKLVVVGAVGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEKMSKDGKKKKKKSKTKC 6ccy A 2.18 BS01 EX4 A 1 L156 G157 G159 G162 K163 V164 A177 T211 M227 E228 A230 E234 M281 F438 F442 L16 G17 G19 G22 K23 V24 A37 T71 M87 E88 A90 E94 M141 F298 F302 D274 K276 N279 D292 T312 D134 K136 N139 D152 T172 2.7.11.1,2.7.11.13 0004672,0004674,0005524,0006468 ic50=0.003uM remove_due_to_license_issue P31749,Q16513 29655979 501 GSLRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTESRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGPSDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSEVDTRYFDEEFTAQMITITEQEMFRDFDYIADWEG 6cd4 A 1.23 BS01 EX1 A 1 W81 P82 L92 L94 Y139 I146 W39 P40 L50 L52 Y97 I104 ? ic50=5.14uM remove_due_to_license_issue O60885 30102854 201 TNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6cd5 A 1.58 BS01 R4L A 1 W81 P82 F83 L92 L94 Y139 N140 I146 W40 P41 F42 L51 L53 Y98 N99 I105 ? remove_due_to_license_issue O60885 30102854 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6cdj A 1.13 BS01 GR8 A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=2pM remove_due_to_license_issue Q5RZ08 29763303 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6cdj B 1.13 BS01 GR8 A 1 D25 A28 D29 D30 I47 G48 P81 V82 I84 D25 A28 D29 D30 I47 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q5RZ08 29763303 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6cdl A 1.25 BS01 GR5 B 1 R8 D25 A28 D30 G48 P81 V82 R8 D25 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q5RZ08 29763303 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6cdl B 1.25 BS01 GR5 B 1 D25 G27 D29 D30 I47 G48 G49 I50 D25 G27 D29 D30 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=0.012nM remove_due_to_license_issue Q5RZ08 29763303 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6ce2 A 2.15 BS01 SVR B 1 L2 G30 L32 G33 R34 K49 Y52 L2 G29 L31 G32 R33 K48 Y51 N28 G30 L32 H48 K49 Y52 Y73 D99 N27 G29 L31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0035821,0042130,0047498,0050482,0090729 remove_due_to_license_issue P82114 29985425 202 SLVELGKMILQETGKNPVKSYGAYGCNCGVLGRGKPKDATDRCCYVHKCCYKKLTNCNPKKDRYSYDWKNKTIVCGEENPCLKQLCECDKAVAICLRENKGTYNKKRDVYLKPFCDKGRDC 6ce2 B 2.15 BS01 SVR B 1 L2 P18 Y22 G30 G33 R34 K49 Y52 P68 K69 K70 L2 P17 Y21 G29 G32 R33 K48 Y51 P59 K60 K61 N28 G30 L32 H48 K49 Y52 Y73 D99 N27 G29 L31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0016042,0035821,0042130,0047498,0050482,0090729 Kd=0.5uM remove_due_to_license_issue P82114 29985425 202 SLVELGKMILQETGKNPVKSYGAYGCNCGVLGRGKPKDATDRCCYVHKCCYKKLTNCNPKKDRYSYDWKNKTIVCGEENPCLKQLCECDKAVAICLRENKGTYNKKRDVYLKPFCDKGRDC 6ce6 A 1.6 BS04 EYP A 1 W1143 G1154 R1155 W1182 Y1184 Y1189 W36 G47 R48 W75 Y77 Y82 3.5.1.-,3.5.1.98 0008270 ic50=5.1uM remove_due_to_license_issue IC50=5100nM, Kd=8000nM Q9UBN7 29741882 1307 SPLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKFG 6ce8 A 1.55 BS04 EYV A 1 W1143 G1154 R1155 W1182 Y1184 Y1189 W36 G47 R48 W75 Y77 Y82 3.5.1.-,3.5.1.98 0008270 ic50=390uM remove_due_to_license_issue IC50=390000nM Q9UBN7 29741882 1308 SPLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKFG 6cea A 1.6 BS04 EYY A 1 W1143 G1154 R1155 W1182 Y1184 Y1189 W35 G46 R47 W74 Y76 Y81 3.5.1.-,3.5.1.98 0008270 remove_due_to_license_issue IC50=>720000nM Q9UBN7 29741882 1305 PLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKF 6cec A 1.55 BS04 EY7 A 1 W1143 R1155 W1182 Y1184 Y1189 W36 R48 W75 Y77 Y82 3.5.1.-,3.5.1.98 0008270 ic50=45uM remove_due_to_license_issue IC50=45000nM Q9UBN7 29741882 1309 SPLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKF 6ced A 1.7 BS04 EYA A 1 W1143 R1155 W1182 Y1184 Y1189 W35 R47 W74 Y76 Y81 3.5.1.-,3.5.1.98 0008270 Kd=1.5uM remove_due_to_license_issue IC50=2300nM, Kd=1500nM Q9UBN7 29741882 1304 PLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKF 6cee A 1.55 BS04 EYM A 1 W1143 G1154 R1155 W1182 Y1184 Y1189 W36 G47 R48 W75 Y77 Y82 3.5.1.-,3.5.1.98 0008270 ic50=65uM remove_due_to_license_issue IC50=65000nM Q9UBN7 29741882 1304 SPLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKF 6cef A 1.8 BS04 EYJ A 1 W1143 G1154 R1155 W1182 Y1184 Y1189 W35 G46 R47 W74 Y76 Y81 3.5.1.-,3.5.1.98 0008270 ic50=180uM remove_due_to_license_issue IC50=180000nM Q9UBN7 29741882 1307 PLPWCPHLVAVCPIPAAGLDVTQPCGDCGTIQENWVCLSCYQVYCGRYINGHMLQHHGNSGHPLVLSYIDLSAWCYYCQAYVHHQALLDVKNIAHQNKFG 6ceh A 1.43 BS02 EZ1 A 1 H94 H119 L198 T199 T200 P202 H93 H118 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=36.5nM remove_due_to_license_issue Ki=37nM P00918 29795760 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ceh A 1.43 BS03 EZ1 A 2 W5 H10 H15 W16 D19 W4 H9 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=36.5nM remove_due_to_license_issue Ki=37nM P00918 29795760 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6cex A 2.57 BS01 NHE A 1 G135 S136 W153 G126 S127 W144 ? 0019031,0019064,0046789 remove_due_to_license_issue Q91MA7 29610325 401 GATLCLGHHAVPNGTLVKTITDDQIEVTNATELVQSSSTGKICNNPHRILDGIDCTLIDALLGDPHCDVFQNETWDLFVERSKAFSNCYPYDVPDYASLRSLVASSGTLEFITEGFTWTGVTQNGGSNACKRGPGSGFFSRLNWLTKSGSTYPVLNVTMPNNDNFDKLYIWGVHHPSTNQEQTSLYVQASGRVTVSTRRSQQTIIPNIGSRPWVRGLSSRISIYWTIVKPGDVLVINSNGNLIAPRGYFKMRTGKSSIMRSDAPIDTCISECITPNGSIPNDKPFQNVNKITYGACPKYVKQNTLKLATGMRNVPEK 6cf5 A 2.04 BS01 NHE A 1 L133A S136 S137 W153 Q226 L132 S135 S136 W152 Q225 ? 0019031,0019064,0046789 remove_due_to_license_issue Q6DQ33 29610325 401 DPGDQICIGYHANNSTEQVDTIMEKNVTVTHAQDILEKKHNGKLCDLDGVKPLILRDCSVAGWLLGNPMCDEFINVPEWSYIVEKANPVNDLCYPGDFNDYEELKHLLSRINHFEKIQIIPKSSWSSHEASLGVSSACPYQGKSSFFRNVVWLIKKNSTYPTIKRSYNNTNQEDLLVLWGIHHPNDAAEQTKLYQNPTTYISVGTSTLNQRLVPRIATRSKVNGQSGRMEFFWTILKPNDAINFESNGNFIAPEYAYKIVKKGDSTIMKSELEYGNCNTKCQTPMGAINSSMPFHNIHPLTIGECPKYVKSNRLVLATGLRNSP 6cf7 A 2.719 BS01 EZ7 B 1 H18 H38 T318 H8 H28 T315 ? 0019031,0019064,0046789 remove_due_to_license_issue A7Y8I1 30846569 201 DTICIGYHANNSTDTVDTVLEKNVTVTHSVNLLEDSHNGKLCRLKGIAPLQLGNCSVAGWILGNPECELLISRESWSYIVEKPNPENGTCYPGHFADYEELREQLSSVSSFERFEIFPKESSWPNHTTTGVSASCSHNGESSFYKNLLWLTGKNGLYPNLSKSYANNKEKEVLVLWGVHHPPNIGDQRALYHKENAYVSVVSSHYSRKFTPEIAKRPKVRDQEGRINYYWTLLEPGDTIIFEANGNLIAPRYAFALSRGFGSGIINSNAPMDECDAKCQTPQGAINSSLPFQNVHPVTIGECPKYVRSAKLRMVTGLRNIPS 6cf7 B 2.719 BS01 EZ7 B 1 V18 G20 W21 I45 I48 T49 V52 N53 I56 V18 G20 W21 I45 I48 T49 V52 N53 I56 ? 0019031,0019064,0046789 remove_due_to_license_issue F2NZB4 30846569 201 GLFGAIAGFIEGGWTGMVDGWYGYHHQNEQGSGYAADQKSTQNAINGITNKVNSVIEKMNTQFTAVGKEFNKLERRMENLNKKVDDGFIDIWTYNAELLVLLENERTLDFHDSNVKNLYEKVKSQLKNNAKEIGNGCFEFYHKCNDECMESVKNGTYDYPKYSEESKLNRE 6cfc A 2.04 BS01 BLG A 1 E390 S399 V400 S401 Q408 F409 M410 L413 Y463 N464 G466 E498 E364 S373 V374 S375 Q382 F383 M384 L387 Y437 N438 G440 E472 0000270,0008933,0016020 Kd=210uM remove_due_to_license_issue 29758058 601 YSIEKLKKEENSLAKDYYIYRLLEKNKISKKDAQDLNSHIFRYIGKIKSELEKINPKYAKCYTYTANTILDANLTCQSVRLNSLVFIASLNSKDRTTLAQTFKNQRPDLTNLLLAFNTSDPMSYIVQKEDINGFFKLYNYSKKYDLDLNTSLVNKLPNHIGFKDFAQNIIIKKENPKFRHSMLEINPENVSEDSAFYLGVNALTYDKTELAYDFFKKAAQSFKSQSNKDNAIFWMWLIKNNEEDLKTLSQSSSLNIYSLYAKELTNTPFPKIESLNPSKKKNNFNMQDPFAWQKINKQIRDANASQLDVLAKEFDTQETLPIYAYILERKNNFKKHYFIMPYYDNIKDYNKTRQALILAIARQESRFIPTAISVSYALGMMQFMPFLANHIGEKELKIPNFDQDFMFKPEIAYYFGNYHLNYLESRLKSPLFVAYAYNGGIGFTNRMLARNDMFKTGKFEPFLSMELVPYQESRIYGKKVLANYIVYRHLLNDSIKISDIFENLIQ 6cfd A 2.57 BS01 EZA A 1 D27 I29 Y61 Y63 M93 L115 M190 D17 I19 Y51 Y53 M83 L105 M180 3.4.21.92 0004176,0004252,0005737,0006508,0006515,0008236,0009368,0051117 remove_due_to_license_issue Q3XX76 29784838 402 IPTVIRAYDIYSRLLKDRIIMLSGQVTDDLANSIIAQLLFLDAQDSEKDIYLYINSPGGSVTAGMAIYDTMNFVKADVQTIVMGMAASMGSFLLTAGTKGKRFALPNAEIMIHQPLGGAQGQATEIEIAARHILQTRERLNKILAERTGQPLEVIEKDTDRDNYMTAEQAKAYGLIDEVME 6cfd B 2.57 BS01 EZA A 1 L49 T80 F83 L40 T71 F74 3.4.21.92 0004176,0004252,0005737,0006508,0006515,0008236,0009368,0051117 remove_due_to_license_issue Q3XX76 29784838 402 IPTVIERAYDIYSRLLKDRIIMLSGQVTDDLANSIIAQLLFLDAQDSEKDIYLYINSPGGSVTAGMAIYDTMNFVKADVQTIVMGMAASMGSFLLTAGTKGKRFALPNAEIMIHQPLGGAQGQATEIEIAARHILQTRERLNKILAERTGQPLEVIEKDTDRDNYMTAEQAKAYGLIDEVME 6cgp A 2.5 BS02 F1Y A 1 S531 H574 G582 F583 H614 F643 D705 L712 Y745 S90 H133 G141 F142 H173 F202 D264 L271 Y304 ? ic50=0.058uM remove_due_to_license_issue A7YT55 29790770 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6cgt A 2.6 BS01 GLC B 1 K232 F259 K232 F259 D135 R227 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 2.4.1.19 0003824,0004556,0005576,0005975,0016757,0030246,0043169,0043895,0046872,2001070 remove_due_to_license_issue P30920 9738912 1 DPDTAVTNKQSFSTDVIYQVFTDRFLDGNPSNNPTGAAYDATCSNLKLYCGGDWQGLINKINDNYFSDLGVTALWISQPVENIFATINYSGVTNTAYHGYWARDFKKTNPYFGTMADFQNLITTAHAKGIKIVIDFAPNHTSPAMETDTSFAENGRLYDNGTLVGGYTNDTNGYFHHNGGSDFSSLENGIYKNTYDLADFNHNNATIDKYFKDAIKLWLDMGVDGIRVDAVKHMPLGWQKSWMSSIYAHKPVFTFGEWFLGSAASDADNTDFANKSGMSLLDFRFNSAVRNVFRDNTSNMYALDSMINSTATDYNQVNDQVTFIDNHDMDRFKTSAVNNRRLEQALAFTLTSRGVPAIYYGTEQYLTGNGDPDNRAKMPSFSKSTTAFNVISKLAPLRKSNPAIAYGSTQQRWINNDVYVYERKFGKSVAVVAVNRNLSTSASITGLSTSLPTGSYTDVLGGVLNGNNITSTNGSINNFTLAAGATAVWQYTTAETTPTIGHVGPVMGKPGNVVTIDGRGFGSTKGTVYFGTTAVTGAAITSWEDTQIKVTIPSVAAGNYAVKVAASGVNSNAYNNFTILTGDQVTVRFVVNNASTTLGQNLYLTGNVAELGNWSTGSTAIGPAFNQVIHQYPTWYYDVSVPAGKQLEFKFFKKNGSTITWESGSNHTFTTPASGTATVTVNWQ 6cgt A 2.6 BS02 DAG B 1 Y195 A230 H233 E257 D328 Y195 A230 H233 E257 D328 D135 R227 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 2.4.1.19 0003824,0004556,0005576,0005975,0016757,0030246,0043169,0043895,0046872,2001070 remove_due_to_license_issue P30920 9738912 2 DPDTAVTNKQSFSTDVIYQVFTDRFLDGNPSNNPTGAAYDATCSNLKLYCGGDWQGLINKINDNYFSDLGVTALWISQPVENIFATINYSGVTNTAYHGYWARDFKKTNPYFGTMADFQNLITTAHAKGIKIVIDFAPNHTSPAMETDTSFAENGRLYDNGTLVGGYTNDTNGYFHHNGGSDFSSLENGIYKNTYDLADFNHNNATIDKYFKDAIKLWLDMGVDGIRVDAVKHMPLGWQKSWMSSIYAHKPVFTFGEWFLGSAASDADNTDFANKSGMSLLDFRFNSAVRNVFRDNTSNMYALDSMINSTATDYNQVNDQVTFIDNHDMDRFKTSAVNNRRLEQALAFTLTSRGVPAIYYGTEQYLTGNGDPDNRAKMPSFSKSTTAFNVISKLAPLRKSNPAIAYGSTQQRWINNDVYVYERKFGKSVAVVAVNRNLSTSASITGLSTSLPTGSYTDVLGGVLNGNNITSTNGSINNFTLAAGATAVWQYTTAETTPTIGHVGPVMGKPGNVVTIDGRGFGSTKGTVYFGTTAVTGAAITSWEDTQIKVTIPSVAAGNYAVKVAASGVNSNAYNNFTILTGDQVTVRFVVNNASTTLGQNLYLTGNVAELGNWSTGSTAIGPAFNQVIHQYPTWYYDVSVPAGKQLEFKFFKKNGSTITWESGSNHTFTTPASGTATVTVNWQ 6cgt A 2.6 BS03 GLC C 1 W101 D371 R375 W101 D371 R375 D135 R227 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 2.4.1.19 0003824,0004556,0005576,0005975,0016757,0030246,0043169,0043895,0046872,2001070 remove_due_to_license_issue P30920 9738912 1 DPDTAVTNKQSFSTDVIYQVFTDRFLDGNPSNNPTGAAYDATCSNLKLYCGGDWQGLINKINDNYFSDLGVTALWISQPVENIFATINYSGVTNTAYHGYWARDFKKTNPYFGTMADFQNLITTAHAKGIKIVIDFAPNHTSPAMETDTSFAENGRLYDNGTLVGGYTNDTNGYFHHNGGSDFSSLENGIYKNTYDLADFNHNNATIDKYFKDAIKLWLDMGVDGIRVDAVKHMPLGWQKSWMSSIYAHKPVFTFGEWFLGSAASDADNTDFANKSGMSLLDFRFNSAVRNVFRDNTSNMYALDSMINSTATDYNQVNDQVTFIDNHDMDRFKTSAVNNRRLEQALAFTLTSRGVPAIYYGTEQYLTGNGDPDNRAKMPSFSKSTTAFNVISKLAPLRKSNPAIAYGSTQQRWINNDVYVYERKFGKSVAVVAVNRNLSTSASITGLSTSLPTGSYTDVLGGVLNGNNITSTNGSINNFTLAAGATAVWQYTTAETTPTIGHVGPVMGKPGNVVTIDGRGFGSTKGTVYFGTTAVTGAAITSWEDTQIKVTIPSVAAGNYAVKVAASGVNSNAYNNFTILTGDQVTVRFVVNNASTTLGQNLYLTGNVAELGNWSTGSTAIGPAFNQVIHQYPTWYYDVSVPAGKQLEFKFFKKNGSTITWESGSNHTFTTPASGTATVTVNWQ 6cgt A 2.6 BS04 DAG C 1 Y89 D371 Y89 D371 D135 R227 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 2.4.1.19 0003824,0004556,0005576,0005975,0016757,0030246,0043169,0043895,0046872,2001070 remove_due_to_license_issue P30920 9738912 2 DPDTAVTNKQSFSTDVIYQVFTDRFLDGNPSNNPTGAAYDATCSNLKLYCGGDWQGLINKINDNYFSDLGVTALWISQPVENIFATINYSGVTNTAYHGYWARDFKKTNPYFGTMADFQNLITTAHAKGIKIVIDFAPNHTSPAMETDTSFAENGRLYDNGTLVGGYTNDTNGYFHHNGGSDFSSLENGIYKNTYDLADFNHNNATIDKYFKDAIKLWLDMGVDGIRVDAVKHMPLGWQKSWMSSIYAHKPVFTFGEWFLGSAASDADNTDFANKSGMSLLDFRFNSAVRNVFRDNTSNMYALDSMINSTATDYNQVNDQVTFIDNHDMDRFKTSAVNNRRLEQALAFTLTSRGVPAIYYGTEQYLTGNGDPDNRAKMPSFSKSTTAFNVISKLAPLRKSNPAIAYGSTQQRWINNDVYVYERKFGKSVAVVAVNRNLSTSASITGLSTSLPTGSYTDVLGGVLNGNNITSTNGSINNFTLAAGATAVWQYTTAETTPTIGHVGPVMGKPGNVVTIDGRGFGSTKGTVYFGTTAVTGAAITSWEDTQIKVTIPSVAAGNYAVKVAASGVNSNAYNNFTILTGDQVTVRFVVNNASTTLGQNLYLTGNVAELGNWSTGSTAIGPAFNQVIHQYPTWYYDVSVPAGKQLEFKFFKKNGSTITWESGSNHTFTTPASGTATVTVNWQ 6cgt A 2.6 BS05 OPG A 1 Y100 H140 D229 E257 H327 D328 Y100 H140 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 D135 R227 D229 E257 H327 D328 2.4.1.19 0003824,0004556,0005576,0005975,0016757,0030246,0043169,0043895,0046872,2001070 remove_due_to_license_issue P30920 9738912 703 DPDTAVTNKQSFSTDVIYQVFTDRFLDGNPSNNPTGAAYDATCSNLKLYCGGDWQGLINKINDNYFSDLGVTALWISQPVENIFATINYSGVTNTAYHGYWARDFKKTNPYFGTMADFQNLITTAHAKGIKIVIDFAPNHTSPAMETDTSFAENGRLYDNGTLVGGYTNDTNGYFHHNGGSDFSSLENGIYKNTYDLADFNHNNATIDKYFKDAIKLWLDMGVDGIRVDAVKHMPLGWQKSWMSSIYAHKPVFTFGEWFLGSAASDADNTDFANKSGMSLLDFRFNSAVRNVFRDNTSNMYALDSMINSTATDYNQVNDQVTFIDNHDMDRFKTSAVNNRRLEQALAFTLTSRGVPAIYYGTEQYLTGNGDPDNRAKMPSFSKSTTAFNVISKLAPLRKSNPAIAYGSTQQRWINNDVYVYERKFGKSVAVVAVNRNLSTSASITGLSTSLPTGSYTDVLGGVLNGNNITSTNGSINNFTLAAGATAVWQYTTAETTPTIGHVGPVMGKPGNVVTIDGRGFGSTKGTVYFGTTAVTGAAITSWEDTQIKVTIPSVAAGNYAVKVAASGVNSNAYNNFTILTGDQVTVRFVVNNASTTLGQNLYLTGNVAELGNWSTGSTAIGPAFNQVIHQYPTWYYDVSVPAGKQLEFKFFKKNGSTITWESGSNHTFTTPASGTATVTVNWQ 6cha C 1.8 BS02 PBA C 1 S190 C191 S195 V213 W215 S42 C43 S47 V65 W67 M192 G193 D194 S195 G196 M44 G45 D46 S47 G48 3.4.21.1 0004252,0006508 Ki=40uM remove_due_to_license_issue Ki=40nM P00766 3584139 1 ANTPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 6cha G 1.8 BS02 PBA G 1 S190 C191 M192 S195 V213 W215 G216 S42 C43 M44 S47 V65 W67 G68 G193 S195 G196 G45 S47 G48 3.4.21.1 0004252,0006508 Ki=40uM remove_due_to_license_issue Ki=40nM P00766 3584139 1 ANTPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 6chh A 2.3 BS01 F0P A 1 Y11 Y20 Y25 G63 S64 G65 T67 Y69 D85 Y86 C141 D142 V143 T163 L164 A169 S201 Y204 S213 Y242 Y20 Y29 Y34 G70 S71 G72 T74 Y76 D92 Y93 C148 D149 V150 T170 L171 A176 S208 Y211 S220 Y249 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0030760,0031100,0032259,0034356,0045722,0090312 remove_due_to_license_issue Ki=89nM, IC50=4360nM, Kd=2700nM P40261 29320176 301 SSGLVPRGSMESGFTSKDTYLSHFNPRDYLEKYYKSRHSAESQILKHLLKNLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIVVTDYSDQNLQELEKWLKAAPAAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPPADCVLSTLCLDAACPDLPTYCRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVARKLSR 6chl A 2.2 BS01 EXJ A 1 G9 A37 S39 F70 S71 D72 L73 M74 L102 G8 A36 S38 F69 S70 D71 L72 M73 L101 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=9nM remove_due_to_license_issue P0A6I6 29551072 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAVD 6chm A 2.28 BS01 F1V A 1 A37 F70 M74 R88 L102 N106 A36 F69 M73 R87 L101 N105 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=199uM remove_due_to_license_issue P0A6I6 29551072 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6chn A 2.03 BS01 F1D A 1 A37 S39 F70 S71 D72 L73 M74 L86 R88 L102 N106 A35 S37 F68 S69 D70 L71 M72 L84 R86 L100 N104 H18 K42 R91 S129 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=11nM remove_due_to_license_issue P0A6I6 29551072 201 KRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6cho A 1.85 BS01 F14 A 1 P8 T10 A37 F70 S71 D72 L73 M74 R88 L102 N106 P8 T10 A37 F70 S71 D72 L73 M74 R88 L102 N106 H18 K42 R91 S129 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=167nM remove_due_to_license_issue P0A6I6 29551072 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6chp A 1.94 BS01 F0Y A 1 A37 A38 S39 S71 D72 L73 M74 L86 R88 L102 N106 A36 A37 S38 S70 D71 L72 M73 L85 R87 L101 N105 H18 K42 R91 S129 H17 K41 R90 S128 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=0.075nM remove_due_to_license_issue P0A6I6 29551072 201 QKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6chq A 1.79 BS01 F0V A 1 G9 T10 A37 L73 M74 Y98 L102 G9 T10 A37 L73 M74 Y98 L102 H18 K42 R91 S129 H18 K42 R91 S129 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 ic50=4.4uM remove_due_to_license_issue P0A6I6 29551072 201 MQKRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLAV 6chv A 2.9 BS01 dna I 0 S23 G24 R25 A36 S39 S20 G21 R22 A33 S36 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 FKVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYG 6chv A 2.9 BS02 dna J 0 T34 A36 T37 R40 T46 A47 T49 L52 T31 A33 T34 R37 T43 A44 T46 L49 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 FKVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYG 6chv B 2.9 BS01 dna E 0 S23 G24 R25 A36 S39 K45 S19 G20 R21 A32 S35 K41 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 KVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYG 6chv B 2.9 BS02 dna F 0 T34 A36 T37 R40 T46 A47 T49 L52 T30 A32 T33 R36 T42 A43 T45 L48 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 KVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYG 6chv C 2.9 BS01 dna I 0 T34 A36 T37 R40 T49 L52 T31 A33 T34 R37 T46 L49 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 FKVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLY 6chv C 2.9 BS02 dna J 0 S23 G24 R25 A36 S39 K45 S20 G21 R22 A33 S36 K42 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 FKVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLY 6chv D 2.9 BS01 dna E 0 V33 T34 A36 T37 R40 T46 T49 L52 V29 T30 A32 T33 R36 T42 T45 L48 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 KVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYGESN 6chv D 2.9 BS02 dna F 0 S23 G24 R25 S39 S19 G20 R21 S35 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 KVSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYGESN 6chv G 2.9 BS01 dna K 0 S23 G24 R25 R26 S39 S18 G19 R20 R21 S34 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 VSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYGESNE 6chv G 2.9 BS02 dna L 0 T34 A36 T37 R40 A47 T49 L52 T29 A31 T32 R35 A42 T44 L47 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 VSHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYGESNE 6chv H 2.9 BS01 dna K 0 T34 T37 R40 T49 L52 T28 T31 R34 T43 L46 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 SHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYG 6chv H 2.9 BS02 dna L 0 S23 G24 R25 A36 S39 S17 G18 R19 A30 S33 ? 0000976,0003677,0003700,0005515,0006355,0046982,0097351 remove_due_to_license_issue Q7A224 30793388 1 ~ 21 SHPGEMIARDLEDMGVSGRRFAHNIGVTPATVSRLLAGKTALTPSLSIRIAAALGSTPEFWLRLQSNYDLRQLENQIDTSGIVLYG 6cis A 1.51 BS01 X26 A 1 W81 P82 Q85 L92 N140 I146 W40 P41 Q44 L51 N99 I105 ? ic50=0.3uM remove_due_to_license_issue O60885 30102854 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6ciy A 1.68 BS01 F3J A 1 W81 P82 Q85 L92 L94 Y139 N140 W40 P41 Q44 L51 L53 Y98 N99 ? ic50=0.41uM remove_due_to_license_issue O60885 30102854 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6cj1 A 1.53 BS01 F2S A 1 W81 P82 Q85 L92 L94 Y139 N140 I146 W40 P41 Q44 L51 L53 Y98 N99 I105 ? remove_due_to_license_issue O60885 30102854 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6cj5 A 2.8 BS01 F4G A 1 L90 A111 M162 G165 C225 D226 L21 A42 M93 G96 C156 D157 D205 K207 N210 D226 S253 D136 K138 N141 D157 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9HBH9 29526098 402 GSTDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6cje A 3.36 BS01 F4A A 1 K113 M162 L212 C225 D226 K43 M92 L142 C155 D156 D205 K207 N210 D226 S253 D135 K137 N140 D156 S162 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9HBH9 29526098 402 STDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGPCGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6cjh A 3.6 BS02 ET8 A 1 L90 D226 L21 D157 D205 K207 N210 D226 S253 D136 K138 N141 D157 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9HBH9 29526098 402 GSTDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6cjj A 1.74 BS01 ADP A 1 N40 A44 M87 N95 G124 V125 G126 F127 T174 N36 A40 M83 N91 G120 V121 G122 F123 T170 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P46598 30679438 303 QGETHEFTAEISQLMSLIINTVYSNKEIFLRELISNASDALDKIRYQALSDPSQLESEPELFIRIIPQKDQKVLEIRDSGIGMTKADLVNNLGTIAKSGTKSFMEALSAGADVSMIGQFGVGFYSLFLVADHVQVISKHNDDEQYVWESNAGGKFTVTLDETNERLGRGTMLRLFLKEDQLEYLEEKRIKEVVKKHSEFVAYPIQLVVTKEVEK 6cjp A 2.6 BS01 F5S A 1 L37 N40 D43 A44 K47 D82 M87 N95 G126 F127 L130 T174 L176 L36 N39 D42 A43 K46 D81 M86 N94 G125 F126 L129 T171 L173 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P46598 30679438 301 LYFQGETHEFTAEISQLMSLIINTVYSNKEIFLRELISNASDALDKIRYQALSDPSQLESEPELFIRIIPQKDQKVLEIRDSGIGMTKADLVNNLGTIAKSGTKSFMEALSAGADVSMIGQFGVGFYSLFLVADHVQVISKHNDDEQYVWESNGKFTVTLDETNERLGRGTMLRLFLKEDQLEYLEEKRIKEVVKKHSEFVAYPIQLVVTKEVE 6cjr A 1.8 BS01 E0G A 1 A44 K47 M87 N95 L96 F127 Y128 W151 A39 K42 M82 N90 L91 F122 Y123 W146 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P46598 30679438 301 GETHEFTAEISQLMSLIINTVYSNKEIFLRELISNASDALDKIRYQALSDPSQLESEPELFIRIIPQKDQKVLEIRDSGIGMTKADLVNNLGTIAKSGTKSFMEALSAGADVSMIGQFGVGFYSLFLVADHVQVISKHNDDEQYVWESNAGGKFTVTLDETNERLGRGTMLRLFLKEDQLEYLEEKRIKEVVKKHSEFVAYPIQLVVTKEVEK 6cjw A 3.38 BS01 FYV A 1 L90 A111 L143 M162 G165 L20 A41 L73 M92 G95 D205 K207 N210 D226 S253 D135 K137 N140 D156 S160 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9HBH9 29526098 402 STDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6cjy A 3.05 BS01 F4J A 1 M162 G165 L212 C225 D226 M93 G96 L143 C156 D157 D205 K207 N210 D226 S253 D136 K138 N141 D157 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9HBH9 29526098 402 GSTDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6ck3 A 2.9 BS01 F67 A 1 M162 D226 M93 D157 D205 K207 N210 D226 S253 D136 K138 N141 D157 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=550nM Q9HBH9 29526098 402 GSTDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6ck6 A 3.32 BS02 N45 A 1 L90 K113 F159 M162 G165 N210 L212 C225 D226 L21 K44 F90 M93 G96 N141 L143 C156 D157 D205 K207 N210 D226 S253 D136 K138 N141 D157 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=1.000000nM, Ki=3.0nM Q9HBH9 29526098 402 GSTDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6ckc A 2.8 BS01 F5J A 1 P314 L315 L319 Y324 F327 G365 E392 K393 D419 M420 E435 L436 C449 P302 L303 L307 Y312 F315 G353 E380 K381 D407 M408 E423 L424 C437 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 remove_due_to_license_issue IC50=25nM, Kd=6.0nM, EC50=40nM O14744 30034588 701 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 6cki A 2.95 BS01 FZJ A 1 V98 A111 K161 M162 L212 C225 D226 V29 A42 K92 M93 L143 C156 D157 D205 K207 N210 D226 S253 D136 K138 N141 D157 S161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=55nM Q9HBH9 29526098 402 GSTDSFSGRFEDVYQLQEDVLGEGAHARVQTCINLITSQEYAVKIIEKQPGHIRSRVFREVEMLYQCQGHRNVLELIEFFEEEDRFYLVFEKMRGGSILSHIHKRRHFNELEASVVVQDVASALDFLHNKGIAHRDLKPENILCEHPNQVSPVKICDFGGSAEYMAPEVVEAFSEEASIYDKRCDLWSLGVILYILLSGYPPFVGRCCGACPACQNMLFESIQEGKYEFPDKDWAHISCAAKDLISKLLVRDAKQRLSAAQVLQHPWVQGC 6ckl A 2.684 BS02 DAN A 1 K142 L161 E162 P164 R165 K142 L161 E162 P164 R165 2.7.7.43 0005737,0008781,0016779 remove_due_to_license_issue P0A0Z8 31583886 703 MEKQNIAVILARQNSKGLPLKNLRKMNGISLLGHTINAAISSKCFDRIIVSTDGGLIAEEAKNFGVEVVLRPAELASDTASSISGVIHALETIGSNSGTVTLLQPTSPLRTGAHIREAFSLFDEKIKGSVVSACPMEHHPLKTLLQINNGEYAPMRHLSDLEQPRQQLPQAFRPNGAIYINDTASLIANNCFFIAPTKLYIMSHQDSIDIDTELDLQQAENILNH 6ckl A 2.684 BS03 DAN B 1 S82 Q104 Y179 S82 Q104 Y179 2.7.7.43 0005737,0008781,0016779 remove_due_to_license_issue P0A0Z8 31583886 301 MEKQNIAVILARQNSKGLPLKNLRKMNGISLLGHTINAAISSKCFDRIIVSTDGGLIAEEAKNFGVEVVLRPAELASDTASSISGVIHALETIGSNSGTVTLLQPTSPLRTGAHIREAFSLFDEKIKGSVVSACPMEHHPLKTLLQINNGEYAPMRHLSDLEQPRQQLPQAFRPNGAIYINDTASLIANNCFFIAPTKLYIMSHQDSIDIDTELDLQQAENILNH 6ckl B 2.684 BS01 DAN A 1 S82 Q104 Y179 F192 S82 Q104 Y179 F192 2.7.7.43 0005737,0008781,0016779 remove_due_to_license_issue P0A0Z8 31583886 703 MEKQNIAVILARQNSKGLPLKNLRKMNGISLLGHTINAAISSKCFDRIIVSTDGGLIAEEAKNFGVEVVLRPAELASDTASSISGVIHALETIGSNSGTVTLLQPTSPLRTGAHIREAFSLFDEKIKGSVVSACPMEHHPLKTLLQINNGEYAPMRHLSDLEQPRQQLPQAFRPNGAIYINDTASLIANNCFFIAPTKLYIMSHQDSIDIDTELDLQQAENILNH 6ckl B 2.684 BS02 DAN B 1 K142 L161 E162 P164 R165 K142 L161 E162 P164 R165 2.7.7.43 0005737,0008781,0016779 remove_due_to_license_issue P0A0Z8 31583886 301 MEKQNIAVILARQNSKGLPLKNLRKMNGISLLGHTINAAISSKCFDRIIVSTDGGLIAEEAKNFGVEVVLRPAELASDTASSISGVIHALETIGSNSGTVTLLQPTSPLRTGAHIREAFSLFDEKIKGSVVSACPMEHHPLKTLLQINNGEYAPMRHLSDLEQPRQQLPQAFRPNGAIYINDTASLIANNCFFIAPTKLYIMSHQDSIDIDTELDLQQAENILNH 6ckr A 1.62 BS01 F5V A 1 W81 P82 Q85 V87 D88 K91 L92 N140 I146 W39 P40 Q43 V45 D46 K49 L50 N98 I104 ? ic50=0.05uM remove_due_to_license_issue IC50=50nM O60885 29657099 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 6cks A 1.72 BS01 F5Y A 1 W81 P82 Q85 V87 D88 L92 N140 I146 W38 P39 Q42 V44 D45 L49 N97 I103 ? ic50=0.015uM remove_due_to_license_issue IC50=15nM O60885 29657099 201 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6ckw A 2.06 BS01 F6D A 1 P8 G9 A37 S39 F70 S71 D72 L73 M74 Y98 L102 M105 P6 G7 A35 S37 F68 S69 D70 L71 M72 Y96 L100 M103 H18 K42 R91 S129 H16 K40 R89 S127 2.7.7.3 0003824,0004595,0005515,0005524,0005737,0009058,0015937,0016779,0042802 Kd=0.83nM remove_due_to_license_issue P0A6I6 29551072 201 KRAIYPGTFDPITNGHIDIVTRATQMFDHVILAIAASPSKKPMFTLEERVALAQQATAHLGNVEVVGFSDLMANFARNQHATVLIRGLRAVADFEYEMQLAHMNRHLMPELESVFLMPSKEWSFISSSLVKEVARHQGDVTHFLPENVHQALMAKLA 6ckx A 2.8 BS02 8M1 A 1 I733 G734 A754 F813 M816 H818 D819 L866 I12 G13 A33 F82 M85 H87 D88 L135 D859 K861 N864 D877 S889 T898 D128 K130 N133 D146 S158 T167 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue IC50=13nM Q9NYV4 30067358 1102 RCVDKFDIIGIIGEGTYGQVYKAKDKDTGELVALKKVRLDNEKEGFPITAIREIKILRQLIHRSVVNMKEIVTDKGAFYLVFEYMDHDLMGLLESGLVHFSEDHIKSFMKQLMEGLEYCHKKNFLHRDIKCSNILLNNSGQIKLADFGLARLYNSEESRPYTNKVITLWYRPPELLLGEERYTPAIDVWSCGCILGELFTKKPIFQANLELAQLELISRLCGSPCPAVWPDVIKLPYFNTMKPKKQYRRRLREEFSFIPSAALDLLDHMLTLDPSKRCTAEQTLQSDFLKDVE 6clv A 2.3 BS01 6MB A 1 R52 D84 N103 M128 D167 F172 A199 K203 R204 R239 R45 D77 N96 M121 D160 F165 A192 K196 R197 R232 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046677,0046872 remove_due_to_license_issue O05701 30065703 300 TKTKIMGILNVTPDSLSNVESAVTRVKAMMDEGADIIDVGGVSTRPGHEMITVEEELNRVLPVVEAIVGFDVKISVDTFRSEVAEACLKLGVDIINDQWAGLYDHRMFQVVAKYDAEIVLMHNGNGNRDEPVVEEMLTSLLAQAHQAKIAGIPSNKIWLDPGIGFAKTRNEEAEVMARLDELVATEYPVLLATSRKRFTKKMMGYDTTPVERDEVTAATTAYGIMKGVRAVRVHNVELNAKLAKGIDFLKENENAR 6cmj A 2.4 BS01 F6J A 1 I171 G174 V179 A192 K194 F267 L269 V270 G273 P274 L319 D330 I11 G14 V19 A32 K34 F92 L94 V95 G98 P99 L144 D155 D312 K314 S316 N317 D330 T350 D137 K139 S141 N142 D155 T175 2.7.11.17 0004672,0005524,0006468 ic50=5nM remove_due_to_license_issue IC50=25nM Q96RR4 29653895 501 QLDQYTLKDEIGKGSYGVVKLAYNENDNTYYAMKVLSKKKLIRQAGGCIQPRGPIEQVYQEIAILKKLDHPNVVKLVEVLDDPNEDHLYMVFELVNQGPVMEVPTLKPLSEDQARFYFQDLIKGIEYLHYQKIIHRDIKPSNLLVGEDGHIKIADFGVSNEFKGSDALLSNTVGTPAFMAPESLSETRKIFSGKALDVWAMGVTLYCFVFGQCPFMDERIMCLHSKIKSQALEFPDQPDIAEDLKDLITRMLDKNPESRIVVPEIKLHPWVTRHGAEPLPSEDENCTL 6cmn A 1.796 BS01 rna D 0 Y13 K22 K23 R47 Q48 R49 R52 Q54 Q85 A87 K88 Y9 K18 K19 R43 Q44 R45 R48 Q50 Q81 A83 K84 ? 0003676,0003723 remove_due_to_license_issue G1TM83 29961805 18 ~ 44 ETRPNHTIYINNLNSKIKKDELKKSLHAIFSRFGQILDILVPRQRTPRGQAFVIFKEVSSATNALRSMQGFPFYDKPMAIQYAKTDKRIPA 6cmr A 2.21 BS01 5OD A 1 E110 R111 F113 T219 E249 E250 T253 L254 Q257 P491 K492 Q495 E106 R107 F109 T212 E233 E234 T237 L238 Q241 P457 K458 Q461 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue IC50=70.0nM Q06124 30375376 601 TSRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLADLVQYYMEHHGQLKEDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQSHPGDFVLSVRTGDDSNDGKSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHSDYINANIIMPEKKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETLQRR 6cms A 2.68 BS01 5OD A 1 R111 F113 T218 T219 T253 L254 Q257 P491 K492 Q495 R107 F109 T214 T215 T241 L242 Q245 P461 K462 Q465 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue IC50=70.0nM Q06124 30375376 601 TSRRWFHPNITGVEAENLLLTRGVDGSFLARPSPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAKLVQYYMEHHGQLKEKNGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQSHPGDFVLSVRTGDDKGESNDGKSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKKQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHSDYINANIIMPEKKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETLQR 6cn5 A 2.3 BS01 F7M A 1 Q286 L287 C320 H323 L324 M365 A368 V376 F377 F388 L396 I397 F401 H479 Q22 L23 C56 H59 L60 M101 A104 V112 F113 F124 L132 I133 F137 H215 ? 0003677,0004879,0005634,0006355 Ki=0.02uM remove_due_to_license_issue IC50=120nM, Ki=20nM P51449 30130103 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQ 6cn6 A 2.45 BS01 F7J A 1 Q286 L287 C320 H323 M365 A368 V376 F377 F388 I400 F401 H479 Q22 L23 C56 H59 M101 A104 V112 F113 F124 I136 F137 H215 ? 0003677,0004879,0005634,0006355 ic50=5nM remove_due_to_license_issue IC50=5.0nM P51449 30130103 4000 ASLTEIEHLVQSVSKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELSQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVV 6cnj A 3.7 BS01 NCT A 1 W156 C199 Y204 W152 C195 Y200 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue Ki=2nM, IC50=430nM, EC50=2400nM P43681 29720657 402 ETRAHAEERLLKKLFSGYNKWSRPVANISDVVLVRFGLSIAQLIDVDEKNQMMTTNVWVKQEWHDYKLRWDPADYENVTSIRIPSELIWRPDIVLYNNADGDFAVTHLTKAHLFHDGRVQWTPPAIYKSSCSIDVTFFPFDQQNCTMKFGSWTYDKAKIDLVNMHSRVDQLDFWESGEWVIVDAVGTYNTRKYECCAEIYPDITYAFVIRRLPLFYTINLIIPCLLISCLTVLVFYLPSECGEKITLCISVLLSLTVFLLLITEIIPSTSLVIPLIGEYLLFTMIFVTLSIVITVFVLNVHHRSPRTHTMPTWVRRVFLDIVPRLLLMKRFERSVKEDWKYVAMVIDRIFLWMFIIVCLLGTVGLFLPPW 6cnk A 3.9 BS03 NCT A 1 W156 Y204 W152 Y200 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 remove_due_to_license_issue Ki=2nM, IC50=430nM, EC50=2400nM P43681 29720657 405 ETRAHAEERLLKKLFSGYNKWSRPVANISDVVLVRFGLSIAQLIDVDEKNQMMTTNVWVKQEWHDYKLRWDPADYENVTSIRIPSELIWRPDIVLYNNADGDFAVTHLTKAHLFHDGRVQWTPPAIYKSSCSIDVTFFPFDQQNCTMKFGSWTYDKAKIDLVNMHSRVDQLDFWESGEWVIVDAVGTYNTRKYECCAEIYPDITYAFVIRRLPLFYTINLIIPCLLISCLTVLVFYLPSECGEKITLCISVLLSLTVFLLLITEIIPSTSLVIPLIGEYLLFTMIFVTLSIVITVFVLNVHHRSPRTHTMPTWVRRVFLDIVPRLLLMKRFERSVKEDWKYVAMVIDRIFLWMFIIVCLLGTVGLFLPPW 6cnp A 2.1 BS01 dna C 0 R166 K167 S168 G169 L170 S171 K186 R19 K20 S21 G22 L23 S24 K39 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6cnp A 2.1 BS02 dna D 0 R188 S189 P191 R41 S42 P44 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6cnp B 2.1 BS01 dna E 0 R166 K167 S168 G169 L170 S171 K186 R14 K15 S16 G17 L18 S19 K34 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 PALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRT 6cnp B 2.1 BS02 dna F 0 R188 S189 P191 R195 R36 S37 P39 R43 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 PALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRT 6cnq A 2.151 BS01 dna D 0 R188 S189 P191 R209 R41 S42 P44 R62 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6cnq A 2.151 BS02 dna C 0 R166 K167 S168 L170 S171 K186 R19 K20 S21 L23 S24 K39 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6cnq B 2.151 BS01 dna E 0 R188 S189 K190 P191 R41 S42 K43 P44 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6cnq B 2.151 BS02 dna F 0 R166 K167 S168 L170 S171 D176 K186 R19 K20 S21 L23 S24 D29 K39 ? 0003677 remove_due_to_license_issue Q9UBB5 29567833 1 ~ 12 KRMDCPALPPGWKKEEVIRKSGLSAGKSDVYYFSPSGKKFRSKPQLARYLGNTVDLSSFDFRTGKMMP 6coj A 1.4 BS01 F8G B 1 W29 Y85 W28 Y84 4.1.99.- 0006707,0008203,0008410,0016829 remove_due_to_license_issue Q0S7P9 29581275 301 VSKRDKRISLDDAVGELRSGMTIGIGGWGSRRKPMALVRALLRSDVTDLTVVTYGGPDLGLLCSAGKVTKAYYGFVSLDSAPFYDPWFAKARTAGEIAVREMDAGMVKCGLEAAAARLPFLPIRAGLGSDVRRFWGDELRTVTSPYPDASGKSETLIAMPALNLDAALVHLNLGDKHGNAAYTGVDPYFDDLYCAAAEKRFVSVERVVETEELVKTVPLQNLILNRMMVDGVVEAPNGAHFTLAGDSYGRDEKFQRHYAESAKTPQAWQQFVATYLSGSEDDYQAAVKKFAEEQA 6coj B 1.4 BS01 F8G B 1 M33 F84 R92 M96 G97 A98 N99 L109 F112 T119 R120 R126 N131 R147 M28 F79 R87 M91 G92 A93 N94 L104 F107 T114 R115 R121 N126 R142 4.1.99.- 0006707,0008203,0016829 remove_due_to_license_issue Q0S7Q0 29581275 301 TEVTRAEYCAIACADIFSGAGEIMASPMATLPLIGARLARLTTEPDLLITDGEALIFADTPAVGAKAPIEGWMPFRKVFDVVASGRRHVVMGANQIDRHGNQNLSAFGPLQQPTRQMFGVRGAPGNTINHPTSYWVGKHTSRVFCDTVDIVSGVGYDQIDPENPAYRFHHLHRVVSNLGVFDFGGPDHTFRALSLHPGVTADQVADNTSFEVAGLADAGVTREPTDEELRLIREVLDPRSLRDREVSV 6cpa A 2.0 BS02 ZAF A 1 H69 E72 R127 N144 R145 E163 H196 I243 Y248 A250 E270 H69 E72 R127 N144 R145 E163 H196 I243 Y248 A250 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=3pM remove_due_to_license_issue P00730 2386784 309 ARSTNTFNYATYHTLDEIYDFMDLLVAQHPELVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 6cpw A 1.85 BS01 F8V A 1 I29 A33 Y34 A50 K52 Y62 T66 E69 D104 M106 E107 T108 L154 D165 I12 A16 Y17 A28 K30 Y40 T44 E47 D82 M84 E85 T86 L132 D143 D147 K149 N152 D165 T188 D125 K127 N130 D143 T166 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 ic50=5.6nM remove_due_to_license_issue P63086 29748051 403 VFDVRYTNLSYIGEGAYGMVCSAYDRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFLDDLPKEKLKELIFEETARFQPG 6cq0 A 3.19 BS01 F8M A 1 L15 A36 F88 C89 P90 M142 L16 A37 F79 C80 P81 M133 D135 K137 N140 D157 T176 D126 K128 N131 D148 T153 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=3760nM Q9UHD2 30270002 801 AMQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFGAGTEEYLHPDMYEDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVELGEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 6cq1 A 1.69921 BS01 F8J A 1 M51 A52 C53 G55 Y58 E115 M46 A47 C48 G50 Y53 E110 ? Kd=219uM remove_due_to_license_issue IC50=142000nM, Kd=219000nM P41182 29969259 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6cq1 A 1.69921 BS02 F8J B 1 D17 N21 D12 N16 ? Kd=219uM remove_due_to_license_issue IC50=142000nM, Kd=219000nM P41182 29969259 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6cq1 B 1.69921 BS01 F8J A 1 N21 L25 N16 L20 ? Kd=219uM remove_due_to_license_issue IC50=142000nM, Kd=219000nM P41182 29969259 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6cq1 B 1.69921 BS02 F8J B 1 M51 A52 C53 G55 Y58 E115 M46 A47 C48 G50 Y53 E110 ? Kd=219uM remove_due_to_license_issue IC50=142000nM, Kd=219000nM P41182 29969259 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6cq4 A 3.2 BS01 F8P A 1 L15 A36 M86 F88 C89 P90 M142 T156 L16 A37 M79 F81 C82 P83 M135 T149 D135 K137 N140 D157 T176 D128 K130 N133 D150 T153 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=370nM Q9UHD2 30270002 801 AMQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFNNVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFGTEEYLHPDMYEDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVELGEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 6cq5 A 3.354 BS01 F8S A 1 L15 A36 F88 C89 P90 M142 T156 L16 A37 F81 C82 P83 M135 T149 D135 K137 N140 D157 D128 K130 N133 D150 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0035175,0035402,0035403,0035979,0042802,0043123,0043231,0044022,0044023,0044024,0044025,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0061470,0072354,0072371,0072518,0106310,0140374,0140823,0140855,0140857,0140896,1902554,1904262,1904263,1904417,1904515,1990244 remove_due_to_license_issue IC50=830nM Q9UHD2 30270002 801 AMQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFNNVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRDIKPGNIMRVIGEDGQSVYKLTDFEEYLHPDMYEDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVELGEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET 6cqf A 2.246 BS01 F97 A 1 L23 G24 A44 M91 F93 C94 G95 G97 D101 L144 L18 G19 A39 M86 F88 C89 G90 G92 D96 L139 D137 K139 A141 N142 D155 T175 D132 K134 A136 N137 D150 T164 2.7.11.1 0004672,0005524,0006468 ic50=0.0045uM remove_due_to_license_issue Q92918 30503777 301 PDIFNRDPRDHYDLLQRLGGGTYGEVFKARDKVSGDLVALKMVKMEPDDDVSTLQKEILILKTCRHANIVAYHGSYLWLQKLWICMEFCGAGSLQDIYQVTGSLSELQISYVCREVLQGLAYLHSQKKIHRDIKGANILINDAGEVRLADFGISAQIRLAFIGTPYWMAPEVAAVALKGGYNELCDIWSLGITAIELAELQPPLFDVHPLRVLFLMTKSGYQPPRLKEKGKWSAAFHNFIKVTLTKSPKKRPSATKMLSHQLVSQPGLNRGLILDLLDKLKN 6cqt A 2.273 BS01 VX A 1 G121 G122 S203 A204 W236 F297 H447 G119 G120 S201 A202 W234 F290 H440 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G119 G120 G152 S201 A202 G240 F290 F292 E327 H440 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P22303 30462502 607 REDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSA 6cqz A 2.216 BS01 VX A 1 G121 G122 S203 A204 W236 F297 G119 G120 S201 A202 W234 F292 G121 G122 G154 S203 A204 G242 F297 F299 E334 H447 G119 G120 G152 S201 A202 G240 F292 F294 E329 H442 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P22303 30462502 605 REDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPGGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSA 6crm A 2.19286 BS01 dna B 0 L74 I75 S97 E124 R125 W154 F158 R159 K222 P223 N244 S245 R246 K248 H267 A268 R275 T293 D312 R315 D344 W347 C351 K355 L70 I71 S93 E120 R121 W150 F154 R155 K218 P219 N240 S241 R242 K244 H263 A264 R271 T289 D308 R311 D340 W343 C347 K351 5.6.2.4 0003676,0003678,0004386,0005524,0006260,0006281,0006310,0009432,0043138 remove_due_to_license_issue A7MQK9 30305632 19 ~ 32 EVYSQETLAKQVLQETFGYQQFRPGQATIIDAVLEGRDCLVVMPTGGGKSLCYQIPALVKTGLTIVVSPLISLMKDQVDQLLANGVAAACLNSTQSREEQQAVLAGCRTGQVRLLYIAPERLMMDNFIDTLGYWDLAMVAVDEAHCISQWGHDFRPEYAALGQLRARFPAVPFMALTATADDTTRRDIVRLLGLDDPLIEISSFDRPNIRYMLMEKFKPLDQLMRYVQEQRGKSGIIYCNSRAKVEDTAARLQSRGISAAAYHAGLEHEVRASVQEKFQRDDLQIVVATVAFGMGINKPNVRFVVHFDIPRNIESYYQETGRAGRDGLPAEAMLFYDPADMAWLRRCLEEKAPGPLQDIERHKLNAMGAFAEAQTCRRLVLLNYFGEGRQAPCGNCDICLDPPRRYDGLVDAQKALSAIARVEQRFGMGYVVEVLRGANNQRIRELGHDKLKVYGIGRDQSQEHWVSVIRQLIHLGVVTQNIAQHSALQLTEAARPFLRGEAPLMLAVPRVA 6cse M 3.24 BS02 ALA M 1 A74 T75 G77 N80 Q170 F273 S274 E276 A57 T58 G60 N63 Q150 F253 S254 E256 ? 0003333,0005283,0005886,0006814,0006865,0015293,0016020,0035725,0055085 remove_due_to_license_issue Q6LX42 30659158 502 WGPYMLVLLLGTGIFLTLRLGFMQIHTLPYALKLAFSKETSEGDISHFQALMTALAATIGTGNIAGVATAYVLGGPGAIFWMWVTAFFGMATKYAEAVLAIKYRTVDDNGEMAGGPMYFLEKGLPLGKILGVAFAFFGAFAAFGIGNMVQTNSVADAVASNFGVDPLITGFVLAIFTAAVILGGIKSIGKATGIIVPFMAVFYILAGLVILAMNIGYIIPAFGTIFSSAFNFSAGFGALIGTAIMWGVKRGVFSNEAGLGSAPIAAAAAKTDHPGRQALVSMTGTFLDTIVVCTITGLVLTIAGLKAFPGLTDLTGASLTAASFDALMPMGGLIVTIGLVFFAYSTVLGWSYYGEKCFEYLIGTKGIRLYRIAFVLVAFWGATASLPLVWNIADTLNGAMAIPNLIGLLLLSGVVVSETKAFNEIRKNEAK 6csf M 3.3 BS02 DAL M 1 T75 G77 G79 N80 Q170 F273 S274 T58 G60 G62 N63 Q150 F253 S254 ? 0003333,0005283,0005886,0006814,0006865,0015293,0016020,0035725,0055085 remove_due_to_license_issue Q6LX42 30659158 502 WGPYMLVLLLGTGIFLTLRLGFMQIHTLPYALKLAFSKETSEGDISHFQALMTALAATIGTGNIAGVATAYVLGGPGAIFWMWVTAFFGMATKYAEAVLAIKYRTVDDNGEMAGGPMYFLEKGLPLGKILGVAFAFFGAFAAFGIGNMVQTNSVADAVASNFGVDPLITGFVLAIFTAAVILGGIKSIGKATGIIVPFMAVFYILAGLVILAMNIGYIIPAFGTIFSSAFNFSAGFGALIGTAIMWGVKRGVFSNEAGLGSAPIAAAAAKTDHPGRQALVSMTGTFLDTIVVCTITGLVLTIAGLKAFPGLTDLTGASLTAASFDALMPMGGLIVTIGLVFFAYSTVLGWSYYGEKCFEYLIGTKGIRLYRIAFVLVAFWGATASLPLVWNIADTLNGAMAIPNLIGLLLLSGVVVSETKAFNEIRKNEAK 6csp A 1.237 BS02 FBM A 1 H573 H574 G582 F583 D612 H614 F643 L712 Y745 H131 H132 G140 F141 D170 H172 F201 L270 Y303 ? Kd=3nM remove_due_to_license_issue F8W4B7 29775292 807 ITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6csq A 2.031 BS02 F9P A 1 H573 H574 G582 F583 D612 H614 F643 Y745 H131 H132 G140 F141 D170 H172 F201 Y303 ? Kd=410nM remove_due_to_license_issue F8W4B7 29775292 804 ITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6csr A 1.619 BS02 BHO A 1 H573 H574 G582 F583 D612 H614 F643 Y745 H132 H133 G141 F142 D171 H173 F202 Y304 ? Kd=144nM remove_due_to_license_issue F8W4B7 29775292 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6css A 1.7 BS02 FBJ A 1 H573 H574 G582 F583 D612 H614 F643 Y745 H132 H133 G141 F142 D171 H173 F202 Y304 ? Kd=25nM remove_due_to_license_issue F8W4B7 29775292 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6cus A -1.00 BS01 IHP A 1 K6 K13 K23 K24 K6 K13 K23 K24 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- remove_due_to_license_issue P03354 30309983 101 SEAVIKVISSACKTYCGKTSPSKKEIGAMLSLLQKEGLLMSPSDLYSPGSWDPITAALSQRAMILGKSGELKTWGLVLGALKAAREE 6cv8 A -1.00 BS01 I3P A 1 K6 S9 K23 K24 K6 S9 K23 K24 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- remove_due_to_license_issue P03354 30309983 101 SEAVIKVISSACKTYCGKTSPSKKEIGAMLSLLQKEGLLMSPSDLYSPGSWDPITAALSQRAMILGKSGELKTWGLVLGALKAAREE 6cvd A 1.78 BS01 4ME A 1 F365 D366 V403 K406 F171 D172 V209 K212 3.6.5.4 0005525,0006614,0016887 Kd~100uM remove_due_to_license_issue P10121 30044812 501 GFARLKRSLLKTKENLGSGFISLFRGKKIDDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFARE 6cvd A 1.78 BS02 4ME A 2 T307 T308 G311 W343 T113 T114 G117 W149 3.6.5.4 0005525,0006614,0016887 Kd~100uM remove_due_to_license_issue P10121 30044812 502 GFARLKRSLLKTKENLGSGFISLFRGKKIDDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFARE 6cve A 2.2 BS01 CTP A 1 T11 G12 V13 G14 K15 T16 V17 E108 G111 G169 P197 G199 A200 A201 T12 G13 V14 G15 K16 T17 V18 E109 G112 G170 P198 G200 A201 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6cvf A 2.3 BS01 CDP A 1 G12 V13 G14 K15 T16 V17 G169 L196 G199 A200 A201 G13 V14 G15 K16 T17 V18 G170 L197 G200 A201 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6cvf B 2.3 BS01 CDP B 1 G12 V13 G14 K15 T16 V17 G169 L196 P197 G199 A201 G13 V14 G15 K16 T17 V18 G170 L197 P198 G200 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6cvv A 2.41 BS01 ATP A 1 G12 G14 K15 T16 R45 D49 G13 G15 K16 T17 R46 D50 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6cvv B 2.41 BS01 ATP B 1 G12 G14 K15 T16 D49 G13 G15 K16 T17 D50 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6cvw A 1.78 BS02 FH1 A 1 Q1041 Y1056 H1057 V1078 D1081 R1123 L1135 K1136 G1137 S1139 F1154 R1155 A1156 A1157 D1168 Q61 Y76 H77 V98 D101 R143 L155 K156 G157 S159 F174 R175 A176 A177 D188 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 Ki=7.1nM remove_due_to_license_issue A0A0B4WYC6 30034602 1206 SHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTM 6cvx A 1.779 BS01 FH4 A 1 Q1041 Y1056 H1057 V1078 D1081 R1123 L1135 K1136 G1137 S1139 F1154 R1155 A1156 A1157 D1168 Q62 Y77 H78 V99 D102 R144 L156 K157 G158 S160 F175 R176 A177 A178 D189 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 Ki=21nM remove_due_to_license_issue A0A0B4WYC6 30034602 1201 GSHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTM 6cvy A 1.798 BS02 FHD A 1 Q1041 Y1056 H1057 V1078 D1081 R1123 L1135 K1136 G1137 S1139 F1154 R1155 A1156 A1157 D1168 Q61 Y76 H77 V98 D101 R143 L155 K156 G157 S159 F174 R175 A176 A177 D188 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0043657,0044423,0046718,0046872,0055036 Ki=3.9nM remove_due_to_license_issue A0A0B4WYC6 30034602 1205 SHMASMKKKGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTMR 6cw4 A -1.00 BS01 FGV A 1 K6 K13 K23 K24 K6 K13 K23 K24 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.26.4,3.4.23.- remove_due_to_license_issue P03354 30309983 101 SEAVIKVISSACKTYCGKTSPSKKEIGAMLSLLQKEGLLMSPSDLYSPGSWDPITAALSQRAMILGKSGELKTWGLVLGALKAAREE 6cw8 A 1.9 BS02 FGY A 1 H463 P464 N530 S531 H574 G582 F583 H614 F643 D705 Y745 H22 P23 N89 S90 H133 G141 F142 H173 F202 D264 Y304 ? remove_due_to_license_issue F8W4B7 30365892 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSL 6cwf A 2.25 BS01 6LA A 1 R61 M107 Q108 G109 K110 E127 K130 W151 R34 M80 Q81 G82 K83 E100 K103 W124 ? Kd=29nM remove_due_to_license_issue C1JZ07 30087354 201 AKTTQEKFDALKEAGVFSGYPGTTDAKLGQDMTRAEFAKVLVKLFGLKEIHGQYSYKDKNYDAKNWAAPFIEAVTAEGLMQGKDLTKKIFDFNGKITVEEASKTLVTALKLEPVKDAQNKATDWAKGYFEAAVNAGLFSKDANPKANATRAQLVEAAFAADEMSK 6cwh A 2.0 BS01 6LA A 1 R61 M107 Q108 G109 K110 E127 K130 W151 R34 M80 Q81 G82 K83 E100 K103 W124 ? Kd=29nM remove_due_to_license_issue C1JZ07 30087354 201 AKTTQEKFDALKEAGVFSGYPGTTDAKLGQDMTRAEFAKVLVKLFGLKEIHGQYSYKDKNYDAKNWAAPFIEAVTAEGLMQGKDLTKKIFDFNGKITVEEASKTLVTALKLEPVKDAQNKATDWAKGYFEAAVNAGLFSKDANPKANATRAQLVEAAFAADEMSK 6cwi A 2.16 BS01 6LA A 1 R61 M107 Q108 G109 K110 L112 E127 K130 W151 R34 M80 Q81 G82 K83 L85 E100 K103 W124 ? Kd=29nM remove_due_to_license_issue C1JZ07 30087354 201 AKTTQEKFDALKEAGVFSGYPGTTDAKLGQDMTRAEFAKVLVKLFGLKEIHGQYSYKDKNYDAKNWAAPFIEAVTAEGLMQGKDLTKKIFDFNGKITVEEASKTLVTALKLEPVKDAQNKATDWAKGYFEAAVNAGLFSKDANPKANATRAQLVEAAFAADEMSK 6cwi A 2.16 BS02 6LA A 2 F44 S45 G46 P48 E63 R177 F17 S18 G19 P21 E36 R150 ? Kd=29nM remove_due_to_license_issue C1JZ07 30087354 202 AKTTQEKFDALKEAGVFSGYPGTTDAKLGQDMTRAEFAKVLVKLFGLKEIHGQYSYKDKNYDAKNWAAPFIEAVTAEGLMQGKDLTKKIFDFNGKITVEEASKTLVTALKLEPVKDAQNKATDWAKGYFEAAVNAGLFSKDANPKANATRAQLVEAAFAADEMSK 6cwn A 1.53 BS01 6LA A 1 F44 S45 G46 Y47 P48 E63 K66 W93 R177 F17 S18 G19 Y20 P21 E36 K39 W66 R150 ? Kd=226nM remove_due_to_license_issue C1JZ07 30087354 301 AKTTQEKFDALKEAGVFSGYPGTTDAKLGQDMTRAEFAKVLVKLFGLKEIHGQYSYKDKNYDAKNWAAPFIEAVTAEGLMQAKDLTKKIFDFNGKITVEEASKTLVTALKLEPVKDAQNKATDWAKGYFEAAVNAGLFSKDANPKANATRAQLVEAAFAADEM 6cyb A 1.62 BS02 FKV A 1 Y655 H656 L770 D808 L809 Q812 I826 Q859 F862 Y82 H83 L197 D235 L236 Q239 I253 Q286 F289 3.1.4.17 0004114,0007165,0008081 ic50=0.96nM remove_due_to_license_issue O00408 30128073 1008 SLYKKAGFYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6cyc A 1.54 BS02 FKJ A 1 Y655 H656 L770 T805 D808 L809 Q812 I826 Q859 F862 Y82 H83 L197 T232 D235 L236 Q239 I253 Q286 F289 3.1.4.17 0004114,0007165,0008081 ic50=14nM remove_due_to_license_issue O00408 30128073 1003 SLYKKAGFYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6cyd A 1.69 BS02 FKG A 1 L770 D808 L809 Q812 I826 Q859 F862 L197 D235 L236 Q239 I253 Q286 F289 3.1.4.17 0004114,0007165,0008081 ic50=2nM remove_due_to_license_issue O00408 30128073 1003 SLYKKAGFYTKLLHDGIQPVAAIDSNFASFTYTPRSLPEDDTSMAILSMLQDMNFINNYKIDCPTLARFCLMVKKGYRDPPYHNWMHAFSVSHFCYLLYKNLELTNYLEDIEIFALFISCMCHDLDHRGTNNSFQVASKSVLAALYSSEGSVMERHHFAQAIAILNTHGCNIFDHFSRKDYQRMLDLMRDIILATDLAHHLRIFKDLQKMAEVGYDRNNKQHHRLLLCLLMTSCDLSDQTKGWKTTRKIAELIYKEFFSQGDLEKAMGNRPMEMMDREKAYIPELQISFMEHIAMPIYKLLQDLFPKAAELYERVASNREHWTKVSHKFTIRGLPSNNSLDFL 6cyg A 1.50392 BS01 N5O A 1 A55 M98 N106 G135 V136 Y139 A40 M83 N91 G120 V121 Y124 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=68uM remove_due_to_license_issue P07900 31501246 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 6cyh A 1.49 BS01 N5A A 1 A55 M98 N106 T109 S113 Y139 A40 M83 N91 T94 S98 Y124 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=708uM remove_due_to_license_issue P07900 31501246 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 6cyi A 1.75658 BS01 N5O A 1 A111 M154 N162 V197 Y200 A39 M82 N90 V125 Y128 ? 0005524,0006457,0016887,0051082,0140662 Kd=9.1uM remove_due_to_license_issue P41148 31501246 404 SEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTEAQEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTETKVEKTVWDWELMN 6cz3 A 1.8 BS01 FLJ A 1 R195 L197 K219 L248 L266 M267 A268 G270 L319 D330 R14 L16 K38 L67 L85 M86 A87 G89 L138 D149 D312 R316 N317 D330 D131 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.056uM remove_due_to_license_issue IC50=70nM Q13882 29879184 9001 DDAERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRDSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHDHNIPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPCFKALRERLSS 6cz4 A 1.5 BS01 FKY A 1 L197 A217 M239 L248 T264 L266 M267 G270 H310 L319 V328 G329 D330 F331 L15 A35 M57 L66 T82 L84 M85 G88 H128 L137 V146 G147 D148 F149 D312 R316 N317 D330 D130 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.076uM remove_due_to_license_issue Q13882 29879184 9001 DAERPREEFTLCRKLGSGYFGEVFEGLWKDRVQVAIKVISRDNLLHQQMLQSEIQAMKKLRHKHILALYAVVSVGDPVYIITELMAKGSLLELLRDSDEKVLPVSELLDIAWQVAEGMCYLESQNYIHRDLAARNILVGENTLCKVGDFGLARLIKEDVYLSHPYKWTAPEALSRGHYSTKSDVWSFGILLHEMFSRGQVPYPGMSNHEAFLRVDAGYRMPCPLECPPSVHKLMLTCWCRDPEQRPCFKALRERLSS 6czb A 2.4 BS02 UTP A 1 T11 G12 V13 G14 K15 T16 V17 E108 T12 G13 V14 G15 K16 T17 V18 E109 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6czb B 2.4 BS02 UTP B 1 G12 V13 G14 K15 T16 E108 G111 G13 V14 G15 K16 T17 E109 G112 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6czc A 2.3 BS02 TTP A 1 T11 G12 G14 K15 T16 K37 D49 E52 E108 G111 T12 G13 G15 K16 T17 K38 D50 E53 E109 G112 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6czc B 2.3 BS02 TTP B 1 G12 G14 K15 T16 V17 D49 E108 G111 G13 G15 K16 T17 V18 D50 E109 G112 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6czd A 2.4 BS02 ADP A 1 T11 G12 V13 G14 K15 T16 M72 A73 E108 A110 G111 T12 G13 V14 G15 K16 T17 M73 A74 E109 A111 G112 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 30289406 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6czd B 2.4 BS02 ADP B 1 T11 G12 G14 K15 T16 M72 A73 E108 G111 T12 G13 G15 K16 T17 M73 A74 E109 G112 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 30289406 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6cze A 2.3 BS01 ITT A 1 G12 V13 G14 K15 T16 E108 G14 V15 G16 K17 T18 E110 T11 G12 K15 T16 K37 T41 G54 E108 T13 G14 K17 T18 K39 T43 G56 E110 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 HGGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6cze B 2.3 BS01 ITT B 1 G12 V13 G14 K15 T16 E108 G13 V14 G15 K16 T17 E109 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6czf A 1.949 BS01 G4P A 1 R45 K46 N48 R62 A82 S83 E84 R45 K46 N48 R62 A82 S83 E84 C1 G27 N101 G102 Y258 R321 K326 M336 D444 C1 G27 N101 G102 Y258 R321 K326 M336 D444 2.4.2.14 0000287,0004044,0005737,0005829,0006164,0006189,0006541,0009113,0016757,0042802,0046872,0097216 Kd=1.6uM remove_due_to_license_issue P0AG16 30559427 502 CGIVGIAGVMPVNQSIYDALTVLQHRGQDAAGIITIDANNCFRLRKANGLVSDVFEARHMQRLQGNMGIGHVRYPTAGSSSASEAQPFYVNSPYGITLAHNGNLTNAHELRKKLFEEKRRHINTTSDSEILLNIFASELDNFRHYPLEADNIFAAIAATNRLIRGAYACVAMIIGHGMVAFRDPNGIRPLVLGKRDIDENRTEYMVASESVALDTLGFDFLRDVAPGEAIYITEEGQLFTRQCADNPVSNPCLFEYVYFARPDSFIDKISVYSARVNMGTKLGEKIAREWEDLDIDVVIPIPETSCDIALEIARILGKPYRQGFVKNRYVGRTFIMPGQQLRRKSVRRKLNANRAEFRDKNVLLVDDSIVRGTTSEQIIEMAREAGAKKVYLASAAPEIRFPNVYGIDMPSATELIAHGREVDEIRQIIGADGLIFQDLNDLIDAVRAENPDIQQFECSVFNGVYVTKDVDQGYLDFLDTLRNDDAKAVQRQNEVENL 6czf C 1.949 BS01 G4P A 1 R45 R58 R62 R45 R58 R62 C1 G27 N101 G102 Y258 R321 K326 M336 D444 C1 G27 N101 G102 Y258 R321 K326 M336 D444 2.4.2.14 0000287,0004044,0005737,0005829,0006164,0006189,0006541,0009113,0016757,0042802,0046872,0097216 remove_due_to_license_issue P0AG16 30559427 502 CGIVGIAGVMPVNQSIYDALTVLQHRGQDAAGIITIDANNCFRLRKANGLVSDVFEARHMQRLQGNMGIGHVRYPTAGSSSASEAQPFYVNSPYGITLAHNGNLTNAHELRKKLFEEKRRHINTTSDSEILLNIFASELDNFRHYPLEADNIFAAIAATNRLIRGAYACVAMIIGHGMVAFRDPNGIRPLVLGKRDIDENRTEYMVASESVALDTLGFDFLRDVAPGEAIYITEEGQLFTRQCADNPVSNPCLFEYVYFARPDSFIDKISVYSARVNMGTKLGEKIAREWEDLDIDVVIPIPETSCDIALEIARILGKPYRQGFVKNRYVGRTFIMPGQQLRRKSVRRKLNANRAEFRDKNVLLVDDSIVRGTTSEQIIEMAREAGAKKVYLASAAPEIRFPNVYGIDMPSATELIAHGREVDEIRQIIGADGLIFQDLNDLIDAVRAENPDIQQFECSVFNGVYVTKDVDQGYLDFLDTLRNDDAKAVQRQNEVENL 6czi A 2.3 BS01 38E A 1 V14 M16 N18 S24 Q25 G26 W28 I46 I52 Y72 L104 V13 M15 N17 S23 Q24 G25 W27 I45 I51 Y71 L103 Kd=0.56uM remove_due_to_license_issue 30209393 201 SRAAQLLPGTWQVTMTNEDGQTSQGQWHFQPRSPYTLDIVAQGTISDGRPITGYGKATVKTDDTLHANLTYPSLGNIKAQGQITYDSPTQFTWNSTTSDGKKLTGTLQR 6czu A 1.47 BS01 FP7 A 1 W81 P82 L92 N140 D145 M149 W40 P41 L51 N99 D104 M108 ? remove_due_to_license_issue O60885 30165024 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEETE 6czv A 1.88 BS01 FOY A 1 W81 P82 F83 N140 I146 M149 W40 P41 F42 N99 I105 M108 ? ic50=0.23uM remove_due_to_license_issue IC50=80nM O60885 30165024 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 6d12 A 2.205 BS01 rna C 0 P449 R468 R472 Y483 V484 D485 R496 Y532 I536 D539 R540 K543 P4 R23 R27 Y38 V39 D40 R51 Y87 I91 D94 R95 K98 ? 0003676,0003723 remove_due_to_license_issue Q4G0J3 29946027 303 ~ 340 ATGPQFVSGVIVKIISTEPLPGRKQVRDTMAAISEVLYVDLLEGDTECHARFKTPLDALAVINAYTEINKKHCWKMEILSGDHEQRYWQKILVDRQAKLN 6d12 B 2.205 BS01 rna C 0 P449 R468 R472 L482 Y483 V484 D485 R496 Y532 I536 D539 R540 K543 L544 R548 P4 R23 R27 L37 Y38 V39 D40 R51 Y87 I91 D94 R95 K98 L99 R103 ? 0003676,0003723 remove_due_to_license_issue Q4G0J3 29946027 303 ~ 340 ATGPQFVSGVIVKIISTEPLPGRKQVRDTMAAISEVLYVDLLEGDTECHARFKTPLDALAVINAYTEINKKHCWKMEILSGDHEQRYWQKILVDRQAKLNQPR 6d15 A 1.3 BS01 TWB A 1 S70 S130 T235 G236 T237 S47 S107 T212 G213 T214 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=32.9uM remove_due_to_license_issue Q9F663 31483651 301 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d15 A 1.3 BS02 TWB A 2 R83 G147 A150 F151 S154 R60 G124 A127 F128 S131 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=32.9uM remove_due_to_license_issue Q9F663 31483651 302 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d16 A 1.4 BS01 FUJ A 1 S70 W105 S130 T235 G236 T237 S47 W82 S107 T212 G213 T214 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=8.4uM remove_due_to_license_issue Q9F663 31483651 301 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d17 A 1.45 BS01 VKE A 1 S70 W105 S130 N132 T235 G236 T237 S47 W82 S107 N109 T212 G213 T214 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=15.3uM remove_due_to_license_issue Q9F663 31483651 301 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d18 A 1.35 BS01 GTV A 1 S70 W105 S130 T235 G236 T237 S47 W82 S107 T212 G213 T214 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.4uM remove_due_to_license_issue Q9F663 31483651 301 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d18 A 1.35 BS02 GTV A 2 N136 W165 N113 W142 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.4uM remove_due_to_license_issue Q9F663 31483651 302 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d18 A 1.35 BS03 GTV A 3 R83 L142 G147 A150 F151 R60 L119 G124 A127 F128 S70 K73 S130 E166 K234 T237 S47 K50 S107 E143 K211 T214 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=1.4uM remove_due_to_license_issue Q9F663 31483651 303 HMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d19 A 1.45 BS01 YKG A 1 S70 W105 S130 T235 G236 T237 S46 W81 S106 T211 G212 T213 S70 K73 S130 E166 K234 T237 S46 K49 S106 E142 K210 T213 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.246uM remove_due_to_license_issue Q9F663 31483651 301 MLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d19 A 1.45 BS02 YKG A 2 R83 G147 A150 F151 R59 G123 A126 F127 S70 K73 S130 E166 K234 T237 S46 K49 S106 E142 K210 T213 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=0.246uM remove_due_to_license_issue Q9F663 31483651 303 MLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6d1a A 1.25 BS03 TWB A 1 M67 F70 H122 D124 H189 N220 M26 F29 H81 D83 H148 N179 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=44.3uM remove_due_to_license_issue C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1b A 1.25 BS03 FUJ A 1 F70 H122 D124 H189 N220 H250 F29 H81 D83 H148 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=123.7uM remove_due_to_license_issue C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1d A 1.4 BS03 GTV A 1 H122 D124 H189 C208 N220 H81 D83 H148 C167 N179 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=33.8uM remove_due_to_license_issue Ki=100000nM C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1g A 1.15 BS03 YKG A 1 M67 V73 H122 D124 H189 C208 N220 H250 M26 V32 H81 D83 H148 C167 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=34.2uM remove_due_to_license_issue Ki=54970nM C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1h A 1.25 BS03 KED A 1 M67 H122 D124 H189 N220 H250 M26 H81 D83 H148 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=190.2uM remove_due_to_license_issue C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1i A 1.1 BS03 T6Z A 1 M67 H122 D124 H189 C208 N220 H250 M26 H81 D83 H148 C167 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=81uM remove_due_to_license_issue C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1k A 1.2 BS03 M3Q A 1 M67 F70 H122 D124 H189 C208 N220 H250 M26 F29 H81 D83 H148 C167 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=741.3uM remove_due_to_license_issue C7C422 31483651 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6d1l A 1.4 BS02 FQV A 1 H94 H96 H119 L198 T199 T200 P202 H93 H95 H118 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.6nM remove_due_to_license_issue Ki=7.6nM P00918 29803994 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6d1l A 1.4 BS03 FQV A 2 W5 N11 H15 W16 D19 W4 N10 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=7.6nM remove_due_to_license_issue Ki=7.6nM P00918 29803994 304 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6d1m A 1.21 BS02 FQY A 1 H94 H119 F131 L198 T199 T200 H93 H118 F129 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=6.3nM remove_due_to_license_issue Ki=6.3nM P00918 29803994 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6d1m A 1.21 BS03 FQY A 2 N11 H15 W16 D19 N10 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=6.3nM remove_due_to_license_issue Ki=6.3nM P00918 29803994 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6d1x A 2.3 BS01 PA7 A 1 A111 M154 N162 V197 Y200 A39 M82 N90 V125 Y128 ? 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P41148 31501246 401 SEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTEAQEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTEKTVWDWELMN 6d28 A 1.75 BS01 NEC A 1 A111 M154 N162 V197 Y200 A40 M83 N91 V126 Y129 ? 0005524,0006457,0016887,0051082,0140662 Kd=200nM remove_due_to_license_issue P41148 12970348 401 KSEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTEAQEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 6d2o A 1.9 BS02 4MZ A 1 C42 D44 H98 C101 G102 G103 C40 D42 H96 C99 G100 G101 C42 D44 R46 H98 C101 C40 D42 R44 H96 C99 4.2.1.1 0004089,0008270,0015976,0016829,0046872 Ki=5uM remove_due_to_license_issue Q9HVB9 30088334 302 ALQQLFENNVRWAEAIKQEDPDFFAKLARQQTPEYLWIGCSDARVPANEIVGMLPGDLFVHRNVANVVLHTDLNCLSVIQFAVDVLKVKHILVTGHYGCGGVRASLHNDQLGLIDGWLRSIRDLAYEYREHLEQLPTEEERVDRLCELNVIQQVANVSHTSIVQNAWHRGQSLSVHGCIYGIKDGLWKNLNVTVSGLDQLPPQYRLSPL 6d3g A 2.398 BS01 NXL A 1 S70 W105 S130 N132 T235 G236 T237 S47 W84 S111 N113 T216 G217 T218 S70 K73 S130 E166 K234 T237 S47 K50 S111 E147 K215 T218 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue A2RP81 31235626 401 SAQSPLLKEQIETIVTGKKATVGVAVWGPDDLEPLLLNPFEKFPMQSVFKLHLAMLVLHQVDQGKLDLNQSVTVNRAAVLQNTWSPMMKDHQGDEFTVAVQQLLQYSVSHSDNVACDLLFELVGGPQALHAYIQSLGVKEAAVVANEAQMHADDQVQYQNWTSMKAAAQVLQKFEQKKQLSETSQALLWKWMVETTTGPQRLKGLLPAGTIVAHKTGTSGVRAGKTAATNDAGVIMLPDGRPLLVAVFVKDSAESERTNEAIIAQVAQAAYQFELKKLS 6d49 A 1.801 BS01 FVP A 1 N20 F21 S68 F117 R119 K126 Y127 S128 K130 N4 F5 S52 F101 R103 K110 Y111 S112 K114 ? Kd=118uM remove_due_to_license_issue P20138 31369984 205 GDPNFWLQVQESVTVQEGLCVLVPCTFFHPIPYYDKNSPVHGYWFREGAIISRDSPVATNKLDQEVQEETQGRFRLLGDPSRNNCSLSIVDARRRDNGSYFFRMERGSTKYSYKSPQLSVHVTDLT 6d4a A 1.751 BS01 FVP A 1 F21 F117 R119 K126 Y127 S128 K130 F2 F98 R100 K107 Y108 S109 K111 ? Kd=118uM remove_due_to_license_issue P20138 31369984 203 NFWLQVQESVTVQEGLCVLVPCTFFHPIPYYDKNSPVHGYWFREGAIISRDSPVATNKLDQEVQEETQGRFRLLGDPSRNNCSLSIVDARRRDNGSYFFRMERGSTKYSYKSPQLSVHVTDLT 6d4o A 2.9 BS01 FUV A 1 M149 D172 H343 E425 Y481 Y485 F486 E516 W561 R574 N578 K580 M151 D163 H322 E404 Y460 Y464 F465 E495 W540 R553 N557 K559 3.2.1.31 0004553,0004565,0004566,0005975,0016798,0030246 remove_due_to_license_issue A0A174ZZA3 30062115 701 NAMLYPVLTQSRLLSDLSGVWNFKLDNGKGFEEKWYEKPLKDADTMPVPASYNDLKEGTDFRDHYGWVFYQRNISVPEYVKSQRIVLRCAAVTHYAMIYLNGKLICEHKGGFLPFEVELNDDLQDGDNLLTIAVNNVIDYTTLPVGGKANMMSGMPQNNPNFDFFNYCGITRPVKIYTTPETYINDITVTADIDFTKEEPSAVLNYNVEVELFDEEGTKLSETEGSEGTFEISNVRLWQPLNAYLYKIKVTAGQDVYTLPYGVRSVRVDGTKFLINEKPFYFKGYGKHEDTFPNGRGINLPMNTKDISIMKWQHANSFRTSHYPYSEEMMRLCDEEGIVVIDETTAVGVNLQFGGGANFGGERIGTFDKEHGVQTQEHHKDVIRDLISRDKNHACVVMWSIANEPDSAAEGAYDYFKPLYDLARELDPQKRPCTLVSVQGTTADTDCSSQLSDVICLNRYYGWYFGGPDLEVSETGLRKELSDWGKLGKPVMFTEYGADTVSGLHDTTSVMYTEEYQVEYYEMNNKVFDEFDFVVGEQAWNFADFATSQSLLRVQGNKKGLFTRDRKPKMVAHYFRNRWSAIPEFGYKT 6d4q A 1.71 BS02 FWG A 1 A145 T203 G285 E318 A131 T189 G271 E280 1.1.1.205 0003824,0003938,0006164,0016491 ic50=0.83uM remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAGL 6d4r A 1.34 BS02 FWY A 1 A145 T203 G285 E318 A131 T189 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 ic50=1.1uM remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAGL 6d4s A 1.63 BS02 FWV A 1 A145 H146 T203 G285 E318 A131 H132 T189 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 ic50=0.9uM remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 6d4t A 1.54 BS02 FWS A 1 A145 T203 G285 E318 A131 T189 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 ic50=0.12uM remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 6d4u A 1.7 BS02 FWP A 1 A145 H146 T203 G285 E318 A131 H132 T189 G271 E280 1.1.1.205 0003824,0003938,0006164,0016491 ic50=1.98uM remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 6d4v A 2.02 BS02 FWM A 1 A145 G285 E318 A131 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 ic50=0.23uM remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 6d4w A 1.8 BS02 FWJ A 1 A145 T203 G285 E318 A131 T189 G271 E281 1.1.1.205 0003824,0003938,0006164,0016491 remove_due_to_license_issue G7CNL4 31055147 402 VPTGGDDPTKIAMLGLTFDDVLLLPAASDVLPANADTSSQLTKKIRLKVPLVSSAMDTVTEARMAIAMARAGGMGVLHRNLPVAEQAAQVETVKRSGGLLVGAAVGVGDDAWERAMALRDAGVDVLVVDTAHAHNRKVLDMVHRLKTTVGDEIEVVGGNVATRAAAAALVEAGADAVKVGVGPGSICTTRVVAGVGAPQITAILEAVAACAPHGVPVIADGGLQYSGDIAKALAAGASTAMLGSLLAGTAESPGELILVNGKQFKSYRGMGSLGAMQLVPEGIEGRVPFRGPLSTVIHQLVGGLRAAMGYTGSATIEELQQAQFVQITAAG 6d50 A 2.5 BS02 GCB A 1 D166 H363 N425 E426 N493 Y495 Y499 E526 W573 N591 K593 D135 H332 N394 E395 N462 Y464 Y468 E495 W542 N560 K562 ? 0004553,0005975 remove_due_to_license_issue A0A078SUX9 30301767 903 QRQTQTINDSWKFLKGECTAAADSAFDDSKWTSIHLPHTWNTDAYTEKDYYRGTGWYRRQLTLPQGWKEKQIILRLDAAGKSATIYINGKNVGEHAGGYTACSFNITPFLSFDTPNTLAVCVDNARQDIAPISGDFTFFGGIYRDVWLTAVPNQHFNLTNHGSDGLFISTPQVSEEQATLSIRGEVKNDAPEKATLELTHTIYRPDGTLLQTLKKNIQLKAGETYAFSNEATPVLKPELWTPETPRLYRVETTLRNRKTKTLLDQSNHYTAFRWFRFDGDEGFFLNGKPYKLRGICRHQDQKPIGPALTDEMHRRDFLLMKEMGANFIRISHYPQDDALLEMCDKLGMLAWEEIPIIDIVPNTPGYGDNCERNLREMIRQHYNHPSIITWGYMNEILLVTQRKYKTEAELKPVLERTLALANRLERVLKEEDSTRISTMAFHGSNSYNETGLSKITDIVGWNLYQGWYGGDLTGFEKFLAQQHQNHPTHPMIVSEYGAGSDKRLHSLHPRAFDFSIEYQQKYLEHYLPVLEDTPYICGGTHWNFIDFSSALRDESMPRINNKGLVYADRTPKDVYHYYQAAWRKDIPVLHIASRDWTDRAGVQQGNAPVYLPVKIYTNLSEVELFIDGISLGKQKTENYTATFEVPFSNRNPFLFAQGNYQGKTVQDGLRINFTPIPACLDANNLKGLELAVNVGSQCFFTSDESQLTWLPDQPYAAGSWGYIGGKEGTAQTEIQNTADGPLFQTLRNEIEGYRFDAPQGVYEIELLFTDIFRESTFGISINGEVVEESLSPCKESGYFRALRKKYYITNDKEYIDIRFHSTSGTCFLNGIKLRNIY 6d55 B 1.68 BS01 FWA B 1 V875 M878 N879 V883 Y884 D887 F890 L901 E902 H905 V298 M301 N302 V306 Y307 D310 F313 L324 E325 H328 ? 0005085,0007264 remove_due_to_license_issue EC50=5900nM, Kd=44nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d56 B 1.68 BS01 FVM B 1 V875 M878 N879 V883 Y884 L886 D887 F890 L901 E902 H905 V298 M301 N302 V306 Y307 L309 D310 F313 L324 E325 H328 ? 0005085,0007264 remove_due_to_license_issue EC50=21100nM, Kd=9.0nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d59 B 1.7 BS01 FVJ B 1 M878 N879 V883 Y884 D887 F890 L901 E902 H905 M301 N302 V306 Y307 D310 F313 L324 E325 H328 ? 0005085,0007264 remove_due_to_license_issue Kd=<100nM, EC50=15600nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d5e B 1.75 BS01 FVG B 1 M878 N879 V883 Y884 D887 F890 L901 H905 M301 N302 V306 Y307 D310 F313 L324 H328 ? 0005085,0007264 remove_due_to_license_issue Kd=140nM, EC50=3200nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d5g B 1.92 BS01 FVD B 1 M878 N879 V883 Y884 D887 F890 L901 E902 H905 M301 N302 V306 Y307 D310 F313 L324 E325 H328 ? 0005085,0007264 remove_due_to_license_issue Kd=250nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d5h B 1.8 BS01 FV7 B 1 M878 N879 V883 Y884 D887 F890 L901 E902 M301 N302 V306 Y307 D310 F313 L324 E325 ? 0005085,0007264 remove_due_to_license_issue EC50=11000nM, Kd=120nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d5j B 1.751 BS01 FV4 B 1 M878 N879 V883 Y884 D887 F890 L901 H905 M301 N302 V306 Y307 D310 F313 L324 H328 ? 0005085,0007264 remove_due_to_license_issue EC50=14500nM, Kd=460nM Q07889 30205005 2001 GQMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIANITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d5w S 2.478 BS01 FVV S 1 V852 V883 Y884 F890 L901 V275 V306 Y307 F313 L324 ? 0005085,0007264 remove_due_to_license_issue EC50=63000nM Q07889 30205005 1101 QMRLPSADVYRFAEPDSEENIIFEEGIPIIKAGTVIKLIERLTYHMYADPNFVRTFLTTYRSFCKPQELLSLIIERFEIPEPEPTEADRIAIENGDQPLSAELKRFRKEYIQPVQLRVLNVCRHWVEHHFYDFERDAYLLQRMEEFIGTVRGKAMKKWVESITKIIQRKKIAHNITFQSSPPTVEWHISRPGHIETFDLLTLHPIEIARQLTLLESDLYRAVQPSELVGSVWTKEDKEINSPNLLKMIRHTTNLTLWFEKCIVETENLEERVAVVSRIIEILQVFQELNNFNGVLEVVSAMNSSPVYRLDHTFEQIPSRQKKILEEAHELSEDHYKKYLAKLRSINPPCVPFFGIYLTNILKTEEGNPEVLKRHGKELINFSKRRKVAEITGEIQQYQNQPYCLRVESDIKRFFENLNPMGNSMEKEFTDYLFNKSLEIEPRNPKPLPRFPKKYSYPLKSPGVRPSNPR 6d6t D 3.86 BS02 FYP D 1 H102 Y160 S205 Y210 H92 Y150 S195 Y200 ? 0004888,0004890,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=0.80nM P14867 29950725 406 NTTVFTRILDRLLDGYDNRLRPGLGERVTEVKTDIFVTSFGPVSDHDMEYTIDVFFRQSWKDERLKFKGPMTVLRLNNLMASKIWTPDTFFHNGKKSVAHNMTMPNKLLRITEDGTLLYTMRLTVRAECPMHLEDFPMDAHACPLKFGSYAYTRAEVVYEWTREPARSVVVAEDGSRLNQYDLLGQTVDSGIVQSSTGEYVVMTTHFHLKRKIGYFVIQTYLPCIMTVILSQVSFWLNRESVPARTVFGVTTVLTMTTLSISARNSLPKVAYATAMDWFIAVCYAFVFSALIEFATVNYFTKSQPARAAKIDRLSRIAFPLLFGIFNLVYWATYLNR 6d6t E 3.86 BS01 FYP D 1 Y58 F77 T142 Y34 F53 T118 ? 0004888,0004890,0005216,0005230,0006811,0006821,0007214,0016020,0034220 remove_due_to_license_issue P18507 29950725 406 GDVTVILNNLLEGYDNKLRPDIGVKPTLIHTDMYVNSIGPVNAINMEYTIDIFFAQTWYDRRLKFNSTIKVLRLNSNMVGKIWIPDTFFRNSKKADAHWITTPNRMLRIWNDGRVLYTLRLTIDAECQLQLHNDEHSCPLEFSSYGYPREEIVYQWKRSSVEVGDTRSWRLYQFSFVGLRNTTEVVKTTSGDYVVMSVYFDLSRRMGYFTIQTYIPCTLIVVLSWVSFWINKDAVPARTSLGITTVLTMTTLSTIARKSLAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAAA 6d6u D 3.92 BS03 FYP D 1 Y160 S205 S206 Y210 Y151 S196 S197 Y201 ? 0004888,0004890,0005216,0005230,0006811,0016020,0034220 remove_due_to_license_issue Ki=0.80nM P14867 29950725 410 DNTTVFTRILDRLLDGYDNRLRPGLGERVTEVKTDIFVTSFGPVSDHDMEYTIDVFFRQSWKDERLKFKGPMTVLRLNNLMASKIWTPDTFFHNGKKSVAHNMTMPNKLLRITEDGTLLYTMRLTVRAECPMHLEDFPMDAHACPLKFGSYAYTRAEVVYEWTREPARSVVVAEDGSRLNQYDLLGQTVDSGIVQSSTGEYVVMTTHFHLKRKIGYFVIQTYLPCIMTVILSQVSFWLNRESVPARTVFGVTTVLTMTTLSISARNSLPKVAYATAMDWFIAVCYAFVFSALIEFATVNYFTKSQPARAAKIDRLSRIAFPLLFGIFNLVYWATYLNR 6d6u E 3.92 BS02 FYP D 1 Y58 T142 Y34 T118 ? 0004888,0004890,0005216,0005230,0006811,0006821,0007214,0016020,0034220 remove_due_to_license_issue P18507 29950725 410 GDVTVILNNLLEGYDNKLRPDIGVKPTLIHTDMYVNSIGPVNAINMEYTIDIFFAQTWYDRRLKFNSTIKVLRLNSNMVGKIWIPDTFFRNSKKADAHWITTPNRMLRIWNDGRVLYTLRLTIDAECQLQLHNFPMDEHSCPLEFSSYGYPREEIVYQWKRSSVEVGDTRSWRLYQFSFVGLRNTTEVVKTTSGDYVVMSVYFDLSRRTIQTYIPCTLIVVLSWVSFWINKDAVPARTSLGITTVLTMTTLSTIARKSYVTAMDLFVSVCFIFVFSALVEYGTLHYFVSSQPARAAKMDSYARIFFPTAFCLFNLVYWVSYL 6d8e A 2.537 BS01 FZP A 1 L718 A743 K745 L788 I789 T790 M793 G796 C797 R841 L844 L23 A48 K50 L89 I90 T91 M94 G97 C98 R142 L145 D837 A839 R841 N842 D855 D138 A140 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 29978938 1101 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEYHAEKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDMHLPSLMDEEDMDDVVDADEYLIP 6d8v A 2.8 BS01 PBE A 1 W109 Y139 F153 W161 Y177 A179 E180 G181 D208 W72 Y102 F116 W124 Y140 A142 E143 G144 D171 ? remove_due_to_license_issue Q92SH9 30442721 402 DRVETLVFDGAKTEARAIASDIAGSVGELAAAARTMSGVLGRGHAGQSTDRAGAINLLKANLEQHGFAFGSWFAEEPKAYDGKDVIDNTERGGNADGAFTPYWSKDRNGNIQLSTFKADYAAEWYGLAAKSGKGAITQPYLAEGTDVPTTMTSIAYPVMSNGRMIGVSGVDISLAALADRLSAVKPFGSGRVYLLSQSGKWLAAPIPELLMKEYDGEGVESVKDALSTGTPRMIENLTYDGNEPFDRVVYPFSLPDVNAQWLVLVDVPR 6d9s A 2.105 BS01 G4P A 1 K43 G44 I101 D103 S104 G105 K131 F152 V153 L158 D159 R165 K44 G45 I102 D104 S105 G106 K132 F153 V154 L159 D160 R166 E99 D100 D103 F152 R165 E100 D101 D104 F153 R166 2.4.2.8 0000166,0000287,0004422,0005737,0005829,0006166,0006178,0016757,0032263,0032264,0046100,0046872,0052657 remove_due_to_license_issue B9ZW32 31552824 201 AMMNQDIEKVLISEEQIQEKVLELGAIIAEDYKNTVPLAIGVLKGAMPFMADLLKRTDTYLEMDFMAVSSYGHSTVSTGEVKILKDLDTSVEGRDILIVEDIIDSGLTLSYLVDLFKYRKAKSVKIVTLLDKPTGRKVDLKADYVGFTVPHEFVVGYGLDYKEQYRNLPYVGVLKPSVYS 6d9x A 1.83 BS01 FZM A 1 S49 S91 F133 S175 C261 F263 I305 S20 S62 F104 S146 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Ki=323uM remove_due_to_license_issue Ki=323000nM P61964 29889518 502 PVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6da4 A 2.9 BS01 G4V A 1 L828 G829 A853 Y904 L905 C909 L956 L14 G15 A39 Y90 L91 C95 L142 D949 A951 R953 N954 D967 D135 A137 R139 N140 D153 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 30423248 1201 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 6dai A 1.63 BS01 G2V A 1 S49 S91 F133 S175 F219 C261 F263 I305 S20 S62 F104 S146 F190 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue Ki=85200nM P61964 29889518 503 PVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6dai A 1.63 BS02 G2V A 2 Y131 F133 F149 P173 V174 S175 Y191 Y102 F104 F120 P144 V145 S146 Y162 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue Ki=85200nM P61964 29889518 504 PVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6dak A 1.6 BS01 G1Y A 1 S49 S91 F133 S175 Y191 F219 Y260 C261 F263 I305 S19 S61 F103 S145 Y161 F189 Y230 C231 F233 I275 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Ki=7.21uM remove_due_to_license_issue Ki=7210nM P61964 29889518 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6dar A 1.88 BS01 G2J A 1 S49 S91 F133 F149 S175 Y191 F219 Y260 C261 F263 I305 S19 S61 F103 F119 S145 Y161 F189 Y230 C231 F233 I275 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Ki=0.219uM remove_due_to_license_issue Ki=219nM P61964 29889518 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKS 6das A 1.8 BS01 G2D A 1 S49 S91 D92 F133 F149 P173 S175 Y191 F219 Y260 C261 F263 I305 S20 S62 D63 F104 F120 P144 S146 Y162 F190 Y231 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Ki=8.37nM remove_due_to_license_issue Ki=30.2nM P61964 29889518 401 PVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6db3 A 1.97 BS01 G54 A 1 L828 A853 K855 M902 Y904 L905 N954 L956 D967 L15 A40 K42 M81 Y83 L84 N133 L135 D146 D949 A951 R953 N954 D967 D128 A130 R132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 ic50=56nM remove_due_to_license_issue IC50=56nM P52333 30423248 4000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQDQQRDFQREIQILKALHSDFIVKYRGVSYGSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 6db4 A 1.662 BS01 G4Y A 1 L828 V836 A853 E903 Y904 L905 C909 D912 R953 L956 D967 L15 V23 A40 E83 Y84 L85 C89 D92 R133 L136 D147 D949 A951 R953 N954 D967 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 30423248 4000 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQGPDQQRDFQREIQILKALHSDFIVKYRGVSYSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 6db9 H 2.025 BS01 rna R 0 Y34 Y57 S58 S60 Q102 Y104 R105 R106 R110 Y31 Y54 S55 S57 Q99 Y101 R102 R103 R107 remove_due_to_license_issue 30382099 1 ~ 60 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPYSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARQGYRRRSGRGFDYWGQGTLVTVSSASTKGPSVFPLAPSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKS 6db9 L 2.025 BS01 rna R 0 S92 F95 S91 F94 remove_due_to_license_issue 30382099 1 ~ 60 DIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSYSFPSTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAQWKVDNALQGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGSSPVTKSFNRGE 6dcb A 1.998 BS01 rna B 0 Y418 C419 K420 Y421 G423 Y424 H456 S482 Q485 N486 R488 H489 Y490 K585 W586 Q618 R626 S671 G673 F674 R676 Y8 C9 K10 Y11 G13 Y14 H46 S72 Q75 N76 R78 H79 Y80 K122 W123 Q155 R163 S208 G210 F211 R213 2.1.1.- 0008168 remove_due_to_license_issue Q7L2J0 30559425 1 ~ 116 RKFQYGNYCKYYGYRNPSCEDGRLRVLKPEWFRGRDVLDLGCNVGHLTLSIACKWGPSRMVGLDIDSRLIHSARQNIRHYLSTSVFPNNVVFVTGNYVLDRDDLVEAQTPEYDVVLCLSLTKWVHLNWGDEGLKRMFRRIYRHLRPGGILVLEPQPWSSYGKRKTLTETIYKNYYRIQLKPEQFSSYLTSPDVGFSSYELVATPHNTSKGFQRPVYLFHKARSPS 6dcc A 2.1 BS01 rna B 0 Y418 C419 K420 Y421 G423 Y424 H456 S482 Q485 N486 R488 H489 Y490 K585 W586 Q618 R626 S671 G673 F674 R676 Y7 C8 K9 Y10 G12 Y13 H45 S71 Q74 N75 R77 H78 Y79 K119 W120 Q152 R160 S205 G207 F208 R210 2.1.1.- 0008168 remove_due_to_license_issue Q7L2J0 30559425 1 ~ 116 KFQYGNYCKYYGYRNPSCEDGRLRVLKPEWFRGRDVLDLGCNVGHLTLSIACKWGPSRMVGLDIDSRLIHSARQNIRHYLSVFPNNVVFVTGNYVLDRDDLVEAQTPEYDVVLCLSLTKWVHLNWGDEGLKRMFRRIYRHLRPGGILVLEPQPWSSYGKRKTLTETIYKNYYRIQLKPEQFSSYLTSPDVGFSSYELVATPHNTSKGFQRPVYLFHKARSP 6dcg A 1.45 BS01 G67 A 1 I29 A33 Y34 A50 K52 Y62 R65 E69 Q103 D104 L105 M106 E107 T108 K112 L154 D165 I14 A18 Y19 A30 K32 Y42 R45 E49 Q83 D84 L85 M86 E87 T88 K92 L134 D145 D147 K149 N152 D165 T188 D127 K129 N132 D145 T168 2.7.11.24 0000165,0001784,0003690,0004672,0004674,0004705,0004707,0005515,0005524,0005634,0005654,0005737,0005739,0005769,0005770,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006974,0007166,0007254,0007507,0008284,0008286,0008353,0009636,0009887,0010759,0014032,0014044,0014069,0015966,0016020,0016301,0018105,0018107,0019233,0019858,0019901,0019902,0030278,0030335,0030424,0030521,0030641,0030878,0031143,0031435,0031647,0031663,0032206,0032355,0032496,0032839,0032872,0032991,0033574,0033598,0034198,0035094,0035556,0036120,0038127,0038133,0042220,0042307,0042473,0042542,0042552,0042802,0043204,0043330,0043401,0043627,0044849,0045542,0045596,0045727,0045893,0046697,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060045,0060291,0060324,0060425,0060440,0060716,0061308,0061431,0070161,0070371,0070849,0071320,0071356,0071364,0071380,0072584,0072686,0090170,0097237,0097305,0106310,0120041,1990314,2000641 ic50=7nM remove_due_to_license_issue P63086 30034615 403 VFDVGPRYTNLSYIGEGAYGMVCSAYDRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFLPKEKLKELIFEETARFQP 6dcl A 2.497 BS01 rna C 0 K15 F17 G19 G20 R55 F57 F59 E85 A89 V90 R92 S95 H101 K9 F11 G13 G14 R49 F51 F53 E79 A83 V84 R86 S89 H95 ? 0003676,0003723 remove_due_to_license_issue P09651 29946118 1 ~ 11 PKEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMAS 6dcl A 2.497 BS02 rna D 0 K106 F108 G110 G111 E114 K145 R146 G147 F148 F150 E176 R178 A180 L181 S182 K183 M186 K100 F102 G104 G105 E108 K139 R140 G141 F142 F144 E170 R172 A174 L175 S176 K177 M180 ? 0003676,0003723 remove_due_to_license_issue P09651 29946118 1 ~ 11 PKEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDRGSGKKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSKQEMAS 6dcl B 2.497 BS01 rna C 0 K106 F108 G110 G111 M137 K145 R146 F148 F150 E176 R178 L181 K99 F101 G103 G104 M130 K133 R134 F136 F138 E164 R166 L169 ? 0003676,0003723 remove_due_to_license_issue P09651 29946118 1 ~ 11 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSK 6dcl B 2.497 BS02 rna D 0 Q12 K15 F17 G20 M46 R55 G56 F57 F59 E85 K87 A89 V90 R92 S95 H101 Q5 K8 F10 G13 M39 R48 G49 F50 F52 E78 K80 A82 V83 R85 S88 H94 ? 0003676,0003723 remove_due_to_license_issue P09651 29946118 1 ~ 11 KEPEQLRKLFIGGLSFETTDESLRSHFEQWGTLTDCVVMRDPNTKRSRGFGFVTYATVEEVDAAMNARPHKVDGRVVEPKRAVSREDSQRPGAHLTVKKIFVGGIKEDTEEHHLRDYFEQYGKIEVIEIMTDKRGFAFVTFDDHDSVDKIVIQKYHTVNGHNCEVRKALSK 6dcy A 2.08 BS03 G5V A 1 H41 E80 D108 E119 K134 H43 E62 D90 E101 K116 3.1.-.- 0003723,0039694 ic50=3.5uM remove_due_to_license_issue C3W5S0 30351002 303 MAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 6dcz A 2.89 BS01 G5Y A 1 H41 E80 D108 E119 K134 H42 E64 D92 E103 K118 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 30351002 301 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 6dd0 A 1.5 BS03 P9T A 1 F61 D120 H196 R228 N233 H263 F31 D87 H148 R174 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 Ki=3.3uM remove_due_to_license_issue Q9K2N0 31483651 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTN 6dd1 A 1.7 BS03 M3Q A 1 F61 W87 H118 D120 H196 N233 F31 W56 H85 D87 H148 N179 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 Ki=22.3uM remove_due_to_license_issue Q9K2N0 31483651 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6dd1 A 1.7 BS04 M3Q A 2 Y67 H196 R228 G232 N233 H263 Y36 H148 R174 G178 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 Ki=22.3uM remove_due_to_license_issue Q9K2N0 31483651 404 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6det A 1.75 BS01 ARG A 1 S29 V32 W70 S87 G88 F89 S90 R95 E134 T137 D179 Y182 S20 V23 W61 S78 G79 F80 S81 R86 E125 T128 D170 Y173 ? Kd=0.006uM remove_due_to_license_issue S3MDF0 30242931 500 IEDPSWSKVQVKSALVIGVSDFVPILSFRNEKNEIVGYDIDIFTELCRRLGIHPIFYPIQWAQKEILLNTGVIDCIASGFSVTEERKQHYRMCTPYLQNAKIVVTLAGRGYQTLAQLQNRTIAVEADTAGDEALLNVEALKDHVIIKAMATIDQLYEALDSGTCDAIVVDLIYSLDTLDKNPQYSIINEAISTEYYTFAFRQADASLVAKIESVLAEMNEDETIPNFSRKWFGSNLSILNVRF 6df4 A 1.3 BS01 G9Y A 1 P1527 F1528 H1530 V1532 N1533 F1536 V1537 Y1582 N1583 Y1589 P27 F28 H30 V32 N33 F36 V37 Y82 N83 Y89 ? 0004402,0005669,0006366,0016251,0017025 ic50=0.023uM remove_due_to_license_issue U3KMH2 30289257 4000 DDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESL 6df7 A 2.0 BS01 G9V A 1 P1527 F1528 H1530 V1532 N1533 F1536 V1537 Y1582 N1583 Y1589 P27 F28 H30 V32 N33 F36 V37 Y82 N83 Y89 ? 0004402,0005669,0006366,0016251,0017025 ic50=0.01uM remove_due_to_license_issue U3KMH2 30289257 4001 DDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESLD 6dge A 1.91 BS01 GBG A 1 L30 D73 F76 E78 D79 R98 G129 R145 V268 C274 L23 D66 F69 E71 D72 R91 G122 R138 V261 C267 3.5.3.18 0000052,0003073,0003824,0005829,0006525,0006527,0007263,0008285,0016403,0016597,0016787,0043116,0045429,0045766,0046209,0046872,0070062,1900038 remove_due_to_license_issue O94760 29983043 301 AAFGRATHAVVRALPESLGQHALRSAKGEEVDVARAERQHQLYVGVLGSKLGLQVVELPADESLPDCVFVEDVAVVCEETALITRPGAPSRRKEVDMMKEALEKLQLNIVEMKDENATLDGGDVLFTGREFFVGLSKRTNQRGAEILADTFKDYAVSTVPVADGLHLKSFCSMAGPNLIAIGSSESAQKALKIMQQMSDHRYDKLTVPDDIAANCIYLNIPNKGHVLLHRTPEEYPESAKVYEKLKDHMLIPVSMSELEKVDGLLTCCSVLINKK 6dgl A 1.95 BS01 GEV A 1 F264 F282 G284 C285 Q286 S289 H323 Y327 L330 I341 M364 H449 Y473 F58 F66 G68 C69 Q70 S73 H107 Y111 L114 I125 M148 H233 Y257 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 31611383 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 6dgo A 3.1 BS01 GD4 A 1 C285 R288 S289 Y327 L330 I341 S342 M348 M364 H449 L453 Y473 C71 R74 S75 Y113 L116 I127 S128 M134 M150 H235 L239 Y259 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 31611383 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 6dgq A 2.45 BS01 GBV A 1 F282 G284 C285 S289 H323 L330 I341 M364 H449 L469 Y473 F64 G66 C67 S71 H105 L112 I123 M145 H230 L250 Y254 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 31611383 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 6dgr A 2.15 BS01 GDY A 1 F282 C285 S289 H323 I341 M364 H449 Y473 F67 C70 S74 H108 I126 M149 H234 Y258 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 31611383 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 6dgt A 2.601 BS01 GFJ A 1 M752 P758 I777 K779 D787 I825 V827 V828 M900 D911 M522 P528 I547 K549 D557 I595 V597 V598 M663 D674 2.7.1.137,2.7.1.153 0001782,0002250,0005524,0005737,0005829,0006629,0006935,0006954,0007166,0010628,0016301,0016303,0030154,0036092,0042113,0043491,0045087,0045766,0046854,0046934,0048872,0050832 remove_due_to_license_issue O35904 30015489 1101 KLINSQISLLIGKGLDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPALLVNVKFEEESFTFQVSTKDMPLALMACALRQPEEYALQVNGRHEYLYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNSLEQPFSIELIEGRKVMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRE 6dgx A 2.001 BS01 017 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 3.1.13.2,3.1.26.13 0004190,0006508 Ki<5pM remove_due_to_license_issue Q72498 30543749 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dgx B 2.001 BS01 017 A 1 D25 A28 D30 P81 I84 D25 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 3.1.13.2,3.1.26.13 0004190,0006508 remove_due_to_license_issue Q72498 30543749 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dgy A 1.954 BS01 K13 A 1 D25 G27 A28 D29 G48 I50 V82 D25 G27 A28 D29 G48 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki<5pM remove_due_to_license_issue Q7ZCR0 30543749 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dgy B 1.954 BS01 K13 A 1 D25 A28 D30 P81 D25 A28 D30 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCR0 30543749 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dgz A 1.994 BS01 A60 A 1 D25 G27 A28 D29 G48 I50 V82 D25 G27 A28 D29 G48 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki<5pM remove_due_to_license_issue Q7ZCR0 30543749 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dgz B 1.994 BS01 A60 A 1 D25 A28 D30 P81 D25 A28 D30 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCR0 30543749 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dh0 A 1.899 BS01 017 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=25.6pM remove_due_to_license_issue Q7ZCI0 30543749 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 6dh0 B 1.899 BS01 017 A 1 D25 A28 D30 V32 V82 D25 A28 D30 V32 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCI0 30543749 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 6dh1 A 1.971 BS01 K13 A 1 D25 G27 A28 D29 I47 G48 I50 V82 D25 G27 A28 D29 I47 G48 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=26.1pM remove_due_to_license_issue Q7ZCI0 30543749 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 6dh1 B 1.971 BS01 K13 A 1 D25 G27 A28 D30 V32 D25 G27 A28 D30 V32 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCI0 30543749 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 6dh2 A 1.978 BS01 A60 A 1 D25 G27 A28 D29 I47 G48 I50 V82 D25 G27 A28 D29 I47 G48 I50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=12.8pM remove_due_to_license_issue Q7ZCI0 30543749 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 6dh2 B 1.978 BS01 A60 A 1 D25 A28 D30 V32 D25 A28 D30 V32 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCI0 30543749 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNVIGRNLLTQIGCTLNF 6dh3 A 1.908 BS01 017 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki<5pM remove_due_to_license_issue Q6B6C5 30543749 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 6dh3 B 1.908 BS01 017 A 1 D25 G27 A28 D30 P81 I84 D25 G27 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q6B6C5 30543749 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 6dh4 A 1.943 BS01 K13 A 1 D25 G27 A28 D29 G48 I50 I82 D25 G27 A28 D29 G48 I50 I82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki<5pM remove_due_to_license_issue Q6B6C5 30543749 104 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 6dh4 B 1.943 BS01 K13 A 1 D25 G27 A28 D30 P81 D25 G27 A28 D30 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q6B6C5 30543749 104 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 6dh5 A 2.008 BS01 A60 A 1 D25 G27 A28 D29 I47 G48 I50 I82 I84 D25 G27 A28 D29 I47 G48 I50 I82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q6B6C5 30543749 104 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 6dh5 B 2.008 BS01 A60 A 1 D25 G27 A28 D30 P81 D25 G27 A28 D30 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q6B6C5 30543749 104 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPINIIGRNLLTQIGCTLNF 6dh6 A 1.97 BS01 017 A 1 D25 G27 A28 D29 D30 G48 V50 D25 G27 A28 D29 D30 G48 V50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=117.2pM remove_due_to_license_issue Q7ZCR0 30543749 104 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dh6 B 1.97 BS01 017 A 1 D25 A28 D30 P81 D25 A28 D30 P81 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCR0 30543749 104 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dh7 A 1.997 BS01 K13 A 1 D25 G27 A28 D29 D30 G48 V50 V82 D25 G27 A28 D29 D30 G48 V50 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=131.3pM remove_due_to_license_issue Q7ZCR0 30543749 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dh7 B 1.997 BS01 K13 A 1 D25 G27 A28 D30 P81 V82 I84 D25 G27 A28 D30 P81 V82 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCR0 30543749 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dh8 A 1.951 BS01 A60 A 1 D25 G27 A28 D29 G48 V50 D25 G27 A28 D29 G48 V50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=146.2pM remove_due_to_license_issue Q7ZCR0 30543749 105 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dh8 B 1.951 BS01 A60 A 1 D25 A28 D30 V32 P81 I84 D25 A28 D30 V32 P81 I84 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q7ZCR0 30543749 105 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGVGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6dha A 1.88 BS01 GFV A 1 I281 F282 G284 C285 Q286 S289 H323 I341 M348 M364 H449 Y473 I60 F61 G63 C64 Q65 S68 H102 I120 M127 M143 H228 Y252 ? 0003677,0004879,0005634,0006355 Kd=708nM remove_due_to_license_issue EC50=1300nM, Ki=1200nM, Kd=708nM, IC50=13000nM P37231 30676741 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 6dhc A 2.85 BS01 GHJ A 1 G11 Q12 G13 L30 D32 G34 P70 Y71 T72 Q73 F108 I110 Y198 D228 G230 T231 T232 G15 Q16 G17 L34 D36 G38 P74 Y75 T76 Q77 F112 I114 Y191 D221 G223 T224 T225 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D221 T224 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 29970308 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6dhu A 1.63 BS01 GHM A 1 Y204 H263 K265 N283 S399 P461 H493 K495 N516 Y43 H102 K104 N122 S238 P295 H327 K329 N350 3.1.4.- 0005634,0006281,0008081 remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6di0 A 1.3 BS01 GJG A 1 L408 T410 G411 A428 Y476 M477 L528 L20 T22 G23 A40 Y88 M89 L140 D521 A523 R525 N526 D539 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>6000nM Q06187 30290988 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6di1 A 1.1 BS01 GJD A 1 L408 T410 G411 A428 Y476 M477 C481 L528 L20 T22 G23 A40 Y88 M89 C93 L140 D521 A523 R525 N526 D539 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30290988 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6die A 1.78 BS01 GHM A 1 Y204 H263 K265 N283 S399 P461 H493 K495 N516 Y43 H102 K104 N122 S238 P295 H327 K329 N350 3.1.4.- 0005634,0006281,0008081 ic50=0.74mM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6dif A 1.2 BS01 TPV B 1 D25 A28 D29 D30 G48 G49 I50 P81 D25 A28 D29 D30 G48 G49 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6dif B 1.2 BS01 TPV B 1 R8 D25 G27 G49 I50 V82 R8 D25 G27 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.019nM remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6dih A 1.78 BS01 GJS A 1 Y204 H263 K265 S399 P461 H493 K495 N516 Y43 H102 K104 S238 P295 H327 K329 N350 3.1.4.- 0005634,0006281,0008081 ic50=1.9mM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6dik A 1.93 BS01 GKP A 1 F3 G6 K7 F3 G6 K7 N28 G30 L32 H48 K49 Y52 Y73 D99 N27 G29 L31 H47 K48 Y51 Y64 D89 ? 0004623,0005509,0005543,0005576,0006644,0008201,0016042,0035821,0042130,0042742,0047498,0050482,0090729 remove_due_to_license_issue Q90249 30251662 201 SLFELGKMILQETGKNPAKSYGAYGCNCGVLGRGKPKDATDRCCYVHKCCYKKLTGCNPKKDRYSYSWKDKTIVCGENNPCLKELCECDKAVAICLRENLGTYNKKYRYHLKPFCKKADPC 6dil A 1.482 BS01 TPV B 1 D25 A28 D29 D30 G48 G49 I50 V82 D25 A28 D29 D30 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dil B 1.482 BS01 TPV B 1 R8 D25 I50 R8 D25 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=7.6nM remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dim A 1.81 BS01 GJP A 1 Y204 H263 K265 N283 P461 H493 W590 Y43 H102 K104 N122 P295 H327 W420 3.1.4.- 0005634,0006281,0008081 remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6dj1 A 1.26 BS01 AB1 B 1 D25 G27 A28 D29 G48 G49 I84 D25 G27 A28 D29 G48 G49 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6dj1 B 1.26 BS01 AB1 B 1 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 V82 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.031nM remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6dj2 A 1.36 BS01 AB1 B 1 D25 G27 A28 D29 I47 G48 P81 V82 I84 D25 G27 A28 D29 I47 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dj2 B 1.36 BS01 AB1 B 1 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 D25 G27 A28 D29 D30 G48 G49 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4.5nM remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dj5 A 1.75 BS01 G52 B 1 R8 D25 A28 D30 G48 P81 V82 I84 R8 D25 A28 D30 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dj5 B 1.75 BS01 G52 B 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dj7 A 1.31 BS01 G10 B 1 D25 G27 A28 D30 G48 G49 P81 V82 I84 D25 G27 A28 D30 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6dj7 B 1.31 BS01 G10 B 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1.9nM remove_due_to_license_issue P04585 30288468 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVVVGPTPVNIIGRNLLTQIGATLNF 6djc A 1.46 BS01 CF6 A 1 W81 P82 F83 V87 L92 L94 N140 I146 M149 W39 P40 F41 V45 L50 L52 N98 I104 M107 ? Ki=232.8nM remove_due_to_license_issue O60885 30012592 501 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEETEIMI 6djd A 1.777 BS01 GJP A 1 Y204 H263 K265 N283 P461 H493 W590 Y43 H102 K104 N122 P295 H327 W421 3.1.4.- 0005634,0006281,0008081 ic50=7.2mM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6dji A 1.75 BS01 GOG A 1 Y204 H263 K265 N283 P461 H493 K495 N516 Y43 H102 K104 N122 P295 H327 K329 N350 3.1.4.- 0005634,0006281,0008081 ic50=3.1mM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6djj A 1.741 BS01 GM7 A 1 Y204 H263 K265 N283 S399 P461 H493 K495 N516 Y43 H102 K104 N122 S238 P295 H327 K329 N350 3.1.4.- 0005634,0006281,0008081 ic50=80uM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6dk1 A 3.12 BS01 GM4 A 1 V84 W89 Y103 F107 E172 F184 A185 V77 W82 Y96 F100 E165 F177 A178 ? 0004985,0005515,0005634,0005635,0005637,0005640,0005783,0005789,0005811,0005829,0005886,0006869,0007399,0014069,0016020,0030426,0031410,0038003,0038023,0042995,0043523,0045202,0045211,0070161,0070207,0098794,0098839,0098978,0150052 remove_due_to_license_issue Ki=3.1nM, Kd=11.6nM, IC50=8.2nM Q99720 30291362 301 RWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRYWAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLF 6dkb A 2.68 BS01 FKY A 1 L516 A542 L564 V573 F589 E590 Y591 M592 G595 H648 L657 I666 G667 D668 F669 L16 A42 L64 V73 F89 E90 Y91 M92 G95 H135 L144 I153 G154 D155 F156 D650 R654 N655 D668 D137 R141 N142 D155 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Kd=0.700000nM, IC50=1900nM P04629 29944371 4000 CVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGSTDYYRMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVLG 6dkg A 2.53 BS02 GO7 A 1 L516 V524 A542 L564 F589 Y591 M592 F646 H648 L657 I666 G667 D668 F669 L17 V25 A43 L65 F90 Y92 M93 F135 H137 L146 I155 G156 D157 F158 D650 R654 N655 D668 D139 R143 N144 D157 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=7700nM, Kd=1.1nM P04629 29944371 802 ACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGYSTDYYRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVLG 6dki A 2.11 BS02 GOD A 1 V524 A542 L564 L567 V573 F589 E590 Y591 M592 L657 I666 G667 D668 F669 V25 A43 L65 L68 V74 F90 E91 Y92 M93 L146 I155 G156 D157 F158 D650 R654 N655 D668 D139 R143 N144 D157 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Kd=5.7nM, IC50=8.4nM P04629 29944371 802 ACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGRDIYSTDYYRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVLG 6dko A 1.556 BS02 GXG A 1 R339 G459 L461 D462 M515 W541 M631 D633 R332 G449 L451 D452 M505 W531 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R332 E424 D452 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=1.6uM remove_due_to_license_issue P9WK17 30137983 804 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAAAVFLRVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKEAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6dl2 A 1.47 BS01 GUJ A 1 W81 P82 V87 L92 N140 I146 M149 W41 P42 V47 L52 N100 I106 M109 ? Ki=33nM remove_due_to_license_issue IC50=100nM, Ki=33nM O60885 30019901 201 SNANPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6dl9 A 1.8 BS02 GXD A 1 V118 R339 E434 G459 L461 D462 M515 W541 M631 D633 V117 R328 E423 G448 L450 D451 M504 W530 M620 D622 D271 E273 R339 E434 D462 D633 D270 E272 R328 E423 D451 D622 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=1uM remove_due_to_license_issue P9WK17 30137983 804 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDVNGPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGASKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6dlj A 2.604 BS02 GXM A 1 V118 R339 E434 G459 F460 L461 D462 W541 M631 D633 V112 R323 E414 G439 F440 L441 D442 W521 M611 D613 D271 E273 R339 E434 D462 D633 D265 E267 R323 E414 D442 D613 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 remove_due_to_license_issue P9WK17 30137983 803 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASDLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGCSKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6dlx A 1.848 BS01 GXY A 1 D359 K406 D165 K212 3.6.5.4 0005525,0006614,0016887 Kd~480uM remove_due_to_license_issue P10121 30044812 501 GFARLKRSLLKTKENLGSGFISLFRGKKIDDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFA 6dlx A 1.848 BS02 GXY A 2 T308 G311 K312 W343 T114 G117 K118 W149 3.6.5.4 0005525,0006614,0016887 Kd~480uM remove_due_to_license_issue P10121 30044812 502 GFARLKRSLLKTKENLGSGFISLFRGKKIDDDLFEELEEQLLIADVGVETTRKIITNLTEGASRKQLRDAEALYGLLKEEMGEILAKVDEPLNVEGKAPFVILMVGVNGVGKTTTIGKLARQFEQQGKSVMLAAGDTFRAAAVEQLQVWGQRNNIPVIAQHTGADSASVIFDAIQAAKARNIDVLIADTAGRLQNKSHLMEELKKIVRVMKKLDVEAPHEVMLTIDASTGQNAVSQAKLFHEAVGLTGITLTKLDGTAKGGVIFSVADQFGIPIRYIGVGERIEDLRPFKADDFIEALFA 6dm8 A 2.7 BS03 6AK A 1 A208 F209 M212 F227 M231 F235 R244 L248 F251 A420 F421 M424 F439 M443 F447 R456 L460 F463 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,P97287 30011190 401 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSDLYRQSLEIISRYLREQATGSKDSKAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEGDVKSFSRVMVHVFKDGVTNWGRIVTLISFGAFVAKHLKSVNQESFIEPLAETITDVLVRTKRDWLVKQRGWDGFVEFFH 6dm8 A 2.7 BS04 6AK A 2 Y-125 P-124 F-123 M106 A109 Q110 Y91 P92 F93 M322 A325 Q326 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,P97287 30011190 403 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSDLYRQSLEIISRYLREQATGSKDSKAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEGDVKSFSRVMVHVFKDGVTNWGRIVTLISFGAFVAKHLKSVNQESFIEPLAETITDVLVRTKRDWLVKQRGWDGFVEFFH 6dm8 A 2.7 BS05 6AK A 3 M212 K215 L216 F227 R229 V230 M424 K427 L428 F439 R441 V442 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,P97287 30011190 404 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSDLYRQSLEIISRYLREQATGSKDSKAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEGDVKSFSRVMVHVFKDGVTNWGRIVTLISFGAFVAKHLKSVNQESFIEPLAETITDVLVRTKRDWLVKQRGWDGFVEFFH 6dm8 A 2.7 BS06 6AK G 3 M212 V230 V234 M424 V442 V446 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,P97287 30011190 404 GKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSDLYRQSLEIISRYLREQATGSKDSKAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEGDVKSFSRVMVHVFKDGVTNWGRIVTLISFGAFVAKHLKSVNQESFIEPLAETITDVLVRTKRDWLVKQRGWDGFVEFFH 6dne A 2.958 BS01 H1V A 1 W81 P82 L92 N93 L94 N140 I146 M149 W38 P39 L49 N50 L51 N97 I103 M106 ? remove_due_to_license_issue O60885 30012592 501 NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 6dnp A 1.711 BS02 GZV A 1 R339 E434 G459 L461 D462 M515 W541 M631 D633 R328 E419 G444 L446 D447 M500 W526 M616 D618 D271 E273 R339 E434 D462 D633 D270 E272 R328 E419 D447 D618 2.3.3.9 0000287,0001968,0003824,0004474,0005515,0005518,0005576,0005737,0005829,0005886,0006097,0006099,0009274,0009436,0009986,0015936,0016740,0042603,0042803,0043236,0044406,0046810,0046872,0120225 ic50=6.6uM remove_due_to_license_issue P9WK17 30137983 803 TDRVSVGNLRIARVLYDFVNNEALPGTDIDPDSFWAGVDKVVADLTPQNQALLNARDELQAQIDKWHRRRVIEPIDMDAYRQFLTEIGYLLPEPDDFTITTSGVDAEITTTAGPQLVVPVLNARFALNAANARWGSLYDALYGTDVIPETDGAEKGPTYNKVRGDKVIAYARKFLDDSVPLSSGSFGDATGFTVQDGQLVVALPDKSTGLANPGQFAGYTGAAESPTSVLLINHGLHIEILIDPESQVGTTDRAGVKDVILESAITTIMDFEDSVAAVDAADKVLGYRNWLGLNKGDLAARVLNRDRNYTAPGGGQFTLPGRSLMFVRNVGHLMTNDAIVDTDGSEVFEGIMDALFTGLIAIHGLKASPLINSRTGSIYIVKPKMHGPAEVAFTCELFSRVEDVLGLPQNTMKIGIMDEERRTTVNLKACIKAAADRVVFINTGFLDRTGDEIHTSMEAGPMVRKGTMKSQPWILAYEDHNVDAGLAAGFSGRAQVGKGMWTMTELMADMVETKIAQPRAGASTAWVPSPTAATLHALHYHQVDVAAVQQGLAGKRRATIEQLLTIPLAKELAWAPDEIREEVDNNCQSILGYVVRWVDQGVGCSKVPDIHDVALMEDRATLRISSQLLANWLRHGVITSADVRASLERMAPLVDRQNAGDVAYRPMAPNFDDSIAFLAAQELILSGAQQPNGYTEPILHRRRREFKARAAE 6dnw A 2.849 BS01 dna B 0 G139 K142 R143 T152 A153 R156 T165 S189 T191 Y207 N208 M254 N261 K262 K286 S290 K293 Y295 Y297 Y299 T308 K313 I318 R320 G6 K9 R10 T19 A20 R23 T32 S56 T58 Y74 N75 M121 N128 K129 K153 S157 K160 Y162 Y164 Y166 T175 K180 I185 R187 ? 0000150,0003677 remove_due_to_license_issue Q928V6 30227134 1 ~ 26 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYLEFREKQLYLKSLINKIYIDGEQVTIEWL 6dnw A 2.849 BS02 dna C 0 K140 T151 R156 R209 N212 Y225 K226 N259 K262 S264 S266 N269 V282 H283 R285 D287 T288 K303 K306 K7 T18 R23 R76 N79 Y92 K93 N126 K129 S131 S133 N136 V149 H150 R152 D154 T155 K170 K173 ? 0000150,0003677 remove_due_to_license_issue Q928V6 30227134 1 ~ 26 DRMVMGKIKRIEAGLPLTTAKGRTFGYDVIDTKLYINEEEAKQLRLIYDIFEEEQSITFLQKRLKKLGFKVRTYNRYNNWLTNDLYCGYVSYKDKVHVKGIHEPIISEEQFYRVQEIFSRMGKNPNMNKESASLLNNLVVCSKCGLGFVHRRKDTVSRGKKYHYRYYSCKTYKHTHELEKCGNKIWRADKLEELIIDRVNNYLEFREKQLYLKSLINKIYIDGEQVTIEWL 6dpt A 1.79 BS01 H7M A 1 S64 Q120 N152 Y221 T316 G317 A318 T319 G320 S61 Q117 N149 Y218 T313 G314 A315 T316 G317 S64 K67 Y150 E272 K315 A318 S61 K64 Y147 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 30728502 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 6dpx A 1.9 BS01 H7G A 1 S64 N152 S212 G317 A318 T319 G320 S61 N149 S209 G314 A315 T316 G317 S64 K67 Y150 E272 K315 A318 S61 K64 Y147 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 30728502 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 6dpy A 1.91 BS01 H7A A 1 S64 L119 N152 Y221 G317 A318 T319 G320 S61 L116 N149 Y218 G314 A315 T316 G317 S64 K67 Y150 E272 K315 A318 S61 K64 Y147 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 30728502 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 6dpz A 1.5 BS01 H7D A 1 S64 L119 Q120 N152 Y221 L293 G317 A318 S61 L116 Q117 N149 Y218 L290 G314 A315 S64 K67 Y150 E272 K315 A318 S61 K64 Y147 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 remove_due_to_license_issue P00811 30728502 401 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 6dq4 A 1.392 BS01 K0I A 1 R73 Y409 A411 D412 Y472 F480 H483 E485 K501 R63 Y137 A139 D140 Y196 F204 H207 E209 K225 Y472 H483 E485 H571 A583 Y196 H207 E209 H295 A307 1.14.11.67 Kd=12uM remove_due_to_license_issue IC50=110000nM, Kd=12000nM P29375 30392349 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRPREAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINVMKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6dq5 A 1.89 BS01 H6G A 1 R73 Y409 Y472 F480 C481 H483 E485 K501 R62 Y125 Y183 F191 C192 H194 E196 K212 Y472 H483 E485 H571 A583 Y183 H194 E196 H282 A294 1.14.11.67 Kd=6.4uM remove_due_to_license_issue Kd=6000nM, IC50=71000nM P29375 30392349 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINVKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFC 6dq6 A 1.587 BS01 H6J A 1 R73 Y409 D412 Y472 F480 C481 H483 E485 K501 L536 R62 Y125 D128 Y182 F190 C191 H193 E195 K211 L246 Y472 H483 E485 H571 A583 Y182 H193 E195 H281 A293 1.14.11.67 Kd=8.5uM remove_due_to_license_issue Kd=9000nM, IC50=83000nM P29375 30392349 601 EFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTRREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLAHINKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6dq8 A 1.46 BS01 H6S A 1 Y409 A411 W470 Y472 F480 C481 H483 K501 W503 H571 Y133 A135 W184 Y186 F194 C195 H197 K215 W217 H285 Y472 H483 E485 H571 A583 Y186 H197 E199 H285 A297 1.14.11.67 Kd=0.26uM remove_due_to_license_issue Kd=260nM, IC50=320nM P29375 30392349 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMTAFGFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6dqa A 1.888 BS01 H6V A 1 Y409 D412 Y472 F480 C481 H483 K501 W503 H571 Y129 D132 Y181 F189 C190 H192 K210 W212 H280 Y472 H483 E485 H571 A583 Y181 H192 E194 H280 A292 1.14.11.67 remove_due_to_license_issue IC50=4900nM P29375 30392349 601 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMFEQAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6dqb A 1.791 BS03 HZM A 1 R73 Y409 A411 D412 Y472 F480 C481 H483 K501 W503 H571 R63 Y126 A128 D129 Y179 F187 C188 H190 K208 W210 H278 Y472 H483 E485 H571 A583 Y179 H190 E192 H278 A290 1.14.11.67 remove_due_to_license_issue P29375 30392349 603 AEFVPPPECPVFEPSWEEFTDPLSFIGRIRPLAEKTGICKIRPPKDWQPPFACEVKSFRFTPRVQRLNELEAMAVREYTLQSFGEMADNFKSDYFNMPVHMVPTELVEKEFWRLVSSIEEDVIVEYGADISSKDFGSGFPVKDGRRKILPEEEEYALSGWNLNNMPVLEQSVLKVPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPSHAAEQLEEVMRELAPELFESQPDLLHQLVTIMNPNVLMEHGVPVYRTNQCAGEFVVTFPRAYHSGFNQGYNFAEAVNFCT 6drx A 3.1 BS01 H8G A 1 W131 L132 D135 V136 S139 F217 A225 W337 F340 W85 L86 D89 V90 S93 F168 A176 W305 F308 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41595 30127358 1201 VEEQGNKLHWAALLILMVIIPTIGGNTLVILAVSLEKKLQYATNYFLMSLAVADLLVGLFVMPIALLTIMFEAMWPLPLVLCPAWLFLDVLFSTASIWHLCAISVDRYIAIKKPIQANQYNSRATAFIKITVVWLISIGIAIPVPIKGIETNPNNITCVLTKERFGDFMLFGSLAAFFTPLAIMIVTYFLTIHALQKKAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLQTISNEQRASKVLGIVFFLFLLMWCPFFITNITLVLCDSCNQTTLQMLLEIFVWIGYVSSGVNPLVYTLFNKTFRDAFGRYITCNYR 6dry A 2.918 BS01 H8D A 1 D135 V136 T140 V208 L209 G221 F340 L362 D93 V94 T98 V162 L163 G175 F330 L352 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41595 30127358 2001 MKQIVEEQGNKLHWAALLILMVIIPTIGGNTLVILAVSLEKKLQYATNYFLMSLAVADLLVGLFVMPIALLTIMFEAMWPLPLVLCPAWLFLDVLFSTASIWHLCAISVDRYIAIKKPIQANNSRATAFIKITVVWLISIGIAIPVPIKGIETDNPNNITCVLTKERFGDFMLFGSLAAFFTPLAIMIVTYFLTIHALQKKAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLVQTISNEQRASKVLGIVFFLFLLMWCPFFITNITLVLCDSCNQTTLQMLLEIFVWIGYVSSGVNPLVYTLFNKTFRDAFGRYITCNYR 6drz A 3.102 BS02 H8J A 1 D135 T140 V208 F340 F341 D97 T102 V167 F328 F329 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41595 30127358 1206 IPEEMKQIVEEQGNKLHWAALLILMVIIPTIGGNTLVILAVSLEKKLQYATNYFLMSLAVADLLVGLFVMPIALLTIMFEAMWPLPLVLCPAWLFLDVLFSTASIWHLCAISVDRYIAIKKPIQANSRATAFIKITVVWLISIGIAIPVPIKGIETDVDNPNNITCVLTKERFGDFMLFGSLAGFFTPLAIMIVTYFLTIHALQKKAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLVQTISNEQRASKVLGIVFFLFLLMWCPFFITNITLVLCDSCNQTTLQMLLEIFVWIGYVSSGVNPLVYTLFNKTFRDAFGRYITCNYR 6ds0 A 3.188 BS02 H8M A 1 T114 D135 V136 F217 G221 F340 L362 E363 V366 T67 D88 V89 F165 G169 F308 L330 E331 V334 ? 0004930,0004993,0005506,0005886,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P41595 30127358 1204 EEQGNKLHWAALLILMVIIPTIGGNTLVILAVSLEKKLQYATNYFLMSLAVADLLVGLFVMPIALLTIMFEAMWPLPLVLCPAWLFLDVLFSTASIWHLCAISVDRYIAIKKPIQANNSRATAFIKITVVWLISIGIAIPVPIKGIETNPNNITCVLTKERFGDFMLFGSLAAFFTPLAIMIVTYFLTIHALQKKAADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAAKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLQTISNEQRASKVLGIVFFLFLLMWCPFFITNITLVLCDSCNQTTLQMLLEIFVWIGYVSSGVNPLVYTLFNKTFRDAFGRYITCNYR 6dsp A 1.37 BS01 PAV A 1 K29 F35 F36 D110 D167 Q168 W171 D224 S225 W271 K8 F14 F15 D89 D146 Q147 W150 D203 S204 W250 ? 0030246,0030288,0030313 Kd=0.81uM remove_due_to_license_issue U5MRH9 30696769 401 VTVTFIPKLTGNAFFESANKGAQKYSEQWGFKVDYEGDANASAASQVSVINKAVQQGTNAICLSSVDAAGVKDALKAAADAGVTVTTWDSDVDPSVRKVMVSQGTPEQLGQMLVQMGYDSLKERGKDPEKDAIKYCWHYSNATVTDQNSWQVEGEKYIKSKYPNWQNVAPDNYYSNQDAEQAISVGESILSAHSDIDLIICNDSTALPGQAQAAQNKGLTAKNVTITGFASPNSMKQYCNDGILTRWGLWDCGIQGAMGCYMAYYIASGNSVKVGDKIEIPTVGTVEVMPNSVLDPKADDSDTSSGVVLLPERTIFTKDNMNNYDF 6dtw A 2.742 BS01 H9Y A 1 L100 K102 K103 V106 V108 V179 Y188 G190 F227 W229 L234 P236 Y318 L94 K96 K97 V100 V102 V173 Y182 G184 F221 W223 L228 P230 Y312 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 31281023 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVICQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDK 6dtx A 3.327 BS01 H9Y A 1 L100 K102 K103 V106 V108 Y181 Y188 F227 W229 P236 Y318 L98 K100 K101 V104 V106 Y179 Y186 F225 W227 P234 Y316 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 31281023 601 SPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQV 6dud A 1.66 BS01 HB4 A 1 L828 A853 Y904 L905 C909 D912 L956 L15 A40 Y83 L84 C88 D91 L135 D949 A951 R953 N954 D967 D128 A130 R132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P52333 30423248 1201 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 6duf A 1.963 BS01 K5C A 1 L100 K101 K103 K104 V179 Y181 Y188 L227 Y318 L102 K103 K105 K106 V181 Y183 Y190 L229 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=7.3nM remove_due_to_license_issue P03366 30044217 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSATVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPLLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 6dug A 2.225 BS01 K5C A 1 L100 P101 K103 K104 S105 V179 Y181 Y188 F227 W229 P236 Y318 L102 P103 K105 K106 S107 V181 Y183 Y190 F229 W231 P238 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=5.4nM remove_due_to_license_issue P03366 30044217 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLPKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 6duh A 2.003 BS01 K5C A 1 L100 K101 K103 V106 V179 I181 Y188 F227 W229 H235 P236 Y318 L102 K103 K105 V108 V181 I183 Y190 F229 W231 H237 P238 Y320 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 ic50=38nM remove_due_to_license_issue P03366 30044217 601 MVPISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIIQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSA 6duk A 2.2 BS03 JBJ A 1 F723 A743 K745 L747 E749 I759 M766 C775 R776 L777 L788 M790 D855 F856 L858 L861 L862 E865 F23 A43 K45 L47 E49 I59 M66 C75 R76 L77 L88 M90 D155 F156 L158 L161 L162 E165 D837 A839 R841 N842 D855 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>1000nM P00533 31092401 1103 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEED 6dvl A 2.1 BS02 HBG A 1 H463 H574 G582 F583 H614 F643 D705 Y745 H21 H132 G140 F141 H172 F201 D263 Y303 ? ic50=11nM remove_due_to_license_issue F8W4B7 30118224 804 ITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6dvm A 1.47 BS02 HBJ A 1 P464 H574 G582 F583 H614 F643 D705 Y745 P22 H132 G140 F141 H172 F201 D263 Y303 ? ic50=3nM remove_due_to_license_issue F8W4B7 30118224 804 ITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6dvn A 2.2 BS02 HB7 A 1 P464 H574 G582 F583 H614 F643 D705 Y745 P23 H133 G141 F142 H173 F202 D264 Y304 ? ic50=14nM remove_due_to_license_issue F8W4B7 30118224 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR 6dvo A 1.98 BS03 HBV A 1 P464 H573 H574 G582 F583 D612 H614 F643 Y745 P22 H131 H132 G140 F141 D170 H172 F201 Y303 ? ic50=60nM remove_due_to_license_issue F8W4B7 30118224 805 ITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLPLKTSATVSINNVLRAHAPFWSSLR 6dxg A 1.905 BS02 HGJ A 1 L159 S162 Y163 Y167 Y240 S241 T263 P264 L7 S10 Y11 Y15 Y78 S79 T101 P102 ? 0002218,0032481 ic50=14uM remove_due_to_license_issue Q86WV6 30405246 402 FNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPAFSLSQEVLRHLRQEEKEEVTV 6dxl A 2.45 BS01 HG4 A 1 S162 Y163 Y167 S241 T263 P264 S10 Y11 Y15 S78 T100 P101 ? 0002218,0032481 Kd=1.6nM remove_due_to_license_issue Q86WV6 30405246 401 FNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADFSLSQEVLRHLRQEEKEEVTV 6dxl B 2.45 BS01 HG4 A 1 S162 Y167 Y240 S241 S10 Y15 Y79 S80 ? 0002218,0032481 remove_due_to_license_issue Q86WV6 30405246 401 FNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPSSFSLSQEVLRHLRQEEKEEVTV 6dxx A 2.7 BS02 WTF B 1 V60 A63 M64 V116 Y120 V32 A35 M36 V88 Y92 3.5.1.23,3.5.1.60 remove_due_to_license_issue IC50=500nM Q02083 30301806 404 SPPAAPRFNVSLDSVPELRWLPVLRHYDLDLVRAAMAQVIGDRVPKWVHVLIGKVVLELERFLPQPFTGEIRGMCDFMNLSLADCLLVNLAYESSVF 6dxx B 2.7 BS01 WTF B 1 Y146 L152 L155 I175 Y177 W181 E195 Y21 L27 L30 I50 Y52 W56 E70 3.5.1.23,3.5.1.60 remove_due_to_license_issue IC50=500nM Q02083 30301806 404 CTSIVAQDSRGHIYHGRNLDYPFGNVLRKLTVDVQFLKNGQIAFTGTTFIGYVGLWTGQSPHKFTVSGDERDKGWWWENAIAALFRRHIPVSWLIRATLSESENFEAAVGKLAKTPLIADVYYIVGGTSPREGVVITRNRDGPADIWPLDPLNGAWFRVETNYDHWKPAPKEDDRRTSAIKALNATGQANLSLEALFQILSVVPVYNNFTIYTTVMSAGSPDKYMTRIRNP 6dy7 A 1.9 BS01 HH7 A 1 V48 S49 S91 F133 S175 Y260 C261 F263 L321 V18 S19 S61 F103 S145 Y230 C231 F233 L291 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=66200nM remove_due_to_license_issue P61964 30865883 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6dya A 2.56 BS01 HHM A 1 S49 F133 F149 Y191 Y260 C261 F263 I305 S20 F104 F120 Y162 Y231 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue P61964 30865883 401 PVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6dyn A 2.102 BS01 HSM A 1 E696 T826 T828 E32 T162 T164 6.3.2.- Kd=638.9uM remove_due_to_license_issue Q9VDC6 30705105 901 MLKMEAVPLRLEHRQEVIDIIVASFYNKADLEQWLKPGVLRTDYSDILNDIWNVLVERDLSFVVYDTNTDRIIGTALNFDARNEPEVDIKSKLLIVFEFLEFCEGPIRDNYLPKGLNQILHSFMMGTAEKLNPRENIACMHFMEHEVLRVAREKQFAGIFTTNTSPLTQQLADVYHYKTLLNFQVNEYVHSDGSRPFGDAPDEQRAIVHWKEV 6dyo A 2.84 BS01 LDP A 1 E696 V760 L764 F787 E32 V96 L100 F123 6.3.2.- remove_due_to_license_issue Q9VDC6 30705105 901 MLKMEAVPLRLEHRQEVIDIIVASFYNKADLEQWLKPGVLRTDYSDILNDIWNVLVERDLSFVVYDTNTDRIIGTALNFDARNEPEVDIKSKLLIVFEFLEFCEGPIRDNYLPKGLNQILHSFMMGTAEKLNPRENIACMHFMEHEVLRVAREKQFAGIFTTNTSPLTQQLADVYHYKTLLNFQVNEYVHSDGSRPFGDAPDEQRAIVHWKEV 6dyr A 2.45 BS01 HJD A 1 F689 E696 Y708 V760 L764 F787 M788 M789 T825 N827 F25 E32 Y44 V96 L100 F123 M124 M125 T161 N163 6.3.2.- Kd=218.6uM remove_due_to_license_issue Q9VDC6 30705105 901 MLKMEAVPLRLEHRQEVIDIIVASFYNKADLEQWLKPGVLRTDYSDILNDIWNVLVERDLSFVVYDTNTDRIIGTALNFDARNEPEVDIKSKLLIVFEFLEFCEGPIRDNYLPKGLNQILHSFMMGTAEKLNPRENIACMHFMEHEVLRVAREKQFAGIFTTNTSPLTQQLADVYHYKTLLNFQVNEYVHSDGSRPFGDAPDEQRAIVHWKEV 6dys A 2.3 BS01 HJ1 A 1 F689 E696 V760 L764 F787 M788 M789 T825 T826 N827 F25 E32 V96 L100 F123 M124 M125 T161 T162 N163 6.3.2.- Kd=56.4uM remove_due_to_license_issue Q9VDC6 30705105 902 MLKMEAVPLRLEHRQEVIDIIVASFYNKADLEQWLKPGVLRTDYSDILNDIWNVLVERDLSFVVYDTNTDRIIGTALNFDARNEPEVDIKSKLLIVFEFLEFCEGPIRDNYLPKGLNQILHSFMMGTAEKLNPRENIACMHFMEHEVLRVAREKQFAGIFTTNTSPLTQQLADVYHYKTLLNFQVNEYVHSDGSRPFGDAPDEQRAIVHWKEV 6dyu A 1.6 BS01 OS2 A 1 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 I54 V80 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.055nM remove_due_to_license_issue Q9ZMY2 30860833 302 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyu B 1.6 BS01 OS2 B 1 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 I54 V80 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.055nM remove_due_to_license_issue Q9ZMY2 30860833 309 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyv A 1.62 BS01 OS3 A 1 M10 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 M12 I54 V80 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.026nM remove_due_to_license_issue Q9ZMY2 30860833 306 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyv B 1.62 BS01 OS3 B 1 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 I54 V80 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.026nM remove_due_to_license_issue Q9ZMY2 30860833 305 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyw A 1.45 BS01 OS5 A 1 I52 A79 G80 F153 V154 E173 M174 E175 D198 F208 I54 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.036nM remove_due_to_license_issue Q9ZMY2 30860833 308 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyw B 1.45 BS01 OS5 B 1 I52 A79 G80 F153 V154 E173 M174 E175 D198 F208 I54 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.036nM remove_due_to_license_issue Q9ZMY2 30860833 307 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyy A 1.61 BS01 OS6 A 1 I52 A79 G80 F153 V154 E173 M174 E175 D198 F208 I54 A81 G82 F155 V156 E175 M176 E177 D200 F210 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.028nM remove_due_to_license_issue Q9ZMY2 30860833 303 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyy A 1.61 BS02 OS6 B 1 F107 H109 P115 F109 H111 P117 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.028nM remove_due_to_license_issue Q9ZMY2 30860833 305 QGVQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyy B 1.61 BS01 OS6 A 1 H109 P115 E116 H109 P115 E116 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.028nM remove_due_to_license_issue Q9ZMY2 30860833 303 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyy B 1.61 BS02 OS6 B 1 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 I52 V78 A79 G80 F153 V154 E173 M174 E175 D198 F208 3.2.2.30,3.2.2.9 0003824,0005829,0008782,0008930,0009086,0009116,0009164,0009234,0016787,0019284,0019509,0102246 Kd=0.028nM remove_due_to_license_issue Q9ZMY2 30860833 305 VQKIGILGAMREEITPILELFGVDFEEIPLGGNVFHKGVYHNKEIIVAYSKIGKVHSTLTTTSMILAFGVQKVLFSGVAGSLVKDLKINDLLVATQLVQHDVDLSAFDHPLGFIPESAIFIETSGSLNALAKKIANEQHIALKEGVIASGDQFVHSKERKEFLVSEFKASAVEMEGASVAFVCQKFGVPCCVLRSISDNADEKAGMSFDEFLEKSAHTSAKFLKSMVDEL 6dyz A 1.62 BS02 OS2 A 1 T18 H65 A94 C95 G96 F177 I194 N195 M196 D220 D222 V236 T10 H57 A86 C87 G88 F169 I186 N187 M188 D212 D214 V228 T18 P41 H65 I67 M68 A94 M196 T197 D220 D222 V233 T10 P33 H57 I59 M60 A86 M188 T189 D212 D214 V225 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Kd=0.63nM remove_due_to_license_issue Kd=0.630000nM Q13126 30860833 307 AVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGRQHTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLP 6dz0 A 1.62 BS02 OS3 A 1 T18 H65 A94 C95 G96 F177 I194 N195 M196 T219 D220 D222 V233 V236 T12 H59 A88 C89 G90 F171 I188 N189 M190 T213 D214 D216 V227 V230 T18 P41 H65 I67 M68 A94 M196 T197 D220 D222 V233 T12 P35 H59 I61 M62 A88 M190 T191 D214 D216 V227 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Kd=0.94nM remove_due_to_license_issue Kd=0.940000nM Q13126 30860833 307 TTAVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGRQHTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLL 6dz2 A 1.99 BS01 OS5 A 1 G16 T18 T92 T93 A94 C95 G96 F177 I194 N195 M196 D220 L240 G8 T10 T81 T82 A83 C84 G85 F166 I183 N184 M185 D209 L229 T18 P41 I67 M68 A94 M196 T197 D220 D222 V233 T10 P33 I56 M57 A83 M185 T186 D209 D211 V222 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Kd=1.4nM remove_due_to_license_issue Kd=1.4nM Q13126 30860833 307 AVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLP 6dz2 C 1.99 BS01 OS5 C 1 T18 A94 C95 G96 F177 I194 N195 M196 D220 D222 V236 L240 T10 A79 C80 G81 F162 I179 N180 M181 D205 D207 V221 L225 T18 P41 I67 M68 A94 M196 T197 D220 D222 V233 T10 P33 I52 M53 A79 M181 T182 D205 D207 V218 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Kd=1.4nM remove_due_to_license_issue Kd=1.4nM Q13126 30860833 308 AVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLP 6dz3 A 1.91 BS01 OS6 A 1 T92 A94 C95 G96 F177 I194 N195 M196 D220 D222 V236 L240 T84 A86 C87 G88 F169 I186 N187 M188 D212 D214 V228 L232 T18 P41 H65 I67 M68 A94 M196 T197 D220 D222 V233 T10 P33 H57 I59 M60 A86 M188 T189 D212 D214 V225 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Kd=1.3nM remove_due_to_license_issue Kd=1.3nM Q13126 30860833 306 AVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGRQHTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLP 6dz3 C 1.91 BS01 OS6 C 1 A94 C95 G96 F177 I194 N195 M196 D220 V236 L237 L240 A86 C87 G88 F169 I186 N187 M188 D212 V228 L229 L232 T18 P41 H65 I67 M68 A94 M196 T197 D220 D222 V233 T10 P33 H57 I59 M60 A86 M188 T189 D212 D214 V225 2.4.2.28 0003824,0004645,0005515,0005634,0005654,0005737,0005829,0006139,0006166,0006738,0009116,0016757,0016763,0017061,0019509,0032259,0033574,0070062 Kd=1.3nM remove_due_to_license_issue Kd=1.3nM Q13126 30860833 307 AVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGRQHTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTLKENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLP 6dzq A 2.25 BS03 HJP A 1 H41 E80 D108 E119 K134 E198 H42 E60 D88 E99 K114 E178 3.1.-.- 0003723,0039694 ic50=0.043uM remove_due_to_license_issue C3W5S0 30351002 203 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERGE 6dzv A 4.2 BS01 HJM A 1 Y95 D98 F335 L337 G338 F341 Y17 D20 F257 L259 G260 F263 ? 0016020 remove_due_to_license_issue P31645 31019304 703 RETWGKKVDFLLSVIGYAVDLGNVWRFPYICYQNGGGAFLLPYTIMAIFGGIPLFYMELALGQYHRNGCISIWRKICPIFKGIGYAICIIAFYIASYYNTIMAWALYYLISSFTDQLPWTSCKNSWNTGNCTNYFSEDNITWTLHSTSPAEEFYTRHVLQIHRSKGLQDLGGISWQLALCIMLIFTVIYFSIWKGVKTSGKVVWVTATFPYIILSVLLVRGATLPGAWRGVLFYLKPNWQKLLETGVWIDAAAQIFFSLGPGFGVLLAFASYNKFNNNCYQDALVTSVVNCMTSFVSGFVIFTVLGYMAEMRNEDVSEVAKDAGPSLLFITYAEAIANMPASTFFAIIFFLMLITLGLDSTFAGLEGVITAVLDEFPHVWAKRRERFVLAVVITCFFGSLVTLTFGGAYVVKLLEEYATGPAVLTVALIEAVAVSWFYGITQFCRDVKEMLGFSPGWFWRICWVAISPLFLLFIICSFLMSPPQLRLFQYNYPYWSIILGYCIGTSSFICIPTYIAYRLIITPGTFKERIIKSITPE 6dzx A 1.678 BS01 MED A 1 Y81 F98 Q99 H100 Y103 N153 R156 N213 N238 Y38 F55 Q56 H57 Y60 N110 R113 N170 N195 ? 0016020 Kd=3.5uM remove_due_to_license_issue C6S9R8 31348565 1001 EIVFGTTVGDFGDMVKEQIQAELEKKGYTVKLVEFTDYVRPNLALAEGELDINVFQHKPYLDDFKKEHNLDITEVFQVPTAPLGLYPGKLKSLEEVKDGSTVSAPNDPSNFARVLVMLDELGWIKLKDGINPLTASKADIAENLKNIKIVELEAAQLPRSRADVDFAVVNGNYAISSGMKLTEALFQEPSFAYVNWSAVKTADKDSQWLKDVTEAYNSDAFKAYAHKRFEGYKSPAAWNE 6dzy A 4.1 BS01 HJM A 1 Y95 A96 D98 I172 A173 Y176 F335 F341 G442 L443 Y17 A18 D20 I94 A95 Y98 F257 F263 G364 L365 ? 0016020 remove_due_to_license_issue P31645 31019304 701 RETWGKKVDFLLSVIGYAVDLGNVWRFPYICYQNGGGAFLLPYTIMAIFGGIPLFYMELALGQYHRNGCISIWRKICPIFKGIGYAICIIAFYIASYYNTIMAWALYYLISSFTDQLPWTSCKNSWNTGNCTNYFSEDNITWTLHSTSPAEEFYTRHVLQIHRSKGLQDLGGISWQLALCIMLIFTVIYFSIWKGVKTSGKVVWVTATFPYIALSVLLVRGATLPGAWRGVLFYLKPNWQKLLETGVWIDAAAQIFFSLGPGFGVLLAFASYNKFNNNCYQDALVTSVVNCMTSFVSGFVIFTVLGYMAEMRNEDVSEVAKDAGPSLLFITYAEAIANMPASTFFAIIFFLMLITLGLDSSFAGLEGVITAVLDEFPHVWAKRRERFVLAVVITCFFGSLVTLTFGGAYVVKLLEEYATGPAVLTVALIEAVAVSWFYGITQFCRDVKEMLGFSPGWFWRICWVAISPLFLLFIIASFLMSPPQLRLFQYNYPYWSIILGYAIGTSSFICIPTYIAYRLIITPGTFKERIIKSITPE 6e05 A 2.5 BS02 CTP A 1 T11 G12 V13 G14 K15 T16 V17 G169 L196 G199 A200 A201 T12 G13 V14 G15 K16 T17 V18 G170 L197 G200 A201 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 30289406 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6e05 B 2.5 BS02 CTP B 1 T11 G12 V13 G14 K15 T16 V17 G169 L196 P197 G199 A201 T12 G13 V14 G15 K16 T17 V18 G170 L197 P198 G200 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 30289406 302 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6e06 A 2.5 BS01 CTP A 1 T11 G12 G14 K15 T16 V17 E108 G169 G199 A200 A201 T12 G13 G15 K16 T17 V18 E109 G170 G200 A201 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 30289406 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLVG 6e06 B 2.5 BS01 CTP B 1 G12 V13 G14 K15 T16 V17 E108 G111 G169 L196 P197 G199 A201 G13 V14 G15 K16 T17 V18 E109 G112 G170 L197 P198 G200 A202 T11 G12 K15 T16 K37 T41 G54 E108 T12 G13 K16 T17 K38 T42 G55 E109 6.3.3.3 0000287,0004141,0005524,0005737,0005829,0009102,0016874,0046872 remove_due_to_license_issue P9WPQ5 30289406 301 GGTILVVTGTGTGVGKTVVCAALASAARQAGIDVAVCKPVQTGTARGDDDLAEVGRLAGVTQLAGLARYPQPMAPAAAAEHAGMALPARDQIVRLIADLDRPGRLTLVEGAGGLLVELAEPGVTLRDVAVDVAAAALVVVTADLGTLNHTKLTLEALAAQQVSCAGLVIGSWPDPPGLVAASNRSALARIAMVRAALPAGAASLDAGDFAAMSAAAFDRNWVAGLV 6e0q A 2.35 BS03 HKD A 1 H41 E80 D108 E119 K134 E198 H42 E60 D88 E99 K114 E178 3.1.-.- 0003723,0039694 ic50=8nM remove_due_to_license_issue C3W5S0 30351002 203 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERGE 6e0r A 2.303 BS01 HKJ A 1 L1122 V1130 M1199 A1200 N1254 L1256 G1269 L24 V28 M90 A91 N145 L147 G160 D1249 R1253 N1254 D1270 D140 R144 N145 D161 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=20nM remove_due_to_license_issue IC50=20nM Q9UM73 31009559 1500 AGKTSSISDLKEVPRKNITLIRGLGHGVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPI 6e13 A 2.349 BS03 HKS A 1 A11 Q16 M229 N271 A12 Q17 M230 N272 1.-.-.- 0018189 remove_due_to_license_issue Q88QV5 30811189 404 MMYIQVLGSAAAGGFPQWNCNCVNCKGYRDGTLKATARTQSSIALSDDGVHWILCNASPDIRAQLQAFAPMQPARALRDTGINAIVLLDSQIDHTTGLLSLREGCPHQVWCTDMVHQDLTTGFPLFNMLSHWNGGLQWNRIELEGSFVIDACPNLKFTPFPLRSAAPPYSPHRFDPHPGDNLGLMVEDTRTGGKLFYAPGLGQVDEKLLAMMHGADCLLVDGTLWEDDEMQRRGVGTRTGREMGHLAQNGPGGTLEVLDGFPRQRKVLIHINNTNPILDENSPERAEVLRRGVEVAFDGMSIELLEHH 6e1a A 3.1 BS01 HL7 A 1 S178 H181 F238 C241 A242 Y276 M278 Y319 M322 Y323 G326 W341 E363 S174 H177 F234 C237 A238 Y272 M274 Y315 M318 Y319 G322 W337 E359 ? 0000122,0000165,0000400,0000403,0000781,0000785,0000976,0001933,0002076,0003677,0003682,0003690,0005515,0005634,0005654,0005737,0005788,0005829,0006281,0006325,0006357,0006974,0008285,0009411,0010332,0016363,0017053,0030511,0030674,0032154,0032991,0035097,0043433,0044665,0045064,0045668,0045736,0045786,0045815,0045892,0045944,0046329,0051219,0070412,0071339 remove_due_to_license_issue Ki=<1.000000nM, IC50=5.0nM, Kd=1400nM O00255 31244110 701 GLKAAQKTLFPLRSIDDVVRLFAAELGREEPDLVLLSLVLGFVEHFLAVNRVIPTNVPELTFQPSPAPDGLTYFPVADLSIIAALYARFTAQIRGAVDLSLYPREGGVSSRELVKKVSDVIWNSLSRSYFKDRAHIQSLFSFITGTKLDSSGVAFAVVGACQALGLRDVHLALSEDHAWVVFGPNGEQTAEVTWHGKGNEDRRGQTVNAGVAERSWLYLKGSYMRCDRKMEVAFMVCAINPSIDLHTDSLELLQLQQKLLWLLYDLGHLERYPMALGNLADLEELEPTPGRPDPLTLYHKGIASAKTYYRDEHIYPYMYLAGYHCRNRNVREALQAWADTATVIQDYNYCREDEEIYKEFFEVANDVIPNLLKEAASLLEASALQDPECFAHLLRFYDGICKWEEGSPTPVLHVGWATFLVQSLGRFEGQVRQKVRIVSGTVAGTARGPVLTFQSEKMKGMKELLVATKINSSAIKLQLTA 6e1y A 1.219 BS01 HLM A 1 S49 S91 F133 F149 S175 Y260 C261 F263 I305 S18 S60 F102 F118 S144 Y225 C226 F228 I270 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=22nM remove_due_to_license_issue Ki=30.8nM P61964 30865883 401 KPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6e1z A 1.1 BS01 HLP A 1 S91 F133 Y260 C261 F263 I305 S64 F106 Y233 C234 F236 I278 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=150000nM remove_due_to_license_issue P61964 30865883 401 PTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6e22 A 1.6 BS01 HLS A 1 S28 S70 F112 F128 S154 Y170 Y239 C240 F242 S19 S61 F103 F119 S145 Y161 Y230 C231 F233 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=1.3nM remove_due_to_license_issue Ki=1.33nM P61964 30865883 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6e23 A 1.66 BS01 HLJ A 1 S49 A65 G89 S91 D92 F133 F149 Y260 C261 F263 I305 S18 A34 G58 S60 D61 F102 F118 Y225 C226 F228 I270 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=0.1nM remove_due_to_license_issue Ki=<0.100nM P61964 30865883 401 KPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6e2m A 2.253 BS01 KK7 A 1 L686 K709 M754 E755 Q756 V757 G760 L810 S821 D822 L17 K40 M79 E80 Q81 V82 G85 L135 S146 D147 D803 K805 D807 N808 D822 T842 D128 K130 D132 N133 D147 T164 2.7.11.25 0004672,0005524,0006468 ic50=2200nM remove_due_to_license_issue Q99683 30024858 1001 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPYSQPLHEEIALHKHLKHKNIVQYLGSFSENFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAPCTETFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6e2m B 2.253 BS01 KK7 B 1 L686 K709 M754 E755 Q756 V757 L810 S821 D822 L16 K39 M77 E78 Q79 V80 L133 S144 D145 D803 K805 D807 N808 D822 T842 D126 K128 D130 N131 D145 T155 2.7.11.25 0004672,0005524,0006468 ic50=2200nM remove_due_to_license_issue Q99683 30024858 1001 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTGTLQYMAPEIIDKGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKV 6e2n A 2.098 BS01 KK8 A 1 L686 A707 K709 M754 E755 Q756 V757 G759 G760 D807 L810 D822 L17 A38 K40 M82 E83 Q84 V85 G87 G88 D135 L138 D150 D803 K805 D807 N808 D822 T842 D131 K133 D135 N136 D150 T167 2.7.11.25 0004672,0005524,0006468 ic50=12.5nM remove_due_to_license_issue Q99683 30024858 1001 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGCTETFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6e2n B 2.098 BS01 KK8 B 1 L686 A707 K709 M754 E755 Q756 V757 G759 G760 D807 L810 D822 L17 A38 K40 M80 E81 Q82 V83 G85 G86 D133 L136 D148 D803 K805 D807 N808 D822 T842 D129 K131 D133 N134 D148 T158 2.7.11.25 0004672,0005524,0006468 ic50=12.5nM remove_due_to_license_issue Q99683 30024858 1001 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPESQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTGTLQYMAPEIIDYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6e2o A 2.389 BS01 S0L A 1 L686 A707 K709 M754 E755 Q756 V757 P758 G759 D807 L810 D822 L17 A38 K40 M83 E84 Q85 V86 P87 G88 D136 L139 D151 D803 K805 D807 N808 D822 T842 D132 K134 D136 N137 D151 T167 2.7.11.25 0004672,0005524,0006468 Kd=2.9nM remove_due_to_license_issue Q99683 30024858 1001 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPESRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLACTETFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6e2o B 2.389 BS01 S0L B 1 A707 K709 M754 E755 Q756 V757 G759 D807 L810 S821 D822 A37 K39 M79 E80 Q81 V82 G84 D132 L135 S146 D147 D803 K805 D807 N808 D822 T842 D128 K130 D132 N133 D147 T157 2.7.11.25 0004672,0005524,0006468 Kd=2.9nM remove_due_to_license_issue Q99683 30024858 1001 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPESQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLTGTLQYMAPEIIDKYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6e3g A 2.1 BS02 HOJ A 1 W317 C320 L324 M358 V361 M365 A368 F377 F378 E379 F388 I400 H479 W55 C58 L62 M96 V99 M103 A106 F115 F116 E117 F126 I138 H217 ? 0003677,0004879,0005634,0006355 ic50=44nM remove_due_to_license_issue IC50=44nM, EC50=53nM P51449 30652849 602 PYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 6e3m A 2.65 BS03 HOG A 1 H41 E80 D108 E119 K134 H43 E63 D91 E102 K117 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 904 MAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 6e3n A 3.19 BS03 HNS A 1 H41 E80 D108 E119 K134 H42 E62 D90 E101 K116 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 903 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 6e3o A 3.19 BS03 HNY A 1 K34 H41 E80 D108 E119 K134 K35 H42 E62 D90 E101 K116 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 903 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 6e3p A 2.8 BS03 HO1 A 1 H41 E80 D108 E119 Y130 K134 E195 R196 H42 E60 D88 E99 Y110 K114 E173 R174 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 903 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 6e3p A 2.8 BS04 HO1 A 2 K34 A37 I38 H41 E80 R124 K35 A38 I39 H42 E60 R104 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 904 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 6e3z A 1.94 BS01 HRV A 1 Q12 G13 L30 D32 Y71 D228 G230 T232 Q17 G18 L35 D37 Y76 D224 G226 T228 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue P56817 401 TGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6e4a A 1.26 BS01 HRY A 1 W81 P82 V87 L92 N140 I146 W40 P41 V46 L51 N99 I105 ? Kd=44nM remove_due_to_license_issue Kd=44nM O60885 30268702 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 6e4c A 2.35 BS03 HRJ A 1 K34 H41 E80 D108 E119 K134 K36 H43 E61 D89 E100 K115 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 903 MAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSER 6e4f A 1.15 BS01 HRA A 1 L408 A428 K430 M449 I472 T474 M477 L528 D539 F540 L20 A40 K42 M61 I84 T86 M89 L140 D151 F152 D521 R525 N526 D539 D133 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.85nM remove_due_to_license_issue IC50=0.850nM Q06187 30093506 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 6e4t A 3.4 BS01 HTV A 1 K31 I46 D88 K23 I38 D80 D139 K141 E143 N144 D157 S176 D131 K133 E135 N136 D149 S168 2.7.11.1,2.7.11.26,2.7.11.31 0004672,0004679,0005524,0006468 remove_due_to_license_issue P54645 30036059 601 GRVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFKWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDDSHTIEFFEMCANLIKILAQ 6e4t B 3.4 BS01 HTV A 1 R83 T106 S108 V113 R5 T28 S30 V35 ? remove_due_to_license_issue P80386 30036059 601 PTVFRWTGGGKEVYLSGSFNNWSKLPLTRSQNNFVAILDLPEGEHQYKFFVDGQWTHDPSEPIVTSQLGTVNNIIQVKKTDFEVFDALMVDSQKAPPILPPHLLQVILNKSCDPALLPEPNHVMLNHLYALSIKDGVMVLSATHRYKKKYVTTLLYKPI 6e4u A 3.27 BS02 HU7 A 1 L18 K29 K31 I46 D88 L10 K21 K23 I38 D80 D139 K141 E143 N144 D157 S176 D131 K133 E135 N136 D149 S168 2.7.11.1,2.7.11.26,2.7.11.31 0004672,0004679,0005524,0006468 remove_due_to_license_issue P54645 30036059 602 GRVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFPEKWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDDPGSHTIEFFEMCANLIKILAQ 6e4v A 2.0 BS01 HWS A 1 R117 L119 R142 W143 W275 Y341 D343 N373 W416 R60 L62 R85 W86 W218 Y284 D286 N316 W359 ? 0006826,0006879,0009279,0015092,0015343,0015344,0015687,0015891,0016020,0033214,0038023,0042928,0044718,0072711,1902495 remove_due_to_license_issue P16869 31098021 806 NDYSVTSTSAGTKMQMTQRDIPQSVTIVSQQRMEDQQLQTLGEVMENTLGISKSQADSDRALYYSRGFQIDNYMVDGIPTYFESRWNLGDALSDMALFERVEVVRGATGLMTGTGNPSAAINMVRKHATSREFKGDVSAEYGSWNKERYVADLQSPLTEDGKIRARIVGGYQNNDSWLDRYNSEKTFFSGIVDADLGDLTTLSAGYEYQRIDVNSPTWGGLPRWNTDGSSNSYDRARSTAPDWAYNDKEINKVFMTLKQQFADTWQATLNATHSEVEFDSKMMYVDAYVNKADGMLVGPYSNYGPGFDYVGGTGWNSGKRKVDALDLFADGSYELFGRQHNLMFGGSYSKQNNRYFSSWANIFPDEIGSFYNFNGNFPQTDWSPQSLAQDDTTHMKSLYAATRVTLADPLHLILGARYTNWRVDTLTYSMEKNHTTPYAGLVFDINDNWSTYASYTSIFQPQNDRDSSGKYLAPITGNNYELGLKSDWMNSRLTTTLAIFRIEQDNVAQSTGTPIPGSNGETAYKAVDGTVSKGVEFELNGAITDNWQLTFGATRYIAEDNEGNAVNPNLPRTTVKMFTSYRLPVMPELTVGGGVNWQNRVYTDTVTPYGTFRAEQGSYALVDLFTRYQVTKNFSLQGNVNNLFDKTYDTNVEGSIVYGTPRNFSITGTYQF 6e4w A 3.35 BS02 HUG A 1 L18 G19 K31 I46 D88 L10 G11 K23 I38 D80 D139 K141 E143 N144 D157 S176 D131 K133 E135 N136 D149 S168 2.7.11.1,2.7.11.26,2.7.11.31 0004672,0004679,0005524,0006468 remove_due_to_license_issue P54645 30036059 602 GRVKIGHYILGDTLGVGTFGKVKVGKHELTGHKVAVKILNRQKIRSLDVVGKIRREIQNLKLFRHPHIIKLYQVISTPSDIFMVMEYVSGGELFDYICKNGRLDEKESRRLFQQILSGVDYCHRHMVVHRDLKPENVLLDAHMNAKIADFGLSNMMSDGEFLRTSCGSPNYAAPEVISGRLYAGPEVDIWSSGVILYALLCGTLPFDDDHVPTLFKKICDGIFYTPQYLNPSVISLLKHMLQVDPMKRATIKDIREHEWFKQDLPKYLFKWHLGIRSQSRPNDIMAEVCRAIKQLDYEWKVVNPYYLRVRRKNPVTSTFSKMSLQLYQVDSRTYLLDFRSIDDSHTIEFFEMCANLIKILAQ 6e59 A 3.4 BS01 L76 A 1 N109 P112 I113 V116 Q165 E193 H197 I204 F264 F268 N82 P85 I86 V89 Q138 E166 H170 I177 F423 F427 ? 0004930,0004995,0005886,0007186,0016020 remove_due_to_license_issue P25103,Q9V2J8 30538204 2001 PAWQIVLWAAAYTVIVVTSVVGNVVVMWIILAHKRMRTVTNYFLVNLAFAEASMAAFNTVVNFTYAVHNEWYYGLFYCKFHNFFPIAAVFASIYSMTAVAFDRYMAIIHPLQPRLSATATKVVICVIWVLALLLAFPQGYYSTTETMPSRVVCMIEWPEHPNKIYEKVYHICVTVLIYFLPLLVIGYAYTVVGITLWASEGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSEQVSAKRKVVKMMIVVVCTFAICWLPFHIFFLLPYINPDLYLKKFIQQVYLAIMWLAMSSTMYNPIIYCCLNDRFRLGFKHAF 6e5b K 2.77 BS01 HUJ K 1 T1 A20 S21 K33 G47 C48 A49 T1 A20 S21 K33 G47 C48 A49 T1 D17 R19 K33 G47 S130 D167 S170 T1 D17 R19 K33 G47 S130 D167 S170 3.4.25.1 0000502,0002376,0004175,0004298,0005515,0005634,0005654,0005737,0005829,0005839,0006508,0019774,0019882,0030154,0043161,0045444,0051603,0052548,0070062,1990111 remove_due_to_license_issue P28062 31283222 901 TTTLAFKFQHGVIAAVDSRASAGSYISALRVNKVIEINPYLLGTMSGCAADCQYWERLLAKECRLYYLRNGERISVSAASKLLSNMMCQYRGMGLSMGSMICGWDKKGPGLYYVDEHGTRLSGNMFSTGSGNTYAYGVMDSGYRPNLSPEEAYDLGRRAIAYATHRDSYSGGVVNMYHMKEDGWVKVESTDVSDLLHQYREAN 6e5g B 2.43 BS01 HUY B 1 F233 A235 V329 K357 S377 P378 C380 L383 I408 Q410 F16 A18 V91 K119 S139 P140 C142 L145 I170 Q172 ? remove_due_to_license_issue Q15562 30581134 501 WQARGLGTARLQLVEFSAFVEPPDAVDSYQRHLFVHISQPPLESVDVRQIYDKFPEKKGGLRELYDRGPPHAFFLVKFWADLNWSGGFYGVSSQYESLEHMTLTCSSKVCSFGKQVVEKVETERAQLEDGRFVYRLLRSPMCEYLVNFLHKLRQLPERYMMNSVLENFTILQVVTNRDTQELLLCTAYVFEVSTSERGAQHHIYRLVR 6e5l A 1.17 BS01 HVD A 1 F16 A33 L36 P38 F57 R58 I77 F16 A33 L36 P38 F57 R58 I77 ? 0002138,0005501,0005504,0005515,0005634,0005654,0005737,0005811,0005829,0006776,0008289,0015908,0016918,0019841,0055088,1904768 Ki=76.3nM remove_due_to_license_issue P09455 30721022 201 PVDFTGYWKMLVNENFEEYLRALDVNVALRKIANLLKPDKEIVQDGDHMIIRTLSTFRNYIMDFQVGKEFEEDLTGIDDRKCMTTVSWDGDKLQCVQKGEKEGRGWTQWIEGDELHLEMRVEGVVCKQVFKKVQHHHHHH 6e5s A 2.061 BS01 RET C 1 F16 Q38 K40 D51 F16 Q38 K40 D51 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 31557439 201 TRDQNGTWEMESNENFEGYMKALDIDFATRKIAVRLTQTKVIDQDGDNFKDKTTSTFRNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 6e5s C 2.061 BS01 RET C 1 L77 W106 K108 L77 W106 K108 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 31557439 201 TRDQNGTWEMESNENFEGYMKALDIDFATRKIAVRLTQTKVIDQDGDNFKDKTTSTFRNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 6e5t A 1.55 BS01 HVJ A 1 F16 A33 P38 F57 R58 F16 A33 P38 F57 R58 ? 0002138,0005501,0005504,0005515,0005634,0005654,0005737,0005811,0005829,0006776,0008289,0015908,0016918,0019841,0055088,1904768 Ki=236.3nM remove_due_to_license_issue P09455 30721022 201 PVDFTGYWKMLVNENFEEYLRALDVNVALRKIANLLKPDKEIVQDGDHMIIRTLSTFRNYIMDFQVGKEFEEDLTGIDDRKCMTTVSWDGDKLQCVQKGEKEGRGWTQWIEGDELHLEMRVEGVVCKQVFKKVQHHHHH 6e6j A 2.44 BS01 HWV A 1 W370 P371 V376 D377 L381 N429 V435 W25 P26 V31 D32 L36 N84 V90 ? remove_due_to_license_issue Ki=4.6nM P25440 31969702 501 HMEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMP 6e6v A 2.25 BS03 HWA A 1 H41 E80 D108 E119 K134 E198 H43 E61 D89 E100 K115 E179 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 203 MAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERGE 6e6w A 2.35 BS03 HWJ A 1 K34 H41 E80 D108 E119 K134 K36 H43 E61 D89 E100 K115 3.1.-.- 0003723,0039694 remove_due_to_license_issue C3W5S0 31536340 203 MAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFGHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 6e7j A 1.3 BS01 HWY A 1 D25 G27 A28 D29 G48 D25 G27 A28 D29 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.33nM remove_due_to_license_issue P04585 30354121 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6e7j B 1.3 BS01 HWY A 1 R8 D25 A28 D30 V82 R8 D25 A28 D30 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30354121 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6e7m B 2.7 BS01 RET D 1 Q38 K40 Q38 K40 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 31557439 203 TRDQNGTWEMESNENFEGYMKALDIDFCTRKIAVRLTQTKVIDQDGDNFKDKTTSTFRNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 6e7m D 2.7 BS01 RET D 1 L77 W106 K108 L77 W106 K108 ? 0005501,0005504,0005634,0005737,0005829,0006776,0008289,0008544,0015908,0016918,0019841 remove_due_to_license_issue P50120 31557439 203 TRDQNGTWEMESNENFEGYMKALDIDFCTRKIAVRLTQTKVIDQDGDNFKDKTTSTFRNYDVDFTVGVEFDEYTKSLDNRHVKALVTWEGDVLVCVQKGEKENRGWKKWIEGDKLYLELTCGDQVCRQVFKKK 6e7r A 2.1 BS01 HYS B 1 Y109 F113 S132 I133 L135 Y84 F88 S107 I108 L110 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 30659174 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPAHLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 6e7r B 2.1 BS01 HYS B 1 P78 Q110 Y175 F176 P177 M207 S208 E236 P47 Q79 Y144 F145 P146 M176 S177 E205 ? remove_due_to_license_issue Q00960 30659174 503 PPSIGIAVILVGTSDEVAIKDAHEKDDFHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPRM 6e7s A 2.72 BS01 HZ4 B 1 Y109 F113 S132 L135 Y84 F88 S107 L110 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPAHLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 6e7s B 2.72 BS01 HZ4 B 1 P78 Q110 F114 Y175 F176 M207 S208 E236 P47 Q79 F83 Y144 F145 M176 S177 E205 ? remove_due_to_license_issue Q00960 503 PPSIGIAVILVGTSDEVAIKDAHEKDDFHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPRM 6e7t A 2.31 BS01 HYY B 1 Y109 F113 S132 L135 Y82 F86 S105 L108 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 506 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 6e7t B 2.31 BS01 HYY B 1 P78 Q110 Y175 F176 M207 S208 E236 P41 Q73 Y138 F139 M170 S171 E199 ? remove_due_to_license_issue Q00960 506 PPSIGIAVILVGTSDEVAIKDAHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPR 6e7u A 2.27 BS01 HX7 B 1 Y109 F113 S132 I133 L135 Y83 F87 S106 I107 L109 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPALTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGGET 6e7u B 2.27 BS01 HX7 B 1 P78 Q110 I111 Y175 F176 M207 S208 E236 P43 Q75 I76 Y140 F141 M172 S173 E201 ? remove_due_to_license_issue Q00960 503 PPSIGIAVILVGTSDEVAIKDAHFHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPRM 6e7v A 2.6 BS01 T88 B 1 Y109 T110 F113 S132 L135 Y84 T85 F88 S107 L110 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 502 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPAHLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 6e7v B 2.6 BS01 T88 B 1 P78 Q110 F114 Y175 F176 P177 D206 M207 S208 E236 P44 Q76 F80 Y141 F142 P143 D172 M173 S174 E202 ? remove_due_to_license_issue Q00960 502 PPSIGIAVILVGTSDEVAIKDAHDFHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPRM 6e7w A 2.67 BS01 HXM B 1 Y109 F113 S132 I133 L135 Y84 F88 S107 I108 L110 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPAHLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 6e7w B 2.67 BS01 HXM B 1 P78 Q110 I111 Y175 F176 P177 M207 S208 E236 P42 Q74 I75 Y139 F140 P141 M171 S172 E200 ? remove_due_to_license_issue Q00960 503 PPSIGIAVILVGTSDEVAIKDAHHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPRM 6e7x A 2.58 BS01 T97 B 1 Y109 F113 S132 I133 L135 Y84 F88 S107 I108 L110 ? 0004930,0007186,0016020 remove_due_to_license_issue A0A1L8F5J9 503 DPKIVNIGAVLSTKKHEQIFREAVNQANKRHFTRKIQLQATSVTHRPNAIQMALSVCEDLISSQVYAILVSHPPAHLTPTPISYTAGFYRIPVIGLTTRMSIYSDKSIHLSFLRTVPPYSHQALVWFEMMRLFNWNHVILIVSDDHEGRAAQKKLETLLEGGPKADKVLQFEPGTKNLTALLLEAKELEARVIILSASEDDATAVYKSAAMLDMTGAGYVWLVGEREISGSALRYAPDGIIGLQLINGKNESAHISDAVAVVAQAIHELFEMENITDPPRGCVGNTNIWKTGPLFKRVLMSSKYPDGVTGRIEFNEDGDRKFAQYSIMNLQNRKLVQVGIFNGSYIIQNDRKIIWPGG 6e7x B 2.58 BS01 T97 B 1 P78 Q110 Y175 F176 P177 M207 S208 E236 P47 Q79 Y144 F145 P146 M176 S177 E205 ? remove_due_to_license_issue Q00960 503 PPSIGIAVILVGTSDEVAIKDAHEKDDFHHLSVVPRVELVAMNETDPKSIITRICDLMSDRKIQGVVFADDTDQEAIAQILDFISAQTLTPILGIHGGSSMIMADKDESSMFFQFGPSIEQQASVMLNIMEEYDWYIFSIVTTYFPGYQDFVNKIRSTIENSFVGWELEEVLLLDMSLDDGDSKIQNQLKKLQSPIILLYCTKEEATYIFEVANSVGLTGYGYTWIVPSLVAGDTDTVPSEFPTGLISVSYDEWDYGLPARVRDGIAIITTAASDMLSEHSFIPEPKSSCYNTHEKRIYQSNMLNRYLINVTFEGRDLSFSEDGYQMHPKLVIILLNKERKWERVGKWKDKSLQMKYYVWPRM 6e8x A 1.6 BS02 J0A A 1 H94 V135 L198 T199 T200 H91 V131 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.07uM remove_due_to_license_issue P00918 30721041 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6e91 A 1.8 BS02 J04 A 1 Q92 H94 H119 V131 L198 T199 T200 P202 Q89 H91 H116 V127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.08uM remove_due_to_license_issue P00918 30721041 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6e92 A 1.772 BS02 HZY A 1 L91 H94 H119 V131 G132 L198 T199 T200 L88 H91 H116 V127 G128 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.002uM remove_due_to_license_issue P00918 30721041 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6e93 A 1.747 BS01 dna C 0 H1028 C1031 R1045 F1047 N1052 H1056 I1059 K1073 H1084 Y1105 T1108 N1111 R1115 H20 C23 R37 F39 N44 H48 I51 K65 H76 Y97 T100 N103 R107 ? remove_due_to_license_issue Q8NAP3 30355731 19 ~ 36 PYACELCAKQFQSPSTLKMHMRCHTGEKPYQCKTCGRCFSVQGNLQKHERIHLGLKEFVCQYCNKAFTLNETLKIHERIHTGEKRYHCQFCFQRFLYLSTKRNHEQRHIREH 6e93 A 1.747 BS02 dna D 0 Y1010 S1021 P1022 S1023 K1055 E1079 R1093 Y2 S13 P14 S15 K47 E71 R85 ? remove_due_to_license_issue Q8NAP3 30355731 1 ~ 18 PYACELCAKQFQSPSTLKMHMRCHTGEKPYQCKTCGRCFSVQGNLQKHERIHLGLKEFVCQYCNKAFTLNETLKIHERIHTGEKRYHCQFCFQRFLYLSTKRNHEQRHIREH 6e94 A 1.594 BS01 dna C 0 K1017 H1028 C1031 R1045 F1047 N1052 R1055 H1056 I1059 K1073 H1084 I1087 Y1105 T1108 N1111 R1115 K9 H20 C23 R37 F39 N44 R47 H48 I51 K65 H76 I79 Y97 T100 N103 R107 ? remove_due_to_license_issue Q8NAP3 30355731 19 ~ 36 PYACELCAKQFQSPSTLKMHMRCHTGEKPYQCKTCGRCFSVQGNLQRHERIHLGLKEFVCQYCNKAFTLNETLKIHERIHTGEKRYHCQFCFQRFLYLSTKRNHEQRHIRE 6e94 A 1.594 BS02 dna D 0 Y1010 P1022 S1023 R1055 E1079 R1093 Y1094 Y2 P14 S15 R47 E71 R85 Y86 ? remove_due_to_license_issue Q8NAP3 30355731 1 ~ 18 PYACELCAKQFQSPSTLKMHMRCHTGEKPYQCKTCGRCFSVQGNLQRHERIHLGLKEFVCQYCNKAFTLNETLKIHERIHTGEKRYHCQFCFQRFLYLSTKRNHEQRHIRE 6e99 A 1.88 BS02 J0G A 1 G53 F55 G56 V58 A71 K73 L75 E128 E171 L174 T184 D185 G35 F37 G38 V40 A53 K55 L57 E110 E153 L156 T166 D167 D167 K169 N172 D185 T202 D149 K151 N154 D167 T184 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 ic50=1uM remove_due_to_license_issue P00517 30384606 601 FLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 6e9a A 1.22 BS01 J0S B 1 D25 G27 A28 D30 P81 V82 D25 G27 A28 D30 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P04585 30354121 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6e9a B 1.22 BS01 J0S B 1 D25 G27 D29 G48 G49 I50 D25 G27 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.0012nM remove_due_to_license_issue P04585 30354121 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6e9l A 2.8 BS02 J0P A 1 G53 S54 F55 G56 V58 A71 K73 V124 L174 T184 D185 G36 S37 F38 G39 V41 A54 K56 V107 L157 T167 D168 D167 K169 N172 D185 T202 D150 K152 N155 D168 T185 2.7.11.11 0000287,0001669,0001707,0001843,0004672,0004674,0004691,0004712,0005515,0005524,0005634,0005737,0005739,0005813,0005829,0005886,0005930,0005952,0006397,0006468,0006611,0007165,0007189,0007193,0016607,0018105,0019901,0019904,0030145,0031594,0031625,0032024,0034237,0034605,0036126,0044853,0045542,0045667,0045722,0045879,0046827,0048240,0048471,0050804,0051726,0061136,0070417,0070613,0071333,0071374,0071377,0097546,0098794,0098978,0099170,0106310,1904262,1904539,1990044,2000810 remove_due_to_license_issue P00517 30384606 401 EFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 6e9w A 2.96 BS01 J0P A 1 I82 G85 A86 F87 G88 V90 A103 K105 L107 Y155 M156 D216 I74 G77 A78 F79 G80 V82 A95 K97 L99 Y147 M148 D208 D198 K200 N203 D216 T237 D190 K192 N195 D208 T229 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=450nM Q13464 30384606 501 TRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLTFPIPKAFVGNQLPFVGFTYYSNRR 6ea1 A 1.815 BS02 J0Y A 1 T305 Q317 E319 A320 V459 G460 A461 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=257nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6ea2 A 1.35 BS02 J1G A 1 T305 Q317 E319 A320 V459 G460 A461 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=285nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6eaa A 1.65 BS02 J1V A 1 T305 Q317 E319 A320 V459 G460 A461 R489 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 R294 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=818nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6eab A 1.85 BS02 J2D A 1 T305 Q317 E319 A320 V459 G460 A461 R489 V493 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 R294 V298 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=431nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6eb1 A 2.2 BS01 J3M A 1 Q95 L102 T124 T125 A129 W132 Q40 L47 T69 T70 A74 W77 ? 0003676,0015074 ic50=4.65uM remove_due_to_license_issue IC50=4650nM F2WR52 30783506 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEFGISMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRYSAGERIVDIIATD 6eb2 A 2.493 BS01 J3P A 1 Q95 L102 T124 T125 A128 A129 W132 Q40 L47 T69 T70 A73 A74 W77 ? 0003676,0015074 ic50=0.48uM remove_due_to_license_issue IC50=23400nM, EC50=<1790nM F2WR52 30783506 301 CSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRGYSAGERIVDIIATDI 6ebe A 1.88 BS02 J3V A 1 A65 Q92 H94 H96 F131 L198 T199 A62 Q89 H91 H93 F127 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.2uM remove_due_to_license_issue P00918 30433782 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ebw A 2.455 BS01 J3Y A 1 A1148 L1196 M1199 A1200 G1202 N1254 L1256 G1269 A42 L90 M93 A94 G96 N146 L148 G161 D1249 R1253 N1254 D1270 D141 R145 N146 D162 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=2.5nM remove_due_to_license_issue Q9UM73 31009559 1500 YCFTSSISDLKEVPRKNITLIRGLGHFGEVYEGQVSSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPI 6ecz A 2.21 BS02 J4D A 1 H64 N67 Q92 H94 H96 L198 T199 P202 H61 N64 Q89 H91 H93 L194 T195 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.27uM remove_due_to_license_issue P00918 30433782 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ed6 A 2.86 BS01 J0P A 1 I98 G101 F103 G104 V106 A119 K121 L123 M169 Y171 M172 L221 D232 I72 G75 F77 G78 V80 A93 K95 L97 M143 Y145 M146 L195 D206 D214 K216 N219 D232 T253 D188 K190 N193 D206 T227 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=37nM O75116 30384606 501 QRKLEALIRDPRSPINVESLLDGLNSLVLDLDFPALRKNKNIDNFLNRYEKIVKKIRGLQMKAEDYDVVKVIGRGAFGEVQLVRHKASQKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWAKFYTAEVVLALDAIHSMGLIHRDVKPDNMLLDKHGHLKLADFGTCMKMDETGMVHCDTAVGTPDYISPEVLKSQFYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMDHKNSLCFPEDAEISKHAKNLICAFLTDREVRLGRNGVEEIRQHPFFKNDQWHWDNIRETAAPVVPELSSDIDSSNFDDIETFPIPKAFVGNQLPFIGFTY 6eda A 1.879 BS02 J3V A 1 A65 Q92 H94 H96 F131 L198 T199 A62 Q89 H91 H93 F127 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.2uM remove_due_to_license_issue P00918 30433782 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6edl A 2.799 BS01 J4M A 1 A1148 M1199 G1202 N1254 L1256 G1269 A47 M98 G101 N153 L155 G168 D1249 R1253 N1254 D1270 D148 R152 N153 D169 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Q9UM73 31009559 1500 NPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVSSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPI 6edr A 2.4 BS01 ZNA A 1 W125 S126 R127 E146 W189 T221 F222 W82 S83 R84 E103 W146 T178 F179 2.4.99.20,3.2.2.-,3.2.2.6 0061809 remove_due_to_license_issue P28907 30568770 401 SRWRQQWSGPGTTKRFPETVLARCVKYTEIHPEMRHVDCQSVWDAFKGAFISKHPCDITEEDYQPLMKLGTQTVPCNKILLWSRIKDLAHQFTQVQRDMFTLEDTLLGYLADDLTWCGEFATSKINYQSCPDWRKDCSNNPVSVFWKTVSRRFAEAACDVVHVMLDGSRSKIFDKDSTFGSVEVHNLQPEKVQTLEAWVIHGGREDSRDLCQDPTIKELESIISKRNIQFSCKNIYRPDKFLQCVKNPE 6eds A 3.18072 BS02 J22 A 1 F202 E205 Y302 Y314 T316 V360 K364 I374 N376 A479 F160 E163 Y260 Y272 T274 V318 K322 I332 N334 A437 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 31086331 1101 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNPINLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 6ee2 A 2.1 BS03 J1V A 1 K374 D379 K386 M392 N457 D459 A460 E461 L487 T488 G489 L492 F583 K290 D295 K302 M308 N373 D375 A376 E377 L403 T404 G405 L408 F499 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=195nM remove_due_to_license_issue W4I9J7 30537832 703 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 6ee2 F 2.1 BS03 J1V F 1 K374 D379 M392 L395 N457 D459 E461 L487 T488 G489 L492 F583 K281 D286 M299 L302 N364 D366 E368 L394 T395 G396 L399 F490 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=195nM remove_due_to_license_issue W4I9J7 30537832 703 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 6ee3 A 1.82 BS02 J4V A 1 T305 Q317 E319 A320 V459 G460 A461 M462 E463 R489 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 M267 E268 R294 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=137nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6ee4 A 1.58 BS02 J4S A 1 T305 Q317 E319 A320 V459 G460 A461 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=202nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6ee6 A 1.5 BS02 J4P A 1 T305 Q317 E319 A320 V459 G460 A461 R489 H496 E497 H500 E519 E572 Y575 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 R294 H301 E302 H305 E324 E377 Y380 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=216nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6eea A 1.63 BS02 J3V A 1 N62 H64 S65 Q67 Q92 H94 H96 L198 T199 T200 N59 H61 S62 Q64 Q89 H91 H93 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.2uM remove_due_to_license_issue P00918 30433782 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6eea A 1.63 BS03 J3V A 2 V135 L141 P202 V131 L137 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.2uM remove_due_to_license_issue P00918 30433782 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6eeb A 1.96 BS01 J6P A 1 L106 M125 M145 L101 M120 M140 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 Kd=5uM remove_due_to_license_issue P0DP23 31337679 201 TEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMT 6eed A 1.5 BS02 J6A A 1 T305 Q317 E319 A320 V459 G460 A461 H496 E497 H500 E519 E572 Y575 T576 Y580 M1034 T110 Q122 E124 A125 V264 G265 A266 H301 E302 H305 E324 E377 Y380 T381 Y385 M839 E463 H496 E497 H500 E519 E572 Y580 E268 H301 E302 H305 E324 E377 Y385 3.4.11.- 0006508,0008237,0008270 Ki=812nM remove_due_to_license_issue O96935 30537832 1102 PKIHYRKDYKPSGFIINQVTLNINIHDQETIVRSVLDMDISKHNVGEDLVFDGVGLKINEISINNKKLVEGEEYTYDNEFLTIFSKFVPKSKFAFSSEVIIHPETNYALTGLYKSKNIIVSQCEATGFRRITFFIDRPDMMAKYDVTVTADKEKYPVLLSNGDKVNEFEIPGGRHGARFNDPPLKPCYLFAVVAGDLKHLSATYITKYTKKKVELYVFSEEKYVSKLQWALECLKKSMAFDEDYFGLEYDLSRLNLVAVSDFNVGAMENKGLNIFNANSLLASKKNSIDFSYARILTVVGHEYFHQYTGNRVTLRDWFQLTLKEGLTVHRENLFSEEMTKTVTTRLSHVDLLRSVQFLEDSSPLSHPIRPESYVSMENFYTTTVYDKGSEVMRMYLTILGEEYYKKGFDIYIKKNDGNTATCEDFNYAMEQAYKMKKADNSANLNQYLLWFSQSGTPHVSFKYNYDAEKKQYSIHVNQYTKPDENQKEKKPLFIPISVGLINPENGKEMISQTTLELTKESDTFVFNNIAVKPIPSLFRGFSAPVYIEDQLTDEERILLLKYDSDAFVRYNSCTNIYMKQILMNYNEFLKAKNEKLESFQLTPVNAQFIDAIKYLLEDPHADAGFKSYIVSLPQDRYIINFVSNLDTDVLADTKEYIYKQIGDKLNDVYYKMFKSLEAKADDLTYFNDESHVDFDQMNMRTLRNTLLSLLSKAQYPNILNEIIEHSKSPYPSNWLTSLSVSAYFDKYFELYDKTYKLSKDDELLLQEWLKTVSRSDRKDIYEILKKLENEVLKDSKNPNDIRAVYLPFTNNLRRFHDISGKGYKLIAEVITKTDKFNPMVATQLCEPFKLWNKLDTKRQELMLNEMNTMLQEPQISNNLKEYLLRLTNK 6eee A 2.3 BS01 J4V A 1 K374 D379 M392 N457 D459 A460 E461 L487 T488 G489 L492 A577 F583 K285 D290 M303 N368 D370 A371 E372 L398 T399 G400 L403 A488 F494 K386 R463 K297 R374 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=28.9nM remove_due_to_license_issue A0A0L7KHE6 30537832 1001 ASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPGKENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSTDEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 6eee F 2.3 BS01 J4V F 1 K374 D379 M392 N457 D459 A460 E461 L487 T488 G489 L492 F583 K280 D285 M298 N363 D365 A366 E367 L393 T394 G395 L398 F489 K386 R463 K292 R369 3.4.11.1 0005737,0006508,0019538,0030145,0046872,0070006 Ki=28.9nM remove_due_to_license_issue A0A0L7KHE6 30537832 1001 SEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGGCNVEEGLTIFLVNNPENGPVKISSKVNDKQVSEFLKDENMEKFNVKLGTSKHFYMFNDNKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLETLFYEYMTDERFKSEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAAPSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYKSKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPENVEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDYIVDIATLTGAMLYSLGTSYAGVFGNNEELINKILQSSKTSNEPVWWLPIINEYRATLNSKYADINQISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFVLND 6eeh A 1.629 BS02 J4D A 1 N62 H64 S65 Q67 H94 H96 V131 V135 L198 T199 T200 P202 N59 H61 S62 Q64 H91 H93 V127 V131 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.29uM remove_due_to_license_issue P00918 30433782 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6eeh A 1.629 BS03 J4D A 2 W5 P201 P202 W2 P197 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.29uM remove_due_to_license_issue P00918 30433782 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6eeh A 1.629 BS04 J4D A 3 G132 K133 P202 G128 K129 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.29uM remove_due_to_license_issue P00918 30433782 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6eeo A 1.719 BS02 J6V A 1 H64 Q92 H94 H96 V135 L198 T199 T200 H61 Q89 H91 H93 V131 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.37uM remove_due_to_license_issue P00918 30433782 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6efj A 1.65 BS03 O5E A 1 W93 D124 H189 C208 K211 N220 H250 W52 D83 H148 C167 K170 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=477uM remove_due_to_license_issue C7C422 30942078 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6ega A 2.512 BS01 J8A A 1 M192 A211 E233 V236 M237 Y262 Y264 M265 G268 I308 H309 L318 S328 D329 F330 M27 A44 E60 V63 M64 Y87 Y89 M90 G93 I133 H134 L143 S153 D154 F155 D311 K313 A315 N316 D329 T351 D136 K138 A140 N141 D154 T158 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue Q9NWZ3 30679311 501 HSFSFYELKNVTNNFDERPISVGGNKMGEGGVVYKGYVNNTTVAVKKLTTEELKQQFDQEIKVMAKCQHENLVELLGFSSDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 6egs A 2.7 BS02 UD2 A 1 T143 D176 R201 L204 D224 H226 G308 G309 V330 G332 E334 N335 H359 H365 T56 D89 R114 L117 D137 H139 G221 G222 V243 G245 E247 N248 H272 H278 2.4.1.41 remove_due_to_license_issue Q10471 29601100 602 AEAKVRWPDFNQEAYVGGQVESDKLRMDRAIPDTRHDQCQRKQWRVDLPATSVVITFHNEARSALLRTVVSVLKKSPPHLIKEIILVDDYSNDPEDGALLGKIEKVRVLRNDRREGLMRSRVRGADAAQAKVLTFLDSHCECNEHWLEPLLERVAEDRTRVVSPIIDVINMDNFQYVGASADLKGGFDWNLVFKWDYMTPEQRRSRQGNPVAPIKTPMIAGGLFVMDKFYFEELGKYDMMMDVWGGENLEISFRVWQCGGSLEIIPCSRVGHVFRKQHPYTFPVFARNTRRAAEVWMDEYKNFYYAAVPSARNVPYGNIQSRLELRKKLSCKPFKWYLENVYPELRVPDHQDIAFGALQQGTNCLDTLGHFADGVVGVYECHNAGGNQEWALTKEKSVKHMDLCLTVVDRAPGSLIKLQGCRENDSRQKWEQIEGNSKLRHVGSNLCLDSRTAKSGGLSVEVCGPALSQQWKFTLNLQ 6ehh A 2.4 BS01 2GE A 1 L9 F27 N33 F72 F74 M81 W117 D119 D120 F139 L8 F26 N32 F71 F73 M80 W116 D118 D119 F138 3.6.1.-,3.6.1.56 0001669,0003723,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0008413,0008584,0008828,0016020,0016787,0016818,0030515,0031410,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=32nM remove_due_to_license_issue P53368 29281266 201 STSRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGAKRELLEESGLSVDTLHKVGHISFEFVGSPELMDVHIFSADHVHGTPTESEEMRPQWFQLDQIPFADMWPDDSYWFPLLLQKKKFCGHFKFQDQDTILSYSLREVDS 6ei4 A 2.0 BS01 B5N A 1 H42 H60 F197 P201 H204 N205 H208 R209 G216 V218 H39 H57 F194 P198 H201 N202 H205 R206 G213 V215 ? 0016491,0046872 remove_due_to_license_issue B2ZB02 29634898 301 KYRVRKNVLHLTDTEKRDFVRTVLILKEKGIYDRYIAWHGAAGKFHTPPGSDRNAAHMSSAFLPWHREYLLRFERDLQSINPEVTLPYWEWETDAQMQDPSQSQIWSADFMGGNGNPIKDFIVDTGPFAAGRWTTIDEQGNPSGGLKRNFGATKEAPTLPTRDDVLNALKITQYDTPPWDMTSQNSFRNQLEGFINGPQLHNRVHRWVGGQMGVVPTAPNDPVFFLHHANVDRIWAVWQIIHRNQNYQPMKNGPFGQNFRDPMYPWNTTPEDVMNHRKLGYVYDIELR 6ei5 A 2.2 BS01 B5Q A 1 N51 G97 M98 D102 N106 L107 F138 W162 T184 N37 G83 M84 D88 N92 L93 F124 W148 T170 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=3.83nM remove_due_to_license_issue P07900 29768913 301 EEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6eif A 2.22 BS01 B5T A 1 I165 A186 K188 L241 L294 V306 I32 A53 K55 L108 L161 V173 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 Ki=104nM remove_due_to_license_issue Ki=104nM, IC50=216nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eij A 2.42 BS01 B5Z A 1 F170 A186 K188 F238 M240 L241 L294 V306 D307 F37 A53 K55 F105 M107 L108 L161 V173 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 Ki=1680nM remove_due_to_license_issue Ki=1680nM, IC50=3500nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eil A 2.465 BS01 B6B A 1 I165 G166 A186 K188 S242 L294 V306 D307 I32 G33 A53 K55 S109 L161 V173 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Ki=>2800nM, IC50=>6000nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eip A 2.56 BS01 B7B A 1 I165 G166 V173 A186 V222 F238 M240 L241 N244 L294 V306 I32 G33 V40 A53 V89 F105 M107 L108 N111 L161 V173 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Ki=2015nM, IC50=4200nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eiq A 2.3 BS01 B6Z A 1 I165 V173 A186 L241 D247 L294 V306 D307 I32 V40 A53 L108 D114 L161 V173 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 Ki=383nM remove_due_to_license_issue Ki=383nM, IC50=800nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eir A 2.4 BS01 B6H A 1 I165 V173 A186 M240 L241 S242 D247 L294 I32 V40 A53 M107 L108 S109 D114 L161 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 Ki=575nM remove_due_to_license_issue Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eis A 2.36 BS01 B6N A 1 I165 G166 V173 K188 F238 E291 L294 V306 D307 I32 G33 V40 K55 F105 E158 L161 V173 D174 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 Ki=252nM remove_due_to_license_issue Ki=252nM, IC50=532nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6ej2 A 1.46 BS01 B7E A 1 G422 D441 Y480 W485 I519 I527 R537 D637 G639 G18 D37 Y76 W81 I115 I123 R133 D223 G225 3.4.23.46 0004190,0006508,0016020 Ki=16nM remove_due_to_license_issue P56817 29617572 901 AGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTDLMEDCGY 6ej3 A 1.94 BS01 B7T A 1 D32 Y71 W76 I110 I118 D228 G230 D32 Y71 W76 I110 I118 D216 G218 3.4.23.46 0004190,0006508,0016020 Ki=1179nM remove_due_to_license_issue P56817 29617572 501 EMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIP 6ej4 A 2.88 BS01 B7W A 1 V173 F238 L241 V306 V40 F105 L108 V173 D287 K289 N292 D307 S324 D154 K156 N159 D174 S191 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue IC50=329nM, Ki=158nM Q13627 30095246 501 KVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDEYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFK 6eji A 2.3 BS01 UD2 A 1 S14 G16 Y46 H118 S119 L146 N166 I189 R191 K196 R246 V247 V250 E267 G268 L269 P270 T271 E275 S14 G16 Y46 H118 S119 L146 N166 I189 R191 K196 R246 V247 V250 E267 G268 L269 P270 T271 E275 ? 0000166,0016757 ic50=303uM remove_due_to_license_issue O86151 29386647 401 MMMKISFIIATLNSGGAERVLVTLANALCKEHEVSIIKFHTGESFYKLENEVKVTSLEQFRFDTLYHKIASRFKKFFALRKALKESKADVFISFLDTTNIACILANIGLKTPLIISEHSNEAYLKPKTWRFLRRVSYPFCDALSVLGSSDKVYYERFVKRVKLLLNPCHFSDEIPFDSSFEKENLVLFIGRLDHNKNPVMFLKAIAHLDKNLQENYKFVIAGDGELRQELEYKVKSLGIKVDFLGRVENVKALYEKAKVLCLCSFVEGLPTVLIESLYFEVCRISSSYYNGAKDLIKDNHDGLLVGCDDEIALAKKLELVLNDENFRKELVNNAKQRCKDFEISNIKEEWLKLIVEVKNA 6ek3 A 1.6 BS01 OUL A 1 H364 G365 Y396 F397 A398 S404 Y409 L464 H78 G79 Y107 F108 A109 S115 Y120 L175 2.4.2.- 0003950 remove_due_to_license_issue IC50=>10000nM Q460N3 30006177 901 LPEHWTDMNHQLFCMVQLEPGQSEYNTIKDKFTRTCSSYAIEKIERIQNAFLWQSYQVKKRQMDIKNDHKNNERLLFHGTDADSVPYVNQHGFNRSCNAVSYGKGTYFAVDASLSAKDTYSKPDSNGRKHMYVVRVLTGVFTKGRAGLVTPPPKNPHNPTDLFDSVTNNTRSPKLFVVFFDNQAYPEYLITFTA 6ekd A 2.1 BS01 B9K A 1 I70 S72 G73 V78 M149 A151 Q155 L206 I25 S27 G28 V33 M104 A106 Q110 L161 D189 K191 N194 D207 T226 D144 K146 N149 D162 T167 2.7.11.24 0004672,0004707,0005524,0006468 ic50=184nM remove_due_to_license_issue P53779 30087925 503 NQFYSVEVGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDDEREHTIEEWKELIYKEVMN 6ekn A 1.2 BS06 B9N A 1 I180 L181 A182 H183 H218 E219 H222 H228 V235 P238 T239 Y240 I76 L77 A78 H79 H114 E115 H118 H124 V131 P134 T135 Y136 H218 E219 H222 H228 H114 E115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=510nM P39900 29727184 306 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 6ekq A 1.65 BS01 B0H A 1 F653 V657 P658 E661 Y707 N708 F714 F29 V33 P34 E37 Y83 N84 F90 ? Kd=10.9uM remove_due_to_license_issue IC50=30600nM, Kd=3500nM P55201 29902720 801 SMEMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGGAVLRQARRQAEKMG 6eks A 1.87 BS04 G39 A 1 R250 D276 Q343 E645 R661 D663 R738 Y766 R197 D223 Q290 E592 R608 D610 R685 Y713 3.2.1.18 0004308,0005576,0005737,0006689,0009313,0016020,0016798,0033691,0043231 ic50=144uM remove_due_to_license_issue P0C6E9 29149072 908 ALFDYNATGDTFDSPAKQGWMQDNTNNGSGVLTNAMPAWLVQGIGGRAQWTYSLSTNQHAQASSFGWRMTTEMKVLSGGMITNYYANGTQRVLPIISLDSSGNLVVEFEGQTGRTVLATGTAATEYHKFELVFLPGSNPSASFYFDGKLIRDNIQPTASKQNMIVWGNGSSNTDGVAAYRDIKFEIQGDVIFRGPDRIPSIVASSVTPGVVTAFAEKRVGGGDPGALSNTNDIITRTSRDGGITWDTELNLTEQINVSDEFDFSDPRPIYDPSSNTVLVSYARWPTDAAQNGDRIKPWMPNGIFYSVYDVASGNWQAPIDVTDQVKERSFQIAGWGGSELYRRNTSLNSQQDWQSNAKIRIVDGAANQIQVADGSRKYVVTLSIDESGGLVANLNGVSAPIILQSEHAKVHSFHDYELQYSALNHTTTLFVDGQQITTWAGEVSQENNIQFGNADAQIDGRLHVQKIVLTQQGHNLVEFDAFYLAQQTPEVEKDLEKLGWTKIKTGNTMSLYGNASVNPGPGHGITLTRQQNISGSQNGRLIYPAIVLDRFFLNVMSIYSDDGGSNWQTGSTLPIPFRWKSSSILETLEPSEADMVELQNGDLLLTARLDFNQIVNGVNYSPRQQFLSKDGGITWSLLEANNANVFSNISTGTVDASITRFEQSDGSHFLLFTNPQGNPAGTNGRQNLGLWFSFDEGVTWKGPIQLVNGASAYSDIYQLDSENAIVIVETDNSNMRILRMPITLLKQKL 6eku A 1.75 BS01 ZMR A 1 R250 I251 E269 R271 D276 D318 N344 R661 D663 R738 Y766 R200 I201 E219 R221 D226 D268 N294 R611 D613 R688 Y716 3.2.1.18 0004308,0005576,0005737,0006689,0009313,0016020,0016798,0033691,0043231 ic50=52uM remove_due_to_license_issue P0C6E9 29149072 901 ALFDYNATGDTEFDSPAKQGWMQDNTNNGSGVLTNADGMPAWLVQGIGGRAQWTYSLSTNQHAQASSFGWRMTTEMKVLSGGMITNYYANGTQRVLPIISLDSSGNLVVEFEGQTGRTVLATGTAATEYHKFELVFLPGSNPSASFYFDGKLIRDNIQPTASKQNMIVWGNGSSNTDGVAAYRDIKFEIQGDVIFRGPDRIPSIVASSVTPGVVTAFAEKRVGGGDPGALSNTNDIITRTSRDGGITWDTELNLTEQINVSDEFDFSDPRPIYDPSSNTVLVSYARWPTDAAQNGDRIKPWMPNGIFYSVYDVASGNWQAPIDVTDQVKERSFQIAGWGGSELYRRNTSLNSQQDWQSNAKIRIVDGAANQIQVADGSRKYVVTLSIDESGGLVANLNGVSAPIILQSEHAKVHSFHDYELQYSALNHTTTLFVDGQQITTWAGEVSQENNIQFGNADAQIDGRLHVQKIVLTQQGHNLVEFDAFYLAQQTPEVEKDLEKLGWTKIKTGNTMSLYGNASVNPGPGHGITLTRQQNISGSQNGRLIYPAIVLDRFFLNVMSIYSDDGGSNWQTGSTLPIPFRWKSSSILETLEPSEADMVELQNGDLLLTARLDFNQIVNGVNYSPRQQFLSKDGGITWSLLEANNANVFSNISTGTVDASITRFEQSDGSHFLLFTNPQGNPAGTNGRQNLGLWFSFDEGVTWKGPIQLVNGASAYSDIYQLDSENAIVIVETDNSNMRILRMPITLLKQKLTLS 6el5 A 1.67 BS01 PU1 A 1 N51 A55 G97 M98 L107 F138 W162 N36 A40 G82 M83 L92 F123 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue EC50=1200nM P07900 29768913 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6ela A 1.485 BS06 B9Z A 1 G179 A182 H218 E219 H222 H228 V235 F237 P238 T239 Y240 G73 A76 H112 E113 H116 H122 V129 F131 P132 T133 Y134 H218 E219 H222 H228 H112 E113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=26nM P39900 29727184 306 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYAYVDINTFRLSADDIRGIQSLYG 6eln A 1.6 BS01 P4A A 1 N51 A55 K58 D93 I96 G97 M98 L107 G108 T184 N35 A39 K42 D77 I80 G81 M82 L91 G92 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29768913 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6elo A 1.8 BS01 BAW A 1 N51 A55 K58 D93 I96 G97 M98 L107 G108 F138 T184 N35 A39 K42 D77 I80 G81 M82 L91 G92 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29768913 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6elp A 1.85 BS01 BA8 A 1 N51 A55 D93 G97 M98 L107 F138 Y139 W162 T184 N35 A39 D77 G81 M82 L91 F122 Y123 W146 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29768913 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6emh A 1.76 BS01 BGE A 1 V78 A91 M146 M149 A151 L206 V27 A40 M95 M98 A100 L155 D189 K191 N194 D207 T226 D138 K140 N143 D156 T170 2.7.11.24 0004672,0004707,0005524,0006468 ic50=833nM remove_due_to_license_issue P53779 30087925 504 NQFYSVEVGDSTFTVLKRYQNLKPIIVCAAYDAVLDRNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIISLLNVFTPQKTLEEFQDVYLVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMVTRYYRAPEVILGMGYKENVDIWSVGCIMGEMVRHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRNYVENRPKYAGLTFPKLFPDSLFPADSEHNKLKASQARDLLSKMLVIDPAKRISVDDALQHPYINVWYDPAEVEAPPPQIYDKQLDEREHTIEEWKELIYKEVMN 6emu A 2.29745 BS01 SAM A 1 L181 D182 P183 W184 I201 G202 I204 D206 K211 K212 T215 K233 I234 D245 I250 L81 D82 P83 W84 I101 G102 I104 D106 K109 K110 T113 K131 I132 D143 I148 2.1.1.218,2.1.1.221 remove_due_to_license_issue Q5JD38 29848639 501 WPYFIIDLYHWDKHTQKEKGKIALQVNQSYGLLRDYFELAVTWANEEFREMFHGPLDRITTYGGPTSEFLKENGINEVVLLDPWAEEVLSEKDFDVKAFIIGGIVDTNKKKTTPKIGEELESAGIKVRRRKIVLRGDVVGVPDRINRILGIILKMMVEGKSMDEAVYEMQ 6en4 C 3.08 BS01 BGZ D 1 K1071 R1074 R1075 V1078 V1110 F1153 Y1157 K609 R612 R613 V616 V648 F691 Y695 ? 0000245,0003729 remove_due_to_license_issue O75533 29656923 104 NLPFLKPDDIQYFDKLLVDVDESTLSPEEQKERKIMKLLLKIKNGTPPMRKAALRQITDKAREFGAGPLFNQILPLLMSPTLEDQERHLLVKVIDRILYKLDDLVRPYVHKILVVIEPLLIDEDYYARVEGREIISNLAKAAGLATMISTMRPDIDNMDEYVRNTTARAFAVVASALGIPSLLPFLKAVCKSKKSWQARHTGIKIVQQIAILMGCAILPHLRSLVEIIEHGLVDEQQKVRTISALAIAALAEAATPYGIESFDSVLKPLWKGIRQHRGKGLAAFLKAIGYLIPLMDAEYANYYTREVMLILIREFQSPDEEMKKIVLKVVKQCCGTDGVEANYIKTEILPPFFKHFWQHRMALDRRNYRQLVDTTVELANKVGAAEIISRIVDDLKDEAEQYRKMVMETIEKIMGNLGAADIDHKLEEQLIDGILYAFQEQTTEDSVMLNGFGTVVNALGKRVKPYLPQICGTVLWRLNNKSAKVRQQAADLISRTAVVMKTCQEEKLMGHLGVVLYEYLGEEYPEVLGSILGALKAIVNVIGMHKMTPPIKDLLPRLTPILKNRHEKVQENCIDLVGRIADRGAEYVSAREWMRICFELLELLKAHKKAIRRATVNTFGYIAKAIGPHDVLATLLNNLKVQERQNRVCTTVAIAIVAETCSPFTVLPALMNEYRVPELNVQNGVLKSLSFLFEYIGEMGKDYIYAVTPLLEDALMDRDLVHRQTASAVVQHMSLGVYGFGCEDSLNHLLNYVWPNVFETSPHVIQAVMGALEGLRVAIGPCRMLQYCLQGLFHPARKVRDVYWKIYNSIYIGSQDALIAHYPRIYNDDKNTYIRYELDYIL 6en5 A 1.75 BS03 BJ2 A 1 Q259 H331 A332 S333 A334 H361 E362 H365 Y369 E389 K489 H491 Y498 Y501 Q254 H326 A327 S328 A329 H356 E357 H360 Y364 E384 K484 H486 Y493 Y496 H331 A332 H361 E362 H365 E389 H491 Y501 H326 A327 H356 E357 H360 E384 H486 Y496 3.4.15.1 0006508,0008237,0008241,0016020 Ki=11.45nM remove_due_to_license_issue P12821 29206036 702 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLPCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 6en6 A 1.8 BS02 BJ2 A 1 Q259 H331 A332 S333 A334 H361 E362 H365 Y369 E389 K489 H491 Y498 Y501 Q254 H326 A327 S328 A329 H356 E357 H360 Y364 E384 K484 H486 Y493 Y496 H331 A332 H361 E362 H365 E389 H491 Y501 H326 A327 H356 E357 H360 E384 H486 Y496 3.4.15.1 0006508,0008237,0008241,0016020 Ki=11.45nM remove_due_to_license_issue P12821 29206036 711 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLPCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 6en8 A 3.29 BS01 dna X 0 K7 T8 K10 S14 V45 A46 G48 L49 F52 Y53 K2 T3 K5 S9 V40 A41 G43 L44 F47 Y48 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 PKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 A 3.29 BS02 dna Y 0 K10 S35 I36 Y47 Y51 K57 K5 S30 I31 Y42 Y46 K52 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 PKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 B 3.29 BS01 dna X 0 S35 I36 Y47 Y51 S56 K57 S23 I24 Y35 Y39 S44 K45 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 KESLNKILDSVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 B 3.29 BS02 dna Y 0 S14 V45 A46 G48 L49 F52 Y53 S3 V33 A34 G36 L37 F40 Y41 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 KESLNKILDSVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 C 3.29 BS01 dna Q 0 S35 I36 Y47 Y51 S56 K57 S30 I31 Y42 Y46 S51 K52 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 PKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 C 3.29 BS02 dna Z 0 K7 T8 G11 S14 V45 A46 Y47 G48 L49 F52 Y53 K2 T3 G6 S9 V40 A41 Y42 G43 L44 F47 Y48 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 PKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 D 3.29 BS01 dna Q 0 S14 V45 A46 Y47 G48 L49 F52 S2 V33 A34 Y35 G36 L37 F40 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 ESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTP 6en8 D 3.29 BS02 dna Z 0 S35 I36 Y47 Y51 S56 K57 S23 I24 Y35 Y39 S44 K45 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 ESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTP 6en8 E 3.29 BS01 dna X 0 K7 T8 S14 A46 G48 L49 F52 Y53 K4 T5 S11 A43 G45 L46 F49 Y50 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 RAPKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 E 3.29 BS02 dna Y 0 S35 I36 Y47 Y51 S56 K57 S32 I33 Y44 Y48 S53 K54 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 RAPKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLTPR 6en8 F 3.29 BS01 dna Q 0 K10 S35 I36 Y47 Y51 S56 K57 K5 S30 I31 Y42 Y46 S51 K52 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 PKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLT 6en8 F 3.29 BS02 dna Z 0 T8 K10 S14 A46 G48 L49 F52 Y53 T3 K5 S9 A41 G43 L44 F47 Y48 ? 0003677 remove_due_to_license_issue Q4J9S1 30948713 1 ~ 21 PKTEKGKESLNKILDASVELIADKGFLSTSINDITSKAGVAYGLFYFYFKSKHDILDEIIRQFNRNMRYYLKTYTQNLDSRIDVEKVGMKKFLEWMNENKKYYKIFIETQVHRPDIYKWHFMKLAERYTTGLSEAMRRGEIINVDPELLSYVLIGIAHMLGKRYVLWSNSGLTLKQQRDLDLIIENMLT 6enm A 1.59 BS01 LPW A 1 I180 A182 L214 T215 H218 E219 H222 H228 V235 P238 T239 Y240 I69 A71 L103 T104 H107 E108 H111 H117 V124 P127 T128 Y129 H218 E219 H222 H228 H107 E108 H111 H117 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=4.8nM P39900 29727184 301 HYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 6enx A 1.95 BS02 BJW A 1 G54 A55 G56 F66 R67 Y98 R101 Q136 I138 H154 V217 W218 F219 G220 E221 T222 G245 T246 S247 V250 Y251 N271 M272 P288 C289 G23 A24 G25 F35 R36 Y67 R70 Q105 I107 H123 V186 W187 F188 G189 E190 T191 G214 T215 S216 V219 Y220 N240 M241 P257 C258 P64 T65 F66 R67 N137 D139 H154 P33 T34 F35 R36 N106 D108 H123 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q6DHI5 29044784 303 PSSDLTAFREHFAKAKHIAIITGAGVSAESGVPTFRGPGGFWRKWQAQDLATPEAFSRDPSLVWEFYHYRREVMRSKMPNPAHLAIAECEARLGQQGRSVVIITQNIDELHHRAGSKHVYEIHGSLFKTRCMSCGEVKANHKSPICPALDGKGAPDPNTKEARIPVELLPRCERKSCNGLLRPHVVWFGETLDSDILTAVERELEKCDLCLVVGTSSIVYPAAMFAPQVASRGVPVAEFNMECTPATQRFKYHFEGPCGSTLPPALE 6eo0 A 2.4 BS03 BVT A 1 G54 A55 G56 A59 F66 R67 Y98 R101 Q136 I138 H154 V217 F219 G220 E221 T222 G245 S247 V250 Y251 N271 M272 E273 C289 G30 A31 G32 A35 F42 R43 Y74 R77 Q112 I114 H130 V193 F195 G196 E197 T198 G221 S223 V226 Y227 N247 M248 E249 C265 P64 T65 F66 R67 N137 D139 H154 P40 T41 F42 R43 N113 D115 H130 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q6DHI5 29044784 304 PFTKMTRPSSDLTAFREHFAKAKHIAIITGAGVSAESGVPTFRGPGGFWRKWQAQDLATPEAFSRDPSLVWEFYHYRREVMRSKMPNPAHLAIAECEARLGQQGRSVVIITQNIDELHHRAGSKHVYEIHGSLFKTRCMSCGEVKANHKSPICPALDGKGAPDPNTKEARIPVELLPRCERKSCNGLLRPHVVWFGETLDSDILTAVERELEKCDLCLVVGTSSIVYPAAMFAPQVASRGVPVAEFNMECTPATQRFKYHFEGPCGSTLPPALE 6eo0 A 2.4 BS04 BVT C 1 E232 M255 F256 E208 M231 F232 P64 T65 F66 R67 N137 D139 H154 P40 T41 F42 R43 N113 D115 H130 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q6DHI5 29044784 303 PFTKMTRPSSDLTAFREHFAKAKHIAIITGAGVSAESGVPTFRGPGGFWRKWQAQDLATPEAFSRDPSLVWEFYHYRREVMRSKMPNPAHLAIAECEARLGQQGRSVVIITQNIDELHHRAGSKHVYEIHGSLFKTRCMSCGEVKANHKSPICPALDGKGAPDPNTKEARIPVELLPRCERKSCNGLLRPHVVWFGETLDSDILTAVERELEKCDLCLVVGTSSIVYPAAMFAPQVASRGVPVAEFNMECTPATQRFKYHFEGPCGSTLPPALE 6eo6 H 1.69 BS01 dna D 0 I372 F382 Q387 L423 R425 T432 R433 Y434 E435 R436 N437 I438 I441 Y477 I9 F19 Q24 L60 R62 T69 R70 Y71 E72 R73 N74 I75 I78 Y114 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 29684204 401 ~ 415 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 6eo7 H 2.24 BS01 dna D 0 I372 R433 Y434 E435 R436 N437 I438 I441 Y477 I9 R70 Y71 E72 R73 N74 I75 I78 Y114 3.4.21.5 0004252,0005509,0006508,0007596 remove_due_to_license_issue P00734 29684204 401 ~ 415 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE 6eo8 H 1.94 BS03 2FN H 1 I174 D189 A190 V213 W215 G216 E217 G219 R221A G226 F227 Y228 I170 D190 A191 V216 W218 G219 E220 G221 R224 G229 F230 Y231 3.4.21.5 0004252,0005509,0006508,0007596 Ki=100nM remove_due_to_license_issue P00734 25268757 307 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQ 6eo9 H 1.84 BS03 2OJ H 1 E97A I174 A190 V213 W215 G216 E217 G219 G226 F227 Y228 E94 I172 A193 V218 W220 G221 E222 G223 G231 F232 Y233 3.4.21.5 0004252,0005509,0006508,0007596 Ki=160nM remove_due_to_license_issue P00734 25268757 307 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 6eog A 1.2 BS01 BKK A 1 R144 I145 A146 H158 R162 N174 W181 E184 S237 G238 R32 I33 A34 H46 R50 N62 W69 E72 S125 G126 ? 0030246 Kd=1.6uM remove_due_to_license_issue P17931 29194992 1001 MLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6eol A 1.5 BS01 BKH A 1 R144 I145 A146 H158 N160 R162 N174 W181 E184 S237 G238 R32 I33 A34 H46 N48 R50 N62 W69 E72 S125 G126 ? 0030246 Kd=0.037uM remove_due_to_license_issue P17931 29194992 303 MLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6eox A 1.3 BS06 BKW A 1 I180 L181 A182 H218 E219 H222 H228 V235 F237 P238 T239 Y240 I75 L76 A77 H113 E114 H117 H123 V130 F132 P133 T134 Y135 H218 E219 H222 H228 H113 E114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=140nM P39900 29727184 306 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 6ep4 A 2.30005 BS02 DME A 1 W82 P285 Y332 H438 W80 P283 Y330 H432 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H432 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 Ki=4.5uM remove_due_to_license_issue P06276 29186056 601 DIIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6ep9 A 2.01 BS01 BNB A 1 Q412 F413 V416 A428 K430 M477 A478 N479 G480 D521 L528 D539 L542 S543 Y551 Q17 F18 V21 A33 K35 M82 A83 N84 G85 D126 L133 D144 L147 S148 Y156 D521 A523 R525 N526 D539 D126 A128 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30756207 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 6epa A 1.82 BS04 BNQ A 1 W30 I51 Y52 F72 F85 T92 W103 L182 W28 I49 Y50 F70 F83 T90 W101 L180 ? 0005509,0005515,0005737,0007268,0007269,0007528,0008021,0008048,0009966,0016192,0046872,0046928 remove_due_to_license_issue Kd=1130nM Q9VWX8 29966094 204 KKNSKLKQDTIDRLTTDTYFTEKEIRQWHKGFLKDCPNGLLTEQGFIKIYKQFFPDGDPSKFASLVFRVFDENNDGAIEFEEFIRALSITSRGNLDEKLHWAFRLYDVDNDGYITREEMYNIVDAIYQMVGQQPQTEDENTPQKRVDKIFDQMDKNHDDRLTLEEFREGSKADPRMVQALSLG 6eq2 A 1.802 BS01 BU8 A 1 N33 F72 W117 D119 D120 N31 F70 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue IC50=1100nM, Kd=1300nM P36639 31077996 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6eq3 A 1.798 BS01 BU5 A 1 Y7 T8 F27 N33 G37 F72 M81 V83 W117 D119 D120 Y5 T6 F25 N31 G35 F70 M79 V81 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue Kd=700nM, IC50=400nM P36639 31077996 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6eq4 A 1.4 BS01 BSW A 1 Y7 N33 F72 M81 W117 D119 D120 Y5 N31 F70 M79 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue Kd=2400nM, IC50=800nM P36639 31077996 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6eq5 A 1.801 BS01 AX7 A 1 F72 F74 M81 W117 D119 F71 F73 M80 W116 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue IC50=44000nM, Kd=18000nM P36639 31077996 201 GASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6eq6 A 2.002 BS01 EV2 A 1 L9 F74 W117 D119 F139 L7 F72 W115 D117 F137 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue Kd=15000nM, IC50=23000nM P36639 31077996 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6eq7 A 1.5 BS01 BS8 A 1 F27 N33 F72 M81 W117 D119 D120 F25 N31 F70 M79 W115 D117 D118 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 remove_due_to_license_issue P36639 31077996 201 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6eq8 D 2.19 BS01 BQZ D 1 W110 G111 W317 R320 N333 E335 Y487 S515 R533 W639 E641 W103 G104 W310 R313 N326 E328 Y480 S508 R526 W632 E634 Kd=0.12uM remove_due_to_license_issue 29602905 708 AFETTTPPEPPQFPAEGKINYVARDTILEFKALPSYSEPDWITEKFEKAGKLPPLKERLPEEPLVYKTGNMPDGVGVYGDTMRHVVGGRPEGWNYIAGQSQGWGGIDIALSECLTRTAPLFQVDAKDTEPLPNLAKSWEWSEDGHTLTMHLVKGAKWSDGEAFNADDVMFYWEDAVVDPNVSPLGGGASPEAFGEGTTLKKIDDYTVEWTFKAAFPKQYLYTMAYPSFCPGPSHILKPQHPKYSKNTYNQFKNAFPPEYMNMPVMGAWVPVSYRPDDLIVLRRNPYYWKVDEKGQQLPYLNEVHYKLSTWADRDVQAVAGSGDFSNLEQPENFVASLKRAADPNAPARLAFGPRLIGYNLQMNFSANGWGNPDERGQAIRELNRNEVFRQAVTSALDRKAIGDSLVKGPFTAIYPGGISSGTSFYDRASTVYYPFNLEGAKAALASIGLKDTDGDGFLNFPKETLGGRNVEITLLVNNGYATDKSLAEGLVGQMAKLGLRVVIHSLDSNQRDAAHYGGQFDWLVRRNSTELSSVVQNTEQLAPVGPRTSWNHRSPEGKELDLMPFEKEMADIVRKFISSQDNAERADLMKQYQKVYTQNLYTIGLTEYPGALIVNKRFSNVPQGTPIFMFNWAEDAIIRERLWVAADKQGKYELFPQQLPGKPGEGGPIN 6eqm A 1.35 BS01 BUH A 1 G11 Q12 G13 Y14 L30 D32 Y71 F108 I110 I118 D228 G230 T231 T232 G14 Q15 G16 Y17 L33 D35 Y74 F111 I113 I121 D221 G223 T224 T225 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 ic50=11nM remove_due_to_license_issue IC50=7.00nM P56817 30224383 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6eqp A 2.34942 BS02 BUW A 1 W82 G116 Q119 T120 S198 W231 L286 F329 Y332 W79 G113 Q116 T117 S195 W228 L283 F326 Y329 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G113 G114 G146 S195 A196 Y234 V285 F287 E322 H435 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 Kd=1.1uM remove_due_to_license_issue IC50=1600nM, Ki=20nM P06276 29186056 601 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6eqs A 1.32 BS02 BV8 A 1 G58 A59 G60 E64 F70 R71 Y102 R105 Q140 I142 H158 V221 F223 G224 E225 N226 G249 T250 S251 V254 Y255 N275 T276 E277 C293 G25 A26 G27 E31 F37 R38 Y69 R72 Q107 I109 H125 V188 F190 G191 E192 N193 G216 T217 S218 V221 Y222 N242 T243 E244 C260 P68 T69 F70 R71 N141 D143 H158 P35 T36 F37 R38 N108 D110 H125 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q9NXA8 29044784 402 ARPSSSMADFRKFFAKAKHIVIISGAGVSAESGVPTFRGAGGYWRKWQAQDLATPLAFAHNPSRVWEFYHYRREVMGSKEPNAGHRAIAECETRLGKQGRRVVVITQNIDELHRKAGTKNLLEIHGSLFKTRCTSCGVVAENYKSPICPALSGKGAPEPGTQDASIPVEKLPRCEEAGCGGLLRPHVVWFGENLDPAILEEVDRELAHCDLCLVVGTSSVVYPAAMFAPQVAARGVPVAEFNTETTPATNRFRFHFQGPCGTTLPEALA 6eqs A 1.32 BS04 BV8 D 1 N226 D236 P256 M259 Q263 N193 D203 P223 M226 Q230 P68 T69 F70 R71 N141 D143 H158 P35 T36 F37 R38 N108 D110 H125 2.3.1.- 0036054,0036055,0070403 remove_due_to_license_issue Q9NXA8 29044784 402 ARPSSSMADFRKFFAKAKHIVIISGAGVSAESGVPTFRGAGGYWRKWQAQDLATPLAFAHNPSRVWEFYHYRREVMGSKEPNAGHRAIAECETRLGKQGRRVVVITQNIDELHRKAGTKNLLEIHGSLFKTRCTSCGVVAENYKSPICPALSGKGAPEPGTQDASIPVEKLPRCEEAGCGGLLRPHVVWFGENLDPAILEEVDRELAHCDLCLVVGTSSVVYPAAMFAPQVAARGVPVAEFNTETTPATNRFRFHFQGPCGTTLPEALA 6equ A 1.65 BS02 BVE A 1 H64 N67 Q92 H94 H119 F131 L198 T199 T200 H65 N68 Q93 H95 H120 F131 L198 T199 T200 H64 H94 H96 E106 H119 T199 H65 H95 H97 E107 H120 T199 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=419nM remove_due_to_license_issue Ki=419nM P00918 29199489 302 GMSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6er3 A 1.37 BS01 SIA C 1 I54 E85 R87 K94 R163 Y169 I48 E79 R81 K88 R152 Y158 ? 0004308,0005975 remove_due_to_license_issue A7B557 29259165 2 GSVLQKEGIEISEGTGYDLSKEPGAATVKALEQGTIVISYKTTSENAIQSLLSVGNGTKGNQDRHFHLYITNAGGVGMELRNTDGEFKYTLDCPAAVRGSVSNTVALKADKENKQYKLFANGELIATLDQEAFKFISDITGVDNVMLGGTMRQGTVAYPFGGSIERMQVYRDVLSDDELIAVTG 6er3 B 1.37 BS01 SIA D 1 I54 E85 R87 K94 R163 Y169 I48 E79 R81 K88 R152 Y158 ? 0004308,0005975 remove_due_to_license_issue A7B557 29259165 2 GSVLQKEGIEISEGTGYDLSKEPGAATVKALEQGTIVISYKTTSENAIQSLLSVGNGTKGNQDRHFHLYITNAGGVGMELRNTDGEFKYTLDCPAAVRGRVSNTVALKADKENKQYKLFANGELIATLDQEAFKFISDITGVDNVMLGGTMRQGTVAYPFGGSIERMQVYRDVLSDDELIAVTGI 6er4 A 1.3 BS01 BGC C 1 D110 D131 D67 D88 ? 0004308,0005975 remove_due_to_license_issue A7B557 29259165 1 MADIGSVLQKEGIEISEGTGYDLSKEPGAATVKALEQGTIVISYKTTSENAIQSLLSVGNGTKGNQDRHFHLYITNAGGVGMELRNTDGEFKYTLDCPAAVRGSYKGERVSNTVALKADKENKQYKLFANGELIATLDQEAFKFISDITGVDNVMLGGTMRQGTVAYPFGGSIERMQVYRDVLSDDELIAVTGK 6er4 A 1.3 BS02 SIA C 1 I95 E126 R128 K135 R204 Y210 I52 E83 R85 K92 R161 Y167 ? 0004308,0005975 remove_due_to_license_issue A7B557 29259165 3 MADIGSVLQKEGIEISEGTGYDLSKEPGAATVKALEQGTIVISYKTTSENAIQSLLSVGNGTKGNQDRHFHLYITNAGGVGMELRNTDGEFKYTLDCPAAVRGSYKGERVSNTVALKADKENKQYKLFANGELIATLDQEAFKFISDITGVDNVMLGGTMRQGTVAYPFGGSIERMQVYRDVLSDDELIAVTGK 6er4 B 1.3 BS01 BGC D 1 D110 D131 D63 D84 ? 0004308,0005975 remove_due_to_license_issue A7B557 29259165 1 GSVLQKEGIEISEGTGYDLSKEPGAATVKALEQGTIVISYKTTSENAIQSLLSVGNGTKGNQDRHFHLYITNAGGVGMELRNTDGEFKYTLDCPAAVRGSYKGERVSNTVALKADKENKQYKLFANGELIATLDQEAFKFISDITGVDNVMLGGTMRQGTVAYPFGGSIERMQVYRDVLSDDELIAVTG 6er4 B 1.3 BS02 SIA D 1 I95 E126 R128 K135 R204 Y210 I48 E79 R81 K88 R157 Y163 ? 0004308,0005975 remove_due_to_license_issue A7B557 29259165 3 GSVLQKEGIEISEGTGYDLSKEPGAATVKALEQGTIVISYKTTSENAIQSLLSVGNGTKGNQDRHFHLYITNAGGVGMELRNTDGEFKYTLDCPAAVRGSYKGERVSNTVALKADKENKQYKLFANGELIATLDQEAFKFISDITGVDNVMLGGTMRQGTVAYPFGGSIERMQVYRDVLSDDELIAVTG 6ert A 1.8 BS02 BVZ A 1 V57 A70 M120 Y122 V123 E127 E170 L173 T183 D184 F327 V45 A58 M108 Y110 V111 E115 E158 L161 T171 D172 F315 D166 K168 N171 D184 T201 D154 K156 N159 D172 T189 2.7.11.11 0004672,0004674,0005524,0006468 remove_due_to_license_issue P25321 401 ESVKEFLAKAKEEFLKKWESPSQNTAQLDHFDRIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFTEF 6es0 A 2.38 BS01 BW8 A 1 R26 A45 K47 E66 L70 L79 T95 Y97 M98 H144 L153 A163 D164 F165 W170 R22 A41 K43 E62 L66 L75 T91 Y93 M94 H140 L149 A159 D160 F161 W166 D146 Q150 N151 D164 D142 Q146 N147 D160 2.7.10.2,2.7.11.1 0004672,0005524,0006468 ic50=2.26uM remove_due_to_license_issue IC50=4870nM O43353 29409752 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLHIHTPLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWGTIIYMPPENYASIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLKKTKLQS 6es2 K 2.95 BS01 dna A 0 R190 V191 Y193 R198 R228 Q229 I232 N236 R4 V5 Y7 R12 R42 Q43 I46 N50 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 1 ~ 18 DKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQQ 6es2 K 2.95 BS02 dna D 0 Y189 R190 Q235 R238 R242 Y3 R4 Q49 R52 R56 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 19 ~ 36 DKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQQ 6es2 L 2.95 BS01 dna B 0 R190 V191 Y193 R198 R228 Q229 I232 N236 R5 V6 Y8 R13 R43 Q44 I47 N51 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 1 ~ 18 KDKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQ 6es2 L 2.95 BS02 dna E 0 Y189 R190 Q235 R238 R242 Y4 R5 Q50 R53 R57 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 19 ~ 36 KDKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQ 6es3 K 2.57 BS01 dna A 0 R184 K186 R190 V191 Y193 R198 R228 Q229 N236 K240 K243 R1 K3 R7 V8 Y10 R15 R45 Q46 N53 K57 K60 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 1 ~ 18 RTKDKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQ 6es3 K 2.57 BS02 dna F 0 Y189 R190 V192 I213 K216 Q235 R238 R242 Y6 R7 V9 I30 K33 Q52 R55 R59 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 19 ~ 36 RTKDKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQ 6es3 M 2.57 BS01 dna B 0 T185 R190 V191 Y193 R198 R228 Q229 N236 K240 T2 R7 V8 Y10 R15 R45 Q46 N53 K57 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 1 ~ 18 RTKDKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQ 6es3 M 2.57 BS02 dna E 0 Y189 R190 V192 I213 K216 Q235 R238 R242 Y6 R7 V9 I30 K33 Q52 R55 R59 ? 0000981,0003677,0006355 remove_due_to_license_issue Q99626 29638214 19 ~ 36 RTKDKYRVVYTDHQRLELEKEFHYSRYITIRRKAELAATLGLSERQVKIWFQNRRAKERKINKKKLQQQQQQ 6esj A 2.97985 BS01 PRM A 1 W82 G116 G117 S198 W231 P285 L286 S287 Y332 H438 W80 G114 G115 S196 W229 P283 L284 S285 Y330 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 29186056 608 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6esm A 1.104 BS06 B9Z A 1 G186 L187 A189 H226 Q227 H230 H236 L243 P246 M247 Y248 R249 G75 L76 A78 H115 Q116 H119 H125 L132 P135 M136 Y137 R138 3.4.24.35 0004222,0006508,0008237,0008270,0031012 remove_due_to_license_issue IC50=2960nM P14780 29727184 306 GDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 6esn A 1.84 BS02 BWE A 1 Q286 L287 H323 M365 R367 A368 V376 F377 F378 E379 F388 I400 F401 S404 Q29 L30 H66 M108 R110 A111 V119 F120 F121 E122 F131 I143 F144 S147 ? 0003677,0004879,0005634,0006355 ic50=0.009uM remove_due_to_license_issue IC50=63nM P51449 30095900 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 6esy A 2.8 BS01 TFX A 1 G117 T120 W231 L286 G115 T118 W229 L284 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue Ki=3.62e+3nM P06276 29186056 612 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6esy A 2.8 BS02 TFX A 2 W82 P285 F329 Y332 W80 P283 F327 Y330 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue Ki=3.62e+3nM P06276 29186056 613 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6et8 A 1.7 BS01 BWH A 1 Y2 F16 W27 L60 L71 N75 H78 T88 I95 T99 L130 M131 W133 P134 V137 W162 Y169 R181 M191 G193 T194 Y3 F17 W28 L61 L72 N76 H79 T89 I96 T100 L131 M132 W134 P135 V138 W163 Y170 R182 M192 G194 T195 ? Kd=5.6nM remove_due_to_license_issue Q8KRS7 30082794 301 HMYDRWFSQQELQVLPFAEQDEQRNQTWLELVGEAQQLMGERCPADEPRAIALATRWMEQLEQDTAGRPEFLTRLNEMHAAEPQMREQTGVTPEMIDFITRAFAESKLAIWARYLNAEELAFTRQHYFDRLMEWPALVADLHRACREKRDPASPEGQQLAQRWLALFQSYAGKDAQTQQKFRYAMEQEPHLMKGTWMTSEVLSWLQQAIGVMMRQ 6etg A 1.279 BS02 BWT A 1 Y136 T187 T188 F189 H192 E194 H280 N284 Y126 T177 T178 F179 H182 E184 H270 N274 1.14.11.66 remove_due_to_license_issue Q6B0I6 31475772 415 AQNPNCNIMIFHPTKEEFNDFDKYIAYMESQGAHRAGLAKIIPPKEWKARETYDNISEILIATPLQQVASGRAGVFTQYHKKKKAMTVGEYRHLANSKKYQTPPHQNFEDLERKYWKNRIYNSPIYGADISGSLFDENTKQWNLGHLGTIQDLLEKECGVVIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHLGEPKTWYVVPPEHGQRLERLARELFPGSSRGCGAFLRHKVALISPTVLKENGIPFNRITQEAGEFMVTFPYGYHAGFNHGFNCAEAINFATPRWIDYGKMASQCSCGEARVTFSMDAFVRILQPERYDLWKRGQD 6etj A 2.51 BS02 BWW A 1 V70 G71 R74 F87 M95 R98 A125 T126 N127 R132 Y193 V58 G59 R62 F75 M83 R86 A113 T114 N115 R120 Y181 R252 H253 N259 S302 E322 H387 R240 H241 N247 S290 E310 H375 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 remove_due_to_license_issue Q16875 30250201 603 ELTQSRVQKIWVPVDHRPSLSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRER 6ets A 1.333 BS02 I1L A 1 Y136 F189 H192 E194 S200 H280 Y126 F179 H182 E184 S190 H270 1.14.11.66 remove_due_to_license_issue Q6B0I6 31475772 416 AQNPNCNIMIFHPTKEEFNDFDKYIAYMESQGAHRAGLAKIIPPKEWKARETYDNISEILIATPLQQVASGRAGVFTQYHKKKKAMTVGEYRHLANSKKYQTPPHQNFEDLERKYWKNRIYNSPIYGADISGSLFDENTKQWNLGHLGTIQDLLEKECGVVIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHLGEPKTWYVVPPEHGQRLERLARELFPGSSRGCGAFLRHKVALISPTVLKENGIPFNRITQEAGEFMVTFPYGYHAGFNHGFNCAEAINFATPRWIDYGKMASQCSCGEARVTFSMDAFVRILQPERYDLWKRGQ 6ety A 1.68 BS04 BXK A 1 R210 N257 E424 L428 S454 G518 Y552 H553 K699 Y700 R156 N203 E370 L374 S400 G464 Y498 H499 K645 Y646 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue IC50=8.9nM Q04609 30552009 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6eu6 A 1.98 BS01 ZDM A 1 P187 L314 K315 P187 L314 K315 2.7.13.3 0005886,0008519,0016020,0072488 remove_due_to_license_issue Q1Q357 29323112 503 MENIQININHLWVIMAACMVFLMQLGFTSYETGFSQSKNAISIALRNLVDTLISSLVFFSVGFGFMFGKSYMGLIGIDLFFANDLALHPNTLSYSFFFFQMVFASTAATILTGAIAERSGFIPNIAGTAFIVAIIYPIFGHWAWGNLFSPDQTGWLKELGFIDFAGATVVHSIGGWFAMAAAIMVGPRIDKYNPDGSSNRIGLHNVPLATLGTFFLWFGWFGFNGGSLLRVSVNIGLVILNTNMAAASAGVSALIFIYATRKRIEAGSLFTAILAGLVAITASSNMVTPVSAVAIGLITGILAIIAEGFIEKTLKIDDPVSAIAVHGVGGVIGTLCVAIFAQKSYLLAENGSRMHQLGIQALGVIVAFSWSFGLGMLFFLCLKKVKRLRVTPEEEKRGLNVAEAA 6euc A 2.21999 BS01 RM0 A 1 Y70 G118 Y121 W279 F330 F331 Y67 G115 Y118 W276 F327 F328 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29672968 604 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6eum A 1.18 BS03 BY5 A 1 W89 H118 D120 H179 C198 N210 H240 W54 H83 D85 H144 C163 N175 H205 H116 H118 D120 H179 C198 K201 N210 H240 H81 H83 D85 H144 C163 K166 N175 H205 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.3uM remove_due_to_license_issue IC50=300nM P04190 29655609 304 KTVIKNETGTISISQLNKNVWVHTELGSFNGEAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 6euv A 2.7 BS01 21G A 1 F323 R355 H357 E361 K376 F404 Q406 M431 N510 V511 F72 R104 H106 E110 K125 F153 Q155 M180 N255 V256 ? remove_due_to_license_issue P31345 29202182 601 NDDIDQSLIIAARNIVRRASVSADPLASLLEMCHSTQIGGTRMVDILRQNPTEEQAVDICKAAMGLRISSSFSFGGFTFKRTSGSSIKREEEVLTGNLQTLKIRVHEGYEEFTMVGKRATAILRKATRRLVQLIVSGRDEQSIAEAIIVAMVFSQEDCMIKAVRGDLNFVNRANQRLNPMHQLLRHFQKDAKVLFQNWGIEHIDNVMGMVGVLPDMTPSTEMSMRGIRVSKMGVSTERVVVSIDRFLRVRDQRGNVLLSPEEVSETHGTERLTITYS 6euv A 2.7 BS02 21G A 2 H285 R293 R299 H34 R42 R48 ? remove_due_to_license_issue P31345 29202182 602 NDDIDQSLIIAARNIVRRASVSADPLASLLEMCHSTQIGGTRMVDILRQNPTEEQAVDICKAAMGLRISSSFSFGGFTFKRTSGSSIKREEEVLTGNLQTLKIRVHEGYEEFTMVGKRATAILRKATRRLVQLIVSGRDEQSIAEAIIVAMVFSQEDCMIKAVRGDLNFVNRANQRLNPMHQLLRHFQKDAKVLFQNWGIEHIDNVMGMVGVLPDMTPSTEMSMRGIRVSKMGVSTERVVVSIDRFLRVRDQRGNVLLSPEEVSETHGTERLTITYS 6euw A 1.0 BS01 BYB A 1 I319 S320 F323 R332 H357 E361 F363 K376 F404 Q406 M427 H428 I1 S2 F5 R14 H39 E43 F45 K58 F86 Q88 M105 H106 ? Kd=0.017uM remove_due_to_license_issue Q2LG68 29202182 501 ISSSFSFGGFTFKRTSGSSVKKEEEVLTGNLQTLKIRVHEGYEEFTMVGRRATAILRKATRRLIQLIVSGRDEQSIAEAIIVAMVFSQEDCMIKAVRGDLNLNPMHQLLRHFQKDAKVLFQNWGIEPIDNVMGMIGILPDMTPSTEMSLRGVRVSK 6eux A 2.05 BS01 BYB A 1 Q325 W359 E363 K378 F406 E511 Q40 W74 E78 K93 F121 E217 ? remove_due_to_license_issue Q5V8X3 29202182 601 SQSMIVACRKIIRRSIVPLELAVEIANVACDIIRAALGRQRFGRLELKRISGRGFKNDEEILIGNGTIQKIGIWDGEEEFHVRCGECRGILKKSKMKLEKLLINSAKKEDMRDLIILCMVFSQDTRMFQGVRGEINFLNRAGQLLSPMYQLQRYFLNRSNDLFDQWGYEESPKASELHGINESMNASDYTLKGVVVTRNVIDDFITKNLSLIKRTGEVIMGANDV 6euz A 1.95 BS01 C8Q B 1 S127 F131 S126 F130 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue IC50=65600nM P22262 29667825 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6euz B 1.95 BS01 C8Q B 1 L60 Q61 Y126 K130 F131 S142 S177 S178 G179 L59 Q60 Y125 K129 F130 S141 S176 S177 G178 ? 0003677,0003700,0005829,0006355 ic50=65.6uM remove_due_to_license_issue IC50=65600nM P22262 29667825 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGYSSGIAHSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6ev0 A 2.3 BS01 BYK A 1 Q61 Y62 Y63 K64 F67 Y126 I149 C229 Q60 Y61 Y62 K63 F66 Y125 I148 C222 ? 0003677,0003700,0005829,0006355 ic50=1.8uM remove_due_to_license_issue P22262 29667825 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGYSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6ev0 B 2.3 BS01 BYK B 1 Q61 Y62 Y63 F67 Y126 I149 W224 C229 Q60 Y61 Y62 F66 Y125 I148 W223 C228 ? 0003677,0003700,0005829,0006355 ic50=1.8uM remove_due_to_license_issue P22262 29667825 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGYSSGIAHSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6evq A -1.00 BS01 C05 A 1 L246 Y247 L56 Y57 ? 0008017 remove_due_to_license_issue Q61166 29138501 301 DEAAELMQQVKVLKLTVEDLEKERDFYFGKLRNIELICQENEGENDPVLQRIVDILYATDEGFVIPDEGG 6evq B -1.00 BS01 C05 B 1 L246 Y247 L56 Y57 ? 0008017 remove_due_to_license_issue Q61166 29138501 301 DEAAELMQQVKVLKLTVEDLEKERDFYFGKLRNIELICQENEGENDPVLQRIVDILYATDEGFVIPDEGG 6evr A 1.5 BS02 BZW A 1 Q92 H94 H119 L131 A132 A135 L198 T199 H200 P202 W209 Q89 H91 H116 L128 A129 A132 L195 T196 H197 P199 W206 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=8.8nM remove_due_to_license_issue Ki=8.8nM P00915 29635168 302 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6ew3 A 2.14 BS03 S3C A 1 W87 H116 D118 H179 C198 N210 H240 W56 H85 D87 H148 C167 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=0.04uM remove_due_to_license_issue D1MEN9 29655609 506 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6ew6 A 1.39 BS01 C0H A 1 M51 A52 C53 G55 Y58 M46 A47 C48 G50 Y53 ? Kd>829uM remove_due_to_license_issue P41182 30335946 201 DSQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTARKFIKAS 6ew7 A 1.6 BS01 C1W A 1 M51 A52 S54 G55 Y58 M45 A46 S48 G49 Y52 ? ic50=2.9uM remove_due_to_license_issue P41182 30335946 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6ew7 A 1.6 BS02 C1W B 1 N21 R24 L25 N15 R18 L19 ? ic50=2.9uM remove_due_to_license_issue P41182 30335946 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6ew7 B 1.6 BS01 C1W A 1 N21 L25 N15 L19 ? ic50=2.9uM remove_due_to_license_issue P41182 30335946 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6ew7 B 1.6 BS02 C1W B 1 M51 A52 S54 G55 Y58 M45 A46 S48 G49 Y52 ? ic50=2.9uM remove_due_to_license_issue P41182 30335946 202 SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAHKTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNILLDFMYTSRLNLREGNIMAVMATAMYLQMEHVVDTCRKFIKAS 6ewe A 1.46 BS03 C0W A 1 H118 D120 H179 C198 N210 D213 H240 H79 D81 H140 C159 N171 D174 H201 H116 H118 D120 H179 C198 K201 N210 H240 H77 H79 D81 H140 C159 K162 N171 H201 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=3.1uM remove_due_to_license_issue IC50=3100nM P04190 29655609 304 KTVIKNETGTISISQLNKNVWVHTELGSAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 6ewk A 2.22 BS01 RM0 A 1 Y70 G118 Y121 W279 F330 F331 Y67 G115 Y118 W276 F327 F328 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29672968 604 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6ex1 A 1.6 BS02 N19 A 1 Q92 H94 H119 L198 T199 H200 Q89 H91 H116 L195 T196 H197 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=49.4nM remove_due_to_license_issue Ki=49nM P00915 29635168 302 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6exi A 1.918 BS01 ADN A 1 H58 T60 Q62 D231 H342 N385 L386 G391 H392 M397 H53 T55 Q57 D226 H337 N380 L381 G386 H387 M392 H58 S81 S86 D135 E197 N222 K227 D231 N232 C236 H342 H392 S400 Q404 H53 S76 S81 D130 E192 N217 K222 D226 N227 C231 H337 H387 S395 Q399 3.13.2.1 0004013,0005737,0005829,0006730,0016787,0033353,0071269 remove_due_to_license_issue A0A087WNH6 29619018 502 GFTDYIVKDIALADFGRKEISLAETEMPGLMATREEYGPKQPLKGARIAGSLHMTIQTAVLIETLAALGADIRWVSCNIYSTQDHAAAAIAAAGIPVFAVKGETLTEYWDYTAKLFDWHGGGTPNMILDDGGDATMLVHAGYRAEQGDTAFLDKPGSEEEEIFYALVKRLLKEKPKGWFAEIAKNIKGVSEETTTGVHRLYEMANKGTLLFPAINVNDSVTKSKFDNLYGCRESLVDGIRRGTDVMLSGKVAMVAGFGDVGKGSAASLRQAGCRVMVSEVDPICALQAAMEGYEVVTMEDAAPRADIFVTATGNKDIITIEHMRAMKDRAIVCNIGHFDNEIQIASLRNLKWTNIKPQVDEIEFPDKHRIIMLSEGRLVNLGNAMGHPSFVMSASFTNQTLAQIELFANNKDSKYAKKVYVLPKTLDEKVARLHLAKIGVKLTELRKDQADYIGVKQEGPYKSDHYRY 6exi A 1.918 BS02 ADN A 2 E284 V285 T317 N319 I322 E279 V280 T312 N314 I317 H58 S81 S86 D135 E197 N222 K227 D231 N232 C236 H342 H392 S400 Q404 H53 S76 S81 D130 E192 N217 K222 D226 N227 C231 H337 H387 S395 Q399 3.13.2.1 0004013,0005737,0005829,0006730,0016787,0033353,0071269 remove_due_to_license_issue A0A087WNH6 29619018 503 GFTDYIVKDIALADFGRKEISLAETEMPGLMATREEYGPKQPLKGARIAGSLHMTIQTAVLIETLAALGADIRWVSCNIYSTQDHAAAAIAAAGIPVFAVKGETLTEYWDYTAKLFDWHGGGTPNMILDDGGDATMLVHAGYRAEQGDTAFLDKPGSEEEEIFYALVKRLLKEKPKGWFAEIAKNIKGVSEETTTGVHRLYEMANKGTLLFPAINVNDSVTKSKFDNLYGCRESLVDGIRRGTDVMLSGKVAMVAGFGDVGKGSAASLRQAGCRVMVSEVDPICALQAAMEGYEVVTMEDAAPRADIFVTATGNKDIITIEHMRAMKDRAIVCNIGHFDNEIQIASLRNLKWTNIKPQVDEIEFPDKHRIIMLSEGRLVNLGNAMGHPSFVMSASFTNQTLAQIELFANNKDSKYAKKVYVLPKTLDEKVARLHLAKIGVKLTELRKDQADYIGVKQEGPYKSDHYRY 6exm A 1.6 BS01 QQH A 1 Y62 Y63 K64 F67 K122 Y126 Q146 I149 W224 C229 Y61 Y62 K63 F66 K121 Y125 Q145 I148 W223 C228 ? 0003677,0003700,0005829,0006355 ic50=3uM remove_due_to_license_issue P22262 29667825 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGYSSGIAHSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6exm B 1.6 BS01 QQH B 1 Y62 Y63 F67 Y126 W224 C229 Y61 Y62 F66 Y125 W216 C221 ? 0003677,0003700,0005829,0006355 ic50=3uM remove_due_to_license_issue P22262 29667825 301 NAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELGYSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6exs A 2.5 BS01 C3H A 1 Y41 N167 A170 Q310 G313 S314 F343 Q344 N347 P348 Y411 Y33 N159 A162 Q302 G305 S306 F335 Q336 N339 P340 Y403 0006857,0015833,0016020,0022857,0055085,1904680 ic50=362uM remove_due_to_license_issue 29966586 514 QTIQSIPQKGFFGHPRGLGVLFFVEFWERFSYYGMRAMLIFYMYFAIHQNGLGIDKTTAMSIMSVYGALIYMSSIPGAWIADRITGTRGATLLGAVLIIIGHICLSLPFALFGLFSSMFFIIIGSGLMKPNISNIVGRLYPENDTRIDAGFVIFYMSVNLGALISPIILQHFVDIRNFHGGFLLAAIGMALGLVWYLLFNRKNLGSVGMAPTNPLSKEEKRKYGMIIGIIVAIVIVVLLVTYYTHTLSFDLISNTVLVLGVALPIIYFTTMLRSKDVTDGERSRVKAFIPLFILGMLFWSIQEQGSNVLNIYGLERSDMQLNLFGWTTRFGEALFQSINPLFILLFAPVISMIWLKMGKKQPSLAIKFSIGTLLAGLSYILIGLVGLGYGHTQFSVNWVILSYVICVIGELCLSPTGNSAAVKLAPKAFNAQMMSVWLLTNASAQAINGTLVKLIKPLGQTNYFIFLGTVAIVITLIILVFSPKITK 6ey7 A 2.9 BS03 C3W A 1 F466 S473 N536 M579 G580 F38 S43 N106 M149 G150 3.1.-.- 0051276 remove_due_to_license_issue P16732 31458978 704 LITDQSREEFDILRYSTLNTNAYDYFGKTLYVYLDPAFTRKASGTGVAAVGAYRHQFLIYGLEHFFLRDLSESSEVAIAECAAHMIISVLSLHPYLDELRIAVEGNTNQAAAVRIACLIRQSVQSSTLIRVLFYHTPDQNHIEQPFYLMGRDKALAVEQFISRFNSGYIKASQELVSYTIKLSHDPIEYLLEQIQNLHRSDDLIIAVIMATYLCDDIHAIRFRVS 6ey8 A 2.16 BS01 C4T A 1 N51 A55 D93 G97 M98 L103 L107 F138 T184 N35 A39 D77 G81 M82 L87 L91 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=1.55uM remove_due_to_license_issue P07900 29768913 302 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6ey9 A 2.0 BS01 C4N A 1 N51 A55 D93 G97 M98 N106 F138 W162 T184 N36 A40 D78 G82 M83 N91 F123 W147 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=1.24uM remove_due_to_license_issue P07900 29768913 302 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6eya A 2.1 BS01 C4K A 1 N51 D54 A55 D93 M98 N106 F138 W162 T184 N35 D38 A39 D77 M82 N90 F118 W142 T164 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=33nM remove_due_to_license_issue P07900 29768913 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6eyb A 1.9 BS01 C3Z A 1 N51 A55 D93 G97 M98 F138 T184 N35 A39 D77 G81 M82 F122 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=4.22uM remove_due_to_license_issue P07900 29768913 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6eyt A 2.21 BS02 UDP A 1 Q51 W52 F53 Y75 F190 D226 A227 D228 S327 S332 S333 W334 R335 Q25 W26 F27 Y49 F164 D200 A201 D202 S301 S306 S307 W308 R309 ? 0000166,0016740,0046872 remove_due_to_license_issue A0A0H3NMP8 29449376 404 SGSANFAGVEYPLLPLDQHTPLLFQWFERNPSRFGENQIPIINTQQNPYLNNIINAAIIEKERTIGVLVDGNFSAGQKKALAKLEKQYENIKVIYNSDLDYSMYDKKLSDIYLENIAKIEAQPANVRDEYLLGEIKKSLNEVLKNNPEESLVSSHDKRLGHVRFDFYRNLFLLKGSNAFLEAGKHGCHHLQPGGGCIYLDADMLLTGKLGTLYLPDGIAVHVSRKGNSMSLENGIIAVNRSEHPALKKGLEIMHSKPYGDPYIDGVCGGLRHYFNCSIRHNYEEFCNFIEFKHEHIFMDTSSLTISSWR 6eyz A 2.2 BS01 C5W A 1 M752 W760 I777 K779 D787 I825 V827 V828 M900 D911 M590 W598 I615 K617 D625 I663 V665 V666 M738 D749 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 29232121 1101 DRVKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSARGNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLVEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNPASLWSLEQPFSIELIEGRKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPHPVYFPALEKILELGRHGERRITEEEQLQLREILERGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVN 6ez6 A 2.04 BS01 C5Z A 1 S754 W760 I777 K779 D787 I825 V827 M900 D911 S593 W599 I616 K618 D626 I664 V666 M739 D750 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 29232121 1101 DRVKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSARGNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLVEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNPASLWSLEQPFSIELIEGRKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPHPVYFPALEKILELGRHGERGRITEEEQLQLREILERGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVN 6ez9 A 1.61 BS04 C68 A 1 R210 M424 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 M370 L374 G464 N465 R480 R482 Y495 H496 K642 Y643 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue IC50=17nM Q04609 30552009 820 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAMEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6ezg A 2.2 BS01 C6K A 1 Y70 W84 G118 E199 I287 F290 F330 F331 Y334 H440 Y67 W81 G115 E196 I284 F287 F327 F328 Y331 H437 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30447434 603 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6ezh A 2.6 BS01 C6H A 1 Y70 W84 G118 Y121 E199 F330 F331 Y334 Y67 W81 G115 Y118 E196 F327 F328 Y331 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30447434 603 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6ezq A 2.39 BS01 C7K A 1 Y150 L198 K199 S202 F211 W214 L238 H242 R257 A291 Y144 L192 K193 S196 F205 W208 L232 H236 R251 A285 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=14uM remove_due_to_license_issue P02768 29193545 601 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPCTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAAL 6ezq A 2.39 BS02 C7K A 2 S342 R348 L387 I388 N391 Y411 L430 L453 L457 R485 F488 S489 S336 R342 L381 I382 N385 Y405 L424 L447 L451 R479 F482 S483 ? 0003677,0005504,0005507,0005515,0005576,0005615,0005634,0005737,0005783,0005788,0005794,0008289,0009267,0015643,0016209,0019825,0030170,0031093,0032991,0042802,0046872,0051087,0051902,0070062,0072562,0072732,0098869,0140272,1903981 Kd=14uM remove_due_to_license_issue P02768 29193545 602 HKSEVAHRFKDLGEENFKALVLIAFAQYLQQCPFEDHVKLVNEVTEFAKTCVADESAENCDKSLHTLFGDKLCTVATYGEMADCCAKQEPERNECFLQHKDDNPNLPRLVRPEVDVMCTAFHDNEETFLKKYLYEIARRHPYFYAPELLFFAKRYKAAFTECCQAADKAACLLPKLDELRDEGKASSAKQRLKCASLQKFGERAFKAWAVARLSQRFPKAEFAEVSKLVTDLTKVHTECCHGDLLECADDRADLAKYICENQDSISSKLKECCEKPLLEKSHCIAEVENDEMPADLPSLAADFVESKDVCKNYAEAKDVFLGMFLYEYARRHPDYSVVLLLRLAKTYETTLEKCCAAADPHECYAKVFDEFKPLVEEPQNLIKQNCELFEQLGEYKFQNALLVRYTKKVPQVSTPTLVEVSRNLGKVGSKCCKHPEAKRMPCAEDYLSVVLNQLCVLHEKTPVSDRVTKCCTESLVNRRPCFSALEVDETYVPCTLSEKERQIKKQTALVELVKHKPKATKEQLKAVMDDFAAFVEKCCKADDKETCFAEEGKKLVAASQAAL 6f05 I 2.2 BS01 GTS I 1 S12 H39 T52 V53 E65 S66 S11 H38 T51 V52 E64 S65 2.5.1.18 0000325,0004364,0004601,0004602,0005507,0005737,0005777,0005829,0005886,0006952,0009407,0009506,0009507,0009570,0009579,0009636,0010043,0016740,0043295,0046686,0048046,0098869,1901149 Ki=34uM remove_due_to_license_issue O80852 29732642 301 VLKVYGPHFASPKRALVTLIEKGVAFETIPVDLMKGEHKQPAYLALQPFGTVPAVVDGDYKIFESRAVMRYVAEKYRSQGPDLLGKTVEDRGQVEQWLDVEATTYHPPLLNLTLHIMFASDEKLIKESEEKLAGVLDVYEAHLSKSKYLAGDFVSLADLAHLPFTDYLVGPIGKAYMIKDRKHVSAWWDDISSRPAWKETVAKYSF 6f1j A 1.25 BS01 EDG A 1 R51 D52 Y75 Q120 D160 E212 R27 D28 Y51 Q96 D136 E188 3.2.1.55 0046373,0046556 Kd=24uM remove_due_to_license_issue A0A2H5BN17 30084398 401 GCALPSTYKWTSTGPLASPKSGLVALRDYSHVIYNGQHLVYGSTANTAGSYGSMNFGLFSDWSEMSSASQNTMSTGAVAPTIFYFAPKSVWILAYQWGPYAFSYRTSTDPSNANGWSSPQPLFTGTISGSSTGVIDQTVIGDSENMYLFFAGDNGHIYRASMPIGDFPGSFGSASTIVLSDSTNNLFEAVEVYTVEGQNQYLMIVEAIGANGRYFRSFTASSLGGTWTAQASTESNPFAGKANSGATWTNDISSGDLVRTNPDQTQTIDACNLQFLYQGRSTSSGGDYNLLPYQPGLLTLA 6f1n A 2.09 BS01 C8W A 1 N51 A55 I96 G97 M98 L107 T109 G135 F138 T184 N37 A41 I82 G83 M84 L93 T95 G121 F124 T170 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=0.000000064M remove_due_to_license_issue P07900 29768913 302 EEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6f1w A 1.864 BS01 CG5 A 1 I15 I23 A36 K38 M80 M82 L85 L135 I13 I19 A32 K34 M73 M75 L78 L128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.011uM remove_due_to_license_issue P48730 30832206 308 LRVGNRYRLGRKIGSGGDIYLGTDIAAGEEVAIKLECVKPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNM 6f1x A 1.9 BS01 C9Q A 1 L9 F27 N33 F72 M81 W117 D119 D120 W123 F124 L7 F25 N31 F70 M79 W115 D117 D118 W121 F122 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=0.02uM remove_due_to_license_issue IC50=20nM P36639 29485874 200 ASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6f20 A 2.0 BS01 C9E A 1 L9 N33 F72 M81 W117 D119 D120 L9 N33 F72 M81 W117 D119 D120 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 Kd=49.5uM remove_due_to_license_issue IC50=9900nM, Kd=49500nM P36639 29485874 201 MGASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6f22 A 1.55 BS01 C9B A 1 T8 L9 F27 N33 F72 M81 W117 D119 D120 T9 L10 F28 N34 F73 M82 W118 D120 D121 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=0.002uM remove_due_to_license_issue P36639 29485874 200 HMGASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6f23 A 1.84 BS01 C8Z A 1 L9 F27 F72 M81 W117 D119 D120 L12 F30 F75 M84 W120 D122 D123 3.6.1.-,3.6.1.56 0001669,0003723,0005515,0005615,0005634,0005737,0005739,0005759,0005829,0006152,0006281,0006979,0008413,0008584,0008828,0016787,0016818,0030515,0031965,0035539,0042262,0046686,0046872,0047693,0106377,0106378,0106431,0106433,0140933 ic50=0.005uM remove_due_to_license_issue EC50=63nM, IC50=5.0nM P36639 29485874 201 GSHMGASRLYTLVLVLQPQRVLLGMKKRGFGAGRWNGFGGKVQEGETIEDGARRELQEESGLTVDALHKVGQIVFEFVGEPELMDVHVFCTDSIQGTPVESDEMRPCWFQLDQIPFKDMWPDDSYWFPLLLQKKKFHGYFKFQGQDTILDYTLREVDTV 6f26 A 1.83 BS01 C9Z A 1 I15 I23 A36 K38 M80 M82 L85 D91 L135 I13 I16 A29 K31 M67 M69 L72 D78 L122 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.024uM remove_due_to_license_issue P48730 30832206 314 LRVGNRYRLGRKIGDIYLGTDIAAGEEVAIKLECVLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML 6f28 A 2.4 BS01 CG8 A 1 E15 Y63 P90 L91 T92 R97 G142 A143 T144 M190 E191 T194 Y217 E11 Y59 P86 L87 T88 R93 G138 A139 T140 M186 E187 T190 Y213 ? 0015276,0016020 Ki=2.15uM remove_due_to_license_issue Ki=2150nM P42264 29451794 302 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 6f29 A 2.6 BS01 CGW A 1 Y63 P90 L91 T92 R97 G142 A143 T144 N174 M190 E191 T194 Y59 P86 L87 T88 R93 G138 A139 T140 N170 M186 E187 T190 ? 0015276,0016020 remove_due_to_license_issue Ki=3250nM P42264 29451794 301 NRSLIVTTLLEEPFVMFRKSDRTLYGNDRFEGYCIDLLKELAHILGFSYEIRLVEDGKYGAQDDKGQWNGMVKELIDHKADLAVAPLTITHVREKAIDFSKPFMTLGVSILYRKGTPIDSADDLAKQTKIEYGAVKDGATMTFFKKSKISTFEKMWAFMSSKPSALVKNNEEGIQRTLTADYALLMESTTIEYITQRNCNLTQIGGLIDSKGYGIGTPMGSPYRDKITIAILQLQEEDKLHIMKEKWWRGSGCP 6f2n A 1.149 BS03 CF8 A 1 V69 H118 D120 H179 C198 N210 H240 V31 H80 D82 H141 C160 N172 H202 H116 H118 D120 H179 C198 K201 N210 H240 H78 H80 D82 H141 C160 K163 N172 H202 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.2uM remove_due_to_license_issue IC50=200nM P04190 29655609 304 EKTVIKNETGTISISQLNKNVWVHTELGSAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 6f34 A 3.13 BS02 ARG A 1 I40 G42 T43 G44 E115 Y116 A119 F231 A232 I234 V317 I40 G42 T43 G44 E115 Y116 A119 F228 A229 I231 V314 ? 0003333,0006865,0015171,0016020,0022857,0055085 remove_due_to_license_issue Q5L1G5 29416041 501 MNLFRKKPIQLLMKESGAKGASLRKELGAFDLTMLGIGAIIGTGIFVLTGVAAAEHAGPALVLSFILSGLACVFAALCYAEFASTVPVSGSAYTYSYATFGELIAWILGWDLILEYGVASSAVAVGWSGYFQGLLSGELPKALTSAYDPAKGTFIDLPAIIIVLFITFLLNLGAKKSARFNAVIVAIKVAVVLLFLAVGVWYVKPENWTPFMPYGFSGVATGAATVFFAYIGFDAVSTAAEEVRNPQRDMPIGIIVSLLVCTLLYIAVSLVLTGIVPYEQLNVKNPVAFALNYIHQDWVAGFISLGAIAGITTVLLVSMYGQTRLFYAISRDGLLPKVFARISPTRQVPYVNTWLTGAAVAVFAGIIPLNKLAELTNIGTLFAFITVSIGVLVLRKTQPDLKRAFRVPFVPVVPILAVLFCGYLVLQLPAMTWIGFVSWLLIGLVIYFIYGRKHSELN 6f3b A 1.4 BS02 CJK A 1 H94 H96 A135 L198 T199 H200 P202 H91 H93 A132 L195 T196 H197 P199 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=273.3nM remove_due_to_license_issue Ki=273nM P00915 29962205 302 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6f3d A 2.38 BS01 CJT A 1 M192 A211 K213 Y262 V263 Y264 M265 D272 L318 M29 A48 K50 Y90 V91 Y92 M93 D100 L146 D311 K313 A315 N316 D329 T351 D139 K141 A143 N144 D157 T172 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=4.0nM Q9NWZ3 29398441 502 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLALKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6f3e A 2.67 BS01 CJQ A 1 V200 A211 K213 Y262 M265 D272 L277 L318 D329 V37 A48 K50 Y84 M87 D94 L99 L140 D151 D311 K313 A315 N316 D329 T351 D133 K135 A137 N138 D151 T165 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=7.5nM, Ki=7.5nM Q9NWZ3 29398441 502 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLLKQQFDQEIKVMAKCQHENLVELLGFSLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLATVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6f3f A 2.41796 BS01 ADP A 1 L273 V281 A293 K295 Y340 M341 A390 L393 L193 V201 A213 K215 Y260 M261 A310 L313 D386 A390 N391 D404 D306 A310 N311 D324 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P05480 29234112 601 RMVTTFVALYDYESRTETDLSFKKGERLQIVNNTEGDWWLAHSLSTGQTGYIPSNYVAPSDSIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPTSKPQTQGLAKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMNKGSLLDFLKGETGKYLRLPQLVDMSAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEDNEYTARQGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKEPEERPTFEYLQAFLEDYFTSTEPQYQP 6f3g A 2.37 BS01 CJN A 1 M192 A211 Y262 Y264 M265 D272 L318 M27 A43 Y87 Y89 M90 D97 L143 D311 K313 A315 N316 D329 T351 D136 K138 A140 N141 D154 T170 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=69nM Q9NWZ3 29398441 501 RFHSFSFYELKNVTNNFDERPISVNKMGEGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARATVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6f3i A 2.14 BS01 CKN A 1 M192 A211 Y262 Y264 M265 D272 L277 L318 S328 D329 M23 A36 Y71 Y73 M74 D81 L86 L127 S137 D138 D311 K313 A315 N316 D329 T351 D120 K122 A124 N125 D138 T153 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=21nM Q9NWZ3 29398441 501 FHSFSFYELKNVTNNFDERGNKMGEVVYKGYVTTVAVKKLLKQQFDQEIKVMAKCQHENLVELLGFSCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6f4h A 2.0 BS01 rna B 0 Y10 N12 N13 E16 T45 L46 K47 M48 R49 Q51 F53 S84 K85 D87 S88 D89 Y9 N11 N12 E15 T44 L45 K46 M47 R48 Q50 F52 S83 K84 D86 S87 D88 ? 0003676,0003723 remove_due_to_license_issue P43332 29880797 1 ~ 22 EMLPNQTIYINNLNEKIKKEELKKSLYAIFSQFGQILDIVALKTLKMRGQAFVIFKEIGSASNALRTMQGFPFYDKPMQIAYSKSDSDIV 6f4h C 2.0 BS01 rna D 0 Y10 N12 N13 E16 K19 K24 V41 L43 T45 L46 K47 M48 R49 Q51 F53 K77 S84 K85 D87 S88 D89 Y12 N14 N15 E18 K21 K26 V43 L45 T47 L48 K49 M50 R51 Q53 F55 K79 S86 K87 D89 S90 D91 ? 0003676,0003723 remove_due_to_license_issue P43332 29880797 1 ~ 22 GAMEMLPNQTIYINNLNEKIKKEELKKSLYAIFSQFGQILDIVALKTLKMRGQAFVIFKEIGSASNALRTMQGFPFYDKPMQIAYSKSDSDIVAKI 6f4h E 2.0 BS01 rna F 0 Y10 N12 N13 E16 K19 T45 L46 K47 M48 R49 Q51 F53 K77 S84 K85 D87 S88 D89 Y9 N11 N12 E15 K18 T44 L45 K46 M47 R48 Q50 F52 K76 S83 K84 D86 S87 D88 ? 0003676,0003723 remove_due_to_license_issue P43332 29880797 1 ~ 22 EMLPNQTIYINNLNEKIKKEELKKSLYAIFSQFGQILDIVALKTLKMRGQAFVIFKEIGSASNALRTMQGFPFYDKPMQIAYSKSDSDIVA 6f4n A 2.541 BS02 AKG A 1 Y272 W310 S318 H321 N327 H400 V402 W414 Y99 W137 S145 H148 N154 H225 V227 W239 1.14.11.73,3.4.-.- remove_due_to_license_issue Q8N371 29563586 502 LIPDVKLEKTVPRLHRPSLQHFREQFLVPGRPVILKGVADHWPCMQKWSLEYIQEIAGCRTVPVEVGSRYTDEEWSQTLMTVNEFISKYIVNEPRDVGYLAQHQLFDQIPELKQDISIPDYCSLGDGEEEEITINAWFGPQGTISPLHQDPQQNFLVQVMGRKYIRLYSPQESGALYPHDTHHNTSQVDVENPDLEKFPKFAKAPFLSCILSPGEILFIPVKYWHYVRALDLSFSVSFWWS 6f4w A 2.293 BS01 FMC A 1 M64 C91 G92 F159 E179 E181 D204 M64 C91 G92 F159 E179 E181 D204 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=2.95uM remove_due_to_license_issue P56463 29430816 300 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f4w A 2.293 BS02 FMC D 1 H4 R43 H4 R43 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=2.95uM remove_due_to_license_issue P56463 29430816 300 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f4w D 2.293 BS01 FMC A 1 H4 R43 H4 R43 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=2.95uM remove_due_to_license_issue P56463 29430816 300 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f4w D 2.293 BS02 FMC D 1 T90 C91 G92 F159 E181 L206 T90 C91 G92 F159 E181 L206 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=2.95uM remove_due_to_license_issue P56463 29430816 300 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f4x A 1.694 BS01 FMC A 1 M64 T90 C91 F159 E179 M180 E181 M64 T90 C91 F159 E179 M180 E181 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=10.7uM remove_due_to_license_issue P56463 29430816 301 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f4x D 1.694 BS01 FMC A 1 H4 R43 H4 R43 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=10.7uM remove_due_to_license_issue P56463 29430816 301 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f4x D 1.694 BS02 FMC D 1 M64 T90 C91 G92 F159 E181 M64 T90 C91 G92 F159 E181 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 H4 G20 R24 R43 E75 R87 T90 S203 D204 L206 R217 2.4.2.1 0003824,0004731,0005829,0006139,0006152,0009116,0009164,0016757,0016763 Kd=10.7uM remove_due_to_license_issue P56463 29430816 301 MTPHINAKIGDFYPQCLLCGDPLRVSYIAKKFLQDAKEITNVRNMLGFSGKYKGRGISLMGHGMGIASCTIYVTELIKTYQVKELLRIGTCGAISPKVGLKDIIMATGASTDSKTNRVRFLNHDLSATPDFELSLRAYQTAKRLGIDLKVGNVFSSDFFYSFETHAFDLMAKYNHLAIEMEAAGLYATAMELNAKALCLCSVSDHLITKEALSPKERVESFDNMIILALEMMS 6f5h A 2.16 BS01 CQ5 A 1 Y224 D295 Q297 M407 R408 F409 K420 H456 N460 H461 Y465 Y514 Y18 D89 Q91 M201 R202 F203 K214 H250 N254 H255 Y259 Y301 3.4.19.12 0004843,0016579 ic50=0.087uM remove_due_to_license_issue EC50=320nM, IC50=90nM Q93009 29541367 1003 SKKHTGYVGLKNQGATCYMNSLLQTLFFTNQLRKAVYMMPTEGDDSSKSVPLALQRVFYELQHSDKPVGTKKLTKSFGWETLDSFMQHDVQELCRVLLDNVENKMKGTCVEGTIPKLFRGKMVSYIQCKEVDYRSDRREDYYDIQLSIKGKKNIFESFVDYVAVEQLDGDNKYDAGEHGLQEAEKGVKFLTLPPVLHLQLMRFMYDPQTDQNIKINDRFEFPEQLPLDEFLQKTDPKDPANYILHAVLVHSGDNHGGHYVVYLNPKGDGKWCKFDDDVVSRCTKEEAIEHNYGGRHCTNAYMLVYIRESKLSEVLQAVTDHDIPQQLVERLQEEKRIEAQKRKERQEHHH 6f5l A 1.63 BS04 CQB A 1 R210 N257 E424 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 N203 E370 L374 G464 N465 R480 R482 Y495 H496 K642 Y643 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue IC50=0.650000nM Q04609 30552009 823 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6f5m A 2.7 BS02 CQH A 1 N61 V62 N62A N45 V46 N47 H57 D102 F192 G193 D194 S195 G196 H41 D88 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 remove_due_to_license_issue P08246 30084397 414 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 6f5m A 2.7 BS03 CQH B 1 G39 H40 N148 G150 I151 G23 H24 N133 G135 I136 H57 D102 F192 G193 D194 S195 G196 H41 D88 F170 G171 D172 S173 G174 3.4.21.37 0000122,0001878,0002020,0002438,0002523,0002812,0003714,0004175,0004252,0005515,0005576,0005615,0005737,0005829,0006508,0006874,0006909,0008201,0008233,0008236,0009411,0009986,0017053,0019955,0022617,0030141,0030163,0031410,0032496,0032682,0032717,0032757,0035578,0035580,0042742,0043406,0045335,0048661,0050728,0050778,0050832,0050900,0050922,0062023,0070062,0070269,0070945,0070947,1903238 remove_due_to_license_issue P08246 30084397 301 IVGGRRARPHAWPFMVSLQLRGGHFCGATLIAPNFVMSAAHCVANVNVRAVRVVLGAHNLSRREPTRQVFAVQRIFENGYDPVNLLNDIVILQLNGSATINANVQVAQLPAQGRRLGNGVQCLAMGWGLLGRNRGIASVLQELNVTVVTSLCRRSNVCTLVRGRQAGVCFGDSGSPLVCNGLIHGIASFVRGGCASGLYPDAFAPVAQFVNWIDSIIQ 6f5u A 2.07 BS01 CQN A 1 R64 V66 A101 R33 V35 A70 ? Kd=0.29mM remove_due_to_license_issue Q05320 29272110 610 SIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQASGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTWAFWELSFTVVAAAAAAA 6f5u B 2.07 BS01 CQN A 1 L515 Y517 M548 L558 L14 Y16 M47 L57 ? remove_due_to_license_issue Q05320 29272110 610 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFVD 6f5w A 1.91 BS01 KG1 A 1 Q77 G98 T99 W104 W118 Q52 G73 T74 W79 W93 ? 0046872 Kd=149uM remove_due_to_license_issue C7BLE4 29341313 413 TIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 6f5w A 1.91 BS02 KG1 A 2 G171 V172 G193 T194 W199 G146 V147 G168 T169 W174 ? 0046872 Kd=149uM remove_due_to_license_issue C7BLE4 29341313 414 TIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 6f5w A 1.91 BS03 KG1 A 3 G267 V268 G289 T290 W295 G242 V243 G264 T265 W270 ? 0046872 Kd=149uM remove_due_to_license_issue C7BLE4 29341313 415 TIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 6f5w A 1.91 BS04 KG1 A 4 G315 V316 G337 T338 W343 G290 V291 G312 T313 W318 ? 0046872 Kd=149uM remove_due_to_license_issue C7BLE4 29341313 416 TIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 6f5w A 1.91 BS05 KG1 A 5 G49 T50 W55 G360 V361 G24 T25 W30 G335 V336 ? 0046872 Kd=149uM remove_due_to_license_issue C7BLE4 29341313 417 TIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 6f5w A 1.91 BS06 KG1 A 6 R186 E188 W202 Q251 G257 W259 R161 E163 W177 Q226 G232 W234 ? 0046872 Kd=149uM remove_due_to_license_issue C7BLE4 29341313 418 TIALSEIVSVVNTSDGRLEVFGVGTDKAVWHNRQMAPHTGSPWSGWSSLKGQVTSKPVVYINTDGRLEVFARGTDNALWHIWQTATNAGWSNWQSLGGVITSNPAIYANTDGRLEVFARGADNALWHISQTTAHSGPWSSWASLNGVITSNPTVHINSDGRLEVFARGTDNALWHIWQTAPDSNLWSSWESLNGIITSDPVVIDTADGRLEVFARGADNALWHIWQTISHSGPWSGWQSLNGVITSAPAVAKNCDNRLEAFARGTDNALWHTWQTVSHSGPWSSWQSLNGVITSAPTAVRDADGRLEVFARGTDNALWLTWQTASSWSPWISLGGVLIDASAIK 6f6i A 2.4 BS01 8PR A 1 R64 V66 L68 A101 G102 R34 V36 L38 A71 G72 ? Kd=0.65mM remove_due_to_license_issue Kd=650000nM Q05320 29272110 509 RSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQASGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTWAFWETLSFTVVAAAAAAA 6f6i B 2.4 BS01 8PR A 1 L515 Y517 M548 L14 Y16 M47 ? remove_due_to_license_issue Kd=650000nM Q05320 29272110 509 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFVD 6f6n A 2.15 BS01 SRE A 1 R64 V66 A101 R33 V35 A70 ? Kd=0.95mM remove_due_to_license_issue Kd=950000nM Q05320 29272110 508 SIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTWAFWETSEELSFTVVAAAAAAA 6f6n B 2.15 BS01 SRE A 1 Y517 M548 L558 Y16 M47 L57 ? remove_due_to_license_issue Kd=950000nM Q05320 29272110 508 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFVD 6f6r A 1.8 BS01 CVE A 1 R179 Q283 C285 R62 Q166 C168 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 29648825 501 QDNPAMPTSSGSEGNVKLCSLEEAQRIWKQKSAEIYPIMDKSSRTRLALIICNEEFDSIPRRTGAEVDITGMTMLLQNLGYSVDVKKNLTASDMTTELEAFAHRPEHKTSDSTFLVFMSHGIREGICGKKHSEQVPDILQLNAIFNMLNTKNCPSLKDKPKVIIIQACRGDSPGVVWFKD 6f6r B 1.8 BS01 CVE A 1 S339 W340 R341 H342 M345 V348 R383 S23 W24 R25 H26 M29 V32 R67 E390 E74 3.4.22.36 0004197,0006508,0008234 remove_due_to_license_issue P29466 29648825 501 AIKKAHIEKDFIAFCSSTPDNVSWRHPTMGSVFIGRLIEHMQEYACSCDVEEIFRKVRFSFEQPDGRAQMPTTERVTLTRCFYLFPGH 6f6s A 2.29 BS01 CXQ B 1 L184 L186 L154 L156 ? Kd=1.3mM remove_due_to_license_issue Q05320 29272110 705 RSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTWAFWETELSFTVVAAAAAA 6f6s B 2.29 BS01 CXQ A 1 Y517 I544 Y16 I41 ? Kd=1.3mM remove_due_to_license_issue Q05320 29272110 507 EAIVNAQPKCNPNLHYWTTQDAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFVD 6f6s B 2.29 BS02 CXQ B 1 Y517 M548 L554 Y16 M45 L51 ? Kd=1.3mM remove_due_to_license_issue Q05320 29272110 705 EAIVNAQPKCNPNLHYWTTQDAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFVD 6f6u A 1.828 BS02 CV8 A 1 Y325 S374 M439 T499 I502 F506 Q535 F538 Y76 S125 M190 T250 I253 F257 Q286 F289 3.1.4.53 0004114,0007165,0008081 ic50=16uM remove_due_to_license_issue Q08499 29652483 604 VKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6f7b A 2.0 BS01 CVQ A 1 V801 V819 K821 E830 G834 F849 M850 F852 L864 Y869 I924 I945 D946 L947 V69 V81 K83 E92 G96 F111 M112 F114 L126 Y131 I186 I207 D208 L209 2.7.11.1 0004672,0005524,0006468,0007094 remove_due_to_license_issue O43683 30429199 1101 APNFIVGNPWDDKLIFKLLSGLSKPVSSYPNTFEWQCKLPAIKPKTEFQLGSKLVYVHHLLGEGAFAQVYEATQKNKQKFVLKVQKPANPWEFYIGTQLMERLKPSMQHMFMKFYSAHLFQNGSVLVGELYSYGTLLNAINLYKNTPEKVMPQGLVISFAMRMLYMIEQVHDCEIIHGDIKPDNFILGNGFLEQDDEDDLSAGLALIDLGQSIDMKLFPKGTIFTAKCETSGFQCVEMLSNKPWNYQIDYFGVAATVYCMLFGTYMKVKNEECKPEGLFRRLPHLDMWNEFFHVMLNIPDCHHLPSLDLLRQKLKKVFQQHYTNKIRALRNRLIVLLLECKRS 6f7c B 2.002 BS02 CVT B 1 C241 L242 A250 D251 L255 N258 V315 A316 I318 K352 C238 L239 A247 D248 L252 N255 V309 A310 I312 K346 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Q6B856 31655259 503 REIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 6f7i A 2.43 BS01 CW5 A 1 V344 A345 K379 V381 E390 N393 A394 E397 L401 Q579 W580 Q676 I712 L715 D716 V8 A9 K43 V45 E54 N57 A58 E61 L65 Q218 W219 Q315 I351 L354 D355 3.4.22.- 0004197,0006508 remove_due_to_license_issue Q9UDY8 30692685 801 QPLAKDKVALLIGNMNYREHPKLKAPLVDVYELTNLLRQLDFKVVSLLDLTEYEMRNAVDEFLLLLDKGVYGLLYYAGHGYENFGNSFMVPVDAPNPYRSENCLCVQNILKLMQEKETGLNVFLLDMCRVTANIVFGYATCQSGLANGIFMKFLKDRLLEDKKITVLLDEVAEDMGKCHLTKGKQALEIRSSLSEKRALTDPIQGTEYSAESLVRNLQWAKAHELPESMCLKFDCGVQIQLGFAAEFSNVMIIYTSIVYKPPEIIMCDAYVTDFPLDLDIDPKDANKGTPEETGSYLVSKDLPKHCLYTRLSSLQKLKEHLVFTVCLSYQYSGLEDTVEDKQEVNVGKPLIAKLD 6f7q A 2.6 BS02 CWQ A 1 H372 Y373 D375 V377 Q517 Q518 H370 Y371 D373 V375 Q515 Q516 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30031971 601 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6f7q A 2.6 BS03 CWQ A 2 I69 D70 W82 G116 G117 T120 S198 W231 L286 F329 Y332 H438 I67 D68 W80 G114 G115 T118 S196 W229 L284 F327 Y330 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30031971 602 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6f7q A 2.6 BS04 CWQ B 1 I462 S466 S507 T508 I460 S464 S505 T506 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30031971 601 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6f7q B 2.6 BS02 CWQ A 1 I462 S466 E506 T508 I460 S464 E504 T506 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30031971 601 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6f7q B 2.6 BS03 CWQ B 1 H372 Y373 D375 V377 Q517 Q518 H370 Y371 D373 V375 Q515 Q516 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30031971 601 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6f7q B 2.6 BS04 CWQ B 2 D70 W82 G116 G117 T120 S198 V288 H438 D68 W80 G114 G115 T118 S196 V286 H436 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G114 G115 G147 S196 A197 Y235 V286 F288 E323 H436 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30031971 602 DIIIATKNGKVRGMNLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDNYTKAEEILSRSIVKRWANFAKYGNPNETQNNSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6f86 A 1.9 BS01 CWW A 1 V43 E50 V71 D73 R76 G77 I78 P79 R136 T165 V29 E36 V57 D59 R62 G63 I64 P65 R104 T133 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.037uM remove_due_to_license_issue P0AES6 31257079 500 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 6f8b A 1.3 BS03 CXH A 1 H140 E141 R198 H223 H140 E141 R198 H223 H140 E141 H144 Y155 E164 D221 H223 H140 E141 H144 Y155 E164 D221 H223 3.4.24.26 0004222,0006508 ic50=6.6uM remove_due_to_license_issue IC50=6600nM P14756 29485268 403 AEAGGPGGNQKIGKYTYGSDYGPLIVNDRCEMDDGNVITVDMNSSTDDSKTTPFRFACPTNTYKQVNGAYSPLNDAHFFGGVVFKLYRDWFGTSPLTHKLYMKVHYGRSVENAYWDGTAMLFGDGATMFYPLVSLDVAAHEVSHGFTEQNSGLIYRGQSGGMNEAFSDMAGEAAEFYMRGKNDFLIGYDIKKGSGALRYMDQPSRDGRSIDNASQYYNGIDVHHSSGVYNRAFYLLANSPGWDTRKAFEVFVDANRYYWTATSNYNSGACGVIRSAQNRNYSAADVTRAFSTVGVTCP 6f8b A 1.3 BS04 CXH A 2 N112 V137 H140 E141 L197 N112 V137 H140 E141 L197 H140 E141 H144 Y155 E164 D221 H223 H140 E141 H144 Y155 E164 D221 H223 3.4.24.26 0004222,0006508 ic50=6.6uM remove_due_to_license_issue IC50=6600nM P14756 29485268 404 AEAGGPGGNQKIGKYTYGSDYGPLIVNDRCEMDDGNVITVDMNSSTDDSKTTPFRFACPTNTYKQVNGAYSPLNDAHFFGGVVFKLYRDWFGTSPLTHKLYMKVHYGRSVENAYWDGTAMLFGDGATMFYPLVSLDVAAHEVSHGFTEQNSGLIYRGQSGGMNEAFSDMAGEAAEFYMRGKNDFLIGYDIKKGSGALRYMDQPSRDGRSIDNASQYYNGIDVHHSSGVYNRAFYLLANSPGWDTRKAFEVFVDANRYYWTATSNYNSGACGVIRSAQNRNYSAADVTRAFSTVGVTCP 6f8j A 1.95 BS01 CZ5 A 1 V43 N46 E50 V71 D73 R76 G77 I78 P79 R136 T165 V29 N32 E36 V57 D59 R62 G63 I64 P65 R104 T133 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.086uM remove_due_to_license_issue P0AES6 31257079 500 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 6f8r A 1.826 BS01 CZK A 1 Y325 H326 S374 I502 F506 M523 Q535 F538 Y70 H71 S119 I247 F251 M268 Q280 F283 3.1.4.53 0004114,0007165,0008081 ic50=20uM remove_due_to_license_issue Q08499 29652483 601 DVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6f8t A 1.8 BS04 CZT A 1 Y325 S374 T499 I502 F506 M523 Q535 F538 Y76 S125 T250 I253 F257 M274 Q286 F289 3.1.4.53 0004114,0007165,0008081 ic50=7uM remove_due_to_license_issue Q08499 29652483 606 VKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6f8u A 2.1 BS03 CZQ A 1 S374 N487 Y495 W498 T499 I502 F506 Q509 M523 S534 Q535 F538 S119 N232 Y240 W243 T244 I247 F251 Q254 M268 S279 Q280 F283 3.1.4.53 0004114,0007165,0008081 ic50=0.8uM remove_due_to_license_issue Q08499 29652483 606 DVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6f8v A 1.85 BS03 D0B A 1 Y325 M439 D484 L485 N487 I502 F506 M523 Q535 F538 Y75 M189 D234 L235 N237 I252 F256 M273 Q285 F288 3.1.4.53 0004114,0007165,0008081 ic50=16uM remove_due_to_license_issue Q08499 29652483 605 KTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6f8w A 1.601 BS02 D0E A 1 M439 D484 L485 T499 I502 M503 F506 M523 S534 Q535 F538 M182 D227 L228 T242 I245 M246 F249 M266 S277 Q278 F281 3.1.4.53 0004114,0007165,0008081 ic50=23uM remove_due_to_license_issue Q08499 29652483 605 LAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQA 6f8x A 1.95 BS03 D08 A 1 Y325 S374 N375 M439 N487 I502 M503 F506 M523 S534 Q535 F538 Y70 S119 N120 M184 N232 I247 M248 F251 M268 S279 Q280 F283 3.1.4.53 0004114,0007165,0008081 ic50=17uM remove_due_to_license_issue Q08499 29652483 605 DVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6f90 A 2.4 BS02 MVL A 1 T91 G92 W198 W352 D353 W390 C399 M400 E535 N582 E595 D637 T72 G73 W179 W333 D334 W371 C380 M381 E516 N561 E574 D616 ? 0005975,0030246 remove_due_to_license_issue Q8A325 29717710 802 AGEITKYVNPFIGTGAIDGGLSGNNYPGATSPFGMIQLSPDTSEAPNWGDASGYDYNRNTIFGFSHTRLSGTGASDLIDITLMPTSSGRTSSAFTHDEEKARPGYYQVMLKDENINAELTTTQRNGIHRYQYPAGKDAEIILDMDHSADKGSWGRRIINSQIRILNDHAVEGYRIITGWAKLRKIYFYMEFSSPILTSTLRDGGRVHENTAVINGTNLHGCFRFGQLNGKPLTCKVALSSVSMENARQNMEQEAPHWDFDRYVAAADADWEKQLGKIEVKGTEVQKEIFYTALYHTMIQPNTMSDVNGEYMAADYTTRKVANNETHYTTFSLWDTFRASHPLYTLLEPERVTDFVKSMIRQYEYYGYLPIWQLWGQDNYCMIGNHSIPVITDAILKGIPGIDMEKAYEAVYNSSVTSHPNSPFEVWEKYGFMPENIQTQSVSITLEQAFDDWCVAQLAAKLNKDADYQRFHKRSEYYRNLFHPKTKFFQSKNDKGEWIEPFDPYQYGGNGGHPFTEGNAWQYFWYVPHNIQALMELTGGTKAFEQKLDTFFTSTYKSMNHNASGFVGQYAHGNEPSHHVAYLYNFAGQPWKTQKYVSHILNTLYNNTSSGYAGNDDCGQMSAWYVFSAMGFYPVNPADGRYIIGSPLLDECTLKLAGNKEFRIRTIRKSPEDIYIQSVTLNGKKHKDFFITHQDIMNGGTMVFKMGKKPSGWGK 6f92 A 1.9 BS02 MVL A 1 T69 G70 W184 W343 D344 W383 C392 M393 E531 D633 T65 G66 W180 W339 D340 W379 C388 M389 E527 D629 ? 0000224,0005829,0005975,0006516,0030246,0046872 remove_due_to_license_issue Q8A0Q6 29717710 804 EKLTDYVNPFVGTDGYGNVYPGAQIPFGGIQISPDTDSRFYDAASGYKYNHLTLMGFSLTHLSGTGIPDLGDFLFIPGTGEMKLEPGTHEDPDQGYRSRYSHDKEWASPNYYAVELADYGVKAEMTSGVRSGMFRFTYPESDNAFIMIDMNHTLWQSCEWSNLRMINDSTITGYKLVKGWGPERHVYFTATFSKKLTGLRFVQDKKPVIYNTSRFRSSYEAWGKNLMACISFDTKAGEEVTVKTAISAVSTDGARNNMKELDGLTFNELRAKGEALWEKELGKYTLTADRKTKETFYTSAYHAALHPFIFQDSDGQFRGLDKNIEKAEGFTNYTVFSLWDTYRALHPWFNLVQQEVNADIANSMLAHYDKSVEKMLPIWSFYGNETWCMIGYHAVSVLADMIVKEVKGFDYERAYEAMKTTAMNSNYDCLPEYREMGYVPFDKEAESVSKTLEYAYDDYCIAQAAKKLGKEDDYHYFLNRALSYQTLIDPETKYMRGRDSKGDWRTPFTPVAYQGPGSVHGWGDITEGFTMQYTWYVPQDVQGYINEAGKELFRKRLDELFTVELPDDIPGAHDIQGRIGAYWHGNEPCHHVAYLYNYLKEPWKCQKWIRTIVDRFYGNTPDALSGNDDCGQMSAWYMFNCIGFYPVAPSSNIYNIGSPCAEAITVRMSNGKNIEMTADNWSPKNLYVKELYVNGKKYDKSYLTYDDIRDGVKLRFVMSGKPNYKRAVSDEAVPPSISLPEKTMKYKSSIGFLEHHHHHH 6f92 D 1.9 BS02 MVL D 1 T69 G70 W184 W343 D344 W383 C392 M393 E531 D633 T65 G66 W180 W339 D340 W379 C388 M389 E527 D629 ? 0000224,0005829,0005975,0006516,0030246,0046872 remove_due_to_license_issue Q8A0Q6 29717710 804 EKLTDYVNPFVGTDGYGNVYPGAQIPFGGIQISPDTDSRFYDAASGYKYNHLTLMGFSLTHLSGTGIPDLGDFLFIPGTGEMKLEPGTHEDPDQGYRSRYSHDKEWASPNYYAVELADYGVKAEMTSGVRSGMFRFTYPESDNAFIMIDMNHTLWQSCEWSNLRMINDSTITGYKLVKGWGPERHVYFTATFSKKLTGLRFVQDKKPVIYNTSRFRSSYEAWGKNLMACISFDTKAGEEVTVKTAISAVSTDGARNNMKELDGLTFNELRAKGEALWEKELGKYTLTADRKTKETFYTSAYHAALHPFIFQDSDGQFRGLDKNIEKAEGFTNYTVFSLWDTYRALHPWFNLVQQEVNADIANSMLAHYDKSVEKMLPIWSFYGNETWCMIGYHAVSVLADMIVKEVKGFDYERAYEAMKTTAMNSNYDCLPEYREMGYVPFDKEAESVSKTLEYAYDDYCIAQAAKKLGKEDDYHYFLNRALSYQTLIDPETKYMRGRDSKGDWRTPFTPVAYQGPGSVHGWGDITEGFTMQYTWYVPQDVQGYINEAGKELFRKRLDELFTVELPDDIPGAHDIQGRIGAYWHGNEPCHHVAYLYNYLKEPWKCQKWIRTIVDRFYGNTPDALSGNDDCGQMSAWYMFNCIGFYPVAPSSNIYNIGSPCAEAITVRMSNGKNIEMTADNWSPKNLYVKELYVNGKKYDKSYLTYDDIRDGVKLRFVMSGKPNYKRAVSDEAVPPSISLPEKTMKYKSSIGFLEHHHHHH 6f94 A 2.35 BS01 D0H A 1 V43 A47 E50 D73 R76 G77 I78 I94 R136 V29 A33 E36 D59 R62 G63 I64 I80 R104 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.099uM remove_due_to_license_issue P0AES6 31257079 500 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 6f96 A 2.5 BS01 D0K A 1 V43 N46 E50 V71 D73 R76 G77 I78 P79 I94 R136 V29 N32 E36 V57 D59 R62 G63 I64 P65 I80 R104 5.6.2.2 0003677,0003918,0005524,0006265 ic50=0.019uM remove_due_to_license_issue P0AES6 31257079 500 GLDAVRKRPGMYIGDTDDGTGLHHMVFEVVDNAIDEALAGHCKEIIVTIHADNSVSVQDDGRGIPTGIHPEEGVSAAEVIMTVLGVGVSVVNALSQKLELVIQREGKIHRQIYEHGVPQAPLAVTGETEKTGTMVRFWPSLETFTNVTEFEYEILAKRLRELSFLNSGVSIRLRDKRDGKEDHFHYE 6f9g A 2.388 BS01 PUT A 1 Y152 M166 M170 W186 Y202 D204 D233 Y100 M114 M118 W134 Y150 D152 D181 ? Kd=2uM remove_due_to_license_issue Q88NI1 29758259 401 SARQRLQAHAETQALRIQRYFMDAYQYGNGFARLVQVLKDRGGSDLRAELTRQARASLAGNPDVIGLYLVFQPNALDQQDSHYLGQDAMGSNESGRFSLYWSQPSPGTLELEAMPETMLGDTSIGSNGAAKNRWLTCPQDTARTCMLEPYLDEVNGRQVLMTSIALPLLEHGKVVGVVGLDIGLANLQQLSVNGRRDLFDGQGQVSIATAAGLLAGNSRDDSVLGKPMDKSVADGLLRVAHPFTPIPDTAPWQVVLELPES 6f9r A 1.85 BS03 D0W A 1 Q259 H331 A332 S333 A334 H361 E362 H365 Y369 E389 D393 K489 H491 Y498 Y501 F505 Q256 H328 A329 S330 A331 H358 E359 H362 Y366 E386 D390 K486 H488 Y495 Y498 F502 H331 A332 H361 E362 H365 E389 H491 Y501 H328 A329 H358 E359 H362 E386 H488 Y498 3.4.15.1 0006508,0008237,0008241,0016020 Ki=10.6uM remove_due_to_license_issue Ki=7400nM P12821 29476645 710 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLTATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEG 6f9t A 1.6 BS03 D0Z A 1 A354 S355 A356 H383 E384 H387 H410 E411 F457 K511 H513 Y520 Y523 F527 A315 S316 A317 H344 E345 H348 H371 E372 F418 K472 H474 Y481 Y484 F488 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H474 Y484 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=14nM P12821 29476645 712 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPNS 6f9u A 1.9 BS03 D0W A 1 Q281 H353 A354 S355 A356 H383 E384 H387 E411 K511 H513 Y520 Y523 Q242 H314 A315 S316 A317 H344 E345 H348 E372 K472 H474 Y481 Y484 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H474 Y484 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=7400nM P12821 29476645 711 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPNS 6f9v A 1.69 BS02 D0Z A 1 Q259 H331 A332 S333 A334 H361 E362 H365 H388 E389 K489 H491 Y498 Y501 F505 Q255 H327 A328 S329 A330 H357 E358 H361 H384 E385 K485 H487 Y494 Y497 F501 H331 A332 H361 E362 H365 E389 H491 Y501 H327 A328 H357 E358 H361 E385 H487 Y497 3.4.15.1 0006508,0008237,0008241,0016020 Ki=171.9nM remove_due_to_license_issue Ki=14nM P12821 29476645 702 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPE 6fa2 A 2.6 BS03 D2W A 1 V7 S39 R41 D54 L56 Q70 T74 V7 S39 R41 D54 L56 Q70 T74 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 30093669 203 MTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGHEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6fa3 B 1.82 BS03 D1Z B 1 K5 V7 S39 Y40 R41 D54 I55 L56 Y71 T74 K9 V11 S43 Y44 R45 D58 I59 L60 Y75 T78 3.6.5.2 0003924,0005525,0007165,0016020 Kd=0.038uM remove_due_to_license_issue P01116 30093669 203 AFQGMTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGHEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKE 6fa4 B 2.02 BS03 D1W B 1 K5 V7 S39 Y40 R41 D54 L56 Y71 T74 K9 V11 S43 Y44 R45 D58 L60 Y75 T78 3.6.5.2 0003924,0005525,0007165,0016020 Kd=0.051uM remove_due_to_license_issue P01116 30093669 203 AFQGMTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGHEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEK 6fa5 A 2.303 BS01 ADP A 1 T322 G323 S324 G325 K326 T327 T328 R362 F558 T580 R628 T37 G38 S39 G40 K41 T42 T43 R77 F273 T295 R343 3.6.4.13 0003676,0005524 Kd=179nM remove_due_to_license_issue G0SEG4 29968674 1001 AQRTIQEVRKSLPVYAYRDAFLDAVKEYQVLILVGETGSGKTTQIPQYLHEAGYTKGNRKIACTQPRRVAAMSVAARVADEMGVRLGHEVGYSIRFEDCTSEKTILKYMTDGMLLREMVTSPDLADYSCIMIDEAHERTVHTDILLALIKDLTRARPELRLIISSATLNAEKFSAYFDDAPIFNVPGRVHPVEVYYTSAPESNYLEAALVTVFQIHATQPEGDILVFLTGQEEIERACERVEEIRRKLGKRVPEIIALPIYSNMPSEMQAKIFEPTPPGARKVVFSTNIAETSLTIDGIVYVIDSGYVKENTFSPVGTTGQSTLAVVPCSRAAANQRMGRAGRVKPGKCFRLYTKYAYLSEMDESPTPEIQRTSLSSVVLQLKALGIDDLLGFDFLDPPPTELLIKSLNMLYALGALNSAGQLTRVGRQMGEFPTEPMLAKALIAATQEGCVSEVLTIVSMLGEVGTLFFRPKDKKVHADSARARFTVRDGGDHLTLLNIYNQWVEAEYSPIWARENFLAQRSLTRARDVRDQLAKLCDRILDGSEASCGGVNNPTPILRALTAAFFLNAARLNRAGDGYRTLKNNITVYVHPSSVVRGMDPPPKVIIYHELVVTSKEYVRSVIPVEPRWLSEFG 6faa A 1.97 BS01 ADP A 1 T322 G323 S324 G325 K326 T327 T328 R362 T580 D582 T40 G41 S42 G43 K44 T45 T46 R80 T298 D300 3.6.4.13 0003676,0005524 Kd=179nM remove_due_to_license_issue G0SEG4 29968674 1001 AERAQRTIQEVRKSLPVYAYRDAFLDAVKEYQVLILVGETGSGKTTQIPQYLHEAGYTKGNRKIACTQPRRVAAMSVAARVADEMGVRLGHEVGYSIRFEDCTSEKTILKYMTDGMLLREMVTSPDLADYSCIMIDEAHERTVHTDILLALIKDLTRARPELRLIISSATLNAEKFSAYFDDAPIFNVPGRVHPVEVYYTSAPESNYLEAALVTVFQIHATQPEGDILVFLTGQEEIERACERVEEIRRKLGKRVPEIIALPIYSNMPSEMQAKIFEPTPPGARKVVFSTNIAETSLTIDGIVYVIDSGYVKENTFSPVTGQSTLAVVPCSRAAANQRMGRAGRVKPGKCFRLYTKYAYLSEMDESPTPEIQRTSLSSVVLQLKALGIDDLLGFDFLDPPPTELLIKSLNMLYALGALNSAGQLTRVGRQMGEFPTEPMLAKALIAATQEGCVSEVLTIVSMLGEVGTLFFRPKDKKVHADSARARFTVRDGGDHLTLLNIYNQWVEAEYSPIWARENFLAQRSLTRARDVRDQLAKLCDRILDGSEASCGGVNNPTPILRALTAAFFLNAARLNRAGDGYRTLKNNITVYVHPSSVVRGMDPPPKVIIYHELVVTSKEYVRSVIPVEPRWLSEFGA 6fac A 2.05 BS01 ADP A 1 T322 G323 S324 G325 K326 T327 T328 R362 F558 T580 D582 T55 G56 S57 G58 K59 T60 T61 R95 F291 T313 D315 3.6.4.13 0003676,0005524 Kd=179nM remove_due_to_license_issue G0SEG4 29968674 1001 PMTPEQRLLKQKIEEAERAQRTIQEVRKSLPVYAYRDAFLDAVKEYQVLILVGETGSGKTTQIPQYLHEAGYTKGNRKIACTQPRRVAAMSVAARVADEMGVRLGHEVGYSIRFEDCTSEKTILKYMTDGMLLREMVTSPDLADYSCIMIDEAHERTVHTDILLALIKDLTRARPELRLIISSATLNAEKFSAYFDDAPIFNVPGRVHPVEVYYTSAPESNYLEAALVTVFQIHATQPEGDILVFLTGQEEIERACERVEEIRRKLGKRVPEIIALPIYSNMPSEMQAKIFEPTPPGARKVVFSTNIAETSLTIDGIVYVIDSGYVKENTFSPVGTTGQSTLAVVPCSRAAANQRMGRAGRVKPGKCFRLYTKYAYLSEMDESPTPEIQRTSLSSVVLQLKALGIDDLLGFDFLDPPPTELLIKSLNMLYALGALNSAGQLTRVGRQMGEFPTEPMLAKALIAATQEGCVSEVLTIVSMLGEVGTLFFRPKDKKVHADSARARFTVRDGGDHLTLLNIYNQWVEAEYSPIWARENFLAQRSLTRARDVRDQLAKLCDRILDGSEASCGGVNNPTPILRALTAAFFLNAARLNRAGDGYRTLKNNITVYVHPSSVVRGMDPPPKVIIYHELVVTSKEYVRSVIPVEPRWLSEFG 6faf A 1.99 BS02 D3B A 1 F91 Q92 H94 H96 H119 L198 T199 H200 P202 F88 Q89 H91 H93 H116 L195 T196 H197 P199 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=306.1nM remove_due_to_license_issue Ki=306nM P00915 29962205 302 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6fag A 1.79 BS02 EON A 1 Q92 H94 H119 L198 T199 H200 P202 W209 Q89 H91 H116 L195 T196 H197 P199 W206 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 remove_due_to_license_issue Ki=255nM P00915 29962205 303 DWGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6fam A 1.13 BS01 MAN A 1 H63 R295 E333 H335 E336 H33 R265 E303 H305 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 29508463 502 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESKQ 6fam A 1.13 BS02 G63 A 1 Y46 W126 H154 E156 Y195 Y252 E333 E336 Y16 W96 H124 E126 Y165 Y222 E303 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 29508463 503 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESKQ 6fap B 2.7 BS03 D3H B 1 L1693 D1695 L18 D20 ? remove_due_to_license_issue Q9UIF9 29529862 1804 KVTCLVCRKGDNDEFLLLCDGCDRGCHIYCHRPKMEAVPEGDWFCTVCLAQ 6fau A 1.25 BS02 D3W B 1 N42 S45 V46 F119 N47 S50 V51 F117 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6fav A 1.4 BS02 D3Q B 1 N42 S45 F119 N47 S50 F117 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6faw A 1.4 BS02 D3K B 1 N42 S45 P167 N47 S50 P164 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6fb0 A 2.15 BS01 dna D 0 S19 D20 G21 S22 I24 Q26 K28 T46 Q47 K48 K75 R77 N136 D137 S138 T140 R141 K142 S18 D19 G20 S21 I23 Q25 K27 T45 Q46 K47 K74 R76 N135 D136 S137 T139 R140 K141 S19 D20 S18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 29980759 501 ~ 524 NTKYNKEFLLYLAGFVDSDGSIIAQIKPNQSVKFKHRLQLTFDVTQKTQRRWFLDKLVDEIGVGYVADSGSVSKYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 6fb0 A 2.15 BS02 dna F 0 S32 V33 R38 Y66 I81 K139 S31 V32 R37 Y65 I80 K138 S19 D20 S18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 29980759 601 ~ 624 NTKYNKEFLLYLAGFVDSDGSIIAQIKPNQSVKFKHRLQLTFDVTQKTQRRWFLDKLVDEIGVGYVADSGSVSKYRLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQIAALNDSKTRKTTSETVRAVLDS 6fb0 B 2.15 BS01 dna D 0 K38 Y66 Y68 I81 K116 D137 K139 K37 Y65 Y67 I80 K115 D136 K138 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 29980759 501 ~ 524 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSGKFKHKLSLTFKVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSNYYLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQVAALNDSKTRKTTSETVRAVLDSL 6fb0 B 2.15 BS02 dna F 0 D20 G21 S22 I24 Q26 K28 T46 Q47 K48 R51 V73 N136 D137 S138 T140 R141 K142 D19 G20 S21 I23 Q25 K27 T45 Q46 K47 R50 V72 N135 D136 S137 T139 R140 K141 G19 D20 G18 D19 3.1.-.- 0004519,0006314,0009507,0042802,0046872 remove_due_to_license_issue P05725 29980759 601 ~ 624 NTKYNKEFLLYLAGFVDGDGSIIAQIKPNQSGKFKHKLSLTFKVTQKTQRRWFLDKLVDEIGVGYVYDSGSVSNYYLSEIKPLHNFLTQLQPFLKLKQKQANLVLKIIEQLPSAKESPDKFLEVCTWVDQVAALNDSKTRKTTSETVRAVLDSL 6fba A 2.0 BS01 D48 A 1 E140 I148 L149 E94 I102 L103 R109 T110 K138 R159 H187 Q190 T294 P333 G359 R63 T64 K92 R113 H141 Q144 T248 P281 G307 2.1.3.2 0004070,0006207,0006221,0006520,0016020,0016597,0016740,0016743,0044205 Kd=19.9uM remove_due_to_license_issue O15804 29476738 402 DLDKIMTKMKNKSVINIDDVDDEELLAILYTSKQFEKILKNNEDSKYLENKVFCSVFLEPSTRTRCSFDAAILKLGSKVLNITDMNSTSFYKGETVEDAFKILSTYVDGIIYRDPSKKNVDIAVSSSSKPIINAGNGTGEHPTQSLLDFYTIHNYFPFILDRNINKKLNIAFVGDLKNGRTVHSLSKLLSRYNVSFNFVSCKSLNIPKDIVNTITYNLKKNNFYSDDSIKYFDNLEEGLEDVHIIYMTRIQKERYNQYKNAFILSNKTLENTRDDTKILHPLPRVNEIKVEVDSNPKSVYFTQAENGLYVRMALLYLIFSS 6fba B 2.0 BS01 D48 A 1 R109 P335 R63 P280 R109 T110 K138 R159 H187 Q190 T294 P333 G359 R63 T64 K92 R113 H141 Q144 T248 P278 G304 2.1.3.2 0004070,0006207,0006221,0006520,0016020,0016597,0016740,0016743,0044205 Kd=19.9uM remove_due_to_license_issue O15804 29476738 402 DLDKIMTKMKNKSVINIDDVDDEELLAILYTSKQFEKILKNNEDSKYLENKVFCSVFLEPSTRTRCSFDAAILKLGSKVLNITDMNSTSFYKGETVEDAFKILSTYVDGIIYRDPSKKNVDIAVSSSSKPIINAGNGTGEHPTQSLLDFYTIHNYFPFILDRNINKKLNIAFVGDLKNGRTVHSLSKLLSRYNVSFNFVSCKSLNIPKDIVNTITYNLKKNNFYSDDSIKYFDNLEEGLEDVHIIYMTRIQYNQYKNAFILSNKTLENTRDDTKILHPLPRVNEIKVEVDSNPKSVYFTQAENGLYVRMALLYLIFS 6fba B 2.0 BS02 D48 B 1 E140 I148 L149 Y152 E94 I102 L103 Y106 R109 T110 K138 R159 H187 Q190 T294 P333 G359 R63 T64 K92 R113 H141 Q144 T248 P278 G304 2.1.3.2 0004070,0006207,0006221,0006520,0016020,0016597,0016740,0016743,0044205 Kd=19.9uM remove_due_to_license_issue O15804 29476738 402 DLDKIMTKMKNKSVINIDDVDDEELLAILYTSKQFEKILKNNEDSKYLENKVFCSVFLEPSTRTRCSFDAAILKLGSKVLNITDMNSTSFYKGETVEDAFKILSTYVDGIIYRDPSKKNVDIAVSSSSKPIINAGNGTGEHPTQSLLDFYTIHNYFPFILDRNINKKLNIAFVGDLKNGRTVHSLSKLLSRYNVSFNFVSCKSLNIPKDIVNTITYNLKKNNFYSDDSIKYFDNLEEGLEDVHIIYMTRIQYNQYKNAFILSNKTLENTRDDTKILHPLPRVNEIKVEVDSNPKSVYFTQAENGLYVRMALLYLIFS 6fbv C 3.52 BS01 FI8 D 1 M1051 I1052 T1096 K1101 E1119 S1120 M1024 I1025 T1069 K1074 E1092 S1093 2.7.7.6 0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005515,0005829,0005886,0006351,0006360,0006366,0006383,0009274,0016779,0032549,0034062,0042793,0046677 remove_due_to_license_issue P9WGY9 29606590 1904 SNNSVPGAPNRVSFAKLREPLEVPGLLDVQTDSFEWLIGSPRWRESAAERGDVNPVGGLEEVLYELSPIEDFSGSMSLSFSDPRFDDVKAPVDECKDKDMTYAAPLFVTAEFINNNTGEIKSQTVFMGDFPMMTEKGTFIINGTERVVVSQLVRSPGVYFDETIDKSTDKTLHSVKVIPSRGAWLEFDVDKRDTVGVRIDRKRRQPVTVLLKALGWTSEQIVERFGFSEIMRSTLEKDNTVGTDEALLDIYRKLRPGEPPTKESAQTLLENLFFKEKRYDLARVGRYKVNKKLGLHVGEPITSSTLTEEDVVATIEYLVRLHEGQTTMTVPGGVEVPVETDDIDHFGNRRLRTVGELIQNQIRVGMSRMERVVRERMTTQDVEAITPQTLINIRPVVAAIKEFFGTSQLSQFMDQNNPLSGLTHKRRLSALGPGGLSRERAGLEVRDVHPSHYGRMCPIETPEGPNIGLIGSLSVYARVNPFGFIETPYRKVVDGVVSDEIVYLTADEEDRHVVAQANSPIDADGRFVEPRVLVRRKAGEVEYVPSSEVDYMDVSPRQMVSVATAMIPFLEHDDANRALMGANMQRQAVPLVRSEAPLVGTGMELRAAIDAGDVVVAEESGVIEEVSADYITVMHDNGTRRTYRMRKFARSNHGTCANQCPIVDAGDRVEAGQVIADGPCTDDGEMALGKNLLVAIMPWEGHNYEDAIILSNRLVEEDVLTSIHIEEHEIDARDTKLGAEEITRDIPNISDEVLADLDERGIVRIGAEVRDGDILVGKVTPKGETELTPEERLLRAIFGEKAREVRDTSLKVPHGESGKVIGIRVFSREDEDELPAGVNELVRVYVAQKRKISDGDKLAGRHGNKGVIGKILPVEDMPFLADGTPVDIILNTHGVPRRMNIGQILETHLGWCAHSGWKVDAAKGVPDWAARLPDELLEAQPNAIVSTPVFDGAQEAELQGLLSCTLPNRDGDVLVDADGKAMLFDGRSGEPFPYPVTVGYMYIMKLHHLVDDKIHARSTGPYSMITQQPLGGKAQFGGQRFGEMECWAMQAYGAAYTLQELLTIKSDDTVGRVKVYEAIVKGENIPEPGIPESFKVLLKELQSLCLNVEVLSSDGAAI 6fbv D 3.52 BS03 FI8 D 1 R84 R89 R412 R82 R87 R410 2.7.7.6 0000287,0000428,0001054,0001055,0001056,0001057,0001058,0001059,0001060,0001066,0003677,0003899,0005829,0005886,0006351,0006360,0006366,0006383,0008270,0009274,0016779,0034062,0042793,0046872 remove_due_to_license_issue P9WGY7 29606590 1904 DVNFFDELRIGLATAEDIRQWSYGEVKKPETINYRTLKPEKDGLFCEKIFGPTRDWECYCGKYKRVRFKGIICERCGVEVTRAKVRRERMGHIELAAPVTHIWYFKGVPSRLGYLLDLAPKDLEKIIYFAAYVITSVDEEMRHNELSTLEAEMAVERKAVEDQRDGELEARAQKLEADLAELEAEGAKADARRKVRDGGEREMRQIRDRAQRELDRLEDIWSTFTKLAPKQLIVDENLYRELVDRYGEYFTGAMGAESIQKLIENFDIDAEAESLRDVIRNGKGQKKLRALKRLKVVAAFQQSGNSPMGMVLDAVPVIPPELRPMVQLDGGRFATSDLNDLYRRVINRNNRLKRLIDLGAPEIIVNNEKRMLQESVDALFDNGRRGRPVTGPGNRPLKSLSDLLKGKQGRFRQNLLGKRVDYSGRSVIVVGPQLKLHQCGLPKLMALELFKPFVMKRLVDLNHAQNIKSAKRMVERQRPQVWDVLEEVIAEHPVLLNRAPTLHRLGIQAFEPMLVEGKAIQLHPLVCEAFNADFDGDQMAVHLPLSAEAQAEARILMLSSNNILSPASGRPLAMPRLDMVTGLYYLTTEVPGDTGEYQPASGDHPETGVYSSPAEAIMAADRGVLSVRAKIKVRLTQLRPPVEIEAELFGHSGWQPGDAWMAETTLGRVMFNELLPLGYPFVNKQMHKKVQAAIINDLAERYPMIVVAQTVDKLKDAGFYWATRSGVTVSMADVLVPPRKKEILDHYEERADKVEKQFQRGALNHDERNEALVEIWKEATDEVGQALREHYPDDNPIITIVDSGATGNFTQTRTLAGMKGLVTNPKGEFIPRPVKSSFREGLTVLEYFINTHGARKGLADTALRTADSGYLTRRLVDVSQDVIVREHDCQTERGIVVELAERAPDGTLIRDPYIETSAYARTLGTDAVDEAGNVIVERGQDLGDPEIDALLAAGITQVKVRSVLTCATSTGVCATCYGRSMATGKLVDIGEAVGIVAAQSIGEPGTQLTMRDITGGLPRVQELFEARVPRGKAPIADVTGRVRLEDGERFYKITIVPDDGGEEVVYDKISKRQRLRVFKHEDGSERVLSDGDHVEVGQQLMEGSADPHEVLRVQGPREVQIHLVREVQEVYRAQGVSIHDKHIEVIVRQMLRRVTIIDSGSTEFLPGSLIDRAEFEAENRRVVAEGGEPAAGRPVLMGITKASLATDSWLSAASFQETTRVLTDAAINCRSDKLNGLKENVIIGKLIPAGTGINRYRNIAVQPTEEARAA 6fbv F 3.52 BS01 FI8 D 1 L423 D424 L199 D200 ? 0003677,0003700,0005515,0005737,0005886,0006352,0006355,0009274,0009415,0010468,0016987,2000142 remove_due_to_license_issue P9WGI1 29606590 1904 ADSVRAYLKQIGKVALLNAEEEVELAKRIEAGLYATQLMTELSERGEKLPAAQRRDMMWICRDGDRAKNHLLEANLRLVVSLAKRYTGRGMAFLDLIQEGNLGLIRAVEKFDYTKGYKFSTYATWWIRQAITRAMADQARTIRIPVHMVEVINKLGRIQRELLQDLGREPTPEELAKEMDITPEKVLEIQQYAREPISLDQQLGDFIEDSVAVDAVSFTLLQDQLQSVLDTLSEREAGVVRLRFGLTDGQPRTLDEIGQVYGVTRERIRQIESKTMSKLRHPSRSQVLRDYLD 6fbw A 1.45 BS02 D4K B 1 N42 S45 V46 F119 N47 S50 V51 F118 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNEGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6fby A 1.5 BS02 D4H B 1 N42 S45 F119 I219 N47 S50 F116 I216 ? remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATGDDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6fcj A 2.49 BS01 D4W A 1 N51 A55 D93 M98 L107 T109 V186 N36 A40 D78 M83 L92 T94 V171 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 6fcl A 1.5 BS01 AMP A 1 F26 R27 R67 D128 L129 A131 T132 G133 T135 F24 R25 R65 D126 L127 A129 T130 G131 T133 2.4.2.7 0002055,0003999,0005515,0005576,0005654,0005737,0005829,0006166,0006168,0007625,0016208,0016757,0032263,0032264,0034774,0044209,0046083,0070062 remove_due_to_license_issue P07741 29576532 200 DSELQLVEQRIRSFPDFPTPGVVFRDISPVLKDPASFRAAIGLLARHLKATHGGRIDYIAGLDSRGFLFGPSLAQELGLGCVLIRKRGKLPGPTLWASYSLEYGKAELEIQKDALEPGQRVVVVDDLLATGGTMNAACELLGRLQAEVLECVSLVELTSLKGREKLAPVPFFSLLQYE 6fcl B 1.5 BS01 AMP B 1 F26 R27 R67 D127 D128 L129 A131 T132 G133 T135 F24 R25 R65 D120 D121 L122 A124 T125 G126 T128 2.4.2.7 0002055,0003999,0005515,0005576,0005654,0005737,0005829,0006166,0006168,0007625,0016208,0016757,0032263,0032264,0034774,0044209,0046083,0070062 remove_due_to_license_issue P07741 29576532 200 DSELQLVEQRIRSFPDFPTPGVVFRDISPVLKDPASFRAAIGLLARHLKATHGGRIDYIAGLDSRGFLFGPSLAQELGLGCVLIRKRGKLPGPTLWASYSAELEIQKDALEPGQRVVVVDDLLATGGTMNAACELLGRLQAEVLECVSLVELTSLKGREKLAPVPFFSLLQYE 6fdc A 1.45 BS03 DD5 A 1 Y325 H326 N487 P488 Y495 W498 T499 I502 F506 P522 M523 Q535 F538 Y77 H78 N239 P240 Y247 W250 T251 I254 F258 P274 M275 Q287 F290 3.1.4.53 0004114,0007165,0008081 ic50=2.3uM remove_due_to_license_issue Q08499 29652483 606 GVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6fdq A 2.3 BS01 2UQ A 1 W247 M262 L265 A266 S270 V271 S274 W276 C345 W85 M100 L103 A104 S108 V109 S112 W114 C183 3.4.22.- 0006508,0008234 remove_due_to_license_issue B0B9A0 30028574 501 VPAWDSDIIFKCLCYFHTLYPGLIPLETFPPATIFNFKQKIISILEDKKAVLRGEPIKGPLPICCSKENYRRHLQRTTLLPVFMWYHPTPKTLSDTMQTMKQLAIKGSVGASHWLLVIVDIQARRLVYFDSLYNYVMPPENMKKELQSFAQQLDQVYPAYDSKKFSVKIAAKEVIQRGSGSSCGAWCCQFLHWYLKDPLTDALNDLPVDSVERHENLASFVQACEAAVQDLPELSWPEA 6fdu B 2.3 BS01 D5W B 1 D167 S168 W247 M262 A266 S274 W276 G342 C345 D5 S6 W85 M100 A104 S112 W114 G180 C183 3.4.22.- 0006508,0008234 remove_due_to_license_issue B0B9A0 30028574 501 VPAWDSDIIFKCLCYFHTLYPGLIPLETFPPATIFNFKQKIISILEDKKAVLRGEPIKGPLPICCSKENYRRHLQRTTLLPVFMWYHPTPKTLSDTMQTMKQLAIKGSVGASHWLLVIVDIQARRLVYFDSLYNYVMPPENMKKELQSFAQQLDQVYPAYDSKKFSVKIAAKEVIQRGSGSSCGAWCCQFLHWYLKDPLTDALNDLPVDSVERHENLASFVQACEAAVQDLPELSWPEA 6fe0 A 1.91 BS02 V90 A 1 N62 H64 Q92 H94 H96 L198 T199 T200 N46 H48 Q72 H74 H76 L179 T180 T181 H64 H94 H96 E106 H119 T199 H48 H74 H76 E86 H99 T180 4.2.1.1 0004089,0008270 Kd=1.1nM remove_due_to_license_issue Kd=15nM Q16790 29928486 302 SPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 6fe1 A 1.95 BS02 V14 A 1 N62 H94 H96 V121 V131 L198 T199 T200 N58 H86 H88 V113 V122 L191 T192 T193 H64 H94 H96 E106 H119 T199 H60 H86 H88 E98 H111 T192 4.2.1.1 0004089,0008270 Kd=0.05nM remove_due_to_license_issue Kd=<10.0nM Q16790 29928486 302 WRYGGDPPWPRVSPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 6fe5 A 1.52 BS04 D6E A 1 R210 M424 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 R156 M370 L374 G464 N465 R480 R482 Y495 H496 K642 Y643 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 remove_due_to_license_issue Ki=0.580000nM, IC50=0.500000nM Q04609 30552009 821 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAMEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6fer A 2.87 BS01 D6Q A 1 L616 V624 M676 I685 M699 T701 Y703 M704 F753 L764 A774 D775 F776 L17 V25 M60 I69 M83 T85 Y87 M88 F126 L137 A147 D148 F149 D757 R761 N762 D775 D130 R134 N135 D148 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue Q16832 30452219 1001 VAVEEFPRKLLTFKEKLGEGQFGEVHLCEVEGPVLVAVKMLRADANKNARNDFLKEIKIMSRLKDPNIIHLLAVCITDDPLCMITEYMENGDLNQFLSRHTVSYTNLKFMATQIASGMKYLSSLNFVHRDLATRNCLVGKNYTIKIADFGMSRNLYSGDYYRIQGRAVLPIRWMSWESILLGKFTTASDVWAFGVTLWETFTFCQEQPYSQLSDEQVIENTGEFFRDQGRQTYLPQPAICPDSVYKLMLSCWRRDTKNRPSFQEIHLLLLQ 6few A 1.44 BS01 D6W A 1 V624 A653 K655 E672 M676 I685 M699 T701 M704 L773 A783 D784 F785 V22 A45 K47 E64 M68 I77 M91 T93 M96 L153 A163 D164 F165 D766 R770 N771 D784 D146 R150 N151 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=1.41uM remove_due_to_license_issue Q08345 30452219 1001 VDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKAAPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALN 6fex A 1.291 BS01 D6Z A 1 V624 A653 K655 M676 I685 M699 Y703 M704 H764 L773 A783 D784 F785 V23 A49 K51 M72 I81 M95 Y99 M100 H145 L154 A164 D165 F166 D766 R770 N771 D784 D147 R151 N152 D165 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.029uM remove_due_to_license_issue IC50=25.6nM Q08345 30452219 1001 RVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVFPLNVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAED 6ffe A 1.76 BS01 D7Q A 1 W370 P371 L383 Y428 N429 V435 M438 W28 P29 L41 Y86 N87 V93 M96 ? remove_due_to_license_issue P25440 29656650 505 MGKLSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 6fff A 1.67 BS01 D7H A 1 W370 P371 L383 Y386 Y428 N429 V435 M438 W28 P29 L41 Y44 Y86 N87 V93 M96 ? remove_due_to_license_issue IC50=100nM P25440 29656650 503 MGKLSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 6ffg A 1.59 BS01 D7B A 1 W370 P371 L383 Y428 N429 H433 V435 W28 P29 L41 Y86 N87 H91 V93 ? remove_due_to_license_issue IC50=2512nM, Kd=32nM P25440 29656650 503 MGKLSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMPD 6ffh A 2.65 BS01 D7W A 1 G624 I625 G628 S654 P655 Y659 W1785 F1788 S1809 A1810 G57 I58 G61 S87 P88 Y92 W367 F370 S391 A392 E1011 D1020 E121 D130 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P41594 29455526 4006 SPVQYLRWGDPAPIAAVVFACLGLLATLFVTVVFIIYRDTPVVKSSSRELCYIILAGICLGYLCTFCLIAKPKQIYCYLQRIGIGLSPAMSYSALVTKTYRAARILAMSKKNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKISACAQLVIAFILICIQLGIIVALFIMEPPDIMHDYPEVYLICNTTNLGVVAPLGYNGLLILACTFYAFKTRNVPANFNEAKYIAFTMYTTCIIWLAFVPIYFGSNYKIITMCFSVSLSATVALGCMFVPKVYIILAKPERN 6ffi A 2.2 BS01 D8B A 1 G624 S654 P655 Y659 W945 F948 S965 S969 G57 S87 P88 Y92 W363 F366 S383 S387 E688 D697 E121 D130 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 ic50=8nM remove_due_to_license_issue P00720,P41594 29455526 4009 SPVQYLRWGDPAPIAAVVFACLGLLATLFVTVVFIIYRDTPVVKSSSRELCYIILAGICLGYLCTFCLIAKPKQIYCYLQRIGIGLSPAMSYSALVTKTYRAARILAMSKKNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKISACAQLVIAFILICIQLGIIVALFIMEPPDIMEVYLICNTTNLGVVAPLGYNGLLILACTFYAFKTRNVPANFNEAKYIAFTMYTTCIIWLAFVPIYFGSNYKIITMCFSVSLSATVALGCMFVPKVYIILAKPERN 6ffn A 1.75 BS01 D8K A 1 H40 E71 L127 S128 N130 T142 C147 V162 G163 G164 N165 G166 F170 H42 E73 L129 S130 N132 T144 C149 V164 G165 G166 N167 G168 F172 H40 E71 G145 C147 H42 E73 G147 C149 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue P04936 29433930 201 GSGPEEEFGMSLIKHNSCVITTENGKFTGLGVYDRFVVVPTHADPGKEIQVDGITTKVIDSYDLYNKNGIKLEITVLKLDRNEKFRDIRRYIPNNEDDYPNCNLALLANQPEPTIINVGDVVSYGNILLSGNQTARMLKYSYPTKSGYCGGVLYKIGQVLGIHVGGNGRDGFSAMLLRSYFT 6ffs A 1.86 BS01 D8E A 1 H40 L127 S128 N130 T142 K143 C147 V162 G163 G164 N165 F170 H42 L129 S130 N132 T144 K145 C149 V164 G165 G166 N167 F172 H40 E71 G145 C147 H42 E73 G147 C149 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0004197,0006508 remove_due_to_license_issue P04936 29433930 201 GSGPEEEFGMSLIKHNSCVITTENGKFTGLGVYDRFVVVPTHADPGKEIQVDGITTKVIDSYDLYNKNGIKLEITVLKLDRNEKFRDIRRYIPNNEDDYPNCNLALLANQPEPTIINVGDVVSYGNILLSGNQTARMLKYSYPTKSGYCGGVLYKIGQVLGIHVGGNGRDGFSAMLLRSYFT 6fg6 A 2.401 BS01 D8Q A 1 P1817 F1818 V1822 N1873 V1879 P22 F23 V27 N78 V84 ? remove_due_to_license_issue Q9UIF9 29770599 1901 HSDLTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 6fgc A 1.5 BS02 D95 A 1 D327 F330 I331 R653 I656 D9 F12 I13 R335 I338 2.10.1.1,2.7.7.75 0006777,0032324 remove_due_to_license_issue Q03555 30704910 816 SPFPLTSMDKAFITVLEMTPVLGTEIINYRDGMGRVLAQDVYAKDNLPPFPASVKDGYAVRAADGPGDRFIIGESQAGEQPTQTVMPGQVMRVTTGAPIPCGADAVVQVEDTELIRESDDGTEELEVRILVQARPGQDIRPIGHDIKRGECVLAKGTHMGPSEIGLLATVGVTEVEVNKFPVVAVMSTGNELLNPEDDLLPGKIRDSNRSTLLATIQEHGYPTINLGIVGDNPDDLLNALNEGISRADVIITSGGVSMGEKDYLKQVLDIDLHAQIHFGRVFMKPGLPTTFATLDIDGVRKIIFALPGNPVSAVVTCNLFVVPALRKMQGILDPRPTIIKARLSCDVKLDPRPEYHRCILTWHHQEPLPWAQSTGLMSMRSANGLLMLPPKTEQYVELHKGEVVDVMVIGRL 6fgf A 2.801 BS01 EN2 A 1 P1817 F1818 V1822 L1826 Y1830 N1873 V1879 P22 F23 V27 L31 Y35 N78 V84 ? remove_due_to_license_issue Q9UIF9 29770599 1901 HSDLTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 6fgg A 1.1 BS01 D9B A 1 W1816 P1817 V1822 N1873 V1879 W18 P19 V24 N75 V81 ? Kd=17uM remove_due_to_license_issue Q9UIF9 29770599 1901 LTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFYQ 6fgl A 2.1 BS01 UO1 A 1 W1816 P1817 P1821 V1822 N1823 L1826 N1873 V1879 W21 P22 P26 V27 N28 L31 N78 V84 ? ic50=24uM remove_due_to_license_issue Q9UIF9 29770599 1901 HSDLTFCEIILMEMESHDAAWPFLEPVNPRLVSGYRRIIKNPMDFSTMRERLLRGGYTSSEEFAADALLVFDNCQTFNEDDSEVGKAGHIMRRFFESRWEEFY 6fgq A 2.37 BS01 D9N A 1 Q286 L287 H323 R364 M365 R367 A368 F377 F378 F388 L396 I397 I400 F401 Q24 L25 H61 R102 M103 R105 A106 F115 F116 F126 L134 I135 I138 F139 ? 0003677,0004879,0005634,0006355 ic50=0.014uM remove_due_to_license_issue IC50=21nM P51449 30095900 601 QGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCHVERLQIFQHLHPIV 6fgy A 1.54 BS01 D9W A 1 G59 Q60 G61 L78 D80 Y119 F156 I166 D276 G278 T280 G13 Q14 G15 L32 D34 Y73 F110 I120 D219 G221 T223 3.4.23.46 0004190,0006508,0016020 ic50=70nM remove_due_to_license_issue IC50=70nM P56817 29764741 501 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIPQ 6fh3 A 1.85 BS01 RPI A 1 V283 D285 S286 R338 D339 R342 V280 D282 S283 R335 D336 R339 R31 E122 R126 C168 T170 R177 R208 E213 R28 E119 R123 C165 T167 R174 R205 E210 2.7.14.1 0003824,0004111,0004672,0005524,0005615,0016301,0016772,0016775,0046314 remove_due_to_license_issue P0DMM5 30962626 401 GKFFNTAVSAWMSQEGPNSDIVLSSRIRLARNIVDFRFPTLFSSEEAKQIVALFERAFVHRPYGEAGRFELLKMSELQPIEKRVLVEKHLISPHLAEDSPFGACLLSENEEISIMINEEDHIRIQCLFPGLQLAEALEAASELDDWIEGHVNYAFDERLGYLTSCPTNVGTGLRASVMMHLPALVLTQQINRIIPAINQLGLVVRGTYGEGSEALGNIFQISNQITLGKSEEDIVADLHTIVEQLIAQERAARQALVKTLGIQLEDKVFRSYGILANCRVIDSKEAAQCLSDVRLGIDLGYIKNVSRNILNELMILTQPGFLQQYAGGVLRPEERDVRRAALIRERLRMETR 6fh3 B 1.85 BS01 RPI B 1 D285 S286 P322 P335 R338 D339 R342 D274 S275 P311 P324 R327 D328 R331 R31 E122 R126 C168 T170 R177 R208 E213 R27 E111 R115 C157 T159 R166 R197 E202 2.7.14.1 0003824,0004111,0004672,0005524,0005615,0016301,0016772,0016775,0046314 remove_due_to_license_issue P0DMM5 30962626 401 KFFNTAVSAWMSQEGPNSDIVLSSRIRLARNIVDFRFPTLFSSEEAKQIVALFERAFVGRFELLKMSELQPIEKRVLVEKHLISPHLAEDSPFGACLLSENEEISIMINEEDHIRIQCLFPGLQLAEALEAASELDDWIEGHVNYAFDERLGYLTSCPTNVGTGLRASVMMHLPALVLTQQINRIIPAINQLGLVVRGTYGEGSEALGNIFQISNQITLGKSEEDIVADLHTIVEQLIAQERAARQALVKTLGIQLEDKVFRSYGILANCRVIDSKEAAQCLSDVRLGIDLGYIKNVSRNILNELMILTQPGFLQQYAGGVLRPEERDVRRAALIRERLRMETR 6fh6 A 2.082 BS01 D8Q A 1 P1888 F1889 Y1901 F1943 N1944 I1950 P33 F34 Y46 F88 N89 I95 ? remove_due_to_license_issue Q9UIF8 29770599 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFK 6fh7 A 2.1 BS01 EN2 A 1 P1888 L1891 V1893 N1944 I1950 P33 L36 V38 N89 I95 ? remove_due_to_license_issue Q9UIF8 29770599 2001 SMSVKKPKRDDSKDLALCSMILTEMETHEDAWPFLLPVNLKLVPGYKKVIKKPMDFSTIREKLSSGQYPNLETFALDVRLVFDNCETFNEDDSDIGRAGHNMRKYFEKKWTDTFKV 6fhk A 1.657 BS01 ADP A 1 T14 Y15 G201 G202 G230 E268 K271 R272 S275 G338 G339 R342 T11 Y12 G198 G199 G227 E265 K268 R269 S272 G335 G336 R339 ? 0005524,0140662 remove_due_to_license_issue P0DMV8 30108182 401 AAAIGIDLGTTYSCVGVFQHGKVEIIANDQGNRTTPSYVAFTDTERLIGDAAKNQVALNPQNTVFDAKRLIGRKFGDPVVQSDMKHWPFQVINDGDKPKVQVSYKGETKAFYPEEISSMVLTKMKEIAEAYLGYPVTNAVITVPAYFNDSQRQATKDAGVIAGLNVLRIINEPTAAAIAYGLDRTGKGERNVLIFDLGGGTFDVSILTIDDGIFEVKATAGDTHLGGEDFDNRLVNHFVEEFKRKHKKDISQNKRAVRRLRTACERAKRTLSSSTQASLEIDSLFEGIDFYTSITRARFEELCSDLFRSTLEPVEKALRDAKLDKAQIHDLVLVGGSTRIPKVQKLLQDFFNGRDLNKSINPDEAVAYGAAVQAAILM 6fhq A 1.95 BS03 DE5 A 1 E1944 L1948 D1950 W1973 E19 L23 D25 W48 ? Kd=3.4mM remove_due_to_license_issue Q9UIF8 29529862 2003 HMSIMKVYCQICRKGDNEELLLLCDGCDKGCHTYCHRPKITTIPDGDWFCPACIAKAS 6fi1 A 2.7 BS03 D3H A 1 E1944 L1948 D1950 I1968 E18 L22 D24 I42 ? remove_due_to_license_issue Q9UIF8 29529862 2003 MSIMKVYCQICRKGDNEELLLLCDGCDKGCHTYCHRPKITTIPDGDWFCPACIAKAS 6fi4 A 2.0 BS02 60H B 1 F119 K122 D215 F113 K116 D205 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSGPEVREYREKVETELQGVCDTVLGLLDSHLIKDAESRVFYLKMKGDYYRYLAEVAKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6fi5 A 1.7 BS02 60H B 1 N42 S45 F119 K122 I168 N47 S50 F118 K121 I165 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 29722962 101 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNEGPEVREYREKVETELQGVCDTVLGLLDSHLIKEAGDAESRVFYLKMKGDYYRYLAEVATDKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6fii D 2.405 BS02 SG9 D 1 P175 D179 T180 V181 E183 P184 M398 P173 D177 T178 V179 E181 P182 M380 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 Kd=9.5nM remove_due_to_license_issue Q6B856 29844393 502 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDATAD 6fil A 1.73 BS01 D6W A 1 V624 A653 K655 E672 M676 I685 M699 T701 M704 L767 A777 D778 F779 V21 A34 K36 E53 M57 I66 M80 T82 M85 L148 A158 D159 F160 D760 R764 N765 D778 D141 R145 N146 D159 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=1.41uM remove_due_to_license_issue Q08345 30452219 1001 DFPRSRLRFKEKLGEGQFGEVHLCEVDSPPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKAAEGAPGDPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNT 6fiv A 1.9 BS01 3TL A 1 G32 A33 D34 M56 I57 G58 V59 G28 A29 D30 M52 I53 G54 V55 2.7.7.-,2.7.7.49,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.-,3.6.1.23 0004190,0006508 Ki=8.3nM remove_due_to_license_issue P16088 10651036 201 GTTTTLEKRPEILIFVNGYPIKFLLDTGADITILNRRDFQVKNSIENGRQNMIGVGGGKRGTNYINVHLEIRDENYKTQCIFGNVCVLEDNSLIVPLLGRDNMIKFNIRLVM 6fjf D 2.402 BS02 DKE D 1 G100 N102 K105 T180 V181 V182 R401 F404 W407 G98 N100 K103 T178 V179 V180 R382 F385 W388 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 Kd=6.8nM remove_due_to_license_issue Q6B856 29844393 503 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDATAD 6fjm D 2.1 BS02 DKN D 1 G100 N102 T180 V181 V182 F404 W407 Y408 G97 N99 T177 V178 V179 F388 W391 Y392 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 Kd=576nM remove_due_to_license_issue Q6B856 29844393 503 REIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSLTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDATAD 6fky A 2.98 BS04 E9N C 1 T65 Y98 R101 Q136 N137 I138 H154 V216 T31 Y64 R67 Q102 N103 I104 H120 V182 P64 T65 F66 R67 N137 D139 H154 P30 T31 F32 R33 N103 D105 H120 2.3.1.- 0000035,0005634,0005737,0005739,0005829,0006476,0008270,0010566,0016740,0017136,0034979,0036047,0036048,0036049,0036054,0036055,0046872,0061697,0070403,1901363 remove_due_to_license_issue Q6DHI5 29494161 101 DLTAFREHFAKAKHIAIITGAGVSAESGVPTFRGPGGFWRKWQAQDLATPEAFSRDPSLVWEFYHYRREVMRSKMPNPAHLAIAECEARLGQQGRSVVIITQNIDELHHRAGSKHVYEIHGSLFKTRCMSCGEVKANHKSPICPALDGKGAPDPNTKEARIPVELLPRCERKSCNGLLRPHVVWFGETLDSDILTAVERELEKCDLCLVVGTSSIVYPAAMFAPQVASRGVPVAEFNMECTPATQKYHFEGPCGSTLPPALE 6fmc A 0.9 BS01 DUE A 1 Y297 T316 D320 S346 E348 T349 K351 Y353 G414 I415 Y28 T47 D51 S77 E79 T80 K82 Y84 G145 I146 ? Kd=1.32uM remove_due_to_license_issue O14786 29648813 501 GHMFKCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 6fmf A 2.811 BS01 DUE A 1 Y297 S298 N300 W301 D320 S346 E348 T349 K351 Y353 G414 Y25 S26 N28 W29 D48 S74 E76 T77 K79 Y81 G142 ? remove_due_to_license_issue O14786 29648813 501 FKCMEALGMESGEIHSDQITASSQYSTNWSAERSRLNYPENGWTPGEDSYREWIQVDLGLLRFVTAVGTQGAISKETKKKYYVKTYKIDVSSNGEDWITIKEGNKPVLFQGNTNPTDVVVAVFPKPLITRFVRIKPATWETGISMRFEVYGCKIT 6fmi C 2.8 BS01 DV2 C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue P40337 29650462 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 6fmj C 2.45 BS01 DV5 C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=0.76uM remove_due_to_license_issue P40337 29650462 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 6fmk C 2.75 BS01 DV8 C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue P40337 29650462 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 6fmn A 1.36 BS02 E4E A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 D92 Y96 D146 C148 G219 L221 A222 M250 G251 D102 D280 C318 C320 C323 H349 D92 D270 C308 C310 C313 H339 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=1120nM remove_due_to_license_issue P28720 29939431 406 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHLDGSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 6fn9 A 2.27 BS01 DW8 A 1 K49 G53 R56 R127 Y128 N173 K48 G52 R55 R126 Y127 N172 ? 0000122,0001525,0003016,0003723,0005515,0005615,0005634,0005654,0005737,0005829,0005925,0006468,0006605,0007165,0008039,0008104,0019901,0019904,0030324,0031625,0031647,0031982,0035148,0042149,0042470,0042802,0043066,0043067,0044325,0045296,0045824,0050815,0051683,0070062,0070371,0070372,0072562,0090128,0090168,0098686,0098978,0140297,0140311,1900181,1904262 ic50=284uM remove_due_to_license_issue P63104 29924885 301 DKNELVQKAKLAEQAERYDDMAACMKSVTEQGAELSNEERNLLSVAYKNVVGARRSSWRVVSSIEQKTEGAEKKQQMAREYREKIETELRDICNDVLSLLEKFLIPNASQAESKVFYLKMKGDYYRYLAEVAAGDDKKGIVDQSQQAYQEAFEISKKEMQPTHPIRLGLALNFSVFYYEILNSPEKACSLAKTAFDEAIAELDTLSEESKDSTLIMQLLRDNLTLWTS 6fne A 2.501 BS01 DY5 A 1 H652 R654 K667 H247 R249 K262 ? 0005085,0032012 ic50=3uM remove_due_to_license_issue Q6DN90 30742123 801 SNDVIRKRHYRIGLNLFNKKPEKGVQYLIERGFVPDTPVGVAHFLLQRKGLSRQMIGEFLGNRQKQFNRDVLDCVVDEMDFSTMELDEALRKFQAHIRVQGEAQKVERLIEAFSQRYCICNPGVVRQFRNPDTIFILAFAIILLNTDMYSPNVKPERKMKLEDFIKNLRGVDDGEDIPREMLMGIYERIRKRELKTNEDHVSQVQKVEKLIVGKKGCVLSLPHRRLVCYCRLFEVPDPNKPQKLGLHQREIFLFNDLLVVTKIFQKKKNSVTYSFRQSFSLYGMQVLLFENQYYPNGIRLTSSVADIKVLINFNAPNPQDRKKFTDDLRESIAEVQEMEKHRIESELEKQ 6fnf A 1.556 BS01 DXH A 1 V627 A644 K646 E663 M667 T692 Y694 M695 Y735 H737 L746 S756 D757 F758 V22 A35 K37 E54 M58 T83 Y85 M86 Y126 H128 L137 S147 D148 F149 D739 A741 R743 N744 D757 P780 D130 A132 R134 N135 D148 P153 2.7.10.1 0004672,0004713,0005524,0006468 Kd=13nM remove_due_to_license_issue P29317 29928781 1001 TEIHPSCVTRQKVIGAGEFGEVYKGMLKTKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLSPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIR 6fng A 1.038 BS01 DWT A 1 V627 A644 K646 E663 M667 T692 Y694 M695 L730 Y735 S756 D757 F758 V29 A41 K43 E60 M64 T89 Y91 M92 L127 Y132 S153 D154 F155 D739 A741 R743 N744 D757 P780 D136 A138 R140 N141 D154 P160 2.7.10.1 0004672,0004713,0005524,0006468 Kd=73nM remove_due_to_license_issue P29317 29928781 1001 QAVLKFTTEIHPSCVTRQKVIGAGEFGEVYKGMLKKEVPVAIKTLKAGYTEKQRVDFLGEAGIMGQFSHHNIIRLEGVISKYKPMMIITEYMENGALDKFLREKDGEFSVLQLVGMLRGIAAGMKYLANMNYVHRDLAARNILVNSNLVCKVSDFGLKIPIRWTAPEAISYRKFTSASDVWSFGIVMWEVMTYGERPYWELSNHEVMKAINDGFRLPTPMDCPSAIYQLMMQCWQQERARRPKFADIVSILDKLIRAPDSLKTLADFDPRVSIRLPS 6fni A 1.468 BS01 DXH A 1 A645 E664 M668 T693 M696 Y736 L747 S757 D758 F759 F764 A39 E53 M57 T82 M85 Y125 L136 S146 D147 F148 F153 D740 A742 R744 N745 D758 P783 D129 A131 R133 N134 D147 P155 2.7.10.1 0004672,0004713,0005524,0006468 Kd=6nM remove_due_to_license_issue P54760 29928781 1001 AKEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLSRFIPIRWTAPEAIAFRKFTSASDVWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQIVSALDKMIRNPASLKIVAR 6fnj A 1.239 BS01 DWT A 1 V629 A645 K647 E664 M668 I677 T693 F695 M696 Y736 S757 D758 F759 V23 A39 K41 E58 M62 I71 T87 F89 M90 Y130 S151 D152 F153 D740 A742 R744 N745 D758 P783 D134 A136 R138 N139 D152 P157 2.7.10.1 0004672,0004713,0005524,0006468 Kd=142nM remove_due_to_license_issue P54760 29928781 1001 AKEIDVSYVKIEEVIGAGEFGEVCRGRLKAPGKKESCVAIKTLKGGYTERQRREFLSEASIMGQFEHPNIIRLEGVVTNSMPVMILTEFMENGALDSFLRLNDGQFTVIQLVGMLRGIASGMRYLAEMSYVHRDLAARNILVNSNLVCKVSDFGLIPIRWTAPEAIAFRKFTSASDVWSYGIVMWEVMSFGERPYWDMSNQDVINAIEQDYRLPPPPDCPTSLHQLMLDCWQKDRNARPRFPQIVSALDKMIRNPASLKIVA 6fnq A 1.75 BS01 AVJ A 1 F47 Y56 T163 N166 Y206 E282 S284 F48 Y57 T164 N167 Y207 E283 S285 2.1.1.44 0008168,0008276,0032259,0052699,0052704,0052706 Kd=26uM remove_due_to_license_issue A0R5M8 29658702 401 HMALSLANYLAADSAAEALRRDVRAGLTATQKSLPPKWFYDAVGSDLFDQITRLPEYYPTRTEAQILRTRSAEIISAAGADTLVELGSGTSEKTRMLLDAMRDAELLRRFIPFDVDAGVLRSAGAAIGAEYPGIEIDAVCGDFEEHLGKIPHVGRRLVVFLGSTIGNLTPAPRAEFLSTLADTLQPGDSLLLGTDLVKDTGRLVRAYDDAAGVTAAFNRNVLAVVNRELSADFDLDAFEHVAKWNSDEERIEMWLRARTAQHVRVAALDLEVDFAAGEEMLTEVSCKFRPENVVAELAEAGLRQTHWWTDPAGDFGLSLAVR 6fnr A 1.83 BS01 DYT A 1 F47 Y56 Y206 E282 S284 F47 Y56 Y206 E282 S284 2.1.1.44 0008168,0008276,0032259,0052699,0052704,0052706 Ki=2.6uM remove_due_to_license_issue A0R5M8 29658702 403 HMALSLANYLAADSAAEALRRDVRAGLTATQKSLPPKWFYDAGSDLFDQITRLPEYYPTRTEAQILRTRSAEIISAAGADTLVELGSGTSEKTRMLLDAMRDAELLRRFIPFDVDAGVLRSAGAAIGAEYPGIEIDAVCGDFEEHLGKIPHVGRRLVVFLGSTIGNLTPAPRAEFLSTLADTLQPGDSLLLGTDLVKDTGRLVRAYDDAAGVTAAFNRNVLAVVNRELSADFDLDAFEHVAKWNSDEERIEMWLRARTAQHVRVAALDLEVDFAAGEEMLTEVSCKFRPENVVAELAEAGLRQTHWWTDPAGDFGLSLAVR 6fns A 1.85 BS01 DY8 A 1 Y39 F47 Y56 G161 T163 N166 Y206 E282 S284 Y40 F48 Y57 G162 T164 N167 Y207 E283 S285 2.1.1.44 0008168,0008276,0032259,0052699,0052704,0052706 Ki=93uM remove_due_to_license_issue A0R5M8 29658702 401 HMALSLANYLAADSAAEALRRDVRAGLTATQKSLPPKWFYDAVGSDLFDQITRLPEYYPTRTEAQILRTRSAEIISAAGADTLVELGSGTSEKTRMLLDAMRDAELLRRFIPFDVDAGVLRSAGAAIGAEYPGIEIDAVCGDFEEHLGKIPHVGRRLVVFLGSTIGNLTPAPRAEFLSTLADTLQPGDSLLLGTDLVKDTGRLVRAYDDAAGVTAAFNRNVLAVVNRELSADFDLDAFEHVAKWNSDEERIEMWLRARTAQHVRVAALDLEVDFAAGEEMLTEVSCKFRPENVVAELAEAGLRQTHWWTDPAGDFGLSLAVR 6fnt A 1.9 BS01 AVO A 1 Y39 F47 Y56 G161 T163 N166 Y206 E282 S284 Y40 F48 Y57 G162 T164 N167 Y207 E283 S285 2.1.1.44 0008168,0008276,0032259,0052699,0052704,0052706 Ki=21uM remove_due_to_license_issue A0R5M8 29658702 401 HMALSLANYLAADSAAEALRRDVRAGLTATQKSLPPKWFYDAVGSDLFDQITRLPEYYPTRTEAQILRTRSAEIISAAGADTLVELGSGTSEKTRMLLDAMRDAELLRRFIPFDVDAGVLRSAGAAIGAEYPGIEIDAVCGDFEEHLGKIPHVGRRLVVFLGSTIGNLTPAPRAEFLSTLADTLQPGDSLLLGTDLVKDTGRLVRAYDDAAGVTAAFNRNVLAVVNRELSADFDLDAFEHVAKWNSDEERIEMWLRARTAQHVRVAALDLEVDFAAGEEMLTEVSCKFRPENVVAELAEAGLRQTHWWTDPAGDFGLSLAVR 6fnx A 1.19 BS01 DYZ A 1 W81 P82 F83 V87 N140 I146 W40 P41 F42 V46 N99 I105 ? ic50=12.6uM remove_due_to_license_issue IC50=12589nM O60885 29883107 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6fo5 A 0.95 BS01 DZH A 1 P82 F83 L92 L94 N140 D145 M149 P41 F42 L51 L53 N99 D104 M108 ? Kd=0.19uM remove_due_to_license_issue IC50=251nM, Kd=190nM O60885 29883107 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6fo7 A 2.59 BS02 LX3 A 1 Y175 L258 S265 I299 R302 S303 S306 W314 C316 Y323 V328 H333 H423 Y22 L45 S52 I86 R89 S90 S93 W101 C103 Y110 V115 H120 H210 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Q9PTN2 29733645 4000 HMLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV 6fo8 1 2.3 BS02 DZT 1 1 Y175 L258 L261 S265 I296 I299 R302 S303 S306 W314 C316 Y323 H333 H423 Y20 L43 L46 S50 I81 I84 R87 S88 S91 W99 C101 Y108 H118 H208 ? 0003677,0004879,0005634,0006355 ic50=18.4nM remove_due_to_license_issue Q9PTN2 29733645 500 LSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSE 6fo9 A 2.701 BS02 E0E A 1 Y175 S265 I299 R302 S303 S306 W314 C316 Y323 V328 H333 H423 Y22 S52 I86 R89 S90 S93 W101 C103 Y110 V115 H120 H210 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Q9PTN2 29733645 500 HMLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV 6fob A 2.75 BS02 DZW A 1 Y175 M254 L258 V262 S265 I299 R302 S303 S306 W314 C316 Y323 V328 H333 H423 F448 Y21 M40 L44 V48 S51 I85 R88 S89 S92 W100 C102 Y109 V114 H119 H209 F234 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Q9PTN2 29733645 501 MLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV 6fod A 2.5 BS02 E05 A 1 Y175 S265 I299 R302 S303 S306 W314 C316 Y323 H333 H423 Y427 F448 Y22 S52 I86 R89 S90 S93 W101 C103 Y110 H120 H210 Y214 F235 ? 0003677,0004879,0005634,0006355 ic50=7.11nM remove_due_to_license_issue Q9PTN2 29733645 4000 HMLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSWSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV 6fpu A 1.36 BS02 E48 A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 V282 D92 Y96 D142 C144 G215 L217 A218 M246 G247 V268 D102 D280 C318 C320 C323 H349 D92 D266 C304 C306 C309 H335 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0046872,0101030 Kd=321nM remove_due_to_license_issue P28720 29939431 405 RPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLSSLTKQSEEGVTFKSHRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 6fq3 A 1.901 BS01 rna B 0 C563 R564 R581 S582 R611 K628 D629 Y658 R676 R707 F722 R752 R770 C129 R130 R147 S148 R177 K194 D195 Y224 R242 R273 F288 R318 R336 2.3.2.27 remove_due_to_license_issue E7FAM5 29674686 1 ~ 13 SSGAFATASKAHGEGIKRALQGKPASFTVVGYDHDGEPRLSGGDSVSVVLMSPDGNLSSAEVSDHQDGTYTVSYLPKGEGEHLLSVLICNQHIEGSPFKVMVKSGRSYGGVGLPMASFGGEGDGDGQLCRPWGICVDKEGYVVVADRSNNRVQIFKPCGTFHHKFGTLGSRPGQFDRPAGVACDSQRRIIVADKDNHRIQIFTFDGQFLLKFGEKGTKNGQFNYPWDVAVNFEGKILVSDTRNHRVQLFGPDGTFLNKYGFEGALWKHFDSPRGVAFNQEGHLVVTDFNNHRLLVIRPDCQSARFLGSEGTGNGQFLRPQGVAVDQEDRIIVADSRNHRIQVFEPNGNFLCKFGTHGNGFGQMDRPSGIAVTPDGVIVAVDFGNNRILMF 6fqo A 1.35 BS01 E2T A 1 L1109 P1110 Q1113 V1115 L1120 N1168 R1173 V1174 L27 P28 Q31 V33 L38 N86 R91 V92 2.3.1.-,2.3.1.48 ic50=0.14uM remove_due_to_license_issue IC50=140nM Q92793 30258543 1201 KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 6fqp A 2.42 BS01 dna L 0 R168 N170 L171 Q210 N217 R221 R1 N3 L4 Q43 N50 R54 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 RGNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRKDGKDP 6fqp A 2.42 BS02 dna M 0 R168 Y191 K197 I216 R219 R220 R1 Y24 K30 I49 R52 R53 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 RGNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRKDGKDP 6fqp B 2.42 BS01 dna L 0 R165 R166 R167 R168 G169 Y191 K197 I216 R219 R220 R2 R3 R4 R5 G6 Y28 K34 I53 R56 R57 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 KRRRRGNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqp B 2.42 BS02 dna M 0 R165 R167 N170 L171 Q210 N217 R221 R2 R4 N7 L8 Q47 N54 R58 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 KRRRRGNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq A 3.25 BS01 dna L 0 L171 Q210 N217 R221 L2 Q41 N48 R52 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 NLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq A 3.25 BS02 dna M 0 Y191 K197 R219 R220 Y22 K28 R50 R51 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 NLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq B 3.25 BS01 dna L 0 Y191 K197 R219 R220 Y23 K29 R51 R52 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 GNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq B 3.25 BS02 dna M 0 N217 R221 N49 R53 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 GNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq D 3.25 BS01 dna G 0 N170 L171 N217 R221 N4 L5 N51 R55 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 AAGNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq D 3.25 BS02 dna H 0 Y191 K197 I216 R219 R220 Y25 K31 I50 R53 R54 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 AAGNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq E 3.25 BS01 dna G 0 G169 N170 Y191 K197 R219 R220 G1 N2 Y23 K29 R51 R52 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 GNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqq E 3.25 BS02 dna H 0 L171 Q210 N213 N217 R221 L3 Q42 N45 N49 R53 ? 0003677,0006355 remove_due_to_license_issue Q15583 30060237 1 ~ 16 GNLPKESVQILRDWLYEHRYNAYPSEQEKALLSQQTHLSTLQVCNWFINARRRLLPDMLRK 6fqr A 2.1 BS01 rna C 0 Y5 L34 Y39 F41 S73 V74 R79 Y6 L35 Y40 F42 S74 V75 R80 ? 0003676,0003723 remove_due_to_license_issue O00425 30135093 1 ~ 3 SMNKLYIGNLSENAAPSDLESIFKDAKIPVSGPFLVKTGYAFVDCPDESWALKAIEALSGKIELHGKPIEVEHSVPKRQRIRKLQIRNIPPHLQWEVLDSLLVQYGVVESCEQVNTDSETAVVNVTYSSKDQARQALDKLNGFQLENFTLKVAYIPDE 6fqu A 1.43 BS01 E3B A 1 P1110 V1115 L1120 N1168 R1173 V1174 F1177 P29 V34 L39 N87 R92 V93 F96 2.3.1.-,2.3.1.48 ic50=2.2uM remove_due_to_license_issue IC50=2200nM Q92793 30258543 1201 KKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 6fr0 A 1.5 BS01 E3H A 1 P1110 Q1113 V1115 L1120 N1168 R1173 V1174 P27 Q30 V32 L37 N85 R90 V91 2.3.1.-,2.3.1.48 ic50=0.146uM remove_due_to_license_issue IC50=146nM Q92793 30258543 1201 IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 6fr2 A 2.262 BS01 E3N A 1 D335 W336 M339 I375 F381 Y383 Q384 M419 Y466 V498 H524 D107 W108 M111 I147 F153 Y155 Q156 M191 Y238 V270 H296 F267 D335 W336 D496 H524 F39 D107 W108 D268 H296 3.1.3.76,3.3.2.10 0003824 ic50=4.99nM remove_due_to_license_issue P34913 30059891 601 PTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 6frf A 2.1 BS01 E3T A 1 P1110 Q1113 V1115 L1120 N1168 R1173 V1174 P31 Q34 V36 L41 N89 R94 V95 2.3.1.-,2.3.1.48 ic50=0.04uM remove_due_to_license_issue IC50=40nM Q92793 30258543 1201 MRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG 6fs0 A 2.25 BS01 E4W A 1 A227 M231 L235 V249 V253 R263 T266 L267 F270 G271 I294 A62 M66 L70 V84 V88 R98 T101 L102 F105 G106 I129 ? 0042981 Kd=0.00017uM remove_due_to_license_issue IC50=<3.00nM, Ki=0.200000nM Q07820 30559424 401 GPLGSEDDLYRQSLEIISRYLREQATGSKDSKPLGEAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6fs1 A 1.6 BS01 E4Q A 1 F228 M231 V249 M250 V253 R263 T266 L267 F270 G271 I294 F57 M60 V78 M79 V82 R92 T95 L96 F99 G100 I123 ? 0042981 Kd=0.098uM remove_due_to_license_issue Ki=42nM, IC50=42nM, Kd=94nM Q07820 30559424 401 DDLYRQSLEIISRYLREQATGSKDSKPLGEAGAAGRRALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6fsd A 2.7 BS01 E5H A 1 Y72 Y124 W286 Y337 F338 Y72 Y124 W279 Y330 F331 G121 G122 S203 A204 E334 H447 G121 G122 S203 A204 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 30339371 601 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 6fse A 2.7 BS01 E5K A 1 Y72 W86 G120 G121 Y124 W286 Y337 F338 Y341 Y72 W86 G120 G121 Y124 W279 Y330 F331 Y334 G121 G122 S203 A204 E334 H447 G121 G122 S203 A204 E327 H440 3.1.1.7 0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005794,0005886,0006581,0007155,0009986,0016020,0016787,0017171,0031594,0031623,0042166,0042802,0042803,0043236,0045202,0048471,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P21836 30339371 601 EGREDPQLLVRVRGGQLRGIRLKAPGGPVSAFLGIPFAEPPVGSRRFMPPEPKRPWSGVLDATTFQNVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPASPTPVLIWIYGGGFYSGAASLDVYDGRFLAQVEGAVLVSMNYRVGTFGFLALPGSREAPGNVGLLDQRLALQWVQENIAAFGGDPMSVTLFGESAGAASVGMHILSLPSRSLFHRAVLQSGTPNGPWATVSAGEARRRATLLARLVGCNDTELIACLRTRPAQDLVDHEWHVLPQESIFRFSFVPVVDGDFLSDTPEALINTGDFQDLQVLVGVVKDEGSYFLVYGVPGFSKDNESLISRAQFLAGVRIGVPQASDLAAEAVVLHYTDWLHPEDPTHLRDAMSAVVGDHNVVCPVAQLAGRLAAQGARVYAYIFEHRASTLTWPLWMGVPHGYEIEFIFGLPLDPSLNYTTEERIFAQRLMKYWTNFARTGDPNDPRDSKSPQWPPYTTAAQQYVSLNLKPLEVRRGLRAQTCAFWNRFLPKLLSA 6fsy A 1.34 BS01 E5Q A 1 W81 P82 F83 L92 N140 M149 W40 P41 F42 L51 N99 M108 ? remove_due_to_license_issue IC50=166nM, Kd=247nM O60885 29776834 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6ft3 A 1.28 BS01 E5T A 1 W81 P82 V87 L92 N140 I146 W40 P41 V46 L51 N99 I105 ? remove_due_to_license_issue IC50=377nM O60885 29776834 202 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6ft4 A 1.34 BS01 E5W A 1 P82 F83 L92 N140 I146 M149 P41 F42 L51 N99 I105 M108 ? remove_due_to_license_issue IC50=235nM O60885 29776834 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6ft7 A 2.02 BS01 E6Q A 1 G163 E164 V170 A184 F236 L239 L290 G35 E36 V42 A56 F108 L111 L162 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P49761 29723265 511 SKRSSRSVEDDKEGHLVCRIGDWLQERYEIVGNLGEGTFGKVVECLDHARGKSQVALKIIRNVGKYREAARLEINVLKKIKEKDKENKFLCVLMSDWFNFHGHMCIAFELLGKNTFEFLKENNFQPYPLPHVRHMAYQLCHALRFLHENQLTHTDLKPENILFVNSEFETLYNEHKSCEEKSVKNTSIRVADFGSATFDHEHHTTIVATRHYRPPEVILELGWAQPCDVWSIGCILFEYYRGFTLFQTHENREHLVMMEKILGPIPSHMIHRTRKQKYFYKGGLVWDENSSDGRYVKENCKPLKSYMLQDSLEHVQLFDLMRRMLEFDPAQRITLAEALLHPFFAGLTPEERSFHT 6ft8 A 1.45 BS01 E6T A 1 L167 G168 V175 A189 F241 L244 D250 L295 L22 G23 V30 A44 F96 L99 D105 L150 D288 K290 N293 D325 T342 D143 K145 N148 D180 T197 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P49759 29723265 501 SMHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKKS 6ft9 A 1.87 BS01 E6W A 1 L167 G168 V175 A189 F241 E242 L244 E292 L295 L21 G22 V29 A43 F95 E96 L98 E146 L149 D288 K290 N293 D325 T342 D142 K144 N147 D179 T196 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P49759 29723265 501 MHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKK 6ftn A 2.0 BS01 E78 A 1 W760 I777 K779 D787 Y813 C815 I825 V828 S831 M900 I910 W569 I586 K588 D596 Y622 C624 I634 V637 S640 M709 I719 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 ic50=200nM remove_due_to_license_issue O35904 29852070 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELGRHLQLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 6ftp A 1.8 BS01 DM2 B 1 L273 S274 F277 E278 L280 L248 S249 F252 E253 L255 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 remove_due_to_license_issue P01011 29760101 501 LASANVDFAFSLYKQLVLKAPDKNVIFSPLSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNQSSDELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKFEMPFDPQDTHQSRFYLSKKKYVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASALFILPDQDKMEEVEAMLSQETLSRFFESLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTERSAATALEVLFQ 6ftp B 1.8 BS01 DM2 B 1 V381 N383 W386 V15 N17 W20 ? remove_due_to_license_issue P01011 29760101 501 RTIVRFNRPFLMIIVDNFTWSIFFMSKVTNPKQA 6ftw A 2.16 BS02 E6Z A 1 M273 I336 M337 M357 S368 Q369 F372 M193 I256 M257 M277 S288 Q289 F292 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 31327675 517 RFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6fty A 1.67 BS01 E7H A 1 L41 C42 H57 S190 C191 K192 S195 S215 S217 R218 C220 L25 C26 H41 S178 C179 K180 S183 S199 S201 R202 C204 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 remove_due_to_license_issue Kd=>2000000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 6ftz A 1.67 BS01 E7E A 1 D189 S190 C191 K192 S195 V213 S215 R218 D177 S178 C179 K180 S183 V197 S199 R202 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=1000uM remove_due_to_license_issue Kd=1000000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 6fu1 A 1.548 BS02 E7Q A 1 D100 G139 W140 H141 H142 G150 F151 D186 H188 F216 H292 G338 G339 Y341 D99 G138 W139 H140 H141 G149 F150 D176 H178 F206 H273 G306 G307 Y309 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=4.4uM remove_due_to_license_issue A5H660 29498707 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6fu1 A 1.548 BS03 E7Q A 2 G238 R239 G219 R220 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=4.4uM remove_due_to_license_issue A5H660 29498707 506 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6fu4 A 2.45 BS01 HSM A 1 Y126 Y158 E170 M172 E176 Y189 W192 Y208 D210 D239 Y79 Y111 E123 M125 E129 Y142 W145 Y161 D163 D192 ? Kd=639nM remove_due_to_license_issue Q9I0I4 30425146 401 QMLDESARLRLEARGELQALRIQRYFMDAFQYGKGFSRQILFLRDQAQKRFLDAYDLREDLTRQVRTALAANPEVLGLYVVFEPNALDGKDELFVDQPALGSNDKGRFSLYWAQATPGQLESESMIESELADTSSGPSGAAYNAWYTCPKESGQPCVLDPYFDKVGERQLLMTSIAFPLELDGKVIGVMGLDINLSNLQALSEQGNRELYDGVGQVGILSPAGLFAGNSRDAGLLGKNLAKADPQHAGELLQLLAAGKSRLFNENDDLKVLQPLQPIPGAKPWGVLLEVPKSALLGP 6fu5 A 3.26 BS01 E7N A 1 L24 V32 A45 K47 L79 T95 M98 G101 E105 L153 D164 L20 V28 A41 K43 L72 T88 M91 G94 E98 L146 D157 D146 Q150 N151 D164 D139 Q143 N144 D157 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43353 30026309 400 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLTPLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLGTIIYMPPENYEPSIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLKKTKLQ 6fug A 2.21 BS01 E85 A 1 I143 H146 D189 S190 C191 K192 S195 V213 R218 V219 C220 I125 H128 D166 S167 C168 K169 S172 V186 R188 V189 C190 H57 D102 K192 G193 D194 S195 G196 H41 D84 K169 G170 D171 S172 G173 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=50uM remove_due_to_license_issue IC50=20000nM, Kd=50000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTRVCGNRKKPGIYTRVASYAAWIDSVLASA 6fuh A 1.37 BS01 E88 A 1 C42 H57 D189 S190 C191 K192 G193 S195 V213 S215 S217 R218 C26 H41 D177 S178 C179 K180 G181 S183 V197 S199 S201 R202 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=170uM remove_due_to_license_issue Kd=170000nM, IC50=75000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 6fui A 1.38 BS01 E7W A 1 H57 C58 D189 S190 C191 K192 G193 S195 S215 S217 R218 C220 H41 C42 D177 S178 C179 K180 G181 S183 S199 S201 R202 C204 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=35uM remove_due_to_license_issue IC50=84000nM, Kd=35000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVL 6fuj A 2.25 BS01 E8B A 1 D189 S190 C191 K192 S215 R218 D177 S178 C179 K180 S199 R202 H57 D102 K192 G193 D194 S195 G196 H41 D89 K180 G181 D182 S183 G184 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 ic50=120uM remove_due_to_license_issue IC50=120000nM, Kd=120000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA 6ful A 1.649 BS01 E7Z A 1 Y1135 K1137 T1143 H1146 N1156 H1226 V1228 Y218 K220 T226 H229 N239 H309 V311 1.14.11.68 remove_due_to_license_issue O15550 30226987 1501 SVSIYPSSAEVLKACRNLSNSSILLDKCPPPRPPSSPYPPLPKDKLNPPTPSIYLENKRDAFFPPLHQFCTNPNNPVTVIRGLAGALKLDLGLFSTKTLVEANNEHMVEVRTQLLQPADENWDPTGTKKIWHCESNRSHTTIAKYAQYQASSFQESLREEPFKTIKFGTNIDLSDDKKWKLQLHELTKLPAFVRVVSAGNLLSHVGHTILGMNTVQLYMKVPGSRTPGHQENNNFCSVNINIGPGDCEWFVVPEGYWGVLNDFCEKNNLNFLMGSWWPNLEDLYEANVPVYRFIQRPGDLVWINAGTVHWVQAIGWCNNIAWNVGPLTACQYKLAVERYEWNKLQSVKSIVPMVHLSWNMARNIKVSDPKLFEMIKYCLLRTLKQCQTLREALIAAGKEIIWHGRTKEEPAHYCSICEVEVFDLLFVTNESNSRKTYIVHCQDCARKTSGNLENFVVLEQYKMEDLMQVYDQFTLAPP 6fut A 1.5 BS01 E82 A 1 H146 S190 C191 K192 S195 S215 S217 R218 V219 C220 H129 S174 C175 K176 S179 S195 S197 R198 V199 C200 H57 D102 K192 G193 D194 S195 G196 H41 D85 K176 G177 D178 S179 G180 3.4.21.46 0004252,0005576,0005615,0006508,0006956,0006957,0008236,0009617,0016787,0031093,0034774,0051604,0070062,1904813 Kd=20uM remove_due_to_license_issue Kd=20000nM, IC50=32000nM P00746 29795765 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASAAA 6fv1 A 2.3 BS01 E8E A 1 H41 F139 N141 G142 C144 H163 Q164 I165 E166 P189 H41 F139 N141 G142 C144 H163 Q164 I165 E166 P189 2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue P0C6X5 32045235 401 SGLKKMAQPSGCVERCVVRVCYGSTVLNGVWLGDTVTCPRHVIAPSTTVLIDYDHAYSTMRLHNFSVSHNGVFLGVVGVTMHGSVLRIKVSQSNVHTPKHVFKTLKPGDSFNILACYEGIASGVFGVNLRTNFTIKGSFINGACGSPGYNVRNDGTVEFCYLHQIELGSGAHVGSDFTGSVYGNFDDQPSLQVESANLMLSDNVVAFLYAALLNGCRWWLCSTRVNVDGFNEWAMANGYTSVSSVECYSILAAKTGVSVEQLLASIQHLHEGFGGKNILGYSSLCDEFTLAEVVKQMYGV 6fv2 A 2.95 BS01 D03 A 1 V26 H41 I51 F139 N141 G142 A143 C144 H163 E166 D187 Q188 S190 V26 H41 I51 F139 N141 G142 A143 C144 H163 E166 D187 Q188 S190 2.1.1.57,2.7.7.48,2.7.7.50,3.1.13.-,3.4.19.12,3.4.22.-,3.6.4.12,3.6.4.13,4.6.1.- 0008233,0019082 remove_due_to_license_issue P0C6X5 32045235 402 SGLKKMAQPSGCVERCVVRVCYGSTVLNGVWLGDTVTCPRHVIAPSTTVLIDYDHAYSTMRLHNFSVSHNGVFLGVVGVTMHGSVLRIKVSQSNVHTPKHVFKTLKPGDSFNILACYEGIASGVFGVNLRTNFTIKGSFINGACGSPGYNVRNDGTVEFCYLHQIELGSGAHVGSDFTGSVYGNFDDQPSLQVESANLMLSDNVVAFLYAALLNGCRWWLCSTRVNVDGFNEWAMANGYTSVSSVECYSILAAKTGVSVEQLLASIQHLHEGFGGKNILGYSSLCDEFTLAEVVKQMYGVN 6fv4 A 1.974 BS02 16G A 1 G132 A133 H134 H188 N212 A213 H244 I301 A302 G303 G135 A136 H137 H191 N215 A216 H247 I304 A305 G306 3.5.1.25 0006040,0006044,0006046,0008448,0016787,0016810,0046872 remove_due_to_license_issue A0QU89 29728457 402 GSHMLLTADTVLTGTELLRPGWLEIASDRVVAVGAGAPPAQADRNLGAATVVPGFVDTHLHGGGGGNFSAATDDETARAVALHRAHGSTTLVASLVTAGPEDLLRQVSGLARQVRAGLIDGIHLEGPWLSTLRCGAHQPVLMRDPDPGEIGRVLDAGEGTVRMVTIAPERDGALAAIAQLVNAGVVAAVGHTEATYDQTRAAIDAGATVGTHLFNAMRPIDRREPGPAVALTEDSRVTVEMIVDGVHVAPAIYRHITQTVGPERLSLITAAMAATGMSDGVYRLGPLDIDVVAGVARVAGTDTIAGSTATMEQVFRLAVAHCGLPRDDALSLAVRQACVNPARALGLPAAGLAAGARADLVVLDHDLAVTAVMRAGEWVVT 6fwr A 2.5 BS01 dna B 0 N85 V86 F113 G114 R117 N223 A225 L226 A229 A542 S543 R545 Q564 L591 Q592 S593 K612 F615 P616 P617 I618 D619 Y636 F638 R673 Y679 N84 V85 F112 G113 R116 N222 A224 L225 A228 A537 S538 R540 Q559 L586 Q587 S588 K607 F610 P611 P612 I613 D614 Y631 F633 R668 Y674 3.6.4.12 0003676,0003677,0003678,0003689,0004386,0005515,0005524,0006139,0006281,0006338,0009378,0009432,0016787,0016818,0016853,0016887,0032508,0033677,0036121,0043139,0044806,0046872,0051539,0061749,0061775,0140584,0140588,0140665,0140849,1990518 remove_due_to_license_issue P27296 30520735 1 ~ 11 ALTAALKAQIAAWYKALQEQIPDFIPRAPQRQMIADVAKTLAGEEGRHLAIEAPTGVGKTLSYLIPGIAIAREEQKTLVVSTANVALQDQIYSKDLPLLKKIIPDLKFTAAFGRGRYVCPRNLTALASTEPTQQDLLAFLDDELTPNNQEEQKRCAKLKGDLDTYKWDGLRDHTDIAIDDDLWRRLSTDKASCLNRNCYYYRECPFFVARREIQEAEVVVANHALVMAAMESEAVLPDPKNLLLVLDEGHHLPDVARDALEMSAEITAPWYRLQLDLFTKLVATCMEQFRPKTIPPLAIPERLNAHCEELYELIASLNNILNLYMPAGQEAEHRFAMGELPDEVLEICQRLAKLTEMLRGLAELFLNDLSEKDIVRLHRLILQMNRALGMFEAQSKLWRLASLAQSSGAPVTKWATREEREGQLHLWFHCVGIRVSDQLERLLWRSIPHIIVTSATLRSLNSFSRLQEMSGLKEKAGDRFVALDSPFNHCEQGKIVIPRMRVEPSIDNEEQHIAEMAAFFREQVESKKHLGMLVLFASGRAMQRFLDYVTDLRLMLLVQGDQPRYRLVELHRKRVANGERSVLVGLQSFAEGLDLKGDLLSQVHIHKIAFPPIDSPVVITEGEWLKSLNRYPFEVQSLPSASFNLIQQVGRLIRSHGCWGEVVIYDKRLLTKNYGKRLLDALPVFPIEQPEVPEGIVKK 6fx1 A 2.1 BS01 FUC M 1 G12 D13 G12 D13 ? 0046872 remove_due_to_license_issue A0A3B6UEU4 29956878 6 APVPVTKLVCDGDTYKCTAYLDFGDGRWVAQWDTNVFHTG 6fx1 A 2.1 BS02 C4W O 1 F23 W28 F23 W28 ? 0046872 remove_due_to_license_issue A0A3B6UEU4 29956878 1 APVPVTKLVCDGDTYKCTAYLDFGDGRWVAQWDTNVFHTG 6fx1 A 2.1 BS03 FUC O 1 A1 F23 A1 F23 ? 0046872 remove_due_to_license_issue A0A3B6UEU4 29956878 6 APVPVTKLVCDGDTYKCTAYLDFGDGRWVAQWDTNVFHTG 6fx1 B 2.1 BS01 C4W M 1 F23 W28 F25 W30 ? 0046872 remove_due_to_license_issue A0A3B6UEU4 29956878 1 AMAPVPVTKLVCDGDTYKCTAYLDFGDGRWVAQWDTNVFHTG 6fx1 B 2.1 BS02 FUC M 1 A1 F23 A3 F25 ? 0046872 remove_due_to_license_issue A0A3B6UEU4 29956878 6 AMAPVPVTKLVCDGDTYKCTAYLDFGDGRWVAQWDTNVFHTG 6fx1 B 2.1 BS03 FUC N 1 G12 D13 G14 D15 ? 0046872 remove_due_to_license_issue A0A3B6UEU4 29956878 8 AMAPVPVTKLVCDGDTYKCTAYLDFGDGRWVAQWDTNVFHTG 6fyi A 2.6 BS01 EAE A 1 F174 A191 K193 L246 L297 F27 A44 K46 L99 L150 D290 K292 N295 D327 T344 D143 K145 N148 D180 T197 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=95nM P49760 29985556 501 EGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGARVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPIPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEEHHQLFDLIESMLEYEPAKRLTLGEALQHPFFARLR 6fyk A 2.39 BS01 EAZ A 1 E171 F174 A191 K193 F243 L246 N295 L297 V326 D327 E35 F38 A55 K57 F107 L110 N159 L161 V190 D191 2.7.12.1 0004672,0005524,0006468 ic50=3nM remove_due_to_license_issue P49760 29985556 501 SRRAKSVEDDAEGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGARVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPIPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEEHHQLFDLIESMLEYEPAKRLTLGEALQHPFFARLRAE 6fyl A 1.95 BS01 3NG A 1 L169 G170 E171 F174 V177 A191 K193 F243 L246 L297 V326 D327 L26 G27 E28 F31 V34 A48 K50 F100 L103 L154 V183 D184 2.7.12.1 0004672,0005524,0006468 ic50=7nM remove_due_to_license_issue IC50=4.0nM P49760 29985556 501 EDDAEGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGARVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPIPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEEHHQLFDLIESMLEYEPAKRLTLGEALQHPFFARLR 6fym A 2.15 BS01 EBB A 1 H1682 G1683 T1684 D1685 Y1701 G1703 Y1714 Y1721 Y1727 L1782 H70 G71 T72 D73 Y89 G91 Y102 Y109 Y115 L170 2.4.2.- 0003950 remove_due_to_license_issue Q460N5 30344052 1901 KQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 6fyp A 2.29 BS01 3NG A 1 L162 G163 E164 F167 V170 A184 K186 V220 F236 L239 N242 L290 D320 L28 G29 E30 F33 V36 A50 K52 V86 F102 L105 N108 L156 D186 2.7.12.1 0004672,0005524,0006468 ic50=143nM remove_due_to_license_issue IC50=41nM P49761 29985556 501 SVEDDKEGHLVCRIGDWLQERYEIVGNLGEGTFGKVVECLDHARGKSQVALKIIRNVGKYREAARLEINVLKKIKEKDKENKFLCVLMSDWFNFHGHMCIAFELLGKNTFEFLKENNFQPYPLPHVRHMAYQLCHALRFLHENQLTHTDLKPENILFVNSEFETLYNEHKSCEEKSVKNTSIRVADFGSATFDHEHHTTIVATRHYRPPEVILELGWAQPCDVWSIGCILFEYYRGFTLFQTHENREHLVMMEKILGPIPSHMIHRTRKQKYFYKGGLVWDENSSDGRYVKENCKPLKSYMLQDSLEHVQLFDLMRRMLEFDPAQRITLAEALLHPFFAGLTPEERSF 6fyv A 2.46 BS01 3NG A 1 L167 G168 E169 F172 V175 A189 K191 F241 L244 L295 V324 D325 L18 G19 E20 F23 V26 A40 K42 F92 L95 L146 V172 D173 D288 K290 N293 D325 T342 D139 K141 N144 D173 T190 2.7.12.1 0004672,0005524,0006468 ic50=11nM remove_due_to_license_issue Q9HAZ1 29985556 501 ICQSGDVLRARYEIVDTLGEGAFGKVVECIDHGMDGMHVAVKIVKNVGRYREAARSEIQVLEHLNSTDPNSVFRCVQMLEWFDHHGHVCIVFELLGLSTYDFIKENSFLPFQIDHIRQMAYQICQSINFLHHNKLTHTDLKPENILFVKSDYVVKYNKRDERTLKNTDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFQTHDSKEHLAMMERILGPIPQHMIQKTRKRKYFHHNQLDWDEHSSAGRYVRRRCKPLKEFMLCHDEEHEKLFDLVRRMLEYDPTQRITLDEALQHPFFDLLK 6fyz A 2.15 BS01 EBE A 1 E677 H802 H803 G811 F812 D840 H842 F871 P942 G974 E28 H121 H122 G130 F131 D159 H161 F190 P261 G293 3.5.1.98 Kd=0.039uM remove_due_to_license_issue IC50=36nM, Kd=80nM P56524 30463802 2001 PRFTTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPLIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELQQRPNANAVRSMEKVMEIHSKYWRCLQRH 6fz4 A 1.85 BS01 EC8 A 1 E13 Y61 P88 L89 T90 R95 D139 G140 S141 T144 Y216 E10 Y58 P85 L86 T87 R92 D136 G137 S138 T141 Y213 ? 0015276,0016020 Ki=1.12uM remove_due_to_license_issue P22756 30620174 307 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRG 6fzg A 2.1 BS01 EDK A 1 F310 G312 C313 Q314 S317 H351 I369 F388 F391 H477 L493 L497 Y501 F81 G83 C84 Q85 S88 H122 I140 F159 F162 H248 L264 L268 Y272 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Ki=1.4nM, EC50=6.2nM P37231 30651555 550 MQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKMKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 6fzm A 2.67 BS01 EE5 A 1 H1682 G1683 K1704 N1705 Y1714 Y1721 S1722 T1726 Y1727 L1782 H71 G72 K93 N94 Y103 Y110 S111 T115 Y116 L171 2.4.2.- 0003950 remove_due_to_license_issue Q460N5 30344052 1901 MKQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 6fzu A 1.8 BS02 EE8 A 1 C320 V376 F377 F378 C57 V113 F114 F115 ? 0003677,0004879,0005634,0006355 ic50=216uM remove_due_to_license_issue IC50=216000nM P51449 29990434 601 YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFST 6fzx A 2.1 BS01 EEK A 1 N112 A113 H140 E141 H144 E164 D221 H223 H224 N112 A113 H140 E141 H144 E164 D221 H223 H224 H140 E141 H144 Y155 E164 D221 H223 H140 E141 H144 Y155 E164 D221 H223 3.4.24.26 0004222,0006508 Ki=12.3uM remove_due_to_license_issue P14756 30088919 401 AEAGGPGGNQKIGKYTYGSDYGPLIVNDRCEMDDGNVITVDMNSSTDDSKTTPFRFACPTNTYKQVNGAYSPLNDAHFFGGVVFKLYRDWFGTSPLTHKLYMKVHYGRSVENAYWDGTAMLFGDGATMFYPLVSLDVAAHEVSHGFTEQNSGLIYRGQSGGMNEAFSDMAGEAAEFYMRGKNDFLIGYDIKKGSGALRYMDQPSRDGRSIDNASQYYNGIDVHHSSGVYNRAFYLLANSPGWDTRKAFEVFVDANRYYWTATSNYNSGACGVIRSAQNRNYSAADVTRAFSTVGVTCP 6g01 A 1.61 BS03 EEW A 1 R118 E119 D151 R152 R225 E277 R293 N295 R368 Y402 R37 E38 D70 R71 R144 E196 R212 N214 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue C6KP13 30404922 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 6g02 A 1.84 BS02 EF8 A 1 R118 E119 D151 R152 R225 E277 R293 R368 Y402 P431 R37 E38 D70 R71 R144 E196 R212 R287 Y321 P350 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 remove_due_to_license_issue C3W6G3 30404922 502 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 6g07 A 1.66 BS03 EEZ A 1 Q286 L287 C320 R364 M365 R367 A368 F377 F378 F388 I400 Q23 L24 C57 R101 M102 R104 A105 F114 F115 F125 I137 ? 0003677,0004879,0005634,0006355 Kd=35.5nM remove_due_to_license_issue IC50=255nM, Kd=36nM P51449 29990434 601 YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFST 6g0v A 1.09 BS01 EGZ A 1 H158 R162 W181 E184 H46 R50 W69 E72 ? 0030246 Kd=166uM remove_due_to_license_issue P17931 30094951 301 MLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6g0w A 2.34 BS01 EGW A 1 H1682 G1683 A1706 Y1714 S1722 Y1727 H1753 D1775 L1782 H70 G71 A92 Y98 S106 Y111 H137 D159 L166 2.4.2.- 0003950 ic50=5.2uM remove_due_to_license_issue IC50=5248nM Q460N5 29748053 1901 KQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRAGKNAVGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK 6g0z A 2.15 BS01 GDP A 1 N58 K59 D61 D86 K88 N130 G132 K133 S134 T135 N57 K58 D60 D85 K87 N129 G131 K132 S133 T134 ? 0003924,0005525,0005737,0006412 Kd=4.84uM remove_due_to_license_issue A0A0H2XK72 30366986 301 VIQWYPGHMAKAKREVSEQLKKVDVVFELVDARIPYSSRNPMIDEVINQKPRVVILNKKDMSNLNEMSKWEQFFIDKGYYPVSVDAKHGKNLKKVEAAAIKATAEKFEREKAKGLKPRAIRAMIVGIPNVGKSTLINKLAKRSIGNKPGVTKQQQWIKVGNALQLLDTPGILWPKFEDEEVGKKLSLTGAIKDSIVHLDEVAIYGLNFLIQNDLARLKSHYNIEVPEDAEIIAWFDAIGKKRGLIRRGNEIDYEAVIELIIYDIRNAKIGNYCFDIFKDMTEELANDANN 6g14 B 1.8 BS01 G4P B 1 N58 K59 D61 D86 K88 N130 G132 K133 S134 T135 N57 K58 D60 D85 K87 N129 G131 K132 S133 T134 ? 0003924,0005525,0005737,0006412 Kd=3.26uM remove_due_to_license_issue A0A0H2XK72 30366986 301 VIQWYPGHMAKAKREVSEQLKKVDVVFELVDARIPYSSRNPMIDEVINQKPRVVILNKKDMSNLNEMSKWEQFFIDKGYYPVSVDAKHGKNLKKVEAAAIKATAEKFEREKAKGLKPRAIRAMIVGIPNVGKSTLINKLAKRSIGNKPGVTKQQQWIKVGNALQLLDTPGILWPKFEDEEVGKKLSLTGAIKDHLDEVAIYGLNFLIQNDLARLKSHYNIEVPEDAEIIAWFDAIGKKRGLIRRGNEIDYEAVIELIIYDIRNAKIGNYCFDIFKDMTEELANDA 6g1l A 2.4 BS01 dna B 0 K206 H209 N210 E213 R217 N221 N242 K243 K7 H10 N11 E14 R18 N22 N43 K44 ? 0046983 remove_due_to_license_issue Q08874 30705290 1 ~ 16 AKERQKKDNHNLIERRRRFNINDRIKELGTLIPKSNDPDMRWNKGTILKASVDYIRKLQREQQRAKDLENRQKKLEHAN 6g1u A 1.79 BS01 E1K A 1 W84 G117 G118 E199 F330 W432 H440 Y442 W81 G114 G115 E196 F327 W429 H437 Y439 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29534488 607 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g1u A 1.79 BS02 E1K A 2 W84 G117 G118 E199 F330 W432 H440 W81 G114 G115 E196 F327 W429 H437 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29534488 608 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g1u A 1.79 BS03 E1K A 3 Y70 W279 Y67 W276 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29534488 609 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g1v A 1.82 BS01 E1N A 1 W84 G118 Y121 F330 Y334 W432 H440 W81 G115 Y118 F327 Y331 W429 H437 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29534488 604 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g1w A 1.9 BS01 E0Z A 1 W84 G118 Y121 L282 S286 I287 F288 R289 F330 F331 Y334 W432 I439 H440 W81 G115 Y118 L279 S283 I284 F285 R286 F327 F328 Y331 W429 I436 H437 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 29534488 604 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g22 A 1.85 BS02 2O2 A 1 D43 F49 F75 W76 V77 W96 S131 I133 K134 R163 D9 F15 F41 W42 V43 W62 S97 I99 K100 R129 D41 D43 D176 D7 D9 D142 3.1.3.- 0008253,0009264 remove_due_to_license_issue Q9NPB1 305 ALRVLVDMDGVLADFEGGFLRKFRARFPDQPFIALEDRRGFWVSEQYGRLRPGLSEKAISIWESKNFFFELEPLPGAVEAVKEMASLQNTDVFICTSPIKMFKYCPYEKYAWVEKYFGPDFLEQIVLTRDKTVVSADLLIDDRPDITGAEPTPSWEHVLFTACHNQHLQLQPPRRRLHSWADDWKAILDSKRP 6g24 A 2.1 BS01 EH2 A 1 F313 S314 N315 Q367 I370 G371 H374 Y390 F392 F48 S49 N50 Q92 I95 G96 H99 Y115 F117 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEATKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYID 6g25 A 1.432 BS01 EHQ A 1 V278 Y281 W284 F312 S314 Q316 E318 V13 Y16 W19 F47 S49 Q51 E53 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEAQKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYID 6g27 A 1.65 BS01 EHE A 1 V278 Y281 W284 F312 S314 E318 R319 V13 Y16 W19 F47 S49 E53 R54 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYID 6g28 A 1.23 BS01 AR6 A 1 D55 D56 A98 G100 G101 A102 S103 H125 G127 G128 C129 G130 H163 T167 Y263 S264 S269 S270 D302 D304 S305 D57 D58 A100 G102 G103 A104 S105 H127 G129 G130 C131 G132 H165 T169 Y265 S266 S271 S272 D304 D306 S307 3.2.2.19 0000287,0003875,0005515,0005615,0016787,0016799,0030955,0036211,0046872,0051725 remove_due_to_license_issue P54922 30472116 401 GGMEKYVAAMVLSAAGDALGYYNGKWEFLQDGEKIHRQLAQLGGLDALDVGRWRVSDDTVMHLATAEALVEAGKAPKLTQLYYLLAKHYQDCMEDMDGRAPGGASVHNAMQLKPGKPNGWRIPFNSHEGGCGAAMRAMCIGLRFPHHSQLDTLIQVSIESGRMTHHHPTGYLGALASALFTAYAVNSRPPLQWGKGLMELLPEAKKYIVQSGYFVEENLQHWSYFQTKWENYLKLRGILDGESAPTFPESFGVKERDQFYTSLSYSGWGGSSGHDAPMIAYDAVLAAGDSWKELAHRAFFHGGDSDSTAAIAGCWWGVMYGFKGVSPSNYEKLEYRNRLEETARALYSLGSKEDTVISL 6g29 A 1.7 BS01 EHK A 1 Y281 W284 F312 S314 E318 Q367 Y16 W19 F47 S49 E53 Q90 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYIDKQ 6g2a A 1.8 BS01 A3R A 1 D55 G100 G101 A102 S103 H125 G127 G128 C129 G130 H163 H165 T167 Y263 S269 S270 D304 S305 D59 G104 G105 A106 S107 H129 G131 G132 C133 G134 H167 H169 T171 Y267 S273 S274 D308 S309 3.2.2.19 0000287,0003875,0005515,0005615,0016787,0016799,0030955,0036211,0046872,0051725 remove_due_to_license_issue P54922 30472116 401 HHGGMEKYVAAMVLSAAGDALGYYNGKWEFLQDGEKIHRQLAQLGGLDALDVGRWRVSDDTVMHLATAEALVEAGKAPKLTQLYYLLAKHYQDCMEDMDGRAPGGASVHNAMQLKPGKPNGWRIPFNSHEGGCGAAMRAMCIGLRFPHHSQLDTLIQVSIESGRMTHHHPTGYLGALASALFTAYAVNSRPPLQWGKGLMELLPEAKKYIVQSGYFVEENLQHWSYFQTKWENYLKLRGILDGESAPTFPESFGVKERDQFYTSLSYSGWGGSSGHDAPMIAYDAVLAAGDSWKELAHRAFFHGGDSDSTAAIAGCWWGVMYGFKGVSPSNYEKLEYRNRLEETARALYSLGSKEDTVISL 6g2b A 1.61 BS01 EH8 A 1 V278 Y281 W284 F312 S314 Q316 E318 V13 Y16 W19 F47 S49 Q51 E53 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEAQKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYIDKQ 6g2c A 1.76 BS01 EHT A 1 V278 Y281 W284 F312 S314 Q316 E318 Q367 V13 Y16 W19 F47 S49 Q51 E53 Q91 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEQKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYIDK 6g2e A 1.85 BS01 EHH A 1 V278 Y281 W284 F312 S314 Q316 E318 V13 Y16 W19 F47 S49 Q51 E53 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEATKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYID 6g2f A 1.74 BS01 EHW A 1 Y281 W284 F312 S314 Q316 E318 Q367 Y16 W19 F47 S49 Q51 E53 Q91 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEQKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYID 6g2k A 2.01 BS01 rna R 0 C245 F247 Y249 I276 F287 Q316 K320 T321 C4 F6 Y8 I35 F46 Q75 K79 T80 ? 0003676,0003723 remove_due_to_license_issue Q15717 30418581 1 ~ 6 MGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTN 6g2k B 2.01 BS01 rna R 0 C245 F247 Y249 I276 F279 F289 Q316 K320 T321 C4 F6 Y8 I35 F38 F48 Q75 K79 T80 ? 0003676,0003723 remove_due_to_license_issue Q15717 30418581 1 ~ 6 MGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTN 6g2l A 1.48 BS02 EJ8 A 1 D41 D43 F49 F75 W76 V77 W96 S131 I133 K134 R163 K165 D12 D14 F20 F46 W47 V48 W67 S102 I104 K105 R134 K136 D41 D43 D176 D12 D14 D147 3.1.3.- 0008253,0009264 remove_due_to_license_issue Q9NPB1 303 SNAGRALRVLVDMDGVLADFEGGFLRKFRARFPDQPFIALEDRRGFWVSEQYGRLRPGLSEKAISIWESKNFFFELEPLPGAVEAVKEMASLQNTDVFICTSPIKMFKYCPYEKYAWVEKYFGPDFLEQIVLTRDKTVVSADLLIDDRPDITGAEPTPSWEHVLFTACHNQHLQLQPPRRRLHSWADDWKAILDSKRP 6g2m A 1.37 BS01 O84 A 1 D41 D43 F49 F75 W76 V77 W96 S131 I133 K134 R163 K165 D11 D13 F19 F45 W46 V47 W66 S101 I103 K104 R133 K135 D41 D43 D176 D11 D13 D146 3.1.3.- 0008253,0009264 remove_due_to_license_issue Q9NPB1 305 SNARALRVLVDMDGVLADFEGGFLRKFRARFPDQPFIALEDRRGFWVSEQYGRLRPGLSEKAISIWESKNFFFELEPLPGAVEAVKEMASLQNTDVFICTSPIKMFKYCPYEKYAWVEKYFGPDFLEQIVLTRDKTVVSADLLIDDRPDITGAEPTPSWEHVLFTACHNQHLQLQPPRRRLHSWADDWKAILDSKRP 6g2n A 1.4 BS02 O84 A 1 D14 D16 F22 F48 A50 Y69 S104 L106 L107 R136 K138 D7 D9 F15 F41 A43 Y62 S97 L99 L100 R129 K131 3.1.3.- 0000166,0000255,0005634,0005737,0005739,0005829,0006204,0006249,0008252,0008253,0009117,0009223,0009264,0016311,0016787,0016791,0019103,0042802,0043605,0046050,0046055,0046074,0046079,0046872,0050483,0070062 remove_due_to_license_issue Q8TCD5 302 SVRVLVDMDGVLADFEAGLLRGFRRRFPEEPHVPLEQRRGFLAREQYRALRPDLADKVASVYEAPGFFLDLEPIPGALDAVREMNDLPDTQVFICTSPLLKYHHCVGEKYRWVEQHLGPQFVERIILTRDKTVVLGDLLIDDKDTVRGQEETPSWEHILFTCCHNRHLVLPPTRRRLLSWSDNWREILDSKR 6g2n B 1.4 BS02 O84 B 1 D14 D16 F22 F48 L49 A50 Y69 S104 L106 L107 R136 K138 D7 D9 F15 F41 L42 A43 Y62 S97 L99 L100 R129 K131 3.1.3.- 0000166,0000255,0005634,0005737,0005739,0005829,0006204,0006249,0008252,0008253,0009117,0009223,0009264,0016311,0016787,0016791,0019103,0042802,0043605,0046050,0046055,0046074,0046079,0046872,0050483,0070062 remove_due_to_license_issue Q8TCD5 302 SVRVLVDMDGVLADFEAGLLRGFRRRFPEEPHVPLEQRRGFLAREQYRALRPDLADKVASVYEAPGFFLDLEPIPGALDAVREMNDLPDTQVFICTSPLLKYHHCVGEKYRWVEQHLGPQFVERIILTRDKTVVLGDLLIDDKDTVRGQEETPSWEHILFTCCHNRHLVLPPTRRRLLSWSDNWREILDSKR 6g2o A 1.81 BS01 EJE A 1 Y281 W284 F312 S314 Q316 E318 Q367 Y16 W19 F47 S49 Q51 E53 Q91 2.1.1.370,2.1.1.371 remove_due_to_license_issue Q9BZ95 31285596 401 VKFQVGDLVWSKVGTYPWWPCMVSSDPQLEVHTKINTRGAREYHVQFFSNQPERAWVHEKRVREYKGHKQYEELLAEQKIRKPRPQRERAQWDIGIAHAEKALKMTREERIEQYTFIYID 6g2r A 2.1 BS01 EJK A 1 F1 N46 Y48 I52 D54 Q133 N135 Y137 D140 F1 N46 Y48 I52 D54 Q133 N135 Y137 D140 ? 0007155,0009289 Kd=0.35nM remove_due_to_license_issue P08191 30710416 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 6g2s A 2.2 BS01 EJN A 1 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 F1 I13 N46 D47 Y48 I52 D54 Q133 N135 D140 ? 0007155,0009289 Kd=4.01nM remove_due_to_license_issue P08191 30710416 301 FACKTANGTAIPIGGGSANVYVNLAPVVNVGQNLVVDLSTQIFCHNDYPETITDYVTLQRGSAYGGVLSNFSGTVKYSGSSYPFPTTSETPRVVYNSRTDKPWPVALYLTPVSSAGGVAIKAGSLIAVLILRQTNNYNSDDFQFVWNIYANNDVVVPT 6g33 A 2.05 BS01 5ID A 1 G168 F172 V175 A189 F241 L244 E292 L295 G23 F27 V30 A44 F96 L99 E147 L150 D288 K290 N293 D325 T342 D143 K145 N148 D180 T197 2.7.12.1 0004672,0005524,0006468 Kd~7nM remove_due_to_license_issue P49759 29601130 501 SMHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKK 6g34 A 1.76 BS01 5ID A 1 I49 A68 F164 F166 G167 D170 G212 L215 I245 I19 A38 F134 F136 G137 D140 G182 L185 I215 2.7.11.1 0004672,0005524,0006468 Kd=5.7nM remove_due_to_license_issue Q8TF76 29601130 401 PVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g35 A 1.55 BS01 EKK A 1 I490 A509 F605 F607 G608 D611 G653 L656 I686 I30 A49 F145 F147 G148 D151 G193 L196 I226 2.7.11.1 0004672,0005524,0006468 Kd=17.5nM remove_due_to_license_issue Q8TF76 29601130 802 FQSMGECSQKGPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g36 A 1.46 BS01 EKH A 1 I49 A68 F164 F166 G167 D170 G212 L215 I245 I30 A49 F145 F147 G148 D151 G193 L196 I226 2.7.11.1 0004672,0005524,0006468 Kd=16.3nM remove_due_to_license_issue Q8TF76 29601130 401 FQSMGECSQKGPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g37 A 1.48 BS01 FTU A 1 A509 F607 G608 D611 G653 L656 I686 A38 F136 G137 D140 G182 L185 I215 2.7.11.1 0004672,0005524,0006468 Kd=42.7nM remove_due_to_license_issue Q8TF76 29601130 801 PVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g38 A 1.47 BS01 TBN A 1 A509 F607 G608 D611 G653 L656 I686 A38 F136 G137 D140 G182 L185 I215 2.7.11.1 0004672,0005524,0006468 Kd=239.2nM remove_due_to_license_issue Q8TF76 29601130 800 PVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g39 A 1.45 BS01 5ID A 1 I490 G491 V498 A509 Y605 F607 G608 D611 G653 L656 I686 I20 G21 V28 A39 Y135 F137 G138 D141 G183 L186 I216 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q8TF76 29601130 802 GPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEYEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g3a A 1.43 BS01 5ID A 1 I490 A509 I557 F607 G608 D611 G653 L656 I686 I20 A39 I87 F137 G138 D141 G183 L186 I216 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q8TF76 29601130 805 GPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLETEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK 6g3c A 1.6 BS01 EKT A 1 L551 G552 L579 K581 Q626 E627 F628 V629 G632 K677 S698 L15 G16 L43 K45 Q90 E91 F92 V93 G96 K141 S162 N673 K677 N678 D699 N137 K141 N142 D163 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue O60674 30763067 901 FHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCFCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSL 6g3o A 2.27 BS03 EL8 A 1 G32 H33 P34 D104 H145 H146 G154 F155 D181 H183 F210 L276 Y308 G22 H23 P24 D94 H135 H136 G144 F145 D171 H173 F200 L266 Y298 3.5.1.-,3.5.1.98 0004407 remove_due_to_license_issue Q92769 30122227 1004 GGKKKVCYYYDGDIGNYYYGQGHPMKPHRIRMTHNLLLNYGLYRKMEIYRPHKATAEEMTKYHSDEYIKFLRSIRPDNMSEYSKQMQRFNVGEDCPVFDGLFEFCQLSTGGSVAGAVKLNRQQTDMAVNWAGGLHHAKKSEASGFCYVNDIVLAILELLKYHQRVLYIDIDIHHGDGVEEAFYTTDRVMTVSFHKYGEYFPGTGDLRDIGAGKGKYYAVNFPMRDGIDDESYGQIFKPIISKVMEMYQPSAVVLQCGADSLSGDRLGCFNLTVKGHAKCVEVVKTFNLPLLMLGGGGYTIRNVARCWTYETAVALDCEIPNELPYNDYFEYFGPDFKLHISPSNMTNQNTPEYMEKIKQRLFENLRMLP 6g3q A 1.01 BS02 FO9 A 1 H94 H119 F131 L198 T199 T200 P202 H94 H119 F130 L197 T198 T199 P201 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=57.9nM remove_due_to_license_issue P00918 30344913 302 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6g3v A 1.69 BS02 FO9 A 1 H94 H119 L198 T199 H200 P202 H90 H115 L194 T195 H196 P198 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=922.4nM remove_due_to_license_issue P00915 30344913 302 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6g3y A 2.51 BS01 ELB A 1 G42 F45 N151 I152 K249 M257 H270 Q315 A316 F319 L323 G33 F36 N142 I143 K240 M248 H261 Q306 A307 F310 L314 K249 D268 K240 D259 3.2.2.-,4.2.99.18 0000702,0000978,0003677,0003684,0003824,0005634,0005654,0005739,0006281,0006284,0006289,0006355,0006974,0006979,0008017,0008534,0009314,0009410,0009416,0016363,0016607,0016798,0016829,0019104,0019899,0032355,0032357,0032991,0034039,0034614,0043066,0044029,0045471,0045944,0051593,0071276,0140078,0140097,1901291 remove_due_to_license_issue O08760 30442810 401 HMRHRTLSSSPALWASIPCPRSELRLDLVLASGQSFRWKEQSPAHWSGVLADQVWTLTQTEDQLYCTVYRGDDSQVSRPTLEELETLHKYFQLDVSLAQLYSHWASVDSHFQRVAQKFQGVRLLRQDPTECLFSFICSSNNNIARITGMVERLCQAFGPRLIQLDDVTYHGFPNLHALAGPEAETHLRKLGLGYRARYVRASAKAILEEQGGPAWLQQLRVAPYEEAHKALCTLPGVGAKVADCICLMALDKPQAVPVDVHVWQIAHRDYGWHPKTSQAKGPSPLANKELGNFFRNLWGPYAGWAQAVLFSADLRQ 6g46 A 2.4 BS03 ELH A 1 D164 N201 H202 H295 H296 H323 H325 D157 N194 H195 H288 H289 H316 H318 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D128 D157 Y160 N194 H195 H279 H288 H289 H316 H318 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 Ki=185uM remove_due_to_license_issue P80366 30107365 515 NRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDDS 6g47 A 1.497 BS01 SIA A 1 R316 N318 R124 N126 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue A0MK70 29674446 401 GIQTLWTPPTSNPNCTVYTESDSLLSLCLTKCGAHVLGSVSLTGVAGTMTNMAETSLAIEFTFDDTGKLLHSPLVNNTFSIRQGDSPASNPTYNALAFMPNSTLYARGGSGEPRNNYYVQTYLRGNVQRPITLTVTFNSAATGYSLSFKWTAVVREKFAAPATSFCYITEQ 6g47 C 1.497 BS01 SIA D 1 R316 N318 R118 N120 ? 0007155,0019028,0019058,0019062 remove_due_to_license_issue A0MK70 29674446 2 SGIEGRPGIQTLWTPPTSNPNCTVYTESDSLLSLCLTKCGAHVLGSVSLTGVAGTMTNMAETSLAIEFTFDDTGKLLHSPLVNNTFYNALAFMPNSTLYARGGSGEPRNNYYVQTYLRGNVQRPITLTVTFNSAATGYSLSFKWTAVVREKFAAPATSFCYITEQ 6g4m A 2.63 BS01 DQ5 A 1 Y70 W279 Y334 G335 Y67 W276 Y331 G332 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30125110 601 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g4m A 2.63 BS02 DQ5 A 2 W84 Y121 E199 S286 I287 F288 R289 F290 F330 F331 Y334 W432 H440 Y442 W81 Y118 E196 S283 I284 F285 R286 F287 F327 F328 Y331 W429 H437 Y439 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30125110 602 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g4n A 2.9 BS01 E2W A 1 Y70 W279 Y67 W276 G118 G119 G151 S200 A201 A239 F290 F292 E327 H440 G115 G116 G148 S197 A198 A236 F287 F289 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30125110 603 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6g4y A 2.65 BS01 ELZ A 1 R410 V416 A429 K431 I469 M471 L473 L474 L524 C535 D536 F537 R63 V69 A82 K84 I122 M124 L126 L127 L177 C188 D189 F190 D517 K519 N522 D536 L553 T561 D170 K172 N175 D189 L200 T208 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 29940120 703 PVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQSLLTGDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 6g4z A 2.84 BS01 ELW A 1 R410 V416 I469 M471 L524 C535 D536 F537 R63 V69 I122 M124 L177 C188 D189 F190 D517 K519 N522 D536 L553 T561 D170 K172 N175 D189 L200 T208 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 29940120 701 PVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQSLLTGDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 6g5j A 1.85 BS02 EM8 A 1 L5 P17 Y20 M21 C27 G28 L29 G30 D47 L5 P17 Y20 M21 C27 G28 L29 G30 D47 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0004623,0005509,0006644,0016042,0050482 ic50=0.2uM remove_due_to_license_issue IC50=200nM O15496 30034586 202 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKC 6g5j A 1.85 BS03 EM8 A 2 R15 T16 I18 Y103 F109 R15 T16 I18 Y103 F109 F26 G28 G30 H46 D47 Y50 Y65 D91 F26 G28 G30 H46 D47 Y50 Y65 D91 3.1.1.4 0004623,0005509,0006644,0016042,0050482 ic50=0.2uM remove_due_to_license_issue IC50=200nM O15496 30034586 203 GILELAGTVGCVGPRTPIAYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGPAENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKC 6g5l A 1.21 BS02 EM5 A 1 W4 H66 H91 H117 A129 L197 T198 T199 W2 H64 H89 H115 A127 L195 T196 T197 H66 H91 H93 E104 H117 T198 H64 H89 H91 E102 H115 T196 4.2.1.1 0004089,0008270 Kd=0.019nM remove_due_to_license_issue Kd=24nM O43570 30006175 302 KWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 6g5u B 1.7 BS02 ENN B 1 Q94 H96 H121 V145 L200 T201 V202 Q89 H91 H116 V140 L195 T196 V197 H66 H96 H98 E108 H121 T201 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005515,0005737,0005829,0006730,0008270,0016829,0043209,0043231,0046872 Kd=6.3nM remove_due_to_license_issue Kd=5.7nM Q8N1Q1 30006175 302 SWGYREHNGPIHWKEFFPIADGDQQSPIEIKTKEVKYDSSLRPLSIKYDPSSAKIISNSGHSFNVDFDDTENKSVLRGGPLTGSYRLRQVHLHWGSADDHGSEHIVDGVSYAAELHVVHWNSDKYPSFVEAAHEPDGLAVLGVFLQIGEPNSQLQKITDTLDSIKEKGKQTRFTNFDLLSLLPPSWDYWTYPGSLTVPPLLESVTWIVLKQPINISSQQLAKFRSLLCTAEGEAAAFLVSNHRPPQPLKGRKVRASFH 6g6t A 1.12 BS02 ENN A 1 Q92 H94 H119 L198 T199 T200 Q89 H91 H116 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=0.16nM remove_due_to_license_issue Kd=20nM P00918 30006175 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6g6w A 2.72 BS01 EO5 A 1 F751 M752 P758 W760 I777 K779 D787 Y813 I825 E826 V827 V828 M900 I910 D911 F669 M670 P676 W678 I695 K697 D705 Y731 I743 E744 V745 V746 M805 I815 D816 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue O00329 30351000 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPSAPNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKATVQPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDESVSLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEDCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHSEEEQLQLREILERELYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSGGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWK 6g6y A 1.8 BS02 EOK A 1 E116 G117 E118 R119 W127 A133 I136 P137 Y211 E95 G96 E97 R98 W106 A112 I115 P116 Y186 ? 0003777,0005524,0007018,0008017 Kd=220nM remove_due_to_license_issue P52732 30031975 403 KNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 6g6z A 2.8 BS02 EOK A 1 E118 R119 A133 Y211 L214 E101 R102 A116 Y194 L197 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue P52732 30031975 403 GKNIQVVVRCRPFNLAERSAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPEVN 6g7a A 1.42 BS02 EOQ A 1 H91 H117 V119 S130 L197 T198 T199 W208 H90 H116 V118 S129 L196 T197 T198 W207 H66 H91 H93 E104 H117 T198 H65 H90 H92 E103 H116 T197 4.2.1.1 0004089,0008270 Kd=0.041nM remove_due_to_license_issue Kd=0.041000nM O43570 30006175 303 SKWTYFGPDGENSWSKKYPSCGGLLQSPIDLHSDILQYDASLTPLEFQGYNLSANKQFLLTNNGHSVKLNLPSDMHIQGLQSRYSATQLHLHWGNPNDPHGSEHTVSGQHFAAELHIVHYNSDLYPDASTASNKSEGLAVLAVLIEMGSFNPSYDKIFSHLQHVKYKGQEAFVPGFNIEELLPERTAEYYRYRGSLTTPPCNPTVLWTVFRNPVQISQEQLLALETALYCTHMDDPSPREMINNFRQVQKFDERLVYTSFSQ 6g7f H 2.7 BS01 EPW H 1 T1 K33 A46 G47 S129 T1 K33 A46 G47 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 30165344 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6g7f H 2.7 BS02 EPW N 1 H114 S118 H114 S118 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 30165344 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6g7f N 2.7 BS01 EPW N 1 T1 T20 T21 K33 S46 G47 S48 A49 T1 T20 T21 K33 S46 G47 S48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0000502,0004175,0004298,0005515,0005634,0005737,0005829,0005839,0006508,0010499,0019774,0034515,0043161,0051603 remove_due_to_license_issue P38624 30165344 201 TSIMAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDKIWCCRSGSAADTQAIADIVQYHLELYTSQYGTPSTETAASVFKELCYENKDNLTAGIIVAGYDDKNKGEVYTIPLGGSVHKLPYAIAGSGSTFIYGYCDKNFRENMSKEETVDFIKHSLSQAIKWDGSSGGVIRMVVLTAAGVERLIFYPDEYEQL 6g8m H 2.7 BS01 EQE H 1 T1 K33 A46 G47 G128 S129 T1 K33 A46 G47 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 30165344 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6g8m N 2.7 BS01 EQE N 1 T1 T20 T21 K33 S46 G47 A49 T1 T20 T21 K33 S46 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0000502,0004175,0004298,0005515,0005634,0005737,0005829,0005839,0006508,0010499,0019774,0034515,0043161,0051603 remove_due_to_license_issue P38624 30165344 201 TSIMAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDKIWCCRSGSAADTQAIADIVQYHLELYTSQYGTPSTETAASVFKELCYENKDNLTAGIIVAGYDDKNKGEVYTIPLGGSVHKLPYAIAGSGSTFIYGYCDKNFRENMSKEETVDFIKHSLSQAIKWDGSSGGVIRMVVLTAAGVERLIFYPDEYEQL 6g8n H 3.0 BS01 EQB H 1 T1 K33 G45 A46 G47 S129 T1 K33 G45 A46 G47 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 30165344 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6g8n H 3.0 BS02 EQB N 1 H114 H116 H114 H116 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 30165344 201 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6g8n N 3.0 BS01 EQB N 1 T1 T20 T21 K33 S46 G47 T1 T20 T21 K33 S46 G47 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0000502,0004175,0004298,0005515,0005634,0005737,0005829,0005839,0006508,0010499,0019774,0034515,0043161,0051603 remove_due_to_license_issue P38624 30165344 201 TSIMAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDKIWCCRSGSAADTQAIADIVQYHLELYTSQYGTPSTETAASVFKELCYENKDNLTAGIIVAGYDDKNKGEVYTIPLGGSVHKLPYAIAGSGSTFIYGYCDKNFRENMSKEETVDFIKHSLSQAIKWDGSSGGVIRMVVLTAAGVERLIFYPDEYEQL 6g91 A 1.8 BS01 EQW A 1 A52 Q105 M108 T110 K114 L156 A45 Q98 M101 T103 K107 L149 D149 K151 N154 D167 T190 D142 K144 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=3200nM remove_due_to_license_issue IC50=3200nM P28482 29775310 403 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFLDDLPKEKLKELIFEETARFQPG 6g92 A 1.99 BS01 ERZ A 1 A52 M108 E109 K114 L156 A45 M101 E102 K107 L149 D149 K151 N154 D167 T190 D142 K144 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=76000nM remove_due_to_license_issue IC50=76000nM P28482 29775310 404 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFDDLPKEKLKELIFEETARFQPG 6g93 A 1.67 BS01 EU2 A 1 A52 K54 Q105 M108 T110 K114 L156 A42 K44 Q95 M98 T100 K104 L146 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=11nM remove_due_to_license_issue IC50=11.0nM P28482 29775310 406 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFLDDLPKEKLKELIFEETARFQPG 6g97 A 1.9 BS01 EQZ A 1 G37 V39 A52 K54 Q105 M108 T110 K114 L156 D167 G27 V29 A42 K44 Q95 M98 T100 K104 L146 D157 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=4.2nM remove_due_to_license_issue IC50=3.90nM P28482 29775310 407 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQPG 6g98 A 2.47 BS02 ER5 A 1 R60 N62 H64 Q67 Q92 H94 H96 V121 V131 L198 T199 T200 R46 N48 H50 Q53 Q74 H76 H78 V103 V112 L181 T182 T183 H64 H94 H96 E106 H119 T199 H50 H76 H78 E88 H101 T182 4.2.1.1 0004089,0008270 Kd=0.16nM remove_due_to_license_issue Q16790 29928486 302 RVSPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 6g99 B -1.00 BS01 rna A 0 S418 G419 Q420 Q421 R422 D425 N435 M436 N437 F438 S439 W440 R441 N445 S5 G6 Q7 Q8 R9 D12 N22 M23 N24 F25 S26 W27 R28 N32 ? 0003723,0006355 remove_due_to_license_issue P35637 30581145 1 ~ 5 GPLGSGQQRAGDWKCPNPTCENMNFSWRNECNQCKAPKPDG 6g9a A 1.91 BS01 ESQ A 1 E33 G37 V39 K54 Q105 M108 E109 T110 K114 L156 C166 D167 E26 G30 V32 K47 Q98 M101 E102 T103 K107 L149 C159 D160 D149 K151 N154 D167 T190 D142 K144 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=21nM remove_due_to_license_issue IC50=12.0nM P28482 29775310 404 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFLPKEKLKELIFEETARFQPG 6g9b A 2.26 BS01 IXX A 1 I38 L43 L184 L186 I8 L13 L154 L156 ? Kd=584uM remove_due_to_license_issue Kd=584000nM Q05320 29741894 609 RSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQASGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTWAFWETLSFTVVSAAAAAAA 6g9b B 2.26 BS01 IXX B 1 Y517 Q521 Y16 Q20 ? Kd=584uM remove_due_to_license_issue Kd=584000nM Q05320 29741894 705 EAIVNAQPKCNPNLHYWTTQGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFV 6g9d A 1.8 BS01 ER8 A 1 Y36 V39 A52 K54 E71 Q105 M108 K114 L156 D167 Y29 V32 A45 K47 E64 Q98 M101 K107 L149 D160 D149 K151 N154 D167 T190 D142 K144 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=4.3nM remove_due_to_license_issue IC50=9.00nM P28482 29775310 406 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFELDDLPKEKLKELIFEETARFQPG 6g9f A 2.35 BS01 NXL A 1 S330 W370 S387 D389 S545 G546 T547 S274 W314 S331 D333 S489 G490 T491 3.4.16.4 0008658,0009002,0009252,0016020 remove_due_to_license_issue P0AD65 30995398 1330 NRIKLVPIAPSRGIIYDRNGIPLALNRTIYQIEMMPEKVDNVQQTLDALRSVVDLTDDDIAAFRKERARSHRFTSIPVKTNLTEVQVARFAVNQYRFPGVEVKGYKRRYYPYGSALTHVIGYVSKINDKDVERLNNDGKLANYAATHDIGKLGIERYYEDVLHGQTGYEEVEVNNRGRVIRQLKEVPPQAGHDIYLTLDLKLQQYIETLLAGSRAAVVVTDPRTGGVLALVSTPSYDPNLFVDGISSKDYSALLNDPNTPLVNRATQGVYPPASTVKPYVAVSALSAGVITRNTTLFDPGWWQLPGSEKRYRDWKKWGHGRLNVTRSLEESADTFFYQVAYDMGIDRLSEWMGKFGYGHYTGIDLAEERSGNMPTREWKQKRFKKPWYQGDTIPVGIGQGYWTATPIQMSKALMILINDGIVKVPHLLMSTAEDGKQVPWVQPHEPPVGDIHSGYWELAKDGMYGVANRPNGTAHKYFASAPYKIAAKSGTAQLRDHKLMTAFAPYNNPQVAVAMILENGGAGPAVGTLMRQILDHIML 6g9h A 1.73 BS01 ERW A 1 I31 Y36 A52 K54 E71 Q105 M108 T110 K114 L156 D167 I21 Y26 A42 K44 E61 Q95 M98 T100 K104 L146 D157 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=4nM remove_due_to_license_issue IC50=3.00nM P28482 29775310 405 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFLDDLPKEKLKELIFEETARFQPG 6g9j A 1.98 BS01 ERK A 1 Y36 V39 A52 K54 I56 Y64 R67 T68 Q105 M108 T110 K114 L156 C166 D167 Y29 V32 A45 K47 I49 Y57 R60 T61 Q98 M101 T103 K107 L149 C159 D160 D149 K151 N154 D167 T190 D142 K144 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=4.1nM remove_due_to_license_issue IC50=4.30nM P28482 29775310 403 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPG 6g9k A 1.94 BS01 ESK A 1 Y36 V39 A52 K54 Y64 R67 T68 Q105 M108 K114 D167 Y26 V29 A42 K44 Y54 R57 T58 Q95 M98 K104 D157 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 remove_due_to_license_issue P28482 29775310 404 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQPG 6g9m A 1.86 BS01 ESW A 1 G34 G37 V39 A52 K54 Q105 M108 T110 K114 D167 G24 G27 V29 A42 K44 Q95 M98 T100 K104 D157 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=7.9nM remove_due_to_license_issue IC50=7.90nM P28482 29775310 404 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFELDDLPKEKLKELIFEETARFQP 6g9n A 1.76 BS01 ESN A 1 I31 Y36 V39 A52 K54 Y64 R67 T68 Q105 M108 T110 K114 D167 G169 I21 Y26 V29 A42 K44 Y54 R57 T58 Q95 M98 T100 K104 D157 G159 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=3nM remove_due_to_license_issue IC50=3.00nM P28482 29775310 407 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKMELDDLPKEKLKELIFEETARFQPG 6g9s A 2.001 BS01 ET5 A 1 S330 W370 S387 D389 S545 G546 T547 S274 W314 S331 D333 S489 G490 T491 3.4.16.4 0004180,0005515,0005886,0006508,0008360,0008658,0009002,0009252,0016020,0030288,0046677,0071555,0071972 remove_due_to_license_issue P0AD65 30995398 701 NRIKLVPIAPSRGIIYDRNGIPLALNRTIYQIEMMPEKVDNVQQTLDALRSVVDLTDDDIAAFRKERARSHRFTSIPVKTNLTEVQVARFAVNQYRFPGVEVKGYKRRYYPYGSALTHVIGYVSKINDKDVERLNNDGKLANYAATHDIGKLGIERYYEDVLHGQTGYEEVEVNNRGRVIRQLKEVPPQAGHDIYLTLDLKLQQYIETLLAGSRAAVVVTDPRTGGVLALVSTPSYDPNLFVDGISSKDYSALLNDPNTPLVNRATQGVYPPASTVKPYVAVSALSAGVITRNTTLFDPGWWQLPGSEKRYRDWKKWGHGRLNVTRSLEESADTFFYQVAYDMGIDRLSEWMGKFGYGHYTGIDLAEERSGNMPTREWKQKRFKKPWYQGDTIPVGIGQGYWTATPIQMSKALMILINDGIVKVPHLLMSTAEDGKQVPWVQPHEPPVGDIHSGYWELAKDGMYGVANRPNGTAHKYFASAPYKIAAKSGTAQRDHKLMTAFAPYNNPQVAVAMILENGGAGPAVGTLMRQILDHIML 6g9u A 1.75 BS02 ETK A 1 R60 N62 H64 Q92 H94 H96 V121 L198 T199 T200 R46 N48 H50 Q74 H76 H78 V103 L181 T182 T183 H64 H94 H96 E106 H119 T199 H50 H76 H78 E88 H101 T182 4.2.1.1 0004089,0008270 Kd=0.2nM remove_due_to_license_issue Q16790 29928486 302 RVSPACAGRFQSPVDIRPQLAAFSPALRPLELLGFQLPPLPELRLRNNGHSVQLTLPPGLEMALGPGREYRALQLHLHWGAAGRPGSEHTVEGHRFPAEIHVVHLSTAFARVDEALGRPGGLAVLAAFLEEGPEENSAYEQLLSRLEEIAEEGSETQVPGLDISALLPSDFSRYFQYEGSLTTPPCAQGVIWTVFNQTVMLSAKQLHTLSDTLWGPGDSRLQLNFRATQPLNGRVIEASFP 6g9x A 2.3 BS01 JKE A 1 Y119 L145 R280 Y331 F335 C362 Y110 L136 R256 Y307 F311 C338 ? 0005886,0015293,0022857,0055085 remove_due_to_license_issue A0LNN5 31201333 507 TMPRWVPLLLGLLGSTTCGMLLYAWSVFIKPLNAESRAEIAMAFAICCLIFGLMTFPAGRLSDKMGPRKVVMTGGVLLAIGFILSGFIQSKYQLYITYGVIAGFGGGMIYLPPIATAPKWWPDRRALATGFAVVGLGLGSFLMGPLATYIIEWRYVFWYCGVAMGIMALIAGAFLEPPPAGWKPAGAAPKVTRDWTYEEAKGDTKFWLLYLAYFCGSFAGLMVIGHLAGFGRDAGLTAMAAAGAVSSLAFSNAATRILSGWFVDKIGIRVYFAALFALQTAAMIAIFQLGGSVVGLSIVAIVIGWNYGAMFTLFPATCLQFYGPTAQGSNYGLLFTACGLAGFAGPWVGGWLKDTTGTYYLPFLCAAALCALGTAIVFMTKPPEKKHALELEVLFQ 6gat A -1.00 BS01 dna B 0 R24 R59 R24 R59 ? 0003700,0006355,0006357,0008270,0043565 remove_due_to_license_issue P17429 9533884 101 ~ 113 MKNGEQNGPTTCTNCFTQTTPVWRRNPEGQPLCNACGLFLKLHGVVRPLSLKTDVIKKRNRNSANS 6gat A -1.00 BS02 dna C 0 P21 N34 F39 R47 I56 R59 R61 P21 N34 F39 R47 I56 R59 R61 ? 0003700,0006355,0006357,0008270,0043565 remove_due_to_license_issue P17429 9533884 114 ~ 126 MKNGEQNGPTTCTNCFTQTTPVWRRNPEGQPLCNACGLFLKLHGVVRPLSLKTDVIKKRNRNSANS 6gbm B -1.00 BS01 rna A 0 N285 T286 F288 K312 K315 K316 Y325 T326 R328 K334 T338 A369 T370 R371 R372 A373 N10 T11 F13 K37 K40 K41 Y50 T51 R53 K59 T63 A94 T95 R96 R97 A98 ? 0003676,0003723,0006355 remove_due_to_license_issue P35637 30581145 1 ~ 23 GSHMDNSDNNTIFVQGLGENVTIESVADYFKQIGIIKTNKKTGQPMINLYTDRETGKLKGEATVSFDDPPSAKAAIDWFDGKEFSGNPIKVSFATRRADFNR 6gbw H 1.45 BS03 EU5 H 1 H57 Y60A W60D L99 A190 S195 V213 S214 W215 G216 E217 G219 F227 H43 Y47 W50 L96 A193 S198 V218 S219 W220 G221 E222 G223 F232 H57 D102 E192 G193 D194 S195 G196 H43 D99 E195 G196 D197 S198 G199 3.4.21.5 0004252,0005509,0006508,0007596 Ki=3.51nM remove_due_to_license_issue Ki=3.5nM P00734 31633354 306 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 6gbx A 1.72 BS02 S77 A 1 K144 D159 E201 W207 D248 Q304 D305 W329 H330 K111 D126 E168 W174 D215 Q271 D272 W296 H297 2.3.2.5 0005515,0005576,0008270,0016603,0016746,0017186,0035580,0036211,0046872,0070062,1904724,1904813 Ki=0.02uM remove_due_to_license_issue IC50=17nM Q16769 30132075 403 SAWPEEKNYHQPAILNSSALRQIAEGTSISEMWQNDLQPLLIERYPGSPGSYAARQHIMQRIQRLQADWVLEIDTFLSQTPEGERSFSNIISTLNPTAKRHLVLACHYDSKYFSHWNNRVFVGATDSAVPCAMMLELARALDKKLLSLKTVSDSKPDLSLQLIFFDGEEAFLHWSPQDSLYGSRHLAAKMASTPHPPGARGTSQLHGMDLLVLLDLIGAPNPTFPNFFPNSARWFERLQAIEHELHELGLLKDHSLEGRYFQNYSYGGVIQDDHIPFLRRGVPVLHLIPSPFPEVWHTMDDNEENLDESTIDNLNKILQVFVLEYLHL 6gc5 A 1.9 BS01 rna E 0 F247 Y249 Q253 I276 R277 K285 F289 Q316 K320 T321 F5 Y7 Q11 I34 R35 K43 F47 Q74 K78 T79 ? 0003676,0003723 remove_due_to_license_issue Q15717 30718402 1 ~ 5 GWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKT 6gc5 B 1.9 BS01 rna F 0 F247 Y249 K274 F289 Q316 K320 T321 F5 Y7 K32 F43 Q70 K74 T75 ? 0003676,0003723 remove_due_to_license_issue Q15717 30718402 2 ~ 4 GWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTN 6gc5 C 1.9 BS01 rna G 0 F247 Y249 K274 K285 F289 Q316 K320 T321 F5 Y7 K32 K43 F47 Q74 K78 T79 ? 0003676,0003723 remove_due_to_license_issue Q15717 30718402 1 ~ 4 GWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKT 6gc5 D 1.9 BS01 rna H 0 F247 Y249 I276 F289 Q316 K320 T321 F6 Y8 I35 F44 Q71 K75 T76 ? 0003676,0003723 remove_due_to_license_issue Q15717 30718402 2 ~ 4 SGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTN 6gch G 2.1 BS02 APF G 1 S190 C191 M192 G193 S195 S214 G216 S217 C220 S40 C41 M42 G43 S45 S64 G66 S67 C70 G193 S195 G196 G43 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 2271520 246 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 6gcl A 1.95 BS02 EUE A 1 S95 F97 Y174 P210 S94 F96 Y156 P192 R14 D161 Y174 K178 R13 D143 Y156 K160 ? 0000166,0016491,0047040 ic50=34.2uM remove_due_to_license_issue O76290 30908048 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 6gcl D 1.95 BS02 EUE D 1 S95 F97 Y174 P210 S94 F96 Y155 P191 R14 D161 Y174 K178 R13 D142 Y155 K159 ? 0000166,0016491,0047040 ic50=34.2uM remove_due_to_license_issue O76290 30908048 302 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 6gcr A 2.3 BS01 EUW A 1 C427 I428 G429 A452 L501 C502 G505 E506 L553 D564 L567 C15 I16 G17 A40 L89 C90 G93 E94 L141 D152 L155 D546 A548 R550 N551 D564 D134 A136 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q00944 29897729 701 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEK 6gcw A 2.0 BS01 EUQ A 1 I428 V436 A452 K454 L501 C502 G505 E506 L553 I15 V23 A39 K41 L88 C89 G92 E93 L140 D546 A548 R550 N551 D564 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4.7nM remove_due_to_license_issue Q00944 29897729 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKL 6gcw B 2.0 BS01 EUQ B 1 I428 A452 M499 L501 C502 G505 E506 L553 G563 D564 L567 I15 A39 M86 L88 C89 G92 E93 L140 G150 D151 L154 D546 A548 R550 N551 D564 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=4.7nM remove_due_to_license_issue Q00944 29897729 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ 6gcx A 1.553 BS01 EUW A 1 R426 L501 C502 T503 G505 L553 L567 R14 L87 C88 T89 G91 L139 L153 D546 A548 R550 N551 D564 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM remove_due_to_license_issue Q00944 29897729 701 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ 6gd3 B 1.35 BS01 rna P 0 F247 K274 I276 F279 F287 F289 K320 T321 F8 K35 I37 F40 F48 F50 K81 T82 ? 0003676,0003723 remove_due_to_license_issue Q15717 30418581 1 ~ 6 GAMGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTN 6gd3 C 1.35 BS01 rna P 0 F247 Y249 K274 K285 F287 F289 K313 Q316 K320 T321 K323 F8 Y10 K35 K46 F48 F50 K74 Q77 K81 T82 K84 ? 0003676,0003723 remove_due_to_license_issue Q15717 30418581 1 ~ 6 GAMGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNK 6gdg A 4.11 BS01 NEC A 1 T88 Q89 M177 W246 L249 N253 M270 I274 H278 T82 Q83 M154 W211 L214 N218 M235 I239 H243 ? 0001609,0001973,0004930,0005515,0005737,0005829,0007186,0015035,0015036,0016020,0030337,0045454 remove_due_to_license_issue P0AA25,P29274 29726815 400 AVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTF 6gdy A 2.04 BS02 AKG A 1 Y131 F133 T184 H187 N197 K204 H273 V275 Y131 F133 T184 H187 N197 K204 H273 V275 1.14.11.- Kd=3.5uM remove_due_to_license_issue Q6NYC1 31147442 402 MNHKSKKRIREAKRSARPELKDSLDWTRHNYYESFSLSPAAVADNVERADALQLSVEEFVERYERPYKPVVLLNAQEGWSAQEKWTLERLKRKYRNQKFKCGEDNDGYSVKMKMKYYIEYMESTRDDSPLYIFDSSYGEHPKRRKLLEDYKVPKFFTDDLFQYAGEKRRPPYRWFVMGPPRSGTGIHIDPLGTSAWNALVQGHKRWCLFPTSTPRELIKVTRDEGGNQQDEAITWFNVIYPRTQLPTWPPEFKPLEILQKPGETVFVPGGWWHVVLNLDTTIAITQNFASSTNFPVVWHKTVRGRPKLSRKWYRILKQEHPELAVLADSVDLQ 6ge0 A 1.82 BS01 EVQ A 1 Y36 V39 A52 K54 I56 Y64 R67 T68 Q105 M108 T110 K114 L156 D167 Y26 V29 A42 K44 I46 Y54 R57 T58 Q95 M98 T100 K104 L146 D157 D149 K151 N154 D167 T190 D139 K141 N144 D157 T180 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=2.1nM remove_due_to_license_issue IC50=2.10nM P28482 29775310 406 PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDLDDLPKEKLKELIFEETARFQPG 6ge7 A 2.3 BS01 EW8 A 1 L46 L54 K69 F105 M107 L46 L54 K69 F105 M107 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=0.867uM remove_due_to_license_issue P02754 29879410 201 LIVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 6gev A 1.54 BS02 EWN A 1 N770 Q776 M807 L810 S811 L814 F829 M845 F941 C942 T945 N36 Q42 M73 L76 S77 L80 F95 M111 F207 C208 T211 ? Ki=1.9nM remove_due_to_license_issue IC50=63nM, Ki=2.0nM P08235 30596500 1104 YFSPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 6gf3 A 2.4 BS03 EX5 B 1 T179 A180 T179 A180 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 30006510 503 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGV 6gf3 B 2.4 BS02 EX5 B 1 C241 A250 L255 N258 M259 A316 I318 N349 N350 K352 C238 A247 L252 N255 M256 A307 I309 N340 N341 K343 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Q6B856 30006510 503 REIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 6gf9 A 2.1 BS01 X90 A 1 L46 L54 I56 V92 F105 M107 L45 L53 I55 V91 F104 M106 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=0.000000064M remove_due_to_license_issue P02754 29879410 201 IVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 6gfs A 2.0 BS01 F15 A 1 V92 F105 M107 V92 F105 M107 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=0.000000064M remove_due_to_license_issue P02754 29879410 201 LIVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 6gfy C 2.7 BS01 EXH C 1 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? remove_due_to_license_issue P40337 29949369 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 6gfz C 2.3 BS01 EXE C 1 P86 W88 Y98 P99 I109 H110 S111 Y112 H115 W117 P25 W27 Y37 P38 I48 H49 S50 Y51 H54 W56 ? Kd=3080nM remove_due_to_license_issue P40337 29949369 301 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLT 6gg3 A 3.72 BS01 ALA A 1 N44 N70 H464 I469 F470 N32 N58 H452 I457 F458 R73 R120 K270 T328 R61 R108 K258 T316 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 29748232 602 IQTQQLHAAMADTFLEHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 6gg4 A 2.46 BS01 PHE A 1 R43 N44 N70 H464 I469 F470 R21 N22 N48 H442 I447 F448 R73 R120 K270 T328 R51 R98 K248 T306 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 29748232 603 ADTFLEHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 6gg5 A 3.2 BS01 TRP A 1 R43 N44 N70 R106 H464 G468 I469 F470 F502 R21 N22 N48 R84 H442 G446 I447 F448 F480 R73 R120 K270 T328 R51 R98 K248 T306 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 29748232 603 ADTFLEHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 6gg8 A 1.8 BS02 EY8 A 1 N770 A773 Q776 M807 S810 S811 L814 F829 M845 L938 F941 C942 T945 N34 A37 Q40 M71 S74 S75 L78 F93 M109 L196 F199 C200 T203 ? Ki=0.79nM remove_due_to_license_issue IC50=25nM, Ki=0.794328nM, EC50=0.050119nM P08235 30596500 1102 SPVMVLENIEPEIVYAGYDSSKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLSSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHRK 6gga A 1.55 BS01 EY2 A 1 L145 V147 T150 C220 E221 P222 P223 D228 C229 L50 V52 T55 C125 E126 P127 P128 D133 C134 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 31633398 401 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 6ggb A 1.32 BS02 EXQ A 1 L145 V147 T150 P151 C220 E221 P222 P223 D228 T230 L51 V53 T56 P57 C126 E127 P128 P129 D134 T136 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 31633398 402 SSVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 6ggd A 1.40001 BS02 EYB A 1 L145 V147 T150 P151 C220 E221 P222 P223 D228 L50 V52 T55 P56 C125 E126 P127 P128 D133 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 31633398 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 6gge A 1.25001 BS02 EYE A 1 L145 V147 T150 C220 E221 P222 P223 D228 C229 L50 V52 T55 C125 E126 P127 P128 D133 C134 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 31633398 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRKK 6ggf A 1.32 BS02 EXQ A 1 L145 V147 T150 C220 E221 P222 P223 D228 L50 V52 T55 C125 E126 P127 P128 D133 ? 0000976,0003677,0003700,0005634,0006355,0006915 remove_due_to_license_issue P04637 31633398 402 SVPSQKTYQGSYGFRLGFLHSGTAKSVTCTYSPALNKLFCQLAKTCPVQLWVDSTPPPGTRVRAMAIYKQSQHMTEVVRRCPHHERCSDSDGLAPPQHLIRVEGNLRAEYLDDRNTFRHSVVVPCEPPEVGSDCTTIHYNYMCYSSCMGGMNRRPILTIITLEDSSGNLLGRDSFEVRVCACPGRDRRTEEENLRK 6ggg A 1.71 BS02 EYN A 1 L766 N770 L772 A773 Q776 M807 S811 L814 F829 L848 M852 L938 F941 C942 T945 L16 N20 L22 A23 Q26 M57 S61 L64 F79 L98 M102 L188 F191 C192 T195 ? Ki=0.63nM remove_due_to_license_issue IC50=20nM, Ki=0.630957nM P08235 30596500 1102 IVYAGYDKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQITLIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQGMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYIKELRKMVTKSPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESHALKVEFPAMLVEIISDQLPKVESGNAKPLYFHR 6ggn A 2.0 BS01 EYH A 1 L54 G58 I61 M62 Y67 Q72 F86 V93 H96 I99 Y100 L37 G41 I44 M45 Y50 Q55 F69 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 ic50=0.08nM remove_due_to_license_issue IC50=0.17nM Q00987 30217415 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 6ggv A 2.69 BS01 ARG A 1 S35 F38 F76 S93 G94 M95 T96 R101 Q142 T145 T146 D183 Y209 S15 F18 F56 S73 G74 M75 T76 R81 Q122 T125 T126 D163 Y189 ? 0015276,0016020 remove_due_to_license_issue Q9WZ62 29860047 301 IDEIKSRGYLLVGLSADFPPFEFVDENGNIVGFDVDLAKEIARRLGVELKIVDMTFDGLIPSLLTKKIDVIISGMTITEERKKVVAFSDPYFDAGQVIVVRKDSDFRPKTYEDLVGKTVAVQIGTTGDIEVSKYDGIKVVRFDKFTDAFLELKRGRADAVVLDSATARAFVAKNPDLVISSGVLSSEQYGIAVRKEDTDLLEFINSVLRELK 6gh9 A 2.09 BS02 MIX A 1 Y855 G856 H862 Y273 G274 H280 3.4.19.12 0004843,0016579 remove_due_to_license_issue Q9Y4E8 30228188 1003 MEQPGLCGLSNLGNTCFMNSAIQCLSNTPPLTEYFLNDKYQEELNFDNPLGMRGEIAKSYAELIKQMWSGKFSYVTPRAFKTQVGRFAPQQELLAFLLDGLHEDLNRIRKKPYIQLKDADGRPDKVVAEEAWENHLKRNDSIIVDIFHGLFKSTLVCPECAKISVTFDPFCYLTLPLASKVKLKDCIELFTTKEKLGAEDPWYCPNCKEHQQATKKLDLWSLPPVLVVHLKRFSDKLDTLVDFPINDLDMSEFLINPNAGPCRYNLIAVSNHYGGMGGGHYTAFAKNKDDGKWYYFDDSSVSTASEDQIVSKAAYVLFYQRQDTFSGTGFF 6ghh A 1.9 BS01 TDA A 1 I84 F105 M107 I84 F105 M107 ? 0005515,0005576,0019841,0036041,0036094,0042802 Kd=0.000000064M remove_due_to_license_issue P02754 29879410 201 LIVTQTMKGLDIQKVAGTWYSLAMAASDISLLDAQSAPLRVYVEELKPTPEGDLEILLQKWENGECAQKKIIAEKTKIPAVFKIDALNENKVLVLDTDYKKYLLFCMENSAEPEQSLACQCLVRTPEVDDEALEKFDKALKALPMHIRLSFNPTQLEEQCHI 6ghp A 1.95 BS02 EZ5 A 1 E39 N42 L43 V46 F119 K122 D215 L218 E44 N47 L48 V51 F115 K118 D208 L211 ? 0000122,0001836,0003334,0005515,0005576,0005615,0005634,0005737,0005829,0006469,0006611,0007165,0008104,0008426,0008630,0010482,0010839,0019901,0022407,0030216,0030307,0031424,0032880,0042802,0043588,0043616,0045296,0045606,0045785,0045824,0046827,0050815,0051219,0051726,0061436,0070062,0072089,0140311,0141156,1903077,1903829,2000647 remove_due_to_license_issue P31947 30025189 301 GAMGSMERASLIQKAKLAEQAERYEDMAAFMKGAVEKGEELSCEERNLLSVAYKNVVGGQRAAWRVLSSIEQKSNGPEVREYREKVETELQGVCDTVLGLLDSHLIKGDAESRVFYLKMKGDYYRYLAEVATKKRIIDSARSAYQEAMDISKKEMPPTNPIRLGLALNFSVFHYEIANSPEEAISLAKTTFDEAMADLHTLSEDSYKDSTLIMQLLRDNLTLWT 6ghv A 2.1 BS01 EZ8 A 1 F313 E347 N349 G352 E354 E358 N365 D367 K368 F61 E95 N97 G100 E102 E106 N113 D115 K116 ? Kd=52uM remove_due_to_license_issue Q9NNX6 31469191 1001 CHPCPWEWTFFQGNCYFMSNSQRNWHDSITACKEVGAQLVVIKSAEEQNFLQLQSSRSNRFTWMGLSDLNQEGTWQWVDGSPLLPSFKQYWNRGEPNNVGEEDCAEFSGNGWNDDKCNLAKFWICKKSAASC 6ghv A 2.1 BS04 EZ8 B 1 Q264 G265 Q12 G13 ? Kd=52uM remove_due_to_license_issue Q9NNX6 31469191 1001 CHPCPWEWTFFQGNCYFMSNSQRNWHDSITACKEVGAQLVVIKSAEEQNFLQLQSSRSNRFTWMGLSDLNQEGTWQWVDGSPLLPSFKQYWNRGEPNNVGEEDCAEFSGNGWNDDKCNLAKFWICKKSAASC 6ghv A 2.1 BS05 EZ8 D 1 N272 R309 S310 N311 R312 F374 N20 R57 S58 N59 R60 F122 ? Kd=52uM remove_due_to_license_issue Q9NNX6 31469191 502 CHPCPWEWTFFQGNCYFMSNSQRNWHDSITACKEVGAQLVVIKSAEEQNFLQLQSSRSNRFTWMGLSDLNQEGTWQWVDGSPLLPSFKQYWNRGEPNNVGEEDCAEFSGNGWNDDKCNLAKFWICKKSAASC 6gi6 A 1.98 BS01 EZB A 1 V222 K235 L263 T283 Y285 H286 L343 A353 V21 K34 L62 T82 Y84 H85 L142 A152 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.194uM remove_due_to_license_issue IC50=194nM Q04771 30085668 501 RTVARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSRHSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKID 6gih A 1.96 BS01 EZN A 1 Q36 Y39 L41 V67 I69 D103 S106 T108 A110 Q34 Y37 L39 V65 I67 D101 S104 T106 A108 D156 K158 N161 D175 S194 D151 K153 N156 D170 S189 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue IC50=44000nM P68400 29759799 403 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK 6gin A 2.2 BS01 IR2 A 1 V214 A233 K235 L263 Y285 H286 G289 L343 A353 V11 A30 K32 L60 Y82 H83 G86 L140 A150 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.032uM remove_due_to_license_issue IC50=32nM, Kd=330nM Q04771 30085668 501 VARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSRHSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKID 6gip A 2.17 BS01 EUN A 1 V222 A233 K235 L263 L281 T283 Y285 H286 G289 L343 V19 A30 K32 L60 L78 T80 Y82 H83 G86 L140 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 ic50=0.042uM remove_due_to_license_issue Kd=640nM, IC50=42nM Q04771 30085668 501 VARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSRHSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKID 6gis A 2.82 BS01 dna D 0 D21 K77 R149 H153 K217 D21 K77 R149 H153 K211 ? 0000122,0000307,0000701,0000781,0000785,0001673,0003677,0003682,0003684,0005515,0005634,0005652,0005654,0005657,0005813,0006260,0006272,0006275,0006281,0006287,0006298,0006979,0007507,0016604,0019899,0019985,0030331,0030337,0030855,0030894,0030971,0031297,0032077,0032139,0032355,0032405,0033993,0034644,0035035,0042802,0043596,0043626,0044849,0044877,0045739,0045740,0046686,0070062,0070182,0070301,0070557,0071466,0071548,0097421,1900264,1902065,1902990 remove_due_to_license_issue P12004 28071730 1 ~ 10 MFEARLVQGSILKKVLEALKDLINEACWDISSSGVNLQSMDSSHVSLVQLTLRSEGFDTYRCDRNLAMGVNLTSMSKILKCAGNEDIITLRAEDNADTLALVFEAPNQEKVSDYEMKLMDLDVEQLGIPEQEYSCVVKMPSGEFARICRDLSHIGDAVVISCAKDGVKFSASGELGNGNIKLSQTEEAVTIEMNEPVQLTFALRYLNFFTKATPLSSTVTLSMSADVPLVVEYKIADMGHLKYYLAPK 6giu A 1.39 BS03 L69 A 1 E70 D90 D93 G94 T95 E162 G194 A196 E213 W219 D220 E68 D88 D91 G92 T93 E160 G192 A194 E211 W217 D218 E70 D90 I92 D93 T95 D220 E68 D88 I90 D91 T93 D218 3.1.3.25,3.1.3.94 0000287,0005515,0005737,0005829,0006020,0006021,0006661,0006796,0007165,0008934,0016787,0030145,0031403,0042802,0042803,0046854,0046872,0052834 remove_due_to_license_issue P29218 30289407 304 DPWQECMDYAVTLARQAGEVVCEAIKNEMNVMLKSSPVDLVTATDQKVEKMLISSIKEKYPSHSFIGEESVAAGEKSILTDNPTWIIDPIDGTTNFVHRFPFVAVSIGFAVNKKIEFGVVYSCVEGKMYTARKGKGAFCNGQKLQVSQQEDITKSLLVTELGSSRTPETVRMVLSNMEKLFCIPVHGIRSVGTAAVNMCLVATGGADAYYEMGIHCWDVAGAGIIVTEAGGVLMDVTGGPFDLMSRRVIAANNRILAERIAKEIQVIPLQRDDED 6giu B 1.39 BS03 L69 B 1 E70 D90 D93 G94 T95 E162 G194 A196 E213 W219 D220 E68 D88 D91 G92 T93 E160 G192 A194 E211 W217 D218 E70 D90 I92 D93 T95 D220 E68 D88 I90 D91 T93 D218 3.1.3.25,3.1.3.94 0000287,0005515,0005737,0005829,0006020,0006021,0006661,0006796,0007165,0008934,0016787,0030145,0031403,0042802,0042803,0046854,0046872,0052834 remove_due_to_license_issue P29218 30289407 305 DPWQECMDYAVTLARQAGEVVCEAIKNEMNVMLKSSPVDLVTATDQKVEKMLISSIKEKYPSHSFIGEESVAAGEKSILTDNPTWIIDPIDGTTNFVHRFPFVAVSIGFAVNKKIEFGVVYSCVEGKMYTARKGKGAFCNGQKLQVSQQEDITKSLLVTELGSSRTPETVRMVLSNMEKLFCIPVHGIRSVGTAAVNMCLVATGGADAYYEMGIHCWDVAGAGIIVTEAGGVLMDVTGGPFDLMSRRVIAANNRILAERIAKEIQVIPLQRDDED 6gj5 A 1.499 BS02 F0N A 1 K5 V7 E37 S39 D54 L56 M67 Q70 Y71 T74 K5 V7 E37 S39 D54 L56 M63 Q66 Y67 T70 3.6.5.2 0003924,0005525,0007165,0016020 Kd=440uM remove_due_to_license_issue P01116 31332011 203 MTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6gj6 A 1.761 BS02 EZZ A 1 K5 L6 V7 E37 D54 L56 Y71 T74 G75 K5 L6 V7 E37 D54 L56 Y67 T70 G71 3.6.5.2 0003924,0005525,0007165,0016020 Kd=20.4uM remove_due_to_license_issue P01116 31332011 204 MTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6gj7 A 1.67 BS02 F0B A 1 K5 V7 E37 S39 D54 L56 Q70 Y71 T74 G75 K5 V7 E37 S39 D54 L56 Q70 Y71 T74 G75 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31332011 203 MTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKH 6gj8 A 1.65 BS01 F0K A 1 K5 V7 E37 S39 D54 L56 Q70 Y71 T74 G75 K6 V8 E38 S40 D55 L57 Q71 Y72 T75 G76 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31332011 201 GMTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKE 6gjb A 1.82 BS01 F0H A 1 G37 A52 K54 Q105 D106 M108 E109 N154 L156 C166 D167 G30 A45 K47 Q98 D99 M101 E102 N147 L149 C159 D160 D149 K151 N154 D167 T190 D142 K144 N147 D160 T183 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.008uM remove_due_to_license_issue P28482 30568786 406 GAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFELDDLPKEKLKELIFEETARFQPG 6gjd A 1.58 BS01 F0E A 1 A35 Y36 R50 A52 K54 I56 Y64 R67 T68 E71 Q105 D106 L107 M108 E109 T110 K114 L156 C166 D167 A26 Y27 R41 A43 K45 I47 Y55 R58 T59 E62 Q96 D97 L98 M99 E100 T101 K105 L147 C157 D158 D149 K151 N154 D167 T190 D140 K142 N145 D158 T181 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 ic50=0.022uM remove_due_to_license_issue P28482 30568786 411 GPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFDDLPKEKLKELIFEETARFQPG 6gji A 1.6 BS01 F1E A 1 G72 A101 N102 A103 Q111 F113 H126 G72 A101 N102 A103 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gjj A 1.38 BS01 L36 A 1 Q63 G72 A101 N102 A103 Q111 F113 H126 Q63 G72 A101 N102 A103 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gjl A 1.16 BS01 F1Q A 1 H54 Q63 G72 A101 N102 F113 H126 H54 Q63 G72 A101 N102 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gjm A 1.354 BS01 L36 A 1 G72 A101 N102 A103 Q111 F113 H126 G72 A101 N102 A103 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gjn A 1.7 BS01 F0Q A 1 H54 R55 M61 Q63 G72 A101 N102 Q111 F113 H126 H54 R55 M61 Q63 G72 A101 N102 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gjr A 1.69 BS01 F0W A 1 H54 R55 Q63 G72 A101 N102 Q111 F113 H126 H54 R55 Q63 G72 A101 N102 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gjw A 1.9 BS02 F2H D 1 R62 C66 H67 S87 P88 N89 R42 C46 H47 S67 P68 N69 2.3.2.27 remove_due_to_license_issue P98170 31011505 102 EEFVEEFNRLKTFANFPSGSPVSASTLARAGFLYTGEGDTVRCFSCHAAVDRWQYGDSAVGRHRKVSPNCRFINGFYL 6gjw D 1.9 BS02 F2H D 1 R62 C66 H67 S87 P88 N89 R42 C46 H47 S67 P68 N69 2.3.2.27 Kd=9uM remove_due_to_license_issue P98170 31011505 102 EEFVEEFNRLKTFANFPSGSPVSASTLARAGFLYTGEGDTVRCFSCHAAVDRWQYGDSAVGRHRKVSPNCRFINGFYL 6gjy A 1.29 BS01 F1Z A 1 G72 A101 N102 A103 Q111 F113 H126 G72 A101 N102 A103 Q111 F113 H126 R55 F60 Q63 N102 F113 L122 H126 R55 F60 Q63 N102 F113 L122 H126 5.2.1.8 0000413,0001933,0001934,0003723,0003755,0005178,0005515,0005576,0005615,0005634,0005737,0005829,0005925,0006357,0006457,0006469,0006915,0016018,0016020,0019076,0030168,0030182,0030593,0030595,0031982,0032148,0032873,0032991,0034389,0034599,0034774,0042118,0043410,0045069,0045070,0046790,0050714,0051082,0051092,0060352,0061944,0070062,0070527,0140839,0140840,1902176,1903901,1904399,1904813,2001233 remove_due_to_license_issue P62937 30746096 201 MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGFMCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTEWLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE 6gl3 A 2.77 BS01 EMW A 1 N390 I562 Y598 V613 H620 G675 L678 I688 N68 I127 Y163 V178 H185 G240 L243 I253 2.7.1.67 0016301,0046854 remove_due_to_license_issue IC50=37nM Q9UBF8 29952567 801 APEREFIKSLMAIGKRLATLPTKEQKTQRLISELSLLNHKLPARVWLPTAGFDHHVVRVPHTQAVVLNSKDKAPYLIYVEVLECENFDTTSVPARIPENEPWQEKVRRIREGSPYGHLPNWRLLSVIVKCGDDLRQELLAFQVLKQLQSIWEQERVPLWIKPYKILVISADSGMIEPVVNAVSIHQVKKQSQLSLLDYFLQEHGSYTTEAFLSAQRNFVQSCAGYCLVCYLLQVKDRHNGNILLDAEGHIIHIDFGFILSSTSAFKLTTEFVDVMGGLDGDMFNYYKMLMLQGLIAARKHMDKVVQIVEIMQQGSQLPCFHGSSTIRNLKERFHMSMTEEQLQLLVEQMVDGSM 6gl8 A 1.4 BS01 F3Q A 1 F104 Y108 D111 F112 M115 Q118 V133 L137 G145 R146 A149 F153 F45 Y49 D52 F53 M56 Q59 V74 L78 G86 R87 A90 F94 ? 0042981 Kd=0.000000064M remove_due_to_license_issue P10415,Q07817 29732004 301 GSYDNREIVMKYIHYKLSQRGYEWDAGADESEVVHKTLREAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 6gl9 A 1.7 BS01 F3W A 1 L828 V836 A853 Y904 L905 C909 R911 R953 L956 L17 V25 A42 Y93 L94 C98 R100 R142 L145 A949 A951 R953 N954 D967 A138 A140 R142 N143 D156 2.7.10.2 0004672,0005524,0006468 ic50=135nM remove_due_to_license_issue IC50=135nM P52333 29852068 1201 QDPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 6gla A 1.92 BS01 F4B A 1 L828 G829 A853 E903 Y904 L905 C909 R911 D912 R953 L956 L16 G17 A41 E91 Y92 L93 C97 R99 D100 R141 L144 A949 A951 R953 N954 D967 A137 A139 R141 N142 D155 2.7.10.2 0004672,0005524,0006468 ic50=27nM remove_due_to_license_issue IC50=0.210000nM, EC50=740nM P52333 29852068 1201 DPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVRQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 6glb A 2.0 BS01 F48 A 1 L828 V836 A853 E903 Y904 L905 C909 R953 N954 L956 L16 V24 A41 E91 Y92 L93 C97 R141 N142 L144 A949 A951 R953 N954 D967 A137 A139 R141 N142 D155 2.7.10.2 0004672,0005524,0006468 ic50=129nM remove_due_to_license_issue IC50=10.0nM P52333 29852068 1201 DPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRALAARNILVESEAHVKIADFGLAKLLPLDKDYYVVRQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGSR 6gmd A 1.66 BS01 A8Q A 1 N118 F121 L124 Y136 P159 V162 I164 M221 M225 N116 F119 L122 Y134 P157 V160 I162 M219 M223 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 29759799 402 GPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTV 6gmq I 2.755 BS01 F4K I 1 L118 R120 G127 L128 L129 E134 L201 L57 R59 G66 L67 L68 E73 L140 ? remove_due_to_license_issue P40337 30040896 302 VLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQER 6gmx B 2.533 BS01 F7B B 1 E64 E102 F109 E39 E77 F84 ? 0006511 remove_due_to_license_issue Kd=6.7nM Q15369 30040896 201 MYVKLISSDGHEFIVKREHALTSGTIKAMLSTNEVNFREIPSHVLSKVCMYFTYKVRYTNSSTEIPEFPIAPEIALELLMAANFLDC 6gn1 B 2.6 BS01 F4N B 1 I62 F67 V70 A83 K85 Y134 V135 Q185 L188 D200 I27 F32 V35 A48 K50 Y94 V95 Q145 L148 D160 D181 K183 N186 D200 S219 D141 K143 N146 D160 S179 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue IC50=10nM P49841 29873877 502 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 6gnm C 2.24 BS01 27M C 1 K15 L17 A108 L109 K6 L8 A99 L100 ? 0005179,0005576,0006144,0007165,0070324 Kd=54.61uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gnm D 2.24 BS01 27M B 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005576,0006144,0007165,0070324 remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gnr A 1.4 BS01 6J3 A 1 K15 A108 K6 A99 ? 0005179,0005576,0006144,0007165,0070324 Kd=3.61uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gnr B 1.4 BS01 6J3 B 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005576,0006144,0007165,0070324 Kd=3.61uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVS 6gnw A 1.75 BS01 F52 C 1 K15 L17 A108 L109 K6 L8 A99 L100 ? 0005179,0005576,0006144,0007165,0070324 remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gnw B 1.75 BS01 F52 D 1 K15 L17 A108 L109 K6 L8 A99 L100 ? 0005179,0005576,0006144,0007165,0070324 remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSSV 6gnw C 1.75 BS01 F52 C 1 L17 A108 L109 L110 L8 A99 L100 L101 ? 0005179,0005576,0006144,0007165,0070324 Kd=10.2uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gnw D 1.75 BS01 F52 D 1 L17 A108 L109 L110 T117 L8 A99 L100 L101 T108 ? 0005179,0005576,0006144,0007165,0070324 Kd=10.2uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gon A 1.65 BS01 8PF A 1 K15 A108 L110 K6 A99 L101 ? 0005179,0005576,0006144,0007165,0070324 Kd=2.16uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVS 6gon B 1.65 BS01 8PF D 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005576,0006144,0007165,0070324 remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVS 6gon C 1.65 BS01 8PF A 1 K15 L17 A108 K6 L8 A99 ? 0005179,0005576,0006144,0007165,0070324 remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6gon D 1.65 BS01 8PF D 1 K15 L17 A108 L110 T117 K6 L8 A99 L101 T108 ? 0005179,0005576,0006144,0007165,0070324 Kd=2.16uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVSS 6goo A 1.8 BS01 8PF A 1 K15 L17 A108 L110 T117 T119 K6 L8 A99 L101 T108 T110 ? 0005179,0005576,0006144,0007165,0070324 Kd=2.16uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVS 6goo B 1.8 BS01 8PF B 1 K15 L17 L110 K6 L8 L101 ? 0005179,0005576,0006144,0007165,0070324 Kd=2.16uM remove_due_to_license_issue Q9PTT3 30226982 201 CPLMVKILDAVKGTPAGSVALKVSQKTADGGWTQIATGVTDATGEIHNLITEQQFPAGVYRVEFDTKAYWTNQGSTPFHEVAEVVFDAHPEGHRHYTLALLLSPFSYTTTAVVS 6gop H 2.9 BS01 F6K H 1 T1 T21 K33 A46 G47 A49 T1 T21 K33 A46 G47 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043 30029468 301 TTIVGVKFNNGVVIAADTRSTQGPIVADKNCAKLHRISPKIWCAGAGTAADTEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6got A 1.56 BS02 F6W A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.4nM remove_due_to_license_issue Kd=25nM P00918 30253337 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6gpb A 2.86 BS04 H2P A 1 G135 H377 N484 R569 Y573 K574 E672 S674 G675 G122 H364 N471 R556 Y560 K561 E659 S661 G662 H377 K568 R569 K574 T676 K680 H364 K555 R556 K561 T663 K667 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 2106586 998 SVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKI 6gqm A 2.0 BS01 F8H A 1 L595 V603 A621 K623 E640 V654 Y672 C673 C674 Y675 G676 L799 I808 C809 D810 F811 L27 V35 A53 K55 E72 V86 Y104 C105 C106 Y107 G108 L165 I174 C175 D176 F177 D792 R796 N797 D810 D158 R162 N163 D176 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue P10721 30204441 1001 SYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAQGLIKSDAAMTVAVKMLKPSAHSTEREALMSELKVLSYLGNHENIVNLLGACTHGGPTLVITEYCCYGDLLNFLRRKRDEFVPYLYKDFLTLEHLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGNITKICDFGLARDIKNDSNYVDKGNARLPVKWMAPESIFNSVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMSSPEYAPAEMYDIMKTCWDADPDKRPTFKQIVQDIEKQISES 6gr7 A 1.4 BS01 F52 A 1 L17 A108 A109 L110 L8 A99 A100 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.19uM remove_due_to_license_issue P02766 30226982 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6gr7 B 1.4 BS01 F52 B 1 A108 A109 L110 A99 A100 L101 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.19uM remove_due_to_license_issue P02766 30226982 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6grp A 1.6 BS01 F4Z A 1 A108 A109 L110 S117 A99 A100 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.34uM remove_due_to_license_issue P02766 30226982 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6grp A 1.6 BS02 F4Z A 2 K15 A108 K6 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.34uM remove_due_to_license_issue P02766 30226982 202 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6grp B 1.6 BS01 F4Z B 1 K15 A108 K6 A99 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.34uM remove_due_to_license_issue P02766 30226982 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6grp B 1.6 BS02 F4Z B 2 A108 L110 S117 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.34uM remove_due_to_license_issue P02766 30226982 202 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6gu2 A 2.0 BS01 F9Z A 1 I10 V18 A31 K33 V64 F80 E81 F82 L83 L135 D146 I13 V21 A34 K36 V67 F83 E84 F85 L86 L138 D149 D128 K130 Q132 N133 D146 V159 T166 D131 K133 Q135 N136 D149 V162 T166 2.7.11.22,2.7.11.23 0000082,0000086,0000226,0000307,0000781,0001618,0003682,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005789,0005813,0005819,0005829,0005856,0005876,0006260,0006281,0006338,0006357,0006468,0006915,0006974,0007077,0007095,0007098,0007344,0008353,0009410,0009636,0010628,0010629,0010971,0014038,0014070,0014075,0014823,0016020,0016301,0016477,0016579,0018105,0018107,0030261,0030332,0030496,0030544,0030855,0031100,0034501,0035173,0042307,0042542,0042752,0043066,0044772,0045471,0045740,0045931,0045995,0046686,0046688,0046718,0048144,0048511,0048678,0051301,0055015,0060045,0062033,0065003,0070062,0070301,0070371,0071407,0072686,0090166,0097121,0097122,0097125,0097472,0106310,0140833,0140834,0140835,0140836,0140837,1900182,1902423,1902850,1905448 Kd=1600nM remove_due_to_license_issue P06493 30472117 301 LGSMEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRHPNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCHSRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIPIRVYTVTLWYRSPEVLLGSARYSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNTFPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFNDLDNQI 6gu3 A 2.65 BS01 FB8 A 1 I10 V18 A31 L83 S84 M85 D86 K89 L135 I13 V21 A34 L86 S87 M88 D89 K92 L138 D128 K130 Q132 N133 D146 V159 T166 D131 K133 Q135 N136 D149 V162 T169 2.7.11.22,2.7.11.23 0000082,0000086,0000226,0000307,0000781,0001618,0003682,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005789,0005813,0005819,0005829,0005856,0005876,0006260,0006281,0006338,0006357,0006468,0006915,0006974,0007077,0007095,0007098,0007344,0008353,0009410,0009636,0010628,0010629,0010971,0014038,0014070,0014075,0014823,0016020,0016301,0016477,0016579,0018105,0018107,0030261,0030332,0030496,0030544,0030855,0031100,0034501,0035173,0042307,0042542,0042752,0043066,0044772,0045471,0045740,0045931,0045995,0046686,0046688,0046718,0048144,0048511,0048678,0051301,0055015,0060045,0062033,0065003,0070062,0070301,0070371,0071407,0072686,0090166,0097121,0097122,0097125,0097472,0106310,0140833,0140834,0140835,0140836,0140837,1900182,1902423,1902850,1905448 remove_due_to_license_issue IC50=62nM P06493 30472117 301 LGSMEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRHPNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCHSRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIPIRVYTHEVVTLWYRSPEVLLGSARYSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNTFPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFND 6gu4 A 2.73 BS01 FC8 A 1 I10 A31 F80 L83 S84 M85 D86 Q132 L135 I13 A34 F83 L86 S87 M88 D89 Q135 L138 D128 K130 Q132 N133 D146 V159 T166 D131 K133 Q135 N136 D149 V162 T169 2.7.11.22,2.7.11.23 0000082,0000086,0000226,0000307,0000781,0001618,0003682,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005789,0005813,0005819,0005829,0005856,0005876,0006260,0006281,0006338,0006357,0006468,0006915,0006974,0007077,0007095,0007098,0007344,0008353,0009410,0009636,0010628,0010629,0010971,0014038,0014070,0014075,0014823,0016020,0016301,0016477,0016579,0018105,0018107,0030261,0030332,0030496,0030544,0030855,0031100,0034501,0035173,0042307,0042542,0042752,0043066,0044772,0045471,0045740,0045931,0045995,0046686,0046688,0046718,0048144,0048511,0048678,0051301,0055015,0060045,0062033,0065003,0070062,0070301,0070371,0071407,0072686,0090166,0097121,0097122,0097125,0097472,0106310,0140833,0140834,0140835,0140836,0140837,1900182,1902423,1902850,1905448 remove_due_to_license_issue IC50=31nM P06493 30472117 301 LGSMEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRHPNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCHSRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIPIRVYTHEVVTLWYRSPEVLLGSARYSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNTFPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFND 6gu6 A 2.33 BS01 1QK A 1 G11 E12 A31 K33 F80 L83 S84 M85 D86 Q132 L135 G11 E12 A31 K33 F80 L83 S84 M85 D86 Q132 L135 D128 K130 Q132 N133 D146 T166 D128 K130 Q132 N133 D146 T163 2.7.11.22,2.7.11.23 0000082,0000086,0000226,0000307,0000781,0001618,0003682,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005789,0005813,0005819,0005829,0005856,0005876,0006260,0006281,0006338,0006357,0006468,0006915,0006974,0007077,0007095,0007098,0007344,0008353,0009410,0009636,0010628,0010629,0010971,0014038,0014070,0014075,0014823,0016020,0016301,0016477,0016579,0018105,0018107,0030261,0030332,0030496,0030544,0030855,0031100,0034501,0035173,0042307,0042542,0042752,0043066,0044772,0045471,0045740,0045931,0045995,0046686,0046688,0046718,0048144,0048511,0048678,0051301,0055015,0060045,0062033,0065003,0070062,0070301,0070371,0071407,0072686,0090166,0097121,0097122,0097125,0097472,0106310,0140833,0140834,0140835,0140836,0140837,1900182,1902423,1902850,1905448 Kd=1810nM remove_due_to_license_issue P06493 30472117 301 MEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRHPNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCHSRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIPITHEVVTLWYRSPEVLLGSARYSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNTFPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFNDLD 6gu7 A 2.75 BS01 FB8 A 1 I10 A31 K33 E81 L83 S84 D86 K89 L135 D146 I10 A31 K33 E81 L83 S84 D86 K89 L135 D146 D128 K130 Q132 N133 D146 T166 D128 K130 Q132 N133 D146 T157 2.7.11.22,2.7.11.23 0000082,0000086,0000226,0000307,0000781,0001618,0003682,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005737,0005739,0005759,0005789,0005813,0005819,0005829,0005856,0005876,0006260,0006281,0006338,0006357,0006468,0006915,0006974,0007077,0007095,0007098,0007344,0008353,0009410,0009636,0010628,0010629,0010971,0014038,0014070,0014075,0014823,0016020,0016301,0016477,0016579,0018105,0018107,0030261,0030332,0030496,0030544,0030855,0031100,0034501,0035173,0042307,0042542,0042752,0043066,0044772,0045471,0045740,0045931,0045995,0046686,0046688,0046718,0048144,0048511,0048678,0051301,0055015,0060045,0062033,0065003,0070062,0070301,0070371,0071407,0072686,0090166,0097121,0097122,0097125,0097472,0106310,0140833,0140834,0140835,0140836,0140837,1900182,1902423,1902850,1905448 remove_due_to_license_issue IC50=62nM P06493 30472117 301 MEDYTKIEKIGEGTYGVVYKGRHKTTGQVVAMKKIRLESEEEGVPSTAIREISLLKELRHPNIVSLQDVLMQDSRLYLIFEFLSMDLKKYLDSIPPGQYMDSSLVKSYLYQILQGIVFCHSRRVLHRDLKPQNLLIDDKGTIKLADFGLARAFGIVTLWYRSPEVLLGSARYSTPVDIWSIGTIFAELATKKPLFHGDSEIDQLFRIFRALGTPNNEVWPEVESLQDYKNTFPKWKPGSLASHVKNLDENGLDLLSKMLIYDPAKRISGKMALNHPYFNDLDNQ 6gub A 2.52 BS01 F9Z A 1 I10 Y15 V18 A31 K33 V64 F80 E81 L83 L134 D145 I11 Y16 V19 A32 K34 V62 F78 E79 L81 L132 D143 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 30472117 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 6guc A 2.0 BS01 SU9 A 1 I10 A31 K33 F80 L83 L134 I11 A32 K34 F76 L79 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=25nM remove_due_to_license_issue IC50=22nM P24941 30472117 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHL 6gue A 1.99 BS01 FB8 A 1 I10 A31 K33 F80 L83 H84 D86 K89 L134 I11 A32 K34 F76 L79 H80 D82 K85 L130 D127 K129 Q131 N132 D145 T158 T165 D123 K125 Q127 N128 D141 T154 T161 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=4nM remove_due_to_license_issue IC50=6nM P24941 30472117 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKITEGVPSTAIREISLLKELNHPNIVKLLDVIHTNNKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 6guf A 2.65 BS01 23D A 1 F80 F82 L83 H84 Q85 D86 L134 F78 F80 L81 H82 Q83 D84 L132 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 remove_due_to_license_issue P24941 30472117 301 SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 6guh A 1.5 BS01 FB8 A 1 I10 V18 A31 F80 L83 H84 Q85 D86 K89 L134 D145 I12 V20 A33 F74 L77 H78 Q79 D80 K83 L128 D139 D127 K129 Q131 N132 D145 T158 T165 D121 K123 Q125 N126 D139 T144 T151 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=26nM remove_due_to_license_issue IC50=6nM P24941 30472117 301 EFMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 6guk A 1.3 BS01 FC8 A 1 I10 G11 E12 A31 F80 L83 H84 D86 L134 I10 G11 E12 A31 F70 L73 H74 D76 L124 D127 K129 Q131 N132 D145 T165 D117 K119 Q121 N122 D135 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=715nM remove_due_to_license_issue IC50=26nM P24941 30472117 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 6gva A 2.15 BS01 FCQ A 1 E8 I10 V18 A31 F80 F82 L83 Q131 L134 E8 I10 V18 A31 F78 F80 L81 Q129 L132 D127 K129 Q131 N132 D145 T158 T165 D125 K127 Q129 N130 D143 T156 T163 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 ic50=5nM remove_due_to_license_issue P24941 30943029 301 MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVT 6gvf A 2.5 BS01 FE5 A 1 D810 Y836 I848 E849 V850 V851 M922 D933 D685 Y711 I723 E724 V725 V726 M787 D798 2.7.11.1,2.7.1.137,2.7.1.153 0016301,0046854 Ki=28nM remove_due_to_license_issue Kd=15nM, Ki=28nM P42336 31749911 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGW 6gvg A 3.0 BS01 FCZ A 1 M772 I800 D810 Y836 V851 M922 D933 M647 I675 D685 Y711 V726 M787 D798 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue Ki=990nM P42336 31749911 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGW 6gvh A 2.74 BS01 FDH A 1 M772 K802 D810 Y836 I848 V851 M922 I932 D933 M650 K680 D688 Y714 I726 V729 M790 I800 D801 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue Ki=920nM P42336 31749911 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRTSTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREAGFSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGW 6gvi A 2.9 BS01 FDW A 1 I800 K802 D810 Y836 I848 V850 V851 M922 D933 I675 K677 D685 Y711 I723 V725 V726 M787 D798 2.7.11.1,2.7.1.137,2.7.1.153 0001525,0001889,0001944,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0005944,0006006,0006629,0006909,0007173,0008286,0010468,0010592,0010629,0014704,0014823,0014870,0016242,0016301,0016303,0030027,0030036,0030168,0030295,0030835,0031295,0032008,0032869,0035005,0035175,0035402,0035403,0035979,0035994,0036092,0038084,0040014,0043201,0043276,0043457,0043491,0043524,0043542,0043560,0044022,0044023,0044024,0044025,0046854,0046934,0048009,0048015,0048471,0048661,0050852,0051897,0055119,0060048,0060612,0071333,0071464,0071548,0072354,0072371,0072518,0086003,0097009,0106310,0110053,0140823,0140855,0140857,0141068,1903544,1905477,1990244,2000270,2000811 remove_due_to_license_issue Ki=150nM P42336 31749911 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSMLLSSEQLKLCVLEYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRRTKSLWVINSALRIKILCATYVNVNIRDIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKGRKGAKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHKKRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGW 6gvx A 2.24 BS01 TAK A 1 A38 L86 E87 C89 P90 G91 L139 A40 L85 E86 C88 P89 G90 L138 D132 K134 N137 D150 S171 D131 K133 N136 D149 S163 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 Ki=24nM remove_due_to_license_issue Q14680 31108049 402 PLGSMKDYDELLKYYELHETIGTFAKVKLACHILTGEMVAIKIMDKNTDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKCGSLAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR 6gvz A 1.54 BS01 CHO A 1 W355 S356 P357 F390 W135 S136 P137 F170 ? Kd=0.4uM remove_due_to_license_issue J9XXB7 30355683 600 GPGSKPFTLPILTIGELSNSRFPVPIDELYTSPNEGVIVQPQNGRSTLDGELLGTTQLVPSNICALRGRINAQVPDDHHQWNLQVTNTNGTPFDPTEDVPAPLGTPDFLANIYGVTSQRNPNNTCRAHDGVLATWSPKFTPKLGSVILGTWEESDLDLNQPTRFTPVGLFNTDHFDQWALPSYSGRLTLNMNLAPSVSPLFPGEQLLFFRSHIPLKGGTSDGAIDCLLPQEWIQHFYQESAPSPTDVALIRYTNPDTGRVLFEAKLHRQGFITVANSGSRPIVVPPNGYFRFDSWVNQFYSLAPM 6gw1 A 1.9 BS01 CHO A 1 H298 R299 Q333 V361 S379 W381 H73 R74 Q108 V132 S150 W152 ? Kd=0.000000064M remove_due_to_license_issue Q5F4T5 30355683 601 PFTLPILTLGELTNSRFPLPIDVLYTNPNESAIVQCQNGRCTLDGELQGTTQLLPTGICAFRGKVTQQVQDEHRGTHWNMTVTNLNGTPFDPTEDVPAPLGTPDFSGQIYGVISQRNTNTGNLPANRAHEAVIATYSPKFTPKLGNIQFSTWETQDVSSGQPTKFTPVGLASVDANSHFDQWTLPSYSGALTLNMNLAPSVAPVFPGECLLFFRSFIPLKGGYGNPAIDCLMPQEWVQHLYQESAPSLSDVALVRYVNPETGRTLFEAKLHRNGFLTVARNSAGPVVAPTNGYFRFDSWVNQFYTLAPM 6gw4 A 2.295 BS01 CHO A 1 H300 Q301 P360 S363 A364 T377 W378 H76 Q77 P136 S139 A140 T153 W154 ? Kd=0.000000064M remove_due_to_license_issue A0ZNP3 30355683 600 KPFTLPVLTIGEMTNSRFPAPIDMLYTSPNGNVVVQPQNGRCTLDGELQGSTQLVPANVCAFRGKITARIVDQAAHQWHMQIDNPNGTLFDPTEDVPAPLGTPDFKAKIFGVISQRNDYNDGSQGPANRAHDAVVPTTSAKFTPKLGSILVGTWENNDIETQPSKFTPVGLLEMNDFNQWSLPNYSGALTLNMGLAPAVFPTFPGEQILFFRSFIPLKGGHGNPAIDCLLPQEWIQHFYQESAPSQTSVALIRYVNPDTGRVLFEGKLHRQGFITIAKSGDGPIVVPPNGYFRFDSWVNQFYSLAPM 6gwr A 2.07 BS01 FEW A 1 V624 K655 E672 I675 M676 L679 I685 M699 T701 Y703 M704 F762 H764 L773 A783 D784 V25 K52 E69 I72 M73 L76 I82 M96 T98 Y100 M101 F150 H152 L161 A171 D172 D766 R770 N771 D784 D154 R158 N159 D172 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd=7.9nM remove_due_to_license_issue Kd=7.9nM, IC50=9.4nM Q08345 30075624 1001 MPRVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSLDFPLGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEDKAAEQGPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDALNT 6gx3 A 2.1 BS02 FF2 A 1 H141 H142 G150 D186 H188 F216 H292 Y341 H139 H140 G148 D175 H177 F205 H275 Y311 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=250nM remove_due_to_license_issue A5H660 29806110 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6gx3 A 2.1 BS03 FF2 A 2 E131 K330 V331 P332 V361 E129 K300 V301 P302 V331 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=250nM remove_due_to_license_issue A5H660 29806110 505 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6gx6 A 2.0 BS01 rna B 0 Y5 K36 Y39 F41 S73 V74 R79 Y7 K38 Y41 F43 S75 V76 R81 ? 0003676,0003723 remove_due_to_license_issue O00425 30135093 1 ~ 4 GSMNKLYIGNLSENAAPSDLESIFKDAKIPVSGPFLVKTGYAFVDCPDESWALKAIEALSGKIELHGKPIEVEHSVPKRQRIRKLQIRNIPPHLQWEVLDSLLVQYGVVESCEQVNTDSETAVVNVTYSSKDQARQALDKLNGFQLENFTLKVAYIPDE 6gxa A 2.1 BS02 TB8 A 1 K20 D100 H141 H142 D186 H188 F216 Y341 K19 D99 H140 H141 D176 H178 F206 Y313 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=60nM remove_due_to_license_issue A5H660 29806110 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6gxb A 1.35 BS02 FF5 A 1 D72 L91 Q92 H94 H119 V121 V130 L197 T198 T199 D69 L88 Q89 H91 H116 V118 V127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6gxe A 1.3 BS02 FFH A 1 H94 H119 V134 L197 T198 T199 P201 H91 H116 V131 L194 T195 T196 P198 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6gxe A 1.3 BS03 FFH A 2 H4 W5 H15 W16 D19 H1 W2 H12 W13 D16 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue P00918 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6gxg A 1.6 BS01 FFN A 1 W39 C40 W70 E107 S108 I109 W41 C42 W72 E109 S110 I111 ? 0004791,0005634,0030178,0031397,0098869 remove_due_to_license_issue O77404 30605929 201 AMGSGLAKYLPGATNLLSKSGEVSLGSLVGKTVFLYFSASWCPPCRGFTPVLAEFYEKHHVAKNFEVVLISWDENESDFHDYYGKMPWLALPFDQRSTVSELGKTFGVESIPTLITINADTGAIIGTQARTRVIEDPDGANFPW 6gxq A 1.96 BS02 FFZ A 1 M785 D822 N825 G873 Q874 F877 M200 D237 N240 G288 Q289 F292 3.1.4.- 0004114,0007165,0008081 Ki=0.00000079M remove_due_to_license_issue Kd=79nM, Ki=158nM Q8WQX9 31378593 1005 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLETR 6gxu A 1.917 BS02 FG8 A 1 K20 D100 H141 H142 D186 H188 F216 P291 H292 Y341 K19 D98 H139 H140 D175 H177 F205 P274 H275 Y312 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=180nM remove_due_to_license_issue A5H660 29806110 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKLTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDY 6gxw A 2.071 BS02 FGN A 1 K20 H142 H188 F216 H292 Y341 K19 H141 H178 F206 H275 Y311 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=440nM remove_due_to_license_issue A5H660 29806110 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6gxy A 1.8 BS01 FFN A 1 W39 C40 W70 V106 E107 S108 I109 W40 C41 W71 V107 E108 S109 I110 ? 0004791,0005634,0030178,0031397,0098869 remove_due_to_license_issue O77404 30605929 201 MGSGLAKYLPGATNLLSKSGEVSLGSLVGKTVFLYFSASWCPPCRGFTPVLAEFYEKHHVAKNFEVVLISWDENESDFHDYYGKMPWLALPFDQRSTVSELGKTFGVESIPTLITINADTGAIIGTQARTRVIEDPDGANFPWPN 6gxy B 1.8 BS01 FFN B 1 W39 C40 W70 V106 E107 S108 I109 W41 C42 W72 V108 E109 S110 I111 ? 0004791,0005634,0030178,0031397,0098869 remove_due_to_license_issue O77404 30605929 201 GMGSGLAKYLPGATNLLSKSGEVSLGSLVGKTVFLYFSASWCPPCRGFTPVLAEFYEKHHVAKNFEVVLISWDENESDFHDYYGKMPWLALPFDQRSTVSELGKTFGVESIPTLITINADTGAIIGTQARTRVIEDPDGANFPWPN 6gy0 A 2.55 BS01 FGE A 1 M752 W760 K779 Y813 I825 V828 S831 M900 I910 M556 W564 K583 Y617 I629 V632 S635 M704 I714 2.7.1.137,2.7.1.153 0001782,0002250,0005524,0005737,0005829,0006629,0006935,0006954,0007166,0010628,0016301,0016303,0030154,0036092,0042113,0043491,0045087,0045766,0046854,0046934,0048872,0050832 remove_due_to_license_issue O35904 30718815 1101 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 6gy1 A 2.1 BS03 FGQ A 1 M40 D141 H142 W143 K144 N170 E199 M38 D139 H140 W141 K142 N168 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 ic50=0.501uM remove_due_to_license_issue P22734 30272964 303 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQG 6gz9 A 3.1 BS01 TXC A 1 Y41 V166 N347 P348 N426 Y33 V158 N339 P340 N418 0006857,0015833,0016020,0022857,0055085,1904680 remove_due_to_license_issue 30602453 501 QTIQSIPQKGFFGHPRGLGVLFFVEFWERFSYYGMRAMLIFYMYFAIHQNGLGIDKTTAMSIMSVYGALIYMSSIPGAWIADRITGTRGATLLGAVLIIIGHICLSLPFALFGLFSSMFFIIIGSGLMKPNISNIVGRLYPENDTRIDAGFVIFYMSVNLGALISPIILQHFVDIRNFHGGFLLAAIGMALGLVWYLLFNRKNLGSVGMKPTNPLSKEEKRKYGMIIGIIVAIVIVVLLVTYYTHTLSFDLISNTVLVLGVALPIIYFTTMLRSKDVTDGERSRVKAFIPLFILGMLFWSIQEQGSNVLNIYGLERSDMQLNLFGWTTRFGEALFQSINPLFILLFAPVISMIWLKMGKKQPSLAIKFSIGTLLAGLSYILIGLVGLGYGHTQFSVNWVILSYVICVIGELCLSPTGNSAAVKLAPKAFNAQMMSVWLLTNASAQAINGTLVKLIKPLGQTNYFIFLGTVAIVITLIILVFSPKITKA 6gzd A 2.28 BS02 LCI A 1 S25 I31 A44 M90 L93 D99 L143 S17 I23 A36 M82 L85 D91 L135 2.7.11.1 0000775,0000776,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005694,0005737,0005813,0005819,0005829,0005847,0005856,0005929,0006338,0006468,0007030,0007165,0007166,0016020,0016055,0016607,0018105,0019082,0030877,0031670,0032436,0035025,0035175,0035402,0035403,0035979,0036064,0042995,0043161,0044022,0044023,0044024,0044025,0045095,0045104,0051301,0072354,0072371,0072518,0090090,0106310,0140823,0140855,0140857,1900226,1904263,1990244 Kd=9.8nM remove_due_to_license_issue P48729 30146162 1018 AEFIVGGKYKLGRKIGSGSFGDIYLATNITNGEEVAVKLESQKARHPQLHYESKLYKILQGGVGIPHIRWYGQEKDYNVLVMDLLGPSLEDLFNFCSRRFTMKTVLMLADQMISRIEYVHTKNFIHRDIKPDNFLMGIGRHCNKLFLIDFGLAKKYRDNRTRQHIPYREDKNLTGTARYASINAHLGIEQSRRDDMESLGYVLMYFNRTSLPWQGLKAATKKQKYEKISEKKMSTPVEVLCKGFPAEFAMYLNYCRGLRFEEAPDYMYLRQLFRILFRTLNHQYDYTFDWTMLKQKA 6gzh A 3.17 BS01 LCI A 1 I25 G26 F30 A46 F103 F105 C106 D109 L156 I18 G19 F23 A39 F90 F92 C93 D96 L143 D149 K151 N154 D167 T191 D136 K138 N141 D154 T175 2.7.11.22,2.7.11.23 0004672,0005524,0006468 remove_due_to_license_issue P50750 30146162 2001 VECPFCDEVSKYEKLAKIGQGTFGEVFKARHRKTGQKVALKKVLMENEKEGFPITALREIKILQLLKHENVVNLIEICRTKASGSIYLVFDFCEHDLAGLLSNVLVKFTLSEIKRVMQMLLNGLYYIHRNKILHRDMKAANVLITRDGVLKLADFGLARAFSLAQPNRYTNRVVTLWYRPPELLLGERDYGPPIDLWGAGCIMAEMWTRSPIMQGNTEQHQLALISQLCGSITPEVWPNVDNYELYEKLELVKGQKRKVKDRLKAYVRDPYALDLIDKLLVLDPAQRIDSDDALNHDFFWSDPMPSDLKG 6gzm A 1.59 BS01 LCI A 1 I23 A36 M82 L85 D91 L135 I148 I19 A32 M78 L81 D87 L131 I144 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue P48730 30146162 1004 VGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF 6gzm B 1.59 BS01 LCI A 1 E2 R10 E2 R10 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue P48730 30146162 1004 MELRVGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF 6gzm B 1.59 BS02 LCI B 1 I15 G16 I23 A36 M82 L85 D91 L135 I148 I15 G16 I23 A36 M82 L85 D91 L135 I148 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue P48730 30146162 1003 MELRVGNRYRLGNKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKF 6gzy A 2.15 BS01 FHH A 1 I869 Y878 C885 H887 F888 H889 T891 S899 Q974 I12 Y21 C28 H30 F31 H32 T34 S42 Q108 2.3.2.31 0004842,0008270,0071797 remove_due_to_license_issue Q96EP0 30657686 4001 QGLAMYLQENGIDCPKCKFSYALARGGCMHFHCTQCRHQFCSGCYNAFYAKNKCPEPNCRVKKSLHGHHPRDCLFYLRDWTALRLQKLLQDNNVMFNTEPPGCRVIEQRDEACGKETPAGYAGLCQAHYKEYLVSLINAHSLDPATLYEVEELETATERYLHVRPQPLAGEDPPAYQARLLQKLTEEVPLGQSIPRRRK 6h0u A 2.3 BS01 FKB A 1 V70 A83 K85 Y134 V135 R141 L188 C199 D200 V35 A48 K50 Y99 V100 R106 L153 C164 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0001837,0001954,0002020,0002039,0003170,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005515,0005524,0005634,0005654,0005737,0005739,0005813,0005829,0005886,0005977,0006338,0006468,0006983,0007005,0007212,0007399,0007623,0008013,0008286,0009968,0010508,0010628,0010629,0010719,0010975,0016055,0016301,0018105,0018107,0019082,0019901,0021766,0030010,0030011,0030154,0030336,0030424,0030425,0030516,0030877,0031175,0031333,0031334,0031398,0031625,0032007,0032092,0032436,0032886,0034236,0034452,0035175,0035402,0035403,0035556,0035979,0036016,0042752,0043066,0043161,0043525,0043547,0044022,0044023,0044024,0044025,0045597,0045668,0045719,0045724,0045732,0046777,0046825,0046827,0048156,0048511,0048814,0050321,0050770,0051059,0051093,0060070,0060079,0061629,0070507,0070885,0071109,0071300,0072354,0072371,0072518,0090090,0097110,0097191,0097192,0098793,0098794,0098978,0099171,0106027,0106310,0140823,0140855,0140857,0150101,1900034,1900181,1900271,1901030,1901984,1902042,1903566,1903940,1904339,1904646,1904781,1904886,1990244,1990909,2000077,2000466,2000740 remove_due_to_license_issue P49841 30548443 501 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR 6h12 A 2.2 BS01 FJK A 1 Y70 Q74 W84 Y121 W279 F330 F331 W432 H440 Y67 Q71 W81 Y118 W276 F327 F328 W429 H437 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30798053 626 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6h13 B 2.8 BS01 FJN B 1 W84 Y121 W279 L282 F284 F330 W432 H440 W81 Y118 W276 L279 F281 F327 W429 H437 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30798053 605 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSQESKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6h14 B 1.86 BS01 FW8 B 1 W84 Y121 W279 L282 F288 F330 F331 W432 H440 W81 Y118 W276 L279 F285 F327 F328 W429 H437 G118 G119 S200 A201 E327 H440 G115 G116 S197 A198 E324 H437 3.1.1.7 0001507,0003990,0004104,0005615,0005886,0006581,0019695,0043083,0045202,0052689,0098552 remove_due_to_license_issue P04058 30798053 609 SELLVNTKSGKVMGTRVPVLSSHISAFLGIPFAEPPVGNMRFRRPEPKKPWSGVWNASTYPNNCQQYVDEQFPGFSGSEMWNPNREMSEDCLYLNIWVPSPRPKSTTVMVWIYGGGFYSGSSTLDVYNGKYLAYTEEVVLVSLSYRVGAFGFLALHGSQEAPGNVGLLDQRMALQWVHDNIQFFGGDPKTVTIFGESAGGASVGMHILSPGSRDLFRRAILQSGSPNCPWASVSVAEGRRRAVELGRNLNCNLNSDEELIHCLREKKPQELIDVEWNVLPFDSIFRFSFVPVIDGEFFPTSLESMLNSGNFKKTQILLGVNKDEGSFFLLYGAPGFSKDSESKISREDFMSGVKLSVPHANDLGLDAVTLQYTDWMDDNNGIKNRDGLDDIVGDHNVICPLMHFVNKYTKFGNGTYLYFFNHRASNLVWPEWMGVIHGYEIEFVFGLPLVKELNYTAEEEALSRRIMHYWATFAKTGNPNEPHSSKWPLFTTKEQKFIDLNTEPMKVHQRLRVQMCVFWNQFLPKLLNAT 6h1d A 1.94 BS01 SAH A 1 Y23 T29 G53 S54 G55 D77 I78 D103 L104 N122 P124 A140 Y17 T23 G47 S48 G49 D71 I72 D97 L98 N116 P118 A134 2.1.1.- 0003676,0005515,0005634,0005829,0006325,0008168,0008276,0008757,0009007,0009404,0018364,0018872,0030307,0030791,0032259,0032775,0032991,0035657,0036009,0042054,0045814,0045815,0140984,1904047 remove_due_to_license_issue Q9Y5N5 31061526 301 STPFHGHVGRGAFSDVYEPAEDTFLLLDALEAAAAELAGVEICLEVGSGSGVVSAFLASMIGPQALYMCTDINPEAAACTLETARCNKVHIQPVITDLVKGLLPRLTEKVDLLVFNPPYVVTPPQEVGSHGIEAAWAGGRNGREVMDRFFPLVPDLLSPRGLFYLVTIKENNPEEILKIMKTKGLQGTTALSRQAGQETLSVLKFTK 6h1h A 1.54 BS02 FJE A 1 D43 F45 F53 H56 E103 Q115 W117 D40 F42 F50 H53 E100 Q112 W114 1.13.11.24 0003712,0005515,0005634,0005654,0005737,0005829,0006366,0007586,0008127,0016604,0030099,0030224,0046872,0051213 remove_due_to_license_issue O00625 30613326 302 SKKVTLSVLSREQSEGVGARVRRSIGRPELKNLDPFLLFDEFKGGRPGGFPDHPHRGFETVSYLLEGGSMAHEDFCGHTGKMNPGDLQWMTAGRGILHAEMPCSEEPAHGLQLWVNLRSSEKMVEPQYQELKSEEIPKPSKDGVTVAVISGEALGIKSKVYTRTPTLYLDFKLDPGAKHSQPIPKGWTSFIYTISGDVYIGPDDAQQKIEPHHTAVLGEGDSVQVENKDPKRSHFVLIAGEPLREPVIQHGPFVMNTNEEISQAILDFRNAKNGFERAKTWKSKIGN 6h1i A 1.69 BS02 FJH A 1 E18 R26 L41 D43 F45 F53 P54 H56 S65 G113 Q115 W117 E15 R23 L38 D40 F42 F50 P51 H53 S62 G110 Q112 W114 1.13.11.24 0003712,0005515,0005634,0005654,0005737,0005829,0006366,0007586,0008127,0016604,0030099,0030224,0046872,0051213 remove_due_to_license_issue IC50=44nM, Kd=38nM O00625 30613326 305 SKKVTLSVLSREQSEGVGARVRRSIGRPELKNLDPFLLFDEFKGGRPGGFPDHPHRGFETVSYLLEGGSMAHEDFCGHTGKMNPGDLQWMTAGRGILHAEMPCSEEPAHGLQLWVNLRSSEKMVEPQYQELKSEEIPKPSKDGVTVAVISGEALGIKSKVYTRTPTLYLDFKLDPGAKHSQPIPKGWTSFIYTISGDVYIGPDDAQQKIEPHHTAVLGEGDSVQVENKDPKRSHFVLIAGEPLREPVIQHGPFVMNTNEEISQAILDFRNAKNGFERAKTWKSKIGN 6h1u A 1.68 BS01 ASP A 1 R147 T162 S164 R169 T211 T212 W232 D250 I253 R106 T121 S123 R128 T170 T171 W191 D209 I212 ? 0005576,0006865,0030288 Kd=4.8uM remove_due_to_license_issue P96257 30065086 401 LPTPVGMEIMPPQPPLPPDSSSQDCDPTASLRPFATKAEADAAVADIRARGRLIVGLDIGSNLFSFRDPITGEITGFDVDIAGEVARDIFGVPSHVEYRILSAAERVTALQKSQVDIVVKTMSITCERRKLVNFSTVYLDANQRILAPRDSPITKVSDLSGKRVCVARGTTSLRRIREIAPPPVIVSVVNWADCLVALQQREIDAVSTDDTILAGLVEEDPYLHIVGPDMADQPYGVGINLDNTGLVRFVNGTLERIRNDGTWNTLYRKWLTVLGPAPAPPTPRYVD 6h29 A 1.46 BS02 FK8 A 1 H94 H96 V121 F131 L141 L198 T199 H94 H96 V121 F130 L140 L197 T198 H64 H94 H96 E106 H119 T199 H64 H94 H96 E106 H119 T198 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.4uM remove_due_to_license_issue P00918 30140816 302 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6h2t A 1.67 BS01 GLU A 1 R147 T162 S164 R169 T211 T212 W232 D250 R107 T122 S124 R129 T171 T172 W192 D210 ? 0005576,0006865,0030288 Kd=15.2uM remove_due_to_license_issue P96257 30065086 401 PLPTPVGMEIMPPQPPLPPDSSSQDCDPTASLRPFATKAEADAAVADIRARGRLIVGLDIGSNLFSFRDPITGEITGFDVDIAGEVARDIFGVPSHVEYRILSAAERVTALQKSQVDIVVKTMSITCERRKLVNFSTVYLDANQRILAPRDSPITKVSDLSGKRVCVARGTTSLRRIREIAPPPVIVSVVNWADCLVALQQREIDAVSTDDTILAGLVEEDPYLHIVGPDMADQPYGVGINLDNTGLVRFVNGTLERIRNDGTWNTLYRKWLTVLGPAPAPPTPRYVD 6h2z A 1.94 BS02 FKE A 1 H94 H119 G132 V135 L198 T199 T200 P202 H91 H116 G128 V131 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.5nM remove_due_to_license_issue Ki=0.500000nM P00918 30530195 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6h33 A 1.58 BS02 FKQ A 1 H94 H119 V135 L198 T199 T200 P202 H95 H120 V135 L198 T199 T200 P202 H64 H94 H96 E106 H119 T199 H65 H95 H97 E107 H120 T199 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.6nM remove_due_to_license_issue Ki=0.600000nM P00918 30530195 302 GMSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6h34 A 1.55 BS02 FKK A 1 H3 F20 Q92 H94 H119 V121 L198 T199 P201 P202 H1 F18 Q90 H92 H117 V119 L195 T196 P198 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.5nM remove_due_to_license_issue Ki=0.500000nM P00918 30530195 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6h36 A 1.85 BS02 FKE A 1 Q92 H94 H119 V121 F131 L198 T199 P202 Q89 H91 H116 V118 F128 L195 T196 P199 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005737,0005829,0006730,0008270,0016829,0032230,0032849,0046872,0051453,0070050,2001225 Ki=0.45nM remove_due_to_license_issue Ki=0.450000nM P43166 30530195 302 GWGYGQDDGPSHWHKLYPIAQGDRQSPINIISSQAVYSPSLQPLELSYEACMSLSITNNGHSVQVDFNDSDDRTVVTGGPLEGPYRLKQFHFHWGKKHDVGSEHTVDGKSFPSELHLVHWNAKKYSTFGEAASAPDGLAVVGVFLETGDEHPSMNRLTDALYMVRFKGTKAQFSCFNPKSLLPASRHYWTYPGSLTTPPLSESVTWIVLREPISISERQMGKFRSLLFTSEDDERIHMVNNFRPPQPLKGRVVKASFRA 6h37 A 1.9 BS02 FKQ A 1 Q92 H94 H119 V121 F131 A135 L198 T199 P202 Q88 H90 H115 V117 F127 A131 L194 T195 P198 H64 H94 H96 E106 H119 T199 H60 H90 H92 E102 H115 T195 4.2.1.1 0004089,0005737,0005829,0006730,0008270,0016829,0032230,0032849,0046872,0051453,0070050,2001225 Ki=2.6nM remove_due_to_license_issue Ki=2.6nM P43166 30530195 302 WGYGQDDGPSHWHKLYPIAQGDRQSPINIISSQAVYSPSLQPLELSYEACMSLSITNNGHSVQVDFNDSDDRTVVTGGPLEGPYRLKQFHFHWGKKHDVGSEHTVDGKSFPSELHLVHWNAKKYSTFGEAASAPDGLAVVGVFLETGDEHPSMNRLTDALYMVRFKGTKAQFSCFNPKSLLPASRHYWTYPGSLTTPPLSESVTWIVLREPISISERQMGKFRSLLFTSEDDERIHMVNNFRPPQPLKGRVVKASFRA 6h38 A 1.7 BS02 FKK A 1 Y20 Q92 H94 H119 V121 F131 L198 T199 T200 P201 P202 Y17 Q89 H91 H116 V118 F128 L195 T196 T197 P198 P199 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T196 4.2.1.1 0004089,0005737,0005829,0006730,0008270,0016829,0032230,0032849,0046872,0051453,0070050,2001225 Ki=7.8nM remove_due_to_license_issue Ki=7.8nM P43166 30530195 302 GWGYGQDDGPSHWHKLYPIAQGDRQSPINIISSQAVYSPSLQPLELSYEACMSLSITNNGHSVQVDFNDSDDRTVVTGGPLEGPYRLKQFHFHWGKKHDVGSEHTVDGKSFPSELHLVHWNAKKYSTFGEAASAPDGLAVVGVFLETGDEHPSMNRLTDALYMVRFKGTKAQFSCFNPKSLLPASRHYWTYPGSLTTPPLSESVTWIVLREPISISERQMGKFRSLLFTSEDDERIHMVNNFRPPQPLKGRVVKASFRA 6h3k A 2.48 BS01 FMW A 1 Q541 G605 I607 D608 S611 L654 Q26 G90 I92 D93 S96 L139 D647 K649 N652 D664 T686 D132 K134 N137 D149 T159 2.7.12.1 0004672,0005524,0006468 Ki=0.11mM remove_due_to_license_issue IC50=3.00nM, Ki=0.110000nM P33981 30199249 801 QSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 6h3q A 1.31 BS02 FMH A 1 H94 H119 F131 L198 T199 T200 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=47.3nM remove_due_to_license_issue Ki=73nM P00918 30193219 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6h4a A 2.65 BS01 FNB A 1 A345 L346 K379 V381 E390 N393 A394 E397 F398 L401 Q676 A6 L7 K40 V42 E51 N54 A55 E58 F59 L62 Q319 3.4.22.- 0004197,0006508 remove_due_to_license_issue IC50=0.005nM Q9UDY8 30692685 801 AKDKVALLIGNMNYREHPKLKAPLVDVYELTNLLRQLDFKVVSLLDLTEYEMRNAVDEFLLLLDKGVYGLLYYAGHGYENFGNSFMVPVDAPNPYRSENCLCVQNILKLMQEKETGLNVFLLDMCRVTANIVFGYATCQEAFEIQHSGLANGIFMKFLKDRLLEDKKITVLLDEVAEDMGKCHLTKGKQALEIRSSLSEKRALTDPIQGTEYSAESLVRNLQWAKAHELPESMCLKFDCGVQIQLGFAAEFSNVMIIYTSIVYKPPEIIMCDAYVTDFPLDLDIDPKDANKGTPEETGSYLVSKDLPKHCLYTRLSSLQKLKEHLVFTVCLSYQYSGLEDTVEDKQEVNVGKPLIAKL 6h4d A 2.9 BS02 GDP A 1 N159 K160 D162 S190 F192 G216 G218 K219 S220 S221 N118 K119 D121 S149 F151 G175 G177 K178 S179 S180 3.6.1.- 0003924,0005525,0005737,0016787,0019843,0042254,0042274,0046872 remove_due_to_license_issue Q9HUL3 31199072 402 DLGPEQTGQVIAHFGVQVEVESADGQVSRCHLRANLPALVTGDQVVWRAGGIGVIVAQLPRRSELCRPDMRGLLKPVAANVDRIVIVFAPRPEPHANLIDRYLIAAEHAGIQPLLLLNKADLVDESNAEGIDALLNVYRTLGYPLIEVSAFNGLAMDELRGALDGHVSVFVGQSGVGKSSLVNALLPGTARLFHFPGGGDLIDSPGIREFGLGHVSRDDVEAGFIEFRDLLGHCRFRDCKHDREPGCALLQALEDGRIMPQRMASYRHILASMP 6h4o A 2.25 BS03 FQH A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 H276 Y125 Y162 F170 H173 E175 K191 W193 K226 H261 G170 Y177 H188 E190 H276 S288 G155 Y162 H173 E175 H261 S273 1.14.11.66,1.14.11.69 ic50=0.128uM remove_due_to_license_issue IC50=128nM O75164 31158747 403 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4p A 2.19 BS03 FQ5 A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 H276 Y127 Y172 F180 H183 E185 K201 W203 K236 H271 G170 Y177 H188 E190 H276 S288 G165 Y172 H183 E185 H271 S283 1.14.11.66,1.14.11.69 Ki=0.003uM remove_due_to_license_issue IC50=102nM, EC50=8500nM, Ki=3.0nM O75164 31158747 403 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4q A 2.31 BS03 FO2 A 1 Y132 Y177 F185 H188 E190 D191 K206 W208 K241 H276 Y125 Y163 F171 H174 E176 D177 K192 W194 K227 H262 G170 Y177 H188 E190 H276 S288 G156 Y163 H174 E176 H262 S274 1.14.11.66,1.14.11.69 ic50=2.06uM remove_due_to_license_issue IC50=2060nM O75164 31158747 403 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEF 6h4r A 2.14 BS03 FQB A 1 Y132 Y177 F185 H188 E190 K206 W208 H276 Y127 Y164 F172 H175 E177 K193 W195 H263 G170 Y177 H188 E190 H276 S288 G157 Y164 H175 E177 H263 S275 1.14.11.66,1.14.11.69 Ki=0.004nM remove_due_to_license_issue Ki=4.0nM, IC50=93nM O75164 31158747 403 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4s A 2.45 BS03 FQE A 1 Y132 D135 Y177 F185 H188 E190 K206 W208 H276 Y125 D128 Y161 F169 H172 E174 K190 W192 H260 G170 Y177 H188 E190 H276 S288 G154 Y161 H172 E174 H260 S272 1.14.11.66,1.14.11.69 Ki=0.002uM remove_due_to_license_issue IC50=60nM, EC50=30300nM, Ki=2.0nM O75164 31158747 403 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4t A 2.38 BS03 FOW A 1 Y132 D135 Y175 Y177 F185 H188 E190 K206 W208 K241 H276 D311 Y126 D129 Y161 Y163 F171 H174 E176 K192 W194 K227 H262 D297 G170 Y177 H188 E190 H276 S288 G156 Y163 H174 E176 H262 S274 1.14.11.66,1.14.11.69 Ki=0.004uM remove_due_to_license_issue IC50=423nM, EC50=4700nM, Ki=4.0nM O75164 31158747 403 TLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4u A 2.21 BS03 FO2 A 1 Y132 D135 Y177 F185 H188 E190 K206 W208 H276 Y125 D128 Y166 F174 H177 E179 K195 W197 H265 G170 Y177 H188 E190 H276 S288 G159 Y166 H177 E179 H265 S277 1.14.11.66,1.14.11.69 remove_due_to_license_issue IC50=2060nM O75164 31158747 403 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEF 6h4v A 2.15 BS03 FQN A 1 Y132 Y177 F185 H188 E190 K206 W208 H276 Y127 Y164 F172 H175 E177 K193 W195 H263 G170 Y177 H188 E190 H276 S288 G157 Y164 H175 E177 H263 S275 1.14.11.66,1.14.11.69 ic50=0.613uM remove_due_to_license_issue IC50=613nM O75164 31158747 403 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4w A 2.81 BS03 FQQ A 1 Y132 D135 Y175 Y177 F185 H188 E190 K206 W208 H276 Y124 D127 Y160 Y162 F170 H173 E175 K191 W193 H261 G170 Y177 H188 E190 H276 S288 G155 Y162 H173 E175 H261 S273 1.14.11.66,1.14.11.69 remove_due_to_license_issue EC50=5900nM, IC50=107nM, Ki=5.0nM O75164 31158747 403 NPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLK 6h4x A 2.34 BS03 FNQ A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 Y127 Y165 F173 H176 E178 K194 W196 K229 G170 Y177 H188 E190 H276 S288 G158 Y165 H176 E178 H264 S276 1.14.11.66,1.14.11.69 ic50=0.131uM remove_due_to_license_issue IC50=131nM O75164 31158747 403 ETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFL 6h4y A 2.38 BS03 FO8 A 1 Y132 Y177 F185 H188 E190 K206 W208 K241 H276 Y125 Y162 F170 H173 E175 K191 W193 K226 H261 G170 Y177 H188 E190 H276 S288 G155 Y162 H173 E175 H261 S273 1.14.11.66,1.14.11.69 ic50=0.077uM remove_due_to_license_issue IC50=77nM O75164 31158747 403 LNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEF 6h4z A 2.3 BS05 FQ5 A 1 Y425 D428 C480 W486 Y488 F496 H499 E501 K517 W519 H587 Y129 D132 C183 W189 Y191 F199 H202 E204 K220 W222 H290 G481 Y488 H499 E501 H587 A599 G184 Y191 H202 E204 H290 A302 1.14.11.67 Ki=0.002uM remove_due_to_license_issue EC50=600nM, Ki=2.0nM, IC50=23nM Q9UGL1 31158747 805 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKARDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAESY 6h4z A 2.3 BS06 FQ5 A 2 P33 Q58 T59 Y525 P10 Q35 T36 Y228 G481 Y488 H499 E501 H587 A599 G184 Y191 H202 E204 H290 A302 1.14.11.67 Ki=0.002uM remove_due_to_license_issue EC50=600nM, Ki=2.0nM, IC50=23nM Q9UGL1 31158747 806 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKARDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAESY 6h50 A 2.19 BS05 FO2 A 1 W486 Y488 F496 H499 E501 K517 W519 H587 W188 Y190 F198 H201 E203 K219 W221 H289 G481 Y488 H499 E501 H587 A599 G183 Y190 H201 E203 H289 A301 1.14.11.67 ic50=0.156uM remove_due_to_license_issue IC50=156nM Q9UGL1 31158747 809 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKRDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAES 6h51 A 2.21 BS05 FQK A 1 Y425 W486 Y488 F496 H499 E501 K517 W519 H587 Y127 W187 Y189 F197 H200 E202 K218 W220 H285 G481 Y488 H499 E501 H587 A599 G182 Y189 H200 E202 H285 A297 1.14.11.67 Ki=0.016uM remove_due_to_license_issue IC50=134nM, EC50=26400nM, Ki=16nM Q9UGL1 31158747 816 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRARDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAES 6h52 A 2.14 BS05 FQN A 1 Y425 W486 Y488 F496 H499 E501 K517 W519 H587 Y128 W188 Y190 F198 H201 E203 K219 W221 H289 G481 Y488 H499 E501 H587 A599 G183 Y190 H201 E203 H289 A301 1.14.11.67 ic50=0.068uM remove_due_to_license_issue IC50=68nM Q9UGL1 31158747 813 SMFLPPPECPVFEPSWEEFADPFAFIHKIRPIAEQTGICKVRPPPDWQPPFACDVDKLHFTPRIQRLNELEAQTRVKRDYTLRTFGEMADAFKSDYFNMPVHMVPTELVEKEFWRLVSTIEEDVTVEYGADIASKEFGSGFPVRDGIKLSPEEEEYLDSGWNLNNMPVMEQSVLAHITADICGMKLPWLYVGMCFSSFCWHIEDHWSYSINYLHWGEPKTWYGVPGYAAEQLENVMKKLAPELFVSQPDLLHQLVTIMNPNTLMTHEVPVYRTNQCAGEFVITFPRAYHSGFNQGFNFAEAVNFCTVDWLPLGRQCVEHYRLLHRYCVFSHDEMICKMASKADVLDVVVASTVQKDMAIMIEDEKALRETVRKLGVIDSERMDFELLPDDERQCVKCKTTCFMSAISCSCKPGLLVCLHHVKELCSCPPYKYKLRYRYTLDDLYPMMNALKLRAESY 6h5w A 1.37 BS03 FT8 A 1 Q281 H353 A354 S355 E384 H387 F457 K511 H513 Y520 Y523 Q242 H314 A315 S316 E345 H348 F418 K472 H474 Y481 Y484 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H474 Y484 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=0.015000nM, IC50=0.100000nM P12821 30372620 710 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPNS 6h5w A 1.37 BS04 FT8 A 2 D121 E123 R124 W220 M223 E403 R522 D82 E84 R85 W181 M184 E364 R483 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H474 Y484 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=0.015000nM, IC50=0.100000nM P12821 30372620 711 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPNS 6h5w A 1.37 BS05 FT8 A 3 N85 E123 V518 N46 E84 V479 H353 A354 H383 E384 H387 E411 H513 Y523 H314 A315 H344 E345 H348 E372 H474 Y484 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=0.015000nM, IC50=0.100000nM P12821 30372620 712 DEAEASKFVEEYDRTSQVVWNEYAGANWNYNTNITTETSKILLQKNMQIAQHTLKYGTQARKFDVNQLQNTTIKRIIKKVQDLERAALPAQELEEYNKILLDMETTYSVATVCHPQGSCLQLEPDLTNVMATSRKYEDLLWAWEGWRDKAGRAILQFYPKYVELINQAARLNGYVDAGDSWRSMYETPSLEQDLERLFQELQPLYLNLHAYVRRALHRHYGAQHINLEGPIPAHLLGNMWAQTWSNIYDLVVPFPSAPSMDTTEAMLKQGWTPRRMFKEADDFFTSLGLLPVPPEFWQKSMLEKPTDGREVVCHASAWDFYNGKDFRIKQCTTVNLEDLVVAHHEMGHIQYFMQYKDLPVALREGANPGFHEAIGDVLALSVSTPKHLHSLNLLSSEGGSDEHDINFLMKMALDKIAFIPFSYLVDQWRWRVFDGSITKENYNQEWWSLRLKYQGLCPPVPRTQGDFDPGAKFHIPSSVPYIRYFVSFIIQFQFHEALCQAAGHTGPLHKCDIYQSKEAGQRLATAMKLGFSRPWPEAMQLITGQPQMSASAMLSYFKPLLDWLRTENELHGEKLGWPQYNWTPNS 6h5x A 1.8 BS03 FT8 A 1 Q259 H331 A332 S333 E362 H365 F435 K489 H491 Y498 Y501 Q256 H328 A329 S330 E359 H362 F432 K486 H488 Y495 Y498 H331 A332 H361 E362 H365 E389 H491 Y501 H328 A329 H358 E359 H362 E386 H488 Y498 3.4.15.1 0006508,0008237,0008241,0016020 remove_due_to_license_issue Ki=0.015000nM, IC50=0.100000nM P12821 30372620 709 LDPGLQPGQFSADEAGAQLFAQSYQSSAEQVLFQSVAASWAHDTNITAENARRQEEAALLSQEFAEAWGQKAKELYEPIWQQFTDPQLRRIIGAVRTLGSANLPLAKRQQYNALLSQMSRIYSTAKVCLPATCWSLDPDLTNILASSRSYAMLLFAWEGWHNAAGIPLKPLYEDFTALSNEAYKQDGFTDTGAYWRSWYNSPTFEDDLEHLYQQLEPLYLNLHAFVRRALHRRYGDRYINLRGPIPAHLLGDMWAQSWENIYDMVVPFPDKPNLDVTSTMLQQGWQATHMFRVAEEFFTSLELSPMPPEFWEGSMLEKPADGREVVCHASAWDFYNRKDFRIKQCTRVTMDQLSTVHHEMGHIQYYLQYKDLPVSLRRGANPGFHEAIGDVLALSVSTPEHLHKIGLLDRVTNDTESDINYLLKMALEKIAFLPFGYLVDQWRWGVFSGRTPPSRYNFDWWYLRTKYQGICPPVTRNETHFDAGAKFHVPNVTPYIRYFVSFVLQFQFHEALCKEAGYEGPLHQCDIYRSTKAGAKLRKVLRAGSSRPWQEVLKDMVGLDALDAQPLLKYFQLVTQWLQEQNQQNGEVLGWPEYQWHPPLPDNYPEGI 6h75 A 1.45 BS01 SLB A 1 N10 D49 E67 R127 R147 F170 N187 Q214 N10 D49 E67 R127 R147 F170 N187 Q214 ? 0030288,0042597,0055085 Kd=42uM remove_due_to_license_issue P44542 31518131 401 ADYDLKFGMNNGTSSNEYKAAEMFAKEVKEKSQGKIEISLYPSSQLGDDRAMLKQLKDGSLDFTFAESARFQLFYPEAAVFALPYVISNYNVAQKALFDTEFGKDLIKKMDKDLGVTLLSQAYNGTRQTTSNRAINSIADMKGLKLRVPNAATNLAYAKYVGASPTPMAFSEVYLALQTNAVDGQENPLAAVQAQKFYEVQKFLAMTNHILNDQLYLVSNETYKELPEDLQKVVKDAAENAAKYHTKLFVDGEKDLVTFFEKQGVKITHPDLVPFKESMKPYYAEFVKQTGQKGESALKQIEAINPHH 6h76 A 1.5 BS01 SLB A 1 N10 D49 E67 R70 R127 R147 F170 N187 Q214 N10 D49 E67 R70 R127 R147 F170 N187 Q214 ? 0030288,0042597,0055085 Kd=0.03uM remove_due_to_license_issue P44542 31518131 401 ADYDLKFGMNAGTSSNEYKAAEMFAKEVKEKSQGKIEISLYPSSQLGDDRAMLKQLKDGSLDFTFAESARFQLFYPEAAVFALPYVISNYNVAQKALFDTEFGKDLIKKMDKDLGVTLLSQAYNGTRQTTSNRAINSIADMKGLKLRVPNAATNLAYAKYVGASPTPMAFSEVYLALQTNAVDGQENPLAAVQAQKFYEVQKFLAMTNHILNDQLYLVSNETYKELPEDLQKVVKDAAENAAKYHTKLFVDGEKDLVTFFEKQGVKITHPDLVPFKESMKPYYAEFVKQTGQKGESALKQIEAINPHH 6h77 A 2.1 BS01 ATP A 1 G80 G82 G83 D104 Y105 D106 N112 R115 K127 N150 D183 N184 G45 G47 G48 D69 Y70 D71 N77 R80 K92 N115 D148 N149 ? 0008641 remove_due_to_license_issue Q9GZZ9 30412706 401 GRVRIEKMSSEVVDSNPYSRLMALKRMGIVSDYEKIRTFAVAIVGVGGVGSVTAEMLTRCGIGKLLLFDYDKVELANMNRLFFQPHQAGLSKVQAAEHTLRNINPDVLFEVHNYNITTVENFQHFMDRISNGGLEEGKPVDLVLSCVDNFEARMTINTACNELGQTWMESGVSENAVSGHIQLIIPGESACFACAPPLVVAANIDEKTLKREGVCAASLPTTMGVVAGILVQNVLKFLLNFGTVSFYLGYNAMQDFFPTMSMKPNPQCDDRNCRKQQEEYKKKVAAEEIIHEDNEWGIELV 6h77 B 2.1 BS01 ATP B 1 G80 G82 G83 D104 Y105 D106 N112 R115 K127 N150 I151 D183 N184 G45 G47 G48 D69 Y70 D71 N77 R80 K92 N115 I116 D148 N149 ? 0008641 remove_due_to_license_issue Q9GZZ9 30412706 401 GRVRIEKMSSEVVDSNPYSRLMALKRMGIVSDYEKIRTFAVAIVGVGGVGSVTAEMLTRCGIGKLLLFDYDKVELANMNRLFFQPHQAGLSKVQAAEHTLRNINPDVLFEVHNYNITTVENFQHFMDRISNGGLEEGKPVDLVLSCVDNFEARMTINTACNELGQTWMESGVSENAVSGHIQLIIPGESACFACAPPLVVAANIDEKTLKREGVCAASLPTTMGVVAGILVQNVLKFLLNFGTVSFYLGYNAMQDFFPTMSMKPNPQCDDRNCRKQQEEYKKKVAALPEIIHEDNEWGIELV 6h78 A 2.7 BS01 ATP A 1 G80 G82 G83 D104 Y105 D106 N112 R115 K127 I151 D183 N184 G45 G47 G48 D69 Y70 D71 N77 R80 K92 I116 D148 N149 ? 0008641 remove_due_to_license_issue Q9GZZ9 30412706 401 GRVRIEKMSSEVVDSNPYSRLMALKRMGIVSDYEKIRTFAVAIVGVGGVGSVTAEMLTRCGIGKLLLFDYDKVELANMNRLFFQPHQAGLSKVQAAEHTLRNINPDVLFEVHNYNITTVENFQHFMDRISNGGLEEGKPVDLVLSCVDNFEARMTINTACNELGQTWMESGVSENAVSGHIQLIIPGESACFACAPPLVVAANIDEKTGVCAASLPTTMGVVAGILVQNVLKFLLNFGTVSFYLGYNAMQDFFPTMSMKPNPQCDDRNCRKQQEEYKKKVAAL 6h78 B 2.7 BS01 ATP B 1 G80 G82 G83 D104 Y105 D106 N112 R115 K127 N150 I151 V182 D183 N184 G45 G47 G48 D69 Y70 D71 N77 R80 K92 N115 I116 V147 D148 N149 ? 0008641 remove_due_to_license_issue Q9GZZ9 30412706 401 GRVRIEKMSSEVVDSNPYSRLMALKRMGIVSDYEKIRTFAVAIVGVGGVGSVTAEMLTRCGIGKLLLFDYDKVELANMNRLFFQPHQAGLSKVQAAEHTLRNINPDVLFEVHNYNITTVENFQHFMDRISNGGLEEGKPVDLVLSCVDNFEARMTINTACNELGQTWMESGVSENAVSGHIQLIIPGESACFACAPPLVVAANEGVCAASLPTTMGVVAGILVQNVLKFLLNFGTVSFYLGYNAMQDFFPTMSMKPNPQCDDRNCRKQQEEYKKKVAA 6h7d A 2.4 BS01 BGC A 1 Q177 I184 Q295 N301 N332 G406 W410 Q157 I164 Q275 N281 N312 G386 W390 ? 0005354,0005886,0008645,0009679,0015144,0015145,0015293,0015578,0015749,0015757,0015761,0016020,0022857,0055055,0055085,0071333 Kd=3.2uM remove_due_to_license_issue Q9LT15 30679446 600 VTAFVIMTCIVAAMGGLLFGYDLGISGGVTSMEEFLTKFFPQVESQMKKAKHDTAYCKFDNQMLQLFTSSLYLAALVASFMASVITRKHGRKVSMFIGGLAFLIGALFNAFAVNVSMLIIGRLLLGVGVGFANQSTPVYLSEMAPAKIRGALNIGFQMAITIGILVANLINYGTSKMAQHGWRVSLGLAAVPAVVMVIGSFILPDTPNSMLERGKNEEAKQMLKKIRGADNVDHEFQDLIDAVEAAKKVENPWKNIMESKYRPALIFCSAIPFFQQITGINVIMFYAPVLFKTLGFGDDAALMSAVITGVVNMLSTFVSIYAVDRYGRRLLFLEGGIQMFICQLLVGSFIGARFGTSGTGTLTPATADWILAFICVYVAGFAWSWGPLGWLVPSEICPLEIRPAGQAINVSVNMFFTFLIGQFFLTMLCHMKFGLFYFFASMVAIMTVFIYFLLPETKGVPIEEMGRVWKQHWFWKKYIPEDAIIGG 6h7f A 2.26 BS01 FV8 A 1 W97 R253 Y312 Y314 L336 Y378 W65 R221 Y280 Y282 L304 Y346 ? 0006826,0009279,0015343,0015344,0015891,0033214,0038023,0044718 remove_due_to_license_issue Q76HJ9 30558715 802 DTYAGGQVATSSNVGFLGSKKFLDTPFNTISYTDKYIEDKQAKDITEVIAATDPSIYTNGASGGWSENYYIRGYASSTNDMSMNGLFGITPFYRTSPEMFGRVEVLKGPSALLNGMPPAGSVGGTVNLVTKYAADEPFARLTTTYMSDAQFGGHVDVGRRFGENKEFGVRINGMYRDGDAAVNDQSKESRLFSLGLDWQGENARVFVDAYDALDHVDGVTRGVNVSTAVGIPKPPKADTLLSPDWGSVETKDKGAMIRGEYDFSDQLMAYAAYGQSTTEYKYNGASAGTITSSTGTLSSTLGQLAFDVDKKSADAGFKGKFETGSVKHQWVANATYYNHTQDDYGYRIIPGFSDPVITNIYDPNPNWGPKPEFTPPFLFHSTLSTSSFGLADTLSFAQDKVQLTLGLRHQTVKATSSVNTLPENAKSATTPGVALLIKATDKISVYANYIEGLTKGDQAPATASNPGEIFPPQKTKQQELGLKVDLGTFAHTLSAFEITKPSSYLDPSKLVNNLPTFVSDGEQRNRGIEWSFFGSPIEHVRLMGGFTYLDPELTKTKSGGNDGHTAVAVPKNQAKLGAEWDTQVAQGTLTLSGNINAVSKQYINAENTLSVPGRTLLDVGARYSTKVEDHPVTFRANIYNLTNKAYWAQPQLTNLALGAPRTYMLSVSYDF 6h7j A 2.8 BS01 5FW A 1 W117 D121 V122 S211 S215 F306 F307 N329 Y333 W78 D82 V83 S172 S176 F239 F240 N262 Y266 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 31072904 401 AAKVMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVYLRVYREAKEQIRKIDRASKRKTSRVMAMKEHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLL 6h7l A 2.7 BS05 Y00 A 1 G98 W117 T118 D121 V122 F201 S211 S215 F306 V326 N329 W330 G59 W78 T79 D82 V83 F162 S172 S176 F239 V259 N262 W263 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 31072904 406 AAKVMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVYLRVYREAKEQIRKIDRASKRKTSRVMAMKEHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLLA 6h7m A 2.76 BS04 68H A 1 D121 V122 F201 S211 S215 F306 F307 N329 D82 V83 F162 S172 S176 F239 F240 N262 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 31072904 504 AAKVMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVYLRVYREAKEQIRKIDRASKRKTSRVMAMKEHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLLA 6h7n A 2.5 BS01 FVK A 1 G98 V102 W117 D121 V122 S211 S215 F306 F307 V326 N329 W330 Y333 G59 V63 W78 D82 V83 S172 S176 F239 F240 V259 N262 W263 Y266 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 401 AAKVMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVYLRVYREAKEQIRKIDRASKRKTSRVMAMKEHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLLA 6h7o A 2.8 BS01 P32 A 1 D121 V122 F201 T203 S211 S215 F306 F307 N310 N329 Y333 D82 V83 F162 T164 S172 S176 F239 F240 N243 N262 Y266 ? 0004930,0004935,0004940,0007186,0007189,0016020,0045823 remove_due_to_license_issue P07700 31072904 401 AAKVMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVYLRVYREAKEQIRKIDRASKRKTSRVMAMKEHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLL 6h7y A 1.81 BS05 FVZ A 1 K207 R210 E424 L428 G518 N519 R536 F546 S547 G548 Y552 H553 K699 Y700 K153 R156 E370 L374 G464 N465 R482 F492 S493 G494 Y498 H499 K645 Y646 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.35nM remove_due_to_license_issue IC50=0.350000nM Q04609 30429952 833 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFDKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6h7z A 2.0 BS04 FVW A 1 G206 R210 E424 L428 G518 N519 R534 R536 S547 Y552 H553 K699 Y700 G152 R156 E370 L374 G464 N465 R480 R482 S493 Y498 H499 K644 Y645 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.075nM remove_due_to_license_issue IC50=0.075000nM Q04609 30429952 832 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFKSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6h8q A 3.631 BS01 dna F 0 H427 S507 N509 H282 S354 N356 ? 0000775,0000785,0003682,0005515,0005634,0005694,0005737,0005829,0006473,0007059,0007062,0007064,0008278,0030892,0030893,0034087,0034089,0051301 remove_due_to_license_issue P40541 30109982 1 ~ 19 TELFDILSTSEDVSIEELLREWLETYSENRDKFLQEFINLLLNCCGSVARVEDHDVHSNESSNETIGEIQLLFQRQKLHEFYLLISKENKKRKNFKMGPLYQNFAEFMTKLLEVANDLQLLYVGNLVLDLLTWLSSFSVCKIRCFRYISTLTLYLFQDYLTQQAVNLEKNYLAKLSKQLSLEEKKKRPNNKTLEKLESTIAETQGSKVVIDSIIDNIVKLCFVHRYKDVSDLIRSESMLHLSIWIKNYPEYFLKVTFLKYFGWLLSDNSVSVRLQVTKILPHLIIQNSAIRQVFERFKTKILEVAIRDVNLDVRIHSIQVLTEASSLGYLDDSEILIISSLMFDEEFDPFKTSSFNKRSKFLSTVAKFLARVIKEKFDEFIKTHEDLPKEVDGLEVGPVVQVGIFIKILNDSLIYHLKDCAEVDSRTKIRMLTQAAEFLSPYISTHLKTICNLLISDTESNELIPIDRNSTILYLNVFHGLCAGANNPKIQTKDSVKEIVLPLFYDLLNAASIESADILCPLLESFITFSLDDWISIGYETELKKITDKTIKAFMDSTIGNSKVDMKYDIFAKFIHHIHHFEKKELQEKFLNQIATLKIHLKKFLQEKMDPNNSRDDYKDLTCSLYELYINKLTILGRDYPIEVDEELLQLFLNNFVSRIPIMFQDFDDSTAQEINFKMLVLLATWNLEKWREIIEKVRDYEISKDLRSVWKPIAAIIGRLNTLVISLAATNETFENINSLFYLKWSACTSLMDIIVAIKIFELKLPADATTWRYSMSEQFPFYLHDNASKVLLKIFLYLESLFAKQVDVQLERVADEDANLNDLPETGFFENIETEFLLFTVKLKGLMKLNILDERFASRVALNKEKLGPLFKKIVDD 6h8q B 3.631 BS02 dna C 0 H427 S507 H282 S354 ? 0000775,0000785,0003682,0005515,0005634,0005694,0005737,0005829,0006473,0007059,0007062,0007064,0008278,0030892,0030893,0034087,0034089,0051301 remove_due_to_license_issue P40541 30109982 1 ~ 19 TELFDILSTSEDVSIEELLREWLETYSENRDKFLQEFINLLLNCCGSVARVEDHDVHSNESSNETIGEIQLLFQRQKLHEFYLLISKENKKRKNFKMGPLYQNFAEFMTKLLEVANDLQLLYVGNLVLDLLTWLSSFSVCKIRCFRYISTLTLYLFQDYLTQQAVNLEKNYLAKLSKQLSLEEKKKRPNNKTLEKLESTIAETQGSKVVIDSIIDNIVKLCFVHRYKDVSDLIRSESMLHLSIWIKNYPEYFLKVTFLKYFGWLLSDNSVSVRLQVTKILPHLIIQNSAIRQVFERFKTKILEVAIRDVNLDVRIHSIQVLTEASSLGYLDDSEILIISSLMFDEEFDPFKTSSFNKRSKFLSTVAKFLARVIKEKFDEFIKTHEDLPKEVDGLEVGPVVQVGIFIKILNDSLIYHLKDCAEVDSRTKIRMLTQAAEFLSPYISTHLKTICNLLISDTESNELIPIDRNSTILYLNVFHGLCAGANNPKIQTKDSVKEIVLPLFYDLLNAASIESADILCPLLESFITFSLDDWISIGYETELKKITDKTIKAFMDSTIGNSKVDMKYDIFAKFIHHIHHFEKKELQEKFLNQIATLKIHLKKFLQEKMDPNNSRDDYKDLTCSLYELYINKLTILGRDYPIEVDEELLQLFLNNFVSRIPIMFQDFDDSTAQEINFKMLVLLATWNLEKWREIIEKVRKDLRSVWKPIAAIIGRLNTLVISLAATNETFENINSLFYLKWSACTSLMDIIVAIKIFELKLPADATTWRYSMSEQFPFYLHDNASKVLLKIFLYLESLFAKQVDVQLERVADEDANLNDLPETGFFENIETEFLLFTVKLKGLMKLNILDERFASRVALNKEKLGPLFKKIVD 6h8s A 1.771 BS01 FSZ A 1 E341 V344 Y345 E455 A458 C465 I468 E93 V96 Y97 E207 A210 C217 I220 3.1.3.48 0004725,0006470,0016311 remove_due_to_license_issue P54830 30207464 601 SAHEYLLSASRVLRAEELHEKALDPFLLQAEFFEIPMNFVDPKEYDIPGLVRKNRYKTILPNPHSRVRLTSPDPEDPLSSYINANYIRGYSGEEKVYIATQGPIVSTVADFWRMVWQERTPIIVMITNIEEMNEKCTEYWPEEQVVHDGVEITVQKVIHTEDYRLRLISLRRGTEERTLKHYWFTSWPDQKTPDRAPPLLHLVREVEEAAQQEGPHCSPIIVHCSAGIGRTGCFIATSICCQQLRREGVVDILKTTCQLRQDRGGMIQTCEQYQFVHHAMSLYEKQLSHQS 6h96 A 1.55 BS01 FWE A 1 W27 L60 L71 N75 H78 I95 T99 L130 M131 W133 P134 V137 W162 R181 M184 G193 T194 W28 L61 L72 N76 H79 I96 T100 L131 M132 W134 P135 V138 W163 R182 M185 G194 T195 ? remove_due_to_license_issue Q8KRS7 30422653 301 KMYDRWFSQQELQVLPFAEQDEQRNQTWLELVGEAQQLMDERCPADEPRAIALATRWMEQLEQDTAGRPEFLTRLNEMHAAEPQMREQTGVTPEMIDFITRAFAESKLAIWARYLNDEELAFTRQHYFDRLMEWPALVADLHRACREKRDPASPGGQQLAQRWLALFQSYAGKDAQTQQKFRYAMEQEPHLMKGTWMTSEVLSWLQQAIGVMM 6h9b A 2.75 BS02 FWH B 1 A180 V181 A173 V174 ? 0000226,0000793,0001764,0001964,0005200,0005525,0005737,0005829,0005856,0005874,0005879,0005881,0005886,0006886,0007017,0007098,0007224,0007613,0007626,0008344,0008542,0009612,0010001,0010467,0015630,0016787,0021542,0021696,0021766,0021859,0021987,0022008,0030182,0030317,0030534,0031594,0034612,0035641,0036126,0036464,0042802,0044877,0045202,0046785,0046872,0046982,0048853,0048873,0050807,0050808,0051402,0055037,0061744,0071277,0072384,0140058,1902065 remove_due_to_license_issue D0VWZ0 30525602 505 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVD 6h9b B 2.75 BS02 FWH B 1 C241 A250 L255 N258 M259 A316 T317 N349 N350 K352 A354 C239 A248 L253 N256 M257 A314 T315 N347 N348 K350 A352 ? 0003924,0005200,0005525,0005737,0005856,0005874,0007010,0007017,0046872 remove_due_to_license_issue D0VWY9 30525602 505 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVATIFRGRMSMKEVDEQMLNIQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSSTFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDATAD 6h9v A 1.52 BS01 MFU A 1 T344 R345 D374 T123 R124 D153 ? remove_due_to_license_issue B5BTR7 30899001 601 TGSKPFTVPILTVEEMTNSRFPIPLEKLFTGPSGAFVVQPQNGRCTTDGVLLGTTQLSPVNICTFRGDVTHIAGSRNYTMNLASLNWNNYDPTEEIPAPLGTPDFVGKIQGLLTQTTKGDGSTRGHKATVYTGSAPFTPKLGSVQFSTDTENDFETHQNTKFTPVGVIQDGSTTHRNEPQQWVLPSYSGRNVHNVHLAPAVAPTFPGEQLLFFRSTMPGCSGYPNMDLDCLLPQEWVQHFYQEAAPAQSDVALLRFVNPDTGRVLFECKLHKSGYVTVAHTGQHDLVIPPNGYFRFDSWVNQFYTLAPM 6h9v B 1.52 BS01 MFU B 1 T344 R345 D374 T121 R122 D149 ? remove_due_to_license_issue B5BTR7 30899001 601 SKPFTVPILTVEEMTNSRFPIPLEKLFTGPSGAFVVQPQNGRCTTDGVLLGTTQLSPVNICTFRGDVTHIAGSRNYTMNLASLNWNNYDPTEEIPAPLGTPDFVGKIQGLLTQTTKGDGSTRGHKATVYTGSAPFTPKLGSVQFSTDTDFETHQNTKFTPVGVIQDTTHRNEPQQWVLPSYSGRNVHNVHLAPAVAPTFPGEQLLFFRSTMPGCSGYPNMDLDCLLPQEWVQHFYQEAAPAQSDVALLRFVNPDTGRVLFECKLHKSGYVTVAHTGQHDLVIPPNGYFRFDSWVNQFYTLAPM 6h9x A 2.1 BS01 SSA A 1 T237 E239 R268 E270 I282 R283 M284 F287 K289 E291 E355 I356 S357 S358 N389 S391 A394 R397 T235 E237 R266 E268 I280 R281 M282 F285 K287 E289 E353 I354 S355 S356 N387 S389 A392 R395 6.1.1.11 0000166,0004812,0004828,0005524,0005737,0006412,0006418,0006434,0016260,0046872 remove_due_to_license_issue W9BNU9 31048140 501 MLDPNLLRTEPDAVAEKLARRGFKLDVDKLRALEERRKVLQVQTENLQAERNSRSKSIGQAKARDIEPLRLEVNKLGEQLDAAKSELETLLAEIRDIALAIPNIPHDDVPVGRDENDNVEVSRWGTPRQFDFEVRDHVTLGEMHGGLDFAAAVKLTGSRFVVMKGQLARLHRALAQFMLDLHTEQHGYSENYVPYLVNQDTLYGTGQLPKFAGDLFHTRPLEEEADSSNYALIPTAEVPLTNLVRDEIIDEDDLPIKMTAHTPCFRSEAGSYGRDTRGLIRMHQFDKVEMVQIVRPEDSMAALEEMTGHAEKVLQLLGLPYRKVALCTGDMGFSACKTYDLEVWVPAQNTYREISSCSNVWDFQARRMQARCRSKSDKKTRLVHTLNGSGLAVGRTLVALMENYQQADGRIEIPEVLRPYMRGLEYIG 6ha4 A 1.33 BS01 T3Y A 1 K30 F31 D32 K30 F31 D32 ? 0050832 Kd=107uM remove_due_to_license_issue B6HWK0 30867921 202 AKYTGKCTKSKNECKYKNDAGKDTFIKCPKFDNKKCTKDNNKCTVDTYNNAVDCD 6hah A 1.45 BS01 FWQ A 1 K27 C28 P29 K30 F31 K27 C28 P29 K30 F31 ? 0050832 Kd=15.4uM remove_due_to_license_issue B6HWK0 30867921 101 AKYTGKCTKSKNECKYKNDAGKDTFIKCPKFDNKKCTKDNNKCTVDTYNNAVDCD 6hai A 2.2 BS01 FWW A 1 F16 L60 N75 H78 T88 I95 T99 L130 W133 P134 V137 W162 R181 M184 M191 G193 T194 M196 L201 Q205 F16 L60 N75 H78 T88 I95 T99 L130 W133 P134 V137 W162 R181 M184 M191 G193 T194 M196 L201 Q205 ? remove_due_to_license_issue Q8KRS7 30422653 302 MYDRWFSQQELQVLPFAEQDEQRNQTWLELVGEAQQLMDERCPADEPRAIALATRWMEQLEQDTAGRPEFLTRLNEMHAAEPQMREQTGVTPEMIDFITRAFAESKLAIWARYLNDEELAFTRQHYFDRLAEWPALVADLHRACREKRDPASPGGQQLAQRWLALFQSYAGKDAQTQQKFRYAMEQEPHLMKGTWMTSEVLSWLQQAIGVMM 6haj B 1.5 BS01 EVB B 1 K27 P29 K30 K27 P29 K30 ? 0050832 Kd=10.6uM remove_due_to_license_issue B6HWK0 30867921 101 AKYTGKCTKSKNECKYKNDAGKDTFIKCPKFDNKKCTKDNNKCTVDTYNNAVDCD 6hax A 2.35 BS01 FWZ B 1 V1408 F1409 L1412 L1418 Y1421 A1460 F1463 N1464 I1470 V33 F34 L37 L43 Y46 A85 F88 N89 I95 3.6.4.- 0006338,0016586 remove_due_to_license_issue P51531 31178587 301 LSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNHKYRSLGDLEKDVMLLCHNAQTFNLEGSQIYEDSIVLQSVFKSARQKIAK 6hax B 2.35 BS01 FWZ B 1 F76 W88 Y98 P99 R107 I109 H110 S111 Y112 H115 W117 F17 W29 Y39 P40 R48 I50 H51 S52 Y53 H56 W58 ? remove_due_to_license_issue P40337 31178587 301 RPVLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQERIAH 6hay A 2.24 BS01 FX8 B 1 V1408 F1409 L1412 L1418 Y1421 V1429 D1430 A1460 F1463 N1464 I1470 V35 F36 L39 L45 Y48 V56 D57 A87 F90 N91 I97 3.6.4.- 0006338,0016586 remove_due_to_license_issue P51531 31178587 301 EKLSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNHKYRSLGDLEKDVMLLCHNAQTFNLEGSQIYEDSIVLQSVFKSARQKIAKEEE 6hay B 2.24 BS01 FX8 B 1 W88 Y98 P99 R107 I109 H110 S111 Y112 H115 W117 W30 Y40 P41 R49 I51 H52 S53 Y54 H57 W59 ? remove_due_to_license_issue P40337 31178587 301 PRPVLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQERIAHQR 6haz A 1.31 BS01 FX5 A 1 V1408 F1409 L1412 Y1421 A1460 F1463 N1464 I1470 V31 F32 L35 Y44 A83 F86 N87 I93 3.6.4.- 0006338,0016586 remove_due_to_license_issue P51531 31178587 1501 PNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNHKYRSLGDLEKDVMLLCHNAQTFNLEGSQIYEDSIVLQSVFKSARQKIAK 6haz B 1.31 BS01 FX5 B 1 V1408 F1409 L1412 Y1421 A1460 F1463 N1464 I1470 V31 F32 L35 Y44 A83 F86 N87 I93 3.6.4.- 0006338,0016586 remove_due_to_license_issue P51531 31178587 1501 PNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNHKYRSLGDLEKDVMLLCHNAQTFNLEGSQIYEDSIVLQSVFKSARQKIAK 6hb4 A 3.05 BS01 dna B 0 L58 K62 L65 K69 T77 K139 R140 M143 K147 R157 Y162 Q179 L182 K183 K186 Y211 R232 R233 T234 K236 L15 K19 L22 K26 T34 K96 R97 M100 K104 R114 Y119 Q136 L139 K140 K143 Y168 R189 R190 T191 K193 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKKQRK 6hb4 A 3.05 BS02 dna C 0 Y57 T78 I81 R82 A85 W88 R89 K146 K147 K156 R157 R159 N163 A167 F170 P178 Y14 T35 I38 R39 A42 W45 R46 K103 K104 K113 R114 R116 N120 A124 F127 P135 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKKQRK 6hb4 A 3.05 BS03 dna F 0 K52 Y103 W107 K9 Y60 W64 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKKQRK 6hb4 D 3.05 BS01 dna C 0 K52 Y103 W107 K9 Y60 W64 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKK 6hb4 D 3.05 BS02 dna E 0 V54 L58 K62 T77 K139 R140 M143 K146 K147 R157 Y162 Q179 L182 K186 W189 Y211 R232 R233 V11 L15 K19 T34 K96 R97 M100 K103 K104 R114 Y119 Q136 L139 K143 W146 Y168 R189 R190 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKK 6hb4 D 3.05 BS03 dna F 0 Y57 T78 I81 R82 A85 W88 R89 R140 K156 R157 R159 N163 V166 A167 F170 P178 Y14 T35 I38 R39 A42 W45 R46 R97 K113 R114 R116 N120 V123 A124 F127 P135 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIKK 6hb4 G 3.05 BS01 dna H 0 K52 V54 L58 T77 R157 Y162 Q179 L182 K183 W189 Y211 R232 R233 T234 K9 V11 L15 T34 R114 Y119 Q136 L139 K140 W146 Y168 R189 R190 T191 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 6hb4 G 3.05 BS02 dna I 0 S56 Y57 T78 I81 R82 A85 W88 R89 M143 K147 K156 R157 R159 N163 A167 F170 P178 S13 Y14 T35 I38 R39 A42 W45 R46 M100 K104 K113 R114 R116 N120 A124 F127 P135 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 6hb4 G 3.05 BS03 dna L 0 Q100 Y103 W107 Q57 Y60 W64 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 6hb4 J 3.05 BS01 dna I 0 Y103 W107 Y60 W64 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 6hb4 J 3.05 BS02 dna K 0 K51 K52 V54 L58 K62 K69 K139 M143 R157 Y162 Q179 L182 K183 K186 W189 Y211 R232 K8 K9 V11 L15 K19 K26 K96 M100 R114 Y119 Q136 L139 K140 K143 W146 Y168 R189 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 6hb4 J 3.05 BS03 dna L 0 S55 Y57 T78 I81 R82 A85 W88 R89 K136 K139 R140 K146 K156 R157 R159 N163 V166 A167 P178 S12 Y14 T35 I38 R39 A42 W45 R46 K93 K96 R97 K103 K113 R114 R116 N120 V123 A124 P135 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRTIK 6hb5 A 1.88 BS01 YSC A 1 Y37 G39 D41 G50 H51 P54 D81 Y175 Q179 D182 G197 G198 D200 Q201 L227 Y33 G35 D37 G46 H47 P50 D77 Y171 Q175 D178 G193 G194 D196 Q197 L223 T43 H48 H51 K85 R89 Q179 D200 K235 K238 T239 T39 H44 H47 K81 R85 Q175 D196 K231 K234 T235 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0016020,0042803,0043039 remove_due_to_license_issue Ki=1484nM P0AGJ9 30995568 501 NLIKQLQERGLVAQVTDEEALAERLAQGPIALYCGFDPTADSLHLGHLVPLLCLKRFQQAGHKPVALVGGATGLIGDPSFKAAERKLNTEETVQEWVDKIRKQVAPFLDFDCGENSAIAANNYDWFGNMNVLTFLRDIGKHFSVNQMINKEAVKQRLNREDQGISFTEFSYNLLQGYDFACLNKQYGVVLQIGGSDQWGNITSGIDLTRRLHQNQVFGLTVPLITKADGTKFGKTEGGAVWLDPKKTSPYKFYQFWINTADADVYRFLKFFTFMSIEEINALEEEPRAQYVLAEQVTRLVHGEEGLQAAKRITECLFSGSLSALSEADFEQLAQDGVPMVEMEKGADLMQALVDSELQPSRGQARKTIASNAITINGEKQSDPEYFFKEEERLFGRFTLLRRGKKNYCLICWK 6hb6 A 1.92 BS01 YSU A 1 Y37 G39 D41 G50 H51 P54 D81 Y175 Q179 D182 G197 G198 D200 Q201 L227 Y33 G35 D37 G46 H47 P50 D77 Y171 Q175 D178 G193 G194 D196 Q197 L223 T43 H48 H51 K85 R89 Q179 D200 K235 K238 T39 H44 H47 K81 R85 Q175 D196 K231 K234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0016020,0042803,0043039 remove_due_to_license_issue Ki=43nM P0AGJ9 30995568 501 NLIKQLQERGLVAQVTDEEALAERLAQGPIALYCGFDPTADSLHLGHLVPLLCLKRFQQAGHKPVALVGGATGLIGDPSFKAAERKLNTEETVQEWVDKIRKQVAPFLDFDCGENSAIAANNYDWFGNMNVLTFLRDIGKHFSVNQMINKEAVKQRLNREDQGISFTEFSYNLLQGYDFACLNKQYGVVLQIGGSDQWGNITSGIDLTRRLHQNQVFGLTVPLITKADGTKFGKGAVWLDPKKTSPYKFYQFWINTADADVYRFLKFFTFMSIEEINALEEEDKAPRAQYVLAEQVTRLVHGEEGLQAAKRITECLFSGSLSALSEADFEQLAQDGVPMVEMEKGADLMQALVDSELQPSRGQARKTIASNAITINGEKQSDPEYFFKEEERLFGRFTLLRRGKKNYCLICWK 6hb7 A 1.9 BS01 Y3U A 1 Y37 G39 D41 G50 H51 P54 D81 Y175 Q179 D182 G197 G198 D200 Q201 L227 Y33 G35 D37 G46 H47 P50 D77 Y171 Q175 D178 G193 G194 D196 Q197 L223 T43 H48 H51 K85 R89 Q179 D200 K235 K238 T39 H44 H47 K81 R85 Q175 D196 K231 K234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0016020,0042803,0043039 remove_due_to_license_issue Ki=149nM P0AGJ9 30995568 501 NLIKQLQERGLVAQVTDEEALAERLAQGPIALYCGFDPTADSLHLGHLVPLLCLKRFQQAGHKPVALVGGATGLIGDPSFKAAERKLNTEETVQEWVDKIRKQVAPFLDFDCGENSAIAANNYDWFGNMNVLTFLRDIGKHFSVNQMINKEAVKQRLNREDQGISFTEFSYNLLQGYDFACLNKQYGVVLQIGGSDQWGNITSGIDLTRRLHQNQVFGLTVPLITKADGTKFGKAVWLDPKKTSPYKFYQFWINTADADVYRFLKFFTFMSIEEINALEEEDKNRAQYVLAEQVTRLVHGEEGLQAAKRITECLFSGSLSALSEADFEQLAQDGVPMVEMEKGADLMQALVDSELQPSRGQARKTIASNAITINGEKQSDPEYFFKEEERLFGRFTLLRRGKKNYCLICWK 6hbm A 2.76 BS06 AHR A 1 E28 S29 D105 R106 R163 N213 D241 E12 S13 D89 R90 R147 N197 D225 ? 0030246,0030313,0046872 remove_due_to_license_issue A0QT50 31006617 408 ALTLGFAQVGAESGWRTANTESIKSAAEEAGVNLKFADANGEQEKQISAIRSFIQQGVDVIAFSPVVRTGWDAVLQETKNAGIPVILTDRAVDTQDTDVYKTFIGADFIEEGRRAGQWVADQYASATGPVNIVQLEGTTGADPAIDRKTGFAEGISKNPNLKIVASQTGDFTRSGGKQVMEAFLKSTPQIDVVFAQNDDMGLGAMEAIEAAGKKPGTDIKIVAVDATHDGMQALADGKFNYIVECNPLLGPELMDLAKKVAAGEPVPERVVTPDEAFDQAQAKAALPNRQYKLAAALEHHHHHH 6hbn A 1.59 BS01 FXB A 1 G46 V53 V66 K68 N118 H160 M163 I174 D175 G44 V51 V64 K66 N116 H158 M161 I172 D173 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 31559376 406 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARMG 6hc3 A 3.1 BS01 dna B 0 K51 K52 V54 L58 K62 R140 K146 R157 Y162 Q179 L182 K186 Y211 R232 R233 T234 K9 K10 V12 L16 K20 R98 K104 R115 Y120 Q137 L140 K144 Y169 R190 R191 T192 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 A 3.1 BS02 dna C 0 S56 Y57 L58 S61 T78 I81 R82 A85 W88 R89 Q100 Y103 W107 K139 M143 K146 K147 K156 R157 R159 N163 A167 F170 P178 S14 Y15 L16 S19 T36 I39 R40 A43 W46 R47 Q58 Y61 W65 K97 M101 K104 K105 K114 R115 R117 N121 A125 F128 P136 ? remove_due_to_license_issue Q00059 31114891 2 ~ 23 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 D 3.1 BS01 dna E 0 K51 K52 V54 L58 K62 T77 I81 H137 M143 K147 R157 Y162 Q179 L182 K186 K190 Y211 R232 R233 T234 K9 K10 V12 L16 K20 T35 I39 H95 M101 K105 R115 Y120 Q137 L140 K144 K148 Y169 R190 R191 T192 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 D 3.1 BS02 dna F 0 S55 Y57 L58 S61 T78 I81 A85 W88 R89 Q100 Y103 W107 R140 K147 K156 R157 N163 F170 P178 L182 S13 Y15 L16 S19 T36 I39 A43 W46 R47 Q58 Y61 W65 R98 K105 K114 R115 N121 F128 P136 L140 ? remove_due_to_license_issue Q00059 31114891 2 ~ 23 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 G 3.1 BS01 dna H 0 K51 K52 V54 L58 K62 I81 K147 R157 P158 S160 Y162 Q179 L182 K183 K186 E208 Y211 R232 R233 T234 K9 K10 V12 L16 K20 I39 K105 R115 P116 S118 Y120 Q137 L140 K141 K144 E166 Y169 R190 R191 T192 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 G 3.1 BS02 dna I 0 S55 Y57 L58 S61 T78 I81 A85 W88 R89 Y103 W107 R140 K156 R157 N163 A167 F170 P178 L182 S13 Y15 L16 S19 T36 I39 A43 W46 R47 Y61 W65 R98 K114 R115 N121 A125 F128 P136 L140 ? remove_due_to_license_issue Q00059 31114891 2 ~ 23 SSVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 J 3.1 BS01 dna K 0 K51 K52 V54 L58 K62 R140 K146 K147 R157 Y162 Q179 L182 K186 Y211 R232 R233 T234 K8 K9 V11 L15 K19 R97 K103 K104 R114 Y119 Q136 L139 K143 Y168 R189 R190 T191 ? remove_due_to_license_issue Q00059 31114891 1 ~ 22 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hc3 J 3.1 BS02 dna L 0 S55 Y57 L58 T78 I81 R82 A85 W88 R89 Q100 Y103 W107 K139 M143 K146 K147 K156 R157 N163 V166 F170 P178 S12 Y14 L15 T35 I38 R39 A42 W45 R46 Q57 Y60 W64 K96 M100 K103 K104 K113 R114 N120 V123 F127 P135 ? remove_due_to_license_issue Q00059 31114891 2 ~ 23 SVLASCPKKPVSSYLRFSKEQLPIFKAQNPDAKTTELIRRIAQRWRELPDSKKKIYQDAYRAEWQVYKEEISRFKEQLTPSQIMSLEKEIMDKHLKRKAMTKKKELTLLGKPKRPRSAYNVYVAERFQEAKGDSPQEKLKTVKENWKNLSDSEKELYIQHAKEDETRYHNEMKSWEEQMIEVGRKDLLRRT 6hck A 2.7 BS01 LEU A 1 K64 Y126 L150 K64 Y126 L150 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue P22262 30759392 301 MNAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELIAHSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6hck A 2.7 BS02 LEU A 2 Y63 K64 F67 W224 Y63 K64 F67 W219 ? 0003677,0003700,0005829,0006355 remove_due_to_license_issue P22262 30759392 302 MNAQAEEFKKYLETNGIKPKQFHKKELIFNQWDPQEYCIFLYDGITKLTSISENGTIMNLQYYKGAFVIMSGFIDTETSVGYYNLEVISEQATAYVIKINELKELLSKNLTHFFYVFQTLQKQVSYSLAKFNDFSINGKLGSICGQLLILTYVYGKETPDGIKITLDNLTMQELIAHSSAVSRIISKLKQEKVIVYKNSCFYVQNLDYLKRYAPKLDEWFYLACPATWGKLN 6hcu A 1.62 BS01 FYB A 1 R330 H338 N339 F342 E500 G554 L555 R559 R249 H257 N258 F261 E419 G457 L458 R462 R330 E332 T337 H338 E500 N503 R559 R249 E251 T256 H257 E419 N422 R462 6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 ic50=0.015uM remove_due_to_license_issue Q8IDJ8 30894487 601 VDPRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKYGLKDTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFLDSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRPA 6hcu B 1.62 BS01 FYB B 1 R330 H338 N339 F342 E500 G554 L555 R559 R251 H259 N260 F263 E421 G457 L458 R462 R330 E332 T337 H338 E500 N503 R559 R251 E253 T258 H259 E421 N424 R462 6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 ic50=0.015uM remove_due_to_license_issue Q8IDJ8 30894487 601 VDPRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSAQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKYGLKDTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAGGANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFSAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRPA 6hcv A 2.2 BS01 FYE A 1 R330 T337 H338 N339 F342 E500 G554 R559 R245 T252 H253 N254 F257 E415 G452 R457 6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 ic50=0.005uM remove_due_to_license_issue Q8IDJ8 30894487 601 PRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKYGLTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPNPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFKLAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRPA 6hcv B 2.2 BS01 FYE B 1 R330 E332 H338 N339 F342 E500 G554 R559 R246 E248 H254 N255 F258 E414 G451 R456 6.1.1.6 0000166,0003676,0004812,0004824,0005524,0005737,0006418,0006430 ic50=0.005uM remove_due_to_license_issue Q8IDJ8 30894487 601 PRLYFENRSKFIQDQKDKGINPYPHKFERTISIPEFIEKYKDLGNGEHLEDTILNITGRIMRVSASGQKLRFFDLVGDGEKIQVLANYSFHNHEKGNFAECYDKIRRGDIVGIVGFPGKSKKGELSIFPKETILLSACLHMLPMKGLTEIRYRQRYLDLLINESSRHTFVTRTKIINFLRNFLNERGFFEVETPMMNLIAANARPFITHHNDLDLDLYLRIATELPLKMLIVGGIDKVYEIGKVFRNEGIDNTHNPEFTSCEFYWAYADYNDLIKWSEDFFSQLVYHLFGTYKISYNKDGPENQPIEIDFTPPYPKVSIVEEIEKVTNTILEQPFDSNETIEKMINIIKEHKIELPPTAAKLLDQLASHFIENKYNDKPFFIVEHPQIMSPLAKYHRTKPGLTERLEMFICGKEVLNAYTELNDPFKQKECFKLAFCTSLEYGLPPTGGLGLGIDRITMFLTNKNSIKDVILFPTMRPA 6hcw A 1.46 BS02 FYB A 1 R295 E297 H303 N304 F307 E464 L465 G518 L519 G520 R523 R251 E253 H259 N260 F263 E420 L421 G474 L475 G476 R479 R295 E297 T302 H303 E464 N467 R523 R251 E253 T258 H259 E420 N423 R479 6.1.1.6 0000049,0000166,0003676,0004812,0004824,0005524,0005737,0005829,0006418,0006430,0016020 ic50=0.13uM remove_due_to_license_issue Q5CR27 30894487 602 SHYTDNRYKMMECIKDAGRPFYPHKFKISMSLPAYALKYGNVENGYIDKDTTLSLSGRVTSIRSSSSKLIFYDIFCEEQKVQIIANIMEHDISTGEFSVSHSEIRRGDVVGFTGFPGKSKRGELSLFSKSVVLLSPCYHMLPTAISGLKDQEVRYRQRYLDLMLNEESRKVFKLRSRAIKYIRNYFDRLGFLEVETPMLNMIYGGAAARPFITYHNELETQLYMRIAPELYLKQLIVGGLDKVYEIGKNFRNEGIDLTHNPEFTAMEFYMAYADYYDLMDLTEELISGLVLEIHGSLKIPYHPDGPEGKCIEIDFTTPWKRFSFVEEIESGLGEKLKRPLDSQENIDFMVEMCEKHEIELPHPRTAAKLLDKLAGHFVETKCTNPSFIIDHPQTMSPLAKWHREKPEMTERFELFVLGKELCNAYTELNEPLQQRKFFEQQADAKASGDVEACPIDETFCLALEHGLPPTGGWGLGIDRLIMFLADKNNIKEVILFPAMRN 6hd4 A 2.03 BS01 FYW A 1 A356 L359 L360 A452 T453 Y454 E481 P484 V487 I521 V525 A114 L117 L118 A210 T211 Y212 E239 P242 V245 I279 V283 D382 A384 R386 N387 D400 P421 D140 A142 R144 N145 D158 P179 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 30137981 603 GAMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKEL 6hd6 A 2.3 BS01 FYH A 1 L359 L360 L448 A452 E481 C483 P484 I521 L115 L116 L204 A208 E237 C239 P240 I277 D382 A384 R386 N387 D400 P421 D138 A140 R142 N143 D156 P177 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00520 30137981 602 AMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKEL 6hdn A 1.9 BS01 FZB A 1 V1008 N1064 D1071 I1074 V30 N86 D93 I96 3.6.1.- ic50=3.16uM remove_due_to_license_issue IC50=25119nM Q6PL18 30226378 1206 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 6hdo A 2.61 BS01 FZH A 1 V1008 V1013 D1014 E1017 V1018 Y1063 N1064 G1070 D1071 I1074 R1077 V30 V35 D36 E39 V40 Y85 N86 G92 D93 I96 R99 3.6.1.- remove_due_to_license_issue IC50=251nM Q6PL18 30226378 1203 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 6hdq A 1.7 BS01 FZE A 1 W81 P82 L92 W38 P39 L49 ? ic50=5.01uM remove_due_to_license_issue IC50=5012nM O60885 30226378 202 NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6hf5 A 1.8 BS03 G1N A 1 F62 Y67 W87 D118 H179 C198 R205 G209 N210 H240 F31 Y36 W56 D87 H148 C167 R174 G178 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 ic50=6.7uM remove_due_to_license_issue Q9K2N0 30427656 306 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6hgf A 1.651 BS01 HCY B 1 A27 S28 R270 A5 S6 R248 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 remove_due_to_license_issue P01011 31103428 501 DRGLASANVDFAFSLYKQLVLKAPDKNVIFSPLSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNQSSDELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKWEMPFDPQDTHQSRFYLSKKKWVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASALFILPDQDKMEEVEAMLSRETLARWGDSLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTEASAATAVKITLL 6hgf B 1.651 BS01 HCY B 1 V381 H383 W386 V16 H18 W21 ? Kd=9.6uM remove_due_to_license_issue P01011 31103428 501 TRTIVRFNRPFLMIIVDHFTWSIFFMSKVTNPKQ 6hgg A 1.787 BS01 HCY A 1 S28 V31 F252 R270 A274 S7 V10 F231 R249 A253 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 Kd=3.8uM remove_due_to_license_issue P01011 31103428 401 VDRGLASANVDFAFSLYKQLVLKAPDKNVIFSPVSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNQSSDELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKWEMPFDPQDTHQSRFYLSKKKWVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASVFFILPDQDKMEEVEAMLSRETLARWGDSLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTEASAATAVKITLL 6hgg B 1.787 BS01 HCY A 1 V381 H383 W386 V15 H17 W20 ? remove_due_to_license_issue P01011 31103428 401 RTIVRFNRPFLMIIVDHFTWSIFFMSKVTNPKQA 6hgi A 1.517 BS01 C0R A 1 S28 V31 F252 R270 L273 S6 V9 F230 R248 L251 ? 0003677,0004867,0005515,0005576,0005615,0005634,0006953,0006954,0019216,0030277,0031093,0034774,0035578,0062023,0070062,0072562 Kd=0.6uM remove_due_to_license_issue P01011 31103428 401 DRGLASANVDFAFSLYKQLVLKAPDKNVIFSPVSISTALAFLSLGAHNTTLTEILKGLKFNLTETSEAEIHQSFQHLLRTLNQSSDELQLSMGNAMFVKEQLSLLDRFTEDAKRLYGSEAFATDFQDSAAAKKLINDYVKNGTRGKITDLIKDLDSQTMMVLVNYIFFKAKWEMPFDPQDTHQSRFYLSKKKWVMVPMMSLHHLTIPYFRDEELSCTVVQLNYTGNASVFFILPDQDKMEEVEAMLSRETLARWGDSLEFREIGELYLPKFSISRDYNLNDILLQLGIEEAFTSKADLSGITGARNLAVSQVVHKAVLDVFEEGTEASAATAVKITLL 6hgi B 1.517 BS01 C0R A 1 V381 H383 W386 V16 H18 W21 ? remove_due_to_license_issue P01011 31103428 401 TRTIVRFNRPFLMIIVDHFTWSIFFMSKVTNPKQA 6hgj B 1.825 BS01 AS4 A 1 H383 W386 H17 W20 ? remove_due_to_license_issue P01011 31103428 401 RTIVRFNRPFLMIIVDHFTWSIFFMSKVTNPKQA 6hgr A 1.52 BS01 IMP A 1 F26 R27 R67 D127 D128 L129 A131 T132 G133 T135 F24 R25 R65 D120 D121 L122 A124 T125 G126 T128 2.4.2.7 0002055,0003999,0005515,0005576,0005654,0005737,0005829,0006166,0006168,0007625,0016208,0016757,0032263,0032264,0034774,0044209,0046083,0070062 Ki=350uM remove_due_to_license_issue P07741 31160323 200 DSELQLVEQRIRSFPDFPTPGVVFRDISPVLKDPASFRAAIGLLARHLKATHGGRIDYIAGLDSRGFLFGPSLAQELGLGCVLIRKRGKLPGPTLWASYKAELEIQKDALEPGQRVVVVDDLLATGGTMNAACELLGRLQAEVLECVSLVELTSLKGREKLAPVPFFSLLQYE 6hgr B 1.52 BS01 IMP B 1 F26 R27 R67 D127 D128 L129 A131 T132 G133 T135 F24 R25 R65 D125 D126 L127 A129 T130 G131 T133 2.4.2.7 0002055,0003999,0005515,0005576,0005654,0005737,0005829,0006166,0006168,0007625,0016208,0016757,0032263,0032264,0034774,0044209,0046083,0070062 Ki=350uM remove_due_to_license_issue P07741 31160323 200 DSELQLVEQRIRSFPDFPTPGVVFRDISPVLKDPASFRAAIGLLARHLKATHGGRIDYIAGLDSRGFLFGPSLAQELGLGCVLIRKRGKLPGPTLWASYSLEYGKAELEIQKDALEPGQRVVVVDDLLATGGTMNAACELLGRLQAEVLECVSLVELTSLKGREKLAPVPFFSLLQYE 6hgv A 2.0 BS02 G3Q A 1 D335 W336 M339 F381 Y383 Q384 M419 Y466 M469 H524 D107 W108 M111 F153 Y155 Q156 M191 Y238 M241 H296 F267 D335 W336 D496 H524 F39 D107 W108 D268 H296 3.1.3.76,3.3.2.10 0003824 ic50=2.8uM remove_due_to_license_issue IC50=2800nM P34913 31223445 602 PTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 6hgx A 2.16 BS02 G3T A 1 D335 W336 M339 I375 Y383 Q384 M419 Y466 M469 D107 W108 M111 I147 Y155 Q156 M191 Y238 M241 F267 D335 W336 D496 H524 F39 D107 W108 D268 H296 3.1.3.76,3.3.2.10 0003824 ic50=0.077uM remove_due_to_license_issue IC50=77nM P34913 31223445 602 PTSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSDAR 6hgy A 2.2 BS01 G4B A 1 G23 C25 G65 G66 Y67 N161 G23 C25 G65 G66 Y67 N161 Q19 C25 H162 N182 Q19 C25 H162 N182 3.4.22.38 0006508,0008234 remove_due_to_license_issue P43235 30628449 301 APDSVDYRKKGYVTPVKNQGQCGSCWAFSSVGALEGQLKKKTGKLLNLSPQNLVDCVSENDGCGGGYMTNAFQYVQKNRGIDSEDAYPYVGQEESCMYNPTGKAAKCRGYREIPEGNEKALKRAVARVGPVSVAIDASLTSFQFYSKGVYYDESCNSDNLNHAVLAVGYGIQKGNKHWIIKNSWGENWGNKGYILMARNKNNACGIANLASFPKM 6hgz A 1.86 BS03 AR6 A 1 D63 G103 G105 F129 S134 Y135 G136 N137 G138 H168 I260 D303 T306 D55 G95 G97 F121 S126 Y127 G128 N129 G130 H160 I234 D277 T280 3.2.1.143,3.2.2.-,3.5.1.- 0000287,0004649,0005634,0005694,0005737,0005739,0005759,0006281,0016787,0046872,0060546,0140290,0140292 remove_due_to_license_issue H3BCW1 30472116 403 MVSLAQVRGALCGALLGDCMGAEFEGSDAVELPDVLEFVRLLEKEKKAGTLFYTDDTAMTRAVIQSLIAKPDFDEVDMAKRFAEEYKKEPTRGYGAGVVQVFKKLLSPKYSDVFQPAREQFDGKGSYGNGGAMRVASIALAYPNIQDVIKFARRSAQLTHASPLGYNGAILQALAVHFALQGELKRDTFLEQLIGEMERIEGLPFCSRLKKIKEFLASSNVPKADIVDELGHGIAALESVPTAIYSFLHCMESDPDIPDLYNNLQRTIIYSISLGGDTDTIATMAGAIAGAYYGMDQVTPSWKRSCEAIVETEESAVKLYELYCKQL 6hh3 A 1.82 BS03 A1R A 1 D63 D64 G103 G105 F129 S134 Y135 G136 N137 G138 H168 D303 D305 T306 D56 D57 G96 G98 F122 S127 Y128 G129 N130 G131 H161 D279 D281 T282 3.2.1.143,3.2.2.-,3.5.1.- 0000287,0004649,0005634,0005694,0005737,0005739,0005759,0006281,0016787,0046872,0060546,0140290,0140292 remove_due_to_license_issue H3BCW1 30472116 403 PMVSLAQVRGALCGALLGDCMGAEFEGSDAVELPDVLEFVRLLEKEKKAGTLFYTDDTAMTRAVIQSLIAKPDFDEVDMAKRFAEEYKKEPTRGYGAGVVQVFKKLLSPKYSDVFQPAREQFDGKGSYGNGGAMRVASIALAYPNIQDVIKFARRSAQLTHASPLGYNGAILQALAVHFALQGELKRDTFLEQLIGEMERIEGKLPFCSRLKKIKEFLASSNVPKADIVDELGHGIAALESVPTAIYSFLHCMESDPDIPDLYNNLQRTIIYSISLGGDTDTIATMAGAIAGAYYGMDQVTPSWKRSCEAIVETEESAVKLYELYCKQL 6hh5 A 1.95 BS02 A3R A 1 E33 D63 G103 A104 G105 F129 S134 Y135 G136 N137 G138 H168 I260 D303 E25 D55 G95 A96 G97 F121 S126 Y127 G128 N129 G130 H160 I234 D277 3.2.1.143,3.2.2.-,3.5.1.- 0000287,0004649,0005634,0005694,0005737,0005739,0005759,0006281,0016787,0046872,0060546,0140290,0140292 remove_due_to_license_issue H3BCW1 30472116 402 MVSLAQVRGALCGALLGDCMGAEFEGSDAVELPDVLEFVRLLEKEKKAGTLFYTDDTAMTRAVIQSLIAKPDFDEVDMAKRFAEEYKKEPTRGYGAGVVQVFKKLLSPKYSDVFQPAREQFDGKGSYGNGGAMRVASIALAYPNIQDVIKFARRSAQLTHASPLGYNGAILQALAVHFALQGELKRDTFLEQLIGEMERIEGLPFCSRLKKIKEFLASSNVPKADIVDELGHGIAALESVPTAIYSFLHCMESDPDIPDLYNNLQRTIIYSISLGGDTDTIATMAGAIAGAYYGMDQVTPSWKRSCEAIVETEESAVKLYELYCKQL 6hhg A 2.3 BS01 G4T A 1 E17 W80 L210 T211 L264 K268 Y272 R273 D274 D292 C310 E15 W74 L155 T156 L209 K213 Y217 R218 D219 D237 C252 D274 K276 N279 D292 T312 D219 K221 N224 D237 T254 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue P31749 30996949 501 DVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDEAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVISRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKTMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTA 6hhh A 2.7 BS01 G4Q A 1 E17 W80 T82 I84 E85 L210 T211 L264 K268 Y272 D292 C296 K297 E16 W76 T78 I80 E81 L161 T162 L215 K219 Y223 D243 C247 K248 D274 K276 N279 D292 T312 D225 K227 N230 D243 T252 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue P31749 30996949 501 SDVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDVEAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFD 6hhi A 2.7 BS01 G4N A 1 E17 W80 I84 E85 L210 T211 L264 K268 Y272 R273 D274 D292 C296 E15 W75 I79 E80 L158 T159 L212 K216 Y220 R221 D222 D240 C244 D274 K276 N279 D292 T312 D222 K224 N227 D240 T257 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue IC50=18.2nM, Kd=79.0nM P31749 30996949 501 DVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDREAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKTMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTA 6hhj A 2.3 BS01 G4H A 1 W80 I84 S205 L210 L264 Y272 R273 D274 D292 C296 C310 W76 I80 S171 L176 L230 Y238 R239 D240 D258 C262 C276 D274 K276 N279 D292 T312 D240 K242 N245 D258 T278 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue P31749 30996949 501 DVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDQREAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKQRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTA 6hhr A 2.0 BS01 G5E A 1 N51 A55 K58 D93 I96 G97 M98 L107 G108 T184 N35 A39 K42 D77 I80 G81 M82 L91 G92 T168 3.6.4.10 0005524,0006457,0016887,0051082,0140662 remove_due_to_license_issue P07900 30500211 301 VETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 6hjj A 2.13 BS01 G7T A 1 L139 G140 A160 K162 V174 Q177 L178 E181 A213 L263 A273 F275 L13 G14 A34 K36 V48 Q51 L52 E55 A87 L137 A147 F149 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T155 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=1.7uM remove_due_to_license_issue O14965 30239186 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLICEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPSNA 6hjk A 2.4 BS01 G7W A 1 F144 K162 V174 L178 L194 Y212 A213 L263 G276 W277 F18 K36 V48 L52 L68 Y86 A87 L137 G150 W151 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T156 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 ic50=25nM remove_due_to_license_issue O14965 30239186 501 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLICEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 6hk3 A 2.35 BS02 G8B A 1 V70 A83 D133 Y134 V135 R141 L188 D200 V36 A49 D99 Y100 V101 R107 L154 D166 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0004672,0005524,0006468 Kd=31.4nM remove_due_to_license_issue Ki=12nM P49841 31246463 401 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 6hk4 A 2.5 BS02 G8E A 1 I62 F67 A83 K85 D133 Y134 V135 R141 L188 D200 I28 F33 A49 K51 D99 Y100 V101 R107 L154 D166 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0004672,0005524,0006468 Kd=2.81nM remove_due_to_license_issue Ki=0.67nM P49841 31246463 408 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 6hk6 A 2.35 BS01 G8H A 1 M101 A121 I191 G193 I235 I245 M100 A120 I180 G182 I224 I234 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9BVS4 30991936 401 GKVNVAKLRYMSRDDFRVLTAVEMGMKNHEIVPGSLIASIASLKHGGCNKVLRELVKHKLIAWERTKTVQGYRLTNAGYDYLALKTLSSRQVVESVGNQMGVGKESDIYIVANEEGQQFALKLHRLGRTSFRNLHNVSWLYLSRLSAMKEFAYMKALYERKFPVPKPIDYNRHAVVMELINGYPLCQIHHVEDPASVYDEAMELIVKLANHGLIHGDFNEFNLILDESDHITMIDFPQMVSTSHPNAEWYFDRDVKCIKDFFMKRFSYESELFPTFKDIRREDTLDVEVS 6hk7 A 3.2 BS01 G8N A 1 I62 F67 V70 A83 K85 V135 P136 T138 R141 L188 D200 I27 F32 V35 A48 K50 V100 P101 T103 R106 L153 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0004672,0005524,0006468 remove_due_to_license_issue Ki=90nM P49841 31246463 403 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA 6hke A 2.11 BS01 MLT A 1 F24 P29 T30 H80 S149 V150 S151 G173 T174 Q192 F12 P17 T18 H68 S137 V138 S139 G161 T162 Q180 ? Kd=21nM remove_due_to_license_issue Q6N446 30471256 401 FPVRTVTVVVPFAKGGPTDTVARLITAEMAKTLGQPIEIENMLGAGGTLAATRVAHAAPDGHTLIVGHLGTHGAAVALFPKLAYRPDKDFTPVALLTEMPVLLLARKQFPPKDLSEFASYVESHTDNLNVAHAGFGSVSYASCLLLNRLLKVDPTGVPFSGTGPALQALVEGQVDYMCDQIVNAVPALREGKVKAYVIAASERDPVVPDVPTAREAGLPGFQVGAWTGLFAPRGTPEPIVAKLNAAVSRALDQSDVRTRLTDLGALVPRPEQRAPVVLAQLVQEEISRWEDVVE 6hkj A 2.09 BS04 G8W A 1 K207 R210 E424 L428 G518 N519 R534 R536 Y552 H553 K699 Y700 K153 R156 E370 L374 G464 N465 R480 R482 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.99nM remove_due_to_license_issue IC50=0.990000nM Q04609 30429952 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6hkm A 2.47 BS01 G92 A 1 I61 A82 K84 I86 E102 L103 L106 V135 L137 M140 D200 I8 A19 K21 I23 E39 L40 L43 V71 L73 M76 D136 D182 K184 S186 N187 D200 T224 D118 K120 S122 N123 D136 T158 2.7.11.24 0004672,0004707,0005524,0006468 ic50=270nM remove_due_to_license_issue IC50=270nM Q13164 30563338 1001 EYEIIETIGNVVSSAQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARREGI 6hkn A 2.33 BS01 G9E A 1 I61 Y66 A82 K84 I86 E102 L103 L106 L137 D138 M140 L189 D200 I8 Y10 A22 K24 I26 E42 L43 L46 L77 D78 M80 L129 D140 D182 K184 S186 N187 D200 T224 D122 K124 S126 N127 D140 T164 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.051uM remove_due_to_license_issue IC50=51nM Q13164 30563338 1001 EYEIIETIAYGVVSSARRQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSPAEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARRE 6hkx A 2.8 BS02 GCE A 1 E116 G117 E118 R119 A133 I136 P137 Y211 L214 E215 G217 A218 R221 E92 G93 E94 R95 A109 I112 P113 Y187 L190 E191 G193 A194 R197 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=6.0nM P52732 31488701 602 KNIQVVVRCRPFNHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTLVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 6hkx B 2.8 BS02 GCE B 1 E116 G117 W127 A133 Y211 L214 E215 G217 A218 R221 F239 E90 G91 W101 A107 Y185 L188 E189 G191 A192 R195 F213 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=6.0nM P52732 31488701 602 KNIQVVVRCRPFNLAHSIVECDPVRKEVSVRTGGSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKETTIDGEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 6hky A 2.75 BS02 GCE A 1 E116 G117 E118 R119 A133 I136 Y211 L214 A218 R221 E101 G102 E103 R104 A118 I121 Y196 L199 A203 R206 ? 0003777,0005524,0007018,0008017 remove_due_to_license_issue IC50=6.0nM P52732 31488701 403 GKNIQVVVRCRPFNLAERKASAHSIVECDPVRKEVSVRTGGLADKSSRKTYTFDMVFGASTKQIDVYRSVVCPILDEVIMGYNCTIFAYGQTGTGKTFTMEGERSPNEEYTWEEDPLAGIIPRTLHQIFEKLTDNGTEFSVKVSLLEIYNEELFDLLNPSSDVSERLQMFDDPRNKRGVIIKGLEEITVHNKDEVYQILEKGAAKRTTAATLMNAYSSRSHSVFSVTIHMKEELVKIGKLNLVDLAGSENNINQSLLTLGRVITALVERTPHVPYRESKLTRILQDSLGGRTRTSIIATISPASLNLEETLSTLEYAHRAKNILNKPE 6hkz A 2.09 BS04 GBZ A 1 R210 N257 E424 L428 R463 D465 G518 N519 R534 R536 S547 G548 Y552 H553 K699 Y700 R156 N203 E370 L374 R409 D411 G464 N465 R480 R482 S493 G494 Y498 H499 K643 Y644 3.4.17.21 0004180,0004181,0005737,0005886,0006508,0006760,0008233,0008237,0009986,0016020,0016805,0035609,0046872,0070062,1904492,1904493 ic50=0.13nM remove_due_to_license_issue IC50=0.130000nM Q04609 30429952 818 KHNMKAFLDELKAENIKKFLYNFTQIPHLAGTEQNFQLAKQIQSQWKEFGLDSVELAHYDVLLSYPNKTHPNYISIINEDGNEIFNTSLFEPPPPGYENVSDIVPPFSAFSPQGMPEGDLVYVNYARTEDFFKLERDMKINCSGKIVIARYGKVFRGNKVKNAQLAGAKGVILYSDPADYFAPGVKSYPDGWNLPGGGVQRGNILNLNGAGDPLTPGYPANEYAYRRGIAEAVGLPSIPVHPIGYYDAQKLLEKMGGSAPPDSSWRGSLKVPYNVGPGFTGNFSTQKVKMHIHSTNEVTRIYNVIGTLRGAVEPDRYVILGGHRDSWVFGGIDPQSGAAVVHEIVRSFGTLKKEGWRPRRTILFASWDAEEFGLLGSTEWAEENSRLLQERGVAYINADSSIEGNYTLRVDCTPLMYSLVHNLTKELKSPDEGFEGKSLYESWTKKSPSPEFSGMPRISKLGSGNDFEVFFQRLGIASGRARYTKNWETNKFSGYPLYHSVYETYELVEKFYDPMFKYHLTVAQVRGGMVFELANSIVLPFDCRDYAVVLRKYADKIYSISMKHPQEMKTYSVSFDSLFSAVKNFTEIASKFSERLQDFSNPIVLRMMNDQLMFLERAFIDPLGLPDRPFYRHVIYAPSSHNKYAGESFPGIYDALFDIESKVDPSKAWGEVKRQIYVAAFTVQAAAETLSEVA 6hlx A 1.65 BS01 G9Z A 1 G45 Y239 Q267 Y355 F357 Q358 W383 R386 G401 T425 N426 R475 G21 Y215 Q243 Y331 F333 Q334 W359 R362 G377 T401 N402 R451 ? 0015031,0015833,0030288,0042597,0043190,0046872,0055085,1904680 remove_due_to_license_issue O50260 30552142 604 GTLYFGLSGEPSTLDTVVQPGTSGRTVKLAIHRGLVNYGIDGKISPELAESYEVSPDAKEFTFHLRQAKFHDGTTVTSADVKASLERILDPKGKASFRNELSSISKIETPDEKTVKLTLSTPSVAMIDYLALPESVIVPAAWLAKNADNPNAAPVGAGPFKFAGWTRGREITVKKFDDYYKKGKPDLDEVHYVFYSDENTRVNALKSGDVDIIDYVPAKDAADIAKGPETQLLRNTGPFMGLQFNTKFEPFSKPEVRQAIAYAVDRSAIINTAFNGLGSPIFGIAIPKGYMGYSDAKANYFSHHVEKAKALLAKAGYPNGFEVRLLATSQYSFQQNTAIAIQSELAKIGIKVKLDLPDWASRMAKASTGDYDFTVMGSLGEITDADWLSNYYYGGDKLVRTNNSPYFNDQQINDLLDKGRATVDKAERVKIYDAFVDRALELSPLVYFMWREQNYAVKKGVTGFTNMPGFLTFQSGLSIENTKIEHHHHHH 6hly A 1.4 BS01 G9Z A 1 Y37 F41 E89 M128 F130 A208 R229 E252 Y288 Y11 F15 E63 M102 F104 A182 R203 E226 Y262 0015846,0019808,0042597 remove_due_to_license_issue 30552142 410 HMMADLVISSYGGSFQDAQTKAYFDPYAKASGVKVTGTTGTGYAKVKAMVESGNVTWDVISAESPAFASEVKDGLLEPIDYSVVKADNVPENFRTKYGVGYMVFGTNLAWNKDKFPNGVTPAQFFDPNVKGRRVLPSDATYSLEFALMGDGVKPADLYPLDVKRALKVIDRVKDQVIGYKGASDIQALMQQGEADIVYAGTGRIKNAIKAGANWSYSWEGALADTEYWAVPKGAPHAAEAMKFINFAVQAEPQAELTRVIAYGPTNVDALRLLDPAVAKDLPSYPANAKLGAVLNSKWWNDNYDAVKAEWTTYIMQHHHH 6hlz A 1.89 BS01 G9Z A 1 Y37 F41 E89 M128 F130 S163 A208 R229 E252 Y288 Y11 F15 E63 M102 F104 S137 A182 R203 E226 Y262 0015846,0019808,0042597 remove_due_to_license_issue 30552142 432 HMMADLVISSYGGSFQDAQTKAYFDPYAKASGVKVTGTTGTGYAKVKAMVESGNVTWDVISAESPAFASEVKDGLLEPIDYSVVKADNVPENFRTKYGVGYMVFGTNLAWNKDKFPNGVTPAQFFDPNVKGRRVLPSDATYSLEFALMGDGVKPADLYPLDVKRALKVIDRVKDQVIGYKGASDIQALMQQGEADIVYAGTGRIKNAIKAGANWSYSWEGALADTEYWAVPKGAPHAAEAMKFINFAVQAEPQAELTRVIAYGPTNVDALRLLDPAVAKDLPSYPANAKLGAVLNSKWWNDNYDAVKAEWTTYIMQ 6hm1 A 1.54 BS01 AO3 A 1 Y28 F58 G113 W114 D151 E153 M220 Y222 D223 Y276 Y325 M393 W395 Y8 F29 G84 W85 D122 E124 M191 Y193 D194 Y247 Y296 M364 W366 ? 0000272,0004553,0004568,0005975,0006032,0008061,0016798 Kd=0.91uM remove_due_to_license_issue A8GFD6 30789732 501 ASYLSVGYFNGGDINKLDVTQITHLNYSFGLIYNDEKQETNPALKDPSRLHQIYLSPKVMADLQLLPVLRKQNPELKVLLSVGGWGARGFSGAAATAESRAVFIRSVQQVIKQYHLDGIDLDWEYPVNGAWGLVESQPADRANFTLLLAELHKALDKGKLLTIAVGANVKSPQEWVDVKGIAPYLDYINLMTYDMAYGTQYFNSNLYDSKQWPTVAAADRYSANFVVDNYLAAGLKPAQLNLGIGFYGRVPKRATEPGIDWDKADAAKNPVTQPYFTARETAVFKAMGLDLTKDSYFKYNDIVSKLLNDPQRRFTAHWDSDAQVPYLTMKSAEGKPLFAISYENPRSVALKADYIKSKGLGGAMFWEYGADDNNRLAHQLAESLGI 6hm2 A 1.74 BS01 G9Z A 1 Y37 F41 E89 M128 F130 A208 R229 E252 Y288 Y12 F16 E64 M103 F105 A183 R204 E227 Y263 0015846,0019808,0042597 remove_due_to_license_issue 30552142 401 SHMMADLVISSYGGSFQDAQTKAYFDPYAKASGVKVTGTTGTGYAKVKAMVESGNVTWDVISAESPAFASEVKDGLLEPIDYSVVKADNVPENFRTKYGVGYMVFGTNLAWNKDKFPNGVTPAQFFDPNVKGRRVLPSDATYSLEFALMGDGVKPADLYPLDVKRALKVIDRVKDQVIGYKGASDIQALMQQGEADIVYAGTGRIKNAIKAGANWSYSWEGALADTEYWAVPKGAPHAAEAMKFINFAVQAEPQAELTRVIAYGPTNVDALRLLDPAVAKDLPSYPANAKLGAVLNSKWWNDNYDAVKAEWTTYIM 6hm6 A 2.1 BS01 GDK A 1 L377 G378 V385 A400 M448 A451 G454 L501 L14 G15 V22 A36 M79 A82 G85 L132 D494 R498 N499 D512 D125 R129 N130 D143 2.7.10.2 0004672,0004713,0005524,0006468 ic50=3.16uM remove_due_to_license_issue IC50=3162nM P43405 30249354 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKVVKTVAVKILDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYD 6hm7 A 1.64 BS01 GDH A 1 V385 A400 A451 G454 P455 L501 D512 V23 A38 A89 G92 P93 L139 D150 D494 R498 N499 D512 D132 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=79.4nM remove_due_to_license_issue IC50=79nM P43405 30249354 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDV 6hmg A 1.27 BS01 GDQ A 1 Y46 H154 E156 Y195 Y252 E333 E336 Y16 H124 E126 Y165 Y222 E303 E306 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 30427198 403 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 6hmg A 1.27 BS02 GLC A 1 H63 W126 R295 E333 H33 W96 R265 E303 ? 0004559,0016020,0016787,0016798 remove_due_to_license_issue D6D1V7 30427198 402 NNLGTELDYDTFCFYYDWYGSEAIDGQYRHWAHAIAPDPNGGSGQNPGTIPGTQESIASNFYPQLGRYSSSDPNILTKHMDMFVMARTGVLALTWWNEQDETEAKRIGLILDAADKKKIKVCFHLEPYPSRNVQNLRENIVKLITRYGNHPAFYRKDGKPLFFIYDSYLIEPSEWEKLLSPGGSITIRNTAYDALMIGLWTSSPTVQRPFILNAHFDGFYTYFAATGFTYGSTPTNWVSMQKWAKENGKIFIPSVGPGYIDTRIRPWNGSVIRTRTDGQYYDAMYRKAIEAGVSAISITSFNEWHEGSQIEPAVPYTSSEFTYLDYENREPDYYLTRTAYWVGKFRESK 6hmp A 2.039 BS01 GEW A 1 S17 G18 I23 A36 K38 M80 M82 L85 K130 D132 L135 I148 S10 G11 I16 A28 K30 M72 M74 L77 K122 D124 L127 I140 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=218nM remove_due_to_license_issue P48730 30924488 301 RYRLGRKIGSGSFGDIYLGTDIAAEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 6hmr A 1.782 BS01 GE5 A 1 S17 I23 A36 M80 M82 L85 D132 L135 I148 S11 I17 A29 M73 M75 L78 D125 L128 I141 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=2.36nM remove_due_to_license_issue P48730 30924488 301 NRYRLGRKIGSGSFGDIYLGTDIAAEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLK 6hmx A 2.53 BS01 GEZ A 1 L24 S25 V32 A45 K47 L79 T95 M98 G101 E105 L153 L20 S21 V28 A41 K43 L70 T86 M89 G92 E96 L144 D146 Q150 N151 D164 D137 Q141 N142 D155 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43353 30344914 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRGGTIIYMPPENYEPSIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 6hmy A 1.6 BS02 SIA K 1 E11 Y12 H13 E11 Y12 H13 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 31439922 6 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 6hmy B 1.6 BS01 SIA K 1 G33 K34 G33 K34 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 31439922 6 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 6hmy B 1.6 BS03 SIA L 1 E11 Y12 H13 I58 E11 Y12 H13 I58 ? 0005515,0005534,0005576,0016020,0020002,0035821,0042531,0042597,0046812,0090729,1902494 remove_due_to_license_issue P01556 31439922 6 TPQNITDLCAEYHNTQIHTLNDKIFSYTESLAGKREMAIITFKNGATFQVEVPGSQHIDSQKKAIERMKDTLRIAYLTEAKVEKLCVWNNKTPHAIAAISMAN 6hni A 1.35 BS01 TYR A 1 H55 S113 T114 A133 S135 D158 N189 T237 D238 N239 A242 E263 Y279 H12 S70 T71 A90 S92 D115 N146 T194 D195 N196 A199 E220 Y236 ? Kd=94uM remove_due_to_license_issue Q18A65 31420448 401 VKKIGITQLVEHPALDATRTGFVKALEKNGFKDGENIDIDFQNAQNDMPTTQSIASKFASDKKDLIFAISTPSAQAAFNATKDIPILITAVSDPVAAGLVKTLEKPGTNVSGTSDFVSVDKGLELLKIFAPKAKTIGVMYNTSEVNSKVQVDALKEYASKNGFKVVEKGITTSNEVNQGISSLVGKIDVLYVPTDNLVASSMPIVSKIATENKIPVIAAESGPVEKGALACQGINYEKLGYKTGEMAVKILNGESVSDMPVATSDDTDIIVNEDILKALGMEKPSNENISYVKTK 6hop A 1.55 BS01 FER A 1 V66 K68 F113 V116 M163 I174 D175 V64 K66 F111 V114 M161 I172 D173 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 31661600 405 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 6hoq A 1.55 BS01 FER A 1 V66 K68 F113 V116 M163 I174 D175 V64 K66 F111 V114 M161 I172 D173 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 31661600 404 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 6hor A 1.8 BS01 GJK A 1 V66 K68 F113 M163 I174 D175 V64 K66 F111 M161 I172 D173 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 31661600 401 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 6hot A 1.5 BS01 CIY A 1 V53 K68 F113 I174 D175 V51 K66 F111 I172 D173 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 31661600 404 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 6hou A 1.8 BS01 V55 A 1 K68 F113 I174 D175 K66 F111 I172 D173 D156 K158 N161 D175 S194 D154 K156 N159 D173 S192 2.7.11.1 0004672,0004674,0005524,0006468 remove_due_to_license_issue P68400 31661600 403 GPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKD 6hov A 1.85 BS01 FER A 1 W81 P82 V87 L92 N140 I146 W40 P41 V46 L51 N99 I105 ? remove_due_to_license_issue O60885 31661600 203 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 6hoy A 1.7 BS03 TSN A 1 A53 S56 F64 V70 W71 N114 D116 A44 S47 F55 V61 W62 N105 D107 P62 D63 F64 R65 N114 D116 H133 P53 D54 F55 R56 N105 D107 H124 2.3.1.-,2.3.1.286,2.4.2.- 0070403 Kd=33uM remove_due_to_license_issue Kd=33000nM, Ki=2000nM Q8N6T7 30395713 409 PFTADKGKCGLPEIFDPPEELERKVWELARLVWQSSSVVFHTGAGISTASGIPDFRGPHGVWTMEERGLAPKFDTTFESARPTQTHMALVQLERVGLLRFLVSQNVDGLHVRSGFPRDKLAELHGNMFVEECAKCKTQYVRDTVVGTMGLKATGRLCTVACRGELRDTILDWEDSLPDRDLALADEASRNADLSITLGTSLQIRPSGNLPLATKRRGGRLVIVNLQPTKHDRHADLRIHGYVDEVMTRLMKHLGLEIPAWDGPRVLERALPPLPRPPTPKL 6hp0 A 1.88 BS03 GJT A 1 E119 K150 D151 R152 R156 W179 R225 E277 R293 N295 R368 Y402 E38 K69 D70 R71 R75 W98 R144 E196 R212 N214 R287 Y321 D151 E278 R293 R368 Y402 D70 E197 R212 R287 Y321 3.2.1.18 0004308,0005975,0016020,0033644,0046761,0055036 Ki=470nM remove_due_to_license_issue C6KP13 31128993 503 SVKLAGNSSLCPVSGWAIYSKDNSVRIGSKGDVFVIREPFISCSPLECRTFFLTQGALLNDKHSNGTIKDRSPYRTLMSCPIGEVPSPYNSRFESVAWSASACHDGINWLTIGISGPDNGAVAVLKYNGIITDTIKSWRNNILRTQESECACVNGSCFTVMTDGPSNGQASYKIFRIEKGKIVKSVEMNAPNYHYEECSCYPDSSEITCVCRDNWHGSNRPWVSFNQNLEYQIGYICSGIFGDNPRPNDKTGSCGPVSSNGANGVKGFSFKYGNGVWIGRTKSISSRNGFEMIWDPNGWTGTDNNFSIKQDIVGINEWSGYSGSFVQHPELTGLDCIRPCFWVELIRGRPKENTIWTSGSSISFCGVNSDTVGWSWPDGAELPFTID 6hp9 A 1.96 BS01 GKB A 1 A653 E672 I675 M676 L679 I685 T701 Y703 M704 H764 A783 D784 A55 E74 I77 M78 L81 I87 T103 Y105 M106 H152 A171 D172 D766 R770 N771 D784 D154 R158 N159 D172 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=5.6nM remove_due_to_license_issue IC50=5.6nM Q08345 31310125 1001 SMPRVDFPRSRLRFKEKLGEGQFGEVHLCEVDSPQDLVSLDFPLNVRKGHPLLVAVKILRPDATKNARNDFLKEVKIMSRLKDPNIIRLLGVCVQDDPLCMITDYMENGDLNQFLSAHQLEQGPTISYPMLLHVAAQIASGMRYLATLNFVHRDLATRNCLVGENFTIKIADFGMSRNLYAGDYYRVQGRAVLPIRWMAWECILMGKFTTASDVWAFGVTLWEVLMLCRAQPFGQLTDEQVIENAGEFFRDQGRQVYLSRPPACPQGLYELMLRCWSRESEQRPPFSQLHRFLAEDA 6hpw A 1.9 BS01 GKT A 1 F28 H56 S58 F59 P60 E75 S76 Y78 A79 F81 F26 H54 S56 F57 P58 E73 S74 Y76 A77 F79 ? Kd~807nM remove_due_to_license_issue Q03111 30407816 209 NQCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6hq3 A 2.79 BS01 CMP D 1 R108 R111 R105 R108 ? remove_due_to_license_issue Q6MLN6 31355487 901 AAQSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRRKNI 6hq3 D 2.79 BS01 CMP D 1 F17 G57 E58 M59 A60 R67 S68 A69 F13 G53 E54 M55 A56 R63 S64 A65 ? remove_due_to_license_issue Q6MLN6 31355487 901 AQSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRR 6hq4 A 2.63 BS01 CMP A 1 F56 G57 E58 M59 A60 R67 S68 A69 N113 F51 G52 E53 M54 A55 R62 S63 A64 N108 ? 0000166,0046872,0071111 remove_due_to_license_issue Q6MLN6 31355487 901 QSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRRKNIGSALDQIKLENQIFQAFQNKEFELFYQPIVNLKNKTITGCEALLRWNSPQHGLVSPNLFIDIIENSSMVIPIGHWIINQALKDLRTIQDQLRLNKKERMADDFMMSINISGRQFTHSDFVNNLEDLREKHDLHTQNIKLEMTERIMMDGAIAIDALNQCRSLGYAISIDDFGTGFSGLQYLTQMPISFLKIDRSFVMKILSDPKSKAVVSSIIHLAHAMDIEVIAEGIEHHEEALVLETLGARFGQGYLFSKPVDLGRFLKLIKL 6hq4 B 2.63 BS01 CMP B 1 F17 F56 G57 E58 M59 A60 R67 S68 A69 F12 F51 G52 E53 M54 A55 R62 S63 A64 ? 0000166,0046872,0071111 remove_due_to_license_issue Q6MLN6 31355487 901 QSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRSALDQIKLENQIFQAFQNKEFELFYQPIVNLKNKTITGCEALLRWNSPQHGLVSPNLFIDIIENSSMVIPIGHWIINQALKDLRTIQDQLRLNKKERMADDFMMSINISGRQFTHSDFVNNLEDLREKHDLHTQNIKLEMTERIMMDGAIAIDALNQCRSLGYAISIDDFGTGFSGLQYLTQMPISFLKIDRSFVMKILSDPKSKAVVSSIIHLAHAMDIEVIAEGIEHHEEALVLETLGARFGQGYLFSKPVDLGRFLKLIK 6hq7 A 2.46 BS01 PCG A 1 F17 I36 L47 F56 G57 E58 M59 A60 R67 S68 A69 L109 F12 I31 L42 F51 G52 E53 M54 A55 R62 S63 A64 L104 ? 0000166,0046872,0071111 remove_due_to_license_issue Q6MLN6 31355487 901 QSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRRPGGSRISSALDQIKLENQIFQAFQNKEFELFYQPIVNLKNKTITGCEALLRWNSPQHGLVSPNLFIDIIENSSMVIPIGHWIINQALKDLRTIQDQLRLNKKERMADDFMMSINISGRQFTHSDFVNNLEDLREKHDLHTQNIKLEMTERIMMDGAIAIDALNQCRSLGYAISIDDFGTGFSGLQYLTQMPISFLKIDRSFVMKILSDPKSKAVVSSIIHLAHAMDIEVIAEGIEHHEEALVLETLGARFGQGYLFSKPVDLGRFLKLIKL 6hq7 A 2.46 BS03 PCG B 1 R108 R111 R103 R106 ? 0000166,0046872,0071111 remove_due_to_license_issue Q6MLN6 31355487 901 QSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRRPGGSRISSALDQIKLENQIFQAFQNKEFELFYQPIVNLKNKTITGCEALLRWNSPQHGLVSPNLFIDIIENSSMVIPIGHWIINQALKDLRTIQDQLRLNKKERMADDFMMSINISGRQFTHSDFVNNLEDLREKHDLHTQNIKLEMTERIMMDGAIAIDALNQCRSLGYAISIDDFGTGFSGLQYLTQMPISFLKIDRSFVMKILSDPKSKAVVSSIIHLAHAMDIEVIAEGIEHHEEALVLETLGARFGQGYLFSKPVDLGRFLKLIKL 6hq7 B 2.46 BS01 PCG A 1 R108 R111 R103 R106 ? 0000166,0046872,0071111 remove_due_to_license_issue Q6MLN6 31355487 901 QSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRRGTQSALDQIKLENQIFQAFQNKEFELFYQPIVNLKNKTITGCEALLRWNSPQHGLVSPNLFIDIIENSSMVIPIGHWIINQALKDLRTIQDQLRLNKKERMADDFMMSINISGRQFTHSDFVNNLEDLREKHDLHTQNIKLEMTERIMMDGAIAIDALNQCRSLGYAISIDDFGTGFSGLQYLTQMPISFLKIDRSFVMKILSDPKSKAVVSSIIHLAHAMDIEVIAEGIEHHEEALVLETLGARFGQGYLFSKPVDLGRFLKLIK 6hq7 B 2.46 BS02 PCG B 1 F17 I36 F56 G57 E58 M59 A60 R67 S68 A69 F12 I31 F51 G52 E53 M54 A55 R62 S63 A64 ? 0000166,0046872,0071111 remove_due_to_license_issue Q6MLN6 31355487 901 QSVDIHKDQIIFSEGDAGDCAYIIEKGRVLIYLTKDKEEIPLTILGEGEIFGEMALIDNQNRSASVRALEDVRLAIVTKQQVLERVSTADKVVQLLMRVLLKRLRRGTQSALDQIKLENQIFQAFQNKEFELFYQPIVNLKNKTITGCEALLRWNSPQHGLVSPNLFIDIIENSSMVIPIGHWIINQALKDLRTIQDQLRLNKKERMADDFMMSINISGRQFTHSDFVNNLEDLREKHDLHTQNIKLEMTERIMMDGAIAIDALNQCRSLGYAISIDDFGTGFSGLQYLTQMPISFLKIDRSFVMKILSDPKSKAVVSSIIHLAHAMDIEVIAEGIEHHEEALVLETLGARFGQGYLFSKPVDLGRFLKLIK 6hqy A 2.501 BS02 GKW A 1 K20 H141 H142 D186 H188 F216 P291 H292 Y341 K19 H140 H141 D176 H178 F206 P274 H275 Y311 3.5.1.98 0004407,0005634,0006325,0031507,0046872 Kd=367nM remove_due_to_license_issue IC50=436nM, Kd=367nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hr2 A 1.76 BS01 FWZ B 1 V1484 F1485 L1488 L1494 Y1497 V1505 A1536 F1539 N1540 I1546 V33 F34 L37 L43 Y46 V54 A85 F88 N89 I95 3.6.4.- 0006338,0016586 remove_due_to_license_issue P51532 31178587 301 SPNPPNLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNHKYRSLNDLEKDVMLLCQNAQTFNLEGSLIYEDSIVLQSVFTSVRQKIEKED 6hr2 B 1.76 BS01 FWZ B 1 F76 W88 Y98 P99 R107 I109 H110 S111 Y112 H115 W117 F16 W28 Y38 P39 R47 I49 H50 S51 Y52 H55 W57 ? remove_due_to_license_issue P40337 31178587 301 PVLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQERIAHQ 6hro A 2.3 BS01 GKZ A 1 L186 P187 K190 K191 L157 P158 K161 K162 ? ic50=0.05uM remove_due_to_license_issue Q05320 30785281 607 GRSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTWAFWESEELSFTVVAAAAAAAA 6hro A 2.3 BS02 GKZ B 1 N61 R64 V66 G67 E100 A101 N32 R35 V37 G38 E71 A72 ? ic50=0.05uM remove_due_to_license_issue Q05320 30785281 709 GRSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQAKKSGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTWAFWESEELSFTVVAAAAAAAA 6hro B 2.3 BS01 GKZ A 1 M548 L554 M47 L53 ? ic50=0.05uM remove_due_to_license_issue Q05320 30785281 607 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFV 6hro B 2.3 BS02 GKZ B 1 L515 Y517 D522 M548 L14 Y16 D21 M47 ? ic50=0.05uM remove_due_to_license_issue Q05320 30785281 709 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFV 6hrp A 1.12 BS01 GMQ A 1 L408 V416 A428 K430 Y476 M477 A478 N479 G480 N526 L528 D539 Y551 L13 V21 A33 K35 Y81 M82 A83 N84 G85 N131 L133 D144 Y156 D521 A523 R525 N526 D539 D126 A128 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=23nM Q06187 30857747 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 6hrq A 1.845 BS02 GM5 A 1 H142 F151 D186 H188 F216 P291 H292 Y341 H141 F150 D177 H179 F207 P276 H277 Y314 3.5.1.98 0004407,0005634,0006325,0031507,0046872 Kd=81.7nM remove_due_to_license_issue IC50=95nM, Kd=82nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPLDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hrt A 1.36 BS01 GMW A 1 L408 V416 A428 K430 Y476 M477 A478 N479 G480 N526 L528 D539 L542 Y551 L13 V21 A33 K35 Y81 M82 A83 N84 G85 N131 L133 D144 L147 Y156 D521 A523 R525 N526 D539 D126 A128 R130 N131 D144 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=<1.000000nM Q06187 30857747 701 EIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREARHAFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASAAVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 6hrw A 2.45 BS01 GNK A 1 E70 V73 M74 W100 A130 S134 L167 D168 E60 V63 M64 W90 A120 S124 L157 D158 ? 0000976,0003677,0003700,0005886,0006355 ic50=1uM remove_due_to_license_issue O53623 30784877 301 RSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLNG 6hrx A 1.87 BS01 GO8 A 1 E70 W100 A130 S134 D168 E62 W92 A122 S126 D160 ? 0000976,0003677,0003700,0005886,0006355 ic50=0.00000001M remove_due_to_license_issue O53623 30784877 301 EERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLNG 6hrx B 1.87 BS01 GO8 B 1 E70 M77 W100 A130 S134 L167 D168 E60 M67 W90 A120 S124 L157 D158 ? 0000976,0003677,0003700,0005886,0006355 ic50=0.00000001M remove_due_to_license_issue O53623 30784877 301 RSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6hry A 1.84 BS01 GOE A 1 E70 M74 W100 L114 A130 S134 D168 E60 M64 W90 L104 A120 S124 D158 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 30784877 301 RSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLNG 6hry B 1.84 BS01 GOE B 1 E70 M74 M77 W100 F126 V129 A130 S134 L167 D168 E67 M71 M74 W97 F123 V126 A127 S131 L164 D165 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 30784877 301 KRRTQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLNG 6hrz A 1.57 BS01 GO2 A 1 W100 T138 I164 L167 D168 W94 T132 I158 L161 D162 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 30784877 301 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLNG 6hrz A 1.57 BS02 GO2 A 2 E70 V73 M74 M77 Y133 S134 M137 E64 V67 M68 M71 Y127 S128 M131 ? 0000976,0003677,0003700,0005886,0006355 remove_due_to_license_issue O53623 30784877 302 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLNG 6hs0 A 1.45 BS01 GNW A 1 A96 V97 W100 S134 L141 I164 L167 D168 A90 V91 W94 S128 L135 I158 L161 D162 ? 0000976,0003677,0003700,0005886,0006355 ic50=0.00000001M remove_due_to_license_issue O53623 30784877 301 TQEERSAATREALITGARKLWGLRGYAEVGTPEIATEAGVTRGAMYHQFADKAALFRDVVEVVEQDVMARMATLVAASGAATPADAIRAAVDAWLEVSGDPEVRQLILLDAPVVLGWAGFRDVAQRYSLGMTEQLITEAIRAGQLARQPVRPLAQVLIGALDEAAMFIATADDPKRARRETRQVLRRLIDGMLN 6hs4 A 2.05 BS01 GON A 1 L186 P187 A189 L157 P158 A160 ? ic50=3.1uM remove_due_to_license_issue Q05320 30785281 607 GRSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQASGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTEWAFWETSEELSFTVVAAAAAAAA 6hs4 A 2.05 BS02 GON A 2 R64 V66 E100 R35 V37 E71 ? ic50=3.1uM remove_due_to_license_issue Q05320 30785281 608 GRSIPLGVIHNSALQVSDVDKLVCRDKLSSTNQLRSVGLNLEGNGVATDVPSATKRWGFRSGVPPKVVNYEAGEWAENCYNLEIKKPDGSECLPAAPDGIRGFPRCRYVHKVSGTGPCAGDFAFHKEGAFFLYDRLASTVIYRGTTFAEGVVAFLILPQASGYYSTTIRYQATGFGTNETEYLFEVDNLTYVQLESRFTPQFLLQLNETIYTSGKRSNTTGKLIWKVNPEIDTTEWAFWETSEELSFTVVAAAAAAAA 6hs4 B 2.05 BS01 GON A 1 M548 L554 M47 L53 ? remove_due_to_license_issue Q05320 30785281 607 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFV 6hs4 B 2.05 BS02 GON A 2 L515 Y517 T519 D522 M548 L14 Y16 T18 D21 M47 ? remove_due_to_license_issue Q05320 30785281 608 EAIVNAQPKCNPNLHYWTTQDEGAAIGLAWIPYFGPAAEGIYIEGLMHNQDGLICGLRQLANETTQALQLFLRATTELRTFSILNRKAIDFLLQRWGGTCHILGPDCCIEPADWTKNITDKIDQIIHDFV 6hsh A 1.545 BS02 GOK A 1 D100 H142 G150 F151 D186 H188 F216 Y341 D99 H141 G149 F150 D177 H179 F207 Y313 3.5.1.98 0004407,0005634,0006325,0031507,0046872 Kd=28.4nM remove_due_to_license_issue Kd=28nM, IC50=303nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPCSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPHESHNDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hsk A 2.096 BS02 GOK A 1 H142 H143 G151 F152 D178 H180 G206 F208 P209 Y306 H129 H130 G138 F139 D165 H167 G193 F195 P196 Y293 3.5.1.-,3.5.1.98 0000118,0000122,0000228,0004407,0005515,0005634,0005654,0005694,0005737,0006325,0007064,0016787,0030544,0031078,0031397,0031647,0032129,0032204,0033558,0034739,0040029,0042903,0046872,0051879,0140297,0140937,0160008,0160009,0180032,0180033,1990162 remove_due_to_license_issue IC50=64nM, Ki=24nM, Kd=23nM Q9BY41 30347148 404 LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYALHKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGYDCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEASGFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSLHKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKEVYQAFNPKAVVLQLGADTISGDRLGCFNMTPVGIGKCLKYILQWQLATLILGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITPSCRPDRNEPHRIQQILNYIKGNLKHVV 6hsz A 2.374 BS02 GOW A 1 K20 H141 H142 G150 D186 H188 F216 H292 Y341 K19 H140 H141 G149 D176 H178 F206 H275 Y311 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=116nM remove_due_to_license_issue IC50=116nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQ 6ht1 A 2.1 BS01 GQ5 A 1 F28 H56 S58 F59 P60 E75 S76 G77 Y78 A79 G80 F27 H55 S57 F58 P59 E74 S75 G76 Y77 A78 G79 ? Kd=0.077uM remove_due_to_license_issue Q03111 30288907 210 DNQCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6ht8 A 2.497 BS02 GQE A 1 K20 D100 H141 H142 G150 D186 H188 F216 H292 Y341 K19 D99 H140 H141 G149 D176 H178 F206 H276 Y312 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=190nM remove_due_to_license_issue IC50=190nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6htc H 2.8 BS01 GQK H 1 T1 T21 E22 C31 K33 G47 T48 A49 G168 T1 T21 E22 C31 K33 G47 T48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6htd H 3.0 BS01 GQH H 1 T1 T21 K33 G47 A49 D53 G128 S129 T1 T21 K33 G47 A49 D53 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6htd I 3.0 BS01 GQH H 1 D124 L125 D124 L125 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6htg A 1.939 BS02 T61 A 1 K20 H142 D186 H188 F216 H292 Y341 K19 H141 D176 H178 F206 H277 Y313 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=67nM remove_due_to_license_issue IC50=68nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hth A 1.95 BS02 GQN A 1 K20 H141 H142 G150 H188 F216 P291 H292 Y341 K19 H140 H141 G149 H178 F206 P274 H275 Y311 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=75nM remove_due_to_license_issue IC50=76nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKL 6hti A 1.693 BS02 GQW A 1 K20 H141 H142 G150 D186 H188 F216 P291 H292 Y341 K19 H140 H141 G149 D175 H177 F205 P276 H277 Y313 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=97nM remove_due_to_license_issue IC50=97nM A5H660 30347148 505 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMKLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6htn A 1.55 BS01 MFU A 1 R16 E29 G40 A41 W82 W87 R15 E28 G39 A40 W81 W86 ? 0030246 Kd=0.86uM remove_due_to_license_issue A0A2T6C3M6 30853410 201 GATSWLDGSGQIHLRIYSLQQSNGKLLERCWDSNKWYDGALTNQFSAISGAGATSWLDSSGQIHIRVYAIGTDGKIIELCWDKDKWYSGALTGQFYGASTPDATSWLDKNGQIHIRVYAYNQDNVQKEYCWDGSKWYVGAYTE 6htn A 1.55 BS02 MFU A 2 R67 E79 A91 W132 W137 R66 E78 A90 W131 W136 ? 0030246 Kd=0.86uM remove_due_to_license_issue A0A2T6C3M6 30853410 202 GATSWLDGSGQIHLRIYSLQQSNGKLLERCWDSNKWYDGALTNQFSAISGAGATSWLDSSGQIHIRVYAIGTDGKIIELCWDKDKWYSGALTGQFYGASTPDATSWLDKNGQIHIRVYAYNQDNVQKEYCWDGSKWYVGAYTE 6htn A 1.55 BS03 MFU A 3 R117 E129 G140 A141 R116 E128 G139 A140 ? 0030246 Kd=0.86uM remove_due_to_license_issue A0A2T6C3M6 30853410 203 GATSWLDGSGQIHLRIYSLQQSNGKLLERCWDSNKWYDGALTNQFSAISGAGATSWLDSSGQIHIRVYAIGTDGKIIELCWDKDKWYSGALTGQFYGASTPDATSWLDKNGQIHIRVYAYNQDNVQKEYCWDGSKWYVGAYTE 6htn A 1.55 BS04 MFU B 3 L15 W32 W37 L14 W31 W36 ? 0030246 Kd=0.86uM remove_due_to_license_issue A0A2T6C3M6 30853410 203 GATSWLDGSGQIHLRIYSLQQSNGKLLERCWDSNKWYDGALTNQFSAISGAGATSWLDSSGQIHIRVYAIGTDGKIIELCWDKDKWYSGALTGQFYGASTPDATSWLDKNGQIHIRVYAYNQDNVQKEYCWDGSKWYVGAYTE 6htp H 3.0 BS01 GQQ H 1 T1 A20 T21 G47 A49 D53 S129 T1 A20 T21 G47 A49 D53 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6htp I 3.0 BS01 GQQ H 1 D124 L125 D124 L125 3.4.25.1 0005839,0019774,0043161,0051603 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6htr H 2.6 BS01 GQT H 1 T1 T21 C31 K33 G45 G47 A49 D53 S129 T1 T21 C31 K33 G45 G47 A49 D53 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6htt A 1.748 BS02 GQZ A 1 K20 H141 H142 D186 H188 F216 P291 H292 Y341 K19 H140 H141 D176 H178 F206 P274 H275 Y312 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=220nM remove_due_to_license_issue A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6htu A 2.888 BS01 rna D 0 E191 P211 H212 F216 K232 S233 K234 E12 P32 H33 F37 K53 S54 K55 ? remove_due_to_license_issue O95793 30456389 75 ~ 93 HMNKSEISQVFEIALKRNLPVNFEVARESGPPHMKNFVTKVSVGEFVGEGEGKSKKISKKNAAIAVLEELKKLPPL 6htu A 2.888 BS02 rna F 0 S184 I186 S187 P211 H212 K238 S5 I7 S8 P32 H33 K59 ? remove_due_to_license_issue O95793 30456389 194 ~ 212 HMNKSEISQVFEIALKRNLPVNFEVARESGPPHMKNFVTKVSVGEFVGEGEGKSKKISKKNAAIAVLEELKKLPPL 6htu B 2.888 BS01 rna D 0 S184 S187 F190 K238 S5 S8 F11 K59 ? remove_due_to_license_issue O95793 30456389 75 ~ 93 HMNKSEISQVFEIALKRNLPVNFEVARESGPPHMKNFVTKVSVGEFVGEGEGKSKKISKKNAAIAVLEELKKLPPL 6htu B 2.888 BS02 rna F 0 M181 E191 L194 F216 K232 S233 K234 M2 E12 L15 F37 K53 S54 K55 ? remove_due_to_license_issue O95793 30456389 194 ~ 212 HMNKSEISQVFEIALKRNLPVNFEVARESGPPHMKNFVTKVSVGEFVGEGEGKSKKISKKNAAIAVLEELKKLPPL 6htu C 2.888 BS01 rna D 0 N336 K337 N46 K47 ? remove_due_to_license_issue O95793 30456389 75 ~ 93 GINPISRLAQIQQAKEPEYTLLTPRRREFVMQVKVGNHTAEGTGTNKKVAKRNAAENMLEILGFK 6htu C 2.888 BS02 rna F 0 N286 I288 S289 N3 I5 S6 ? remove_due_to_license_issue O95793 30456389 194 ~ 212 GINPISRLAQIQQAKEPEYTLLTPRRREFVMQVKVGNHTAEGTGTNKKVAKRNAAENMLEILGFK 6htz A 1.841 BS02 GRK A 1 K20 H141 H142 G150 D186 H188 F216 Y341 K19 H140 H141 G149 D177 H179 F207 Y314 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=183nM remove_due_to_license_issue IC50=183nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPLDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hu0 A 1.746 BS02 T86 A 1 K20 D100 H141 H142 G150 D186 H188 F216 H292 Y341 K19 D99 H140 H141 G149 D175 H177 F205 H274 Y311 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=122nM remove_due_to_license_issue IC50=120nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPNLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLI 6hu1 A 1.996 BS02 GT2 A 1 K20 H141 H142 G150 D186 H188 F216 H292 Y341 K19 H140 H141 G149 D176 H178 F206 H276 Y313 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=191nM remove_due_to_license_issue IC50=191nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPHEDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQ 6hu2 A 1.986 BS02 T34 A 1 K20 H142 G150 D186 H188 F216 H292 Y341 K19 H141 G149 D178 H180 F208 H278 Y315 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=1260nM remove_due_to_license_issue A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTRQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hu3 A 1.655 BS02 GRZ A 1 H141 H142 D186 H188 F216 P291 H292 Y341 H140 H141 D175 H177 F205 P276 H277 Y315 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=504nM remove_due_to_license_issue IC50=504nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMKLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPNLLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hu3 A 1.655 BS03 GRZ B 1 Q48 W49 D50 Q47 W48 D49 3.5.1.98 0004407,0005634,0006325,0031507,0046872 ic50=504nM remove_due_to_license_issue IC50=504nM A5H660 30347148 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNMKLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPNLLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6hub H 2.9 BS01 GRW H 1 T1 T21 G47 T48 A49 D53 S129 T1 T21 G47 T48 A49 D53 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6huc H 3.0 BS01 GRT H 1 T1 T21 C31 G47 A49 D53 S129 T1 T21 C31 G47 A49 D53 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6huc I 3.0 BS01 GRT H 1 D124 I126 D124 I126 3.4.25.1 0005839,0019774,0043161,0051603 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6huq H 3.0 BS01 GT5 H 1 T1 T21 E22 G47 A49 D53 G128 S129 T1 T21 E22 G47 A49 D53 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6huq I 3.0 BS01 GT5 H 1 D124 L125 D124 L125 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6huu H 2.8 BS01 GTW H 1 T1 T21 G47 A49 D53 G128 S129 T1 T21 G47 A49 D53 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6huu I 2.8 BS01 GTW H 1 D124 L125 D124 L125 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6huu Z 2.8 BS01 GTW Y 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 30657666 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 6huv H 3.1 BS01 GT8 H 1 T1 T21 C31 H35 G45 A46 G47 A49 G168 T1 T21 C31 H35 G45 A46 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue Q99436 30657666 301 TTIAGVVYKDGIVLGADTRATEGMVVADKNCSKIHFISPNIYCCGAGTAADTDMTTQLISSNLELHSLSTGRLPRVVTANRMLKQMLFRYQGYIGAALVLGGVDVTGPHLYSIYPHGSTDKLPYVTMGSGSLAAMAVFEDKFRPDMEEEEAKNLVSEAIAAGIFNDLGSGGNIDLCVISKNKLDFLRPYTVPNKKGTRLGRYRCEKGTTAVLTEKITPL 6hv0 A 2.73 BS01 GUK A 1 L577 K599 I642 L644 C645 F712 L714 L16 K38 I68 L70 C71 F135 L137 D688 K690 N693 D711 T734 D111 K113 N116 D134 T157 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 remove_due_to_license_issue O75460 30779566 1001 SVVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPECSDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFGLEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCKKLAVGRHSFSRRSGVPGTEGWIAPEMNPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDLRRTYKGGSVRDLLRAMRNKKHHYRELPAEVRETLGSLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFH 6hv4 H 3.0 BS01 GQK H 1 T1 A20 T21 G47 V48 A49 T1 A20 T21 G47 V48 A49 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hv5 H 3.0 BS01 GQH H 1 T1 A20 T21 N22 K33 G47 A49 S129 T1 A20 T21 N22 K33 G47 A49 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hv7 H 3.4 BS01 GQQ H 1 T1 A20 T21 N22 G47 V48 A49 E53 S129 T1 A20 T21 N22 G47 V48 A49 E53 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hv7 I 3.4 BS01 GQQ H 1 D124 L125 C128 D124 L125 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6hv7 Z 3.4 BS01 GQQ Y 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 30657666 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 6hva H 2.9 BS01 GQT H 1 T1 A20 T21 N22 A27 K33 G47 V48 A49 G128 S129 T1 A20 T21 N22 A27 K33 G47 V48 A49 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hvh A 2.36 BS01 GV2 A 1 R45 Y49 I50 S152 C154 V159 N163 E166 V167 V214 V217 I241 V243 R30 Y34 I35 S137 C139 V144 N148 E151 V152 V199 V202 I226 V228 R252 H253 N259 S302 E322 H387 R237 H238 N244 S287 E307 H372 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=0.047uM remove_due_to_license_issue Q16875 30378281 601 ELTQSRVQKIWVPVDHNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERSE 6hvi A 1.96 BS01 GV5 A 1 R45 G46 Y49 I50 S152 C154 V159 N163 E166 V214 V217 I241 V243 R32 G33 Y36 I37 S139 C141 V146 N150 E153 V201 V204 I228 V230 R252 H253 N259 S302 E322 H387 R239 H240 N246 S289 E309 H374 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=0.38uM remove_due_to_license_issue Q16875 30378281 601 PLELTQSRVQKIWVPVHRNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERSE 6hvj A 2.28 BS01 GV8 A 1 R45 Y49 I50 S152 C154 V159 N163 V167 V214 I241 A423 R29 Y33 I34 S136 C138 V143 N147 V151 V198 I225 A407 R252 H253 N259 S302 E322 H387 R236 H237 N243 S286 E306 H371 2.7.1.105,3.1.3.46 0003824,0003873,0004331,0005515,0005524,0005654,0005829,0006000,0006003,0006096,0006915,0010001,0016301,0016787,0046835,0061744 ic50=0.028uM remove_due_to_license_issue Q16875 30378281 601 ELTQSRVQKIWVPVHNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERSE 6hvr H 2.7 BS01 GRW H 1 T1 A20 T21 G47 A49 G128 T1 A20 T21 G47 A49 G128 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hvr I 2.7 BS01 GRW H 1 D124 L125 C128 D124 L125 C128 3.4.25.1 0005839,0019774,0043161,0051603 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6hvs H 3.1 BS01 GRT H 1 T1 T21 N22 C31 K33 G45 G47 A49 S129 T1 T21 N22 C31 K33 G45 G47 A49 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hvs I 3.1 BS01 GRT H 1 D124 L125 C128 D124 L125 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6hvt H 2.9 BS01 GT5 H 1 T1 A20 T21 N22 G47 A49 G128 S129 T1 A20 T21 N22 G47 A49 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hvt I 2.9 BS01 GT5 H 1 D124 L125 C128 D124 L125 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6hvt Z 2.9 BS01 GT5 Y 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 30657666 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 6hvu H 2.9 BS01 GTW H 1 T1 A20 T21 N22 G47 A49 G128 S129 T1 A20 T21 N22 G47 A49 G128 S129 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hvu I 2.9 BS01 GTW H 1 L125 C128 L125 C128 3.4.25.1 0000502,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603,0061133 remove_due_to_license_issue P25451 30657666 301 SDPSSINGGIVVAMTGKDCVAIACDLRLGSQSLGVSNKFEKIFHYGHVFLGITGLATDVTTLNEMFRYKTNLYKLKEERAIEPETFTQLVSSSLYERRFGPYFVGPVVAGINSKSGKPFIAGFDLIGCIDEAKDFIVSGTASDQLFGMCESLYEPNLEPEDLFETISQALLNAADRDALSGWGAVVYIIKKDEVVKRYLKMRQD 6hvu Z 2.9 BS01 GTW Y 1 D126 P127 D126 P127 3.4.25.1 0000502,0003674,0005515,0005634,0005737,0005829,0005839,0010499,0019774,0043161,0051603 remove_due_to_license_issue P23724 30657666 301 QFNPYGDNGGTILGIAGEDFAVLAGDTRNITDYSINSRYEPKVFDCGDNIVMSANGFAADGDALVKRFKNSVKWYHFDHNDKKLSINSAARNIQHLLYGKRFFPYYVHTIIAGLDEDGKGAVYSFDPVGSYEREQCRAGGAAASLIMPFLDNQVNFKNQYEPGTNGKVKKPLKYLSVEEVIKLVRDSFTSATERHIQVGDGLEILIVTKDGVRKEFYELKRD 6hvv H 2.7 BS01 GT8 H 1 T1 A20 T21 K33 G45 G47 V48 A49 G168 T1 A20 T21 K33 G45 G47 V48 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hvw H 3.0 BS01 GVW H 1 T1 T21 C31 G45 G47 A49 G168 T1 T21 C31 G45 G47 A49 G168 T1 D17 R19 K33 G47 S129 D166 S169 T1 D17 R19 K33 G47 S129 D166 S169 3.4.25.1 0004298,0005839,0051603 remove_due_to_license_issue P25043,P40306 30657666 301 TTIAGLVFQDGVILGADTRATNDSVVADKSCEKIHFIAPKIYCCGAGVAADAEAVTQLIGSNIELHSLYTSREPRVVSALQMLKQHLFKYQGHIGAYLIVAGVDPTGSHLFSIHAHGSTDVGYYLSLGSGSLAAMAVLESHWKQDLTKEEAIKLASDAIQAGIWNDLGSGSNVDVCVMEIGKDAEYLRNYLTPNVREEKQKSYKFPRGTTAVLKESIVNICDIQEE 6hwu A 2.3 BS01 GE5 A 1 V30 G33 A34 A51 K53 L104 V105 T106 M109 F169 G170 L171 V26 G29 A30 A47 K49 L100 V101 T102 M105 F160 G161 L162 D150 K152 N155 D168 T185 D141 K143 N146 D159 T165 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=54.7nM remove_due_to_license_issue Q16539 30924488 404 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNILTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 6hwv A 1.7 BS01 GEW A 1 Y35 A51 K53 L104 V105 T106 M109 G110 F169 A172 Y31 A47 K49 L100 V101 T102 M105 G106 F165 A168 D150 K152 N155 D168 T185 D146 K148 N151 D164 T169 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=115nM remove_due_to_license_issue Q16539 30924488 404 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 6hwz A 1.64 BS02 GXE A 1 H95 L199 T200 H90 L194 T195 H65 H95 H97 E107 H120 T200 H60 H90 H92 E102 H115 T195 4.2.1.1,4.2.1.69 0004064,0004089,0005515,0005737,0005829,0006730,0008270,0016829,0016836,0018820,0046872,0070062 Ki=6.7uM remove_due_to_license_issue P00915 30560259 302 WGYDDKNGPEQWSKLYPIANGNNQSPVDIKTSETKHDTSLKPISVSYNPATAKEIINVGHSFHVNFEDNDNRSVLKGGPFSDSYRLFQFHFHWGSTNEHGSEHTVDGVKYSAELHVAHWNSAKYSSLAEAASKADGLAVIGVLMKVGEANPKLQKVLDALQAIKTKGKRAPFTNFDPSTLLPSSLDFWTYPGSLTHPPLYESVTWIICKESISVSSEQLAQFRSLLSNVEGDNAVPMQHNNRPTQPLKGRTVRASF 6hx1 A 2.14 BS01 GXK A 1 L577 G578 K599 Y628 I642 C645 A646 F712 L714 H723 L16 G17 K38 Y57 I71 C74 A75 F141 L143 H150 D688 K690 N693 D711 T734 D117 K119 N122 D140 T161 2.7.11.1,3.1.26.- 0004521,0004540,0004672,0004674,0005524,0006397,0006468,0030968 ic50=1.6uM remove_due_to_license_issue O75460 30779566 1001 SVVIVGKISFCPKDVLGHGAEGTIVYRGMFDNRDVAVKRILPECFRESDEHPNVIRYFCTEKDRQFQYIAIELCAATLQEYVEQKDFAHLGLEPITLLQQTTSGLAHLHSLNIVHRDLKPHNILISMPNAHGKIKAMISDFGLCKKVGRHSFSRRSGVPGTEGWIAPEMLSENPTYTVDIFSAGCVFYYVISEGSHPFGKSLQRQANILLGACSLDCLHPEKHEDVIARELIEKMIAMDPQKRPSAKHVLKHPFFWSLEKQLQFFQDVSDRIEKESLDGPIVKQLERGGRAVVKMDWRENITVPLQTDLRKFRTYKGGSVRDLLRAMRNKKHHYRELPAEVRETLGSLPDDFVCYFTSRFPHLLAHTYRAMELCSHERLFQPYYFHE 6hx5 A 1.44 BS02 GXE A 1 H94 V121 L198 T199 H91 V118 L194 T195 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=2.2uM remove_due_to_license_issue P00918 30560259 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6hx8 A 2.402 BS03 GXN B 1 S178 T179 A180 V181 S178 T179 A180 V181 3.6.5.- 0000226,0000278,0003725,0003924,0005200,0005525,0005737,0005829,0005856,0005874,0005881,0007017,0015630,0016787,0031625,0046872,0071353 remove_due_to_license_issue P81947 30775645 502 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGV 6hx8 B 2.402 BS02 GXN B 1 V238 C241 L248 N258 A317 I318 N349 K352 A354 I378 V236 C239 L246 N256 A310 I311 N342 K345 A347 I363 ? 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0007399,0015630,0046872,0046982,1902669 remove_due_to_license_issue Q6B856 30775645 502 MREIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQD 6hys A 2.6 BS01 ADP A 1 L565 T590 G591 S592 G593 K594 T595 T596 R629 F825 D849 R893 L11 T36 G37 S38 G39 K40 T41 T42 R75 F271 D295 R339 3.6.4.13 0000398,0003676,0003724,0005524 remove_due_to_license_issue Q14562 31409651 1301 QMSILEQRESLPIYKLKEQLVQAVHDNQILIVIGETGSGKTTQITQYLAEAGYTSRGKIGCTQPRRVAAMSVAKRVSEEFGCCLGQEVGYTIRFEDCTSPETVIKYMTDGMLLRECLIDPDLTQYAIIMLDEAHERTIHTDVLFGLLKKTVQKRQDMKLIVTSATLDAVKFSQYFYEAPIFTIPGRTYPVEILYTKEPETDYLDASLITVMQIHLTEPPGDILVFLTGQEEIDTACEILYERMKSLGPDVPELIILPVYSALPSEMQTRIFDPAPPGSRKVVIATNIAETSLTIDGIYYVVDPGFVKQKVYNSKTGIDQLVVTPISQAQAKQRAGRAGRTGPGKCYRLYTERAYRDEMLTTNVPEIQRTNLASTVLSLKAMGINDLLSFDFMDAPPMETLITAMEQLYTLGALDDEGLLTRLGRRMAEFPLEPMLCKMLIMSVHLGCSEEMLTIVSMLSVQNVFYRPKDKQALADQKKAKFHQTEGDHLTLLAVYNSWKNNKFSNPWCYENFIQARSLRRAQDIRKQMLGIMDRHKLDVVSCGKSTVRVQKAICSGFFRNAAKKDPQEGYRTLIDQQVVYIHPSSALFNRQPEWVVYHELVLTTKEYMREVTTIDPRWLVEFAPAFFKVSDP 6hzp A 2.5 BS01 FVT A 1 N167 N347 N159 N339 0006857,0015833,0016020,0022857,0055085,1904680 remove_due_to_license_issue 30602453 501 QTIQSIPQKGFFGHPRGLGVLFFVEFWERFSYYGMRAMLIFYMYFAIHQNGLGIDKTTAMSIMSVYGALIYMSSIPGAWIADRITGTRGATLLGAVLIIIGHICLSLPFALFGLFSSMFFIIIGSGLMKPNISNIVGRLYPENDTRIDAGFVIFYMSVNLGALISPIILQHFVDIRNFHGGFLLAAIGMALGLVWYLLFNRKNLGSVGMKPTNPLSKEEKRKYGMIIGIIVAIVIVVLLVTYYTHTLSFDLISNTVLVLGVALPIIYFTTMLRSKDVTDGERSRVKAFIPLFILGMLFWSIQEQGSNVLNIYGLERSDMQLNLFGWTTRFGEALFQSINPLFILLFAPVISMIWLKMGKKQPSLAIKFSIGTLLAGLSYILIGLVGLGYGHTQFSVNWVILSYVICVIGELCLSPTGNSAAVKLAPKAFNAQMMSVWLLTNASAQAINGTLVKLIKPLGQTNYFIFLGTVAIVITLIILVFSPKITK 6hzu A 2.2 BS01 GYQ A 1 L881 G882 E883 G887 V889 A906 M956 E957 F958 G962 E966 L1010 D1021 L29 G30 E31 G35 V37 A54 M96 E97 F98 G102 E106 L150 D161 D1003 A1005 R1007 N1008 D1021 D143 A145 R147 N148 D161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=5.5nM remove_due_to_license_issue P23458 31609613 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6hzv A 2.46 BS01 GYW A 1 L828 A853 V884 M902 Y904 L905 G908 C909 D912 R953 L956 L14 A39 V68 M82 Y84 L85 G88 C89 D92 R133 L136 D949 R953 N954 D967 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 ic50=59nM remove_due_to_license_issue IC50=59nM P52333 31609613 1101 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQGPDQQRDFQREIQILKALHSDFIVKYRGVSYQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVRPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML 6hzy A 1.7 BS01 GYZ A 1 H66 E87 W88 H135 W227 D229 R262 G286 E288 W316 H31 E52 W53 H100 W192 D194 R227 G251 E253 W281 ? 0004553,0004560,0005764,0005975,0006004,0016139,0016798 Ki=121uM remove_due_to_license_issue Q8A3I4 30663832 512 IPLKYGATNEGKRQDPAMQKFRDNRLGAFIHWGLYAIPGGEWNGKVYGGAAEWLKSWAKVPADEWLKLMDQWNPTKFDAKKWAKMAKEMGTKYVKITTKHHEGFCLWPSKYTKYTVANTPYKRDILGELVKAYNDEGIDVHFYFSVMDWSNPDYRYDIKSKEDSIAFSRFLEFTDNQLKELATRYPTVKDFWFDGTWDASVKKNGWWTAHAEQMLKELVPGVAINSRLRADDKGKRHFDSNGRLMGDYESGYERRLPDPVKDLKVTQWDWEACMTIPENQWGYHKDWSLSYVKTPIEVIDRIVHAVSMGGNMVVNFGPQADGDFRPEEKAMATAIGKWMNRYGKAVYACDYAGFEKQDWGYYTRGKNDEVYMVVFNQPYSERLIVKTPKGITVEKATLLTTGEDITVVETTRNEYNVSVPKKNPGEPYVIQLKVRAAK 6i0c A 2.675 BS02 GZ5 A 1 W82 G116 G117 P285 L286 S287 A328 Y332 W430 H438 W79 G113 G114 P282 L283 S284 A325 Y329 W427 H435 G116 G117 G149 S198 A199 Y237 V288 F290 E325 H438 G113 G114 G146 S195 A196 Y234 V285 F287 E322 H435 3.1.1.8 0001540,0003824,0003990,0004104,0005515,0005576,0005615,0005641,0005783,0005788,0005886,0006581,0006805,0007584,0007612,0008285,0009410,0014016,0016486,0016788,0019695,0019899,0033265,0042802,0043279,0050783,0050805,0051384,0051593,0052689,0072562 remove_due_to_license_issue P06276 30851693 613 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6i0k A 1.64 BS02 GZ8 A 1 H19 F21 D35 S36 M59 N109 S124 H193 S209 T210 H22 F24 D38 S39 M62 N112 S127 H196 S212 T213 2.5.1.72 0005737,0005829,0008987,0009435,0016740,0016765,0019363,0019805,0034628,0046872,0051539 remove_due_to_license_issue Q9X1X7 30855610 302 HHHMVDEILKLKKEKGYIILAHNFQIPELQDIADFVGDSLQLARKAMELSEKKILFLGVDFMAELVKILNPDKKVIVPDRSATCPMANRLTPEIIREYREKFPDAPVVLYVNSTSECKTLADVICTSANAVEVVKKLDSSVVIFGPDRNLGEYVAEKTGKKVITIPENGHCPVHQFNAESIDAVRKKYPDAKVIVHPECPKPVRDKADYVGSTGQMEKIPERDPSRIFVIGTEIGMIHKLKKKFPDREFVPLEMAVCVNMKKNTLENTLHALQTESFEVILPKEVIEKAKKPILRMFELMG 6i0p A 1.9 BS02 QAS A 1 H19 F21 D35 S36 M59 N109 H193 S209 T210 H22 F24 D38 S39 M62 N112 H196 S212 T213 2.5.1.72 0005737,0005829,0008987,0009435,0016740,0016765,0019363,0019805,0034628,0046872,0051539 remove_due_to_license_issue Q9X1X7 30855610 302 HHHMVDEILKLKKEKGYIILAHNFQIPELQDIADFVGDSLQLARKAMELSEKKILFLGVDFMAELVKILNPDKKVIVPDRSATCPMANRLTPEIIREYREKFPDAPVVLYVNSTSECKTLADVICTSANAVEVVKKLDSSVVIFGPDRNLGEYVAEKTGKKVITIPENGHCPVHQFNAESIDAVRKKYPDAKVIVHPECPKPVRDKADYVGSTGQMEKIPERDPSRIFVIGTEIGMIHKLKKKFPDREFVPLEMAVCVNMKKNTLENTLHALQTESFEVILPKEVIEKAKKPILRMFELMG 6i0r A 2.1 BS02 QAT A 1 H19 D35 S36 Y107 H193 S209 T210 H24 D40 S41 Y112 H198 S214 T215 2.5.1.72 0005737,0005829,0008987,0009435,0016740,0016765,0019363,0019805,0034628,0046872,0051539 remove_due_to_license_issue Q9X1X7 30855610 309 HHHHHMVDEILKLKKEKGYIILAHNFQIPELQDIADFVGDSLQLARKAMELSEKKILFLGVDFMAELVKILNPDKKVIVPDRSATCPMANRLTPEIIREYREKFPDAPVVLYVNSTSECKTLADVICTSANAVEVVKKLDSSVVIFGPDRNLGEYVAEKTGKKVITIPENGHCPVHQFNAESIDAVRKKYPDAKVIVHPECPKPVRDKADYVGSTGQMEKIPERDPSRIFVIGTEIGMIHKLKKKFPDREFVPLEMAVCVNMKKNTLENTLHALQTESFEVILPKEVIEKAKKPILRMFELMG 6i0x A 1.6 BS01 BFB A 1 W127 D130 R152 R154 Y233 I234 H236 D238 T346 C351 W84 D87 R109 R111 Y190 I191 H193 D195 T303 C308 3.5.3.- 0004668,0009446 remove_due_to_license_issue Q9RQJ2 30638292 502 AFQETNPPAGPVRAIAEYERSAAVLVRYPFGIPMELIKELAKNDKVITIVASESQKNTVITQYTQSGVNLSNCDFIIAKTDSYWTRDYTGWFAMYDTNKVGLVDFIYNRPRPNDDEFPKYEAQYLGIEMFGMKLKQTGGNYMTDGYGSAVQSHIAYTENSSLSQAQVNQKMKDYLGITHHDVVQDPNNTYIDHVDCWGKYLAPNKILIRKVPDNHPQHQALEDMAAYFAAQTCAWGTKYEVYRALATNEQPYTNSLILNNRVFVPVNGPASVDNDALNVYKTAMPGYEIIGVKGASGTPWLGTDALHCRTHEVADKGYLYIKHYPILGEQAGPDYKIEADVVSCANATISPVQCYYRINGSGSFKAADMTMESTGHYTYSFTGLNKNDKVEYYISAADNSGRKETYPFIGEPDPFKFTCM 6i0z A 1.77 BS01 GZQ A 1 F14 I93 W101 V134 F181 Y186 L214 F9 I88 W96 V129 F176 Y181 L209 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=92uM remove_due_to_license_issue Kd=92000nM Q16658 30773430 501 TAEAVQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i10 A 2.1 BS01 GZK A 1 F14 L48 A58 I93 W101 V134 E215 F216 R217 F4 L38 A48 I83 W91 V124 E205 F206 R207 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=29.5uM remove_due_to_license_issue IC50=734nM, Kd=29300nM Q16658 30773430 501 QIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i11 A 1.67 BS01 H0H A 1 F14 L48 I93 W101 V134 L214 E215 F216 R217 F5 L39 I84 W92 V125 L205 E206 F207 R208 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=29.3uM remove_due_to_license_issue IC50=67900nM, Kd=29300nM Q16658 30773430 502 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i12 A 1.65 BS01 H08 A 1 L48 I93 W101 V134 E215 F216 R217 L39 I84 W92 V125 E206 F207 R208 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=2.7uM remove_due_to_license_issue IC50=4600nM, Kd=2700nM Q16658 30773430 502 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i13 A 1.79 BS01 H0Q A 1 L48 I93 W101 V134 E215 F216 R217 L39 I84 W92 V125 E206 F207 R208 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=7.6uM remove_due_to_license_issue IC50=11400nM, Kd=7600nM Q16658 30773430 505 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i14 A 1.73 BS01 GZN A 1 F14 L48 I93 W101 V134 E215 F216 R217 F5 L39 I84 W92 V125 E206 F207 R208 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=1.5uM remove_due_to_license_issue IC50=1300nM, Kd=1500nM Q16658 30773430 502 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i15 A 1.91 BS01 GZT A 1 L48 I93 W101 V134 E215 F216 R217 L39 I84 W92 V125 E206 F207 R208 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 remove_due_to_license_issue Q16658 30773430 504 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i16 A 2.0 BS01 H0B A 1 F14 L48 Q50 S57 A58 I93 W101 V134 E215 F216 F5 L39 Q41 S48 A49 I84 W92 V125 E206 F207 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 remove_due_to_license_issue Kd=>100000nM Q16658 30773430 502 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i17 A 1.56 BS01 GZW A 1 F14 L48 A58 I93 A95 W101 V134 L214 E215 F216 R217 R224 F5 L39 A49 I84 A86 W92 V125 L205 E206 F207 R208 R215 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=0.25uM remove_due_to_license_issue Q16658 30773430 503 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i18 A 1.49 BS01 H0N A 1 F14 L16 L48 I93 W101 V134 E215 F216 R217 F5 L7 L39 I84 W92 V125 E206 F207 R208 ? 0001725,0001726,0002102,0003723,0003779,0005515,0005737,0005829,0005856,0005902,0005911,0005938,0007015,0007043,0007163,0008144,0010592,0015629,0016477,0030027,0030035,0030036,0030046,0030175,0030426,0030674,0031253,0032534,0032956,0035089,0042995,0044393,0045296,0048870,0051015,0051017,0051491,0070062,0070161,0071803,0090091 Kd=85nM remove_due_to_license_issue Kd=90nM, IC50=240nM Q16658 30773430 507 VQIQFGLINCGNKYLTAEAFGFKVNASASSLKKKQIWTLEQPPDEAGSAAVCLRSHLGRYLAADKDGNVTCEREVPGPDCRFLIVAHDDGRWSLQSEAHRRYFGGTEDRLSCFAQTVSPAEKWSVHIAMHPQVNIYSVTRKRYAHLSARPADEIAVDRDVPWGVDSLITLAFQDQRYSVQTADHRFLRHDGRLVARPEPATGYTLEFRSGKVAFRDCEGRYLAPSGPSGTLKAGKATKVGKDELFALEQSCAQVVLQAANERNVSTRQGMDLSANQDEETDQETFQLEIDRDTKKCAFRTHTGKYWTLTATGGVQSTASSKNASCYFDIEWRDRRITLRASNGKFVTSKKNGQLAASVETAGDSELFLMKLINRPIIVFRGEHGFIGCRKVTGTLDANRSSYDVFQLEFNDGAYNIKDSTGKYWTVGSDSAVTSSGDTPVDFFFEFCDYNKVAIKVGGRYLKGDHAGVLKASAETVDPASLWEY 6i1r A 2.8 BS01 C5P A 1 P38 E42 S79 Y82 L83 N86 N206 W209 P34 E38 S75 Y78 L79 N82 N202 W205 ? 0000139,0015165,0016020,0090481 remove_due_to_license_issue B4FZ94 31133698 401 MQWYLVAALLTILTSSQGILTTLSQSNYDYATIPFLAELFKLSVSGFFLWKECRTSPSVRMTKEWRSVRLYVVPSVIYLIHNNVQFATLTYVDPSTYQIMGNLKIVTTGILFRLVLKRKLSNIQWMAIVLLAVGTTTSQVKGCGDSPCDSLFSAPLEGYLLGILSACLSALAGVYTEYLMKKNNDSLYWQNVQLYTFGVIFNMGWLIYGDFKAGFELGPWWQRLFNGYSITTWMVVFNLGSTGLLVSWLMKYSDNIVKVYSTSMAMLLTMVLSIYLFSVKATIQLFLGIIICIISLQMYFMPVHMLIEL 6i3s A 1.77 BS01 H28 A 1 L54 L57 G58 I61 M62 Y67 F86 V93 H96 I99 Y100 L37 L40 G41 I44 M45 Y50 F69 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 remove_due_to_license_issue Q00987 30458062 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 6i3u A 2.09 BS01 H2E A 1 L634 Y670 Q683 W684 I685 S688 P690 I761 L319 Y355 Q368 W369 I370 S373 P375 I446 2.7.1.137 0016301,0016303,0046854 ic50=0.0006uM remove_due_to_license_issue Q8NEB9 30840447 901 KLARSLRSGPSDHDLKPNAATRDQLNIIVSYPPTKQLTYEEQDLVWKFRYYLTNQEKALTKFLKCVNWDLPQEAKQALELLGKWKPMDVEDSLELLSSHYTNPTVRRYAVARLRQADDEDLLMYLLQLVQALKYENFDDIKNGLIDSSQIITSPLPEQDLCTFLISRACKNSTLANYLYWYVIVECEDQDTQQRDPKTHEMYLNVMRRFSQALLKGDKSVRVMRSLLAAQQTFVDRLVHLMKAVQRESGNRKKKNERLQALLGDNEKMNLSDVELIPLPLEPQVKIRGIIPETATLAKSANMPAQLFFKTEDGGKYPVLFKHGDDLRQDQLILQIISLMDKLLRKENLDLKLTPYKVLATSTKHGFLQWIQGSVPVAEVLDTEGSIQNFFRKYAPSENGPNGISAEVMDTYVKSCAGYCVITYILGVGDRHLDNLLLTKTGKLFHIDFGYILGRDPKPLPPPMKLNKEMVEGMGGTQSEQYQEFRKQCYTAFLHLRRYSNLILNLFSLMVDANIPDIALEPDKTVKKVQDKFRLDLSDEEAVHYMQSLIDESVHALF 6i5g A 2.0 BS01 PTG A 1 F387 S415 L417 M419 D496 F497 V498 H524 W525 F158 S186 L188 M190 D267 F268 V269 H295 W296 F267 D335 W336 D496 H524 F38 D106 W107 D267 H295 3.1.3.76,3.3.2.10 0003824 Ki=8.56uM remove_due_to_license_issue P34913 31123712 607 TSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD 6i5i A 1.6 BS01 H3E A 1 L167 G168 F172 V175 A189 K191 F241 L244 E292 L295 V324 L22 G23 F27 V30 A44 K46 F96 L99 E147 L150 V179 D288 K290 N293 D325 T342 D143 K145 N148 D180 T197 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P49759 30569600 501 SMHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKKS 6i5y A 1.9 BS01 YSA A 1 Y37 G39 D41 G50 H51 P54 D81 Y175 Q179 D182 G197 G198 D200 Q201 L227 I228 Y33 G35 D37 G46 H47 P50 D77 Y171 Q175 D178 G193 G194 D196 Q197 L223 I224 T43 H48 H51 K85 R89 Q179 D200 K235 K238 T39 H44 H47 K81 R85 Q175 D196 K231 K234 6.1.1.1 0000166,0003723,0004812,0004831,0005524,0005737,0005829,0006412,0006418,0006437,0016020,0042803,0043039 remove_due_to_license_issue Ki=2.9nM P0AGJ9 30995568 501 NLIKQLQERGLVAQVTDEEALAERLAQGPIALYCGFDPTADSLHLGHLVPLLCLKRFQQAGHKPVALVGGATGLIGDPSFKAAERKLNTEETVQEWVDKIRKQVAPFLDFDCGENSAIAANNYDWFGNMNVLTFLRDIGKHFSVNQMINKEAVKQRLNREDQGISFTEFSYNLLQGYDFACLNKQYGVVLQIGGSDQWGNITSGIDLTRRLHQNQVFGLTVPLITKADGTKFGKAVWLDPKKTSPYKFYQFWINTADADVYRFLKFFTFMSIEEINALEEEDKNRAQYVLAEQVTRLVHGEEGLQAAKRITECLFSGSLSALSEADFEQLAQDGVPMVEMEKGADLMQALVDSELQPSRGQARKTIASNAITINGEKQSDPEYFFKEEERLFGRFTLLRRGKKNYCLICWK 6i61 A 1.65 BS01 H3W A 1 L268 E275 M306 L309 Y326 L345 N346 I349 F435 F450 L35 E42 M73 L76 Y93 L112 N113 I116 F202 F217 ? Kd=569nM remove_due_to_license_issue P62508 31127318 501 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAK 6i64 A 1.91 BS01 H48 A 1 E275 M306 L309 Y326 N346 I349 F435 E42 M73 L76 Y93 N113 I116 F202 ? Kd=48.7nM remove_due_to_license_issue P62508 31127318 501 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAK 6i65 A 1.5 BS01 H3Z A 1 E275 L309 V313 Y326 F435 E42 L76 V80 Y93 F202 ? Kd=390.4nM remove_due_to_license_issue P62508 31127318 501 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAK 6i66 A 1.6 BS01 H4Q A 1 A272 E275 L309 V313 Y326 F435 F450 A39 E42 L76 V80 Y93 F202 F217 ? Kd=182.5nM remove_due_to_license_issue P62508 31127318 501 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEA 6i67 A 1.75 BS01 H42 A 1 E275 L309 V313 Y326 F435 E42 L76 V80 Y93 F202 ? Kd=201.4nM remove_due_to_license_issue P62508 31127318 501 YNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAKV 6i74 A 0.959 BS01 H5Z A 1 R144 I145 A146 H158 N160 R162 N174 W181 E184 S237 G238 R32 I33 A34 H46 N48 R50 N62 W69 E72 S125 G126 ? 0030246 Kd=3.4uM remove_due_to_license_issue P17931 30632578 901 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6i75 A 1.171 BS01 H5T A 1 R144 A146 H158 N160 R162 N174 W181 E184 S237 G238 R32 A34 H46 N48 R50 N62 W69 E72 S125 G126 ? 0030246 Kd=23uM remove_due_to_license_issue P17931 30632578 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6i76 A 1.2 BS01 H5N A 1 R144 A146 H158 N160 R162 N174 W181 E184 G238 R32 A34 H46 N48 R50 N62 W69 E72 G126 ? 0030246 Kd=8.5uM remove_due_to_license_issue P17931 30632578 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6i77 A 1.219 BS01 H5Q A 1 R144 A146 H158 N160 R162 N174 W181 E184 G238 R32 A34 H46 N48 R50 N62 W69 E72 G126 ? 0030246 Kd=11uM remove_due_to_license_issue P17931 30632578 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6i78 A 1.15 BS01 H5H A 1 R144 H158 N160 R162 N174 W181 E184 R32 H46 N48 R50 N62 W69 E72 ? 0030246 Kd=18uM remove_due_to_license_issue P17931 30632578 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6i8b B 1.76 BS01 H7T B 1 W62 W72 Y91 F94 Y98 H139 F141 W151 Y170 Y179 D184 W13 W23 Y42 F45 Y49 H84 F86 W95 Y114 Y123 D128 ? 0007276 remove_due_to_license_issue Kd=111nM, EC50=270nM, IC50=33nM Q9Y657 31550156 301 RRNIVGCRIQHGWKEGNGPVTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELNKDERVSALEVLPDRVATHLADTMIGKAVEHMFETDGSKDEWRGMVLARAPVMNTWFYITYEKDPVLYMYQLLDDYKEGDLRIMPDSLVGKQVEYAGSKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLVKTSAENLYFQ 6i8b B 1.76 BS02 H7T E 1 R51 A119 R2 A70 ? 0007276 remove_due_to_license_issue Kd=111nM, EC50=270nM, IC50=33nM Q9Y657 31550156 302 RRNIVGCRIQHGWKEGNGPVTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELNKDERVSALEVLPDRVATHLADTMIGKAVEHMFETDGSKDEWRGMVLARAPVMNTWFYITYEKDPVLYMYQLLDDYKEGDLRIMPDSLVGKQVEYAGSKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLVKTSAENLYFQ 6i8l B 1.58 BS01 H7Q B 1 D95 H139 F141 W151 Y170 Y179 D184 D44 H81 F83 W93 Y112 Y121 D126 ? 0007276 remove_due_to_license_issue IC50=390nM Q9Y657 31550156 304 NIVGCRIQHGWKEGNGPVTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELNKDERVSALEVLPDRVATLADTMIGKAVEHMFETEDGSKDEWRGMVLARAPVMNTWFYITYEKDPVLYMYQLLDDYKEGDLRIMPDSSLVGKQVEYAKSKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLVKTSAENLYFQ 6i8m A 2.1 BS01 H7W A 1 H862 G863 G888 Y889 Y896 F897 S904 Y907 H201 G202 G227 Y228 Y235 F236 S243 Y246 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue P26446 30996792 1101 KSKLAKPIQDLIKMIFDVESMKKAMVEFEIDLQKMPLGKLSKRQIQSAYSILNEVQQAVSDGGSESQILDLSNRFYTLIPHDFGMKKPPLLSNLEYIQAKVQMLDNLLDIEVAYSLLRGGNEDGDKDPIDINYEKLRTDIKVVDKDSEEAKIIKQYVKNTHAATHNAYDLKVVEIFRIEREGESQRYKPFKQLHNRQLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQADPIGLILLGEVALGNMYELKNASHITKLPKGKHSVKGLGKTAPDPTATTTLDGVEVPLGNGISTGINDTCLLYNEYIVYDVAQVNLKYLLKLKFNY 6i8t A 2.1 BS01 H7Z A 1 Q759 Q763 H862 G863 G888 Y896 F897 K903 S904 Y907 Q98 Q102 H201 G202 G227 Y235 F236 K242 S243 Y246 S904 Y907 E988 S243 Y246 E327 2.4.2.-,2.4.2.30 0003950 remove_due_to_license_issue P26446 30996792 1101 KSKLAKPIQDLIKMIFDVESMKKAMVEFEIDLQKMPLGKLSKRQIQSAYSILNEVQQAVSDGGSESQILDLSNRFYTLIPHDFGMKKPPLLSNLEYIQAKVQMLDNLLDIEVAYSLLRGGNEDGDKDPIDINYEKLRTDIKVVDKDSEEAKIIKQYVKNTHAATHNAYDLKVVEIFRIEREGESQRYKPFKQLHNRQLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQADPIGLILLGEVALGNMYELKNASHITKLPKGKHSVKGLGKTAPDPTATTTLDGVEVPLGNGISTGINDTCLLYNEYIVYDVAQVNLKYLLKLKFNY 6i8z A 1.99 BS01 H82 A 1 I428 A452 M499 E500 L501 C502 T503 G505 E506 L553 G563 D564 L567 I15 A39 M86 E87 L88 C89 T90 G92 E93 L140 G150 D151 L154 D546 R550 N551 D564 D133 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=17nM remove_due_to_license_issue Q05397 30739444 701 DYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPALAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKYSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSSNDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKAQQE 6i96 A 1.85 BS01 0UE A 1 V210 Y216 Y218 T245 F246 H374 G375 Q441 Y443 S460 W503 F803 Y805 V67 Y73 Y75 T102 F103 H231 G232 Q298 Y300 S317 W360 F660 Y662 ? 0009279,0015343,0015891,0038023 Kd=100nM remove_due_to_license_issue Q9I116 31385808 901 VFALGNNLGSTDGYLATHSQIATKTSKPLLETSQTVSVITREQIDDTASKTVQQAMRYTPGIFTGQVGASNRYDYVVMRGFADNSVDNIYLDGLKAMGDSGTFSSMQVDPYFLERIDVLKGPSSVLYGRSLPGGLVALTSKKPLYEDYRQITGSIGNMGQKEMGFDFSGPLDEEKRIAYRLIGLGKGSDTQFDHVKEERYAIAPTLAIDFSDDTTLTLQGYLQHDPNGGYHGGVPADGTLSHHNGRHISREFFDGEPSKDDFDRTQRMFGYQLEHRIDDVWSARQNFRYLDSDVDLSQVYAYGWSASEPNKLNRYFSGAREHLQAYIVDNMLQAEFATGAARHTLLTGLDYQRRRTVVDWRSGSASALDAFNPVYGDDAISYFPDDNHTRRLEQTGVYLQDLIDIDQWRFSLGLRQDWVSVTDKNRSTGSKADDDWEKFTGRIGALYLFDNGLAPYVSYSESFNPNAYSDASGTPLAPTEGKQWELGLKFQAPGSNSFYTASLFHITQENVASKEPQDNFYTSVGEVRSQGLELEAHTQLSDNLKLLGSYTYTDITYTKSLDGNQGHTPNQAPKHMASLWADYAFDAGPLSGLSIGGGARYVGETWADKENTLRVPDYTLVDARIGYDLGKLGLKGLDVSLNANNLLDKDYVASCYSLDFCYFGEKRNVTATVNYQF 6i97 A 3.35 BS01 0UE A 1 Y216 Y218 T245 F246 H374 G375 Y443 K657 P659 Y799 Y159 Y161 T188 F189 H317 G318 Y386 K600 P602 Y742 ? 0006826,0007166,0009279,0015343,0015344,0015891,0019867,0033214,0038023,0044718 remove_due_to_license_issue Q9I116 31385808 901 EQARPYAIPAGQLGDVLNRFAREAGITLSATPAQTGGYSSQGLRGSFTVQQGLARLLADTPLEAEDQGDGSFVLREAPAKDGDVLNMQAVEVFALGNDGYLATHSQIATKTSKPLLETSQTVSVITREQIDDTASKTVQQAMRYTPGIFTGQVGASNRYDYVVMRGFADNSVDNIYLDGLKAMGDSGTFSSMQVDPYFLERIDVLKGPSSVLYGRSLPGGLVALTSKKPLYEDYRQITGSIGNMGQKEMGFDFSGPLDEEKRIAYRLIGLGKGSDTQFDHVKEERYAIAPTLAIDFSDDTTLTLQGYLQHDPNGGYHGGVPADGTLSHHNGRHISREFFDGEPSKDDFDRTQRMFGYQLEHRIDDVWSARQNFRYLDSDVDLSQVYAYGWSASEPNKLNRYFSGAREHLQAYIVDNMLQAEFATGAARHTLLTGLDYQRRRTVVDWRSGSASALDAFNPVYGDDAISYFPDDNHTRRLEQTGVYLQDLIDIDQWRFSLGLRQDWVSVTDKNRSTGSKADDDWEKFTGRIGALYLFDNGLAPYVSYSESFNPNAYSDASGTPLAPTEGKQWELGLKFQAPGSNSFYTASLFHITQENVASKEPQDNFYTSVGEVRSQGLELEAHTQLSDNLKLLGSYTYTDITYTKSLDGNQGHTPNQAPKHMASLWADYAFDAGPLSGLSIGGGARYVGETWADKENTLRVPDYTLVDARIGYDLGKLGLKGLDVSLNANNLLDKDYVASCYSLDFCYFGEKRNVTATVNYQF 6i9a A 1.2 BS03 H8E A 1 A443 H444 G445 N475 C477 I478 N510 S511 Y512 W513 D516 H575 A215 H216 G217 N247 C249 I250 N282 S283 Y284 W285 D288 H347 D388 H444 G445 C477 D160 H216 G217 C249 3.4.22.47 0006508,0008233,0008234 remove_due_to_license_issue Q51817 30894633 707 DVYTDHGDLYNTPVRMLVVAGAKFKEALKPWLTWKAQKGFYLDVHYTDEAEVGTTNASIKAFIHKKYNDGLAASAAPVFLALVGDTDVISGEKGKKTKKVTDLYYSAVDGDYFPEMYTFRMSASSPEELTNIIDKVLMYEKATMPDKSYLEKVLLIAGADYSWNSQVGQPTIKYGMQYYYNQEHGYTDVYNYLKAPYTGCYSHLNTGVSFANYTAHGSETAWADPLLTTSQLKALTNKDKYFLAIGNCCITAQFDYVQPCFGEVITRVKEKGAYAYIGSSPNSYWGEDYYWSVGANAVFGVQPTFEGTSMGSYDATFLEDSYNTVNSIMWAGNLAATHAGNIGNITHIGAHYYWEAYHVLGDGSVMPYRAMPKTNTYTLPASLPQNQASYSIQASAGSYVAISKDGVLYGTGVANASGVATVSMTKQITENGNYDVVITRSNYLPVIKQIQVG 6ia7 A 2.3 BS01 GTP A 1 S14 K15 S16 G17 K18 S19 T20 T39 H143 S145 L174 D175 Y176 S10 K11 S12 G13 K14 S15 T16 T27 H96 S98 L127 D128 Y129 ? 0003924,0005525,0005737,0005856,0005929,0006886,0012505,0030992,0031514,0036064,0060271 remove_due_to_license_issue Q381A3 30940671 301 LVKILVLGPSKSGKSTVTNFLAGTRETNPLRVLEVEIALDAVVQLWDVGGWPAIASNADGIIYVFNPEVKGSEKELLLWYKNFARVTDGHSLIFSHHSSLPEFAVGDNAIPPMPKQLQGIRALETSLDYQSDNFKEAFDALVEQIIASRLAAE 6iae A 2.49 BS01 GTP A 1 S14 K15 S16 G17 K18 S19 T20 T39 H143 H144 S145 L174 D175 S12 K13 S14 G15 K16 S17 T18 T30 H101 H102 S103 L132 D133 ? 0003924,0005525,0005737,0005856,0005929,0006886,0012505,0030992,0031514,0036064,0060271 remove_due_to_license_issue Q381A3 30940671 301 DDLVKILVLGPSKSGKSTVTNFLAGTRDETNPLRVLEVEIALKAVVQLWDVGGSWPAIASNADGIIYVFNPEVKGSEKELLLWYKNFAMRVTDGHSLIFSHHSSLPEFAVGDNAIPPMPKQLQGIRALETSLDYQSDNFKEAFDALVEQIIASRL 6iar A 1.84 BS01 H8W A 1 L346 T347 E353 L387 M421 V533 V534 L37 T38 E44 L78 M112 V223 V224 ? remove_due_to_license_issue P03372 30640465 601 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPSYDLLLEMLDAH 6ib0 A 2.6 BS01 H8Z A 1 M142 M215 C218 K221 L266 M26 M99 C102 K105 L150 D259 K261 N264 D277 C296 D143 K145 N148 D161 C170 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue O14733 30768270 501 KQTGYLTIGGQRYQAEINDLENLGEMGSGTCGQVWKMRFRKTGHVIAVKQMRRSGNKEENKRILMDLDVVLKSHDCPYIVQCFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGKMTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCDFGISGRAGCAAYMAPERIDPPDPTKPDYDIRADVWSLGISLVELATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQSFVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFKDVMAK 6ibk A 1.99 BS01 YTW A 1 W47 D92 D93 C142 K168 D170 E203 R227 D231 W16 D61 D62 C111 K137 D139 E172 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue P06280 525 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTM 6ibk B 1.99 BS01 YTW B 1 W47 D92 D93 C142 K168 D170 E203 R227 D231 W16 D61 D62 C111 K137 D139 E172 R196 D200 D170 D231 D139 D200 3.2.1.22 0003824,0004553,0004557,0005102,0005515,0005576,0005737,0005764,0005794,0005975,0006629,0009311,0016020,0016139,0016787,0016798,0016936,0019915,0030168,0030431,0031133,0035578,0042803,0043202,0045019,0046477,0046479,0051001,0070062,0070527,0090325 remove_due_to_license_issue P06280 520 LDNGLARTPTMGWLHWERFMCNLDCQEEPDSCISEKLFMEMAELMVSEGWKDAGYEYLCIDDCWMAPQRDSEGRLQADPQRFPHGIRQLANYVHSKGLKLGIYADVGNKTCAGFPGSFGYYDIDAQTFADWGVDLLKFDGCYCDSLENLADGYKHMSLALNRTGRSIVYSCEWPLYMWPFQKPNYTEIRQYCNHWRNFADIDDSWKSIKSILDWTSFNQERIVDVAGPGGWNDPDMLVIGNFGLSWNQQVTQMALWAIMAAPLFMSNDLRHISPQAKALLQDKDVIAINQDPLGKQGYQLRQGDNFEVWERPLSGLAWAVAMINRQEIGGPRSYTIAVASLGKGVACNPACFITQLLPVKRKLGFYEWTSRLRSHINPTGTVLLQLENTMQM 6ibl A 2.7 BS01 H98 A 1 D121 V122 V125 D200 F201 S211 S215 F306 F307 N310 N329 Y333 D188 V189 V192 D267 F268 S278 S282 F345 F346 N349 N368 Y372 ? 0004930,0004935,0004940,0005515,0005737,0005829,0007186,0007189,0015035,0015036,0016020,0030337,0045454,0045823 remove_due_to_license_issue P07700,P0AA25 32555462 501 KIIHLTDDSFDTDVLKADGAILVDFWAEWSGPSKMIAPILDEIADEYQGKLTVAKLNIDQNPGTAPKYGIRGIPTLLLFKNGEVAATKVGALSKGQLKEFLDANLAEAKVMSLLMALVVLLIVAGNVLVIAAIGSTQRLQTLTNLFITSLACADLVVGLLVVPFGATLVVRGTWLWGSFLCELWTSLDVLCVTASIETLCVIAIDRYLAITSPFRYQSLMTRARAKVIICTVWAISALVSFLPIMMHWWRDEDPQALKCYQDPGCCDFVTNRAYAIASSIISFYIPLLIMIFVYLRVYREAKEQIRKIDRASKRKTSRVMAMKEHKALKTLGIIMGVFTLCWLPFFLVNIVNVFNRDLVPDWLFVAFNWLGYANSAMNPIIYCRSPDFRKAFKRLLA 6ibs A 1.37 BS03 HB8 A 1 L65 W93 H122 D124 H189 C208 H250 L24 W48 H77 D79 H144 C163 H205 H120 H122 D124 H189 C208 K211 N220 H250 H75 H77 D79 H144 C163 K166 N175 H205 3.5.2.6 remove_due_to_license_issue C7C422 30996812 303 GDQRFGDLVFRQLAPNVWQHTSYLDGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6ibv A 1.4 BS01 H9E A 1 L65 W93 H122 D124 H189 L26 W50 H79 D81 H146 H120 H122 D124 H189 C208 K211 N220 H250 H77 H79 D81 H146 C165 K168 N177 H207 3.5.2.6 remove_due_to_license_issue C7C422 30996812 301 ETGDQRFGDLVFRQLAPNVWQHTSYLDGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6ibx A 2.11 BS01 H9Z A 1 R45 Y49 I50 S152 C154 V159 N163 E166 V167 V214 I241 R28 Y32 I33 S135 C137 V142 N146 E149 V150 V197 I224 2.7.1.105,3.1.3.46 0003824,0003873,0005524,0006000,0006003 ic50=2nM remove_due_to_license_issue IC50=2.0nM Q16875 30626557 501 ELTQSRVQKIWVPVNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERSE 6iby A 2.51 BS01 HAT A 1 R45 Y49 I50 S152 C154 N163 E166 V214 V217 G218 I241 R27 Y31 I32 S134 C136 N145 E148 V196 V199 G200 I223 2.7.1.105,3.1.3.46 0003824,0003873,0005524,0006000,0006003 remove_due_to_license_issue IC50=8280nM Q16875 30626557 501 ELTQSRVQKIWVPNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERSE 6ibz A 2.44 BS02 HAW A 1 R45 Y49 I50 S152 C154 V159 N163 V167 V214 V217 I241 V243 R30 Y34 I35 S137 C139 V144 N148 V152 V199 V202 I226 V228 2.7.1.105,3.1.3.46 0003824,0003873,0005524,0006000,0006003 ic50=22nM remove_due_to_license_issue IC50=22nM Q16875 30626557 503 ELTQSRVQKIWVPVDHNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERSE 6ic0 A 2.6 BS01 HAK A 1 R45 G46 Y49 I50 S152 C154 N163 E166 V214 V217 I241 V243 P421 R28 G29 Y32 I33 S135 C137 N146 E149 V197 V200 I224 V226 P404 2.7.1.105,3.1.3.46 0003824,0003873,0005524,0006000,0006003 remove_due_to_license_issue IC50=22nM Q16875 30626557 501 ELTQSRVQKIWVPVNSPTVIVMVGLPARGKTYISKKLTRYLNWIGVPTKVFNVGEYRREAVKQYSSYNFFRPDNEEAMKVRKQCALAALRDVKSYLAKEGGQIAVFDATNTTRERRHMILHFAKENDFKAFFIESVCDDPTVVASNIMEVKISSPDYKDCNSAEAMDDFMKRISCYEASYQPLDPDKCDRDLSLIKVIDVGRRFLVNRVQDHIQSRIVYYLMNIHVQPRTIYLCRHGENEHNLQGRIGGDSGLSSRGKKFASALSKFVEEQNLKDLRVWTSQLKSTIQTAEALRLPYEQWKALNEIDAGVCEELTYEEIRDTYPEEYALREQDKYYYRYPTGESYQDLVQRLEPVIMELERQENVLVICHQAVLRCLLAYFLDKSAEEMPYLKCPLHTVLKLTPVAYGCRVESIYLNVESVCTHRERS 6ic2 A 1.15 BS02 BBJ A 1 Q92 H94 H96 V121 F131 L198 T199 P202 Q90 H92 H94 V119 F128 L195 T196 P199 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=917.4nM remove_due_to_license_issue P00918 31038135 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ic5 A 2.0 BS01 HB5 B 1 D1 P3 D1 P3 3.4.14.1 remove_due_to_license_issue P53634 30978322 403 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKV 6ic5 B 2.0 BS01 HB5 B 1 G232 C234 E275 G276 G277 F278 A349 G27 C29 E70 G71 G72 F73 A144 Q228 C234 Q23 C29 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 30978322 403 HLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6ic5 C 2.0 BS01 HB5 B 1 T379 N380 I429 T8 N9 I58 H381 N403 H10 N32 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 30978322 403 PFNPFELTNHAVLLVGYGTDSASGMDYWIVKNSWGTGWGENGYFRIRRGTDECAIESIAVAATPIPKL 6ic6 A 1.898 BS01 H9B B 1 D1 P3 D1 P3 3.4.14.1 remove_due_to_license_issue P53634 30978322 403 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKV 6ic6 B 1.898 BS01 H9B B 1 G232 C234 E275 G276 G277 F278 G27 C29 E70 G71 G72 F73 Q228 C234 Q23 C29 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 30978322 403 HLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6ic7 A 2.0 BS01 H9H B 1 D1 P3 D1 P3 3.4.14.1 remove_due_to_license_issue P53634 30978322 403 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKV 6ic7 B 2.0 BS01 H9H B 1 G232 C234 E275 G276 G277 F278 G27 C29 E70 G71 G72 F73 Q228 C234 Q23 C29 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 30978322 403 HLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6ic7 C 2.0 BS01 H9H B 1 T379 N380 T8 N9 H381 N403 H10 N32 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 30978322 403 PFNPFELTNHAVLLVGYGTDSASGMDYWIVKNSWGTGWGENGYFRIRRGTDECAIESIAVAATPIPKL 6idb A 2.502 BS01 SIA C 1 Y88 A125 T126 S127 W142 H174 E181 Q217 Y88 A125 T126 S127 W142 H174 E181 Q217 ? 0019031,0019064,0046789 remove_due_to_license_issue R4NN21 31747596 3 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSSCRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARTQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPEI 6ido A 3.748 BS01 dna C 0 R37 L48 R59 E60 R63 R22 L33 R44 E45 R48 ?,2.7.7.6 0003700,0006352,0006355 remove_due_to_license_issue A6TGP0,P13445 31293000 1 ~ 15 KQSIVKWLFELNAKQREVLARRFGLLGYEAATLEDVGREIGLTRERVRQIQVEGLRRLREILQGQGLNIEALTQLTPEEKLLRAIF 6ido A 3.748 BS02 dna D 0 L57 T58 E60 R61 Q64 L42 T43 E45 R46 Q49 ?,2.7.7.6 0003700,0006352,0006355 remove_due_to_license_issue A6TGP0,P13445 31293000 1 ~ 15 KQSIVKWLFELNAKQREVLARRFGLLGYEAATLEDVGREIGLTRERVRQIQVEGLRRLREILQGQGLNIEALTQLTPEEKLLRAIF 6ido B 3.748 BS01 dna E 0 R37 T47 L48 R59 R63 R21 T31 L32 R43 R47 ?,2.7.7.6 0003700,0006352,0006355 remove_due_to_license_issue A6TGP0,P13445 31293000 1 ~ 15 QSIVKWLFELNAKQREVLARRFGLLGYEAATLEDVGREIGLTRERVRQIQVEGLRRLREILQGTQLTPEEKLLRAIF 6ido B 3.748 BS02 dna F 0 L57 T58 E60 R61 Q64 L41 T42 E44 R45 Q48 ?,2.7.7.6 0003700,0006352,0006355 remove_due_to_license_issue A6TGP0,P13445 31293000 1 ~ 15 QSIVKWLFELNAKQREVLARRFGLLGYEAATLEDVGREIGLTRERVRQIQVEGLRRLREILQGTQLTPEEKLLRAIF 6idz A 2.707 BS01 SIA C 1 Y88 A125 T126 S127 W142 H174 E181 Q217 Y88 A125 T126 S127 W142 H174 E181 Q217 ? 0019031,0019064,0046789 remove_due_to_license_issue R4NN21 31747596 3 DKICLGHHAVSNGTKVNTLTERGVEVVNATETVERTNIPRICSKGKRTVDLGQCGLLGTITGPPQCDQFLEFSADLIIERREGSDVCYPGKFVNEEALRQILRESGGIDKEAMGFTYSGIRTNGATSSCRRSGSSFYAEMKWLLSNTDNAAFPQMTKSYKNTRKSPALIVWGIHHSVSTAEQTKLYGSGNKLVTVGSSNYQQSFVPSPGARTQVNGQSGRIDFHWLMLNPNDTVTFSFNGAFIAPDRASFLRGKSMGIQSGVQVDANCEGDCYHSGGTIISNLPFQNIDSRAVGKCPRYVKQRSLLLATGMKNVPEI 6iez A 1.9 BS01 A50 A 1 F436 E446 H469 V472 V525 Y553 V557 V571 E575 Y576 F73 E83 H106 V109 V162 Y184 V188 V202 E206 Y207 ? 0008289 remove_due_to_license_issue Q9Y5P4 600 THRFVQKVEEMVQNHMTYSLQDVGGDANWQLVVEEGEMKVYRREVEENGIVLDPLKATHAVKGVTGHEVCNYFWNVDVRNDWETTIENFHVVETLADNAIIIYQTHKRVWPASQRDVLYLSVIRKIPALTENDPETWIVCNFSVDHDSAPLNNRCVRAKINVAMICQTLVSEISRDNILCKITYVANVNPGGWAPASVLRAVAKREYPKFLKRFTSYVQEKTAGKPILF 6if0 A 1.8 BS01 A59 A 1 F436 E446 T448 H469 N504 V571 E575 Y576 F73 E83 T85 H106 N141 V202 E206 Y207 ? 0008289 remove_due_to_license_issue Q9Y5P4 600 THRFVQKVEEMVQNHMTYSLQDVGGDANWQLVVEEGEMKVYRREVEENGIVLDPLKATHAVKGVTGHEVCNYFWNVDVRNDWETTIENFHVVETLADNAIIIYQTHKRVWPASQRDVLYLSVIRKIPALTENDPETWIVCNFSVDHDSAPLNNRCVRAKINVAMICQTLVSEISRDNILCKITYVANVNPGGWAPASVLRAVAKREYPKFLKRFTSYVQEKTAGKPILF 6ift A 1.9 BS01 SAM A 1 L26 G27 Q28 N29 F30 L31 G56 P57 G58 F76 E77 I78 D102 V103 N127 P129 Y131 L26 G27 Q28 N29 F30 L31 G56 P57 G58 F76 E77 I78 D102 V103 N127 P129 Y131 2.1.1.182 0000154,0000179,0003723,0005737,0005829,0006364,0008168,0016433,0031167,0032259,0052908 remove_due_to_license_issue P37468 30624914 301 MNKDIATPIRTKEILKKYGFSFKKSLGQNFLIDTNILNRIVDHAEVTEKTGVIEIGPGIGALTEQLAKRAKKVVAFEIDQRLLPILKDTLSPYENVTVIHQDVLKADVKSVIEEQFQDCDEIMVVANLPYYVTTPIIMKLLEEHLPLKGIVVMLQKEVAERMAADPSSKEYGSLSIAVQFYTEAKTVMIVPKTVFVPQPNVDSAVIRLILRDGPAVDVENESFFFQLIKASFAQRRKTLLNNLVNNLPEGKAQKSTIEQVLEETNIDGKRRGESLSIEEFAALSNGLYKALF 6iid A 2.986 BS01 dna E 0 R109 S137 R138 G139 A144 G145 K148 F168 N171 S172 N176 M180 R183 L311 R314 R52 S80 R81 G82 A87 G88 K91 F111 N114 S115 N119 M123 R126 L254 R257 C112 A140 N162 N171 E179 C55 A83 N105 N114 E122 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 10 EKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEE 6iid A 2.986 BS02 dna F 0 K113 K115 S172 L311 R320 R324 K56 K58 S115 L254 R263 R267 C112 A140 N162 N171 E179 C55 A83 N105 N114 E122 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 2 ~ 12 EKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEKKLEE 6iid B 2.986 BS01 dna G 0 R109 S137 R138 G139 P143 G145 F168 N171 S172 N176 R183 L311 R314 R52 S80 R81 G82 P86 G88 F111 N114 S115 N119 R126 L254 R257 C112 A140 N162 N171 E179 C55 A83 N105 N114 E122 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 7 EKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGLEKIMENLKNAEIEPDDYFMSRYEKKLEE 6iid B 2.986 BS02 dna H 0 D169 S172 K315 D112 S115 K258 C112 A140 N162 N171 E179 C55 A83 N105 N114 E122 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 5 ~ 12 EKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGLEKIMENLKNAEIEPDDYFMSRYEKKLEE 6iid C 2.986 BS01 dna I 0 R109 S137 R138 G139 A144 G145 F168 N171 S172 N176 M180 R183 R314 R51 S79 R80 G81 A86 G87 F110 N113 S114 N118 M122 R125 R256 C112 A140 N162 N171 E179 C54 A82 N104 N113 E121 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 11 KAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEK 6iid C 2.986 BS02 dna J 0 K113 S172 L311 R320 K55 S114 L253 R262 C112 A140 N162 N171 E179 C54 A82 N104 N113 E121 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 4 ~ 12 KAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKIEGARSVLRLEKIMENLKNAEIEPDDYFMSRYEK 6iid D 2.986 BS01 dna K 0 R109 K110 S137 R138 G139 A144 G145 K148 F168 N171 S172 N176 R183 Y310 L311 R314 R53 K54 S81 R82 G83 A88 G89 K92 F112 N115 S116 N120 R127 Y254 L255 R258 C112 A140 N162 N171 E179 C56 A84 N106 N115 E123 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 1 ~ 5 AEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKVLRLEKIMENLKNAEIEPDDYFMSRYEKK 6iid D 2.986 BS02 dna L 0 S172 L311 K315 S116 L255 K259 C112 A140 N162 N171 E179 C56 A84 N106 N115 E123 3.1.30.- 0003676,0016787,0046872 remove_due_to_license_issue Q9Y2C4 30949702 9 ~ 12 AEKAVLEQFGFPLTGTEARCYTNHALSYDQAKRVPRWVLEHISKSKIMGDADRKHCKFKPDPNIPPTFSAFNEDYVGSGWSRGAMAPAGNNKFSSKAMAETFYLSNIVPQDFDNNSGYWNRIEMYCRELTERFEDVWVVSGPLTLPQTRGDGKKIVSYQVIGEDNVAVPSHLYKVILARRSSVSTEPLALGAFVVPNEAIGFQPQLTEFQVSLQDLEKLSGLVFFPHLDRTSDIRNICSVDTCKLLDFQEFTLYLSTRKVLRLEKIMENLKNAEIEPDDYFMSRYEKK 6iik A 1.97 BS01 IU1 A 1 Q197 Q198 D199 F331 H426 S431 Y436 Y476 Q96 Q97 D98 F211 H276 S281 Y286 Y326 3.4.19.12 0004843,0016579,0043161 ic50=12.25uM remove_due_to_license_issue IC50=4000nM P54578 30254335 501 ELPCGLTNLGNTCYMNATVQCIRSVPELKDALKRYAGALRASGEMASAQYITAALRDLFDSMDKTSSSIPPIILLQFLHMAFPQFAEKGEQGQYLQQDANECWIQMMRVLQQKLEAIEDKSLIDQFFGVEFETTMKCTESEEEEVTKGKENQLQLSCFINQEVKYLFTGLKLRLQEEITKQSPTLQRNALYIKSSKISRLPAYLTIQMVRFFNAKVLKDVKFPLMLDMYELCTPELQEKMVSFRSKFKDLYEPFSFADDIGSNNCGYYDLQAVLTHQGRSSSSGHYVSWVKRKQDEWIKFDDDKVSIVTPEDILRLSGGGDWHIAYVLLYGPRRV 6iil A 2.2 BS01 A8F A 1 Q197 Q198 D199 F331 H426 S431 S432 Y436 Y476 Q96 Q97 D98 F211 H280 S285 S286 Y290 Y330 3.4.19.12 0004843,0016579,0043161 ic50=0.68uM remove_due_to_license_issue P54578 30254335 501 ELPCGLTNLGNTCYMNATVQCIRSVPELKDALKRYAGALRASGEMASAQYITAALRDLFDSMDKTSSSIPPIILLQFLHMAFPQFAEKGEQGQYLQQDANECWIQMMRVLQQKLEAIEDKSLIDQFFGVEFETTMKCTESEEEEVTKGKENQLQLSCFINQEVKYLFTGLKLRLQEEITKQSPTLQRNALYIKSSKISRLPAYLTIQMVRFFNAKVLKDVKFPLMLDMYELCTPELQEKMVSFRSKFKDLEDKKYEPFSFADDIGSNNCGYYDLQAVLTHQGRSSSSGHYVSWVKRKQDEWIKFDDDKVSIVTPEDILRLSGGGDWHIAYVLLYGPRRVEI 6iin A 2.53 BS01 A8O A 1 Q197 Q198 D199 F331 H426 S431 S432 Y436 Y476 Q97 Q98 D99 F211 H277 S282 S283 Y287 Y327 3.4.19.12 0004843,0016579,0043161 remove_due_to_license_issue P54578 30254335 501 MELPCGLTNLGNTCYMNATVQCIRSVPELKDALKRYAGALRASGEMASAQYITAALRDLFDSMDKTSSSIPPIILLQFLHMAFPQFAEKGEQGQYLQQDANECWIQMMRVLQQKLEAIEKSLIDQFFGVEFETTMKCTESEEEEVTKGKENQLQLSCFINQEVKYLFTGLKLRLQEEITKQSPTLQRNALYIKSSKISRLPAYLTIQMVRFFYNAKVLKDVKFPLMLDMYELCTPELQEKMVSFRSKFKDLYEPFSFADDIGSNNCGYYDLQAVLTHQGRSSSSGHYVSWVKRKQDEWIKFDDDKVSIVTPEDILRLSGGGDWHIAYVLLYGPRRV 6iiq A 1.85 BS01 dna E 0 K20 G21 P23 N76 K20 G21 P23 N76 ? remove_due_to_license_issue Q9Y3E1 11 ~ 15 MARPRPREYKAGDLVFAKMKGYPHWPARIDELPEGAVKPPANKYPIFFFGTHETAFLGPKDLFPYKEYKDKFGKSNKRKGFNEGLWEIENNPGVKFTGY 6iiq B 1.85 BS01 dna F 0 K18 G21 P23 K17 G20 P22 ? remove_due_to_license_issue Q9Y3E1 1 ~ 10 ARPRPREYKAGDLVFAKMKGYPHWPARIDELPEGAVKPPANKYPIFFFGTHETAFLGPKDLFPYKEYKDKFGKSNKRKGFNEGLWEIENNPGVKFTGY 6iiq B 1.85 BS02 dna G 0 K77 R78 K79 K76 R77 K78 ? remove_due_to_license_issue Q9Y3E1 1 ~ 10 ARPRPREYKAGDLVFAKMKGYPHWPARIDELPEGAVKPPANKYPIFFFGTHETAFLGPKDLFPYKEYKDKFGKSNKRKGFNEGLWEIENNPGVKFTGY 6iir A 2.2 BS01 dna C 0 K77 R78 K79 K76 R77 K78 ? remove_due_to_license_issue Q9Y3E1 1 ~ 10 ARPRPREYKAGDLVFAKMKGYPHWPARIDELPEGAVKPPANKYPIFFFGTHETAFLGPKDLFPYKEYKDKFGKSNKRKGFNEGLWEIENNPGVKFTGY 6iir A 2.2 BS02 dna D 0 K20 G21 P23 K19 G20 P22 ? remove_due_to_license_issue Q9Y3E1 1 ~ 10 ARPRPREYKAGDLVFAKMKGYPHWPARIDELPEGAVKPPANKYPIFFFGTHETAFLGPKDLFPYKEYKDKFGKSNKRKGFNEGLWEIENNPGVKFTGY 6iir B 2.2 BS01 dna C 0 R78 K79 R78 K79 ? remove_due_to_license_issue Q9Y3E1 1 ~ 10 MARPRPREYKAGDLVFAKMKGYPHWPARIDELPEGAVKPPANKYPIFFFGTHETAFLGPKDLFPYKEYKDKFGKSNKRKGFNEGLWEIENNPGVKFTGY 6iiu A 2.5 BS01 A8X A 1 A31 G77 T81 V85 M112 S181 W258 L291 L294 R295 T298 Q301 A128 G168 T172 V176 M203 S272 W395 L428 L431 R432 T435 Q438 ? 0004930,0004960,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0043448,0046872 Ki=11nM remove_due_to_license_issue P00268,P0ABE7,P21731 30510189 9001 ADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGATRSSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPLLLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPGSWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGMKKYTCTVCGYIYNPEDGDPDNGVNPGTDFKDIPDDWVCPLCGVGKDQFEEVEERDSEVEMMAQALGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWNQILDPWVYILFRRAVLRRLQPRL 6iiv A 3.0 BS01 A90 A 1 T81 V85 H89 M112 G116 S181 W182 F184 W258 L294 R295 T298 Q301 T173 V177 H181 M204 G208 S273 W274 F276 W396 L432 R433 T436 Q439 ? 0004930,0004960,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0043448,0046872 remove_due_to_license_issue P00268,P0ABE7,P21731 30510189 9001 PADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARRSSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPLLLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPGSWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGMKKYTCTVCGYIYNPEDGDPDNGVNPGTDFKDIPDDWVCPLCGVGKDQFEEVEERDSEVEMMAQALGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWNQILDPWVYILFRRAVLRRLQPRL 6ijh A 2.6 BS02 AEO A 1 L675 I692 Y693 F696 M713 G725 Q726 F729 L229 I246 Y247 F250 M267 G279 Q280 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=68nM Q9Y233 30888810 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRG 6iji B 2.7 BS02 AEL B 1 L675 I692 Y693 M713 G725 F729 L218 I235 Y236 M256 G268 F272 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=0.440000nM Q9Y233 30888810 803 GLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 6ijl A 2.351 BS01 A8U A 1 F183 T184 C186 M190 I214 F216 Y239 Y257 D332 V368 F181 T182 C184 M188 I212 F214 Y237 Y255 D330 V366 2.1.1.354 0000978,0000993,0001162,0005515,0005634,0005654,0005737,0005829,0006325,0006334,0008168,0014904,0032259,0042054,0045184,0045944,0046872,0071549,0140939,0140954,0140999 remove_due_to_license_issue Q9H7B4 31223458 501 PLKVEKFATANRGNGLRAVTPLRPGELLFRSDPLAYTVCKGSRGVVCDRCLLGKEKLMRCSQCRVAKYCSAKCQKKAWPDHKRECKCLKSCKPRYPPDSVRLLGRVVFKLMDGAPSESEKLYSFYDLESNINKLTEDRKEGLRQLVMTFQHFMREEIQDASQLPPAFDLFEAFAKVICNSFTICNAEMQEVGVGLYPSISLLNHSCDPNCSIVFNGPHLLLRAVRDIEVGEELTICYLDMLMTSEERRKQLRDQYCFECDCFRCQTQDKDADMLTGDEQVWKEVQESLKKIEELKAHWKWEQVLAMCQAIISSNSERLPDINIYQLKVLDCAMDACINLGLLEEALFYGTRTMEPYRIFFPGSHPVRGVQVMKVGKLQLHQGMFPQAMKNLRLAFDIMRVTHGREHSLIEDLILLLEECDANI 6ilq A 2.408 BS02 AE0 A 1 C285 R288 S289 A292 I326 M329 I341 E343 M364 C58 R61 S62 A65 I99 M102 I114 E116 M137 ? 0003677,0004879,0005634,0006355 ic50=0.44uM remove_due_to_license_issue IC50=440nM, EC50=1730nM P37231 30594432 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTSPFVIYDMNSLMMVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETSLHPLLQEIYKDL 6ilz A 3.261 BS01 AFU A 1 I260 Y334 T395 D396 F552 D553 I7 Y78 T139 D140 F285 D286 D378 K380 N383 D396 T416 D122 K124 N127 D140 T160 2.7.11.13 0004672,0004674,0005524,0006468,0007163 remove_due_to_license_issue IC50=340nM P41743 30891133 601 FDLLRVIGRGSYAKVLLVRLDRIYAMKVVKKELVNDDEDIDWVQTEKHVFEQASNHPFLVGLHSCFQTESRLFFVIEYVNGGDLMFHMQRQRKLPEEHARFYSAEISLALNYLHERGIIYRDLKLDNVLLDSEGHIKLTDYGMCKEGLRPGDTTSTFCGTPNYIAPEILRGEDYGFSVDWWALGVLMFEMMAGRSPFDIEDYLFQVILEKQIRIPRSLSVKAASVLKSFLNKDPKERLGCHPQTGFADIQGHPFFRNVDWDMMEQKQVVPPFKPNISGEFGLDNFDSQFTNEPVQLTPDDDDIVRKIDQSEFEGFEYINP 6im6 A 1.702 BS04 AH3 A 1 H160 N321 T333 I336 Q369 F372 H74 N235 T247 I250 Q283 F286 3.1.4.53 0004114,0007165,0008081 ic50=20.7uM remove_due_to_license_issue IC50=20700nM Q08499 31099559 505 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6imb A 1.549 BS02 AH9 A 1 H160 I336 Q369 F372 H73 I249 Q282 F285 3.1.4.53 0004114,0007165,0008081 ic50=58.5uM remove_due_to_license_issue IC50=58500nM Q08499 31099559 503 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6imd A 1.499 BS03 AH9 A 1 H160 I336 Q369 F372 H74 I250 Q283 F286 3.1.4.53 0004114,0007165,0008081 ic50=58.5uM remove_due_to_license_issue IC50=58500nM Q08499 31099559 505 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6imi A 1.46 BS03 AH6 A 1 N321 T333 I336 Q369 F372 N235 T247 I250 Q283 F286 3.1.4.53 0004114,0007165,0008081 ic50=26.1uM remove_due_to_license_issue IC50=26100nM Q08499 31099559 504 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6imo A 1.55 BS03 AJL A 1 Y159 I336 M357 Q369 F372 Y72 I249 M270 Q282 F285 3.1.4.53 0004114,0007165,0008081 ic50=0.65uM remove_due_to_license_issue IC50=650nM Q08499 31099559 504 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6imr A 1.503 BS02 AJX A 1 Y159 H160 M273 H276 I336 F340 Q369 F372 I376 Y73 H74 M187 H190 I250 F254 Q283 F286 I290 3.1.4.53 0004114,0007165,0008081 ic50=4.3uM remove_due_to_license_issue IC50=4300nM Q08499 31099559 503 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6imt A 1.483 BS02 AK0 A 1 Y159 I336 F340 M357 Q369 F372 Y72 I249 F253 M270 Q282 F285 3.1.4.53 0004114,0007165,0008081 ic50=0.25uM remove_due_to_license_issue IC50=250nM Q08499 31099559 508 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6ind A 1.872 BS01 AKO A 1 H160 M273 I336 F340 M357 Q369 F372 H74 M187 I250 F254 M271 Q283 F286 3.1.4.53 0004114,0007165,0008081 ic50=0.24uM remove_due_to_license_issue IC50=240nM Q08499 31099559 501 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIP 6ink A 1.7 BS02 AKU A 1 Y159 H160 I336 M357 Q369 F372 Y72 H73 I249 M270 Q282 F285 3.1.4.53 0004114,0007165,0008081 ic50=0.27uM remove_due_to_license_issue IC50=510nM Q08499 31099559 503 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTI 6inm A 1.999 BS02 AKU A 1 H160 M273 I336 M357 Q369 F372 H73 M186 I249 M270 Q282 F285 3.1.4.53 0004114,0007165,0008081 ic50=0.51uM remove_due_to_license_issue IC50=510nM Q08499 31099559 503 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTI 6inz A 2.289 BS01 GCD B 1 W284 A286 S287 L389 Q405 Y409 E410 W258 A260 S261 L363 Q379 Y383 E384 ? 0030313,0046872 remove_due_to_license_issue D1AWE0 31204616 2 PKETTIFAMHLGKALDPNLPVFVKAEKDTNIKLVNVASQNQTDQIQAYNLMLTEGKLPDIVSYELSADLENLGIEGGLIPLEDLINQHAPNLKKFFEENPRYKKDAVAVDGHIYMIPNYYDYFNIKVSQGYFIRQDWLEKLGLKEPRTVDELYTTLKAFREKDPNGNGKKDEVPFFVRANNVRKVLTSLVDLFKASPIWYEENGMVKYGPAQKEFKHAIKELSKWYKEGLIDEEIFTRGLESRDYLLSNNLGGATDDWIASTSSYNRNLADKIPGFNLKLVLPYELNGNAKTRHARTTYLGGWGISKDAKDPVSLIKYFDYWYSVEGRRLWNFGIEGSEYTLVDGKPVFTDKVLKNPDGKTPLAVLREVGAQYRLGAFQDAQYELGWASESAKAGYKYYMDNDVVLDELPILKYTKEKSKEFVSIDTAMRAVVEEKAQQWILGSGDIDKEWDAYIKRLENLGLSKAEQIQNEAF 6ior A 2.5 BS01 ASN A 1 Y120 R125 W127 Y143 D145 F170 D172 Y93 R98 W100 Y116 D118 F143 D145 ? Kd=6.3uM remove_due_to_license_issue Q9KQ43 30745373 501 GSVREEIESLVQDSLMEMVKGVKNTIESDLASKKGLAQSTTEILQLDPTNKAFAKSVLESPNLKGSFLAIGLGYESDATVVENDDGWEPNADYDPRKRPWYVDAKRERKLVVTEPYVDISTKKIIISIGTPVYQQSNFVGAMFYDVELTQLAQLVNSVNLFDAGYLFITTKDGVTIAHPNAENNGEKFSQFLPNVDLKEGTQRIELDGKYYLVKFAQVPSESWYIGAVVDESIAFAMVDDL 6ios A 2.35 BS01 PRO A 1 W114 Y120 R125 W127 D145 F170 D172 W85 Y91 R96 W98 D116 F141 D143 ? Kd=23.8uM remove_due_to_license_issue Q9KQ43 30745373 501 VREEIESLVQDSLMEMVKGVKNTIESDLASKKGLAQSTTEILQLDPTNKAFAKSVLESPNLKGSFLAIGLGYESDATVVENDDGWEPNADYDPRKRPWYVDAKRERKLVVTEPYVDISTKKIIISIGTPVYQQSNFVGAMFYDVELTQLAQLVNSVNLFDAGYLFITTKDGVTIAHPNAENNGEKFSQFLPNVDLKEGTQRIELDGKYYLVKFAQVPSESWYIGAVVDESIAFAMVD 6iot A 2.7 BS01 ARG A 1 A96 D111 W114 Y120 R125 W127 Y143 D145 S147 D172 A69 D84 W87 Y93 R98 W100 Y116 D118 S120 D145 ? remove_due_to_license_issue Q9KQ43 30745373 501 GSVREEIESLVQDSLMEMVKGVKNTIESDLASKKGLAQSTTEILQLDPTNKAFAKSVLESPNLKGSFLAIGLGYESDATVVENDDGWEPNADYDPRKRPWYVDAKRERKLVVTEPYVDISTKKIIISIGTPVYQQSNFVGAMFYDVELTQLAQLVNSVNLFDAGYLFITTKDGVTIAHPNAENNGEKFSQFLPNVDLKEGTQRIELDGKYYLVKFAQVPSESWYIGAVVDESIAFAMV 6iou A 2.1 BS01 SER A 1 Y120 R125 W127 Y143 D145 I146 F170 D172 Y88 R93 W95 Y111 D113 I114 F138 D140 ? Kd=18.3uM remove_due_to_license_issue Q9KQ43 30745373 501 EIESLVQDSLMEMVKGVKNTIESDLASKKGLAQSTTEILQLDPTNKAFAKSVLESPNLKGSFLAIGLGYESDATVVENDDGWEPNADYDPRKRPWYVDAKRERKLVVTEPYVDISTKKIIISIGTPVYQQSNFVGAMFYDVELTQLAQLVNSVNLFDAGYLFITTKDGVTIAHPNAENNGEKFSQFLPNVDLKEGTQRIELDGKYYLVKFAQVPSESWYIGAVVDESIAFAMVDDLR 6iph A 1.65 BS03 DTP A 1 G319 G320 R323 H329 D330 D332 D418 W434 G183 G184 R187 H193 D194 D196 D256 W272 D330 D332 D418 D194 D196 D256 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=0.22uM remove_due_to_license_issue Q9NP87 31067051 503 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHSCAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ipi A 1.8 BS03 DCP A 1 G319 G320 R323 H329 D330 D332 G433 W434 G436 K438 G183 G184 R187 H193 D194 D196 G272 W273 G275 K277 D330 D332 D418 D194 D196 D257 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=1.95uM remove_due_to_license_issue Q9NP87 31067051 503 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHSCCAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ipj A 1.98 BS03 TTP A 1 G319 G320 R323 H329 D330 D332 G433 W434 G183 G184 R187 H193 D194 D196 G272 W273 D330 D332 D418 D194 D196 D257 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=1.62uM remove_due_to_license_issue Q9NP87 31067051 503 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHSCCAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ipl A 1.64 BS02 DTP A 1 G320 R323 K325 H329 D330 D332 G433 W434 T435 G436 K438 G184 R187 K189 H193 D194 D196 G270 W271 T272 G273 K275 D330 D332 D418 D194 D196 D255 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=153uM remove_due_to_license_issue Q9NP87 31067051 502 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHSAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6ipm A 1.72 BS01 DCP A 1 G319 G320 R323 K325 H329 D330 D332 G433 W434 T435 G436 K438 G183 G184 R187 K189 H193 D194 D196 G270 W271 T272 G273 K275 D330 D332 D418 D194 D196 D255 2.7.7.7 0003677,0003887,0005634,0006281,0016779,0034061 Kd=206uM remove_due_to_license_issue Q9NP87 31067051 501 WMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHSAFERSFCIFRLPQPGSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA 6iql A 3.5 BS01 L74 A 1 S91 G96 W98 D112 V113 F330 F331 S61 G66 W68 D82 V83 F293 F294 ? 0004930,0004952,0005506,0005886,0007186,0007195,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,P51436 31750832 1201 GAAALVGGVLLIGLVLAGNSLVCVSVASERTLQTPTNYFIVSLAAADLLLAVLVLPLFVYSEVQGGVWLLSPRLCDTLMAMDVMLCTASIWNLCAISVDRFVAVTGQCQLLLIAATWLLSAAVASPVVCGLNDVPGRDPENRDYVVYSSVCSFFLPCILMLLLYWATFRGLRRWEADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKAKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLKITGRERKAMRVLAVVVGAFLVCWTPFFVVHITRALCPACFVSPRLVSAVTWLGYVNSALNPIIYTIFNAEFRSV 6ir8 A 2.3 BS01 dna B 0 R124 K125 Y126 G127 Q128 R15 K16 Y17 G18 Q19 ? 0003700,0006355,0043565 remove_due_to_license_issue B9FNW2 30783673 1 ~ 14 NSVVVKNLDDGQAWRKYGQKEIQNSKHPKAYFRCTHKYDQLCTAQRQVQRCDDDPASYRVTYIGEHTCR 6ir8 A 2.3 BS02 dna C 0 Y126 K129 Q132 Y140 Y17 K20 Q23 Y31 ? 0003700,0006355,0043565 remove_due_to_license_issue B9FNW2 30783673 1 ~ 14 NSVVVKNLDDGQAWRKYGQKEIQNSKHPKAYFRCTHKYDQLCTAQRQVQRCDDDPASYRVTYIGEHTCR 6irt B 3.5 BS01 AUU B 1 G65 G67 S144 F252 G255 G15 G17 S94 F202 G205 ? 0002720,0003333,0005515,0005764,0005765,0005829,0005886,0006865,0009925,0010507,0010629,0014850,0015171,0015173,0015175,0015179,0015190,0015196,0015297,0015349,0015804,0015807,0015818,0015820,0015821,0015823,0015824,0015827,0015828,0015829,0016020,0016323,0016324,0022857,0031528,0032328,0032729,0032740,0032753,0042149,0042605,0042908,0043231,0055085,0055093,0060252,0070062,0070327,0071222,0071230,0089718,0097421,0098591,0150104,1902024,1902475,1903577,1903801,1904556,1905460,1905534,1990184 remove_due_to_license_issue IC50=112000nM Q01650 30867591 603 TLLNGVAIIVGTIIGSGIFVTPTGVLKEAGSPGLALVVWAACGVFSIVGALCYAELGTTISKSGGDYAYMLEVYGSLPAFLKLWIELLIIRPSSQYIVALVFATYLLKPLFPTCPVPEEAAKLVACLCVLLLTAVNCYSVKAATRVQDAFAAAKLLALALIILLGFVQIGKGDVSNLDPNFSFEGTKLDVGNIVLALYSGLFAYGGWNYLNFVTEEMINPYRNLPLAIIISLPIVTLVYVLTNLAYFTTLSTEQMLSSEAVAVDFGNYHLGVMSWIIPVFVGLSCFGSVNGSLFTSSRLFFVGSREGHLPSILSMIHPQLLTPVPSLVFTCVMTLLYAFSKDIFSVINFFSFFNWLCVALAIIGMIWLRHRKPELERPIKVNLALPVFFILACLFLIAVSFWKTPVECGIGFTIILSGLPVYFFGVWWKNKPKWLLQGIFSTTVLCQKLMQVVPQET 6itj A 1.994 BS01 AXU A 1 F489 V492 A512 K514 V561 Y563 A564 L630 F25 V28 A48 K50 V97 Y99 A100 L154 D623 A625 R627 N628 D641 D147 A149 R151 N152 D165 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=10.8nM remove_due_to_license_issue IC50=11nM P11362 31335138 801 LPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLARDIHHIDYYKKTTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 6itp A 1.572 BS01 HCY A 1 T28 G29 S30 T31 G32 W34 T53 N77 S101 T102 T28 G29 S30 T31 G32 W34 T52 N76 S100 T101 Kd=22.4uM remove_due_to_license_issue 31049949 201 QVQLQESGGGSVQAGGSLRLSCVVSGNTGSTGYWAWFRQGPTEREGVAATYTAGSGTSMTYYADSVKGRFTISQDNAKKTLYLQMNSLKPEDTGMYRCASTRFAGRWYRDSEYRAWGQGTQVTVS 6itp B 1.572 BS01 HCY B 1 T28 G29 S30 T31 G32 W34 T53 N77 S101 T102 T28 G29 S30 T31 G32 W34 T52 N76 S100 T101 Kd=22.4uM remove_due_to_license_issue 31049949 201 QVQLQESGGGSVQAGGSLRLSCVVSGNTGSTGYWAWFRQGPTEREGVAATYTAGSGTSMTYYADSVKGRFTISQDNAKKTLYLQMNSLKPEDTGMYRCASTRFAGRWYRDSEYRAWGQGTQVTVS 6itq A 1.526 BS01 HCY A 1 T28 G29 S30 T31 G32 W34 T53 N77 S101 T102 T28 G29 S30 T31 G32 W34 T50 N73 S97 T98 Kd=20.5uM remove_due_to_license_issue 31049949 201 QVQLQESGGGSVQAGGSLRLSCVVSGNTGSTGYWAWFRQGPREGVAATYTAGSTSMTYYADSVKGRFTISQDNAKKTLYLQMNSLKPEDTGMYRCASTRFAGRWYRDSEYRAWGQGTQVTVS 6itq C 1.526 BS01 HCY C 1 T28 G29 S30 T31 G32 W34 T53 N77 S101 T102 T28 G29 S30 T31 G32 W34 T53 N76 S100 T101 Kd=20.5uM remove_due_to_license_issue 31049949 201 QVQLQESGGGSVQAGGSLRLSCVVSGNTGSTGYWAWFRQGPGTEREGVAATYTAGSTSMTYYADSVKGRFTISQDNAKKTLYLQMNSLKPEDTGMYRCASTRFAGRWYRDSEYRAWGQGTQVTVS 6iuo A 2.3 BS01 AWX A 1 C477 Q480 V481 A501 E520 V550 C552 A553 L619 C34 Q37 V38 A56 E75 V105 C107 A108 L161 D612 R616 N617 D630 D154 R158 N159 D172 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>200nM P22455 31335138 801 GLLAGLVSLDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 6iup A 2.0 BS01 AX0 A 1 C477 V481 A501 K503 V550 C552 A553 L619 D630 C26 V30 A50 K52 V97 C99 A100 L157 D168 D612 R616 N617 D630 D150 R154 N155 D168 2.7.10.1 0004672,0004713,0005524,0006468 ic50=23.1nM remove_due_to_license_issue IC50=23nM P22455 31335138 801 LDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDPARPDQASTVAVKMLKASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPRSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 6ixd A 1.0 BS01 B0F B 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 V82 D25 G27 A28 D29 D30 V32 I47 G48 I50 V82 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 remove_due_to_license_issue Q5RZ08 30990716 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6ixd B 1.0 BS01 B0F B 1 D25 G27 A28 D29 D30 I47 G49 I50 D25 G27 A28 D29 D30 I47 G49 I50 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508 Ki=0.16nM remove_due_to_license_issue Q5RZ08 30990716 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6iyw A 1.6 BS01 IM2 A 1 M303 Y308 Y318 S331 H352 C354 M163 Y168 Y178 S191 H212 C214 2.3.2.- 0016740 remove_due_to_license_issue I6Y9J2 30686533 501 LTFQTSSPAHLTMPYVMPGDGEVVGVGEPVAIRFDENIADRGAAEKAIKITTNPPVEGAFYWLNNREVRWRPEHFWKPGTAVDVAVNTYGVDLGEGMFGEDNVQTHFTIGDEVIATADDNTKILTVRVNGEVVKSMPTSMGKDSTPTANGIYIVGSRYKHIIMDSSTYGVPVNSPNGYRTDVDWATQISYSGVFVHSAPWSVGAQGHTNTSHGCLNVSPSNAQWFYDHVKRGDIVEVVNTVGGTLPGIDGLGDWNIPWDQWRAGNA 6izq A 2.449 BS01 XJ2 A 1 F152 Y153 Q158 M162 E257 M259 Y261 E266 M268 H414 W415 F8 Y9 Q14 M18 E113 M115 Y117 E122 M124 H270 W271 2.1.1.319 0016274,0018216 ic50=3.19uM remove_due_to_license_issue IC50=3190nM Q86X55 31117515 501 SAVQYFQFYGYLSQQQNMMQDYVRTGTYQRAILQNHTDFKDKIVLDVGCGSGILSFFAAQAGARKIYAVEASTMAQHAEVLVKSNNLTDRIVVIPGKVEEVSLPEQVDIIISEPMGYMLFNERMLESYLHAKKYLKPSGNMFPTIGDVHLAPFTDEQLYMEQFTKANFWYQPSFHGVDLSALRGAAVDEYFRQPVVDTFDIRILMAKSVKYTVNFLEAKEGDLHRIEIPFKFHMLHSGLVHGLAFWFDVAFIGSIMTVWLSTAPTEPLTHWYQVRCLFQSPLFAKAGDTLSGTCLLIANKRQSYDISIVAQVDQTGSKSSNLLDLKNPFFRY 6j0g A 1.6 BS01 H6P A 1 H351 Y352 K394 R413 R419 R470 L472 H56 Y57 K99 R118 R124 R175 L177 ? Kd=2.3uM remove_due_to_license_issue O00478 30902636 501 GAAYHEWKMALFKPADVILDPDTANAILLVSEDQRSVQRAEEPRDLPDNPERFEWHYCVLGCENFTSGRHYWEVEVGDRKEWHIGVCSKNVERKKGWVKMTPENGYWTMGLTDGNKYRALTEPRTNLKLPEPPRKVGIFLDYETGEISFYNATDGSHIYTFPHASFSEPLYPVFRILTLEPTALTICPIP 6j0k A 2.0 BS01 H6P A 1 H351 Y352 K394 R413 R419 R470 L472 H57 Y58 K100 R119 R125 R176 L178 ? remove_due_to_license_issue O00478 30902636 501 AGAAYHEWKMALFKPADVILDPDTANAILLVSEDQRSVQRAEEPRDLPDNPERFEWHYCVLGCENFTSGRHYWEVEVGDRKEWHIGVCSKNVERKKGWVKMTPENGYWTMGLTDGNKYRALTEPRTNLKLPEPPRKVGIFLDYETGEISFYNATDGSHIYTFPHASFSEPLYPVFRILTLEPTALTICPIP 6j0o A 1.8 BS01 XAF A 1 E446 H469 K470 V472 I523 E575 Y576 E83 H106 K107 V109 I160 E206 Y207 ? 0008289 remove_due_to_license_issue Q9Y5P4 600 THRFVQKVEEMVQNHMTYSLQDVGGDANWQLVVEEGEMKVYRREVEENGIVLDPLKATHAVKGVTGHEVCNYFWNVDVRNDWETTIENFHVVETLADNAIIIYQTHKRVWPASQRDVLYLSVIRKIPALTENDPETWIVCNFSVDHDSAPLNNRCVRAKINVAMICQTLVSEISRDNILCKITYVANVNPGGWAPASVLRAVAKREYPKFLKRFTSYVQEKTAGKPILF 6j10 B 2.3 BS01 B4O B 1 L19 F23 F24 P25 W102 Y118 F122 L19 F23 F24 P25 W102 Y118 F122 ? 0005198 Kd=445nM remove_due_to_license_issue P03147 31097716 801 MDIDPYKEFGATVELLSFLPSDFFPSVRDLLDTAAALYRDALESPEHCSPHHTALRQAILCWGDLMTLATWVGTNLEDPASRDLVVSYVNTNVGLKFRQLLWFHISCLTFGRETVLEYLVSFGVWIRTPPAARPPNAPILS 6j1l A 2.3 BS01 B6L A 1 Q286 L287 C320 L324 R364 M365 R367 A368 F377 L391 L396 H479 Q21 L22 C55 L59 R99 M100 R102 A103 F112 L126 L131 H214 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue IC50=750nM, Kd=380nM P51449 30964293 601 SLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLEKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQ 6j3o A 2.11 BS01 B4L A 1 P747 E756 N803 Y809 P22 E31 N78 Y84 2.3.1.48,2.3.1.57 0004402 Kd=2.4uM remove_due_to_license_issue Kd=2400nM Q92831 30998845 900 DQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLID 6j3p A 1.598 BS01 B8O A 1 W751 P752 V757 E761 N808 Y814 W23 P24 V29 E33 N80 Y86 2.3.1.-,2.3.1.48 0004402 Kd=105nM remove_due_to_license_issue Kd=105nM Q92830 30998845 900 DPDQLYTTLKNLLAQIKSHPSAWPFMEPVKKSEAPDYYEVIRFPIDLKTMTERLRSRYYVTRKLFVADLQRVIANCREYNPPDSEYCRCASALEKFFYFKLKEGGLID 6j5b A 2.7 BS01 dna B 0 M228 W230 H269 S272 M3 W5 H44 S47 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 ARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b A 2.7 BS02 dna U 0 T252 P253 K254 K271 Q275 R278 T27 P28 K29 K46 Q50 R53 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 ARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b C 2.7 BS01 dna E 0 K225 R227 M228 W230 H269 S272 K276 K2 R4 M5 W7 H46 S49 K53 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 GKARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b C 2.7 BS02 dna G 0 T252 P253 K254 K271 Q275 R278 T29 P30 K31 K48 Q52 R55 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 GKARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b D 2.7 BS01 dna B 0 R227 T252 P253 K254 K271 Q275 R278 R2 T27 P28 K29 K46 Q50 R53 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 ARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b D 2.7 BS02 dna U 0 R227 M228 R229 W230 S272 R2 M3 R4 W5 S47 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 ARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b F 2.7 BS01 dna E 0 T252 P253 K254 K271 Q275 R278 T28 P29 K30 K47 Q51 R54 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 KARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b F 2.7 BS02 dna G 0 R227 M228 R229 W230 H269 S272 R3 M4 R5 W6 H45 S48 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 KARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b H 2.7 BS01 dna I 0 M228 W230 H269 S272 M4 W6 H45 S48 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 KARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b H 2.7 BS02 dna K 0 R227 T252 P253 K254 K271 Q275 R278 R3 T28 P29 K30 K47 Q51 R54 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 KARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARY 6j5b J 2.7 BS01 dna I 0 T252 K254 K271 Q275 R278 T27 K29 K46 Q50 R53 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 ARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARYR 6j5b J 2.7 BS02 dna K 0 R227 M228 R229 W230 H269 S272 R2 M3 R4 W5 H44 S47 ? 0003677,0003700 remove_due_to_license_issue Q94CL7 30974511 1 ~ 20 ARMRWTPELHEAFVEAVNSLGGSERATPKGVLKIMKVEGLTIYHVKSHLQKYRTARYR 6j5l A 2.3 BS01 B9C A 1 L516 G517 F521 V524 A542 Y591 M592 G595 R654 L657 L19 G20 F24 V27 A41 Y90 M91 G94 R153 L156 D650 R654 N655 D668 D149 R153 N154 D167 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=1.6nM remove_due_to_license_issue IC50=1.6nM P04629 31235262 801 SGIRVHHIKRRDIVLKWELGEGAFGKVFLAECHNLDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGIYSTDYYRVTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPV 6j63 A 2.624 BS02 NTD A 1 N282 H308 Q379 F381 F392 E394 F419 F424 N226 H248 Q319 F321 F332 E334 F352 F357 1.13.11.27 0003868,0005506,0005737,0006559,0006572,0009072,0016701,0042802,0046872,0051213 remove_due_to_license_issue P93836 30632699 502 SKFVRKNPKSDKFKVKRFHHIEFWCGDATNVARRFSWGLGMRFSAKSDLSTGNMVHASYLLTSGDLRFLFTAPYSPSLTTTASIPSFDHGSCRSFFSSHGLGVRAVAIEVEDAESAFSISVANGAIPSSPPIVLNEAVTIAEVKLYGDVVLRYVSYKEFLPGFERVEDPLDYGIRRLDHAVGNVPELGPALTYVAGFTGFHQFAEFSGLNSAVLASNDEMVLLPINEPVRKSQIQTYLEHNEGAGLQHLALMSEDIFRTLREMRKRSSIGGFDFMPSPPPTYYQNLKKRVGDVLSDDQIKECEELGILVDRDDQGTLLQIFTKPLGDRPTIFIEIIQRVGCMMYQSGGCGGFGKGNFSELFKSIEEY 6j6m A 1.25 BS01 BA0 A 1 V416 A428 K430 M449 T474 Y476 M477 G480 C481 L528 S538 D539 F540 V24 A36 K38 M57 T82 Y84 M85 G88 C89 L136 S146 D147 F148 D521 R525 N526 D539 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 31381333 701 GSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6j72 A 2.2 BS01 GTP A 1 K46 G48 K49 S50 Q51 V64 T70 K200 D202 S232 V233 K48 G50 K51 S52 Q53 V66 T72 K202 D204 S234 V235 ? 0005525,0016020,0046872 Kd=0.74uM remove_due_to_license_issue I7FE16 31467269 701 MGVIVELIDHTSAIAAAKDRADLVERLRAAKARISDPQIRVVIAGQLKQGKSQLLNSLLNIPVARVGDDESTVLATVVSYGEQASARLVVARPDGAEPELIEIPPSEVTTDLRRAPQASGRQVLRVEVTAPSPLLKGGLAFVDTPGVGGHGQPHLSATLGLLPDADAMLMISDTSQEFTEPEMKFIRQALEICPVAAIVATKTDLYPHWRQIVDANIAHLQRAGLNVPVIPASSVLRSHAISLNDKELNEESNFPAIVKFLSEHVLSRQNDRIRDQIVDEIRSAAEHLLLAVESELSSFNDPGERERLTAELERRKQEAQDALQQTALWQQVLSDGIADLTADVDHDLRHRFRIIAAHTEKVIDGCDPTLHWAEIGAELEDAVATAVGDNFVWAYQRAEALAAEVARTFTEAGLDAVQMPQIDYGGVLMFGMLTSFAGLGMFNPLSLGAGFVLGRKAYKEDMENRMLRVRNEAKANVRKFVDDVAFVVGKESRDRLKGIQRQLRDHYREIANQTTRSLNESLQAAIAAAKVEEAERNTRVKELERQQNILKQVVDHAAKLA 6j7e A 2.4 BS01 AGS A 1 S145 L146 V147 S176 G177 G179 K180 E181 V182 L327 R334 V362 R363 S3 L4 V5 S34 G35 G37 K38 E39 V40 L185 R192 V220 R221 ? 0005524,0006355,0008134,0016887 remove_due_to_license_issue G3XCV0 31268665 401 FRSLVGTSRAIQQVRQMMQQVADTDASVLILGESGTGKEVVARNLHYHSKRREGPFVPVNCGAIPAELLESELFGHEKGAFTGAITSRAGRFELANGGTLFLDEIGDMPLPMQVKLLRVLQERTFERVGSNKTQNVDVRIIAATHKNLEKMIEDGTFREDLYYRLNVFPIEMAPLRERVEDIALLLNELISRMEHEKRGSIRFNSAAIMSLCRHDWPGNVRELANLVERLAIMHPYGVIGVGELPKKFRHV 6j7l A 1.851 BS01 TYD A 1 N13 Y14 G15 F190 Y192 F251 M252 Q254 Y257 R270 E272 D273 S274 N16 Y17 G18 F193 Y195 F254 M255 Q257 Y260 R273 E275 D276 S277 2.4.1.- 0016757,0106361 remove_due_to_license_issue Q9HZZ1 31010899 401 FQHMASWDIFCSVVDNYGDIGVTWRLARQLAAEHGQAVRLWVDEPQAFARICPRADPVAHVQCLDGVEVRAWGRPWAPVAAADVVIEAFACELPEAHRQAMRERKRPSLWLNLEYLSAEEWIGSCHALPSLQACGLSKYFFFPGFREPSGGLLREAGLLERRRRFQASVSAQDEFLASLGVRRKVGERLISLFAYENPALPGWLEQLRDARQPSLLLVPEGRVLADVADWLRVATLAVGDVHVRDALRVQVLPFMAQDDYDRLLWCCDLNAVRGEDSFVRAQWAGRPLLWHIYRTHLAKLEAFLELYCAGLPADLAENLRTFWLAWNAGGGLAGAWEGLERQLPEWRREAQRWADEQGMRPDLAARLVQFYADWLLEHHHHHH 6j81 A 1.8 BS01 B8X A 1 T448 H469 Y553 V571 E575 Y576 T85 H106 Y181 V199 E203 Y204 ? 0008289 remove_due_to_license_issue Q9Y5P4 600 THRFVQKVEEMVQNHMTYSLQDVGGDANWQLVVEEGEMKVYRREVEENGIVLDPLKATHAVKGVTGHEVCNYFWNVDVRNDWETTIENFHVVETLADNAIIIYQTHKRVWPASQRDVLYLSVIRKIPALDPETWIVCNFSVDHDSAPLNNRCVRAKINVAMICQTLVSEISRDNILCKITYVANVNPGGWAPASVLRAVAKREYPKFLKRFTSYVQEKTAGKPILF 6j8q A 1.787 BS01 BHU A 1 C69 S70 N132 E166 N170 T237 C44 S45 N107 E141 N145 T212 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31269398 301 STNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGL 6j8r A 1.575 BS03 BHU A 1 F62 Y67 W87 H116 D118 H179 N210 H240 F31 Y36 W56 H85 D87 H148 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 Ki=0.76uM remove_due_to_license_issue Q9K2N0 31269398 303 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6j9a A 2.915 BS01 dna B 0 R309 R347 W349 P350 N351 R19 R57 W59 P60 N61 ? 0003677 remove_due_to_license_issue Q8W4L5 30962525 1 ~ 15 IVPLFEKTLSASDAGRIGRLVLPKACAEAYFPPISQSEGIPLKIQDVRGREWTFQFRYWPNNNSRMYVLEGVTPCIQSMMLQAGDTVTFSRVDPGGKLIMGSRKAA 6j9a A 2.915 BS02 dna C 0 K297 S300 A301 S302 P313 N351 S354 M356 K7 S10 A11 S12 P23 N61 S64 M66 ? 0003677 remove_due_to_license_issue Q8W4L5 30962525 1 ~ 15 IVPLFEKTLSASDAGRIGRLVLPKACAEAYFPPISQSEGIPLKIQDVRGREWTFQFRYWPNNNSRMYVLEGVTPCIQSMMLQAGDTVTFSRVDPGGKLIMGSRKAA 6j9b A 1.9 BS01 dna C 0 K94 K97 S99 I108 K111 N149 M154 K6 K9 S11 I20 K23 N61 M66 ? 0003677,0003700 remove_due_to_license_issue Q9LW31 30962525 1 ~ 15 RFLFQKELKNSDVSSLRRMILPKKAAEAHLPALECKEGIPIRMEDLDGFHVWTFKYRYWPNNNSRMYVLENTGDFVNAHGLQLGDFIMVYQDLYSNNYVIQARKAS 6j9b A 1.9 BS02 dna B 0 R106 K124 R145 W147 N149 R18 K36 R57 W59 N61 ? 0003677,0003700 remove_due_to_license_issue Q9LW31 30962525 1 ~ 15 RFLFQKELKNSDVSSLRRMILPKKAAEAHLPALECKEGIPIRMEDLDGFHVWTFKYRYWPNNNSRMYVLENTGDFVNAHGLQLGDFIMVYQDLYSNNYVIQARKAS 6j9b D 1.9 BS01 dna F 0 K94 K97 N98 S99 I108 K111 N149 M154 K6 K9 N10 S11 I20 K23 N61 M66 ? 0003677,0003700 remove_due_to_license_issue Q9LW31 30962525 1 ~ 15 RFLFQKELKNSDVSSLRRMILPKKAAEAHLPALECKEGIPIRMEDLDGFHVWTFKYRYWPNNNSRMYVLENTGDFVNAHGLQLGDFIMVYQDLYSNNYVIQARKAS 6j9b D 1.9 BS02 dna E 0 R106 K124 R145 W147 P148 R18 K36 R57 W59 P60 ? 0003677,0003700 remove_due_to_license_issue Q9LW31 30962525 1 ~ 15 RFLFQKELKNSDVSSLRRMILPKKAAEAHLPALECKEGIPIRMEDLDGFHVWTFKYRYWPNNNSRMYVLENTGDFVNAHGLQLGDFIMVYQDLYSNNYVIQARKAS 6jad A 1.9 BS02 GLC B 1 D70 D118 G175 E230 W248 G285 G286 W287 R356 D68 D116 G173 E228 W246 G283 G284 W285 R354 ? remove_due_to_license_issue Q5SLD7 31608555 2 GPVIRVAGDSTAVGEGGRWMKEMVEAWGKKTGTRVEYIDSPADTNDRLALYQQYWAARSPDVDVYMIDVIWPGIVAPHALDLKPYLTEAELKEFFPRIVQNNTIRGKLTSLPFFTDAGILYYRKDLLEKYGYTSPPRTWNELEQMAERVMEGERRAGNRDFWGFVFQGKPYEGLTCDALEWIYSHGGGRIVEPDGTISVNNGRAALALNRAHGWVGRIAPQGVTSYAEEEARNVWQQGNSLFMRNWPYAYALGQAEGSPIRGKFGVTVLPKASADAPNAATLGGWQLMVSAYSRYPKEAVDLVKYLASYEVQKDNAVRLSRLPTRPALYTDRDVLARNPWFRDLLPVFQNAVSRPSDVAGARYNQVSEAIWTEVHSVLTGRKKGEQAVRDLEARIRRILRHHHH 6jao A 1.77 BS02 GLC B 1 D70 D118 G175 E230 W248 G285 G286 W287 D68 D116 G173 E228 W246 G283 G284 W285 ? remove_due_to_license_issue Q5SLD7 31608555 2 GPVIRVAGDSTAVGEGGRWMKEMVEAWGKKTGTRVEYIDSPADTNDRLALYQQYWAARSPDVDVYMIDVIWPGIVAPHALDLKPYLTEAELKEFFPRIVQNNTIRGKLTSLPFFTDAGILYYRKDLLEKYGYTSPPRTWNELEQMAERVMEGERRAGNRDFWGFVFQGKPYEGLTCDALEWIYSHGGGRIVEPDGTISVNNGRAALALNRAHGWVGRIAPQGVTSYAEEEARNVWQQGNSLFMRNWPYAYALGQAEGSPIRGKFGVTVLPKASADAPNAATLGGWQLMVSAYSRYPKEAVDLVKYLASYEVQKDNAVRLSRLPTRPALYTDRDVLARNPWFRDLLPVFQNAVSAPSDVAGARYNQVSEAIWTEVHSVLTGRKKGEQAVRDLEARIRRILRHHHH 6jaq A 1.95 BS01 GLC A 1 D70 D118 G175 E230 W248 G285 G286 W287 D68 D116 G173 E228 W246 G283 G284 W285 ? Kd=111.23uM remove_due_to_license_issue Q5SLD7 31608555 501 GPVIRVAGDSTAVGEGGRWMKEMVEAWGKKTGTRVEYIDSPADTNDRLALYQQYWAARSPDVDVYMIDVIWPGIVAPHALDLKPYLTEAELKEFFPRIVQNNTIRGKLTSLPFFTDAGILYYRKDLLEKYGYTSPPRTWNELEQMAERVMEGERRAGNRDFWGFVFQGKPYEGLTCDALEWIYSHGGGRIVEPDGTISVNNGRAALALNRAHGWVGRIAPQGVTSYAEEEARNVWQQGNSLFMRNWPYAYALGQAEGSPIRGKFGVTVLPKASADAPNAATLGGWQLMVSAYSRYPKEAVDLVKYLASYEVQKDNAVRLSRLPTRPALYTDRDVLARNPWFRDLLPVFQNAVSAPSDVAGARYNQVSEAIWTEVHSVLTGRKKGEQAVRDLEARIRRILRHHH 6jav A 1.437 BS01 BC0 A 1 W1621 W1691 W1809 W16 W86 W204 3.2.1.14 0004553,0005975,0008061 Ki=1.72uM remove_due_to_license_issue A0A221ZS22 31053640 2101 SLLNSRYKLVCYYTNWSWYRPGIGKYSPEDIDPSLCTHIVYGFAVLGNDGLMTAHDTWSDYDNRFYERVVEYKRYGIKVSLALGGWNDSAGDKYSKLVNDPAARAKFVQHAVAFLEKYGFDGLDLDWEYPKCWQVDCSKGPDSDKQGFADLVHELSAVLKPKGLLLSAAVSPNKMVIDAGYDVPVLARLLDWIAVMTYDYHGQWDKKTGHVAPLYYHPDDDTTYFNANYTIHYWMEKGTPASKIVMGMPMYGQSFTIENRGIHGLNIPVSDGGEPGEYTRAKGFLAYYEICDRIRNSGWTVVKDPYQRMGPYAYKGNQWVSFDDVEIIKKKVNFIKSLNLGGGMIWALDLDDYRNRCGQGKHPLLNAIKTELLNPKI 6jaw A 1.981 BS01 BBO A 1 W1691 D1804 W1809 Y1856 W1961 W86 D199 W204 Y251 W346 3.2.1.14 0004553,0005975,0008061 Ki=2.18uM remove_due_to_license_issue A0A221ZS22 31053640 2101 SLLNSRYKLVCYYTNWSWYRPGIGKYSPEDIDPSLCTHIVYGFAVLGNDGLMTAHDTWSDYDNRFYERVVEYKRYGIKVSLALGGWNDSAGDKYSKLVNDPAARAKFVQHAVAFLEKYGFDGLDLDWEYPKCWQVDCSKGPDSDKQGFADLVHELSAVLKPKGLLLSAAVSPNKMVIDAGYDVPVLARLLDWIAVMTYDYHGQWDKKTGHVAPLYYHPDDDTTYFNANYTIHYWMEKGTPASKIVMGMPMYGQSFTIENRGIHGLNIPVSDGGEPGEYTRAKGFLAYYEICDRIRNSGWTVVKDPYQRMGPYAYKGNQWVSFDDVEIIKKKVNFIKSLNLGGGMIWALDLDDYRNRCGQGKHPLLNAIKTELLNPKI 6jax A 1.7 BS01 GCS C 1 W1621 W1691 W16 W86 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue A0A221ZS22 31053640 3 SLLNSRYKLVCYYTNWSWYRPGIGKYSPEDIDPSLCTHIVYGFAVLGNDGLMTAHDTWSDYDNRFYERVVEYKRYGIKVSLALGGWNDSAGDKYSKLVNDPAARAKFVQHAVAFLEKYGFDGLDLDWEYPKCWQVDCSKGPDSDKQGFADLVHELSAVLKPKGLLLSAAVSPNKMVIDAGYDVPVLARLLDWIAVMTYDYHGQWDKKTGHVAPLYYHPDDDTTYFNANYTIHYWMEKGTPASKIVMGMPMYGQSFTIENRGIHGLNIPVSDGGEPGEYTRAKGFLAYYEICDRIRNSGWTVVKDPYQRMGPYAYKGNQWVSFDDVEIIKKKVNFIKSLNLGGGMIWALDLDDYRNRCGQGKHPLLNAIKTELLNPKI 6jax A 1.7 BS02 GCS C 2 V1740 W1809 V135 W204 3.2.1.14 0004553,0005975,0008061 remove_due_to_license_issue A0A221ZS22 31053640 5 SLLNSRYKLVCYYTNWSWYRPGIGKYSPEDIDPSLCTHIVYGFAVLGNDGLMTAHDTWSDYDNRFYERVVEYKRYGIKVSLALGGWNDSAGDKYSKLVNDPAARAKFVQHAVAFLEKYGFDGLDLDWEYPKCWQVDCSKGPDSDKQGFADLVHELSAVLKPKGLLLSAAVSPNKMVIDAGYDVPVLARLLDWIAVMTYDYHGQWDKKTGHVAPLYYHPDDDTTYFNANYTIHYWMEKGTPASKIVMGMPMYGQSFTIENRGIHGLNIPVSDGGEPGEYTRAKGFLAYYEICDRIRNSGWTVVKDPYQRMGPYAYKGNQWVSFDDVEIIKKKVNFIKSLNLGGGMIWALDLDDYRNRCGQGKHPLLNAIKTELLNPKI 6jay A 1.498 BS01 JUK A 1 W1691 Q1808 W1809 W86 Q203 W204 3.2.1.14 0004553,0005975,0008061 Ki=1.99uM remove_due_to_license_issue A0A221ZS22 31053640 2102 SLLNSRYKLVCYYTNWSWYRPGIGKYSPEDIDPSLCTHIVYGFAVLGNDGLMTAHDTWSDYDNRFYERVVEYKRYGIKVSLALGGWNDSAGDKYSKLVNDPAARAKFVQHAVAFLEKYGFDGLDLDWEYPKCWQVDCSKGPDSDKQGFADLVHELSAVLKPKGLLLSAAVSPNKMVIDAGYDVPVLARLLDWIAVMTYDYHGQWDKKTGHVAPLYYHPDDDTTYFNANYTIHYWMEKGTPASKIVMGMPMYGQSFTIENRGIHGLNIPVSDGGEPGEYTRAKGFLAYYEICDRIRNSGWTVVKDPYQRMGPYAYKGNQWVSFDDVEIIKKKVNFIKSLNLGGGMIWALDLDDYRNRCGQGKHPLLNAIKTELLNPKI 6jbe A 1.75 BS01 GLC A 1 D70 D118 G175 E230 W248 G285 G286 R356 D68 D116 G173 E228 W246 G283 G284 R354 ? Kd=19.8uM remove_due_to_license_issue Q5SLD7 31608555 501 GPVIRVAGDSTAVGEGGRWMKEMVEAWGKKTGTRVEYIDSPADTNDRLALYQQYWAARSPDVDVYMIDVIWPGIVAPHALDLKPYLTEAELKEFFPRIVQNNTIRGKLTSLPFFTDAGILYYRKDLLEKYGYTSPPRTWNELEQMAERVMEGERRAGNRDFWGFVFQGKPYEGLTCDALEWIYSHGGGRIVEPDGTISVNNGRAALALNRAHGWVGRIAPQGVTSYAEEEARNVWQQGNSLFMRNWPYAYALGQAEGSPIRGKFGVTVLPKASADAPNAATLGGAQLMVSAYSRYPKEAVDLVKYLASYEVQKDNAVRLSRLPTRPALYTDRDVLARNPWFRDLLPVFQNAVSRPSDVAGARYNQVSEAIWTEVHSVLTGRKKGEQAVRDLEARIRRILRHHHH 6jdi A 1.95 BS01 AGS A 1 S145 L146 V147 S176 G177 G179 K180 E181 V182 L327 R334 V362 R363 S4 L5 V6 S35 G36 G38 K39 E40 V41 L186 R193 V221 R222 ? 0005524,0006355,0008134,0016887 remove_due_to_license_issue G3XCV0 31268665 401 LFRSLVGTSRAIQQVRQMMQQVADTDASVLILGESGTGKEVVARNLHYHSKRREGPFVPVNCGAIPAELLESELFGHEKGAFTGAITSRAGRFELANGGTLFLDEIGDMPLPMQVKLLRVLQERTFERVGSNKTQNVDVRIIAATNKNLEKMIEDGTFREDLYYRLNVFPIEMAPLRERVEDIALLLNELISRMEHEKRGSIRFNSAAIMSLCRHDWPGNVRELANLVERLAIMHPYGVIGVGELPKKFRHV 6jdl A 2.249 BS01 AGS A 1 S145 L146 V147 S176 G177 G179 K180 E181 V182 R334 V362 R363 S4 L5 V6 S35 G36 G38 K39 E40 V41 R193 V221 R222 ? 0005524,0006355,0008134,0016887 remove_due_to_license_issue G3XCV0 31268665 401 LFRSLVGTSRAIQQVRQMMQQVADTDASVLILGESGTGKEVVARNLHYHSKRREGPFVPVNCGAIPAELLESELFGHEKGAFTGAITSRAGRFELANGGTLFLDEIGDMPLPMQVKLLRVLQERTFERVGSNKTQNVDVRIIAATAKNLEKMIEDGTFREDLYYRLNVFPIEMAPLRERVEDIALLLNELISRMEHEKRGSIRFNSAAIMSLCRHDWPGNVRELANLVERLAIMHPYGVIGVGELPKKFRHV 6jfk A 1.997 BS01 GDP A 1 S106 G108 K109 S110 T111 S124 I126 N258 R259 D261 S305 K307 S83 G85 K86 S87 T88 S101 I103 N235 R236 D238 S282 K284 3.6.5.- 0003924,0005525,0005741,0008053,0016020 remove_due_to_license_issue O95140 31664033 801 VNASPLKHFVTAKKKINGIFEQLGAYIQESATFLEDTYRNAELDPVTTEEQVLDVKGYLSKVRGISEVLARRHMKVAFFGRTSNGKSTVINAMLWDKVLPSGIGHTTNCFLRVEGTDGHEAFLLTEGSEEKRSAKTVNQLAHALHQDKQLHAGSLVSVMWPNSKCPLLKDDLVLMDSPGIDVTTELDSWIDKFCLDADVFVLVANSESTLMQTEKHFFHKVSERLSRPNIFILNNRWDASASEPEYMEEVRRQHMERCTSFLVDELGVVDRSQAGDRIFFVSAKEVLNARIQKAQGMPEGGGALAEGFQVRMFEFQNFERRFEECISQSAVKTKFEQHTVRAKQIAEAVRLIMDSLHMAAREQQVYCEEMREERQDRTRENLEQEIAAMNKKIEVLDSLQSKAKLLRNKAGWLDSELNMFTHQYLQPS 6jg8 A 2.097 BS01 dna C 0 N32 K77 T78 K79 R82 N109 N32 K77 T78 K79 R82 N109 ? 0098689 remove_due_to_license_issue O64094 31149347 1 ~ 30 MELIRIAMKKDLENDNSLMNKWATVAGLKNPNPLYDFLNHDGKTFNEFSSIVNIVKSQYPDREYELMKDYCLNLDVKTKAARSALEYADANMFFEIEDVLIDSMISCSNMKSKEYGKVYKIHRELSNSVITEFEAVKRLGKLNIKTPEMNSFSRLLLLYHYLSTGNFSPMAQLIKQIDLSEISENMYIRNTYQTRVHVLMSNIKLNENSLEECREYSKKALESTNILRFQVFSYLTIGNSLLFSNYELAQENFLKGLSISVQNENYNMIFQQALCFLNNVWRKENKWINFESDSIMDLQEQAHCFINFNENSKAKEVLDKLDLLVHNDNELAMHYYLKGRLEQNKACFYSSIEYFKKSNDKFLIRLPLLELQKMGENQKLLELLLL 6jg8 A 2.097 BS02 dna D 0 L28 K29 N30 N32 P33 K43 T44 F45 N46 L28 K29 N30 N32 P33 K43 T44 F45 N46 ? 0098689 remove_due_to_license_issue O64094 31149347 1 ~ 30 MELIRIAMKKDLENDNSLMNKWATVAGLKNPNPLYDFLNHDGKTFNEFSSIVNIVKSQYPDREYELMKDYCLNLDVKTKAARSALEYADANMFFEIEDVLIDSMISCSNMKSKEYGKVYKIHRELSNSVITEFEAVKRLGKLNIKTPEMNSFSRLLLLYHYLSTGNFSPMAQLIKQIDLSEISENMYIRNTYQTRVHVLMSNIKLNENSLEECREYSKKALESTNILRFQVFSYLTIGNSLLFSNYELAQENFLKGLSISVQNENYNMIFQQALCFLNNVWRKENKWINFESDSIMDLQEQAHCFINFNENSKAKEVLDKLDLLVHNDNELAMHYYLKGRLEQNKACFYSSIEYFKKSNDKFLIRLPLLELQKMGENQKLLELLLL 6jg8 B 2.097 BS01 dna C 0 L28 K29 N30 N32 P33 K43 T44 F45 N46 L29 K30 N31 N33 P34 K44 T45 F46 N47 ? 0098689 remove_due_to_license_issue O64094 31149347 1 ~ 30 MMELIRIAMKKDLENDNSLMNKWATVAGLKNPNPLYDFLNHDGKTFNEFSSIVNIVKSQYPDREYELMKDYCLNLDVKTKAARSALEYADANMFFEIEDVLIDSMISCSNMKSKEYGKVYKIHRELSNSVITEFEAVKRLGKLNIKTPEMNSFSRLLLLYHYLSTGNFSPMAQLIKQIDLSEISENMYIRNTYQTRVHVLMSNIKLNENSLEECREYSKKALESTNILRFQVFSYLTIGNSLLFSNYELAQENFLKGLSISVQNENYNMIFQQALCFLNNVWRKENKWINFESDSIMDLQEQAHCFINFNENSKAKEVLDKLDLLVHNDNELAMHYYLKGRLEQNKACFYSSIEYFKKSNDKFLIRLPLLELQKMGENQKLLELLLLLEHHHH 6jg8 B 2.097 BS02 dna D 0 T78 K79 R82 N109 T79 K80 R83 N110 ? 0098689 remove_due_to_license_issue O64094 31149347 1 ~ 30 MMELIRIAMKKDLENDNSLMNKWATVAGLKNPNPLYDFLNHDGKTFNEFSSIVNIVKSQYPDREYELMKDYCLNLDVKTKAARSALEYADANMFFEIEDVLIDSMISCSNMKSKEYGKVYKIHRELSNSVITEFEAVKRLGKLNIKTPEMNSFSRLLLLYHYLSTGNFSPMAQLIKQIDLSEISENMYIRNTYQTRVHVLMSNIKLNENSLEECREYSKKALESTNILRFQVFSYLTIGNSLLFSNYELAQENFLKGLSISVQNENYNMIFQQALCFLNNVWRKENKWINFESDSIMDLQEQAHCFINFNENSKAKEVLDKLDLLVHNDNELAMHYYLKGRLEQNKACFYSSIEYFKKSNDKFLIRLPLLELQKMGENQKLLELLLLLEHHHH 6jib A 2.25 BS01 BQF A 1 Y84 N87 K88 Q132 P309 G310 G313 P314 V317 Y49 N52 K53 Q97 P269 G270 G273 P274 V277 1.5.1.15,3.5.4.9 0003824,0004488 ic50=1.6uM remove_due_to_license_issue IC50=1600nM P13995 31223444 401 EAVVISGRKLAQQIKQEVRQEVEEWVASGNKRPHLSVILVGENPASHSYVLNKTRAAAVVGINSETIMKPASISEEELLNLINKLNNDDNVDGLLVQLPLPEHIDERRICNAVSPDKDVDGFHVINVGRMCLDQYSMLPATPWGVWEIIKRTGIPTLGKNVVVAGRSKNVGMPIAMLLHTDGAHERPGGDATVTISHRYTPKEQLKKHTILADIVISAAGIPNLITADMIKEGAAVIDVGINRVHKPKLVGDVDFEGVRQKAGYITPVPGGVGPMTVAMLMKNTIIAAKKVLR 6jib A 2.25 BS02 BQF A 2 G200 S231 H232 R233 T235 K237 L240 A254 I256 L259 G165 S196 H197 R198 T200 K202 L205 A219 I221 L224 1.5.1.15,3.5.4.9 0003824,0004488 ic50=1.6uM remove_due_to_license_issue IC50=1600nM P13995 31223444 403 EAVVISGRKLAQQIKQEVRQEVEEWVASGNKRPHLSVILVGENPASHSYVLNKTRAAAVVGINSETIMKPASISEEELLNLINKLNNDDNVDGLLVQLPLPEHIDERRICNAVSPDKDVDGFHVINVGRMCLDQYSMLPATPWGVWEIIKRTGIPTLGKNVVVAGRSKNVGMPIAMLLHTDGAHERPGGDATVTISHRYTPKEQLKKHTILADIVISAAGIPNLITADMIKEGAAVIDVGINRVHKPKLVGDVDFEGVRQKAGYITPVPGGVGPMTVAMLMKNTIIAAKKVLR 6jid A 2.5 BS01 BQC A 1 Y84 N87 K88 Q132 I276 P309 G313 P314 V317 Y49 N52 K53 Q97 I241 P270 G274 P275 V278 1.5.1.15,3.5.4.9 0003824,0004488 ic50=8.3uM remove_due_to_license_issue P13995 31223444 401 EAVVISGRKLAQQIKQEVRQEVEEWVASGNKRPHLSVILVGENPASHSYVLNKTRAAAVVGINSETIMKPASISEEELLNLINKLNNDDNVDGLLVQLPLPEHIDERRICNAVSPDKDVDGFHVINVGRMCLDQYSMLPATPWGVWEIIKRTGIPTLGKNVVVAGRSKNVGMPIAMLLHTDGAHERPGGDATVTISHRYTPKEQLKKHTILADIVISAAGIPNLITADMIKEGAAVIDVGINRVHDKPKLVGDVDFEGVRQKAGYITPVPGGVGPMTVAMLMKNTIIAAKKVLR 6jio A 2.6 BS01 BQ3 A 1 L274 A275 M312 F329 H435 L49 A50 M87 F104 H210 ? 0003677,0004879,0006629 remove_due_to_license_issue Ki=28000nM, EC50=57000nM P55055 31202993 501 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPSASQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDVHKILHRLLQD 6jip A 1.659 BS01 dna B 0 F12 W30 M58 G59 F2 W20 M48 G49 ? 0003677,0006355 remove_due_to_license_issue Q8DQG2 31713614 2 ~ 4 EFTFEIEEHLLTLSENEKGWTKEINRVSFNGAPAKFDIRAWSPDHTKMGKGITLSNEEFQTMVDAFK 6jki A 2.59 BS01 SFG A 1 Y91 L92 S93 P94 G118 Y120 E121 I138 L143 G145 G146 P149 Y89 L90 S91 P92 G116 Y118 E119 I136 L141 G143 G144 P147 P94 E121 R159 D174 P92 E119 R157 D165 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q9HXQ1 31399541 301 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 6jki A 2.59 BS02 SFG A 2 S175 D182 S166 D173 P94 E121 R159 D174 P92 E119 R157 D165 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q9HXQ1 31399541 306 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 6jki B 2.59 BS01 SFG A 1 D174 S175 D182 D168 S169 D176 P94 E121 R159 D174 P92 E119 R157 D168 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q9HXQ1 31399541 301 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALSAEEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 6jki B 2.59 BS02 SFG A 2 L92 S93 P94 G118 Y120 E121 I138 L143 G145 G146 P149 L90 S91 P92 G116 Y118 E119 I136 L141 G143 G144 P147 P94 E121 R159 D174 P92 E119 R157 D168 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 remove_due_to_license_issue Q9HXQ1 31399541 306 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALSAEEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 6jn3 A 2.216 BS01 BX6 A 1 C69 S70 W105 E166 N170 T237 C238 C44 S45 W80 E141 N145 T212 C213 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31269398 301 STNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGL 6jn4 A 1.9 BS01 BX9 A 1 C69 S70 K73 W105 S130 N132 E166 N170 T237 C44 S45 K48 W80 S105 N107 E141 N145 T212 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31269398 301 STNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGL 6jn5 A 1.97 BS01 BXU A 1 S70 W105 S130 E166 L167 N170 T237 S44 W79 S104 E140 L141 N144 T211 S70 K73 S130 E166 K234 T237 S44 K47 S104 E140 K208 T211 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31269398 301 TNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGL 6jn6 A 1.602 BS03 BY0 A 1 F62 W87 H116 D118 H179 R205 N210 F31 W56 H85 D87 H148 R174 N179 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0042597,0046677,0046872 Ki=0.07uM remove_due_to_license_issue Q9K2N0 31269398 304 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6jnl A 2.15 BS01 dna D 0 F1277 F1278 Y1282 H1286 V1289 W1309 S1312 H1316 R1338 F1339 D1342 F13 F14 Y18 H22 V25 W45 S48 H52 R74 F75 D78 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnl A 2.15 BS02 dna C 0 W1311 Y1326 V1340 S1341 S1344 R1348 W47 Y62 V76 S77 S80 R84 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 11 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnm A 2.05 BS01 dna D 0 F1277 F1278 Y1282 H1286 V1289 R1294 W1309 S1312 E1315 H1316 R1338 F1339 D1342 F13 F14 Y18 H22 V25 R30 W45 S48 E51 H52 R74 F75 D78 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnm A 2.05 BS02 dna C 0 K1281 W1311 Y1326 V1340 S1341 S1344 K1347 R1348 K17 W47 Y62 V76 S77 S80 K83 R84 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnm B 2.05 BS01 dna F 0 F1277 F1278 Y1282 H1286 V1289 R1294 W1309 S1312 E1315 H1316 R1338 F1339 D1342 F13 F14 Y18 H22 V25 R30 W45 S48 E51 H52 R74 F75 D78 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnm B 2.05 BS02 dna E 0 K1281 W1311 Y1326 V1340 S1341 S1344 K1347 R1348 K17 W47 Y62 V76 S77 S80 K83 R84 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn A 2.6 BS01 dna D 0 F1277 F1278 Y1282 W1309 S1312 H1316 F1339 D1342 F13 F14 Y18 W45 S48 H52 F75 D78 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn A 2.6 BS02 dna C 0 W1311 Y1326 V1340 S1341 S1344 R1348 W47 Y62 V76 S77 S80 R84 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn B 2.6 BS01 dna F 0 K1275 F1277 F1278 Y1282 H1286 W1309 S1312 H1316 F1339 D1342 K11 F13 F14 Y18 H22 W45 S48 H52 F75 D78 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn B 2.6 BS02 dna E 0 W1311 Y1326 V1340 S1341 S1344 K1347 R1348 W47 Y62 V76 S77 S80 K83 R84 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn G 2.6 BS01 dna L 0 F1277 F1278 Y1282 H1286 V1289 W1309 S1312 H1316 F1339 D1342 F12 F13 Y17 H21 V24 W44 S47 H51 F74 D77 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 NICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn G 2.6 BS02 dna K 0 W1311 V1340 S1341 S1344 W46 V75 S76 S79 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 NICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn N 2.6 BS01 dna I 0 F1277 F1278 Y1282 H1286 V1289 S1312 H1316 F1339 F13 F14 Y18 H22 V25 S48 H52 F75 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jnn N 2.6 BS02 dna H 0 W1311 V1340 S1341 S1344 R1348 W47 V76 S77 S80 R84 1.14.11.- remove_due_to_license_issue Q9STM3 31048693 1 ~ 12 RNICPIKGCGKNFFSHKYLVQHQRVHSDDRPLKCPWKGCKMTFKWAWSRTEHIRVHTGARPYVCAEPDCGQTFRFVSDFSRHKRKTGHS 6jno A 2.65 BS01 WY5 A 1 F439 K440 D444 F176 K177 D181 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue Kd=233nM, EC50=22nM, Ki=230nM P19793 31483660 501 PVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 6jno D 2.65 BS01 WY5 A 1 R302 W305 L433 R52 W55 L181 ? 0003677,0003707,0005634,0006355,0008270 remove_due_to_license_issue Kd=233nM, EC50=22nM, Ki=230nM P19793 31483660 501 PVERILEAELANDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEML 6joe A 2.21 BS01 BWR A 1 L92 S93 P94 Y120 E121 S137 I138 Y141 V142 L143 G145 G146 P149 L90 S91 P92 Y118 E119 S135 I136 Y139 V140 L141 G143 G144 P147 P94 E121 R159 D174 P92 E119 R157 D166 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.091uM remove_due_to_license_issue Q02RL6 31442049 301 SMLWVGVVSIFPEMFRAISDYGITSRAVKQGLLTLTCWNPRVYTEDRHQTVDDRPFGGGPGMVMKIKPLEGALADARQAAGGRKAKVIYLSPQGRQLTQAGVRELAEEEALILIAGRYEGIDERFIEEHVDEEWSIGDYVLSGGELPAMVLVDAVTRLLPGALEEDSFTDGLLDCPHYTRPEVYADKRVPEVLLSGNHEHIRRWRLQQALGRTWERRADLLDSRSLSGEEQKLLAEYIRQRD 6jof A 2.2 BS01 BWR A 1 P83 T84 P85 E112 S132 I133 Y136 V137 L138 G140 G141 P83 T84 P85 E112 S132 I133 Y136 V137 L138 G140 G141 P85 E112 R154 P85 E112 R154 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=10.4uM remove_due_to_license_issue Kd=10400nM P9WFY7 31442049 301 MRIDIVTIFPACLDPLRQSLPGKAIESGLVDLNVHDLRRWTHDVHHSVDDAPYGGGPGMVMKAPVWGEALDEICSSETLLIVPTPAGVLFTQATAQRWTTESHLVFACGRYEGIDQRVVQDAARRMRVEEVSIGDYVLPGGESAAVVMVEAVLRLLAGLEGPSYTRPASWRGLDVPEVLLSGDHARIAAWRREVSLQRTRERRPDL 6jon A 2.34 BS01 DTP A 1 K27 D78 D80 S108 P109 S110 H115 R145 Y146 M147 T148 K28 D79 D81 S109 P110 S111 H116 R146 Y147 M148 T149 2.7.7.-,2.7.7.7,3.6.4.12 Kd=13.2uM remove_due_to_license_issue M5AAG8 31176489 401 HMIMEIPAIKALSRYAQWVIWKKERDTKIPYNPNNGKKASSTDPLAWGDIDEAQAGLVRYGANGLGFVLTKSDPFVFIDLDHVLDENKRVKCEWARQLLKEIKSYTEISPSGDGLHVVVSGKLPDYIKHKTKFDDGSALEVYESGRYMTITGEVFDGRDDIKELDLSILGEFAEHKILDDEAIIDLMKRKGQWPDAPKDGDDWSSLDMSFANRLAFWCGKDIERMDRIFRQSPLMRQKWDRPTAGSTYGRITLKKACDFVDSVYDPALRNESDCPFEPYN 6jpj A 2.638 BS01 FGF A 1 L473 V481 R483 C552 A553 A554 L619 L20 V28 R30 C99 A100 A101 L166 D612 R616 N617 D630 D159 R163 N164 D177 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=1.9nM P22455 31041948 800 LPLDPLWEFPRDRLVLGKPLGEGAFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPDLSPDGPRSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAVSE 6jse A 2.0 BS01 C6R A 1 G35 Q36 G37 L54 D56 G58 Y95 F132 I142 D252 G254 T255 T256 A359 G16 Q17 G18 L35 D37 G39 Y76 F113 I123 D223 G225 T226 T227 A325 D56 S59 N61 A63 Y95 D252 T255 D37 S40 N42 A44 Y76 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=1.7nM remove_due_to_license_issue IC50=2.3nM P56817 31021626 508 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 6jsf A 2.3 BS01 C7X A 1 G35 G37 D56 Y95 Q97 G98 K131 F132 I142 D252 G254 T256 A359 G16 G18 D37 Y76 Q78 G79 K112 F113 I123 D222 G224 T226 A322 D56 S59 N61 A63 Y95 D252 T255 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=3.3nM remove_due_to_license_issue IC50=2.0nM P56817 31021626 510 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIP 6jsg A 2.3 BS01 C6U A 1 G35 Q36 G37 L54 D56 Y95 F132 D252 G254 T256 G16 Q17 G18 L35 D37 Y76 F113 D223 G225 T227 D56 S59 N61 A63 Y95 D252 T255 D37 S40 N42 A44 Y76 D223 T226 3.4.23.46 0004190,0006508,0016020 ic50=4.6nM remove_due_to_license_issue IC50=27nM P56817 31021626 507 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 6jsn A 2.6 BS01 C7O A 1 G35 G37 D56 Y95 F132 I142 D252 G254 T255 T256 G16 G18 D37 Y76 F113 I123 D224 G226 T227 T228 D56 S59 N61 A63 Y95 D252 T255 D37 S40 N42 A44 Y76 D224 T227 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=3.8nM, Ki=1.9nM P56817 31021626 508 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 6jsz A 1.53 BS01 C7O A 1 G27 R28 G29 L46 D48 Y87 I134 D241 G243 T245 A347 G13 R14 G15 L32 D34 Y73 I120 D218 G220 T222 A312 D48 S51 N53 A55 Y87 D241 T244 D34 S37 N39 A41 Y73 D218 T221 3.4.23.45 0004190,0006508,0016020 ic50=1.9nM remove_due_to_license_issue IC50=2090nM, Ki=1740nM Q9Y5Z0 31021626 401 ANFLAMVDNLQGGRGYYLEMLIGTPPQKLQILVDTGSSNFAVAGTPHSYIDTYFDTERSSTYRSKGFDVTVKYTQGSWTGFVGEDLVTIPKGFNTSFLVNIATIFESENFFLPGIKWNGILGLAYATLAKPSSSLETFFDSLVTQANIPNVFSMQMCGAGGGSLVLGGIEPSLYKGDIWYTPIKEEWYYQIEILKLEIGGQSLNLDCREYNADKAIVDSGTTLLRLPQKVFDAVVEAVARASLIPEFSDGFWTGSQLACWWSYFPKISIYLRDENSSRSFRITILPQLYIQPMYECYRFGISPSTNALVIGATVMEGFYVIFDRAQKRVGFAASPCAEIAGAAVSEISGPFSTEDVASNCVPA 6jt3 A 2.4 BS01 C83 A 1 G11 Q12 G13 L30 D32 Y71 F108 I118 D228 G230 T231 T232 A335 G16 Q17 G18 L35 D37 Y76 F113 I123 D222 G224 T225 T226 A329 D32 S35 N37 A39 Y71 D228 T231 D37 S40 N42 A44 Y76 D222 T225 3.4.23.46 0004190,0006508,0016020 ic50=5nM remove_due_to_license_issue IC50=0.380000nM P56817 31549838 505 RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6jtc A 2.39 BS01 C8O A 1 H85 W219 T650 T651 S655 D672 R673 H64 W198 T629 T630 S634 D651 R652 3.4.14.- 0008239,0070009 Ki=8.45uM remove_due_to_license_issue B2RID1 31537874 802 DEGMWLMQQLGRKYAQMKERGLKMKEYDLYNPNGTSLKDAVVLFDGGCTGEVVSDRGLVLTNHHCGYDMIQAHSTLEHNYLENGFWAMREADELPNKDISVVFIDKIEDVTDYVKKELKAIKDPNSMDYLSPKYLQKLADKKAGKNFSAKNPGLSVEIKAFYGGNLYLMFTKKTYTDVRLVGAPPSSIGKFGADTDNWIWPRHTGDFSIFRIYADKNGNPAPYSEDNVPLKPKRFFNISLGGVQENDYAMIMGFPGTTHRYFTASEVDEWKSIDNDIRIRMRDIRQGVMLREMLADPQIKIMYSAKYAASQNAYKRAIGANWAIKTRGLRQNKQAMQDRLIAWGAKQGTPRYEEAVHEIDATVAKRADLRRRYWMIEEGIIRGIEFARSPIPTEDETKALQGNDASARKEAIDKIRTRYSKFANKDYSAEVDKKVAVAMLTEYLKEIPYENLPLHLRLVKDRFAGDVQAYVDDIFARSVFGSEAQFDAFAAVPSVEKLAEDPMVLFASSVFDEYRKLYNELRPYDDPILRAQRTYIAGLLEMDGDQDQFPDANLTLRFTYGQVKGYSPRDNVYYGHQTTLDGVMEKEDPDNWEFVVDPKLKAVYERKDFGRYADRSGRMPVAFCATTHTTGGNSGSPVMNANGELIGLNFDRNWEGVGGDIQYLADYQRSIIVDIRYVLLVIDKVGGCQRLLDEMNIVP 6jut A 2.1 BS01 C9O A 1 C22 V30 A43 K45 A54 L57 S58 I66 F68 I80 T82 Y84 A85 V140 C150 D151 F152 G153 C15 V23 A36 K38 A47 L50 S51 I59 F61 I73 T75 Y77 A78 V133 C143 D144 F145 G146 D133 R137 N138 D151 D126 R130 N131 D144 2.7.11.25 0004672,0005524,0006468 ic50=2.1nM remove_due_to_license_issue IC50=2.1nM Q9NYL2 31244114 401 FVQIKFDDLQFFENCGGGSFGSVYRAKWISQDKEVAVKKLLKIEKEAEILSVLSHRNIIQFYGVILEPPNYGIVTEYASLGSLYDYINSNRSEEMDMDHIMTWATDVAKGMHYLHMEAPVKVIHRDLKSRNVVIAADGVLKICDFGASRFHNHTTHMSLVGTFPWMAPEVIQSLPVSETCDTYSYGVVLWEMLTREVPFKGLEGLQVAWLVVEKNERLTIPSSCPRSFAELLHQCWEADAKKRPSFKQIISILESMSNDTSLPDKCNSFLHNKAEWRCEIEATLERLKKLERDLSFK 6jz0 A 2.86 BS01 CKO A 1 L718 V726 A743 T790 M793 C797 D800 R841 L844 D855 L23 V31 A48 T94 M97 C101 D104 R145 L148 D159 D837 R841 N842 D855 D141 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=0.043000nM P00533 31560541 1100 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLMDEEDMDDVVDADEYLIP 6k04 A 1.251 BS01 CQF A 1 W370 P371 F372 V376 L383 N429 H433 V435 M438 W24 P25 F26 V30 L37 N83 H87 V89 M92 ? Ki=3.1nM remove_due_to_license_issue Ki=9.1nM, Kd=45nM P25440 31461688 501 SEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMP 6k05 A 1.935 BS01 CQF A 1 W97 P98 F99 K107 L108 L110 N156 W22 P23 F24 K32 L33 L35 N81 ? Ki=95.5nM remove_due_to_license_issue Ki=9.1nM, Kd=45nM P25440 31461688 201 TNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQE 6k0j A 2.352 BS01 CQO A 1 F233 V236 A249 L304 E352 L355 D368 F22 V25 A38 L93 E141 L144 D157 D348 K350 N353 D368 S385 D137 K139 N142 D157 S174 2.7.12.1 0004672,0005524,0006468 ic50=13nM remove_due_to_license_issue Q92630 31754034 601 QVPHDHVAYRYEVLKVIGKGSFGQVVKAYDHKVHQHVALKMVRNNKRFHRQAAEEIRILEHLRKQDKDNTMNVIHMLENFTFRNHICMTFELLSMNLYELIKKNKFQGFSLPLVRKFAHSILQCLDALHKNRIIHCDAKPENILLKQQGRSGIKVIDFGSSCYEHQRVYTYIQSRFYRAPEVILGARYGMPIDMWSLGCILAELLTGYPLLPGEDEGDQLACMIELLGMPSQKLLDASKRAKNFVSSKGYPRYCTVTTLSDGSVVLNGGRSRRGKLRGPPESREWGNALKGCDDPLFLDFLKQCLEWDPAVRMTPGQALRHPWLRAA 6k1q A 2.7 BS01 D2U A 1 D147 H150 N158 K161 P178 Q181 K182 S184 V185 F240 Y281 W336 L339 R343 A375 S376 S379 D57 H60 N68 K71 P88 Q91 K92 S94 V95 F144 Y185 W343 L346 R350 A382 S383 S386 3.2.1.17 0003796,0004930,0007186,0016020,0016998 remove_due_to_license_issue P00720,P24530 31263780 1201 QGPIEIKETFKYINTVVSCLVFVLGIIGNSTLLYIIYKNKCMRNGPNILIASLALGDLLHIVIDIPINVYKLLAEDWPFGAEMCKLVPFIQKASVGITVLSLCALSIDRYRAVASWSVPKWTAVEIVLIWVVSVVLAVPEAIGFDIITMDYKGSYLRICLLHPVQKTAFMQFYATAKDWWLFSFYFCLPLAITAFFYTLMTCEMLRKNIFEMLRIDEGAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYLNDHLKQRREVAKTVFCLVLVFALCWLPLHLARILKLTLYNQNDPNRCELLSFLLVLDYIGINMASLNSCANPIALYLVSKRFKNAFKSALCC 6k1s A 2.6 BS01 CUX A 1 P314 L315 L319 Y324 G365 E392 K393 D419 M420 E435 C449A P302 L303 L307 Y312 G353 E380 K381 D407 M408 E423 C437 2.1.1.320 0000387,0000785,0002039,0003714,0005515,0005634,0005654,0005694,0005737,0005794,0005829,0006325,0006338,0006353,0006355,0006479,0007088,0008168,0008327,0008469,0010468,0016274,0018216,0032259,0032922,0032991,0034709,0035097,0035243,0035246,0035642,0042054,0042118,0042802,0043021,0044020,0044027,0044877,0045596,0045892,0046982,0048026,0048511,0048714,0062122,0070372,0070611,0070888,0090161,0097421,0140592,0140759,0140903,0140938,0140984,1901796,1904992,1990259 remove_due_to_license_issue IC50=20nM O14744 31312404 700 RVSSGRDLNCVPEIADTLGAVAKQGFDFLCMPVFHPRFKREFIQEPAKNRPGPQTRSDLLLSGRDWNTLIVGKLSPWIRPDSKVEKIRRNSEAAMLQELNFGAYLGLPAFLLPLNQEDNTNLARVLTNHIHTGHHSSMFWMRVPLVAPEDLRDDIIENAPTTHTEEYSGEEKTWMWWHNFRTLCDYSKRIAVALEIGADLPSNHVIDRWLGEPIKAAILPTSIFLTNKKGFPVLSKMHQRLIFRLLKLEVQFIITGTNHHSEKEFCSYLQYLEYLSQNRPPPNAYELFAKGYEDYLQSPLQPLMDNLESQTYEVFEKDPIKYSQYQQAIYKCLLDRVPEEEKDTNVQVLMVLGAGRGPLVNASLRAAKQADRRIKLYAVEKNPNAVVTLENWQFEEWGSQVTVVSSDMREWVAPEKADIIVSELLGSFADNELSPECLDGAQHFLKDDGVSIPGEYTSFLAPISSSKLYNEVRACREKDRDPEAQFEMPYVVRLHNFHQLSAPQPCFTFSHPNRDPMIDNNRYCTLEFPVEVNTVLHGFAGYFETVLYQDITLSIRPETHSPGMFSWFPILFPIKQPITVREGQTICVRFWRCSNSKKVWYEWAVTAPVCSAIHNPTGRSYTIGL 6k4r A 3.109 BS01 AMP A 1 R352 K367 N534 R536 D542 D545 R254 K269 N420 R422 D428 D431 6.-.-.- 0000166,0006508,0008234,0016740,0016874,0046872,0106437,0106438 remove_due_to_license_issue Q5ZTK6 31330531 901 VKQYYFARRGETSTHDTSLPPPVKVLSGRSIPLKEIPFEATRNELVQIYLTSIDKLIKSNKLNSIPSQQIASHYLFLRSLANSETDGIKKNQILSLAKPLGTYLASKEPHVWKMINELIEKSEYPIIHYLKNNRAHSNFMLALIHEYHKEPLTKNQSAFVQKFRDSSVFLFPNPIYTAWLAHSYDEDSSFNPMFRERLSTNFYHSTLTDNLLLRTEPKEVTLSSEHHYKKEKGPIDSSFRYQMSSDRLLRIQGRTLLFSTPQNDVVAVKVQKKGEPKSTLEEEFEMADYLLKHQRRLDVHSKLPQPLGQYSVKKSEILEISRGSLTLIDDSKDLEVYVYKAPQSYFTYLHDKNQDLEDLTASVKTNVHDLFVLLREGIVFPQLADIFHKGRYQALVQLLNVLQFQLGRIDKWQKAVEYVNLRSSGLADLGDSLPITSLFTSSDFTKHYFSELLTGGYHPTFFDKSSGTANSLFTGKRRLFGNYLYLNTIAEYLLVIQLTLGSYGDKVTRDMDKPKKEAVWRELANVMFTSCAEAIHIMTGIPQSRALTLLKQRANIEKHFRQTQFWMTPDYSKLDEDTLQMEQYSIYSGEPEYEFTDKLVSGVGLSVDGVHQDLGGYNRESPLRELEKLLYATVTLIEGTMQLDKEFFKQLEQVEKILSGEIKTDANSCFEAVAQLLDLARPGCHFQKRLVLSYYEEAKLKYPSAPTDAYDSRFQVVARTNAAITIQRFWR 6k4t A 1.39 BS03 JKE A 1 H72 D76 H77 H150 S175 T177 V179 H215 H70 D74 H75 H148 S173 T175 V177 H213 H72 H74 D76 H77 H150 Y184 H215 H70 H72 D74 H75 H148 Y182 H213 3.5.2.6 0046872 remove_due_to_license_issue G5ELM3 31405855 303 RDWSSPQQPFTIYGNTHYVGTGGISAVLLSSPQGHILVDGTTEKGAQVVAANIRAMGFKLSDVKYILSTHSHEDHAGGISAMQKLTGATVLAGAANVDTLRTGVSPKSDPQFGSLSNFPGSAKVRAVADGELVKLGPLAVKAHATPGHTEGGITWTWQSCEQGKCKDVVFADSLTAVSADSYRFSDHPEVVASLRGSFEAVEKLSCDIAIAAHPEVNDMWTRQQRAAKEGNSAYVDNGACRAIAAAGRKRLETRLASEKR 6k4x A 1.17 BS03 D0U A 1 H72 D76 H150 S175 T177 V179 H215 H70 D74 H148 S173 T175 V177 H213 H72 H74 D76 H77 H150 Y184 H215 H70 H72 D74 H75 H148 Y182 H213 3.5.2.6 0046872 remove_due_to_license_issue G5ELM3 31405855 304 RDWSSPQQPFTIYGNTHYVGTGGISAVLLSSPQGHILVDGTTEKGAQVVAANIRAMGFKLSDVKYILSTHSHEDHAGGISAMQKLTGATVLAGAANVDTLRTGVSPKSDPQFGSLSNFPGSAKVRAVADGELVKLGPLAVKAHATPGHTEGGITWTWQSCEQGKCKDVVFADSLTAVSADSYRFSDHPEVVASLRGSFEAVEKLSCDIAIAAHPEVNDMWTRQQRAAKEGNSAYVDNGACRAIAAAGRKRLETRLASEKR 6k9u A 2.35 BS03 D4L A 1 L665 S667 Y683 P702 M703 E711 G715 F719 L207 S209 Y225 P244 M245 E253 G257 F261 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue Q9QYJ6 31235264 803 LPARICRDIELFHFDIGPFENMWPGIFVYMIHRSFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNNGLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLHNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKRDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLNQWEKVIRGEE 6kbs B 1.601 BS01 dna D 0 G3 R4 P40 W67 W68 K70 L73 N75 R77 S84 R85 M86 F87 W106 K113 T149 H160 R162 G209 G2 R3 P39 W66 W67 K69 L72 N74 R76 S83 R84 M85 F86 W105 K112 T148 H159 R161 G208 0003697,0006974,0106300 remove_due_to_license_issue 31504793 -1 ~ 7 CGRFAQSQTREDYLALLAEDIERDIPYDPEPIGRYNVAPGTKVLLLSERDEHLHLDPVFWGYAPGWWDKPPLINARVETAATSRMFKPLWQHGRAICFADGWFEWKKEGDKKQPFFIYRADGQPIFMAAIGSTPFERGDEAEGFLIVTAAADQGLVDIHDRRPLVLSPEAAREWMRQEISGKEASEIAASGCVPANQFSWHPVSRAVGNVKNQGAELIQPVLEVLFQ 6kdx A 2.44 BS03 D6X A 1 Y693 M713 E721 F729 Y247 M267 E275 F283 3.1.4.17 0004114,0007165,0008081 ic50=294nM remove_due_to_license_issue IC50=294nM Q9Y233 31301949 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 6kdz A 3.1 BS02 D79 A 1 Y693 M713 E721 V722 G725 F729 Y247 M267 E275 V276 G279 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=2.9nM Q9Y233 31301949 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 6ke0 A 2.95 BS02 D7C A 1 Y693 P712 M713 G725 F729 Y247 P266 M267 G279 F283 3.1.4.17 0004114,0007165,0008081 remove_due_to_license_issue IC50=69nM Q9Y233 31301949 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEE 6ki6 A 2.5 BS01 dna C 0 K749 N756 Y777 Q781 K784 R787 H788 T814 K10 N17 Y38 Q42 K45 R48 H49 T71 ? remove_due_to_license_issue Q9H165 31467406 1 ~ 13 RSDTCEYCGKVFKNCSNLTVHRRSHTGERPYKCELCNYACAQSSKLTRHMKTHGDVYKCEICKMPFSVYSTLEKHMKKWHS 6ki6 A 2.5 BS02 dna D 0 S755 S783 S16 S44 ? remove_due_to_license_issue Q9H165 31467406 1 ~ 13 RSDTCEYCGKVFKNCSNLTVHRRSHTGERPYKCELCNYACAQSSKLTRHMKTHGDVYKCEICKMPFSVYSTLEKHMKKWHS 6ki6 B 2.5 BS01 dna E 0 N753 S755 S783 N12 S14 S42 ? remove_due_to_license_issue Q9H165 31467406 1 ~ 13 DTCEYCGKVFKNCSNLTVHRRSHTGERPYKCELCNYACAQSSKLTRHMKTHG 6ki6 B 2.5 BS02 dna F 0 K749 N756 H760 Y777 Q781 K784 R787 H788 T791 K8 N15 H19 Y36 Q40 K43 R46 H47 T50 ? remove_due_to_license_issue Q9H165 31467406 1 ~ 13 DTCEYCGKVFKNCSNLTVHRRSHTGERPYKCELCNYACAQSSKLTRHMKTHG 6kjd B 2.299 BS01 LVA B 1 A57 Y127 F129 Y170 I236 E241 H253 F309 G345 G347 A58 Y128 F130 Y171 I237 E242 H254 F310 G346 G348 3.1.1.- 0016787 remove_due_to_license_issue B6H6L7 401 HMDTTFQAAIDTGKINGAVVCATDAQGHFVYNKATGERTLLSGEKQPQQLDDVLYLAAATKLITTIAALQCVEDGLLSLDGDLSSIAPELAAKYVLTGFTDDESPLDDPPARPITLKMLLTHSSGTSYHFLDPSIAKWRAQYANPENEKPRLVEEMFTYPLSFQPGTGWMYGPGLDWAGRVVERVTGGTLMEFMQKRIFDPLGITDSQFYPVTREDLRARLVDLNPSDPGALGSAVIGGGGEMNLRGRGAFGGHGLFLTGLDFVKILRSLLANDGMLLKPAAVDNMFQQHLGPEAAASHRAALASPLGPFFRVGTDPETKVGYGLGGLLTLEDVDGWYGERTLTWGGGLTLTWFIDRKNNLCGVGAIQAVLPVDGDLMADLKQTFRHDIYRKYSAWKGQQ 6kjf B 2.4 BS01 SIM B 1 A56 S57 F129 Y170 I236 E241 F309 W344 G345 G346 G347 A57 S58 F130 Y171 I237 E242 F310 W345 G346 G347 G348 3.1.1.- 0016787 remove_due_to_license_issue B6H6L7 404 HMDTTFQAAIDTGKINGAVVCATDAQGHFVYNKATGERTLLSGEKQPQQLDDVLYLASATKLITTIAALQCVEDGLLSLDGDLSSIAPELAAKYVLTGFTDDESPLDDPPARPITLKMLLTHSSGTSYHFLDPSIAKWRAQYANPENEKPRLVEEMFTYPLSFQPGTGWMYGPGLDWAGRVVERVTGGTLMEFMQKRIFDPLGITDSQFYPVTREDLRARLVDLNPSDPGALGSAVIGGGGEMNLRGRGAFGGHGLFLTGLDFVKILRSLLANDGMLLKPAAVDNMFQQHLGPEAAASHRAALASPLGPFFRVGTDPETKVGYGLGGLLTLEDVDGWYGERTLTWGGGLTLTWFIDRKNNLCGVGAIQAVLPVDGDLMADLKQTFRHDIYRKYSAWKGQQ 6kks A 2.15 BS01 dna B 0 K18 G19 L20 W21 K55 S56 R60 N106 N110 T114 K5 G6 L7 W8 K42 S43 R47 N93 N97 T101 ? remove_due_to_license_issue Q9SEI0 31733060 3 ~ 21 NEYKKGLWTVEEDKILMDYVKAHGKGHWNRIAKKTGLKRCGKSCRLRWMNYLSPNVKRGNFTEQEEDLIIRLHKLLGNRWSLIAKRVPGRTDNQVKNYWNTHLSKK 6kks A 2.15 BS02 dna C 0 L20 H40 W41 N42 K55 R58 N91 R92 W93 S94 K109 L7 H27 W28 N29 K42 R45 N78 R79 W80 S81 K96 ? remove_due_to_license_issue Q9SEI0 31733060 1 ~ 21 NEYKKGLWTVEEDKILMDYVKAHGKGHWNRIAKKTGLKRCGKSCRLRWMNYLSPNVKRGNFTEQEEDLIIRLHKLLGNRWSLIAKRVPGRTDNQVKNYWNTHLSKK 6kla A 2.109 BS01 DJX A 1 T670 Y672 C673 G676 L799 D810 F811 T117 Y119 C120 G123 L177 D188 F189 D792 R796 N797 D810 D170 R174 N175 D188 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue P10721 31721578 1001 EVQWKVVEEINGNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSEDDELALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISES 6klk A 1.759 BS01 URF A 1 Y155 M288 S289 D316 C318 N337 Y154 M287 S288 D315 C317 N336 3.5.2.2 0004157,0005737,0005829,0016787,0016810,0016812,0046872 Kd=133.2uM remove_due_to_license_issue Q9I676 31481233 501 SLLIRGATVVTHEESYRADVLCANGLIQAIGENLETPSGCDVLDGGGQYLMPGGIDPHTHMQLPFMGTVASEDFFSGTAAGLAGGTTSIIDFVIPNPRQSLLEAFHTWRGWAQKSAADYGFHVAITWWSDEVAREMGELVAQHGVNSFKHFMAYKNAIMAADDTLVASFERCLELGAVPTVHAENGELVFHLQQKLLAQGLTGPEAHPLSRPPQVEGEAASRAIRIAETLGTPLYLVHISSREALDEIAYARAKGQPVYGEVLAGHLLLDDSVYRHPDWATAAGYVMSPPFRPVEHQEALWRGLQSGNLHTTATDHCCFCAEQKAMGRDDFSKIPNGTAGIEDRMALLWDAGVNSGRLSMHEFVALTSTNTAKIFNLFPRKGAIRVGADADLVLWDPQGSRTLSAATHHQRVDFNIFEGRTVRGIPSHTISQGKLLWAAGDLRAEPGAGRYVERPAYPSVYEVLGRRAERQRPVAVER 6kwq A 1.76 BS01 rna B 0 N18 P20 T21 K24 H44 S45 K46 E108 T114 S115 K126 K127 Y157 K159 I176 A178 R188 H199 G211 C212 N213 R277 S289 G290 C291 S292 Y327 R416 L420 N18 P20 T21 K24 H44 S45 K46 E108 T114 S115 K126 K127 Y157 K159 I176 A178 R188 H199 G211 C212 N213 R277 S289 G290 C291 S292 Y327 R416 L420 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0003723,0003968,0006351,0039694 remove_due_to_license_issue M4QLY4 31863580 581 ~ 611 GEIQWVKPNKETGRLNINGPTRTKLEPSVFHDIFEGNKEPAVLHSKDPRLEVDFEQALFSKYVGNTLHEPDEYIKEAALHYANQLKQLEINTSQMSMEEACYGTENLEAIDLHTSAGYPYSALGIKKRDILDPTTRDVSKMKFYMDKYGLDLPYSTYVKDELRSIDKIKKGKSRLIEASSLNDSVYLRMAFGHLYEAFHANPGTITGSAVGCNPDTFWSKLPILLPGSLFAFDYSGYDASLSPVWFRALELVLREIGYSEEAVSLIEGINHTHHVYRNKTYCVLGGMPSGCSGTSIFNSMINNIIIRALLIKTFKGIDLDELNMVAYGDDVLASYPFPIDCLELAKTGKEYGLTMTPADKSPCFNEVNWGNATFLKRGFLPDEQFPFLIHPTMPMREIHESIRWTKDARNTQDHVRSLCLLAWHNGKQEYEKFVSTIRSVPVGRALAIPNYENLRRNWLELF 6kwq A 1.76 BS02 rna C 0 H113 R128 Y327 G328 D330 L375 K376 S401 K406 N410 D413 H414 S417 H113 R128 Y327 G328 D330 L375 K376 S401 K406 N410 D413 H414 S417 2.7.7.48,3.4.22.28,3.4.22.29,3.6.1.15 0003723,0003968,0006351,0039694 remove_due_to_license_issue M4QLY4 31863580 691 ~ 701 GEIQWVKPNKETGRLNINGPTRTKLEPSVFHDIFEGNKEPAVLHSKDPRLEVDFEQALFSKYVGNTLHEPDEYIKEAALHYANQLKQLEINTSQMSMEEACYGTENLEAIDLHTSAGYPYSALGIKKRDILDPTTRDVSKMKFYMDKYGLDLPYSTYVKDELRSIDKIKKGKSRLIEASSLNDSVYLRMAFGHLYEAFHANPGTITGSAVGCNPDTFWSKLPILLPGSLFAFDYSGYDASLSPVWFRALELVLREIGYSEEAVSLIEGINHTHHVYRNKTYCVLGGMPSGCSGTSIFNSMINNIIIRALLIKTFKGIDLDELNMVAYGDDVLASYPFPIDCLELAKTGKEYGLTMTPADKSPCFNEVNWGNATFLKRGFLPDEQFPFLIHPTMPMREIHESIRWTKDARNTQDHVRSLCLLAWHNGKQEYEKFVSTIRSVPVGRALAIPNYENLRRNWLELF 6kzc A 2.0 BS01 DZC A 1 L544 A570 K572 E588 L591 L592 V601 F617 E618 Y619 M620 H677 L686 G696 D697 F698 L17 A43 K45 E61 L64 L65 V74 F90 E91 Y92 M93 H138 L147 G157 D158 F159 D679 R683 N684 D697 D140 R144 N145 D158 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=11.46nM remove_due_to_license_issue Q16288 31271959 901 TYVQHIKRRDIVLKRELGEGAFGKVFLAECYNLSPTKDKMLVAVKALKDPTLAARKDFQREAELLTNLQHEHIVKFYGVCGDGDPLIMVFEYMKHGDLNKFLRAHGPDAGELGLSQMLHIASQIASGMVYLASQHFVHRDLATRNCLVGANLLVKIGDFGMSRVYSTDYYRLHTMLPIRWMPPESIMYRKFTTESDVWSFGVILWEIFTYGKQPWFQLSNTEVIECITQGRVLERPRVCPKEVYDVMLGCWQREPQQRLNIKEIYKILHALGKATPIYLDI 6kzd A 1.708 BS01 DZ6 A 1 A570 K572 E588 L592 V601 F617 Y619 M620 L686 G696 D697 F698 A43 K45 E61 L65 V74 F90 Y92 M93 L147 G157 D158 F159 D679 R683 N684 D697 D140 R144 N145 D158 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=2.95nM remove_due_to_license_issue Q16288 31271959 901 TYVQHIKRRDIVLKRELGEGAFGKVFLAECYNLSPTKDKMLVAVKALKDPTLAARKDFQREAELLTNLQHEHIVKFYGVCGDGDPLIMVFEYMKHGDLNKFLRAHGPDAGELGLSQMLHIASQIASGMVYLASQHFVHRDLATRNCLVGANLLVKIGDFGMSRDVYSTDYYRLHTMLPIRWMPPESIMYRKFTTESDVWSFGVILWEIFTYGKQPWFQLSNTEVIECITQGRVLERPRVCPKEVYDVMLGCWQREPQQRLNIKEIYKILHALGKATPIYLDI 6lc1 A 3.12 BS01 dna C 0 R293 R316 N317 R346 G347 R348 R28 R51 N52 R81 G82 R83 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 25 RCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPS 6lc1 A 3.12 BS02 dna F 0 Q277 H278 Y279 K288 K292 Q296 V336 R338 R345 R346 G347 R348 Q12 H13 Y14 K23 K27 Q31 V71 R73 R80 R81 G82 R83 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 26 RCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPS 6lc1 D 3.12 BS01 dna C 0 Q277 H278 Y279 K292 Q296 V336 V337 R338 R346 Q13 H14 Y15 K28 Q32 V72 V73 R74 R82 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 25 GRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLP 6lc1 D 3.12 BS02 dna F 0 E285 F290 R293 R316 N317 Q320 R323 R345 R346 G347 R348 P350 E21 F26 R29 R52 N53 Q56 R59 R81 R82 G83 R84 P86 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 26 GRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLP 6lc1 G 3.12 BS01 dna I 0 E285 G286 F290 R293 R316 N317 R323 R345 G347 R348 S351 E20 G21 F25 R28 R51 N52 R58 R80 G82 R83 S86 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 26 RCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPS 6lc1 G 3.12 BS02 dna L 0 C276 Q277 H278 Y279 K288 K292 R338 R345 R346 R348 C11 Q12 H13 Y14 K23 K27 R73 R80 R81 R83 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 25 RCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPS 6lc1 G 3.12 BS03 dna F 0 D340 S341 D75 S76 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 26 RCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPS 6lc1 J 3.12 BS01 dna I 0 Q277 H278 Y279 Q296 V336 V337 R338 R346 Q13 H14 Y15 Q32 V72 V73 R74 R82 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 26 GRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLP 6lc1 J 3.12 BS02 dna L 0 R293 R316 N317 Q320 R323 R346 G347 R348 R29 R52 N53 Q56 R59 R82 G83 R84 ? 0003700,0006355,0008270,0043565 remove_due_to_license_issue P22736 31822342 1 ~ 25 GRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAKYICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLP 6m7h A 1.6 BS01 KN9 A 1 E11 M109 M124 E127 A128 M144 E8 M106 M121 E124 A125 M141 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 remove_due_to_license_issue P0DP23 31401388 201 LTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTA 6m7h A 1.6 BS02 KN9 A 2 E11 A15 M72 I100 M124 M144 E8 A12 M69 I97 M121 M141 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 remove_due_to_license_issue P0DP23 31401388 202 LTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTA 6m7h A 1.6 BS03 KN9 A 3 F19 L32 M36 L39 M71 A88 F92 M109 L112 M145 F16 L29 M33 L36 M68 A85 F89 M106 L109 M142 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 remove_due_to_license_issue P0DP23 31401388 203 LTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTA 6m7i A 1.701 BS01 J84 A 1 G255 R256 A257 G230 R231 A232 S70 K73 S130 E166 K234 T237 S46 K49 S106 E142 K210 T213 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=386uM remove_due_to_license_issue Q9F663 30942078 301 MLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGV 6m7i A 1.701 BS02 J84 A 2 L167 N170 S171 T237 C238 G239 L143 N146 S147 T213 C214 G215 S70 K73 S130 E166 K234 T237 S46 K49 S106 E142 K210 T213 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=386uM remove_due_to_license_issue Q9F663 30942078 302 MLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGV 6m7i A 1.701 BS03 J84 A 3 S70 W105 S130 L167 T235 G236 T237 S46 W81 S106 L143 T211 G212 T213 S70 K73 S130 E166 K234 T237 S46 K49 S106 E142 K210 T213 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=386uM remove_due_to_license_issue Q9F663 30942078 303 MLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGV 6m7i A 1.701 BS04 J84 A 4 W105 P107 W81 P83 S70 K73 S130 E166 K234 T237 S46 K49 S106 E142 K210 T213 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=386uM remove_due_to_license_issue Q9F663 30942078 304 MLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGV 6m88 A 1.9 BS01 MYC A 1 V73 P111 E131 D132 V133 I142 R182 L254 I384 V9 P47 E67 D68 V69 I78 R118 L190 I205 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=1.1uM remove_due_to_license_issue IC50=1100nM Q8NFU5 30624931 501 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m89 A 1.85 BS01 QUE A 1 K75 P111 E131 D132 V133 I142 L254 I384 K11 P47 E67 D68 V69 I78 L190 I205 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=2.3uM remove_due_to_license_issue IC50=2300nM Q8NFU5 30624931 1001 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m8a A 1.75 BS01 LU2 A 1 I65 Q67 K75 P111 E131 D132 V133 I142 L254 I384 I1 Q3 K11 P47 E67 D68 V69 I78 L190 I206 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=5.5uM remove_due_to_license_issue IC50=5500nM Q8NFU5 30624931 501 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m8b A 1.8 BS01 KMP A 1 I65 Q67 P111 E131 D132 V133 I142 L254 I384 I1 Q3 P47 E67 D68 V69 I78 L190 I206 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=4.4uM remove_due_to_license_issue IC50=4400nM Q8NFU5 30624931 501 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m8c A 1.8 BS01 IRH A 1 I65 Q67 K75 P111 E131 D132 V133 I142 L254 I384 I1 Q3 K11 P47 E67 D68 V69 I78 L190 I206 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=2.2uM remove_due_to_license_issue IC50=2200nM Q8NFU5 30624931 501 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m8d A 2.0 BS01 J8D A 1 I65 K75 P111 E131 D132 V133 I142 L254 I384 I1 K11 P47 E67 D68 V69 I78 L190 I206 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=7.2uM remove_due_to_license_issue IC50=7200nM Q8NFU5 30624931 501 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m8e A 2.0 BS01 J8G A 1 I65 K75 P111 E131 D132 L254 I384 D385 I1 K11 P47 E67 D68 L190 I206 D207 2.7.1.140,2.7.1.151,2.7.1.153 0016301,0032958 ic50=14uM remove_due_to_license_issue IC50=14000nM Q8NFU5 30624931 501 ILQHPDGTVLKQLQPPPRGPRELEFYNMVYAADCFDGVLLELRKYLPKYYGIWSPPTAPNDLYLKLEDVTHKFNKPCIMDVKIGQKSYDPFASSEKIQQQVSKYPLMEEIGFLVLGMRVYHVHSDSYETENQHYGRSLTKETIKDGVSRFFHNGYCLRKDAVAASIQKIEKILQWFENQKQLNFYASSLLFVYEGSSGGEVEVRMIDFAHVFPSNTIDEGYVYGLKHLISVLRSILDN 6m8q A 2.49 BS03 JBG A 1 P45 L47 E48 Y110 V240 F241 P329 G330 M331 Q333 G356 P37 L39 E40 Y102 V232 F233 P321 G322 M323 Q325 G348 3.1.27.- remove_due_to_license_issue Q9UKF6 31819276 503 SDQLLIRPLGAGQEVGRSCIILEFKGRKIMLDCGIHPGLEGMDALPYIDLIDPAEIDLLLISHFHLDHCGALPWFLQKTSFKGRTFMTHATKAIYRWLLSDYVKVSNISADDMLYTETDLEESMDKIETINFHEVKEVAGIKFWCYHAGHVLGAAMFMIEIAGVKLLYTGDFSRQEDRHLMAAEIPNIKPDILIIESTYGTHIHEKREEREARFCNTVHDIVNRGGRGLIPVFALGRAQELLLILDEYWQNHPELHDIPIYYASSLAKKCMAVYQTYVNAMNDKIRKQININNPFVFKHISNLKSMDHFDDIGPSVVMASPGMMQSGLSRELFESWCTDKRNGVIIAGYCVEGTLAKHIMSEPEEITTMSGQKLPLKMSVDYISFSAHTDYQQTSEFIRALKPPHVILVHGEQNEMARLKAALIREYEDNDEVHIEVHNPRNTEAVTLNFR 6m95 A 1.8 BS01 J8S A 1 Y35 A51 K53 L104 T106 M109 G110 A111 D112 N115 A157 Y31 A47 K49 L100 T102 M105 G106 A107 D108 N111 A153 D150 K152 N155 D168 T185 D146 K148 N151 D164 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=140nM remove_due_to_license_issue Q16539 30945818 501 RPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 6m9l A 2.45 BS01 J9G A 1 V30 V38 A51 K53 L104 T106 M109 G110 A111 L167 V26 V31 A44 K46 L97 T99 M102 G103 A104 L160 D150 K152 N155 D168 T185 D143 K145 N148 D161 T164 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=29nM remove_due_to_license_issue Q16539 30945818 501 RPTFYRQELNKTIWEVPERYQNLSPVGYGSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGTRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 6m9t A 2.5 BS01 J9P A 1 T106 T107 Y114 M137 F140 G141 T206 W207 L329 R333 S336 Q339 T61 T62 Y69 M92 F95 G96 T161 W162 L413 R417 S420 Q423 3.2.1.17 0003796,0004930,0007186,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659 remove_due_to_license_issue P00720,P43115 30510194 2101 DCGSVSVAFPITMLLTGFVGNALAMLLVSRSYRRRESKRKKSFLLCIGWLALTDLVGQLLTTPVVIVVYLSKQRWEHIDPSGRLCTFFGLTMTVFGLSSLFIASAMAVERALAIRAPHWYASHMKTRATRAVLLGVWLAVLAFALLPVLGVGQYTVQWPGTWCFISTNWGNLFFASAFAFLGLLALTVTFSCNLATIKALVSRGSNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDATVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYGSWGRITTETAIQLMAIMCVLSVCWSPLLIMMLKMIFNEKQKECNFFLIAVRLASLNQILDPWVYLLLRKILGRPLEVL 6ma1 A 2.75 BS02 JA4 A 1 H558 P559 H562 Q839 L866 F868 V895 A896 K898 H901 R904 H246 P247 H250 Q508 L535 F537 V564 A565 K567 H570 R573 2.4.1.255 0006493,0016757 remove_due_to_license_issue O15294 30285435 1101 CPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 6ma2 A 2.1 BS02 J9S A 1 N557 H558 P559 H562 L866 F868 V895 A896 K898 H901 N245 H246 P247 H250 L535 F537 V564 A565 K567 H570 2.4.1.255 0006493,0016757 Kd=4.1uM remove_due_to_license_issue O15294 30285435 1101 CPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 6ma3 A 2.0 BS02 JAJ A 1 H558 P559 H562 Q839 L866 F868 V895 A896 K898 H901 T921 H246 P247 H250 Q508 L535 F537 V564 A565 K567 H570 T590 2.4.1.255 0006493,0016757 Kd=0.005uM remove_due_to_license_issue O15294 30285435 1101 CPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 6ma4 A 2.0 BS02 JA7 A 1 H558 P559 H562 Q839 F868 V895 A896 K898 H901 R904 H920 T921 H247 P248 H251 Q509 F538 V565 A566 K568 H571 R574 H590 T591 2.4.1.255 0006493,0016757 Kd=0.045uM remove_due_to_license_issue O15294 30285435 1101 SCPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 6ma5 A 2.0 BS02 J9V A 1 H558 P559 H562 Q839 L866 F868 V895 A896 K898 H901 H246 P247 H250 Q508 L535 F537 V564 A565 K567 H570 2.4.1.255 0006493,0016757 Kd~140nM remove_due_to_license_issue O15294 30285435 1101 CPTHADSLNNLANIKREQGNIEEAVRLYRKALEVFPEFAAAHSNLASVLQQQGKLQEALMHYKEAIRISPTFADAYSNMGNTLKEMQDVQGALQCYTRAIQINPAFADAHSNLASIHKDSGNIPEAIASYRTALKLKPDFPDAYCNLAHCLQIVCDWTDYDERMKKLVSIVADQLEKNRLPSVHPHHSMLYPLSHGFRKAIAERHGNLCLDKINVLHKPPYEHPKDLKLSDGRLRVGYVSSDFGNHPTSHLMQSIPGMHNPDKFEVFCYALSPDDGTNFRVKVMAEANHFIDLSQIPCNGKAADRIHQDGIHILVNMNGYTKGARNELFALRPAPIQAMWLGYPGTSGALFMDYIITDQETSPAEVAEQYSEKLAYMPHTFFIGDHANMFPHLKKKAVIDFKIYDNRIVLNGIDLKAFLDSLPDVKIVKMLNMPVIPMNTIAEAVIEMINRGQIQITINGFSISNGLATTQINNKAATGEEVPRTIIVTTRSQYGLPEDAIVYCNFNQLYKIDPSTLQMWANILKRVPNSVLWLLRFPAVGEPNIQQYAQNMGLPQNRIIFSPVAPKEEHVRRGQLADVCLDTPLCNGHTTGMDVLWAGTPMVTMPGETLASRVAASQLTCLGCLELIAKNRQEYEDIAVKLGTDLEYLKKVRGKVWKQRISSPLFNTKQYTMELERLYLQMWEHYAAGNKPDHMIK 6maj A 2.139 BS03 JAV A 1 T477 R483 G485 G487 K488 S512 L514 G515 S518 E525 T143 R149 G151 G153 K154 S178 L180 G181 S184 E191 2.3.1.48 0004402,0006355 remove_due_to_license_issue O95251 31827282 704 SMIKTIAFGRYELDTWYHSPYPEEYARLGRLYMCEFCLKYMKSQTILRRHMAKCVWKHPPGDEIYRKGSISVFEVDGKKNKIYCQNLCLLAKLFLDHKTLYYDVEPFLFYVMTEADNTGCHLIGYFSKEKNSFLNYNVSCILTMPQYMRQGYGKMLIDFSYLLSKVEEKVGSPERPLSDLGLISYRSYWKEVLLRYLHNFQGKEISIKEISQETAVNPVDIVSTLQALQMLKYWKGKHLVLKRQDLIDEWIAKENKTMDPSCLKWTP 6mbo A 1.591 BS01 JDG A 1 T1026 Y1030 T52 Y56 Y1124 Y1211 Y150 Y237 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Q9H9B1 30753076 1301 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 6mbo A 1.591 BS02 JDG A 2 Y1124 A1134 D1135 D1140 S1141 L1143 D1145 V1153 C1155 F1209 R1214 F1215 I1218 Y150 A160 D161 D166 S167 L169 D171 V179 C181 F235 R240 F241 I244 Y1124 Y1211 Y150 Y237 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Q9H9B1 30753076 1302 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 6mbo B 1.591 BS01 JDG A 1 K1008 F1160 Y1161 K33 F183 Y184 Y1124 Y1211 Y149 Y234 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Q9H9B1 30753076 1301 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 6mbo B 1.591 BS02 JDG B 1 I1034 D1036 W1081 N1083 I59 D61 W106 N108 Y1124 Y1211 Y149 Y234 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Q9H9B1 30753076 1301 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 6mbo B 1.591 BS03 JDG B 2 Y1124 A1134 D1135 D1140 S1141 L1143 D1145 R1214 F1215 Y149 A159 D160 D165 S166 L168 D170 R237 F238 Y1124 Y1211 Y149 Y234 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Q9H9B1 30753076 1302 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 6mbp A 1.947 BS01 JDG A 1 Y1124 D1131 A1134 R1137 D1140 S1141 L1143 D1145 V1153 R1214 F1215 Y150 D157 A160 R163 D166 S167 L169 D171 V179 R240 F241 Y1124 Y1211 Y150 Y237 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054 remove_due_to_license_issue Q9H9B1 30753076 2001 VERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDNKDGEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGKLFSCRCGSPKCRHS 6mck A 3.77 BS01 JDP A 1 D478 I479 C522 G523 L526 I656 A659 N660 R662 G684 A685 T688 D247 I248 C291 G292 L295 I416 A419 N420 R422 G444 A445 T448 3.6.4.6 0005524,0016887 remove_due_to_license_issue IC50=1030nM, Ki=26nM P55072 30591537 900 RKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRVTMDDFRWALSQSNPSALRETVVEVPQVTWEDIGGLEDVKRELQELVQYPVEHPDKFLKFGMTPSKGVLFYGPPGCGKTLLAKAIANECQANFISIKGPELLTMWFGESEANVREIFDKARQAAPCVLFFDELDSIAKARAADRVINQILTEMDGMSTKKNVFIIGATNRPDIIDPAILRPGRLDQLIYIPLPDEKSRVAILKANLRKSPVAKDVDLEFLAKMTNGFSGADLTEICQRACKLAIRESIESEIRRERERQTEIRRDHFEEAMRFARRSVSDNDIRKYEMFAQTLQ 6mck B 3.77 BS01 JDP B 1 D478 I479 C522 G523 L526 I656 A659 N660 G684 A685 T688 D247 I248 C291 G292 L295 I416 A419 N420 G444 A445 T448 3.6.4.6 0005524,0016887 remove_due_to_license_issue IC50=1030nM, Ki=26nM P55072 30591537 900 RKQLAQIKEMVELPLRHPALFKAIGVKPPRGILLYGPPGTGKTLIARAVANETGAFFFLINGPEIMSKLAGESESNLRKAFEEAEKNAPAIIFIDELDAIAPKREKTHGEVERRIVSQLLTLMDGLKQRAHVIVMAATNRPNSIDPALRRFGRFDREVDIGIPDATGRLEILQIHTKNMKLADDVDLEQVANETHGHVGADLAALCSEAALQAIRVTMDDFRWALSQSNPSALRETVVEVPQVTWEDIGGLEDVKRELQELVQYPVEHPDKFLKFGMTPSKGVLFYGPPGCGKTLLAKAIANECQANFISIKGPELLTMWFGESEANVREIFDKARQAAPCVLFFDELDSIAKARAADRVINQILTEMDGMSTKKNVFIIGATNRPDIIDPAILRPGRLDQLIYIPLPDEKSRVAILKANLRKSPVAKDVDLEFLAKMTNGFSGADLTEICQRACKLAIRESIESEIRRERERQTEIRRDHFEEAMRFARRSVSDNDIRKYEMFAQTLQ 6md4 A 2.24 BS01 BRL A 1 F282 C285 S289 H323 M364 H449 Y473 F66 C69 S73 H107 M148 H233 Y257 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue EC50=40nM, IC50=1.000000nM, Ki=8nM, Kd=0.145000nM P37231 30575522 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 6md7 A 1.96 BS01 JE1 A 1 T108 R111 F113 T219 E250 T253 Q257 P491 K492 Q495 T105 R108 F110 T211 E234 T237 Q241 P462 K463 Q466 D425 C459 R465 T466 Q506 D396 C430 R436 T437 Q477 3.1.3.48 0004725,0006470,0016311 ic50=0.181uM remove_due_to_license_issue IC50=181nM Q06124 30688459 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHHGQLKENGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQSHPGDFVLSVRTGDNDGKSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPPVSDYINANIIMPEKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6md8 A 1.4 BS01 J84 A 1 N104 Y105 S130 T235 G236 S237 N79 Y80 S105 T210 G211 S212 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677,0046872 Ki=4200uM remove_due_to_license_issue Q9L5C7 30942078 601 PTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 6md8 A 1.4 BS02 J84 A 2 E25 T26 T55 Q56 V57 G289 L290 E1 T2 T31 Q32 V33 G262 L263 S70 K73 S130 E166 K234 S237 S45 K48 S105 E141 K209 S212 3.5.2.6 0008800,0016787,0017001,0030655,0046677,0046872 Ki=4200uM remove_due_to_license_issue Q9L5C7 30942078 602 PTSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERFPMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKPADLVNYNPIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPGGVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAMAQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLPTSWTVGDKTGSGDYGTTNDIAVIWPQGRAPLVLVTYFTQPQQNAESRRDVLASAARIIAEGL 6mdb A 2.34 BS01 JE4 A 1 R111 F113 H114 T219 E249 E250 T253 L254 Q257 P491 K492 Q495 R106 F108 H109 T203 E225 E226 T229 L230 Q233 P453 K454 Q457 D425 C459 R465 T466 Q506 D387 C421 R427 T428 Q468 3.1.3.48 0004725,0006470,0016311 ic50=0.064uM remove_due_to_license_issue Q06124 30688459 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHHGQLKGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQPGDFVLSVRTGDSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPPVSDYINANIIMPKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6mdc A 2.14 BS01 JEA A 1 T108 E110 R111 F113 T219 E249 E250 T253 L254 Q257 P491 K492 T94 E96 R97 F99 T192 E214 E215 T218 L219 Q222 P449 K450 D425 C459 R465 T466 Q506 D383 C417 R423 T424 Q464 3.1.3.48 0004725,0006470,0016311 ic50=0.036uM remove_due_to_license_issue Q06124 30688462 601 RRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESGDFVLSVRTGDSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKLQGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDGDPNEPVSDYINANIIMPEFKPKKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6mdd A 2.05 BS01 JE7 A 1 R111 T218 T219 E250 T253 L254 P491 K492 Q495 R101 T199 T200 E221 T224 L225 P443 K444 Q447 D425 C459 R465 T466 Q506 D377 C411 R417 T418 Q458 3.1.3.48 0004725,0006470,0016311 ic50=47uM remove_due_to_license_issue Q06124 30688462 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQSHPGDFVLSVRTGDSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDSDYINANIIMPKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6mdq A 2.15 BS01 TES A 1 R208 A212 G327 E353 R205 A209 G324 E350 ? 0003677,0005504,0005576,0005615,0005737,0008289,0009267,0015643,0019825,0030170,0032991,0046872,0051902,0072732,1903981 remove_due_to_license_issue P35747 30842823 604 KSEIAHRFNDLGEKHFKGLVLVAFSQYLQQCPFEDHVKLVNEVTEFAKKCAADESAENCDKSLHTLFGDKLCTVATLRATYGELADCCEKQEPERNECFLTHKDDHPNLPKLKPEPDAQCAAFQEDPDKFLGKYLYEVARRHPYFYGPELLFHAEEYKADFTECCPADDKLACLIPKLDALKERILLSSAKERLKCSSFQNFGERAVKAWSVARLSQKFPKADFAEVSKIVTDLTKVHKECCHGDLLECADDRADLAKYICEHQDSISGKLKACCDKPLLQKSHCIAEVKEDDLPSDLPALAADFAEDKEICKHYKDAKDVFLGTFLYEYSRRHPDYSVSLLLRIAKTYEATLEKCCAEADPPACYRTVFDQFTPLVEEPKSLVKKNCDLFEEVGEYDFQNALIVRYTKKAPQVSTPTLVEIGRTLGKVGSRCCKLPESERLPCSENHLALALNRLCVLHEKTPVSEKITKCCTDSLAERRPCFSALELDEGYVPKEFKAETFTFHADICTLPEDEKQIKKQSALAELVKHKPKATKEQLKTVLGNFSAFVAKCCGAEDKEACFAEEGPKLVASSQLALA 6mdq A 2.15 BS02 TES A 2 K17 G21 L134 G135 E158 K14 G18 L131 G132 E155 ? 0003677,0005504,0005576,0005615,0005737,0008289,0009267,0015643,0019825,0030170,0032991,0046872,0051902,0072732,1903981 remove_due_to_license_issue P35747 30842823 605 KSEIAHRFNDLGEKHFKGLVLVAFSQYLQQCPFEDHVKLVNEVTEFAKKCAADESAENCDKSLHTLFGDKLCTVATLRATYGELADCCEKQEPERNECFLTHKDDHPNLPKLKPEPDAQCAAFQEDPDKFLGKYLYEVARRHPYFYGPELLFHAEEYKADFTECCPADDKLACLIPKLDALKERILLSSAKERLKCSSFQNFGERAVKAWSVARLSQKFPKADFAEVSKIVTDLTKVHKECCHGDLLECADDRADLAKYICEHQDSISGKLKACCDKPLLQKSHCIAEVKEDDLPSDLPALAADFAEDKEICKHYKDAKDVFLGTFLYEYSRRHPDYSVSLLLRIAKTYEATLEKCCAEADPPACYRTVFDQFTPLVEEPKSLVKKNCDLFEEVGEYDFQNALIVRYTKKAPQVSTPTLVEIGRTLGKVGSRCCKLPESERLPCSENHLALALNRLCVLHEKTPVSEKITKCCTDSLAERRPCFSALELDEGYVPKEFKAETFTFHADICTLPEDEKQIKKQSALAELVKHKPKATKEQLKTVLGNFSAFVAKCCGAEDKEACFAEEGPKLVASSQLALA 6mdu A 1.15 BS03 N1G A 1 L65 M67 V73 W93 Q123 H189 C208 K211 N220 H250 L24 M26 V32 W52 Q82 H148 C167 K170 N179 H209 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 Ki=56uM remove_due_to_license_issue C7C422 30942078 303 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6me2 A 2.8 BS01 JEV A 1 M107 G108 N162 F179 Q181 V191 L254 M86 G87 N141 F158 Q160 V170 L420 ? 0004930,0007186,0008502,0016020 remove_due_to_license_issue P48039,Q9V2J8 31019306 1201 RPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVANLVVAIYPYPLVLMSIFNNGWNFGYLHCQVSAFLMGLSVIGSIWNITGIAIDRYLYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKLKPQDFRNFVTMFVVFVLFAICFAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNPIIYGLLDQNFRKEYRRIIVSLCTARVFF 6me3 A 2.9 BS01 JEY A 1 G108 V111 N162 L168 F179 Q181 L254 Y281 Y285 G86 V89 N140 L146 F157 Q159 L419 Y446 Y450 ? 0004930,0007186,0008502,0016020 remove_due_to_license_issue P48039,Q9V2J8 31019306 1201 PSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVANLVVAIYPYPLVLMSIFNNGWNFGYLHCQVSAFLMGLSVIGSIWNITGIAIDRYLYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKLKPQDFRNFVTMFVVFVLFAICFAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNPIIYGLLDQNFRKEYRRIIVSLCTARV 6me4 A 3.2 BS01 ML2 A 1 A104 G108 N162 F179 Q181 L254 A82 G86 N140 F157 Q159 L419 ? 0004930,0007186,0008502,0016020 remove_due_to_license_issue P48039,Q9V2J8 31019306 1201 PSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVANLVVAIYPYPLVLMSIFNNGWNFGYLHCQVSAFLMGLSVIGSIWNITGIAIDRYLYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKLKPQDFRNFVTMFVVFVLFAICFAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNPIIYGLLDQNFRKEYRRIIVSLCTARVFF 6me5 A 3.2 BS01 AWY A 1 A104 M107 G108 N162 T178 F179 Q181 V191 L254 A82 M85 G86 N140 T156 F157 Q159 V169 L419 ? 0004930,0007186,0008502,0016020 remove_due_to_license_issue P48039,Q9V2J8 31019306 1201 PSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRNAGNIFVVSLAVANLVVAIYPYPLVLMSIFNNGWNFGYLHCQVSAFLMGLSVIGSIWNITGIAIDRYLYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFAQSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRGIDCSFWNESYLTGSRDERKKSLLSKFGMDEGVTFMFIGRFDRGQKGVDVLLKAIEILSSKKEFQEMRFIIIGKGDPELEGWARSLEEKHGNVKVITEMLSREFVRELYGSVDFVIIPSYFEPFGLVALEAMCLGAIPIASAVGGLRDIITNETGILVKAGDPGELANAILKALELSRSDLSKFRENCKKRAMSFSKLKPQDFRNFVTMFVVFVLFAICFAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNPIIYGLLDQNFRKEYRRIIVSLCTARVFF 6mey A 1.42 BS01 O5E A 1 P94 T115 P65 T86 S70 K73 S130 E166 K234 T237 S41 K44 S101 E137 K205 T208 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=479uM remove_due_to_license_issue Q9F663 30942078 301 VAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHEAVIAAAARLALEGLGVNG 6mey A 1.42 BS02 O5E A 2 S84 Q85 Q87 A88 G89 L90 L91 A200 S55 Q56 Q58 A59 G60 L61 L62 A171 S70 K73 S130 E166 K234 T237 S41 K44 S101 E137 K205 T208 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=479uM remove_due_to_license_issue Q9F663 30942078 302 VAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHEAVIAAAARLALEGLGVNG 6mey A 1.42 BS03 O5E A 3 S70 S130 N170 T235 G236 T237 S41 S101 N141 T206 G207 T208 S70 K73 S130 E166 K234 T237 S41 K44 S101 E137 K205 T208 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=479uM remove_due_to_license_issue Q9F663 30942078 303 VAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHEAVIAAAARLALEGLGVNG 6mg1 A 1.75 BS01 dna C 0 Y274 R278 N282 R289 Y6 R10 N14 R21 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 1 ~ 16 KHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPEPL 6mg1 A 1.75 BS02 dna D 0 R280 A284 K287 S288 K291 R12 A16 K19 S20 K23 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 101 ~ 116 KHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPEPL 6mg1 B 1.75 BS01 dna C 0 A284 K287 S288 K291 A16 K19 S20 K23 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 1 ~ 16 KHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPEPL 6mg1 B 1.75 BS02 dna D 0 Y274 R278 N282 R286 R289 K293 Y6 R10 N14 R18 R21 K25 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 101 ~ 116 KHSDEYKIRRERNNIAVRKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPEPL 6mg3 A 2.05 BS01 dna C 0 Y274 R278 N281 N282 R286 R289 K293 Y6 R10 N13 N14 R18 R21 K25 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 1 ~ 16 KHSDEYKIRRERNNIAARKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFK 6mg3 A 2.05 BS02 dna D 0 R280 N281 A284 A285 K287 S288 R289 R12 N13 A16 A17 K19 S20 R21 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 101 ~ 116 KHSDEYKIRRERNNIAARKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFK 6mg3 B 2.05 BS01 dna C 0 R280 N281 A284 S288 R289 K291 R12 N13 A16 S20 R21 K23 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 1 ~ 16 KHSDEYKIRRERNNIAARKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 6mg3 B 2.05 BS02 dna D 0 Y274 R278 N281 N282 Y6 R10 N13 N14 ? 0003700,0006351,0006355 remove_due_to_license_issue P17676 30566668 101 ~ 116 KHSDEYKIRRERNNIAARKSRDKAKMRNLETQHKVLELTAENERLQKKVEQLSRELSTLRNLFKQLPE 6mh1 A 1.6 BS01 JQP A 1 W81 F83 V87 L92 L94 Y97 C136 N140 I146 W40 F42 V46 L51 L53 Y56 C95 N99 I105 ? ic50=1.7uM remove_due_to_license_issue Kd=1200nM, IC50=1700nM O60885 30253095 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6mh7 A 1.74 BS01 JQY A 1 W81 P82 F83 L92 Y97 C136 N140 I146 W40 P41 F42 L51 Y56 C95 N99 I105 ? ic50=1.3uM remove_due_to_license_issue IC50=1300nM, Kd=1800nM O60885 30253095 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6mhb A 2.75 BS01 JR7 A 1 C32 P33 R183 W222 F225 L226 C27 P28 R175 W214 F217 L218 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue P78417 30735370 601 ARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 6mhc A 2.0 BS01 JRM A 1 C32 L56 G128 R132 Y229 C35 L59 G131 R135 Y232 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue P78417 30735370 301 SNAMSGESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 6mhd A 2.16 BS01 JRD A 1 C32 L56 G128 I131 Y229 C35 L59 G131 I134 Y232 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue P78417 30735370 401 SNAMSGESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 6mhm B 2.743 BS01 JRY B 1 C143 M161 F163 E225 C1 M19 F21 E83 3.5.1.-,3.5.1.109,3.5.1.23 remove_due_to_license_issue Q13510 30525581 407 CTSIVAEDKKGHLIHGRNMDFGVFLGWNINNDTWVITEQLKPLTVNLDFQRNNKTVFKASSFAGYVGMLTGFKPGLFSLTLNERFSINGGYLGILEWILGKKDAMWIGFLTRTVLENSTSYEEAKNLLTKTKILAPAYFILGGNQSGEGCVITRDRKESLDVYELDAKQGRWYVVQTNYDRWKHPFFLDDRRTPAKMCLNRTSQENISFETMYDVLSTKPVLNKLTVYTTLIDVTKGQFETYLRDCPDPCIGW 6mht A 2.05 BS01 dna C 0 I86 S126 G236 Q237 E239 G257 S296 I86 S126 G236 Q237 E239 G257 S296 C81 E119 R163 R165 C81 E119 R163 R165 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 9207024 402 ~ 413 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNFASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAITLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 6mht A 2.05 BS02 dna D 0 F79 C81 S85 S87 K89 R97 E119 V121 R165 R228 Q237 R240 Y242 T250 A253 Y254 G303 N304 F79 C81 S85 S87 K89 R97 E119 V121 R165 R228 Q237 R240 Y242 T250 A253 Y254 G303 N304 C81 E119 R163 R165 C81 E119 R163 R165 2.1.1.37 0003677,0003886,0008168,0009307,0032259,0051719,0051720 remove_due_to_license_issue P05102 9207024 422 ~ 433 MIEIKDKQLTGLRFIDLFAGLGGFRLALESCGAECVYSNEWDKYAQEVYEMNFGEKPEGDITQVNEKTIPDHDILCAGFPCQAFSISGKQKGFEDSRGTLFFDIARIVREKKPKVVFMENVKNFASHDNGNTLEVVKNTMNELDYSFHAKVLNALDYGIPQKRERIYMICFRNDLNIQNFQFPKPFELNTFVKDLLLPDSEVEHLVIDRKDLVMTNQEIEQTTPKTVRLGIVGKGGQGERIYSTRGIAITLSAYGGGIFAKTGGYLVNGKTRKLHPRECARVMGYPDSYKVHPSTSQAYKQFGNSVVINVLQYIAYNIGSSLNFKPY 6mi6 A 2.95 BS01 JSJ A 1 A410 G414 I454 S492 M507 A58 G62 I102 S140 M151 N409 N57 2.7.13.3 0016310,0016772 remove_due_to_license_issue Q56310 30686862 602 IRMVPISFVFNRFPRMVRDLAKKMNKEVNFIMRGEDTELDRTFVEEIGEPLLHLLRNAIDHGIEPKEERIAKGKPPIGTLILSARHEGNNVVIEVEDDGRGIDKEKIIRKAIEKGLIDESKAATLSDQEILNFLFVPGFSVSEVSGRGVGMDVVKNVVESLNGSISIESEKDKGTKVTIRLPL 6miv A 2.05 BS02 JU1 A 1 F70 Y73 S76 D80 D153 G155 T156 F171 F64 Y67 S70 D74 D147 G149 T150 F165 ? remove_due_to_license_issue P11609 30556652 307 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6miv C 2.05 BS01 JU1 A 1 P29 N31 R95 P28 N30 R94 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 307 TQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKFACANAFNNSIIPEDTFFPS 6miy A 2.75 BS02 JTV A 1 F10 Q14 F70 Y73 S76 D80 A102 F120 W133 L150 D153 G155 T156 L163 F171 F5 Q9 F65 Y68 S71 D75 A97 F115 W128 L145 D148 G150 T151 L158 F166 ? remove_due_to_license_issue P11609 30556652 308 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6miy C 2.75 BS01 JTV A 1 P29 N31 R95 P28 N30 R94 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 308 TQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNFACANAFNNSIIPEDTFFPS 6mj4 A 2.0 BS02 JTG A 1 F70 Y73 S76 D80 A102 D153 G155 T156 F171 F64 Y67 S70 D74 A96 D147 G149 T150 F165 ? remove_due_to_license_issue P11609 30556652 309 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6mj4 C 2.0 BS01 JTG A 1 P29 N31 R95 P29 N31 R95 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 309 KTQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNFACANAFNNSIIPEDTFFPS 6mj7 A 1.412 BS03 ARG A 1 V126 I127 D129 N132 D147 D149 V9 I10 D12 N15 D30 D32 ? 0008270 remove_due_to_license_issue Q13501 30349045 204 GSNMVHPNVICDGCNGPVVGTRYKCSVCPDYDLCSVCEGKGLHRGHTKLAFPSP 6mja A 2.35 BS02 JTJ A 1 F10 C12 V30 F70 Y73 S76 D80 L100 W133 D153 G155 T156 F171 F5 C7 V25 F65 Y68 S71 D75 L95 W128 D148 G150 T151 F166 ? remove_due_to_license_issue P11609 30556652 308 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6mja C 2.35 BS01 JTJ A 1 P29 N31 R95 P28 N30 R94 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 308 TQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNFACANAFNNSIIPEDTFFPS 6mjf A 2.198 BS01 SAH A 1 Y97 G98 H99 V102 F103 S128 A129 F170 Q171 Y210 I211 A212 G241 V242 S243 T244 Y90 G91 H92 V95 F96 S121 A122 F163 Q164 Y203 I204 A205 G234 V235 S236 T237 2.1.1.- 0008168,0032259 Kd=6.88uM remove_due_to_license_issue A0A4S8L4Q5 30204409 500 PGSLIVVGTGIESIGQMTLQALSYIEAASKVFYCVIDPATEAFILTKNKNCVDLYQYYDNGKSRMDTYTQMAELMLKEVRNGLDVVGVFYGHPGVFVNPSHRALAIARSEGYQARMLPGVSAEDCLFADLCIDPSNPGCLTYEASDFLIRERPVNVHSHLILFQVGCVGIADFNFSGFDNSKFTILVDRLEQEYGPDHTVVHYIAAMMPHQDPVTDKFTIGQLREPEIAKRVGGVSTFYIPPKARKDINTDIIRLLEFLPAGKVPDKHTQIYPPNQWEPDVPTLPPYGQNEQAAITRLEAHAPPEEYQPLATSKAMTDVMTKLALDPKALAEYKADHRAFAQSVPDLTPQERAALELGDSWAIRCAMKNMP 6mjf B 2.198 BS01 SAH B 1 Y97 G98 H99 V102 F103 S128 A129 F170 Q171 Y210 I211 A212 G241 V242 S243 T244 Y89 G90 H91 V94 F95 S120 A121 F162 Q163 Y202 I203 A204 G233 V234 S235 T236 2.1.1.- 0008168,0032259 Kd=6.88uM remove_due_to_license_issue A0A4S8L4Q5 30204409 500 GSLIVVGTGIESIGQMTLQALSYIEAASKVFYCVIDPATEAFILTKNKNCVDLYQYYDNGKSRMDTYTQMAELMLKEVRNGLDVVGVFYGHPGVFVNPSHRALAIARSEGYQARMLPGVSAEDCLFADLCIDPSNPGCLTYEASDFLIRERPVNVHSHLILFQVGCVGIADFNFSGFDNSKFTILVDRLEQEYGPDHTVVHYIAAMMPHQDPVTDKFTIGQLREPEIAKRVGGVSTFYIPPKARKDINTDIIRLLEFLPAGKVPDKHTQIYPPNQWEPDVPTLPPYGQNEQAAITRLEAHAPPEEYQPLATSKAMTDVMTKLALDPKALAEYKADHRAFAQSVPDLTPQERAALELGDSWAIRCAMKNMP 6mji A 2.3 BS02 JTD A 1 C12 S28 V30 W63 F70 Y73 S76 D80 F120 W133 D153 G155 T156 F171 C7 S23 V25 W58 F65 Y68 S71 D75 F115 W128 D148 G150 T151 F166 ? remove_due_to_license_issue P11609 30556652 310 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6mji C 2.3 BS01 JTD A 1 P29 R95 P29 R95 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 310 KTQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNKDFACANAFNNSIIPEDTFFPS 6mjj A 1.93 BS02 JU4 A 1 F10 F70 Y73 S76 D80 W133 D153 G155 T156 C168 F171 F4 F64 Y67 S70 D74 W127 D147 G149 T150 C162 F165 ? remove_due_to_license_issue P11609 30556652 308 NYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6mjj C 1.93 BS01 JU4 A 1 P29 N31 R95 P29 N31 R95 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 308 KTQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNFACANAFNNSIIPEDTFFPS 6mjq A 3.0 BS02 JUD A 1 Q14 F70 Y73 S76 D80 A102 D153 G155 T156 V160 F171 Q9 F65 Y68 S71 D75 A97 D148 G150 T151 V155 F166 ? remove_due_to_license_issue P11609 30556652 308 KNYTFRCLQMSSFANRSWSRTDSVVWLGDLQTHRWSNDSATISFTKPWSQGKLSNQQWEKLQHMFQVYRVSFTRDIQELVKMMSPKEDYPIEIQLSAGCEMYPGNASESFLHVAFQGKYVVRFWGTSWQTVPGAPSWLDLPIKVLNADQGTSATVQMLLNDTCPLFVRGLLEAGKSDLEKQEKPVAWLSSVPSSAHGHRQLVCHVSGFYPKPVWVMWMRGDQEQQGTHRGDFLPNADETWYLQATLDVEAGEEAGLACRVKHSSLGGQDIILYW 6mjq C 3.0 BS01 JUD A 1 P29 N31 R95 P29 N31 R95 ? 0002376,0003674,0005575,0005886,0008150,0042101 remove_due_to_license_issue A0A0B4J1J9,K7N5M3 30556652 308 KTQVEQSPQSLVVRQGENCVLQCNYSVTPDNHLRWFKQDTGKGLVSLTVLVDQKDKTSNGRYSATLDKDAKHSTLHITATLLDDTATYICVVGDRGSALGRLHFGAGTQLIVIPDIQNPDPAVYQLRDSKSSDKSVCLFTDFDSQTNVSQSKDSDVYITDKCVLDMRSMDFKSNSAVAWSNFACANAFNNSIIPEDTFFPS 6mju A 2.45 BS01 JUM A 1 R376 S434 Y436 L490 R186 S244 Y246 L300 2.7.7.86 ic50=0.0275uM remove_due_to_license_issue Q8N884 31113940 601 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKNPLSQFLEGEILSASKMLSKFRKIIKEEGSPAVTLISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDEEHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 6mjw A 2.405 BS02 JUJ A 1 Y248 R376 L377 Y436 N482 F488 L495 Y87 R184 L185 Y244 N290 F296 L303 2.7.7.86 ic50=0.0102uM remove_due_to_license_issue Q8N884 31113940 602 ASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKNPLSQFLEGEILSASKMLSKFRKIIKEEGSPAVTLLISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDEEHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFD 6mkq A 1.9 BS01 NXL A 1 C42 S43 S103 T190 T209 G210 T211 C39 S40 S100 T187 T206 G207 T208 S43 K46 S103 E140 K208 T211 S40 K43 S100 E137 K205 T208 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue A0A0U3IB62 30782990 301 NKNMADIEAAFEGRVGVYAINTGSGKAYSYRANERFPLCSSFKAFLAAAVLKMDQDSPGVLLEKVNYHNRTMEPHSPITEKFQSQGMAVGELAAATLQYSDNGAANLLMEKYIKGPEGMTQFMNSIGDTKFRLDRWELDLNSAIPGDERDTSTPKAVAESLNKLISNTVLDNYHQEIFKKWMIGNTTGDNRIRAAVPDGWVVGDKTGTCGKYGTANDHAFILQGNNAAPLILSIYTTRKGEHMKHDDEVIAKAARIAIENVK 6mku E 1.727 BS01 ARG E 1 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=70nM remove_due_to_license_issue P02911 31348608 301 ALPQTVRIGTATTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mkw A 2.32 BS01 HIS A 1 Y14 F52 S70 L71 S72 R77 L117 S120 T121 D161 Y13 F51 S69 L70 S71 R76 L116 S119 T120 D160 ? 0006865,0030288,0042597,0071705 Kd=17uM remove_due_to_license_issue P02911 31348608 301 LPQTVRIGTATTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6ml9 E 1.687 BS01 ARG E 1 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 D10 Y13 F51 S68 S69 S71 R76 L116 S119 T120 Q121 D160 ? 0006865,0030288,0042597,0071705 Kd=5uM remove_due_to_license_issue P02911 31348608 301 LPQTVRIGTDTTYAPFSSKDAKGEFIGFAIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mla E 1.582 BS01 ARG E 1 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 ? 0006865,0030288,0042597,0071705 Kd=42uM remove_due_to_license_issue P02911 31348608 301 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQAEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mle E 1.858 BS01 ARG E 1 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 D11 Y14 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=1nM remove_due_to_license_issue P02911 31348608 303 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mlf A 1.75 BS01 JV4 A 1 R280 G302 E320 H324 R414 S416 T418 R423 R280 G302 E320 H324 R414 S416 T418 R423 R12 S97 H98 K107 D237 D239 D241 R242 H324 R12 S97 H98 K107 D237 D239 D241 R242 H324 0000287,0005975,0016868 Ki=53uM remove_due_to_license_issue 31264865 501 MTLPAFKAYDIRGRVPDELNEDLARRIGVALAAQLDQGPVVLGHDVRLASPALQEALSAGLRASGRDVIDIGLCGTEEVYFQTDYLKAAGGVMVTASHNPMDYNGMKLVREQARPISSDTGLFAIRDTVAADTAAPGEPTASEQSRTDKTAYLEHLLSYVDRSTLKPLKLVVNAGNGGAGLIVDLLAPHLPFEFVRVFHEPDGNFPNGIPNPLLPENRDATAKAVKDNGADFGIAWDGDFDRCFFFDHTGRFIEGYYLVGLLAQAILAKQPGGKVVHDPRLTWNTVEQVEEAGGIPVLCKSGHAFIKEKMRSENAVYGGEMSAHHYFREFAYADSGMIPWLLIAELVSQSGRSLADLVEARMQKFPCSGEINFKVADAKASVARVMEHYASLSPELDYTDGISADFGQWRFNLRSSNTEPLLRLNVETRGDAALLETRTQEISNLLRG 6mlg E 1.892 BS01 ARG E 1 D11 Y14 F52 S69 S70 L71 S72 L117 S120 T121 Q122 D161 D11 Y14 F52 S69 S70 L71 S72 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=9uM remove_due_to_license_issue P02911 31348608 301 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKAQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mlh A 1.65 BS01 GPM A 1 R280 G302 E320 H324 R414 S416 N417 T418 R423 R280 G302 E320 H324 R414 S416 N417 T418 R423 R12 S97 H98 K107 D237 D239 D241 R242 H324 R12 S97 H98 K107 D237 D239 D241 R242 H324 0000287,0005975,0016868 Ki=213uM remove_due_to_license_issue 31264865 501 MTLPAFKAYDIRGRVPDELNEDLARRIGVALAAQLDQGPVVLGHDVRLASPALQEALSAGLRASGRDVIDIGLCGTEEVYFQTDYLKAAGGVMVTASHNPMDYNGMKLVREQARPISSDTGLFAIRDTVAADTAAPGEPTASEQSRTDKTAYLEHLLSYVDRSTLKPLKLVVNAGNGGAGLIVDLLAPHLPFEFVRVFHEPDGNFPNGIPNPLLPENRDATAKAVKDNGADFGIAWDGDFDRCFFFDHTGRFIEGYYLVGLLAQAILAKQPGGKVVHDPRLTWNTVEQVEEAGGIPVLCKSGHAFIKEKMRSENAVYGGEMSAHHYFREFAYADSGMIPWLLIAELVSQSGRSLADLVEARMQKFPCSGEINFKVADAKASVARVMEHYASLSPELDYTDGISADFGQWRFNLRSSNTEPLLRLNVETRGDAALLETRTQEISNLLRG 6mli E 1.883 BS01 HIS E 1 Y14 F52 S70 S72 L117 S120 T121 Q122 D161 Y14 F52 S70 S72 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=3700uM remove_due_to_license_issue P02911 31348608 301 ALPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKAQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mlj A 1.6 BS01 ARG A 1 D11 Y14 F52 S69 A70 S72 R77 S120 T121 D161 D10 Y13 F51 S68 A69 S71 R76 S119 T120 D160 ? 0006865,0030288,0042597,0071705 Kd=55nM remove_due_to_license_issue P02911 31348608 301 LPQTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISALSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mll A 1.86 BS01 N1G A 1 S70 P104 S130 L167 N170 T235 G236 T237 C238 S48 P82 S108 L145 N148 T213 G214 T215 C216 S70 K73 S130 E166 K234 T237 S48 K51 S108 E144 K212 T215 3.5.2.6 0008800,0016787,0017001,0030655,0046677 Ki=239uM remove_due_to_license_issue Q9F663 30942078 301 SHMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLG 6mln E 1.721 BS01 ARG E 1 D11 Y14 F52 S69 S70 A72 R77 L117 S120 T121 Q122 D161 D8 Y11 F49 S66 S67 A69 R74 L114 S117 T118 Q119 D158 ? 0006865,0030288,0042597,0071705 Kd=29nM remove_due_to_license_issue P02911 31348608 301 QTVRIGTDTTYAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLAITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mlo E 1.717 BS01 ARG E 1 D11 A14 F52 S69 S70 L71 S72 R77 L117 S120 T121 Q122 D161 D11 A14 F52 S69 S70 L71 S72 R77 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=0.8uM remove_due_to_license_issue P02911 31348608 302 ALPQTVRIGTDTTAAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mlp E 1.485 BS01 HIS E 1 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 F52 S69 S70 S72 R77 L117 S120 T121 Q122 D161 ? 0006865,0030288,0042597,0071705 Kd=200uM remove_due_to_license_issue P02911 31348608 301 ALPQTVRIGTDTTAAPFSSKDAKGEFIGFDIDLGNEMCKRMQVKCTWVASDFDALIPSLKAKKIDAIISSLSITDKRQQEIAFSDKLYAADSRLIAAKGSPIQPTLESLKGKHVGVLQGSTQEAYANDNWRTKGVDVVAYANQDLIYSDLTAGRLDAALQDEVAASEGFLKQPAGKEYAFAGPSVKDKKYFGDGTGVGLRKDDTELKAAFDKALTELRQDGTYDKMAKKYFDFNVYGD 6mlw A 1.9 BS02 JVA A 1 G302 H303 E320 S322 H324 R414 S416 N417 T418 R423 G303 H304 E321 S323 H325 R415 S417 N418 T419 R424 R12 S97 H98 K107 D237 D239 D241 R242 H324 R13 S98 H99 K108 D238 D240 D242 R243 H325 0000287,0005975,0016868 Ki=184uM remove_due_to_license_issue 31264865 502 HMTLPAFKAYDIRGRVPDELNEDLARRIGVALAAQLDQGPVVLGHDVRLASPALQEALSAGLRASGRDVIDIGLCGTEEVYFQTDYLKAAGGVMVTASHNPMDYNGMKLVREQARPISSDTGLFAIRDTVAADTAAPGEPTASEQSRTDKTAYLEHLLSYVDRSTLKPLKLVVNAGNGGAGLIVDLLAPHLPFEFVRVFHEPDGNFPNGIPNPLLPENRDATAKAVKDNGADFGIAWDGDFDRCFFFDHTGRFIEGYYLVGLLAQAILAKQPGGKVVHDPRLTWNTVEQVEEAGGIPVLCKSGHAFIKEKMRSENAVYGGEMSAHHYFREFAYADSGMIPWLLIAELVSQSGRSLADLVEARMQKFPCSGEINFKVADAKASVARVMEHYASLSPELDYTDGISADFGQWRFNLRSSNTEPLLRLNVETRGDAALLETRTQEISNLLRG 6mm2 A 1.04 BS01 ATP A 1 G39 E40 G41 S42 R43 N44 V45 R46 E50 Y57 N59 S88 C89 I90 G39 E40 G41 S42 R43 N44 V45 R46 E50 Y57 N59 S88 C89 I90 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SSQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSRNVRSTGEPSVSHAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEAL 6mmc A 1.42 BS01 ADP A 1 G39 E40 G41 S42 Y57 N59 S88 C89 I90 G37 E38 G39 S40 Y42 N44 S73 C74 I75 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 203 QQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6mmo A 1.86 BS03 AMP B 1 G30 Y31 T32 L64 G31 Y32 T33 L52 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SSQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6mmo A 1.86 BS04 AMP D 1 G38 E39 G40 S41 N58 S87 I89 G39 E40 G41 S42 N46 S75 I77 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SSQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6mmo B 1.86 BS02 AMP B 1 G38 E39 G40 S41 N58 S87 I89 G38 E39 G40 S41 N45 S74 I76 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEA 6mmo B 1.86 BS04 AMP D 2 G30 Y31 T32 L64 G30 Y31 T32 L51 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 202 SQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEA 6mmq A 2.02 BS01 CMP A 1 G31 Y32 T33 L65 G29 Y30 T31 L49 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 QQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEA 6mmq A 2.02 BS02 CMP B 1 G39 E40 N59 S88 I90 G37 E38 N43 S72 I74 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 QQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEA 6mmq D 2.02 BS01 CMP A 1 G39 E40 N59 S88 I90 G38 E39 N44 S73 I75 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEAL 6mmq D 2.02 BS02 CMP D 1 G31 Y32 T33 L65 G30 Y31 T32 L50 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEAL 6mnc B 2.4 BS01 J3Z B 1 V143 P187 H221 F259 E282 V143 P187 H213 F251 E274 1.1.1.51,1.1.1.62 0003824,0004303,0005496,0005515,0005737,0005829,0006629,0006694,0006703,0007040,0007519,0008210,0010467,0016491,0030283,0036094,0042803,0047035,0047045,0050661,0060348,0060612,0061370,0070401,0071248,0072582,1903924 remove_due_to_license_issue IC50=810nM, Ki=3nM P14061 30768851 401 ARTVVLITGCSSGIGLHLAVRLASDPSQSFKVYATLRDLKTQGRLWEAARALACPPGSLETLQLDVRDSKSVAAARERVTEGRVDVLVCNAGLGLLGPLEALGEDAVASVLDVNVVGTVRMLQAFLPDMKRRGSGRVLVTGSVGGLMGLPFNDVYCASKFALEGLCESLAVLLLPFGVHLSLIECGPVHTSPEEVLDRTDIHTFHRFYQYLAHSKQVFREAAQNPEEVAEVFLTALRAPKPTLRYFTTERFLPLLRMRLDDPSGSNYVTAMHREVF 6mnf M 2.758 BS01 MAN A 1 A31 S100A D100B A31 S105 D106 remove_due_to_license_issue 16174734 3 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6mnf M 2.758 BS02 MAN A 2 A31 H32 T33 K95 G96 S100A D100B N100C D100D A31 H32 T33 K99 G100 S105 D106 N107 D108 remove_due_to_license_issue 16174734 4 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6mnv A 1.65 BS01 JVS A 1 R280 G302 E320 S322 H324 R414 S416 N417 T418 R423 R280 G302 E320 S322 H324 R414 S416 N417 T418 R423 0000287,0005975,0016868 Ki=428uM remove_due_to_license_issue 31264865 501 MTLPAFKAYDIRGRVPDELNEDLARRIGVALAAQLDQGPVVLGHDVRLASPALQEALSAGLRASGRDVIDIGLCGTEEVYFQTDYLKAAGGVMVTASHNPMDYNGMKLVREQARPISSDTGLFAIRDTVAADTAAPGEPTASEQSRTDKTAYLEHLLSYVDRSTLKPLKLVVNAGNGGAGLIVDLLAPHLPFEFVRVFHEPDGNFPNGIPNPLLPENRDATAKAVKDNGADFGIAWDGDFDRCFFFDHTGRFIEGYYLVGLLAQAILAKQPGGKVVHDPRLTWNTVEQVEEAGGIPVLCKSGHAFIKEKMRSENAVYGGEMSAHHYFREFAYADSGMIPWLLIAELVSQSGRSLADLVEARMQKFPCSGEINFKVADAKASVARVMEHYASLSPELDYTDGISADFGQWRFNLRSSNTEPLLRLNVETRGDAALLETRTQEISNLLRG 6mny A 2.8 BS01 JVP A 1 L408 T410 V416 A428 K430 M449 I472 T474 M477 C481 L528 S538 D539 F540 L542 L14 T16 V22 A34 K36 M55 I78 T80 M83 C87 L134 S144 D145 F146 L148 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue P35991 30655951 701 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIREGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSEAAEHIAQGLRLYRPHLASERVYTIMYSCWHEKADERPSFKILLSNILDVMD 6mo0 A 2.7 BS01 JVJ A 1 K1074 D1075 L1076 G1148 L1149 G1151 I1165 K81 D82 L83 G155 L156 G158 I159 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue A0A0B4L2Y4,Q91H74 31017399 1201 MADLELERAADVRWEEQAEISGSSLEDGAYRIKQKGILGYSQIGAGVYKEGTFHTMWHVTRGAVLMHKGKRIEPSWADVKKDLISYGGGWKLEGEWKEGEEVQVLALEPGKNPRAVQTKPGLFKTNTGTIGAVSLDFSPGTSGSPIVDKKGKVVGLYGIANTEK 6mo1 A 3.0 BS01 I16 A 1 K1073 K1074 D1075 G1148 L1149 G1151 I1165 K80 K81 D82 G155 L156 G158 I159 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue B3RFT3,Q91H74 31017399 1201 MADLELERAADVRWEEQAEISGSSLEDGAYRIKQKGILGYSQIGAGVYKEGTFHTMWHVTRGAVLMHKGKRIEPSWADVKKDLISYGGGWKLEGEWKEGEEVQVLALEPGKNPRAVQTKPGLFKTNTGTIGAVSLDFSPGTSGSPIVDKKGKVVGLYGIANTEK 6mo2 A 2.8 BS01 JVM A 1 K1073 K1074 D1075 L1076 L1149 G1151 I1165 K80 K81 D82 L83 L156 G158 I159 3.4.21.91,3.6.1.15,3.6.4.13 0003723,0003724,0004252,0005524,0044423 remove_due_to_license_issue A0A0B4L2Y4,Q91H74 31017399 1201 MADLELERAADVRWEEQAEISGSSLEDGAYRIKQKGILGYSQIGAGVYKEGTFHTMWHVTRGAVLMHKGKRIEPSWADVKKDLISYGGGWKLEGEWKEGEEVQVLALEPGKNPRAVQTKPGLFKTNTGTIGAVSLDFSPGTSGSPIVDKKGKVVGLYGIANTEK 6mo4 A 1.844 BS02 JWM A 1 H19 M62 E77 T190 F191 I197 G209 V216 H237 D241 H264 H23 M66 E81 T190 F191 I197 G209 V216 H237 D241 H264 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=4.6nM remove_due_to_license_issue P47205 31283109 302 HHHATIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRTQQASVDFTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 6mo5 A 1.851 BS01 JWP A 1 L18 H19 M62 E77 H78 T190 F191 G192 F193 I197 G209 S210 H237 D241 H264 L23 H24 M67 E82 H83 T194 F195 G196 F197 I201 G213 S214 H241 D245 H268 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=0.3nM remove_due_to_license_issue P47205 31283109 301 HHHHATIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFVRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 6mo7 A 1.85 BS01 JWA A 1 W97 P98 F99 V103 L108 N156 I162 W24 P25 F26 V30 L35 N83 I89 ? remove_due_to_license_issue P25440 30606676 201 RVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQEL 6mo8 A 1.8 BS01 JWD A 1 W97 F99 L108 N156 I162 W24 F26 L35 N83 I89 ? remove_due_to_license_issue P25440 30606676 201 RVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQEL 6mo8 A 1.8 BS02 JWD A 2 N77 Q80 L187 N4 Q7 L114 ? remove_due_to_license_issue P25440 30606676 202 RVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQEL 6mo9 A 1.801 BS01 JVY A 2 W97 F99 L108 N156 I162 M165 W24 F26 L35 N83 I89 M92 ? remove_due_to_license_issue P25440 30606676 202 RVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQEL 6moa A 1.271 BS01 JW4 A 1 W370 P371 F372 N429 H433 V435 W25 P26 F27 N84 H88 V90 ? Kd=2.5nM remove_due_to_license_issue P25440 30606676 501 LSEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMDLSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDVFEFRYAKMP 6mob A 1.8 BS01 JWY A 1 V603 A621 K623 E640 L644 T670 C673 L783 L799 I808 C809 D810 F811 V37 A55 K57 E74 L78 T104 C107 L159 L175 I184 C185 D186 F187 D792 R796 N797 D810 D168 R172 N173 D186 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 remove_due_to_license_issue P10721 31085175 1015 NYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFICSKTSPAIMEDDELALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISE 6mod A 1.85 BS02 JWV A 1 M62 E77 T190 F191 M194 I197 G209 V216 H237 K238 D241 H264 M63 E78 T189 F190 M193 I196 G208 V215 H236 K237 D240 H263 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=0.71nM remove_due_to_license_issue P47205 31283109 302 ATIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFVRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 6mom A 2.1 BS01 JX4 A 1 M192 G195 V200 A211 Y262 Y264 M265 A315 N316 L318 D329 M29 G32 V37 A48 Y94 Y96 M97 A147 N148 L150 D161 D311 K313 A315 N316 D329 T351 D143 K145 A147 N148 D161 T180 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=0.8nM remove_due_to_license_issue Q9NWZ3 31484791 500 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTAS 6moo A 2.2 BS02 A5F A 1 E77 T190 F191 I197 G209 S210 H237 D241 H264 E83 T192 F193 I199 G211 S212 H239 D243 H266 3.5.1.108 0006796,0009245,0016020,0016787,0019637,0046872,0103117,1901135 ic50=19nM remove_due_to_license_issue P47205 31283109 302 HHEGAGTIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFSRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFIRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP 6mq3 A 3.56915 BS01 J22 A 1 F202 E205 Y302 T316 K364 I374 N376 R477 A479 F160 E163 Y260 T274 K322 I332 N334 R435 A437 3.4.24.56 0001618,0004175,0004222,0005515,0005524,0005576,0005615,0005634,0005737,0005739,0005777,0005782,0005829,0005886,0006508,0008237,0008270,0008286,0009897,0009986,0010815,0010992,0016323,0019885,0030163,0032092,0042277,0042447,0042803,0043171,0043559,0045732,0046718,0046872,0050435,0051603,0070062,0097242,0150094,1901142,1901143,1903715 remove_due_to_license_issue P14735 31086331 1101 NNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFLQHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLSPLFDESAKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVVVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQELKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKANLNFEFFSPFAYVDPLHSNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNSGIEIYYQTDMQSTSENMFLELFAQIISEPAFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAESAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSNPINLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPH 6mr5 A 1.85 BS02 W45 A 1 P464 S531 H573 H574 F583 D612 H614 F643 G743 Y745 P23 S90 H132 H133 F142 D171 H173 F202 G302 Y304 ? remove_due_to_license_issue F8W4B7 30613344 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDTPLKTSATVSINNVLRAHAPFWSSLR 6mr5 A 1.85 BS03 W45 B 1 D460 H462 D19 H21 ? remove_due_to_license_issue F8W4B7 30613344 804 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDTPLKTSATVSINNVLRAHAPFWSSLR 6mrg A 2.77 BS01 JXV A 1 S193 Y194 G239 L404 I407 F432 T488 M495 W531 S162 Y163 G208 L373 I376 F401 T457 M464 W500 L79 P188 V458 P484 G489 A490 L48 P157 V427 P453 G458 A459 3.1.1.-,3.5.1.99 0000139,0004040,0005515,0005543,0005783,0005789,0005794,0006631,0008289,0009062,0016020,0016042,0016787,0016788,0017064,0031090,0042802,0045907,0047372,0052651,0098793,0098794,0098978,0150036 remove_due_to_license_issue P97612 30289722 601 TGRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMTP 6msa A 2.06 BS02 JY4 A 1 L635 L675 I692 Q726 F729 L189 L229 I246 Q280 F283 3.1.4.17 0004114,0007165,0008081 ic50=5nM remove_due_to_license_issue Q9Y233 30587449 803 HMSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGEETATW 6msc A 2.36 BS02 JY7 A 1 L675 F696 M713 Q726 F729 L228 F249 M266 Q279 F282 3.1.4.17 0004114,0007165,0008081 ic50=21nM remove_due_to_license_issue IC50=21nM Q9Y233 30587449 803 MSICTSEEWQGLMQFTLPVRLCKEIELFHFDIGPFENMWPGIFVYMVHRSCGTSCFELEKLCRFIMSVKKNYRRVPYHNWKHAVTVAHCMYAILQNNHTLFTDLERKGLLIACLCHDLDHRGFSNSYLQKFDHPLAALYSTSTMEQHHFSQTVSILQLEGHNIFSTLSSSEYEQVLEIIRKAIIATDLALYFGNRKQLEEMYQTGSLNLNNQSHRDRVIGLMMTACDLCSVTKLWPVTKLTANDIYAEFWAEGDEMKKLGIQPIPMMDRDKKDEVPQGQLGFYNAVAIPCYTTLTQILPPTEPLLKACRDNLSQWEKVIRGE 6msn A 1.591 BS02 JYD A 1 Q134 D135 R173 G216 R421 T467 T468 R471 Q107 D108 R146 G189 R385 T431 T432 R435 4.2.1.2 0004333,0005737,0005829,0006091,0006106,0006108,0016829,0016836,0020015,0042803,0046872,0051539,0097014 Ki=8.9uM remove_due_to_license_issue E9AE57 30645090 602 DFHFSAIFQPTDPHHHQTEFAKVEGSEKYVEEVEVFGRQALKVNPEALTILAHRAFSDVHHFFRKDHLEGWRRAIEDPEASDNDRYVATTLLKNACIAAGRVLPSCQDTGTAIVLGKRGELCWTGGEDEKYLSKGIWNAYRYHNLRYSQTAALDMFKECNTGDNLPAQLDLLAVPGSDYEFLFIAKGGGSANKAYLYQETKALLNPKSLRAFIEEKLKTLGTAACPPYHIALVIGGTSAEMTMKTVKLASCRYYDSLPTTGDKYGRAFRDPEWEKIVMEVAQKSGIGAQFGGKYFAHQARVIRLPRHGASCPVGLAVSCSADRQILAHINKSGIYIEQLEQNPAQYLPTSVKVDLKRPIDKVRQQLSQYPVGTRVMLNGTLIVARDIAHAKIKEMMDNGEPLPEYMKTSPIYYAGPAKTPEGYASGSFGPTTAGRMDSYVDLFQSHGGSYITLAKGNRSKQVTDACKKHGGFYLGSIGGPAAILAKDSIKQVTCLAFPELGMEAVWKIEVEDFPAFIVVDDKGNDMYSKTLA 6msn B 1.591 BS02 JYD B 1 Q134 D135 R173 G216 R421 T467 T468 R471 Q107 D108 R146 G189 R384 T430 T431 R434 4.2.1.2 0004333,0005737,0005829,0006091,0006106,0006108,0016829,0016836,0020015,0042803,0046872,0051539,0097014 Ki=8.9uM remove_due_to_license_issue E9AE57 30645090 602 DFHFSAIFQPTDPHHHQTEFAKVEGSEKYVEEVEVFGRQALKVNPEALTILAHRAFSDVHHFFRKDHLEGWRRAIEDPEASDNDRYVATTLLKNACIAAGRVLPSCQDTGTAIVLGKRGELCWTGGEDEKYLSKGIWNAYRYHNLRYSQTAALDMFKECNTGDNLPAQLDLLAVPGSDYEFLFIAKGGGSANKAYLYQETKALLNPKSLRAFIEEKLKTLGTAACPPYHIALVIGGTSAEMTMKTVKLASCRYYDSLPTTGDKYGRAFRDPEWEKIVMEVAQKSGIGAQFGGKYFAHQARVIRLPRHGASCPVGLAVSCSADRQILAHINKSGIYIEQLEQNPAQYLPSVKVDLKRPIDKVRQQLSQYPVGTRVMLNGTLIVARDIAHAKIKEMMDNGEPLPEYMKTSPIYYAGPAKTPEGYASGSFGPTTAGRMDSYVDLFQSHGGSYITLAKGNRSKQVTDACKKHGGFYLGSIGGPAAILAKDSIKQVTCLAFPELGMEAVWKIEVEDFPAFIVVDDKGNDMYSKTLA 6mso A 2.053 BS02 JYD A 1 Q115 D116 R154 G197 R404 T451 K474 Q106 D107 R145 G188 R395 T442 K465 4.2.1.2 0003824,0004333,0005737,0005739,0006091,0006099,0006106,0006108,0016829,0016836,0042803,0046872,0051539 Ki=3uM remove_due_to_license_issue Q4QAU9 30645090 608 AEFNFVPLVSKVSHKETKYRLLTKDYVSVVQPGAGLPEMLRVDPAALTLLSSTAFDDVEHLLRSSHLMSLRKIFDDPEASDNDKFVALQLLKNANISSARLLPGCQDTGTAIIAGYRGDQVFVPGNDEEALSRGVYDIFQKRNFRYSQNVPLSMYDEKNTGTNLPAQIDLYASKGMEYSFMFVAKGGGSANKSFLLQETKSVLNPKSLRNFLKEKLAMFGTSACPPYHVAVVIGGTSAEMTMKVLKYASCHYYDDLITKPDMKTGYTFRDLELEEEVLKVCQNIGMGAQFGGKYYAHDVRVIRMPRHGASCPIGIGVSCSADRQALGKINKDGVWLEELEMEPSQYLPDLKEDELLKTPAVMVNLNRPMPEVLQELSKHPVRTRLSLTGTIIVARDSAHARMREMLEAGKPLPQYMKEHPVYYAGPAKQPDGLPSGSFGPTTAGRMDPFVDLFQSHGGSMVMLAKGNRSKQVTKACHKYGGFYLGSIGGPAAVLAQNAIKKVECLDMKDLGMEAVWRIEVENFPAFIVVDDKGNDFFEQL 6mso B 2.053 BS02 JYD B 1 Q115 D116 R154 G197 R404 T451 R454 K474 Q106 D107 R145 G188 R395 T442 R445 K465 4.2.1.2 0003824,0004333,0005737,0005739,0006091,0006099,0006106,0006108,0016829,0016836,0042803,0046872,0051539 Ki=3uM remove_due_to_license_issue Q4QAU9 30645090 604 AEFNFVPLVSKVSHKETKYRLLTKDYVSVVQPGAGLPEMLRVDPAALTLLSSTAFDDVEHLLRSSHLMSLRKIFDDPEASDNDKFVALQLLKNANISSARLLPGCQDTGTAIIAGYRGDQVFVPGNDEEALSRGVYDIFQKRNFRYSQNVPLSMYDEKNTGTNLPAQIDLYASKGMEYSFMFVAKGGGSANKSFLLQETKSVLNPKSLRNFLKEKLAMFGTSACPPYHVAVVIGGTSAEMTMKVLKYASCHYYDDLITKPDMKTGYTFRDLELEEEVLKVCQNIGMGAQFGGKYYAHDVRVIRMPRHGASCPIGIGVSCSADRQALGKINKDGVWLEELEMEPSQYLPDLKEDELLKTPAVMVNLNRPMPEVLQELSKHPVRTRLSLTGTIIVARDSAHARMREMLEAGKPLPQYMKEHPVYYAGPAKQPDGLPSGSFGPTTAGRMDPFVDLFQSHGGSMVMLAKGNRSKQVTKACHKYGGFYLGSIGGPAAVLAQNAIKKVECLDMKDLGMEAVWRIEVENFPAFIVVDDKGNDFFEQL 6msy H 1.999 BS01 MAN A 1 A31 H32 T33 K95 G96 S100A D100B N100C D100D A31 H32 T33 K99 G100 S105 D106 N107 D108 ? remove_due_to_license_issue P0DOX5 16174734 4 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSQTYICNVNHKPSNTKVDKKVEP 6mt0 A 2.2 BS01 JYG A 1 L44 F49 A65 K67 V126 L174 I185 D186 L12 F17 A33 K35 V94 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 remove_due_to_license_issue IC50=0.050000nM P11309 30624936 401 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 6mu1 A 4.1 BS01 JYP A 1 G268 R269 Q270 A272 T273 S274 A275 R504 Q507 K508 D566 Y567 R568 K569 N570 G265 R266 Q267 A269 T270 S271 A272 R470 Q473 K474 D519 Y520 R521 K522 N523 ? 0000902,0001666,0005216,0005220,0005262,0005509,0005515,0005524,0005635,0005637,0005730,0005737,0005783,0005789,0005886,0005955,0006811,0006816,0006915,0007200,0007204,0007207,0007338,0009791,0010976,0014069,0015278,0016020,0016358,0016529,0019722,0019855,0019903,0019904,0030425,0030658,0030667,0030868,0031088,0031094,0031410,0032024,0032469,0032991,0035091,0036444,0042045,0042802,0043025,0043065,0043066,0044325,0044877,0045202,0046872,0048471,0050849,0050882,0051209,0051289,0051480,0051928,0055085,0070059,0070588,0070679,0071320,0071456,0097060,0097421,0098685,0098695,0098793,0098794,0098982,0099105,0099566,1903514,1990806,2000347 remove_due_to_license_issue P29994 30470765 2801 KMSSFLHIGDICSLYAEGSTNGFISTLGLVDDRCVVQPEAGDLNNPPKKFRDCLFKLCPMNRYSAQKQFWKAAKPGANSTTDAVLLNKLHHAADLEKKQNETENRKLLGTVIQYGNVIQLLHLKSNKYLTVNKRLPALLEKNAMRVTLDEAGNEGSWFYIQPFYKLRSIGDSVVIGDKVVLNPVNAGQPLHASSHQLVDNPGCNEVNSVNCNTSWKIVLFMKWSDNKDDILKGGDVVRLFHAEQEKFLTCDEHRKKQHVFLRTTGRQSATSATSSKALWEVEVVQHDPCRGGAGYWNSLFRFKHLATGHYLAAEVDPDYSLVSVPEGNDISSIFELDPTTLRGGDSLVPRNSYVRLRHLCTNTWVHSTNIPIDKEEEKPVMLKIGTSPLKEDKEAFAIVPVSPAEVRDLDFANDASKVLGSIAGKLEKGTITQNERRSVTKLLEDLVYFVTGGTNSGQDVLEVVFSKPNRERQKLMREQNILKQIFKLLQAPFTDCGDHAPFRHICRLCYRVLRHSQQDYRKNQEYIAKQFGFMQKQITALLHNNRKLLEKHITAAEIDTFVSLVRKNREPRFLDYLSDLCVSMNKSIPVTQELICKAVLNPTNADILIRSKSVRELAQDAKEGQKEDRDVLSYYRYQLNLFARMCLDRQYLAINEISGQLDVDLILRCMSDENLPYDLRASFCRLMLHMHVDRDPQEQVTPVKYARLWSEIPSEIAIDDYDSSGASKDEIKERFAQTMEFVEEYLRDVVCQRFPFSDKEKNKLTFEVVNLARNLIYFGFYNFSDLLRLTKILLAILDCVPEKEDIMVMDTKLKIIEILQFILNVRLDYRISCLLCIFKREFDESNSQSVPGALDFEHIEEQAEGIFGHGGRTFLRVLLHLTMHDYPPLVSGALQLLFRHFSQRQEVLQAFKQVQLSQDVDNYKQIKQDLDQLRSIVEKSESYNYRVVKEILIRLSKLCVQESASVRKSRKQQQRLLRNMGKAEDTKMQEIMRLAHEFLQNFCAGNQQNQALLHKHINLFLNPGILEAVTMQHIFMNNFQLCSEINERVVQHFVHCIETHGRNVQYIKFLQTIVKIKKCQDMVMAELVNSGEDVLVFYNDRASFQTLIQMMRLFMYHIHLVELLAVCTEGKNVYTEIKCNSLLPLDDIVRVVTHEDCIPEVKIAYINFLNHCYVDTEVEMKEIYTSNHMWKLFENFLVDSVLEKYVTEIVMSIVTTFLQTRQPVFVQLLQGVFRVYHCNWLMPSQKASVESCIRRNIIERLQDIVSALEDRLRPLVQAELSVLVDVLHRPELLFPENTDARRKCESGGFICKLIKHTKQLLEENEEKLCIKVLQTLREMMTKDRGYGSRGEMSLAEVQCHLDKEGASNLVIDLIMNASSDRVFHESILLAIALLEGGNTTIQHSFFCRLTEDKKSEKFFKVFYDRMKVAQQEIKATVTVNTDDLEMSAVITIMQPILRFLQLLCENHNRDLQNFLRCQNNKTNYNLVCETLQFLDCICGSTTGGLGLLGLYINEKNVALINQTLESLTEYCQGPCHENQNCIATHESNGIDIITALILNDINPLGKKRMDLVLELKNNASKLLLAIMESRHDSENAERILYNMRPKELVEVIKKAYMQGEVEFEDGENGEDGAASPRNVGHNIYILAHQLARHNKELQTMLKPGGQVDGDEALEFYAKHTAQIEIVRLDRTMEQIVFPVPSICEFLTKESKLRIYYTTERDEQGSKINDFFLRSEDLFNEMNWQKKLRAQPVLYWCARNMSFWSSISFNLAVLMNLLVAFFYPFKGVRGGTLALIASTILRLIFSVGLQPTLFLLGAFNVCNKIIFLMSFVGNCGTFTRGYRAMVLDVEFLYHLLYLLICAMGLFVHEFFYSLLLFDLVYREETLLNVIKSVTRNGRPIILTAALALILVYLFSIVGYLFFKDDFILEETEQDKEHTCETLLMCIVTVLSHGLRSGGGVGDVLRKPSKEEPLFAARVIYDLLFFFMVIIIVLNLIFGVIIDTFADLRSEKQKKEEILKTTCFICGLERDKFDNKTVTFEEHIKEEHNMWHYLCFIVLVKVKDSTEYTGPESYVAEMIRERNLDWFPRMRAMSLVSSDSEGEQNELRNLQEKLESTMKLVTNLSGQLSELKDQMTEQRKQKQRIGLLGHP 6mu3 H 2.327 BS01 MAN A 1 A31 D100B A31 D106 ? remove_due_to_license_issue P0DOX5 16174734 3 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 6mu3 H 2.327 BS02 MAN A 2 A31 H32 T33 K95 G96 S100A D100B N100C D100D A31 H32 T33 K99 G100 S105 D106 N107 D108 ? remove_due_to_license_issue P0DOX5 16174734 4 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 6mub H 2.503 BS01 MAN A 1 A31 D100B A31 D106 ? remove_due_to_license_issue P0DOX5 16174734 4 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKS 6mub H 2.503 BS02 MAN A 2 T33 K95 D100B N100C D100D T33 K99 D106 N107 D108 ? remove_due_to_license_issue P0DOX5 16174734 5 EVQLVESGGGLVKAGGSLILSCGVSNFRISAHTMNWVRRVPGGGLEWVASISTSSTYRDYADAVKGRFTVSRDDLEDFVYLQMHKMRVEDTAIYYCARKGSDRLSDNDPFDAWGPGTVVTVSPASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKS 6mul A 3.09 BS01 K4A A 1 F751 M752 W760 I777 Y813 I825 V828 N836 M900 I910 D911 F555 M556 W564 I581 Y617 I629 V632 N640 M704 I714 D715 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 30986068 9001 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 6mum A 3.06 BS01 K47 A 1 T750 W760 I777 Y813 I825 V828 M900 I910 T557 W567 I584 Y620 I632 V635 M707 I717 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 30986068 9001 VKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNLWSLEQPFSIELIEGRKVNAMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPVYFPALEKILELQLQLREILERELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFKRVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESW 6mv3 A -1.00 BS02 WW7 A 1 F27 L41 M45 M60 E63 V64 M80 S84 R147 I148 M153 F27 L41 M45 M60 E63 V64 M80 S84 R102 I103 M108 ? 0005509,0005861 remove_due_to_license_issue P19429,P63316 30376637 201 MDDIYKAAVEQLTEEQKNEFKAAFDIFVLGAEDGSISTKELGKVMRMLGQNPTPEELQEMIDEVDEDGSGTVDFDEFLVMMVRSMKDDSKGKFKRPTLRRVRISADAMMQALLGARAKGHHHHHH 6mvu A 1.488 BS01 K4V A 1 G221 G224 E225 V228 V243 R246 I247 A250 G207 G210 E211 V214 V229 R232 I233 A236 N165 E261 A295 E464 N151 E247 A281 E450 ? 0000166,0016491,0016620 remove_due_to_license_issue A0A0Q3EUQ3 30529746 801 APESAKEAYAWLAEKGDFGHFIGGAWTAPGDLFATVNPATGQTLAQVSQATQADVDAAVKAARKAQPAWAKDGAARARVLYALARLLQKHARLFAVLETLDNGKPIREARDIDVPLAQRHFYHHAGYAQLMGTEMPDRAPLGVCGQVIPWNFPLLMLAWKIAPALAMGNTVVLKPAEWTPLTALLFADICGQAGVPAGVVNIVTGDGAVGEMIVTAQVDKVAFTGSTAVGRRIREATAGTGKALSLELGGKGPYVVCDDADIDSAVEGLVDAIWFNQGQVACAGSRLLVQEGIADVFHAKLRARMDSLRIGDPLDKCIDIGAMVHPDQLARVRDMVAANTDGEVYQTAVPAGCYYPPTLISGLAPASPLMQQEIFGPVLVSTTFRTPAEAVEIANNTAYGLAASVWSENVNLALDLAPKLVAGIVWINGTNMMDAAAPFGGVRESGFGREGGWEGLAGYTRPAIATKSPAAVAAYTGDGAADGLDRTAKLYIGGKQTRPDGGYSRAVYGPKGKLLGHASLSNRKDLRNAVEAMNAASGWSRTTGHLRAQILYFIGENLSARADEFANRIKDMTGKDGKAEVAASIDRLFSAAAWADKYDGQVKGVPLRGVALAMKEPVGKIGILCPDAAPLLGLVSLMAPAIAMGNRVTLAASEAFPLAATDFYQVLDTSDVPAGVVNILTGAHADLAEPMARHLDLDAVWGLSGHAQVIEAASAGNLKRSWTGPFDPAHDHTRDILSHATEVKTIWVPYGA 6mwe A 2.05 BS01 919 A 1 A853 K855 E872 E903 A905 L971 A981 D982 F983 G984 R987 Q989 A38 K40 E44 E75 A77 L143 A153 D154 F155 G156 R159 Q161 D964 A966 R968 N969 D982 D136 A138 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q02763 28838996 1203 YPVLDWNDIKFQDVIGEGNFGQVLKARIKKDGLRMDAAIKRMGELEVLCKLGHHPNIINLLGACEHRGYLYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLSRGQEVYKTMGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGIDCSAEE 6mwn C 2.838 BS01 rna A 0 E4 T205 E1 T202 remove_due_to_license_issue 31399592 593 ~ 684 EVQLVESGGGLVQPGGSLRLSCAASGFSLSSSSMHWVRQAPGKGLEWVASISPYSGSTSYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARTKYHYKNYYWWALDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6mwn C 2.838 BS02 rna B 0 S33 S55 Y57 S58 Y104 H105 Y106 K107 N108 Y109 Y110 W111 W112 S30 S52 Y54 S55 Y101 H102 Y103 K104 N105 Y106 Y107 W108 W109 remove_due_to_license_issue 31399592 593 ~ 684 EVQLVESGGGLVQPGGSLRLSCAASGFSLSSSSMHWVRQAPGKGLEWVASISPYSGSTSYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARTKYHYKNYYWWALDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6mwn D 2.838 BS01 rna A 0 S57 G58 S61 S56 G57 S60 remove_due_to_license_issue 31399592 593 ~ 684 DIQMTQSPSSLSASVGDRVTITCRASQSVYYSVAWYQQKPGKAPKLLIYSASYLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYRRRPITFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGE 6mwn D 2.838 BS02 rna B 0 Q28 S29 Y31 R67 R93 R95 Q27 S28 Y30 R66 R92 R94 remove_due_to_license_issue 31399592 593 ~ 684 DIQMTQSPSSLSASVGDRVTITCRASQSVYYSVAWYQQKPGKAPKLLIYSASYLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYRRRPITFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGE 6mwn H 2.838 BS01 rna A 0 S33 S55 Y57 S58 Y104 H105 Y106 K107 N108 Y109 Y110 W111 W112 S30 S52 Y54 S55 Y101 H102 Y103 K104 N105 Y106 Y107 W108 W109 remove_due_to_license_issue 31399592 593 ~ 684 EVQLVESGGGLVQPGGSLRLSCAASGFSLSSSSMHWVRQAPGKGLEWVASISPYSGSTSYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARTKYHYKNYYWWALDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6mwn H 2.838 BS02 rna B 0 E4 L173 S175 S201 T205 Q206 E1 L170 S172 S198 T202 Q203 remove_due_to_license_issue 31399592 593 ~ 684 EVQLVESGGGLVQPGGSLRLSCAASGFSLSSSSMHWVRQAPGKGLEWVASISPYSGSTSYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARTKYHYKNYYWWALDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6mwn L 2.838 BS01 rna A 0 Q28 S29 Y31 R67 G69 R93 R94 Q27 S28 Y30 R66 G68 R92 R93 remove_due_to_license_issue 31399592 593 ~ 684 DIQMTQSPSSLSASVGDRVTITCRASQSVYYSVAWYQQKPGKAPKLLIYSASYLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYRRRPITFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGE 6mwn L 2.838 BS02 rna B 0 S57 G58 P60 S61 K170 S56 G57 P59 S60 K169 remove_due_to_license_issue 31399592 593 ~ 684 DIQMTQSPSSLSASVGDRVTITCRASQSVYYSVAWYQQKPGKAPKLLIYSASYLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYRRRPITFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGE 6mx3 A 1.362 BS01 K5P A 1 S162 T263 P264 Q266 T267 S9 T94 P95 Q97 T98 ? 0002218,0032481 remove_due_to_license_issue IC50=7300nM Q86WV6 30655953 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLDPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPSFSLSQEVLRHLRQE 6mx3 A 1.362 BS02 K5P B 1 S162 Y163 G166 Y167 S9 Y10 G13 Y14 ? 0002218,0032481 remove_due_to_license_issue IC50=7300nM Q86WV6 30655953 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLDPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPSFSLSQEVLRHLRQE 6mx3 B 1.362 BS01 K5P A 1 S162 G166 Y167 S9 G13 Y14 ? 0002218,0032481 remove_due_to_license_issue IC50=7300nM Q86WV6 30655953 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQE 6mx3 B 1.362 BS02 K5P B 1 S162 T263 P264 Q266 T267 S9 T97 P98 Q100 T101 ? 0002218,0032481 remove_due_to_license_issue IC50=7300nM Q86WV6 30655953 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQE 6mx8 A 1.96 BS01 6GY A 1 L1122 A1148 M1199 A1200 G1202 E1210 L1256 D1270 L29 A45 M96 A97 G99 E107 L151 D165 D1249 R1253 N1254 D1270 D144 R148 N149 D165 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=0.37nM remove_due_to_license_issue IC50=0.370000nM Q9UM73 27144831 1500 PNYCFAGKTSSISDLKEVPRKNITLIRGLGHGEVYEGQVSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMACAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIE 6mxb A 2.192 BS01 XMP A 1 I149 D151 T152 G153 T155 K180 Y201 V202 E208 I131 D133 T134 G135 T137 K162 Y183 V184 E190 E147 D148 D151 Y201 R214 E129 D130 D133 Y183 R196 ? 0000166,0000287,0000310,0004422,0005737,0005829,0006178,0016757,0020015,0032263,0032264,0042301,0046100,0046872,0052657 Ki=26uM remove_due_to_license_issue Q38CA1 31287615 301 PLKPNFVGRDADGNVTVDGRSYPMAESVVATESTIHRSMKEMAQTLANAYKTLKHRDTHNKGNSALAPITDENPLIIISVLKGSYIFTADMVRYLGDCGLPNVVDFIRITVLDNLRFTELTGKHVLIMEDIADTGRTMKLLVEKIRREYRPASLKVCVLVDKPGGRVVDFKPEFVCLTAPTRYVVGYGFEVNDRYRNYRHVFVLKPEYAKRYPSKL 6mxd A 2.96 BS01 IMP A 1 I149 D151 T152 G153 T155 K180 Y201 V202 I132 D134 T135 G136 T138 K163 Y184 V185 E147 D148 D151 Y201 R214 E130 D131 D134 Y184 R197 ? 0000166,0000287,0000310,0004422,0005737,0005829,0006178,0016757,0020015,0032263,0032264,0042301,0046100,0046872,0052657 remove_due_to_license_issue Q38CA1 31287615 301 PLKPNFVGRDADGNVTVDGRSYPMAESVVATESTIHRSMKEMAQTLANAYKTLKHRDTHNKGNSALAPITDENPLIIISVLKGSYIFTADMVRYLGDCGLPNVVDFIRITQVLDNLRFTELTGKHVLIMEDIADTGRTMKLLVEKIRREYRPASLKVCVLVDKPGGRVVDFKPEFVCLTAPTRYVVGYGFEVNDRYRNYRHVFVLKPEYAKRYPSKL 6mxe A 2.47 BS01 K5S B 1 L159 S162 T263 P264 Q266 T267 L6 S9 T97 P98 Q100 T101 ? 0002218,0032481 remove_due_to_license_issue IC50=68nM, EC50=>30000nM Q86WV6 30655953 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQESFSLSQEVLRHLRQ 6mxe A 2.47 BS02 K5S B 2 S162 Y163 G166 Y167 S9 Y10 G13 Y14 ? 0002218,0032481 remove_due_to_license_issue IC50=68nM, EC50=>30000nM Q86WV6 30655953 402 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQESFSLSQEVLRHLRQ 6mxe B 2.47 BS01 K5S B 1 S162 Y163 G166 Y167 S9 Y10 G13 Y14 ? 0002218,0032481 remove_due_to_license_issue IC50=68nM, EC50=>30000nM Q86WV6 30655953 401 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 6mxe B 2.47 BS02 K5S B 2 L159 S162 T263 P264 Q266 T267 L6 S9 T97 P98 Q100 T101 ? 0002218,0032481 remove_due_to_license_issue IC50=68nM, EC50=>30000nM Q86WV6 30655953 402 SVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQ 6myn A 2.744 BS01 K6Y A 1 R410 G411 V416 A429 V455 M471 E472 L473 L474 G477 L524 C535 D536 F537 R63 G64 V69 A82 V108 M124 E125 L126 L127 G130 L177 C188 D189 F190 D517 L553 D170 L200 2.7.11.25 0004672,0004674,0005524,0006468 remove_due_to_license_issue Q9WUL6 31531194 703 PVEEYLVHALQGSVSSGQAHSLASLAKTWSDNEGVLLTEKLKPVDYEYREEVHWMTHQPRVGRGSFGEVHRMKDKQTGFQCAVKKVRLEVFRVEELVACAGLSSPRIVPLYGAVREGPWVNIFMELLEGGSLGQLIKQMGCLPEDRALYYLGQALEGLEYLHTRRILHGDVKADNVLLSSDGSRAALCDFGHALCLQSLLTGDYIPGTETHMAPEVVMGKPCDAKVDIWSSCCMMLHMLNGCHPWTQYFRGPLCLKIASEPPPIREIPPSCAPLTAQAIQEGLRKEPVHRASAMELRRKVGKALQEVGGLKSPWKGEYKEPR 6mzq A 2.0 BS01 TZ0 A 1 L484 A512 K514 E531 M535 I545 E562 Y563 A564 N568 L630 A640 D641 L21 A46 K48 E65 M69 I79 E96 Y97 A98 N102 L161 A171 D172 D623 A625 R627 N628 D641 D154 A156 R158 N159 D172 2.7.10.1 0004672,0004713,0005007,0005524,0006468 ic50=3.9nM remove_due_to_license_issue IC50=3.6nM P11362 30600916 801 ELPEDPRWELPRDRLVLGKPLGEGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSYNPSEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSQE 6mzw A 2.2 BS01 TZ0 A 1 L484 G485 C488 V492 A512 K514 E531 M535 I545 Y563 A564 L630 D641 F642 L21 G22 C25 V29 A49 K51 E68 M72 I82 Y100 A101 L165 D176 F177 D623 R627 N628 D641 D158 R162 N163 D176 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue IC50=3.6nM P11362 30600916 801 ELPEDPRWELPRDRLVLGKPLGEGCFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPGLEYSYNPSPEEQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 6n0j A 1.79 BS02 K8S A 1 E18 V24 R26 D43 F45 F53 S65 L114 Q115 W117 Q252 E16 V22 R24 D41 F43 F51 S63 L112 Q113 W115 Q250 1.13.11.24 0003712,0005515,0005634,0005654,0005737,0005829,0006366,0007586,0008127,0016604,0030099,0030224,0046872,0051213 remove_due_to_license_issue O00625 302 SSKKVTLSVLSREQSEGVGARVRRSIGRPELKNLDPFLLFDEFKGGRPGGFPDHPHRGFETVSYLLEGGSMAHEDFCGHTGKMNPGDLQWMTAGRGILHAEMPCSEEPAHGLQLWVNLRSSEKMVEPQYQELKSEEIPKPSKDGVTVAVISGEALGIKSKVYTRTPTLYLDFKLDPGAKHSQPIPKGWTSFIYTISGDVYIGPDDAQQKIEPHHTAVLGEGDSVQVENKDPKRSHFVLIAGEPLREPVIQHGPFVMNTNEEISQAILDFRNAKNGFERAKTWKSKIGN 6n0k A 1.46 BS02 K8M A 1 E18 V24 R26 D43 F45 F53 S65 M73 L114 Q115 W117 Q252 G254 E16 V22 R24 D41 F43 F51 S63 M71 L112 Q113 W115 Q250 G252 1.13.11.24 0003712,0005515,0005634,0005654,0005737,0005829,0006366,0007586,0008127,0016604,0030099,0030224,0046872,0051213 remove_due_to_license_issue O00625 302 SSKKVTLSVLSREQSEGVGARVRRSIGRPELKNLDPFLLFDEFKGGRPGGFPDHPHRGFETVSYLLEGGSMAHEDFCGHTGKMNPGDLQWMTAGRGILHAEMPCSEEPAHGLQLWVNLRSSEKMVEPQYQELKSEEIPKPSKDGVTVAVISGEALGIKSKVYTRTPTLYLDFKLDPGAKHSQPIPKGWTSFIYTISGDVYIGPDDAQQKIEPHHTAVLGEGDSVQVENKDPKRSHFVLIAGEPLREPVIQHGPFVMNTNEEISQAILDFRNAKNGFERAKTWKSKIGN 6n0m A 3.3 BS01 K94 A 1 T374 Y375 T377 T386 R390 W444 E451 T260 Y261 T263 T272 R276 W330 E337 1.11.1.- 0005634,1901031 remove_due_to_license_issue P58004 30858438 900 GLEALMSSGRVDNLAVVMGLHPDYFTSFWRLHYLLLHTDGPLASSWRHYIAIMAAARHQCSYLVGSHMAEFLQTGGDPEWLLGLHRAPEKLRKLSEINKLLAHRPWLITKEHIQALLKTGEHTWSLAELIQALVLLTHCHSLSSFVFGCGILPEGDPPSEQSSPRDVEALMERMQQLQESEEMESRFELEKSESLPDMLCFVEDPTFGYEDFTRRGAQAPPTFRAQDYTWEDHGYSLIQRLYPEGGQLLDEKFQAAYSLTYNTIAMHSGVDTSVLRRAIWNYIHCVFGIRYDDYDYGEVNQLLERNLKVYIKTVACYPEKTTRRMYNLFWRHFRHSEKVHVNLLLLEARMQAALLYALRAITRYMT 6n0p A 2.37 BS01 K81 A 1 V471 A481 K483 E501 L505 L514 I527 T529 Q530 C532 D594 F595 V23 A33 K35 E53 L57 L66 I79 T81 Q82 C84 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S163 2.7.11.1 0004672,0005524,0006468 Kd=1.3nM remove_due_to_license_issue IC50=0.400000nM, Kd=1.3nM P15056 31059256 801 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSEQLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 6n0q A 2.04 BS01 K7S A 1 I463 V471 A481 K483 E501 L505 L514 I527 T529 G593 D594 F595 I18 V26 A36 K38 E56 L60 L69 I82 T84 G148 D149 F150 D576 K578 N580 N581 D594 S616 D131 K133 N135 N136 D149 S154 2.7.11.1 0004672,0005524,0006468 ic50=0.04uM remove_due_to_license_issue P15056 31059256 801 SSDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGSGSILWMAPEVIRMKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL 6n17 A 1.639 BS01 K8Y A 1 Y204 H263 K265 N283 S399 S400 P461 H493 K495 N516 Y43 H102 K104 N122 S238 S239 P295 H327 K329 N350 3.1.4.- 0005634,0006281,0008081 ic50=1.01mM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6n19 A 1.501 BS01 K8V A 1 Y204 H263 K265 N283 S399 S400 P461 H493 K495 N516 S518 Y43 H102 K104 N122 S238 S239 P295 H327 K329 N350 S352 3.1.4.- 0005634,0006281,0008081 ic50=0.96mM remove_due_to_license_issue Q9NUW8 31199869 701 NPFQFYLTRVSGVKPKYNSGALHIKDILSPLFGTLVSSAQFNYCFDVDWLVKQYPPEFRKKPILLVHGDKREAKAHLHAQAKPYENISLCQAKLDIAFGTHHTKMMLLLYEEGLRVVIHTSNLIHADWHQKTQGIWLSPLYPRIADGTHKSGESPTHFKADLISYLMAYNAPSLKEWIDVIHKHDLSETNVYLIGSTPGRFQGSQKDNWGHFRLKKLLKDHASSMPNAESWPVVGQFSSVGSLGADESKWLCSEFKESMLTLGKESSSVPLYLIYPSVENVRTSLEGYPAGGSLPYSIQTAEKQNWLHSYFHKWSAETSGRSNAMPHIKTYMRPSPDFSKIAWFLVTSANLSKAAWGALEKNGTQLMIRSYELGVLFLPSAFGLDSFKVKQKFFAGPMATFPVPYDLPPELYGSKDRPWIWNIPYVKAPDTHGNMWVP 6n3k A 2.2 BS01 K9V A 1 W46 D116 W117 H144 F165 Y167 Q168 M193 Y252 W46 D116 W117 H144 F165 Y167 Q168 M193 Y252 ? 0003824 ic50=29nM remove_due_to_license_issue G0R7E2 30771398 401 MDTSKLKPNDPRVKYETKQIRGKTYSYILGEPAGPKLETVVLVHGWPDMAFGWRHQIPYLMSLGFQVVAPNMLGYAGTDAPRDLSQFTLKSVSADIAELARSFVGQDGQIVLGGHDWGGAVVWRTAYYHPELVKAVFSVCTPLHPLSAEYKPLEDIVAAGHMLNFKYQLQLKGPDVEARIQGKDMLRRFFRAMFGGRGPNGEAGFSTSDGVHFDVLDKIGAPPLLDEQELEYYVEQYALQEAPELRGPLNWYRTRELNAKDEMDRAKNGPPLRFEMPALFVAASKDNALPPAMSKGMDAFYKDLTRAEVDATHWALTQAGDEVNRVIGEWLNKALG 6n3l A 2.61 BS01 KAV A 1 L596 A617 E636 L640 M802 E803 Y804 C805 F855 I864 G865 D866 F867 L13 A34 E53 L57 M83 E84 Y85 C86 F136 I145 G146 D147 F148 N848 K850 N853 D866 A904 N129 K131 N134 D147 A149 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9P2K8 31620240 2501 SRYFIEFEELQLLGKGAFGAVIKVQNKLDGCCYAVKRIPINPASRQFRRIKGEVTLLSRLHHENIVRYYNAWIENVHYLYIQMEYCEASTLRDTIDQGLYRDTVRLWRLFREILDGLAYIHEKGMIHRNLKPVNIFLDSDDHVKIGDFAALYVSPEYNQKVDLFSLGIIFFEMSYHPMVTASERIFVLNQLRDPFPEDFHAKQKSVISWLLNHDPAKRPTATELLKSELLP 6n3n A 3.01 BS01 KA4 A 1 L596 A617 K619 L640 Y651 I800 M802 Y804 C805 F855 D866 F867 L13 A34 K36 L55 Y66 I79 M81 Y83 C84 F134 D145 F146 N848 K850 N853 D866 E904 N127 K129 N132 D145 E156 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q9P2K8 31620240 2500 SRYFIEFEELQLLGKGAFGAVIKVQNKLDGCCYAVKRIPINPASFRRIKGEVTLLSRLHHENIVRYYNAWIENVHYLYIQMEYCEASTLRDTIDQGLYRDTVRLWRLFREILDGLAYIHEKGMIHRNLKPVNIFLDSDDHVKIGDFGLATDHLAFEALYVSPEYNQKVDLFSLGIIFFEMSYHPMVTASERIFVLNQLRDPTSPKFPEDHAKQKSVISWLLNHDPAKRPTATELLKSELLPP 6n3o A 2.4 BS01 KA7 A 1 L596 A617 K619 L640 Y651 M802 Y804 C805 F855 D866 F867 L13 A34 K36 L57 Y68 M84 Y86 C87 F137 D148 F149 N848 K850 N853 D866 E904 N130 K132 N135 D148 E160 2.7.11.1 0004672,0005524,0006468 ic50=2.4nM remove_due_to_license_issue Q9P2K8 31620240 2500 SRYFIEFEELQLLGKGAFGAVIKVQNKLDGCCYAVKRIPINPASRQFRRIKGEVTLLSRLHHENIVRYYNAWIENAVHYLYIQMEYCEASTLRDTIDQGLYRDTVRLWRLFREILDGLAYIHEKGMIHRNLKPVNIFLDSDDHVKIGDFGLATDHLAFSEALYVSPEYNQKVDLFSLGIIFFEMSYHPMVTASERIFVLNQLRDPTSPKFPEDFDDGEHAKQKSVISWLLNHDPAKRPTATELLKSELLPPP 6n3v A 1.45 BS01 KB7 A 1 I18 F19 F41 D43 I44 N99 G105 Q106 S107 H112 H114 I7 F8 F30 D32 I33 N88 G94 Q95 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=2.45uM remove_due_to_license_issue P49773 31503445 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 6n3w A 1.75 BS01 KBJ A 1 I18 F41 D43 I44 N99 G105 Q106 S107 H112 H114 I7 F30 D32 I33 N88 G94 Q95 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=1.56uM remove_due_to_license_issue P49773 31503445 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 6n3x A 1.1 BS01 KBD A 1 I18 F41 D43 I44 N99 G105 Q106 S107 H112 H114 I7 F30 D32 I33 N88 G94 Q95 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=8.09uM remove_due_to_license_issue P49773 31503445 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 6n3y A 1.8 BS01 HHJ A 1 I18 F41 D43 I44 N99 G105 Q106 S107 H112 H114 I7 F30 D32 I33 N88 G94 Q95 S96 H101 H103 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 Kd=3.65uM remove_due_to_license_issue P49773 31503445 201 RPGGDTIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 6n3y B 1.8 BS01 HHJ A 1 M121 W123 M105 W107 3.4.22.-,3.9.1.- 0000118,0000166,0003824,0005080,0005515,0005634,0005654,0005737,0005829,0005856,0005886,0006355,0006508,0006915,0007165,0008234,0009154,0016787,0016926,0016929,0043530,0050850,0070062,0072332 remove_due_to_license_issue P49773 31503445 201 TIFGKIIRKEIPAKIIFEDDRCLAFHDISPQAPTHFLVIPKKHISQISVAEDDDESLLGHLMIVGKKCAADLGLNKGYRMVVNEGSDGGQSVYHVHLHVLGGRQMHWPPG 6n3z A 2.238 BS01 KC4 A 1 W46 D116 W117 H144 Y167 F205 Y252 A288 W46 D116 W117 H144 Y167 F205 Y252 A288 ? 0003824 ic50=259.3nM remove_due_to_license_issue G0R7E2 30771398 401 MDTSKLKPNDPRVKYETKQIRGKTYSYILGEPAGPKLETVVLVHGWPDMAFGWRHQIPYLMSLGFQVVAPNMLGYAGTDAPRDLSQFTLKSVSADIAELARSFVGQDGQIVLGGHDWGGAVVWRTAYYHPELVKAVFSVCTPLHPLSAEYKPLEDIVAAGHMLNFKYQLQLKGPDVEARIQGKDMLRRFFRAMFGGRGPNGEAGFSTSDGVHFDVLDKIGAPPLLDEQELEYYVEQYALQEAPELRGPLNWYRTRELNAKDEMDRAKNGPPLRFEMPALFVAASKDNALPPAMSKGMDAFYKDLTRAEVDATHWALTQAGDEVNRVIGEWLNKALG 6n48 A 3.2 BS03 KBY A 1 V1126 D1130 F1133 S1137 L1144 K1149 I1153 V269 D273 F276 S280 L287 K292 I296 3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016998,0097746 remove_due_to_license_issue P07550 31249059 1403 DAENLYFQGNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYAADEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILTKTWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLQKFALKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6n4b R 3.0 BS01 KCA R 1 S173 F177 H178 V196 T197 F268 S65 F69 H70 V88 T89 F154 ? 0004930,0004949,0007186,0016020 remove_due_to_license_issue P21554 30639101 501 MVLNPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVFHRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLMWTIAIVIAVLPLLGWNCCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWKAHSHAVRMIQRGTARMDIRLAKTLVLILVVLIICWGPLLAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSM 6n4e A 1.65 BS02 KCD A 1 F9 M11 G13 R14 M99 W104 A105 Y152 F9 M11 G13 R14 M99 W104 A105 Y152 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 ic50=9.9nM remove_due_to_license_issue IC50=9.9nM, Kd=0.500000nM O60760 30858025 202 MPNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGNSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 6n4t A 1.945 BS03 KD7 A 1 H57 F99 Y146 Q175 D189 S190 C191 Q192 G193 D194 S195 W215 G216 G219 H42 F94 Y141 Q169 D185 S186 C187 Q188 G189 D190 S191 W212 G213 G215 H57 D102 Q192 G193 D194 S195 G196 H42 D97 Q188 G189 D190 S191 G192 3.4.21.109 0004252,0006508 remove_due_to_license_issue Q9Y5Y6 31543462 304 VVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV 6n53 A 2.7 BS01 UZR A 1 T29 K33 D62 Y65 D84 I137 R166 T11 K15 D39 Y42 D61 I114 R143 2.7.1.48 0004849,0005524,0005737,0005829,0009224,0016301,0042802,0043771,0044206,0044211 remove_due_to_license_issue Q9BZX2 32015544 304 EPFLIGVSGGTASGKSSVCAKIVQLLGQNQKQVVILSQDSFYRVLTSEQKAKALKGQFNFDHPDAFDNELILKTLKEITEGKTVQIPVYDFVSHSRKEETVTVYPADVVLFEGILAFYSQEVRDLFQMKLFVDTDADTRLSRRVLRDISERGRDLEQILSQYITFVKPAFEEFCLPTKKYADVIIPRGADNLVAINLIVQHIQDILN 6n54 A 2.424 BS01 KEA A 1 T29 K33 D62 Y65 F83 D84 F114 H117 R166 T12 K16 D41 Y44 F62 D63 F93 H96 R145 2.7.1.48 0004849,0005524,0005737,0005829,0009224,0016301,0042802,0043771,0044206,0044211 remove_due_to_license_issue Q9BZX2 32015544 304 GEPFLIGVSGGTASGKSSVCAKIVQLLGQNRQKQVVILSQDSFYRVLTSEQKAKALKGQFNFDHPDAFDNELILKTLKEITEGKTVQIPVYDFVSHSRKEETVTVYPADVVLFEGILAFYSQEVRDLFQMKLFVDTDADTRLSRRVLRDISERGRDLEQILSQYITFVKPAFEEFCLPTKKYADVIIPRGADNLVAINLIVQHIQDILNG 6n55 F 3.085 BS01 UZ0 F 1 Y65 F114 R174 Y46 F95 R155 2.7.1.48 0004849,0005524,0005737,0005829,0009224,0016301,0042802,0043771,0044206,0044211 remove_due_to_license_issue Q9BZX2 32015544 307 GEPFLIGVSGGTASGKSSVCAKIVQLLGQNDYRQKQVVILSQDSFYRVLTSEQKAKALKGQFNFDHPDAFDNELILKTLKEITEGKTVQIPVYDFVSHSRKEETVTVYPADVVLFEGILAFYSQEVRDLFQMKLFVDTDADTRLSRRVLRDISERGRDLEQILSQYITFVKPAFEEFCLPTKKYADVIIPRGADNLVAINLIVQHIQDILNG 6n5c A 1.95 BS05 KDJ A 1 K53 K54 R213 K214 K248 R262 S326 K329 K11 K12 R171 K172 K206 R220 S284 K287 2.7.4.24 0000829 remove_due_to_license_issue O43314 31391889 406 QIVVGICSMAKKSKSKPMKEILERISLFKYITVVVFEEEVILNEPVENWPLCDCLISFHSKGFPLDKAVAYAKLRNPFVINDLNMQYLIQDRREVYSILQAEGILLPRYAILNRDPNNPKECNLIEGEDHVEVNGEVFQKPFVEKPVSAEDHNVYIYYPTSAGGGSQRLFRKIGSRSSVYSPESNVRKTGSYIYEEFMPTDGTDVKVYTVGPDYAHAEARKSPALDGKVERDSEGKEVRYPVILNAREKLIAWKVCLAFKQTVCGFDLLRANGQSYVCDVNGFSFVKNSMKYYDDCAKILGNIVMRELAPQFHIPWS 6n5f A 1.93 BS01 KJ1 A 1 D116 W117 Y167 M193 Y252 H313 D116 W117 Y167 M193 Y252 H313 ? 0003824 ic50=138.8nM remove_due_to_license_issue G0R7E2 30771398 401 MDTSKLKPNDPRVKYETKQIRGKTYSYILGEPAGPKLETVVLVHGWPDMAFGWRHQIPYLMSLGFQVVAPNMLGYAGTDAPRDLSQFTLKSVSADIAELARSFVGQDGQIVLGGHDWGGAVVWRTAYYHPELVKAVFSVCTPLHPLSAEYKPLEDIVAAGHMLNFKYQLQLKGPDVEARIQGKDMLRRFFRAMFGGRGPNGEAGFSTSDGVHFDVLDKIGAPPLLDEQELEYYVEQYALQEAPELRGPLNWYRTRELNAKDEMDRAKNGPPLRFEMPALFVAASKDNALPPAMSKGMDAFYKDLTRAEVDATHWALTQAGDEVNRVIGEWLNKALG 6n5g A 2.6 BS01 KDS A 1 W46 D116 W117 T141 H144 Y167 M193 F205 Y252 A288 L289 H313 W314 W46 D116 W117 T141 H144 Y167 M193 F205 Y252 A288 L289 H313 W314 ? 0003824 remove_due_to_license_issue G0R7E2 30771398 401 MDTSKLKPNDPRVKYETKQIRGKTYSYILGEPAGPKLETVVLVHGWPDMAFGWRHQIPYLMSLGFQVVAPNMLGYAGTDAPRDLSQFTLKSVSADIAELARSFVGQDGQIVLGGHDWGGAVVWRTAYYHPELVKAVFSVCTPLHPLSAEYKPLEDIVAAGHMLNFKYQLQLKGPDVEARIQGKDMLRRFFRAMFGGRGPNGEAGFSTSDGVHFDVLDKIGAPPLLDEQELEYYVEQYALQEAPELRGPLNWYRTRELNAKDEMDRAKNGPPLRFEMPALFVAASKDNALPPAMSKGMDAFYKDLTRAEVDATHWALTQAGDEVNRVIGEWLNKALG 6n5h A 1.717 BS01 AUB A 1 D116 W117 F165 Y167 M193 G195 F205 Y252 H313 D116 W117 F165 Y167 M193 G195 F205 Y252 H313 ? 0003824 ic50=357.9nM remove_due_to_license_issue G0R7E2 30771398 401 MDTSKLKPNDPRVKYETKQIRGKTYSYILGEPAGPKLETVVLVHGWPDMAFGWRHQIPYLMSLGFQVVAPNMLGYAGTDAPRDLSQFTLKSVSADIAELARSFVGQDGQIVLGGHDWGGAVVWRTAYYHPELVKAVFSVCTPLHPLSAEYKPLEDIVAAGHMLNFKYQLQLKGPDVEARIQGKDMLRRFFRAMFGGRGPNGEAGFSTSDGVHFDVLDKIGAPPLLDEQELEYYVEQYALQEAPELRGPLNWYRTRELNAKDEMDRAKNGPPLRFEMPALFVAASKDNALPPAMSKGMDAFYKDLTRAEVDATHWALTQAGDEVNRVIGEWLNKALG 6n69 A 2.0 BS02 KDV A 1 G13 R14 M99 W104 G12 R13 M98 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005737,0006693,0009624,0010269,0016740,0016853,0042803,2000255 ic50=220000nM remove_due_to_license_issue O35543 30858025 202 PNYKLLYFNMRGRAEIIRYIFAYLDIKYEDHRIEQADWPKIKPTLPFGKIPVLEVEGLTLHQSLAIARYLTKNTDLAGKTELEQCQVDAVVDTLDDFMSLFPWAEENQDLKERTFNDLLTRQAPHLLKDLDTYLGDKEWFIGNYVTWADFYWDICSTTLLVLKPDLLGIYPRLVSLRNKVQAIPAISAWILKRPQTKL 6n6o A 2.6 BS01 KE7 A 1 I531 Q541 A551 M602 E603 G605 N606 I607 D608 L654 I17 Q27 A37 M88 E89 G91 N92 I93 D94 L140 D647 K649 N652 D664 T686 D133 K135 N138 D150 T156 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.700000nM P33981 30998356 801 NECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANTVNYMPPEAIKDMSKISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ 6n77 A 1.64 BS01 KEJ A 1 L881 G882 G887 V889 A906 M956 L959 E966 L1010 G1020 D1021 L16 G17 G22 V24 A41 M82 L85 E92 L136 G146 D147 D1003 A1005 R1007 N1008 D1021 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.57nM remove_due_to_license_issue P23458 30981576 1201 DPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n78 A 1.83 BS01 KEP A 1 L881 G882 E883 G887 V889 A906 M956 L959 E966 R1007 L1010 G1020 D1021 L16 G17 E18 G22 V24 A41 M81 L84 E91 R132 L135 G145 D146 D1003 A1005 R1007 N1008 D1021 D128 A130 R132 N133 D146 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.21nM remove_due_to_license_issue P23458 30981576 1201 DPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n79 A 2.27 BS01 KES A 1 L881 G882 G887 V889 A906 V938 M956 L959 E966 R1007 N1008 L1010 G1020 D1021 L16 G17 G22 V24 A41 V69 M83 L86 E93 R134 N135 L137 G147 D148 D1003 A1005 R1007 N1008 D1021 D130 A132 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.21nM remove_due_to_license_issue P23458 30981576 1201 DPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIEKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n7a A 1.33 BS01 KEV A 1 L881 G882 G887 V889 A906 M956 L959 E966 L1010 G1020 D1021 L17 G18 G23 V25 A42 M82 L85 E92 L136 G146 D147 D1003 R1007 N1008 D1021 D129 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Ki=4.3nM remove_due_to_license_issue P23458 30981576 1203 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n7b A 1.81 BS01 KEY A 1 L881 G882 E883 G887 V889 A906 M956 L959 E966 L1010 G1020 D1021 L17 G18 E19 G23 V25 A42 M82 L85 E92 L136 G146 D147 D1003 A1005 R1007 N1008 D1021 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.6nM remove_due_to_license_issue P23458 30981576 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n7c A 1.69 BS01 KF1 A 1 L881 G882 G887 V889 A906 M956 L959 E966 L1010 L17 G18 G23 V25 A42 M82 L85 E92 L136 D1003 A1005 R1007 N1008 D1021 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.67nM remove_due_to_license_issue P23458 30981576 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n7d A 1.78 BS01 KF4 A 1 L881 G882 V889 A906 M956 L959 E966 L1010 G1020 D1021 L17 G18 V25 A42 M82 L85 E92 L136 G146 D147 D1003 A1005 R1007 N1008 D1021 D129 A131 R133 N134 D147 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.3nM remove_due_to_license_issue P23458 30981576 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK 6n7y F 2.0 BS01 KFA F 1 N59 F206 F239 L246 L344 K347 N47 F192 F225 L232 L330 K333 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K45 F86 D91 D95 R100 D162 K186 F225 D229 D230 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=7.7uM remove_due_to_license_issue IC50=7700nM P14324 31577901 402 YAQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6n7z F 2.55 BS01 KF7 F 1 K57 N59 F206 F239 D243 K44 N46 F192 F225 D229 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F85 D90 D94 R99 D161 K186 F225 D229 D230 2.5.1.1,2.5.1.10 0004659,0008299,0016765 remove_due_to_license_issue IC50=2800nM P14324 31577901 402 AQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6n82 F 2.0 BS01 YF7 F 1 N59 F206 F239 D243 T255 N52 F197 F230 D234 T246 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K191 F230 D234 D235 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.1uM remove_due_to_license_issue IC50=860nM P14324 31577901 402 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6n82 F 2.0 BS02 YF7 F 2 L315 E318 Y322 A345 R346 Y349 K350 L306 E309 Y313 A336 R337 Y340 K341 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K191 F230 D234 D235 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.1uM remove_due_to_license_issue IC50=860nM P14324 31577901 403 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6n83 F 2.0 BS01 YL6 F 1 N59 R60 S205 F206 F239 Q242 L344 N50 R51 S196 F197 F230 Q233 L335 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K48 F89 D94 D98 R103 D165 K191 F230 D234 D235 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=0.54uM remove_due_to_license_issue P14324 31577901 401 SDVYAQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6n8x A 1.49484 BS01 KFY A 1 N51 A55 M98 L107 F138 Y139 W162 T184 N36 A40 M83 L92 F123 Y124 W147 T169 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=2uM remove_due_to_license_issue P07900 31141217 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 6n8y A 1.55391 BS01 KFY A 1 N46 A50 M93 L102 F133 Y134 W157 T179 N36 A40 M83 L92 F123 Y124 W147 T169 ? 0005524,0006457,0016887,0051082,0140662 Kd=4.2uM remove_due_to_license_issue P08238 31141217 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELKIDIIPNPQERTLTLVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVVVITKHNDDEQYAWESSAGGSFTVRADHGEPIGRGTKVILHLKEDQTEYLEERRVKEVVKKHSQFIGYPITLYLEKE 6n92 A 1.7 BS01 KFV A 1 L25 A64 H66 D67 I68 H69 W108 G109 G110 T132 P133 Y140 F250 K253 L24 A63 H65 D66 I67 H68 W107 G108 G109 T131 P132 Y139 F249 K252 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=10.8uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n92 C 1.7 BS01 KFV C 1 K24 L25 A64 H66 D67 I68 H69 L71 W108 L136 V138 Y140 F250 K23 L24 A63 H65 D66 I67 H68 L70 W107 L135 V137 Y139 F249 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=10.8uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n92 C 1.7 BS02 KFV C 2 W108 T128 S130 S165 P166 W107 T127 S129 S164 P165 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=10.8uM remove_due_to_license_issue P52045 30869886 303 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n93 A 1.7 BS01 KGA A 1 L25 A64 H66 D67 I68 H69 W108 T132 L136 F250 K253 L24 A63 H65 D66 I67 H68 W107 T131 L135 F249 K252 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=20.6uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n94 A 1.75 BS01 KGJ A 1 K24 L25 A64 H66 D67 I68 H69 W108 G109 G110 T132 P133 Y140 K23 L24 A63 H65 D66 I67 H68 W107 G108 G109 T131 P132 Y139 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=19.8uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n94 C 1.75 BS01 KGJ C 1 L25 A64 G65 H66 D67 I68 W108 G110 T132 P133 L136 Y140 F250 L24 A63 G64 H65 D66 I67 W107 G109 T131 P132 L135 Y139 F249 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=19.8uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n94 C 1.75 BS02 KGJ C 2 W108 T128 F129 S130 S165 P166 W107 T127 F128 S129 S164 P165 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=19.8uM remove_due_to_license_issue P52045 30869886 302 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n95 A 1.798 BS01 YXS A 1 K24 L25 K60 A64 H66 D67 I68 H69 W108 G109 G110 T132 P133 L136 V138 Y140 F250 K253 K23 L24 K59 A63 H65 D66 I67 H68 W107 G108 G109 T131 P132 L135 V137 Y139 F249 K252 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=7.5uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n95 C 1.798 BS01 YXS C 1 L25 A64 H66 D67 I68 W108 G109 G110 T132 P133 Y140 F250 L24 A63 H65 D66 I67 W107 G108 G109 T131 P132 Y139 F249 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=7.5uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n96 C 1.7 BS01 LCV C 1 L25 A64 H66 D67 I68 W108 G109 G110 T132 P133 L136 Y140 L24 A63 H65 D66 I67 W107 G108 G109 T131 P132 L135 Y139 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=3.8uM remove_due_to_license_issue P52045 30869886 301 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n96 C 1.7 BS03 LCV C 2 W108 T128 F129 S130 S165 P166 W107 T127 F128 S129 S164 P165 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=3.8uM remove_due_to_license_issue P52045 30869886 303 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n97 A 1.75 BS02 KGP A 1 L25 K60 A64 H66 D67 I68 W108 G109 G110 T132 P133 L136 Y140 F250 K253 L24 K59 A63 H65 D66 I67 W107 G108 G109 T131 P132 L135 Y139 F249 K252 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=7.1uM remove_due_to_license_issue P52045 30869886 302 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n97 C 1.75 BS02 KGP C 1 L25 A64 H66 D67 I68 W108 G109 G110 T132 P133 Y140 F250 L24 A63 H65 D66 I67 W107 G108 G109 T131 P132 Y139 F249 H66 L71 G110 E113 P133 V138 Y140 E228 Y238 H65 L70 G109 E112 P132 V137 Y139 E227 Y237 4.1.1.- 0003824,0004492,0005829,0006635,0016829,0016831 Ki=7.1uM remove_due_to_license_issue P52045 30869886 302 AYQYVNVVTINKVAVIEFNYGRKLNALSKVFIDDLMQALSDLNRPEIRCIILRAPSGSKVFSAGHDIHELPSGGRDPLSYDDPLRQITRMIQKFPKPIISMVEGSVWGGAFEMIMSSDLIIAASTSTFSMTPVNLGVPYNLVGIHNLTRDAGFHIVKELIFTASPITAQRALAVGILNHVVEVEELEDFTLQMAHHISEKAPLAIAVIKEELRVLGEAHTMNSDEFERIQGMRRAVYDSEDYQEGMNAFLEKRKPNFVGH 6n9l A 2.01 BS02 ADP A 1 H12 N13 S33 G34 S35 G36 K37 S38 S39 Y796 Q801 H11 N12 S32 G33 S34 G35 K36 S37 S38 Y505 Q510 ? 0003677,0005524,0006289,0009380,0016887 Kd=0.1uM remove_due_to_license_issue Q9WYV0 30892613 1002 NEIVVKGARVHNLKNITVRIPKNRLVVITGVSGSGKSSLAMDTIYAEGQRRYLESLSTYKKPDVDEIEGLSPAIAIDQKTVSHNPRSTVGTVTEIYDYLRVLYARIGKKINGLNIHEFTELSISEELEFLKNLNLTEREREIVGELLKEIEKRLEFLVDVGLEYLTLSRSATTLSGGESQRIRLATQIGSGLTGVIYVLDEPTIGLHPRDTERLIKTLKKLRDLGNTVIVVEHDEEVIRNADHIIDIGPGGGTNGGRVVFQGTVDELLKNPDSSLTGEYLSGKRKITVNKTRRLPYASLKIKGVRHNNLKNIDVEIPLGVFVCVTGVSGSGKSSLVMETLYPALMNLLHKTKLPAGEFDSIEGHENIDKMIAIDQSPIGRTPRSNPATYTKVFDEIRSLFAMTPAAKARGYNKSRFSFNLKGGRCEACQGQGYVKIEMLFLPDVYVECDVCKGKRYNRETLEITYKGKNISDILDMTVDEALEFFKNIPSIKRTLQVLHDVGLGYVKLGQPATTLSGGEAQRIKLASELRKRDTGRTLYILDEPTVGLHFEDVRKLVEVLHRLVDRGNTVIVIEHNLDVIKNADHIIDLGPEGGKEGGYIVATGTPEEIAKNPHSYTGRFLKNVL 6n9l A 2.01 BS03 ADP A 2 Y455 R460 N598 N599 S619 G620 S621 G622 K623 S624 S625 Y164 R169 N307 N308 S328 G329 S330 G331 K332 S333 S334 ? 0003677,0005524,0006289,0009380,0016887 Kd=0.1uM remove_due_to_license_issue Q9WYV0 30892613 1003 NEIVVKGARVHNLKNITVRIPKNRLVVITGVSGSGKSSLAMDTIYAEGQRRYLESLSTYKKPDVDEIEGLSPAIAIDQKTVSHNPRSTVGTVTEIYDYLRVLYARIGKKINGLNIHEFTELSISEELEFLKNLNLTEREREIVGELLKEIEKRLEFLVDVGLEYLTLSRSATTLSGGESQRIRLATQIGSGLTGVIYVLDEPTIGLHPRDTERLIKTLKKLRDLGNTVIVVEHDEEVIRNADHIIDIGPGGGTNGGRVVFQGTVDELLKNPDSSLTGEYLSGKRKITVNKTRRLPYASLKIKGVRHNNLKNIDVEIPLGVFVCVTGVSGSGKSSLVMETLYPALMNLLHKTKLPAGEFDSIEGHENIDKMIAIDQSPIGRTPRSNPATYTKVFDEIRSLFAMTPAAKARGYNKSRFSFNLKGGRCEACQGQGYVKIEMLFLPDVYVECDVCKGKRYNRETLEITYKGKNISDILDMTVDEALEFFKNIPSIKRTLQVLHDVGLGYVKLGQPATTLSGGEAQRIKLASELRKRDTGRTLYILDEPTVGLHFEDVRKLVEVLHRLVDRGNTVIVIEHNLDVIKNADHIIDLGPEGGKEGGYIVATGTPEEIAKNPHSYTGRFLKNVL 6n9p A 2.23 BS01 KHD A 1 V416 A428 K430 M449 T474 M477 C481 R525 L528 S538 D539 F540 V28 A40 K42 M61 T86 M89 C93 R137 L140 S150 D151 F152 D521 A523 R525 N526 D539 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30521698 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6nad A 2.90197 BS01 KHY A 1 Q286 L287 C320 H323 L324 V361 R364 M365 F377 F378 E379 F388 I400 Q22 L23 C56 H59 L60 V97 R100 M101 F113 F114 E115 F124 I136 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue Kd=0.500000nM, IC50=14nM P51449 31010722 601 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQI 6nao A 3.23 BS02 KHM A 1 A247 K362 R376 S434 Y436 H437 N482 F488 A87 K198 R212 S270 Y272 H273 N318 F324 2.7.7.86 remove_due_to_license_issue Kd=200nM, IC50=4900nM Q8N884 28934246 602 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKRNPKENPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEGNGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDEF 6nce A 2.598 BS01 dna C 0 S118 F119 N160 H164 S8 F9 N50 H54 ? 0003700,0006355,0043565 remove_due_to_license_issue O00409 30826165 1 ~ 16 GNCKPPYSFSCLIFMAIEDSPTKRLPVKDIYNWILEHFPYFANAPTGWKNSVRHNLSLNKCFKKVDKGSLWCIDPEYRQNLIQALKKTP 6nce A 2.598 BS02 dna D 0 K138 R163 H164 S167 K174 S187 W189 K28 R53 H54 S57 K64 S69 W71 ? 0003700,0006355,0043565 remove_due_to_license_issue O00409 30826165 1 ~ 16 GNCKPPYSFSCLIFMAIEDSPTKRLPVKDIYNWILEHFPYFANAPTGWKNSVRHNLSLNKCFKKVDKGSLWCIDPEYRQNLIQALKKTP 6ncj A 2.0 BS01 KJJ A 1 Q95 T124 T125 A128 A129 W132 Q40 T69 T70 A73 A74 W77 ? 0003676,0015074 ic50=0.024uM remove_due_to_license_issue F2WR52 30609350 305 SSPGIWQLDCTHLEGKVILVAVHVASGYIEAEVIPAETGQETAYFLLKLAGRWPVKTVHTDNGSNFTSTTVKAACWWAGIKQEDGIVIESMNKELKKIIGQVRDQAEHLKTAVQMAVFIHNHKRKGGYSAGERIVDIIATDI 6ncm A 2.704 BS01 dna C 0 V137 K138 R163 H164 S167 S187 V25 K26 R51 H52 S55 S68 ? 0003700,0006355,0043565 remove_due_to_license_issue O00409 30826165 1 ~ 16 CKPPYSFSCLIFMAIEDSPTKRLPVKDIYNWILEHFPYFANAPTGWKNSVRHNLSLNKCFKKVDKKGSLWCIDPEYRQNLIQALKKTPYHP 6ncm A 2.704 BS02 dna D 0 K114 S118 F119 N160 S161 H209 K2 S6 F7 N48 S49 H90 ? 0003700,0006355,0043565 remove_due_to_license_issue O00409 30826165 1 ~ 16 CKPPYSFSCLIFMAIEDSPTKRLPVKDIYNWILEHFPYFANAPTGWKNSVRHNLSLNKCFKKVDKKGSLWCIDPEYRQNLIQALKKTPYHP 6ncm B 2.704 BS01 dna D 0 S118 F119 S120 S161 H164 S7 F8 S9 S50 H53 ? 0003700,0006355,0043565 remove_due_to_license_issue O00409 30826165 1 ~ 16 NCKPPYSFSCLIFMAIEDSPTKRLPVKDIYNWILEHFPYFANAPTGWKNSVRHNLSLNKCFKKVDGSLWCIDPEYRQNLIQALKKTP 6ncn A 1.82 BS01 KJM A 1 L30 W34 D153 Q156 L7 W11 D130 Q133 ? 0005576,0006869,0008289,0042157 Kd=900uM remove_due_to_license_issue P02649 30933499 201 QRWELALGRFWDYLRWVQTLSEQVQEELLSSQVTQELRALMDETMKELKAYKSELEEQLTPVAEETRARLSKELQAAQARLGADMEDVRGRLVQYRGEVQAMLGQSTEELRVRLASHLRKLRKRLLRDADDLQKRLAVYQA 6nco A 1.707 BS01 KQP A 1 E27 L30 G31 W34 D35 D153 Q156 E4 L7 G8 W11 D12 D130 Q133 ? 0005576,0006869,0008289,0042157 Kd=30uM remove_due_to_license_issue P02649 30933499 201 QRWELALGRFWDYLRWVQTLSEQVQEELLSSQVTQELRALMDETMKELKAYKSELEEQLTPVAEETRARLSKELQAAQARLGADMEDVRGRLVQYRGEVQAMLGQSTEELRVRLASHLRKLRKRLLRDADDLQKRLAVYQA 6nd3 A 2.364 BS01 BTL A 1 Y208 F395 C489 E491 T502 Y157 F344 C438 E440 T451 F395 G488 C489 G821 F344 G437 C438 G770 4.3.99.4 0003824,0005829,0016829,0016840,0033265,0042426,0042803,0120525 remove_due_to_license_issue Q30W70 30557011 901 SGIPDGPTPRHVKLKENFLKQVPSITVQRAVAITKIAKENPGLPKPLLRAKTFRYCCETAPLVIQDHELIVGSPNGAPRAGAFSPEVAWRWLQDELDTIGSRPQDPFYISEEDKKVLREEVFPFWQNKSVDEFCEGQYREADLWEMSGESFVSDCSYHAVNGGGDSNPGYDVILMKKGMLDIQREAREKLEQLDYANPEDIDKIYFYKSVIETAEGVMIYARRLSAYAAELAARETDPRRKAELQKISEVNARVPAHAPSNFWEAIQAVWTVESLLVVEENQTGMSIGRVDQYMYPFYRADIDSGRLTEYEAFDLAGCMLVKMSEMMWITSEGASKFFAGYQPFVNMCVGGVTREGHDATNDLTYMLMDAVRHVRIYQPTLATRVHNKSPQKYLKKIVDVIRSGMGFPAVHFDDAHIKMMLAKGVSIEDARDYCLMGCVEPQKSGRLYQWTSTGYTQWPICIELVLNHGVPLWYGKKVTPDMGDLSQYDTYEKFEAAVKEQIRWITKNTSVATVISQRAHRELAPKPLMSLMYEGCMESGRDVSAGGAMYNFGPGVVWSGLATYVDSMAAIKKLVYDDRKYTLAQLNEALKADFAGYDQILADCLAAPKYGNDDDYADMIAADLVHFTETEHRKYKTLYSVLSHGTLSISNNTPFGQLLGASANGRRAWMPLSDGISPTQGADYKGPTAIIKSVSKMANDNMNIGMVHNFKLMSGLLDTPEGENGLITLIRTACMLGNGEMQFNYLDNELLLDAQKHPEKYRDLVVRVAGYSAFFVELCKDVQDEIISRTMLHGF 6ndl A 2.0 BS01 BQX A 1 S93 T94 Q116 R120 G121 R125 W127 S128 M137 D180 K187 G190 F191 G208 I209 G210 N212 I224 S92 T93 Q115 R119 G120 R124 W126 S127 M136 D179 K186 G189 F190 G207 I208 G209 N211 I223 6.3.4.15 0003677,0004077,0005524,0005737,0006355,0016740,0016874,0036211 Ki=0.065uM remove_due_to_license_issue Q2G258 31407891 406 SKYSQDVLQLLYKNKPNYISGQSIAESLNISRTAVKKVIDQLKLEGCKIDSVNHKGHLLQQLPDIWYQGIIDQYTKSSALFDFSEVYDSIDSTQLAAKKSLVGNQSSFFILSDEQTKGRGRFNRHWSSSKGQGLWMSVVLRPNVAFSMISKFNLFIALGIRDAIQHFSQDEVKVKWPNDIYIDNGKVCGFLTEMVANNDGIEAIICGIGINLTQQLENFDESIRHRATSIQLHDKNKLDRYQFLERLLQEIEKRYNQFLTLPFSEIREEYIAASNIWNRTLLFTENDKQFKGQAIDLDYDGYLIVRDEAGESHRLISADIDFG 6ne5 A 1.85 BS01 KJP A 1 H224 A227 F228 M231 M250 V253 F254 N260 R263 T266 L267 F270 G271 I294 H53 A56 F57 M60 M79 V82 F83 N89 R92 T95 L96 F99 G100 I123 ? 0042981 Ki=0.058nM remove_due_to_license_issue Ki=0.058000nM Q07820 30929420 400 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 6nel A 2.0 BS03 KKV A 1 Y24 K34 A37 I38 H41 E80 D108 E119 K134 Y29 K39 A42 I43 H46 E85 D113 E124 K139 ? 0003723,0039694 ic50=11nM remove_due_to_license_issue C6H0Y9 30983160 304 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSERG 6nem A 1.95 BS03 KKS A 1 A20 Y24 K34 A37 I38 H41 E80 D108 E119 R124 K134 A25 Y29 K39 A42 I43 H46 E85 D113 E124 R129 K139 ? 0003723,0039694 ic50=12nM remove_due_to_license_issue C6H0Y9 30983160 304 GPLGSMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 6nfg A 2.76 BS02 KKP A 1 R376 S434 Y436 N482 F488 R203 S261 Y263 N309 F315 2.7.7.86 remove_due_to_license_issue IC50=69000nM, Kd=78000nM Q8N884 602 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFKPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKRAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHAKEFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFDE 6nfh A 1.4 BS01 KLM A 1 L408 G409 V416 A428 K430 T474 M477 G480 L528 L20 G21 V28 A40 K42 T86 M89 G92 L140 D521 A523 R525 N526 D539 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30817167 701 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6nfi A 2.41 BS01 KLP A 1 L408 A428 K430 I472 T474 M477 G480 C481 L528 F540 L17 A33 K35 I72 T74 M77 G80 C81 L128 F140 D521 R525 N526 D539 D121 R125 N126 D139 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30817167 701 YGSWEIDPKDLTFLKELGTVVKYGKWRGQYDVAIKMISMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6nfn H 2.63 BS01 BCG L 1 W33 E99 L100 W33 E99 L100 remove_due_to_license_issue 31702583 301 EVQLVESGGGLVQPGGSLRLSCAASGFIFSSDWMNWVRQAPGKGLEWVANINQDGSEKYYVDSVKGRFTISRDNAQNSLYLQMNSLRAEDTAVYYCAKELGPWGQGTLVTVSSASTKGPSVFPLAPSALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEP 6nfn L 2.63 BS01 BCG L 1 Y34 A52 W93 Y98 Y32 A50 W91 Y96 remove_due_to_license_issue 31702583 301 VVIQESALTTSPGGTVILTCRSSTGTITTSNYANWVQKKPNHVFTGLIGATSIRAPGVPVRFSGFLIGGKAALTITGAQTEDDAMYFCALWYNTHYVFGGGTKVTVLGQPKAAPSVTLFPPSSEELQANKATLVCLISDFYPGAVTVAWKADSSPVKAGVETTTPSKQSNNKYAASSYLSLTPEQWKSHRSYSCQVTHEGSTVEKTVAPTE 6nfo A 2.93 BS02 KKM A 1 A247 R376 S434 Y436 H437 N482 F488 L490 A87 R203 S261 Y263 H264 N309 F315 L317 2.7.7.86 remove_due_to_license_issue IC50=8100nM, Kd=2700nM Q8N884 602 GASKLRAVLEKLKLSRDDISTAAGMVKGVVDHLLLRLKCDSAFRGVGLLNTGSYYEHVKISAPNEFDVMFKLEVPRIQLEEYSNTRAYYFVKFNPLSQFLEGEILSASKMLSKFRKIIKEEINDIKDTDVIMKRKPAVTLLISEKISVDITLALESKSSWPASTQEGLRIQNWLSAKVRKQLRLKPFYLVPKHANGFQEETWRLSFSHIEKEILNNHGKSKTCCENKEEKCCRKDCLKLMKYLLEQLKERFKDKKHLDKFSSYHVKTAFFHVCTQNPQDSQWDRKDLGLCFDNCVTYFLQCLRTEKLENYFIPEFNLFSSNLIDKRSKEFLTKQIEYERNNEFPVFD 6nfy A 2.17 BS01 B49 A 1 L23 A44 E92 F93 C94 G95 G97 D101 L144 L16 A34 E82 F83 C84 G85 G87 D91 L134 D137 K139 A141 N142 D155 A164 T175 D127 K129 A131 N132 D145 A154 T165 2.7.11.1 0004672,0005524,0006468 Kd=16nM remove_due_to_license_issue Kd=16nM Q92918 31018963 9000 GSNRDPRDHYDLLQRLGGGEVFKARDKVSGDLVALKMVKMEPDDDVSTLQKEILILKTCRHANIVAYHGSYLWLQKLWICMEFCGAGSLQDIYQVTGSLSELQISYVCREVLQGLAYLHSQKKIHRDIKGANILINDAGEVRLADFGISAQIGATLARRLSFIGTPYWMAPEVAAVALKGGYNELCDIWSLGITAIELAELQPPLFDVHPLRVLFLMTKSGYQPPRLKEKGKWSAAFHNFIKVTLTKSPKKRPSATKMLSHQLVSQPGLNRGLILDLLDKLK 6nfy B 2.17 BS01 B49 B 1 L23 A44 M91 E92 F93 C94 G95 A96 G97 D101 L144 A154 L16 A37 M84 E85 F86 C87 G88 A89 G90 D94 L137 A147 D137 K139 A141 N142 D155 A164 T175 D130 K132 A134 N135 D148 A157 T168 2.7.11.1 0004672,0005524,0006468 Kd=16nM remove_due_to_license_issue Kd=16nM Q92918 31018963 9000 GSNRDPRDHYDLLQRLGGGTYGEVFKARDKVSGDLVALKMVKMEPDDDVSTLQKEILILKTCRHANIVAYHGSYLWLQKLWICMEFCGAGSLQDIYQVTGSLSELQISYVCREVLQGLAYLHSQKKIHRDIKGANILINDAGEVRLADFGISAQIGATLARRLSFIGTPYWMAPEVAAVALKGGYNELCDIWSLGITAIELAELQPPLFDVHPLRVLFLMTKSGYQPPRLKEKGKWSAAFHNFIKVTLTKSPKKRPSATKMLSHQLVSQPGLNRGLILDLLDKLK 6nfz A 2.966 BS01 B49 A 1 L23 V31 M91 C94 G95 G97 D101 L144 L17 V23 M69 C72 G73 G75 D79 L122 D137 K139 A141 N142 D155 A164 T175 D115 K117 A119 N120 D133 A142 T153 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=16nM Q92918 31018963 401 DIFNRDPRDHYDLLQRLGTYGEVFKARDKVSGDLVALKMVTLQKEILILKTCRHANIVAYHGSYLWICMEFCGAGSLQDIYQVTGSLSELQISYVCREVLQGLAYLHSQKKIHRDIKGANILINDAGEVRLADFGISAQIGATLARRLSFIGTPYWMAPEVAAVALKGGYNELCDIWSLGITAIELAELQPPLFDVHPLRVLFLMTKSGYQPPRLKEKGKWSAAFHNFIKVTLTKSPKKRPSATKMLSHQLVSQPGLNRGLILDLLDKLK 6ng0 A 2.05 BS01 B49 A 1 L23 A44 M91 F93 C94 G95 G97 D101 L144 D155 L18 A36 M83 F85 C86 G87 G89 D93 L136 D147 D137 K139 A141 N142 D155 T175 D129 K131 A133 N134 D147 T162 2.7.11.1 0004672,0005524,0006468 Ki=10nM remove_due_to_license_issue Kd=16nM Q92918 31018963 9000 PDIFNRDPRDHYDLLQRLGGGEVFKARDKVSGDLVALKMVKMEPDDDVSTLQKEILILKTCRHANIVAYHGSYLWLQKLWICMEFCGAGSLQDIYQVTGSLSELQISYVCREVLQGLAYLHSQKKIHRDIKGANILINDAGEVRLADFGISALARRLEFIGTPYWMAPEVAAVALKGGYNELCDIWSLGITAIELAELQPPLFDVHPLRVLFLMTKSGYQPPRLKEKGKWSAAFHNFIKVTLTKSPKKRPSATKMLSHQLVSQPGLNRGLILDLLDKLKNPGKGPSIGD 6nj0 A 1.83 BS01 KOY A 1 L182 S188 R195 L223 L244 G246 A248 A249 G268 Y269 G270 T272 S276 T277 V289 D336 R350 L177 S183 R190 L218 L239 G241 A243 A244 G263 Y264 G265 T267 S271 T272 V283 D330 R344 T142 E273 F356 G361 T140 E268 F350 G355 6.2.1.26 0005524,0008756,0009234,0016874,0016877,0032991,0042802 ic50=8.1uM remove_due_to_license_issue P37353 30912442 501 IFSDWPWRHWRQVRGETIALRLNDEQLNWRELCARVDELASGFAVQGVVEGSGVMLRAWNTPQTLLAWLALLQCGARVLPVNPQLPQPLLEELLPNLTLQFALVPGENTFPALTSLHIQLVEGAHAATWQPTRLCSMTLTSGLPKAAVHTYQAHLASAQGVLSLIPFGDHDDWLLSLPLFHVSGQGIMWRWLYAGARMTVRDKQPLEQMLAGCTHASLVPTQLWRLLVNRSSVSLKAVLLGGAAIPVELTEQAREQGIRCFCGYGLTEFASTVCAKEADLADVGSPLPGREVKIVNNEVWLRAASMAEGYWRNGQLVSLVNDEGWYATRDRGEMHNGKLTIVGRLDNLFFSGGEGIQPEEVERVIAAHPAVLQVFIVPVADKEFGHRPVAVMEYDHESVDLSEWVKDKLARFQQPVRWLTLPPELKNSRQALKEWVQRQ 6njh A 2.15 BS02 KRD A 1 H326 T499 Q535 F538 F599 H73 T243 Q279 F282 F327 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 31013090 703 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPNQVSEFISNTFLD 6nji A 2.45 BS02 KR4 A 1 N487 T499 Q535 F538 F599 N235 T247 Q283 F286 F332 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue Q08499 31013090 702 EQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQNQVSEFISNTFLD 6njj A 2.3 BS02 KR7 A 1 M439 N487 W498 T499 I502 Q535 F538 F599 T603 M186 N231 W242 T243 I246 Q279 F282 F327 T331 3.1.4.53 0004114,0007165,0008081 remove_due_to_license_issue IC50=127nM Q08499 31013090 703 QEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPNQVSEFISNTFLD 6nlj D 1.65 BS01 KTV D 1 L68 P69 Q72 L68 P69 Q72 1.16.3.1 0004322,0005506,0005737,0005829,0006826,0006879,0006880,0008199,0015093,0016491,0020037,0034755,0046872,0070288 Kd=15uM remove_due_to_license_issue Q9HY79 31038945 201 MKGDKKVIQHLNKILGNELIAINQYFLHSRMWNDWGLKRLGAHEYHESIDEMKHADKLIERILFLEGLPNLQDLGKLLIGENTQEMLQCDLNLELKATKDLREAIVHCEQVHDYVSRDLLKDILESEEEHIDYLETQLGLIQKVGLENYLQSHMHE 6nm4 A 2.58 BS03 KS7 A 1 W293 C321 A322 D324 W356 W99 C127 A128 D130 W162 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 0042054 remove_due_to_license_issue Q9NQV7 31848333 403 SEPQDDDYLYCEMCQNFFIDSCAAHGPPTFVKDSAVDKGHPNRSALSLPPGLRIGPSGIPQAGLGVWNEASDLPLGLHFGPYEGRITEDEEAANNGYSWLITKGRNCYEYVDGKDKSWANWMRYVNCARDDEEQNLVAFQYHRQIFYRTCRVIRPGCELLVWYGDEYGQELGIKWGSKWKKELMA 6nm4 A 2.58 BS04 KS7 B 1 D214 S215 A217 A218 P221 D20 S21 A23 A24 P27 2.1.1.-,2.1.1.354,2.1.1.355,2.1.1.359,2.1.1.361,2.1.1.362 0042054 remove_due_to_license_issue Q9NQV7 31848333 403 SEPQDDDYLYCEMCQNFFIDSCAAHGPPTFVKDSAVDKGHPNRSALSLPPGLRIGPSGIPQAGLGVWNEASDLPLGLHFGPYEGRITEDEEAANNGYSWLITKGRNCYEYVDGKDKSWANWMRYVNCARDDEEQNLVAFQYHRQIFYRTCRVIRPGCELLVWYGDEYGQELGIKWGSKWKKELMA 6nmb A 2.3 BS01 AMH A 1 D189 S190 S195 W215 G226 D197 S198 S203 W223 G234 H57 D102 Q192 G193 D194 S195 H51 D102 Q200 G201 D202 S203 3.4.21.73 0004252,0006508 Ki=2.01mM remove_due_to_license_issue Ki=2000000nM P00749 30814058 302 FQCGQIIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTICLPSMYNDPQFGTSCEITGFGKENSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK 6nng A 2.397 BS03 DJ9 B 1 T179 V181 T179 V181 3.6.5.- 0000226,0000278,0003924,0005200,0005525,0005737,0005856,0005874,0007017,0015630,0016787,0046872 remove_due_to_license_issue Q2XVP4 31043459 505 MRECISIHVGQAGVQIGNACWELYCLEHGIQPDGQMPSDKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRQLFHPEQLITGKEDAANNYARGHYTIGKEIIDLVLDRIRKLADQCTGLQGFLVFHSFGGGTGSGFTSLLMERLSVDYGKKSKLEFSIYPAPQVSTAVVEPYNSILTTHTTLEHSDCAFMVDNEAIYDICRRNLDIERPTYTNLNRLISQIVSSITASLRFDGALNVDLTEFQTNLVPYPRIHFPLATYAPVISAEKAYHEQLSVAEITNACFEPANQMVKCDPRHGKYMACCLLYRGDVVPKDVNAAIATIKTKRSIQFVDWCPTGFKVGINYQPPTVVPGGDLAKVQRAVCMLSNTTAIAEAWARLDHKFDLMYAKRAFVHWYVGEGMEEGEFSEAREDMAALEKDYEEVGVDS 6nng B 2.397 BS02 DJ9 B 1 V236 C239 L240 L246 A248 D249 K252 L253 N256 I316 N348 K350 V235 C238 L239 L245 A247 D248 K251 L252 N255 I315 N347 K349 ? 0000226,0000278,0003924,0005200,0005515,0005525,0005737,0005856,0005874,0007017,0046872 remove_due_to_license_issue P02554 31043459 505 REIVHIQAGQCGNQIGAKFWEVISDEHGIDPTGSYHGDSDLQLERINVYYNEATGNKYVPRAILVDLEPGTMDSVRSGPFGQIFRPDNFVFGQSGAGNNWAKGHYTEGAELVDSVLDVVRKESESCDCLQGFQLTHSLGGGTGSGMGTLLISKIREEYPDRIMNTFSVMPSPKVSDTVVEPYNATLSVHQLVENTDETYCIDNEALYDICFRTLKLTTPTYGDLNHLVSATMSGVTTCLRFPGQLNADLRKLAVNMVPFPRLHFFMPGFAPLTSRGSQQYRALTVPELTQQMFDSKNMMAACDPRHGRYLTVAAIFRGRMSMKEVDEQMLNVQNKNSSYFVEWIPNNVKTAVCDIPPRGLKMSATFIGNSTAIQELFKRISEQFTAMFRRKAFLHWYTGEGMDEMEFTEAESNMNDLVSEYQQYQDA 6nnr A 1.05 BS01 UMC A 1 R21 C146 Q165 R166 S167 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 E58 W80 Y94 C146 R166 D169 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 23611499 901 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 6nnr A 1.05 BS02 UMC B 1 R126 R127 R126 R127 E58 W80 Y94 C146 R166 D169 E58 W80 Y94 C146 R166 D169 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 23611499 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 6nnr B 1.05 BS01 UMC A 1 R126 R127 R126 R127 E58 W80 Y94 C146 R166 D169 E58 W80 Y94 C146 R166 D169 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 23611499 901 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 6nnr B 1.05 BS02 UMC B 1 R21 C146 Q165 R166 S167 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 E58 W80 Y94 C146 R166 D169 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 remove_due_to_license_issue P0A884 23611499 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 6no9 A 1.712 BS01 KUV A 1 L44 F49 A65 K67 L120 E121 R122 V126 E171 L174 I185 D186 L12 F17 A33 K35 L88 E89 R90 V94 E139 L142 I153 D154 D167 K169 N172 D186 L193 T204 D135 K137 N140 D154 L161 T172 2.7.11.1 0004672,0004674,0005524,0006468,0043066 Ki=0.03nM remove_due_to_license_issue Ki=0.030000nM P11309 30715878 504 PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLH 6noc A 2.849 BS01 rna B 0 K201 E208 F242 N244 Y245 K284 R288 Q291 H326 Q329 K360 Y361 Y364 Q367 N415 Y416 Q419 K450 S453 H454 E457 F498 N500 Y501 K35 E42 F76 N78 Y79 K118 R122 Q125 H160 Q163 K194 Y195 Y198 Q201 N249 Y250 Q253 K284 S287 H288 E291 F332 N334 Y335 ? 0003723 remove_due_to_license_issue Q09312 30652968 1 ~ 8 VLPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGAYVVQTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRST 6nod A 2.547 BS01 rna D 0 Q206 Q213 N246 Y247 Y280 R283 Q286 H319 R358 Q361 N393 Y394 K426 Y427 S429 N430 E433 Y470 N472 Y473 Q476 H506 H509 K513 Q33 Q40 N73 Y74 Y107 R110 Q113 H146 R185 Q188 N220 Y221 K253 Y254 S256 N257 E260 Y297 N299 Y300 Q303 H333 H336 K340 ? 0003723 remove_due_to_license_issue Q09487 30652968 1 ~ 8 DDLLTRYRANPAMMKNLKLSDIRGALLKFAKDQVGSRFIQQELASSKDRFEKDSIFDEVVSNADELVDDIFGNYVVQKFFEYGEERHWARLVDAIIDRVPEYAFQMYACRVLQKALEKINEPLQIKILSQIRHVIHRCMKDQNGNHVVQKAIEKVSPQYVQFIVDTLLESSNTIYEMSVDPYGCRVVQRCLEHCSPSQTKPVIGQIHKRFDEIANNQYGNYVVQHVIEHGSEEDRMVIVTRVSNNLFEFATHKYSSNVIEKCLEQGAVYHKSMIVGAACHHQEGSVPIVVQMMKDQYANYVVQKMFDQVTSEQRRELILTVRPHIPVLRQFPHGKHILAKLEKY 6nod B 2.547 BS01 rna E 0 Q206 Q213 N246 Y247 Y280 R283 Q286 H319 R358 Q361 N393 Y394 K426 Y427 S429 N430 E433 Y470 N472 Y473 H506 H509 Q33 Q40 N73 Y74 Y107 R110 Q113 H146 R185 Q188 N220 Y221 K253 Y254 S256 N257 E260 Y297 N299 Y300 H333 H336 ? 0003723 remove_due_to_license_issue Q09487 30652968 1 ~ 8 DDLLTRYRANPAMMKNLKLSDIRGALLKFAKDQVGSRFIQQELASSKDRFEKDSIFDEVVSNADELVDDIFGNYVVQKFFEYGEERHWARLVDAIIDRVPEYAFQMYACRVLQKALEKINEPLQIKILSQIRHVIHRCMKDQNGNHVVQKAIEKVSPQYVQFIVDTLLESSNTIYEMSVDPYGCRVVQRCLEHCSPSQTKPVIGQIHKRFDEIANNQYGNYVVQHVIEHGSEEDRMVIVTRVSNNLFEFATHKYSSNVIEKCLEQGAVYHKSMIVGAACHHQEGSVPIVVQMMKDQYANYVVQKMFDQVTSEQRRELILTVRPHIPVLRQFPHGKHILAKLEKY 6nod C 2.547 BS01 rna F 0 Q206 Q213 N246 Y247 Y280 R283 Q286 H319 R358 Q361 Y391 N393 Y394 K426 Y427 S429 N430 E433 Y470 N472 Y473 Q476 H506 Q33 Q40 N73 Y74 Y107 R110 Q113 H146 R185 Q188 Y218 N220 Y221 K253 Y254 S256 N257 E260 Y297 N299 Y300 Q303 H333 ? 0003723 remove_due_to_license_issue Q09487 30652968 1 ~ 8 DDLLTRYRANPAMMKNLKLSDIRGALLKFAKDQVGSRFIQQELASSKDRFEKDSIFDEVVSNADELVDDIFGNYVVQKFFEYGEERHWARLVDAIIDRVPEYAFQMYACRVLQKALEKINEPLQIKILSQIRHVIHRCMKDQNGNHVVQKAIEKVSPQYVQFIVDTLLESSNTIYEMSVDPYGCRVVQRCLEHCSPSQTKPVIGQIHKRFDEIANNQYGNYVVQHVIEHGSEEDRMVIVTRVSNNLFEFATHKYSSNVIEKCLEQGAVYHKSMIVGAACHHQEGSVPIVVQMMKDQYANYVVQKMFDQVTSEQRRELILTVRPHIPVLRQFPHGKHILAKLEKY 6nof A 2.251 BS01 rna B 0 K201 E208 N244 Y245 Q248 F285 R288 Q291 H326 Q329 K360 Y364 Y413 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 S554 K557 K34 E41 N77 Y78 Q81 F118 R121 Q124 H159 Q162 K193 Y197 Y246 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 S387 K390 ? 0003723 remove_due_to_license_issue Q09312 30652968 1 ~ 8 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGAYVVSTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRSTH 6noh A 2.249 BS01 rna B 0 N244 Y245 Q248 R288 Q291 Q322 N323 H326 Q329 K360 Y361 Y364 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 S554 N77 Y78 Q81 R121 Q124 Q155 N156 H159 Q162 K193 Y194 Y197 N248 Y249 Q252 K283 S286 H287 E290 N333 Y334 S387 ? 0003723 remove_due_to_license_issue Q09312 30652968 1 ~ 8 LPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGSYVVSTIIEKLTADSMNVDLTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRSTH 6np2 A 1.2 BS01 SIS A 1 Y85 Y113 D136 H189 S225 N226 Y67 Y95 D118 H171 S207 N208 2.3.1.81 0008080,0016746,0046353,0046677,0046872 Kd=0.16uM remove_due_to_license_issue Q47030 31515870 301 TPWSKSELVRQLRDLGVRSGDMVMPHVSLRAVGPLADGPQTLVDALIEAVGPTGNILAFVSWRDSPYEQTLGHDAPPAAIAQSWPAFDPDHAPAYPGFGAINEFIRTYPGCRRSAHPDASMAAIGPDAAWLVAPHEMGAAYGPRSPIARFLAHAGKILSIGAGPDAVTALHYAEAVARIEGKRRVTYSMPLLREGKRVWVTTSDWDSNGILDEYAAPDGPDAVERIARDYLARTRVAQGPVGGAQSRLIDAADIVSFGIEWLEARHAA 6np3 A 1.15 BS01 LLL A 1 Y85 E86 Y113 D136 D183 H189 S225 N226 Y67 E68 Y95 D118 D165 H171 S207 N208 2.3.1.81 0008080,0016746,0046353,0046677,0046872 Kd=0.34uM remove_due_to_license_issue Q47030 31515870 301 TPWSKSELVRQLRDLGVRSGDMVMPHVSLRAVGPLADGPQTLVDALIEAVGPTGNILAFVSWRDSPYEQTLGHDAPPAAIAQSWPAFDPDHAPAYPGFGAINEFIRTYPGCRRSAHPDASMAAIGPDAAWLVAPHEMGAAYGPRSPIARFLAHAGKILSIGAGPDAVTALHYAEAVARIEGKRRVTYSMPLLREGKRVWVTTSDWDSNGILDEYAAPDGPDAVERIARDYLARTRVAQGPVGGAQSRLIDAADIVSFGIEWLEARHAA 6np4 A 1.151 BS01 TOY A 1 Y85 E86 D136 H189 S225 N226 Y67 E68 D118 H171 S207 N208 2.3.1.81 0008080,0016746,0046353,0046677,0046872 Kd=36uM remove_due_to_license_issue Q47030 31515870 301 TPWSKSELVRQLRDLGVRSGDMVMPHVSLRAVGPLADGPQTLVDALIEAVGPTGNILAFVSWRDSPYEQTLGHDAPPAAIAQSWPAFDPDHAPAYPGFGAINEFIRTYPGCRRSAHPDASMAAIGPDAAWLVAPHEMGAAYGPRSPIARFLAHAGKILSIGAGPDAVTALHYAEAVARIEGKRRVTYSMPLLREGKRVWVTTSDWDSNGILDEYAAPDGPDAVERIARDYLARTRVAQGPVGGAQSRLIDAADIVSFGIEWLEARHAA 6npe A 2.15 BS02 KWD A 1 A356 L359 L360 I451 A452 Y454 E481 G482 P484 V487 A101 L104 L105 I196 A197 Y199 E226 G227 P229 V232 D382 A384 R386 N387 D400 P421 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.00000001M remove_due_to_license_issue IC50=1259nM, EC50=5012nM P00519 30689376 604 YDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 6npf D 2.57 BS01 KVM D 1 S41 Q166 E167 E208 D245 E289 D316 K341 H369 R370 S371 K392 S49 Q169 E170 E211 D248 E291 D318 K343 H371 R372 S373 K394 S41 E167 E208 D245 E289 D316 K341 H369 K392 S49 E170 E211 D248 E291 D318 K343 H371 K394 4.2.1.11 0000015,0000287,0004634,0005515,0005576,0005737,0005829,0005856,0006096,0006396,0006401,0009986,0016020,0016829,0042802,0042803,0046872,1990061 remove_due_to_license_issue P0A6P9 31745118 601 QQMGRGSMSKIVKIIGREIIDSRGNPTVEAEVHLEGGFVGMAAAPSGASTGSREALELRDGDKSRFLGKGVTKAVAAVNGPIAQALIGKDAKDQAGIDKIMIDLDGTENKSKFGANAILAVSLANAKAAAAAKGMPLYEHIAELNGTPGKYSMPVPMMNIINGGDNDIQEFMIQPVGAKTVKEAIRMGSEVFHHLAKVLKAKGMNTAVGDEGGYAPNLGSNAEALAVIAEAVKAAGYELGKDITLAMDCAASEFYKDGKYVLAGENKAFTSEEFTHFLEELTKQYPIVSIEDGLDESDWDGFAYQTKVLGDKIQLVGDDLFVTNTKILKEGIEKGIANSILIKFNQIGSLTETLAAIKMAKDAGYTAVISHRSGETEDATIADLAVGTAAGQIKTGSMSRSDRVAKYNQLIRIEEALGEKAPYNGRKEIKGQ 6npm B 1.603 BS01 KVD B 1 N480 I481 G484 S516 N519 L582 K586 T590 N7 I8 G11 S43 N46 L109 K113 T117 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 Ki=110uM remove_due_to_license_issue P03211 30842315 701 SNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6npp B 1.35 BS01 KWG B 1 K477 N480 I481 S516 N519 L582 K586 T590 K4 N7 I8 S43 N46 L109 K113 T117 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 Ki=0.89uM remove_due_to_license_issue P03211 30842315 701 SNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6npt A 2.19 BS01 KWY A 1 F646 D668 G670 R673 F139 D161 G163 R166 D650 R654 N655 D668 D143 R147 N148 D161 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=68.3pM remove_due_to_license_issue P04629 31059222 801 IENCVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 6npu A 2.33 BS02 KWV A 1 A356 L359 L360 A452 Y454 E481 G482 P484 V487 A101 L104 L105 A197 Y199 E226 G227 P229 V232 D382 A384 R386 N387 D400 P421 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.00000001M remove_due_to_license_issue IC50=398nM, EC50=794nM P00519 30689376 602 YDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 6npv A 1.86 BS02 KWP A 1 A356 I451 A452 Y454 E481 G482 P484 V487 A101 I196 A197 Y199 E226 G227 P229 V232 D382 A384 R386 N387 D400 P421 D127 A129 R131 N132 D145 P166 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.00000001M remove_due_to_license_issue IC50=158nM, EC50=3162nM P00519 30689376 603 YDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 6nrf A 2.0 BS01 KYV A 1 H862 G863 N868 G888 Y889 Y896 F897 S904 Y907 H92 G93 N98 G118 Y119 Y126 F127 S134 Y137 S904 Y907 E988 S134 Y137 E218 2.4.2.-,2.4.2.30 0003950 ic50=18nM remove_due_to_license_issue P09874 31042381 1103 KSKLPKPVQDLIKMIFGDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 6nrg A 1.7 BS01 KYY A 1 H862 G863 G888 Y889 Y896 F897 S904 Y907 H92 G93 G118 Y119 Y126 F127 S134 Y137 S904 Y907 E988 S134 Y137 E218 2.4.2.-,2.4.2.30 0003950 ic50=56nM remove_due_to_license_issue P09874 31042381 1101 KSKLPKPVQDLIKMIFGDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 6nrh A 1.5 BS01 KYP A 1 H862 G863 N868 G888 Y889 Y896 F897 S904 Y907 H92 G93 N98 G118 Y119 Y126 F127 S134 Y137 S904 Y907 E988 S134 Y137 E218 2.4.2.-,2.4.2.30 0003950 ic50=55nM remove_due_to_license_issue P09874 31042381 1101 KSKLPKPVQDLIKMIFGDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 6nri A 2.2 BS01 KYM A 1 H862 G863 N868 G888 Y889 Y896 F897 S904 Y907 H93 G94 N99 G119 Y120 Y127 F128 S135 Y138 S904 Y907 E988 S135 Y138 E219 2.4.2.-,2.4.2.30 0003950 ic50=27nM remove_due_to_license_issue IC50=27nM P09874 31042381 1101 KSKLPKPVQDLIKMIFGGDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 6nrj A 1.65 BS01 KYJ A 1 H862 G863 R878 A880 G888 Y889 Y896 F897 S904 Y907 H92 G93 R108 A110 G118 Y119 Y126 F127 S134 Y137 S904 Y907 E988 S134 Y137 E218 2.4.2.-,2.4.2.30 0003950 ic50=36nM remove_due_to_license_issue IC50=36nM P09874 31042381 1101 KSKLPKPVQDLIKMIFGDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFK 6nsp A 2.31 BS01 L0P A 1 K544 E560 L564 M587 F589 G667 D668 G670 K45 E61 L65 M88 F90 G165 D166 G168 D650 R654 N655 D668 D148 R152 N153 D166 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=44.1pM remove_due_to_license_issue P04629 31059222 801 ACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 6nsq B 3.05 BS01 KZP B 1 A481 K483 E501 L505 L514 T529 W531 C532 G593 D594 F595 A35 K37 E55 L59 L68 T83 W85 C86 G147 D148 F149 D576 K578 N580 N581 D594 S616 D130 K132 N134 N135 D148 S152 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=420nM P15056 31312411 801 SDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARELS 6nss A 1.97 BS01 L0M A 1 G488 H489 I490 F521 K544 E560 L564 V573 M587 F589 D668 G670 G4 H5 I6 F32 K55 E68 L72 V81 M95 F97 D176 G178 D650 R654 N655 D668 D158 R162 N163 D176 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=1.4nM remove_due_to_license_issue P04629 31059222 801 GLQGHIIENPQCVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 6nt2 A 2.48 BS02 KZS A 1 Y57 I62 M66 E162 W163 M164 H311 Y16 I21 M25 E121 W122 M123 H270 2.1.1.319 0001701,0003723,0005515,0005634,0005654,0005737,0005764,0005765,0005829,0006338,0006355,0006479,0006974,0007166,0008168,0008170,0008276,0008284,0008327,0008380,0016020,0016274,0018216,0019082,0019899,0030510,0031175,0032259,0034709,0035241,0035242,0035642,0042054,0042802,0044020,0045648,0045652,0045653,0045727,0046329,0046985,0048273,0048738,0051260,0061431,0062122,0070611,0106080,0140592,0140759,0140903,0140984,1900745,1904047,1904263,1905168,1990259 remove_due_to_license_issue Q99873 31257072 402 PNAEDMTSKDYYFDSYAHFGIHEEMLKDEVRTLTYRNSMFHNRHLFKDKVVLDVGSGTGILCMFAAKAGARKVIGIECSSISDYAVKIVKANKLDHVVTIIKGKVEEVELPVEKVDIIISEWMGYCLFYESMLNTVLYARDKWLAPDGLIFPDRATLYVTAIEDRQYKDYKIHWWENVYGFDMSCIKDVAIKEPLVDVVDPKQLVTNACLIKEVDIYTVKVEDLTFTSPFCLQVKRNDYVHALVAYFNIEFTRCHKRTGFSTSPESPYTHWKQTVFYMEDYLTVKTGEEIFGTIGMRPNAKNNRDLDFTIDLDFKGQLCELSCSTDYRMR 6nt2 D 2.48 BS02 KZS D 1 Y57 I62 E65 M66 E162 W163 M164 E171 H311 Y16 I21 E24 M25 E121 W122 M123 E130 H270 2.1.1.319 0001701,0003723,0005515,0005634,0005654,0005737,0005764,0005765,0005829,0006338,0006355,0006479,0006974,0007166,0008168,0008170,0008276,0008284,0008327,0008380,0016020,0016274,0018216,0019082,0019899,0030510,0031175,0032259,0034709,0035241,0035242,0035642,0042054,0042802,0044020,0045648,0045652,0045653,0045727,0046329,0046985,0048273,0048738,0051260,0061431,0062122,0070611,0106080,0140592,0140759,0140903,0140984,1900745,1904047,1904263,1905168,1990259 remove_due_to_license_issue Q99873 31257072 402 PNAEDMTSKDYYFDSYAHFGIHEEMLKDEVRTLTYRNSMFHNRHLFKDKVVLDVGSGTGILCMFAAKAGARKVIGIECSSISDYAVKIVKANKLDHVVTIIKGKVEEVELPVEKVDIIISEWMGYCLFYESMLNTVLYARDKWLAPDGLIFPDRATLYVTAIEDRQYKDYKIHWWENVYGFDMSCIKDVAIKEPLVDVVDPKQLVTNACLIKEVDIYTVKVEDLTFTSPFCLQVKRNDYVHALVAYFNIEFTRCHKRTGFSTSPESPYTHWKQTVFYMEDYLTVKTGEEIFGTIGMRPNAKNNRDLDFTIDLDFKGQLCELSCSTDYRMR 6ntb A 1.9 BS01 ATP A 1 G39 E40 G41 S42 R43 N44 R46 N59 S88 C89 I90 G38 E39 G40 S41 R42 N43 R45 N50 S79 C80 I81 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSRNVRSTGSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6ntb A 1.9 BS02 ATP B 1 G31 Y32 T33 V64 L65 H102 F104 G30 Y31 T32 V55 L56 H93 F95 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSRNVRSTGSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6ntb C 1.9 BS01 ATP A 1 G31 Y32 T33 L65 H102 G31 Y32 T33 L65 H102 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SSQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSRNVRSTGEPSVSHAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6ntb C 1.9 BS02 ATP C 1 G39 E40 G41 S42 R43 N44 V45 R46 E50 N59 S88 C89 I90 G39 E40 G41 S42 R43 N44 V45 R46 E50 N59 S88 C89 I90 ? 0005524,0006808,0030234,0046872 remove_due_to_license_issue B5II98 201 SSQQVWKLVIITEEILLKKVSKIIKEAGASGYTVLAAAGEGSRNVRSTGEPSVSHAYSNIKFEVLTASRELADQIQDKVVAKYFDDYSCITYISTVEALRAHKF 6ntj A 1.9 BS01 LLL A 1 Y85 E86 Y113 D136 Y159 H189 S225 N226 Y67 E68 Y95 D118 Y141 H171 S207 N208 2.3.1.81 0016746,0046353,0046677 remove_due_to_license_issue C4NV15 31515870 301 TPWSKSELVRQLRDLGVRSGDMVMPHVSLRAVGPLADGPQTLVDALIEAVGPTGNILAFVSWRDSPYEQTLGHDAPPAAIAQSWPAFDPDHAPAYPGFGAINEFIRTYPGCRRSAHPDASMAAIGPDAAWLVAPHEMGAAYGPRSPIARFLAHAGKILSIGAGPDAVTALHYAEAVARIEGKRRVTYSMPLLREGKRVWVTTSDWDSNGILDEYAAPDGPDAVERIARDYLARTRVAQGPVGGAQSRLIDAADIVSFGIEWLEARHA 6nu1 D 2.25 BS01 CYS D 1 R43 N44 N70 H464 I469 R30 N31 N57 H448 I453 R73 R120 K270 T328 R60 R107 K254 T312 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 31386812 601 QTQQLHAAMADTFLEHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP 6nu5 A 1.6 BS01 CYS A 1 R43 N44 N70 H464 G468 I469 F470 R37 N38 N64 H458 G462 I463 F464 R73 R120 K270 T328 R67 R114 K264 T322 2.7.10.2,2.7.11.1,2.7.1.40 0000287,0003723,0003729,0003824,0004743,0005515,0005524,0005576,0005634,0005737,0005739,0005791,0005829,0005929,0006096,0006338,0006417,0012501,0016301,0023026,0030955,0031982,0032869,0034774,0035401,0045296,0046872,0061621,0062023,0070062,0140801,1903561,1903672,1904813,2000767 remove_due_to_license_issue P14618 31386812 601 EAGTAFIQTQQLHAAMADTFLEHMCRLDIDSPPITARNTGIICTIGPASRSVETLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRTATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKQKGADFLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKASDVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAIYHLQLFEELRRLAPITSDPTEATAVGAVEASFKCCSGAIIVLTKSGRYAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDPVQEAWAEDVDLRVNFAMNVGKARGFFKKGDVVIVLTGWRPFTNTMRVVPVP 6nv7 A 2.132 BS01 L3J A 1 G11 Q12 L30 D32 G34 Y71 T72 Q73 F108 D228 G230 T231 T232 N233 R235 G14 Q15 L33 D35 G37 Y74 T75 Q76 F111 D220 G222 T223 T224 N225 R227 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D220 T223 3.4.23.46 0004190,0006508,0016020 Ki=5nM remove_due_to_license_issue P56817 31549827 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6nv9 A 2.13 BS01 L3M A 1 G11 Q12 L30 D32 G34 P70 Y71 T72 Q73 F108 Y198 D228 G230 T231 T232 N233 R235 G14 Q15 L33 D35 G37 P73 Y74 T75 Q76 F111 Y191 D221 G223 T224 T225 N226 R228 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 Ki=7nM remove_due_to_license_issue P56817 31549827 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6nvg A 1.99 BS01 XL8 A 1 L473 V481 R483 A501 K503 E520 M524 I534 V550 C552 A553 G556 L610 D621 L21 V29 R31 A49 K51 E68 M72 I82 V98 C100 A101 G104 L158 D169 D603 R607 N608 D621 D151 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 31413803 804 DLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAVS 6nvh A 1.9 BS01 XL6 A 1 V481 R483 A501 K503 E520 M524 I534 V550 C552 A553 G556 L610 A620 D621 V26 R28 A46 K48 E65 M69 I79 V95 C97 A98 G101 L155 A165 D166 D603 R607 N608 D621 D148 R152 N153 D166 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 31413803 803 DLPLDPLWEFPRDRLVLGKPLGEGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 6nvi A 2.117 BS01 XL7 A 1 V481 R483 A501 K503 E520 M524 I534 V550 C552 A553 G556 L610 A620 D621 V25 R27 A45 K47 E64 M68 I78 V94 C96 A97 G100 L152 A162 D163 D603 R607 N608 D621 D145 R149 N150 D163 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 31413803 801 DLPLDPLWEFPRDRLVLGKPLGEQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV 6nvj A 2.3 BS01 XL5 A 1 L473 R483 E520 M524 I534 V550 C552 A553 G556 L610 A620 D621 L21 R29 E66 M70 I80 V96 C98 A99 G102 L156 A166 D167 D603 R607 N608 D621 D149 R153 N154 D167 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P22455 31413803 805 DLPLDPLWEFPRDRLVLGKPLGEGGQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAVS 6nvl A 2.7 BS01 XL6 A 1 C488 V492 A512 K514 E531 M535 I545 V561 Y563 A564 N568 L630 A640 D641 F642 C26 V30 A50 K52 E69 M73 I83 V99 Y101 A102 N106 L154 A164 D165 F166 D623 R627 N628 D641 D147 R151 N152 D165 2.7.10.1 0004672,0004713,0005007,0005524,0006468 remove_due_to_license_issue P11362 31413803 802 YELPEDPRWELPRDRLVLGKPLGEGCFGQVVLAEAIGLDKDKPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLYYKKTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTSNQE 6nw3 A 2.352 BS01 L4J A 1 L30 D32 G34 P70 Y71 T72 Q73 F108 Y198 D228 G230 T231 T232 N233 R235 T329 L33 D35 G37 P73 Y74 T75 Q76 F111 Y191 D221 G223 T224 T225 N226 R228 T315 D32 S35 N37 A39 Y71 D228 T231 D35 S38 N40 A42 Y74 D221 T224 3.4.23.46 0004190,0006508,0016020 Ki=21nM remove_due_to_license_issue IC50=4nM P56817 31549827 401 SFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGY 6nwc A 2.35 BS01 L6P A 1 K56 L79 L83 I106 H111 Y116 L159 N163 K32 L55 L59 I82 H87 Y92 L135 N139 ? ic50=18nM remove_due_to_license_issue Q8H1R0 31649167 201 SQCSSTLVKHIKAPLHLVWSIVRRFDEPQKYKPFISRCVVQGKKLEVGSVREVDLKSGLPATKSTEVLEILDDNEHILGIRIVGGDHRLKNYSSTISLHSETIDGKTGTLAIESFVVDVPEGNTKEETCFFVEALIQCNLNSLADVTERLQAESM 6nwk A 1.65 BS02 DEX A 1 M29 L32 N33 Q39 M70 M73 F92 Q111 F204 C205 T208 M32 L35 N36 Q42 M73 M76 F95 Q114 F207 C208 T211 Ki=20nM remove_due_to_license_issue 31391291 301 FPTLISLLEVIEPEVLYSGYDSTLPDTSTRLMSTLNRLGGRQVVSAVKWAKALPGFRNLHLDDQMTLLQYSWMSLMAFSLGWRSYKQSNGNMLCFAPDLVINEERMQLPYMYDQCQQMLKISSEFVRLQVSYDEYLCMKVLLLLSTVPKDGLKSQAVFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEMVGGLLQFCFYTFVNKSLSVEFPEMLAEIISNQLPKFKAGSVKPLLFHQK 6nwl A 1.595 BS02 HCY A 1 M29 L32 N33 G36 Q39 M70 F92 Q111 F204 C205 T208 M32 L35 N36 G39 Q42 M73 F95 Q114 F207 C208 T211 Ki=43nM remove_due_to_license_issue 31391291 301 FPTLISLLEVIEPEVLYSGYDSTLPDTSTRLMSTLNRLGGRQVVSAVKWAKALPGFRNLHLDDQMTLLQYSWMSLMAFSLGWRSYKQSNGNMLCFAPDLVINEERMQLPYMYDQCQQMLKISSEFVRLQVSYDEYLCMKVLLLLSTVPKDGLKSQAVFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEMVGGLLQFCFYTFVNKSLSVEFPEMLAEIISNQLPKFKAGSVKPLLFHQK 6nxz A 1.75 BS01 D49 A 1 Q67 I68 Q46 I47 K32 Q67 I68 Y69 K11 Q46 I47 Y48 1.5.1.3 0004146,0009410 Ki=3.5uM remove_due_to_license_issue P00383 31460098 101 ATFGMGDRVRKKSGAAWQGQIVGWYCTNLTPEGYAVESEAHPGSVQIYPVAALERI 6ny0 A 1.4 BS01 LBA A 1 Q67 I68 Q47 I48 1.5.1.3 0004146,0009410 Ki=4uM remove_due_to_license_issue P00383 31460098 101 DATFGMGDRVRKKSGAAWQGQIVGWYCTNLTPEGYAVESEAHPGSVQIYPVAALERIN 6ny4 A 2.33 BS01 Z3A A 1 L828 A853 M902 E903 Y904 L905 G908 L956 L14 A39 M84 E85 Y86 L87 G90 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 ic50~3nM remove_due_to_license_issue IC50=3.0nM P52333 30891131 4000 TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLW 6ny5 A 3.002 BS01 rna C 0 Q162 F163 S166 R169 Y203 N206 K239 N240 W243 Q246 F277 N279 Y280 Q283 R315 R318 E322 Q66 F67 S70 R73 Y107 N110 K143 N144 W147 Q150 F181 N183 Y184 Q187 R219 R222 E226 ? 0003723 remove_due_to_license_issue O60059 31294800 -1 ~ 12 SEFELRRQACGRSQLLKSRVDILEVARQFEMRINLDIVDSMIASAIENNKVATEILPPVETLRSRQFEASKLREIRKNIDSGFYTQEEIEVIARSMLDDVAELSSDYLGNTVVQKFFEYCSDPIKEAMLERIAPYLAAIGIHKNGTWAAQKIIDVASTEKQMDLIVKHLRPYTALLYFDQFGNYVAQCCLRFKYPKNTFLFEVMARHCCEIGQSRFGARAIRACLENENATFEQQALVVASIIINSHLLATNSNGMLLLTWLLDNSFFRNRHRLLAIHLATHLHTTCTHKLASTLIFKLINNKQEPESRNLLLKNLFFSEKDNVLTYILQDQAVGPSFIHKVITYPSIGREFLAQFHLVIKRVLINIHAQPNAVYCRLMEEVGMTS 6ny5 B 3.002 BS01 rna C 0 N206 N240 W243 Q246 F277 N279 Y280 R311 R315 N101 N135 W138 Q141 F172 N174 Y175 R206 R210 ? 0003723 remove_due_to_license_issue O60059 31294800 -1 ~ 12 SEFELRRQACGRSQLLKSRVDILEVARQFEMRINLDIVDSMIASAIENNKVATEILPFEASKLREIRKNIDSGFYTQEEIEVIARSMLDDVAELSSDYLGNTVVQKFFEYCSDPIKEAMLERIAPYLAAIGIHKNGTWAAQKIIDVASTEKQMDLIVKHLRPYTALLYFDQFGNYVAQCCLRFKYPKNTFLFEVMARHCCEIGQSRFGARAIRACLENENATFEQQALVVASIIINSHLLATNSNGMLLLTWLLDNSFFRNRHRLLAIHLATHLHTTCTHKLASTLIFKLINNKQEPESRNLLLKNLFFSEKDNVLTYILQDQAVGPSFIHKVITYGREFLAQFHLVIKRVLINIHAQPNAVYCRLMEEV 6nyh A 2.1 BS01 L8D A 1 I43 K45 M67 V75 V76 L78 L90 M92 H136 D156 L157 I26 K28 M50 V58 V59 L61 L73 M75 H119 D139 L140 D138 K140 E142 N143 D156 T189 D121 K123 E125 N126 D139 T160 2.7.11.1 0004672,0005524,0006468 Ki=21nM remove_due_to_license_issue Q13546 31101885 301 NVIKMKSSDFLEKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNEGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 6nyv B 2.425 BS01 LBD B 1 D484 I485 A486 Q488 G526 N527 L531 P651 L659 G688 D25 I26 A27 Q29 G67 N68 L72 P179 L187 G216 5.6.1.1 0005524,0016887 ic50=0.21uM remove_due_to_license_issue Q8I0P1 30875216 802 GVEQKLVQLILDEIVEGGAKVEWTDIAGQDVAKQALQEMVILPSVRPELFTGLRAPAKGLLLFGPPGNGKTLLARAVATECSATFLNISAASLTSKYDGEKLVRALFAVARHMQPSIIFIDEVDSLLASRRLKTEFLVEFDGLPGNGDRIVVLAATNRPQELDEAALRRFTKRVYVSLPDEQTRELLLNRLLQKQGSPLDTEALRRLAKITDGYSGSDLTALAKDAALEPIRELNVEQVKCLDISAMRAITEQDFHSSLKRIRRSVAPQSLNSYEKWSQDYGD 6nyw B 2.189 BS01 L8M B 1 D484 I485 A486 G487 Q488 G526 C527 L531 P651 T655 R662 G688 D25 I26 A27 G28 Q29 G67 C68 L72 P175 T179 R186 G212 5.6.1.1 0005524,0016887 ic50=0.23uM remove_due_to_license_issue Q8I0P1 30875216 802 GVEQKLVQLILDEIVEGGAKVEWTDIAGQDVAKQALQEMVILPSVRPELFTGLRAPAKGLLLFGPPGCGKTLLARAVATECSATFLNISAASLTSKYDGEKLVRALFAVARHMQPSIIFIDEVDSLLSRRLKTEFLVEFDGLPDRIVVLAATNRPQELDEAALRRFTKRVYVSLPDEQTRELLLNRLLQKQGSPLDTEALRRLAKITDGYSGSDLTALAKDAALEPIRELNVEQVKCLDISAMRAITEQDFHSSLKRIRRSVAPQSLNSYEKWSQDYGD 6nze A 1.96 BS01 L8Y A 1 V603 K642 T687 E688 Y689 V690 G693 R738 L741 S758 V23 K35 T80 E81 Y82 V83 G86 R131 L134 S151 N734 R738 N739 D759 N127 R131 N132 D152 2.7.10.2 0004672,0005524,0006468 ic50=0.0013uM remove_due_to_license_issue IC50=1.3nM P29597 31314518 901 FHRVDQKEITQLSHLGQGTRTNVYEGRLRLRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTIL 6nzf A 2.39 BS01 L91 A 1 L595 V603 V640 K642 T687 E688 Y689 V690 G693 R738 L741 S758 L16 V24 V34 K36 T79 E80 Y81 V82 G85 R130 L133 S150 N734 R738 N739 D759 N126 R130 N131 D151 2.7.10.2 0004672,0005524,0006468 ic50=0.00092uM remove_due_to_license_issue IC50=63nM P29597 31314518 901 SFHRVDQKEITQLSHLGQGTRTNVYEGRLRLRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPLATLTSQCLTYEPTQRPSFRTILRD 6nzg A 2.43 BS01 L9D A 1 D166 H363 N425 E426 Y495 Y499 E526 W573 N591 K593 D135 H332 N394 E395 Y464 Y468 E495 W542 N560 K562 D166 H329 H363 I388 I390 E426 Y495 E526 S586 I590 K593 D135 H298 H332 I357 I359 E395 Y464 E495 S555 I559 K562 3.2.1.23,3.2.1.31 0004553,0005975 remove_due_to_license_issue A0A414F142 31774274 901 QRQTQTINDSWKFLKGECTAAADSAFDDSKWTSIHLPHTWNTDAYTEKDYYRGTGWYRRQLTLPQGWKEKQIILRLDAAGKSATIYINGKNVGEHAGGYTACSFNITPFLSFDTPNTLAVCVDNARQDIAPISGDFTFFGGIYRDVWLTAVPNQHFNLTNHGSDGLFISTPQVSEEQATLSIRGEVKNDAPEKATLELTHTIYRPDGTLLQTLKKNIQLKAGETYAFSNEATPVLKPELWTPETPRLYRVETTLRNRKTKTLLDQSNHYTAFRWFRFDGDEGFFLNGKPYKLRGICRHQDQKPIGPALTDEMHRRDFLLMKEMGANFIRISHYPQDDALLEMCDKLGMLAWEEIPIIDIVPNTPGYGDNCERNLREMIRQHYNHPSIITWGYMNEILLVTQRKYKTEAELKPVLERTLALANRLERVLKEEDSTRISTMAFHGSNSYNETGLSKITDIVGWNLYQGWYGGDLTGFEKFLAQQHQNHPTHPMIVSEYGAGSDKRLHSLHPRAFDFSIEYQQKYLEHYLPVLEDTPYICGGTHWNFIDFSSALRDESMPRINNKGLVYADRTPKDVYHYYQAAWRKDIPVLHIASRDWTDRAGVQQGNAPVYLPVKIYTNLSEVELFIDGISLGKQKTENYTATFEVPFSNRNPFLFAQGNYQGKTVQDGLRINFTPIPACLDANNLKGLELAVNVGSQCFFTSDESQLTWLPDQPYAAGSWGYIGGKEGTAQTEIQNTADGPLFQTLRNEIEGYRFDAPQGVYEIELLFTDIFRESTFGISINGEVVEESLSPCKESGYFRALRKKYYITNDKEYIDIRFHSTSGTCFLNGIKLRNIY 6nzh A 2.73 BS01 L9A A 1 L595 G596 V603 V640 K642 T687 E688 Y689 V690 E691 G693 R738 L741 S758 L15 G16 V23 V32 K34 T79 E80 Y81 V82 E83 G85 R130 L133 S150 N734 R738 N739 D759 N126 R130 N131 D151 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue IC50=390nM P29597 31314518 4000 FHRVDQKEITQLSHLGQGTRTNVYEGRLLRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDL 6nzk A 2.8 BS01 MJJ A 1 N27 K29 K81 S83 L85 L86 S87 W90 N13 K15 K67 S69 L71 L72 S73 W76 ? 0003700,0006355,0016020,0019031,0019062,0019064,0020002,0039654,0044173,0046718,0046813,0055036,0075509 remove_due_to_license_issue Q696P8 31160783 9999 VIGDLKCTSDNINDKDTGPPPISTDTVDVTNGLGTYYVLDRVYLNTTLFLNGYYPTSGSTYRNMALKGSVLLSRLWFKPPFLSDFINGIFAKVKNTKVIKDRVMYSEFPAITIGSTFVNTSYSVVVQPRTINKLQGLLEVSVCQYNMCEYPQTICHPNLGNHRKELWHLDTGVVSCLYKRNFTYDVNADYLYFHFYQEGGTFYAYFTDTGVVTKFLFNVYLGMALSHYYVMPLTCNSKLTLEYWVTPLTSRQYLLAFNQDGIIFNAVDCMSDFMSEIKCKTQSIAPPTGVYELNGYTVQPIADVYRRKPNLPNCNIEAWLNDKSVPSPLNWERKTFSNCNFNMSSLMSFIQADSFTCNNIDAAKIYGMCFSSITIDKFAIPNGRKVDLQLGNLGYLQSFNYRIDTTATSCQLYYNLPAANVSVSRFNPSTWNKRFGFIEDSVFKPRPAGVLTNHDVVYAQHCFKAPKNFCPCKLNNGIGTCPAGTNYLTCTPDPITFTGTYKCPQTKSLVGIGEHCSGLAVKSDYCGGNSCTCRPQAFLGWSADSCLQGDKCNIFANFILHDVNSGLTCSTDLQKANTDIILGVCVNYDLYGILGQGIFVEVNATYYNSWQNLLYDSNGNLYGFRDYITNRTFMIRSCYSGRVSAAFHANSSEPALLFRNIKCNYVFNNSLTRQLQPINYFDSYLGCVVNAYNSTAISVQTCDLTVGSGYCVDYSTTGYRFTNFEPFTVNSVNDSLEPVGGLYEIQIPSEFTIGNMVEFIQTSSPKVTIDCAAFVCGDYAACKSQLVEYGSFCDNINAILTEVNELLDTTQLQVANSLMNGVTLSTKLKDGVNFNVDDINFSPVLGCLGSASSRSAIEDLLFDKVKLSDVGFVEAYNNCTGGAEIRDLICVQSYKGIKVLPPLLSENQFSGYTLAATSASLFPPWTAAAGVPFYLNVQYRINGLGVTMDVLSQNQKLIANAFNNALYAIQEGFDATNSALVKIQAVVNANAEALNNLLQQLSNRFGAISASLQEILSRLDALEAEAQIDRLINGRLTALNAYVSQQLSDSTLVKFSAAQAMEKVNECVKSQSSRINFCGNGNHIISLVQNAPYGLYFIHFSYVPTKYVTARVSPGLCIAGDRGIAPKSGYFVNVNNTWMYTGSGYYYPEPITENNVVVMSTCAVNYTKAPYVMLN 6nzm A 1.72 BS01 L9S A 1 L408 F413 V416 A428 I432 M477 L528 D539 L542 V546 L14 F19 V22 A34 I38 M81 L132 D143 L146 V150 D521 R525 N526 D539 D125 R129 N130 D143 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.001uM remove_due_to_license_issue IC50=<100nM Q06187 31138459 701 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6nzp A 2.35 BS01 LB7 A 1 L595 Q597 V603 V640 K642 T687 E688 Y689 V690 E691 H692 G693 R738 L741 L16 Q18 V24 V35 K37 T82 E83 Y84 V85 E86 H87 G88 R133 L136 N734 R738 N739 D759 N129 R133 N134 D154 2.7.10.2 0004672,0005524,0006468 ic50=0.2nM remove_due_to_license_issue P29597 31318208 901 SFHRVDQKEITQLSHLGQGTRTNVYEGRLRELRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPGSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLTRL 6nzp B 2.35 BS01 LB7 B 1 L595 Q597 V603 V640 K642 T687 E688 Y689 V690 E691 G693 R738 L741 S758 L16 Q18 V24 V37 K39 T84 E85 Y86 V87 E88 G90 R135 L138 S155 N734 R738 N739 D759 N131 R135 N136 D156 2.7.10.2 0004672,0005524,0006468 ic50=0.2nM remove_due_to_license_issue P29597 31318208 901 SFHRVDQKEITQLSHLGQGTRTNVYEGRLRVQELRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPLSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLTR 6nzq A 2.11 BS01 LB4 A 1 L595 G598 V603 V640 K642 T687 E688 Y689 V690 E691 G693 R738 N739 L741 S758 L16 G19 V24 V35 K37 T82 E83 Y84 V85 E86 G88 R133 N134 L136 S153 N734 R738 N739 D759 N129 R133 N134 D154 2.7.10.2 0004672,0005524,0006468 ic50=0.3nM remove_due_to_license_issue IC50=180nM P29597 31318208 4000 SFHRVDQKEITQLSHLGQGTRTNVYEGRLRELRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLT 6nzr A 2.56 BS01 LAJ A 1 L595 V603 V640 K642 T687 E688 Y689 V690 G693 L741 L18 V26 V37 K39 T84 E85 Y86 V87 G90 L138 N734 R738 N739 D759 N131 R135 N136 D156 2.7.10.2 0004672,0005524,0006468 remove_due_to_license_issue P29597 31318208 901 QLSFHRVDQKEITQLSHLGQGTRTNVYEGRLRELRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPGLSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLT 6nzt A 1.4 BS01 L9P A 1 Q1041 H1057 D1081 L1135 G1137 S1139 F1154 R1155 A1156 A1157 Q53 H69 D93 L147 G149 S151 F166 R167 A168 A169 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue S4UY05 31133531 1201 KGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVQFIPVESLETTM 6nzv A 1.55 BS01 L9J A 1 Q1041 F1043 H1057 V1078 D1081 R1123 L1135 G1137 S1139 F1154 R1155 A1156 A1157 Q53 F55 H69 V90 D93 R135 L147 G149 S151 F166 R167 A168 A169 3.4.21.98,3.6.1.15,3.6.4.13 0006508,0008236,0019087 remove_due_to_license_issue S4UY05 31133531 1201 KGSVVIVGRINLSGDTAYAQQTRGEEGCQETSQTGRDKNQVEGEVQIVSTATQTFLATSINGVLWTVYHGAGTRTIASPKGPVTQMYTNVDKDLVGWQAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVSTRGVAKAVQFIPVESLETTM 6o0h A 3.67 BS01 LBG A 1 M278 Y307 I340 G341 G342 F347 T353 F354 I357 R378 R379 G380 M277 Y306 I339 G340 G341 F346 T352 F353 I356 R377 R378 G379 2.3.3.8 0003824,0003878,0005515,0005524,0005576,0005654,0005737,0005829,0006085,0006101,0006107,0006629,0006633,0006695,0008610,0015936,0016020,0016740,0035578,0046872,0046912,0070062,1904813 remove_due_to_license_issue P53396 30944472 2001 SAKAISEQTGKELLYKFICTTSAIQNRFKYARVTPDTDWARLLQDHPWLLSQNLVVKPDQLIKRRGKLGLVGVNLTLDGVKSWLKPRLGQEATVGKATGFLKNFLIEPFVPHSQAEEFYVCIYATREGDYVLFHHEGGVDVGDVDAKAQKLLVGVDEKLNPEDIKKHLLVHAPEDKKEILASFISGLFNFYEDLYFTYLEINPLVVTKDGVYVLDLAAKVDATADYICKVKWGDIEFPPPFGREAYPEEAYIADLDAKSGASLKLTLLNPKGRIWTMVAGGGASVVYSDTICDLGGVNELANYGEYSGAPSEQQTYDYAKTILSLMTREKHPDGKILIIGGSIANFTNVAATFKGIVRAIRDYQGPLKEHEVTIFVRRGGPNYQEGLRVMGEVGKTTGIPIHVFGTETHMTAIVGMALGHRPIPGKSTTLFSRHTKAIVWGMQTRAVQGMLDFDYVCSRDEPSVAAMVYPFTGDHKQKFYWGHKEILIPVFKNMADAMRKHPEVDVLINFASLRSAYDSTMETMNYAQIRTIAIIAEGIPEALTRKLIKKADQKGVTIIGPATVGGIKPGCFKIGNTGGMLDNILASKLYRPGSVAYVSRSGGMSNELNNIISRTTDGVYEGVAIGGDRYPGSTFMDHVLRYQDTPGVKMIVVLGEIGGTEEYKICRGIKEGRLTKPIVCWCIGTCATMFQASETAVAKNQALKEAGVFVPRSFDELGEIIQSVYEDLVANGVIVPAQEVPPPTVPMDYSWARELGLIRKPASFMTSICDERGQELIYAGMPITEVFKEEMGIGGVLGLLWFQKRLPKYSCQFIEMCLMVTADHGPAVSGAHNTIICARAGKDLVSSLTSGLLTIGDRFGGALDAAAKMFSKAFDSGIIPMEFVNKMKKEGKLIMGIGHRVKSINNPDMRVQILKDYVRQHFPATPLLDYALEVEKITTSKKPNLILNVDGLIGVAFVDMLRNCGSFTREEADEYIDIGALNGIFVLGRSMGFIGHYLDQKRLKQGLYRHPWDDISYVLPEHM 6o0k A 1.62 BS01 LBM A 1 A100 D103 F104 R107 Y108 D111 M115 L137 W144 G145 V148 E152 F153 Y202 A38 D41 F42 R45 Y46 D49 M53 L75 W82 G83 V86 E90 F91 Y140 ? 0042981,0043066 Ki=0.018nM remove_due_to_license_issue P10415,Q07817 31160589 301 YDNREIVMKYIHYKLSQRGYEWDAGDDSEVVHLTLRQAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 6o0m A 1.75 BS01 LBM A 1 A100 L104 F112 M115 E136 W144 G145 E152 F153 Y202 A38 L42 F50 M53 E74 W82 G83 E90 F91 Y140 ? 0042981,0043066 Ki=0.46nM remove_due_to_license_issue P10415,Q07817 31160589 301 GYDNREIVMKYIHYKLSQRGYEWDAGDSEVVHLTLRQAGDDLSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 6o0o A 1.998 BS01 F3Q A 1 F63 Y67 D70 F71 M74 R88 V92 E95 L96 G104 R105 A108 F112 F38 Y42 D45 F46 M49 R63 V67 E70 L71 G79 R80 A83 F87 ? 0042981,0043066 Ki=5.3nM remove_due_to_license_issue P10415,Q07817 31160589 201 YDNREIVMKYIHYKLSQRGYEWDAEVVHLTLRQAVDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 6o0p A 1.8 BS01 LBM A 1 A100 D103 F104 Y108 D111 M115 E136 W144 G145 V148 E152 F153 Y202 A38 D41 F42 Y46 D49 M53 E74 W82 G83 V86 E90 F91 Y140 ? 0042981,0043066 Ki=0.11nM remove_due_to_license_issue P10415,Q07817 31160589 301 YDNREIVMKYIHYKLSQRGYEWDAGDDSEVVHLTLRQAADDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYG 6o16 A 2.875 BS01 rna C 0 P302 R303 R304 R330 T345 D346 G347 V348 S374 Y376 G474 Q475 S588 T613 N614 V615 S619 K635 F648 R696 P772 R803 E804 R811 Q887 N946 H960 P961 F966 K967 L969 T981 K983 Y985 P72 R73 R74 R100 T115 D116 G117 V118 S144 Y146 G238 Q239 S263 T287 N288 V289 S293 K309 F322 R370 P433 R464 E465 R472 Q544 N595 H609 P610 F615 K616 L618 T630 K632 Y634 3.6.4.13 0003676,0005524 remove_due_to_license_issue Q6NZL1 30910870 1 ~ 10 VFIPVNRTPEMQEERLKLPILAEEQAIMEAVAEHPIVIVCGETGSGKTTQVPQFLYEAGYSSEDSIIGVTEPRRVAAVAMSQRVAKEMNLSHRVVSYQIRYEGNVTEETRIKFMTDGVLLKEIQKDFLLLKYKVVIIDEAHERSVYTDILLGLLSRIVALRAKRHLPLKLLIMSATLRVEDFTQNQRLFTTPPPVIKVESRFPVTVHFNDDYSGECFRKVCKIHRMLPAGGILVFLTGQAEVHALCRRLRKAFLPLHVLPLYSLLAPEKQAQVFKPPPGTRLCVVATNVAETSLTIPGIKYVVDCGKVKKRYYDRVTGVSSFRVTWVSQASADQRAGRAGRTEPGHCYRLYSSAVFGDFEQFPPPEITRRPVEDLILQMKALSIEKVINFPFPTPPSVEALVAAEELLVALGALQAQLSCPITALGRTMSTFPVAPRYAKMLALSQQHGCLPYTIAIVAAMTVRELFEELDREKELAELKGRRARVAQMKRTWAGQGPSLKLGDLMVLLGAVGACEYAGCSPQFCQANGLRYKAMLEIRRLRGQLTTAVNAVCPEDPKMQPPTESQVTYLRQIMAAGLGDHLARRVQSLDPKWKNAYKTPLLDDPVFIHPSSVLFKELPEFVVYQEIVETTKMYMKGVSTVEIQWIPSLLPSYCQFDAPLEEPAPSYCPESGQVLCHRASVFYRVGWPLPAVQVDFPEGIDRYKYFAKFLLEGQVFRKLASFKSCLLSSPSTMLKTWARLQPRTETLLRALVAHKADSRDSLLAAWKKNPKYLLAEYCEWLPKAMHSDVEKNWPPTTD 6o16 B 2.875 BS01 rna D 0 P302 R303 R304 R330 T345 G347 V348 Y376 G474 Q475 S588 T613 N614 S619 K635 F648 P772 R803 E804 Q887 N946 H960 P961 F966 K967 T981 K983 Y985 P72 R73 R74 R100 T115 G117 V118 Y146 G241 Q242 S268 T290 N291 S296 K312 F325 P439 R470 E471 Q546 N595 H609 P610 F615 K616 T630 K632 Y634 3.6.4.13 0003676,0005524 remove_due_to_license_issue Q6NZL1 30910870 1 ~ 10 VFIPVNRTPEMQEERLKLPILAEEQAIMEAVAEHPIVIVCGETGSGKTTQVPQFLYEAGYSSEDSIIGVTEPRRVAAVAMSQRVAKEMNLSHRVVSYQIRYEGNVTEETRIKFMTDGVLLKEIQKDFLLLKYKVVIIDEAHERSVYTDILLGLLSRIVALRAKRHLPLKLLIMSATLRVEDFTQNQRLFTTPPPVIKVESFPVTVHFNKRTPLDYSGECFRKVCKIHRMLPAGGILVFLTGQAEVHALCRRLRKAFPSLPLHVLPLYSLLAPEKQAQVFKPPPRLCVVATNVAETSLTIPGIKYVVDCGKVKKRYYDRVTGVSSFRVTWVSQASADQRAGRAGRTEPGHCYRLYSSAVFGDFEQFPPPEITRRPVEDLILQMKALSIEKVINFPFPTPPSVEALVAAEELLVALGALQAQMSQLSCPITALGRTMSTFPVAPRYAKMLALSQQHGCLPYTIAIVAAMTVRELFEELDLAELKGRRARVAQMKRTWAGQGPSLKLGDLMVLLGAVGACEYAGCSPQFCQANGLRYKAMLEIRRLRGQLTTAVNAVCPPKMQPPTESQVTYLRQIMAAGLGDHLARRVQSLDPKWKNAYKTPLLDDPVFIHPSSVLFKELPEFVVYQEIVETTKMYMKGVSTVEIQWIPSLLPSYCQFDAPLEEPAPSYCPESGQVLCHRASVFYRVGWPLPAVQVDFPEGIDRYKYFAKFLLEGQVFRKLASFKSCLLSSPSTMLKTWARLQPRTETLLRALVAHKADSRDSLLAAWKKNPKYLLAEYCEWLPKAMHSDVEKNWPPTT 6o2p A 3.3 BS06 VX7 A 1 F305 A309 F312 F931 F932 F305 A309 F312 F687 F688 5.6.1.6 0003689,0005254,0005260,0005515,0005524,0005634,0005737,0005765,0005768,0005769,0005783,0005789,0005829,0005886,0006338,0006695,0006811,0006821,0006904,0009986,0010008,0015106,0015108,0015701,0016020,0016324,0016853,0016887,0017081,0019869,0019899,0030165,0030301,0030660,0030669,0031901,0032991,0034220,0034707,0034976,0035377,0035774,0042626,0043225,0045921,0048240,0050891,0051087,0051454,0051649,0055037,0055038,0055085,0060081,0061775,0070175,0071320,0071889,0097186,0106138,0140359,0140584,0140588,0140665,0140849,1902161,1902476,1902943,1904322 remove_due_to_license_issue EC50=236nM P13569 31221859 1512 MQRSPLEKASVVSKLFFSWTRPILRKGYRQRLELSDIYQIPSVDSADNLSEKLEREWDRELASKKNPKLINALRRCFFWRFMFYGIFLYLGEVTKAVQPLLLGRIIASYDPDNKEERSIAIYLGIGLCLLFIVRTLLLHPAIFGLHHIGMQMRIAMFSLIYKKTLKLSSRVLDKISIGQLVSLLSNNLNKFDEGLALAHFVWIAPLQVALLMGLIWELLQASAFCGLGFLIVLALFQAGLGRMMMKYRDQRAGKISERLVITSEMIENIQSVKAYCWEEAMEKMIENLRQTELKLTRKAAYVRYFNSSAFFFSGFFVVFLSVLPYALIKGIILRKIFTTISFCIVLRMAVTRQFPWAVQTWYDSLGAINKIQDFLQKQEYKTLEYNLTTTEVVMENVTAFWEEGFGELFGTPVLKDINFKIERGQLLAVAGSTGAGKTSLLMVIMGELEPSEGKIKHSGRISFCSQFSWIMPGTIKENIIFGVSYDEYRYRSVIKACQLEEDISKFAEKDNIVLGEGGITLSGGQRARISLARAVYKDADLYLLDSPFGYLDVLTEKEIFESCVCKLMANKTRILVTSKMEHLKKADKILILHEGSSYFYGTFSELQNLQTWNTYLRYITVHKSLIFVLIWCLVIFLAEVAASLVVLWLLGNTPLNNSYAVIITSTSSYYVFYIYVGVADTLLAMGFFRGLPLVHTLITVSKILHHKMLHSVLQAPMSTLNTLKAGGILNRFSKDIAILDDLLPLTIFDFIQLLLIVIGAIAVVAVLQPYIFVATVPVIVAFIMLRAYFLQTSQQLKQLESEGRSPIFTHLVTSLKGLWTLRAFGRQPYFETLFHKALNLHTANWFLYLSTLRWFQMRIEMIFVIFFIAVTFISILTTGEGEGRVGIILTLAMNIMSTLQWAVNSSIDVDSLMRSVSRVFKFIDMPTEGDIWPSGGQMTVKDLTAKYTEGGNAILENISFSISPGQRVGLLGRTGSGKSTLLSAFLRLLNTEGEIQIDGVSWDSITLQQWRKAFGVIPQKVFIFSGTFRKNLDPYEQWSDQEIWKVADEVGLRSVIEQFPGKLDFVLVDGGCVLSHGHKQLMCLARSVLSKAKILLLDQPSAHLDPVTYQIIRRTLKQAFADCTVILCEHRIEAMLECQQFLVIEENKVRQYDSIQKLLNERSLFRQAISPSDRVKLFP 6o4w A 2.35 BS01 E20 A 1 Y72 W86 Y124 E202 W286 F295 Y337 F338 Y341 Y69 W83 Y121 E199 W283 F292 Y334 F335 Y338 G121 G122 S203 A204 E334 H447 G118 G119 S200 A201 E331 H444 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue IC50=10.0nM, Ki=20.5nM, EC50=43nM P22303 31176713 604 EDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPGGTGGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDPKAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSAT 6o4x A 2.3 BS01 AA A 1 W86 G121 E202 Y337 W439 H447 W83 G118 E199 Y334 W436 H444 G121 G122 S203 A204 E334 H447 G118 G119 S200 A201 E331 H444 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue P22303 31176713 605 EDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPGGTGGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDPKAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSAT 6o50 A 2.352 BS01 EBW A 1 Y72 W86 E202 S203 W286 F297 Y337 F338 Y341 H447 Y69 W83 E199 S200 W283 F294 Y334 F335 Y338 H444 G121 G122 S203 A204 E334 H447 G118 G119 S200 A201 E331 H444 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Ki=10nM, IC50=30nM P22303 31176713 601 EDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPGGTGGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDPKAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSAT 6o50 B 2.352 BS01 EBW B 1 Y72 W86 Y124 E202 S203 W286 F297 Y337 F338 Y341 H447 Y69 W83 Y121 E199 S200 W283 F294 Y334 F335 Y338 H444 G121 G122 S203 A204 E334 H447 G118 G119 S200 A201 E331 H444 3.1.1.7 0001507,0001540,0001919,0002076,0003990,0004104,0005515,0005518,0005576,0005604,0005615,0005634,0005794,0005886,0006581,0007155,0007399,0007416,0009986,0016020,0016787,0017171,0031594,0031623,0032223,0042166,0042802,0042803,0042982,0043083,0043236,0045202,0048471,0050714,0052689,0060041,0095500,0098552,0120162 remove_due_to_license_issue Ki=10nM, IC50=30nM P22303 31176713 601 EDAELLVTVRGGRLRGIRLKTPGGPVSAFLGIPFAEPPMGPRRFLPPEPKQPWSGVVDATTFQSVCYQYVDTLYPGFEGTEMWNPNRELSEDCLYLNVWTPYPRPTSPTPVLVWIYGGGFYSGASSLDVYDGRFLVQAERTVLVSMNYRVGAFGFLALPGSREAPGNVGLLDQRLALQWVQENVAAFGGDPTSVTLFGESAGAASVGMHLLSPPSRGLFHRAVLQSGAPNGPWATVGMGEARRRATQLAHLVGCPPGGTGGNDTELVACLRTRPAQVLVNHEWHVLPQESVFRFSFVPVVDGDFLSDTPEALINAGDFHGLQVLVGVVKDEGSYFLVYGAPGFSKDNESLISRAEFLAGVRVGVPQVSDLAAEAVVLHYTDWLHPEDPARLREALSDVVGDHNVVCPVAQLAGRLAAQGARVYAYVFEHRASTLSWPLWMGVPHGYEIEFIFGIPLDPSRNYTAEEKIFAQRLMRYWANFARTGDPNEPRDPKAPQWPPYTAGAQQYVSLDLRPLEVRRGLRAQACAFWNRFLPKLLSAT 6o5g A 1.89 BS01 LMJ A 1 L106 M110 M125 F142 M145 M146 L102 M106 M121 F138 M141 M142 ? 0000086,0000922,0002027,0005509,0005513,0005515,0005576,0005634,0005654,0005737,0005813,0005819,0005829,0005856,0005876,0005886,0007186,0008076,0010800,0010801,0010856,0010880,0010881,0016020,0016240,0019855,0019901,0021762,0030017,0031432,0031514,0031954,0031982,0032465,0032991,0034704,0035458,0043209,0043539,0044305,0044325,0046427,0046872,0048306,0050848,0051592,0055117,0060314,0060315,0060316,0071346,0071902,0072542,0097225,0097720,0098901,0099523,0140056,0140238,1901842,1901844,1902494,1905913,1990456 Kd=2uM remove_due_to_license_issue P0DP23 31337679 201 LTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMT 6o5t A 2.1 BS03 L8J A 1 F62 Y67 R205 N210 H240 F32 Y37 R175 N180 H210 H114 H116 D118 H179 C198 Y201 N210 H240 H84 H86 D88 H149 C168 Y171 N180 H210 3.5.2.6 0016787,0017001,0042597,0046677,0046872 Ki=0.316uM remove_due_to_license_issue Q9K2N0 31483651 503 GEYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRS 6o5u A 1.4 BS01 KAN A 1 Y85 E86 D136 D183 H189 S225 N226 Y67 E68 D118 D165 H171 S207 N208 2.3.1.81 0008080,0016746,0046353,0046677,0046872 Kd=42uM remove_due_to_license_issue Q47030 31515870 301 TPWSKSELVRQLRDLGVRSGDMVMPHVSLRAVGPLADGPQTLVDALIEAVGPTGNILAFVSWRDSPYEQTLGHDAPPAAIAQSWPAFDPDHAPAYPGFGAINEFIRTYPGCRRSAHPDASMAAIGPDAAWLVAPHEMGAAYGPRSPIARFLAHAGKILSIGAGPDAVTALHYAEAVARIEGKRRVTYSMPLLREGKRVWVTTSDWDSNGILDEYAAPDGPDAVERIARDYLARTRVAQGPVGGAQSRLIDAADIVSFGIEWLEARHAA 6o68 A 2.78 BS01 LO4 A 1 G284 C285 R288 I341 M364 G69 C70 R73 I126 M149 ? 0003677,0004879,0005634,0006355 remove_due_to_license_issue P37231 31611383 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 6o6f A 1.6 BS01 LOD A 1 F228 V249 M250 V253 R263 T266 L267 F270 F58 V79 M80 V83 R93 T96 L97 F100 ? 0042981 ic50=0.04uM remove_due_to_license_issue IC50=40nM Q07820 30254093 401 SDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6o6g A 2.4 BS01 LOJ A 1 M231 M250 V253 R263 L267 F270 M55 M74 V77 R87 L91 F94 ? 0042981 ic50=0.3uM remove_due_to_license_issue IC50=300nM Q07820 30254093 401 DELYRQSLEIISRYLREQATGAKDRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6o8i A 1.42 BS01 LTJ A 1 A428 Y476 M477 G480 C481 V546 L547 A38 Y78 M79 G82 C83 V148 L149 D521 R525 N526 D539 D123 R127 N128 D141 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue Q06187 30893553 4000 GYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEE 6o8u A 1.8 BS01 LS7 A 1 M192 G193 V200 A211 Y262 M265 P266 G268 L318 M29 G30 V37 A48 Y93 M96 P97 G99 L149 D311 K313 A315 N316 D329 T351 D142 K144 A146 N147 D160 T176 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=5.3nM remove_due_to_license_issue IC50=3.6nM, Ki=5.00nM Q9NWZ3 31082230 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLTTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6o94 A 1.98 BS01 LRS A 1 I185 M192 G193 E194 V200 A211 Y262 Y264 M265 P266 G268 L318 I23 M30 G31 E32 V38 A49 Y100 Y102 M103 P104 G106 L156 D311 K313 A315 N316 D329 T351 D149 K151 A153 N154 D167 T185 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=7.4nM remove_due_to_license_issue IC50=97nM, Ki=1.8nM Q9NWZ3 31082230 502 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6o95 A 1.77 BS01 LSV A 1 M192 G193 V200 A211 Y262 M265 P266 G268 L318 M31 G32 V39 A50 Y99 M102 P103 G105 L155 D311 K313 A315 N316 D329 T351 D148 K150 A152 N153 D166 T183 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=5.1nM remove_due_to_license_issue Ki=5.1nM, IC50=400nM Q9NWZ3 31082230 502 DTRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA 6o96 A 3.5 BS01 dna I 0 R40 Y41 V46 R49 R63 K64 L65 P66 R69 R4 Y5 V10 R13 R27 K28 L29 P30 R33 ? 0000786,0003677,0005515,0005634,0005654,0005694,0030527,0046982 remove_due_to_license_issue P84233 30981630 2 ~ 147 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGER 6o96 A 3.5 BS02 dna J 0 Y41 R42 R72 R83 F84 R116 V117 T118 M120 Y5 R6 R36 R47 F48 R80 V81 T82 M84 ? 0000786,0003677,0005515,0005634,0005654,0005694,0030527,0046982 remove_due_to_license_issue P84233 30981630 1 ~ 146 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGER 6o96 B 3.5 BS01 dna I 0 R35 R45 I46 G48 R78 K79 T80 R18 R28 I29 G31 R61 K62 T63 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 30981630 2 ~ 147 HRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFG 6o96 B 3.5 BS02 dna J 0 P32 R36 R45 P15 R19 R28 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 30981630 1 ~ 146 HRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFG 6o96 C 3.5 BS01 dna I 0 R29 R42 V43 G44 A45 K75 T76 R77 R18 R31 V32 G33 A34 K64 T65 R66 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 30981630 2 ~ 147 AKAKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPK 6o96 C 3.5 BS02 dna J 0 K15 R17 R20 R32 R77 K4 R6 R9 R21 R66 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 30981630 1 ~ 146 AKAKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPK 6o96 D 3.5 BS01 dna I 0 R33 K34 I39 Y40 R2 K3 I8 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 30981630 2 ~ 147 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTCYTSA 6o96 D 3.5 BS02 dna J 0 T32 Y42 S56 S87 T88 T1 Y11 S25 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 30981630 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTCYTSA 6o96 E 3.5 BS01 dna I 0 Y41 R42 T45 R72 R83 F84 R116 V117 T118 Y5 R6 T9 R36 R47 F48 R80 V81 T82 ? 0000786,0003677,0005515,0005634,0005654,0005694,0030527,0046982 remove_due_to_license_issue P84233 30981630 2 ~ 147 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGER 6o96 E 3.5 BS02 dna J 0 H39 R40 Y41 G44 V46 R49 K56 R63 K64 L65 P66 R69 H3 R4 Y5 G8 V10 R13 K20 R27 K28 L29 P30 R33 ? 0000786,0003677,0005515,0005634,0005654,0005694,0030527,0046982 remove_due_to_license_issue P84233 30981630 1 ~ 146 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEASEAYLVALFEDTNLCAIHAKRVTIMPKDIQLARRIRGER 6o96 F 3.5 BS01 dna I 0 P32 R36 R45 P15 R19 R28 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 30981630 2 ~ 147 HRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFG 6o96 F 3.5 BS02 dna J 0 R35 R45 I46 S47 G48 R78 K79 T80 R18 R28 I29 S30 G31 R61 K62 T63 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P62799 30981630 1 ~ 146 HRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFG 6o96 G 3.5 BS01 dna I 0 K15 T16 R17 G28 R32 R77 K4 T5 R6 G17 R21 R66 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 30981630 2 ~ 147 AKAKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPK 6o96 G 3.5 BS02 dna J 0 R29 R42 V43 G44 A45 K75 T76 R77 R18 R31 V32 G33 A34 K64 T65 R66 ? 0000786,0003677,0005634,0005694,0030527,0046982 remove_due_to_license_issue P06897 30981630 1 ~ 146 AKAKTRSSRAGLQFPVGRVHRLLRKGNYAERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAVRNDEELNKLLGRVTIAQGGVLPNIQSVLLPK 6o96 H 3.5 BS01 dna I 0 T32 Y42 S55 S56 R86 S87 T88 T1 Y11 S24 S25 R55 S56 T57 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 30981630 2 ~ 147 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTCYTSA 6o96 H 3.5 BS02 dna J 0 R33 K34 Y40 R2 K3 Y9 ? 0000786,0003677,0005515,0005634,0005694,0030527,0046982 remove_due_to_license_issue P02281 30981630 1 ~ 146 TRKESYAIYVYKVLKQVHPDTGISSKAMSIMNSFVNDVFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTCYTSA 6o9d A 2.51 BS01 LTY A 1 M192 V200 A211 Y262 Y264 M265 P266 G268 A315 L318 M31 V39 A50 Y94 Y96 M97 P98 G100 A147 L150 D311 K313 A315 N316 D329 T351 D143 K145 A147 N148 D161 T179 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=41nM, Ki=2.0nM Q9NWZ3 31082230 501 DTRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6o9x A 1.7 BS01 M0S A 1 T725 I726 Q754 Y795 N869 F900 F902 T265 I266 Q294 Y335 N409 F440 F442 3.2.1.143 0004649,0005975,0006282 ic50=0.9uM remove_due_to_license_issue Q86W56 31827085 1001 DKKWLGTPIEEMRRMPRCGIRLPLLRPSANHTVTIRVDLLRAGEVPKPFPTHYKDLWDNKHVKMPCSEQNLYPVTAGSRWELIQTALLNKFTRPQNLKDAILKYNVAYSKKWDFTALIDFWDKVLEEAEAQHLYQSILPDMVKIALCLPNICTQPIPLLAAAMNHSITMSQEQIASLLANAFFCTFPRRNAKYSSYPDINFNRLFEGRSSRKPEKLKTLFCYFRRVTAAAPTGLVTFTRQSLEDFPEWERCEKPLTRLHVTYEGTIEENGQGMLQVDFANRFVGGGVTSAGLVQEEIRFLINPELIISRLFTEVLDHNECLIITGTEQYSEYTGYAETYRWSRSHEDGSERDDWQRRCTEIVAIDALHFRRYLDQFVPEKMRRELNKAYCGFLRPGVSSENLSAVATGNWGCGAFGGDARLKALIQILAAAAAERDVVYFTFGDSELMRDIYSMHIFLTERKLTVGDVYKLLLRYYNEECRNCSTPGPDIKLYPFIYHAVESC 6oa1 A 1.8 BS01 M0P A 1 T725 I726 E727 F738 Q754 Y795 N869 F900 F902 T262 I263 E264 F275 Q291 Y332 N406 F437 F439 3.2.1.143 0004649,0005975,0006282 ic50=25.7uM remove_due_to_license_issue Q86W56 31827085 1001 DKKWLGTPIEEMRRMPRCGIRLPLLRPSANHTVTIRVDLLRAGEVPKPFPTHYKDLWDNKHVKMPCSEQNLYPVTAGSRWELIQTALLNKFTRPQNLKDAILKYNVAYSKKWDFTALIDFWDKVLEEAEAQHLYQSILPDMVKIALCLPNICTQPIPLLAAAMNHSITMSQEQIASLLANAFFCTFPRRNSSYPDINFNRLFEGRSSRKPEKLKTLFCYFRRVTAAAPTGLVTFTRQSLEDFPEWERCEKPLTRLHVTYEGTIEENGQGMLQVDFANRFVGGGVTSAGLVQEEIRFLINPELIISRLFTEVLDHNECLIITGTEQYSEYTGYAETYRWSRSHEDGSERDDWQRRCTEIVAIDALHFRRYLDQFVPEKMRRELNKAYCGFLRPGVSSENLSAVATGNWGCGAFGGDARLKALIQILAAAAAERDVVYFTFGDSELMRDIYSMHIFLTERKLTVGDVYKLLLRYYNEECRNCSTPGPDIKLYPFIYHAVESC 6oa3 A 1.9 BS01 M0M A 1 I726 E727 F738 Q754 Y795 N869 C872 F900 F902 I263 E264 F275 Q291 Y332 N406 C409 F437 F439 3.2.1.143 0004649,0005975,0006282 ic50=0.4uM remove_due_to_license_issue Q86W56 31827085 1001 DKKWLGTPIEEMRRMPRCGIRLPLLRPSANHTVTIRVDLLRAGEVPKPFPTHYKDLWDNKHVKMPCSEQNLYPVTAGSRWELIQTALLNKFTRPQNLKDAILKYNVAYSKKWDFTALIDFWDKVLEEAEAQHLYQSILPDMVKIALCLPNICTQPIPLLAAAMNHSITMSQEQIASLLANAFFCTFPRRNSSYPDINFNRLFEGRSSRKPEKLKTLFCYFRRVTAAAPTGLVTFTRQSLEDFPEWERCEKPLTRLHVTYEGTIEENGQGMLQVDFANRFVGGGVTSAGLVQEEIRFLINPELIISRLFTEVLDHNECLIITGTEQYSEYTGYAETYRWSRSHEDGSERDDWQRRCTEIVAIDALHFRRYLDQFVPEKMRRELNKAYCGFLRPGVSSENLSAVATGNWGCGAFGGDARLKALIQILAAAAAERDVVYFTFGDSELMRDIYSMHIFLTERKLTVGDVYKLLLRYYNEECRNCSTPGPDIKLYPFIYHAVESC 6oac A 3.15 BS01 M1J A 1 M772 I800 K802 D810 I848 E849 V850 V851 I932 D933 M597 I625 K627 D635 I673 E674 V675 V676 I750 D751 2.7.11.1,2.7.1.137,2.7.1.153 0016301,0046854 remove_due_to_license_issue P42336 31244112 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSPNNDKQKYTLKINHDCVPEQVIAEAIRKKTRSYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRKSLWVINSALRIKILCATYVNIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVKEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSLRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKGFNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDRVPFVLTQDFLIVISTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDA 6oag F 2.3 BS01 M2Y F 1 K57 N59 F206 F239 D243 K50 N52 F199 F232 D236 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K193 F232 D236 D237 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=3.7uM remove_due_to_license_issue P14324 31577901 401 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6oag F 2.3 BS02 M2Y F 2 E318 Y322 Y349 K350 E311 Y315 Y342 K343 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K193 F232 D236 D237 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=3.7uM remove_due_to_license_issue P14324 31577901 402 DVYAQEKQDFVQHFSQIVRVLTEDEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6oah F 2.2 BS01 M2V F 1 N59 R60 F206 F239 Q242 K347 I348 K350 N52 R53 F199 F232 Q235 K340 I341 K343 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K50 F91 D96 D100 R105 D167 K193 F232 D236 D237 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=1.5uM remove_due_to_license_issue P14324 31577901 402 SDVYAQEKQDFVQHFSQIVRVLTEEMGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6ob0 A 2.81 BS01 M3D A 1 W82 V84 L263 W53 V55 L234 W82 S159 L160 D183 H268 W53 S130 L131 D154 H239 3.1.1.32,3.1.1.34 0004465,0004620,0004806,0005102,0005509,0005515,0005576,0005615,0005886,0006629,0006631,0006633,0006641,0006644,0008201,0008970,0009617,0009749,0009986,0010744,0010884,0010886,0010890,0016042,0016298,0016787,0019433,0031670,0032722,0032731,0032755,0032760,0034185,0034361,0034371,0034372,0034375,0042627,0042632,0042803,0043395,0043495,0045600,0046872,0050729,0052689,0052739,0055096,0070328,0071398,0071813,1902494,1904179,2000343 remove_due_to_license_issue P06858 31072929 503 QRRDFIDIESKFALRTPEDTAEDTCHLIPGVAESVATCHFNHSSKTFMVIHGWTVTGMYESWVPKLVAALYKREPDSNVIVVDWLSRAQEHYPVSAGYTKLVGQDVARFINWMEEEFNYPLDNVHLLGYSLGAHAAGIAGSLTNKKVNRITGLDPAGPNFEYAEAPSRLSPDDADFVDVLHTFTRGSPGRSIGIQKPVGHVDIYPNGGTFQPGCNIGEAIRVIAERGLGDVDQLVKCSHERSIHLFIDSLLNEENPSKAYRCSSKEAFEKGLCLSCRKNRCNNLGYEINKVRAKRSSKMYLKTRSQMPYKVFHYQVKIHFSGTESETHTNQAFEISLYGTVAESENIPFTLPEVSTNKTYSFLIYTEVDIGELLMLKLKWKSDSYFSWSDWWSSPGFAIQKIRVKAGETQKKVIFCSREKVSHLQKGKAPAVFVKCHDKSLN 6ob0 A 2.81 BS02 M3D A 2 W82 Y121 S159 K265 H268 W53 Y92 S130 K236 H239 W82 S159 L160 D183 H268 W53 S130 L131 D154 H239 3.1.1.32,3.1.1.34 0004465,0004620,0004806,0005102,0005509,0005515,0005576,0005615,0005886,0006629,0006631,0006633,0006641,0006644,0008201,0008970,0009617,0009749,0009986,0010744,0010884,0010886,0010890,0016042,0016298,0016787,0019433,0031670,0032722,0032731,0032755,0032760,0034185,0034361,0034371,0034372,0034375,0042627,0042632,0042803,0043395,0043495,0045600,0046872,0050729,0052689,0052739,0055096,0070328,0071398,0071813,1902494,1904179,2000343 remove_due_to_license_issue P06858 31072929 504 QRRDFIDIESKFALRTPEDTAEDTCHLIPGVAESVATCHFNHSSKTFMVIHGWTVTGMYESWVPKLVAALYKREPDSNVIVVDWLSRAQEHYPVSAGYTKLVGQDVARFINWMEEEFNYPLDNVHLLGYSLGAHAAGIAGSLTNKKVNRITGLDPAGPNFEYAEAPSRLSPDDADFVDVLHTFTRGSPGRSIGIQKPVGHVDIYPNGGTFQPGCNIGEAIRVIAERGLGDVDQLVKCSHERSIHLFIDSLLNEENPSKAYRCSSKEAFEKGLCLSCRKNRCNNLGYEINKVRAKRSSKMYLKTRSQMPYKVFHYQVKIHFSGTESETHTNQAFEISLYGTVAESENIPFTLPEVSTNKTYSFLIYTEVDIGELLMLKLKWKSDSYFSWSDWWSSPGFAIQKIRVKAGETQKKVIFCSREKVSHLQKGKAPAVFVKCHDKSLN 6ob0 A 2.81 BS04 M3D B 1 F415 W417 F386 W388 W82 S159 L160 D183 H268 W53 S130 L131 D154 H239 3.1.1.32,3.1.1.34 0004465,0004620,0004806,0005102,0005509,0005515,0005576,0005615,0005886,0006629,0006631,0006633,0006641,0006644,0008201,0008970,0009617,0009749,0009986,0010744,0010884,0010886,0010890,0016042,0016298,0016787,0019433,0031670,0032722,0032731,0032755,0032760,0034185,0034361,0034371,0034372,0034375,0042627,0042632,0042803,0043395,0043495,0045600,0046872,0050729,0052689,0052739,0055096,0070328,0071398,0071813,1902494,1904179,2000343 remove_due_to_license_issue P06858 31072929 503 QRRDFIDIESKFALRTPEDTAEDTCHLIPGVAESVATCHFNHSSKTFMVIHGWTVTGMYESWVPKLVAALYKREPDSNVIVVDWLSRAQEHYPVSAGYTKLVGQDVARFINWMEEEFNYPLDNVHLLGYSLGAHAAGIAGSLTNKKVNRITGLDPAGPNFEYAEAPSRLSPDDADFVDVLHTFTRGSPGRSIGIQKPVGHVDIYPNGGTFQPGCNIGEAIRVIAERGLGDVDQLVKCSHERSIHLFIDSLLNEENPSKAYRCSSKEAFEKGLCLSCRKNRCNNLGYEINKVRAKRSSKMYLKTRSQMPYKVFHYQVKIHFSGTESETHTNQAFEISLYGTVAESENIPFTLPEVSTNKTYSFLIYTEVDIGELLMLKLKWKSDSYFSWSDWWSSPGFAIQKIRVKAGETQKKVIFCSREKVSHLQKGKAPAVFVKCHDKSLN 6ob0 A 2.81 BS05 M3D B 2 W420 W421 W391 W392 W82 S159 L160 D183 H268 W53 S130 L131 D154 H239 3.1.1.32,3.1.1.34 0004465,0004620,0004806,0005102,0005509,0005515,0005576,0005615,0005886,0006629,0006631,0006633,0006641,0006644,0008201,0008970,0009617,0009749,0009986,0010744,0010884,0010886,0010890,0016042,0016298,0016787,0019433,0031670,0032722,0032731,0032755,0032760,0034185,0034361,0034371,0034372,0034375,0042627,0042632,0042803,0043395,0043495,0045600,0046872,0050729,0052689,0052739,0055096,0070328,0071398,0071813,1902494,1904179,2000343 remove_due_to_license_issue P06858 31072929 504 QRRDFIDIESKFALRTPEDTAEDTCHLIPGVAESVATCHFNHSSKTFMVIHGWTVTGMYESWVPKLVAALYKREPDSNVIVVDWLSRAQEHYPVSAGYTKLVGQDVARFINWMEEEFNYPLDNVHLLGYSLGAHAAGIAGSLTNKKVNRITGLDPAGPNFEYAEAPSRLSPDDADFVDVLHTFTRGSPGRSIGIQKPVGHVDIYPNGGTFQPGCNIGEAIRVIAERGLGDVDQLVKCSHERSIHLFIDSLLNEENPSKAYRCSSKEAFEKGLCLSCRKNRCNNLGYEINKVRAKRSSKMYLKTRSQMPYKVFHYQVKIHFSGTESETHTNQAFEISLYGTVAESENIPFTLPEVSTNKTYSFLIYTEVDIGELLMLKLKWKSDSYFSWSDWWSSPGFAIQKIRVKAGETQKKVIFCSREKVSHLQKGKAPAVFVKCHDKSLN 6oco A 2.58 BS01 M5V A 1 T750 M752 W760 V828 D832 M900 I910 T668 M670 W678 V746 D750 M807 I817 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue O00329 31757666 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPLPNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKAVEQPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEKAKDCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHTEEEQLQLREILERRYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSGGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKV 6ocq A 2.793 BS01 M5J A 1 L70 V76 H136 I154 A155 D156 L57 V63 H123 I141 A142 D143 D138 K140 E142 N143 D156 T189 D125 K127 E129 N130 D143 T157 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13546 31013427 301 NVIKMKSSDFLESAEGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 6ocu A 2.77 BS01 M5D A 1 T750 M752 W760 Y813 V828 M900 I910 T657 M659 W667 Y717 V732 M791 I801 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue O00329 31757666 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDESVSLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEDCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHSEEQLQLREILERLYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWK 6ocw H 2.6 BS01 M6M H 1 T1 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 A52 T1 S20 T21 Q22 S27 V31 K33 I45 G47 T48 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocw H 2.6 BS02 M6M N 1 S122 F123 D124 A125 G128 W129 N130 S122 F123 D124 A125 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocw I 2.6 BS01 M6M H 1 F123 D124 A125 G128 W129 F123 D124 A125 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocw I 2.6 BS02 M6M I 1 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 A52 T1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocw Y 2.6 BS01 M6M X 1 F123 D124 A126 G128 W129 F123 D124 A126 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 6ocw Y 2.6 BS02 M6M Y 1 T1 S20 T21 Q22 S27 K33 G47 A49 A52 T1 S20 T21 Q22 S27 K33 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 6ocz H 2.65 BS01 M6Y H 1 S20 T21 Q22 S27 V31 K33 I45 G47 A49 A52 S20 T21 Q22 S27 V31 K33 I45 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocz H 2.65 BS02 M6Y N 1 D124 A125 G128 W129 N130 D124 A125 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocz I 2.65 BS01 M6Y H 1 S122 D124 A126 G128 W129 N130 S122 D124 A126 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocz I 2.65 BS02 M6Y I 1 S20 T21 Q22 S27 V31 I45 G47 A49 A52 S20 T21 Q22 S27 V31 I45 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ocz Y 2.65 BS01 M6Y X 1 S122 F123 D124 A126 G128 W129 S122 F123 D124 A126 G128 W129 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 6ocz Y 2.65 BS02 M6Y Y 1 T1 S20 T21 Q22 S27 V31 G47 A49 A52 T1 S20 T21 Q22 S27 V31 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 6od6 A 2.0 BS01 M7D A 1 Q12 G13 L30 D32 Y71 F108 I118 D228 G230 T232 Q18 G19 L36 D38 Y77 F114 I124 D223 G225 T227 3.4.23.46 0004190,0006508,0016020 ic50=0.00000001M remove_due_to_license_issue P56817 31413800 401 TTGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVETSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6ode H 2.9 BS01 M9G H 1 S20 T21 Q22 V31 K33 I45 G47 A49 A52 S20 T21 Q22 V31 K33 I45 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ode H 2.9 BS02 M9G N 1 S122 F123 D124 A126 G128 W129 N130 S122 F123 D124 A126 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ode I 2.9 BS01 M9G H 1 S122 F123 D124 A126 G128 W129 N130 S122 F123 D124 A126 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ode I 2.9 BS02 M9G I 1 S20 T21 V31 K33 I45 G47 A49 A52 S20 T21 V31 K33 I45 G47 A49 A52 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRS 6ode Y 2.9 BS01 M9G X 1 S122 F123 D124 A126 G128 W129 N130 S122 F123 D124 A126 G128 W129 N130 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 6ode Y 2.9 BS02 M9G Y 1 S20 T21 Q22 V31 K33 I45 G47 A49 S20 T21 Q22 V31 K33 I45 G47 A49 3.4.25.1 0004298,0005839,0010498,0051603 remove_due_to_license_issue P9WHT9 31560200 301 TTIVALKYPGGVVMAGDRRSTQGNMISGRDVRKVYITDDYTATGIAGTAAVAVEFARLYAVELEHYEKLEGVPLTFAGKINRLAIMVRGNLAAAMQGLLALPLLAGYDIHASDPQSAGRIVSFDAAGGWNIEEEGYQAVGSGSLFAKSSMKKLYSQVTDGDSGLRVAVEALYDAADDDSATGGPDLVRGIFPTAVIIDADGAVDVPESRIAELARAIIESRSG 6odz A 1.3 BS02 M8J A 1 H94 H96 H119 F131 L198 T199 T200 H93 H95 H118 F129 L196 T197 T198 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.7nM remove_due_to_license_issue P00918 31136893 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6odz A 1.3 BS03 M8J A 2 H4 H15 W16 D19 H3 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.7nM remove_due_to_license_issue P00918 31136893 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6oe0 A 1.3 BS02 M8S A 1 N67 I91 Q92 H94 H96 H119 F131 L198 T199 T200 N65 I89 Q90 H92 H94 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1.2nM remove_due_to_license_issue P00918 31136893 302 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6oe1 A 1.45 BS02 M8V A 1 H94 H96 H119 F131 L198 T199 T200 H92 H94 H117 F128 L195 T196 T197 H64 H94 H96 E106 H119 T199 H62 H92 H94 E104 H117 T196 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=3.1nM remove_due_to_license_issue P00918 31136893 303 HHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6oe3 A 2.9 BS01 M9A A 1 L100 K101 K102 K103 V106 V108 V179 Y181 Y188 G190 F227 W229 L234 P236 Y318 L94 K95 K96 K97 V100 V102 V173 Y175 Y182 G184 F221 W223 L228 P230 Y312 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0003676,0003964,0004523,0006278 remove_due_to_license_issue P03366 31034849 601 SPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKTKWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFAAQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLSKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNKGRQKVVPLTNTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDKSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLV 6oeb A 2.1 BS01 dna B 0 W81 F92 N93 N96 R98 K105 R106 S107 T199 H210 R212 W80 F91 N92 N95 R97 K104 R105 S106 T186 H197 R199 3.4.-.-,4.-.-.- 0003697,0006974,0106300 remove_due_to_license_issue Q96FZ2 31235913 1 ~ 9 CGRTSCHLPRDVLTRACAYQDRRGQQRLPEWRDPDKYCPSYNKSPQSNSPVLLSRLHFEKDADSSERIIAPMRWGLVPSWFKESDPSKLQFNTTNCRSDTVMEKRSFKVPLGKGRRCVVLADGFYEWQRCQGTNQRQPYFIYFPQIKPENWEKVWDNWRLLTMAGIFDCWEPPEGGDVLYSYTIITVDSCKGLSDIHHRMPAILDGEEAVSKWLDFGEVSTQEALKLIHPTENITFHAVSSVVNNSRNNTPECLAPV 6oeb A 2.1 BS02 dna C 0 W81 R106 K109 W80 R105 K108 3.4.-.-,4.-.-.- 0003697,0006974,0106300 remove_due_to_license_issue Q96FZ2 31235913 1 ~ 6 CGRTSCHLPRDVLTRACAYQDRRGQQRLPEWRDPDKYCPSYNKSPQSNSPVLLSRLHFEKDADSSERIIAPMRWGLVPSWFKESDPSKLQFNTTNCRSDTVMEKRSFKVPLGKGRRCVVLADGFYEWQRCQGTNQRQPYFIYFPQIKPENWEKVWDNWRLLTMAGIFDCWEPPEGGDVLYSYTIITVDSCKGLSDIHHRMPAILDGEEAVSKWLDFGEVSTQEALKLIHPTENITFHAVSSVVNNSRNNTPECLAPV 6of5 A 2.3 BS03 MFJ A 1 D164 Y167 R170 N201 H202 H295 H296 H323 H325 Y365 D157 Y160 R163 N194 H195 H288 H289 H316 H318 Y358 D135 D164 Y167 N201 H202 H286 H295 H296 H323 H325 D128 D157 Y160 N194 H195 H279 H288 H289 H316 H318 3.1.3.2 0003993,0005576,0008199,0008270,0016787,0046872 Ki=4.5uM remove_due_to_license_issue P80366 31445230 528 NRDMPLDSDVFRVPPGYNAPQQVHITQGDLVGRAMIISWVTMDEPGSSAVRYWSEKNGRKRIAKGKMSTYRFFNYSSGFIHHTTIRKLKYNTKYYYEVGLRNTTRRFSFITPPQTGLDVPYTFGLIGDLGQSFDSNTTLSHYELSPKKGQTVLFVGDLSYADRYPNHDNVRWDTWGRFTERSVAYQPWIWTAGNHEIEFAPEINETEPFKPFSYRYHVPYEASQSTSPFWYSIKRASAHIIVLSSYSAYGRGTPQYTWLKKELRKVKRSETPWLIVLMHSPLYNSYNHHFMEGEAMRTKFEAWFVKYKVDVVFAGHVHAYERSERVSNIAYKITNGLCTPVKDQSAPVYITIGDAGNYGVIDSNMIQPQPEYSAFREASFGHGMFDIKNRTHAHFSWNRNQDGVAVEADSVWFFNRHWYPVDDS 6oh2 A 2.58 BS01 C5P A 1 K55 Y98 Q101 N102 Y121 K124 S188 F195 Y214 G257 S261 K272 K41 Y84 Q87 N88 Y107 K110 S170 F177 Y196 G239 S243 K254 ? 0000139,0005456,0005794,0006055,0015165,0015297,0015782,0016020,0090481 remove_due_to_license_issue Q61420 30985278 401 YCLTVMTLVAAAYTVALRYTRTTAEELYFSTTAVCITEVIKLLISVGLLAKETGSLGRFKASLSENVLGSPKELAKLSVPSLVYAVQNNMAFLALSNLDAAVYQVTYQLKIPCTALCTVLMLNRTLSKLQWISVFMLCGGVTLVQWKPAVVVAQNPLLGFGAIAIAVLCSGFAGVYFEKVLKSSDTSLWVRNIQMYLSGIVVTLAGTYLSDGAEIQEKGFFYGYTYYVWFVIFLASVGGLYTSVVVKYTDNIMKGFSAAAAIVLSTIASVLLFGLQITLSFALGALLVCVSIYLYGLPR 6oh3 A 2.75 BS01 NCC A 1 A24 Y27 K55 Y98 Q101 N102 Y121 K124 S188 F195 Y214 G257 T260 S261 K272 A18 Y21 K49 Y92 Q95 N96 Y115 K118 S175 F182 Y201 G244 T247 S248 K259 ? 0000139,0005456,0005794,0006055,0015165,0015297,0015782,0016020,0090481 remove_due_to_license_issue Q61420 30985278 401 NVSLFFKLYCLTVMTLVAAAYTVALRYTRTTAEELYFSTTAVCITEVIKLLISVGLLAKETGSLGRFKASLSENVLGSPKELAKLSVPSLVYAVQNNMAFLALSNLDAAVYQVTYQLKIPCTALCTVLMLNRTLSKLQWISVFMLCGGVTLVQWVVVAQNPLLGFGAIAIAVLCSGFAGVYFEKVLKSSDTSLWVRNIQMYLSGIVVTLAGTYLSDGAEIQEKGFFYGYTYYVWFVIFLASVGGLYTSVVVKYTDNIMKGFSAAAAIVLSTIASVLLFGLQITLSFALGALLVCVSIYLYGLPR 6ohd A 2.5 BS01 MKP A 1 A51 K53 E71 L75 T106 M109 G110 A111 L167 D168 F169 L171 A42 K44 E62 L66 T97 M100 G101 A102 L158 D159 F160 L162 D150 K152 N155 D168 T185 D141 K143 N146 D159 T166 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 ic50=0.42nM remove_due_to_license_issue Q16539 31697454 900 ERPTFYRQELNKTIWEVPERYQNLSPVSVCAAFDTKTGLRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKSQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDSELKILDFGLARATRWYRAPEIMLHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPP 6oht A 3.2 BS01 MKM A 1 I31 L32 L100 Y104 M121 D162 Y165 Y188 M192 N193 W196 I25 L26 L87 Y91 M108 D149 Y152 Y175 M179 N180 W183 5.3.3.5 0000247,0004769,0005515,0005634,0005635,0005783,0005789,0006695,0008203,0016020,0016125,0016126,0016853,0030097,0031410,0031965,0033489,0033490,0033963,0042802,0043931,0047750 remove_due_to_license_issue Q15125 31165728 301 PLHPYWPQHLRLDNFVPNDRPTWHILAGLFSVTGVLVVTTWLLSGRTWRRLSLCWFAVCGFIHLVIEGWFVLYYEDLLGDQAFLSQLWKEYAKGDSRYILGDNFTVCMETITACLWGPLSLWVVIAFLRQHPLRFILQLVVSVGQIYGDVLYFLTEHRDGFQHGELGHPLYFWFYFVFMNALWLVLPGVLVLDAVKHLTHAQSTLD 6oht B 3.2 BS01 MKM B 1 I31 L35 E80 L100 M121 D162 Y188 M192 N193 W196 I25 L29 E67 L87 M108 D149 Y175 M179 N180 W183 5.3.3.5 0000247,0004769,0005515,0005634,0005635,0005783,0005789,0006695,0008203,0016020,0016125,0016126,0016853,0030097,0031410,0031965,0033489,0033490,0033963,0042802,0043931,0047750 remove_due_to_license_issue Q15125 31165728 301 PLHPYWPQHLRLDNFVPNDRPTWHILAGLFSVTGVLVVTTWLLSGRTWRRLSLCWFAVCGFIHLVIEGWFVLYYEDLLGDQAFLSQLWKEYAKGDSRYILGDNFTVCMETITACLWGPLSLWVVIAFLRQHPLRFILQLVVSVGQIYGDVLYFLTEHRDGFQHGELGHPLYFWFYFVFMNALWLVLPGVLVLDAVKHLTHAQSTLD 6ohu A 3.526 BS01 CTX A 1 L35 F36 T39 I75 I79 W101 Y188 M192 N193 W196 L29 F30 T33 I62 I66 W88 Y175 M179 N180 W183 5.3.3.5 0000247,0004769,0005515,0005634,0005635,0005783,0005789,0006695,0008203,0016020,0016125,0016126,0016853,0030097,0031410,0031965,0033489,0033490,0033963,0042802,0043931,0047750 remove_due_to_license_issue Ki=5nM Q15125 31165728 301 PLHPYWPQHLRLDNFVPNDRPTWHILAGLFSVTGVLVVTTWLLSGRTWRRLSLCWFAVCGFIHLVIEGWFVLYYEDLLGDQAFLSQLWKEYAKGDSRYILGDNFTVCMETITACLWGPLSLWVVIAFLRQHPLRFILQLVVSVGQIYGDVLYFLTEHRDGFQHGELGHPLYFWFYFVFMNALWLVLPGVLVLDAVKHLTHAQSTLD 6oi8 A 2.5 BS01 MQV A 1 I157 K159 M169 E201 Y203 L204 H209 Q233 E276 L278 E288 I437 I157 K159 M164 E196 Y198 L199 H204 Q228 E271 L273 E283 I432 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D191 H204 R230 T269 E271 E283 N285 R287 E291 R333 6.3.4.14 0003824,0003989,0004075,0005524,0006633,0016874,0046872,2001295 remove_due_to_license_issue P43873 31306011 502 MLEKVVIANRGEIALRILRACKELGIKTVAVHSTADRDLKHVLLADETICIGPAPSAKSYLNIPAIIAAAEVTGADAIHPGYGFLSENADFAEQVERSGFTFIGPTADVIRLMGDKVSAIKAMKKAGVPCVPGSDGPVSNDIAKNKEIAKRIGYPIIIKASGGMRVVRSEDALEESIAMTKAEAKAAFNNDMVYMEKYLENPRHVEIQVLADTHGNAVYLAERDCSMQRRHQKVVEEAPAPGITEEVRRDIGSRCANACVEIGYRGAGTFEFLYENGEFYFIEMNTRIQVEHPVTEMITGVDLVKEQLRIAAGLPISFKQEDIKVKGHAMECRINAEDPKTFLPSPGKVNHLHSPGGLGVRWDSHVYGGYTVPPHYDSMIAKLITYGDTREVAIRRMQNALSETIIDGIKTNIPLHELILEDENFQKGGTNIHYLEKKLG 6oi9 A 2.06 BS01 MQM A 1 K159 M169 E201 Y203 L204 H209 Q233 H236 E276 L278 E288 I437 K159 M169 E201 Y203 L204 H209 Q233 H236 E276 L278 E288 I437 E276 E288 N290 E296 R338 E276 E288 N290 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 remove_due_to_license_issue P24182 31306011 501 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 6oim A 1.65 BS02 MOV A 1 C12 K16 P34 A59 G60 Q61 E62 E63 M72 H95 Y96 Q99 C13 K17 P35 A60 G61 Q62 E63 E64 M73 H96 Y97 Q100 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31666701 303 GMTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEK 6oin A 1.7 BS02 MQJ A 1 Q654 R655 G657 G659 R660 L686 S690 S693 Y694 Q148 R149 G151 G153 R154 L180 S184 S187 Y188 2.3.1.-,2.3.1.48 0004402,0006355 remove_due_to_license_issue Q9H7Z6 31256587 802 KYVDKIHIGNYEIDAWYFSPFPEDYGKQPKLWLCEYCLKYMKYEKSYRFHLGQCQWRQPPGKEIYRKSNISVHEVDGKDHKIYCQNLCLLAKLFLDHKTLYFDVEPFVFYILTEVDRQGAHIVGYFSKEKESPDGNNVSCIMILPPYQRRGYGRFLIAFSYELSKLESTVGSPEKPLSDLGKLSYRSYWSWVLLENLRDFRGTLSIKDLSQMTSITQNDIISTLQSLNMVKYWKGQHVICVTPKLVEEHLKSAQYKKPPITVDSVCLKWAPP 6oio A 1.7 BS01 ML7 A 1 L601 I649 Q654 R655 G657 G659 R660 S684 S690 S693 L96 I144 Q149 R150 G152 G154 R155 S179 S185 S188 2.3.1.-,2.3.1.48 0004402,0006355 remove_due_to_license_issue Q9H7Z6 31256587 801 VKYVDKIHIGNYEIDAWYFSPFPEDYGKQPKLWLCEYCLKYMKYEKSYRFHLGQCQWRQPPGKEIYRKSNISVHEVDGKDHKIYCQNLCLLAKLFLDHKTLYFDVEPFVFYILTEVDRQGAHIVGYFSKEKESPDGNNVSCIMILPPYQRRGYGRFLIAFSYELSKLESTVGSPEKPLSDLGKLSYRSYWSWVLLENLRDFRGTLSIKDLSQMTSITQNDIISTLQSLNMVKYWKGQHVICVTPKLVEEHLKSAQYKKPPITVDSVCLKWAPP 6oip A 1.8 BS02 MLS A 1 Q324 R325 G327 G329 R330 L356 S360 S363 Y364 Q148 R149 G151 G153 R154 L180 S184 S187 Y188 2.3.1.-,2.3.1.48 0004402,0006355 remove_due_to_license_issue Q9H7Z6 31256587 504 KYVDKIHIGNYEIDAWYFSPFPEDYGKQPKLWLCEYCLKYMKYEKSYRFHLGQCQWRQPPGKEIYRKSNISVHEVDGKDHKIYCQNLCLLAKLFLDHKTLYFDVEPFVFYILTEVDRQGAHIVGYFSKEKESPDGNNVSCIMILPPYQRRGYGRFLIAFSYELSKLESTVGSPEKPLSDLGKLSYRSYWSWVLLENLRDFRGTLSIKDLSQMTSITQNDIISTLQSLNMVKYWKGQHVICVTPKLVEEHLKSAQYKKPPITVDSVCLKWAPP 6oiq A 1.75 BS02 MLV A 1 L601 I649 Q654 R655 G657 G659 R660 S684 L686 S690 S693 L95 I143 Q148 R149 G151 G153 R154 S178 L180 S184 S187 2.3.1.-,2.3.1.48 0004402,0006355 remove_due_to_license_issue Q9H7Z6 31256587 802 KYVDKIHIGNYEIDAWYFSPFPEDYGKQPKLWLCEYCLKYMKYEKSYRFHLGQCQWRQPPGKEIYRKSNISVHEVDGKDHKIYCQNLCLLAKLFLDHKTLYFDVEPFVFYILTEVDRQGAHIVGYFSKEKESPDGNNVSCIMILPPYQRRGYGRFLIAFSYELSKLESTVGSPEKPLSDLGKLSYRSYWSWVLLENLRDFRGTLSIKDLSQMTSITQNDIISTLQSLNMVKYWKGQHVICVTPKLVEEHLKSAQYKKPPITVDSVCLKWAPP 6oir A 2.03 BS02 MNJ A 1 L601 I649 Q654 R655 G657 G659 R660 S684 L686 S690 L95 I143 Q148 R149 G151 G153 R154 S178 L180 S184 2.3.1.-,2.3.1.48 0004402,0006355 remove_due_to_license_issue Q9H7Z6 31256587 802 KYVDKIHIGNYEIDAWYFSPFPEDYGKQPKLWLCEYCLKYMKYEKSYRFHLGQCQWRQPPGKEIYRKSNISVHEVDGKDHKIYCQNLCLLAKLFLDHKTLYFDVEPFVFYILTEVDRQGAHIVGYFSKEKESPDGNNVSCIMILPPYQRRGYGRFLIAFSYELSKLESTVGSPEKPLSDLGKLSYRSYWSWVLLENLRDFRGTLSIKDLSQMTSITQNDIISTLQSLNMVKYWKGQHVICVTPKLVEEHLKSAQYKKPPITVDSVCLKWAPP 6oja A 1.55 BS01 MET A 1 Y81 F98 Q99 H100 Y103 N153 N213 N215 N238 Y39 F56 Q57 H58 Y61 N111 N171 N173 N196 ? 0016020 Kd=0.2nM remove_due_to_license_issue Q9JPG4 31348565 1001 KEIVFGTTVGDFGDMVKEQIQAELEKKGYTVKLVEFTDYVRPNLALAEGELDINVFQHKPYLDDFKKEHNLDITEVFQVPTAPLGLYPGKLKSLEEVKDGSTVSAPNDPSNFARVLVMLDELGWIKLKDGINPLTASKADIAENLKNIKIVELEAAQLPRSRADVDFAVVNGNYAISSGMKLTEALFQEPSFAYVNWSAVKTADKDSQWLKDVTEAYNSDAFKAYAHKRFEGYKSPAAWNE 6olx A 1.43761 BS01 KFY A 1 N51 A55 M98 L107 F138 Y139 W162 N36 A40 M83 L92 F123 Y124 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 Kd=4.15uM remove_due_to_license_issue P07900 31141217 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNASDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEK 6om8 A 2.449 BS01 UDX A 1 G18 Y19 V20 D41 M42 K46 V94 N95 T96 Y113 S135 T136 K286 R353 G11 Y12 V13 D34 M35 K39 V87 N88 T89 Y106 S128 T129 K279 R346 T136 E172 K227 N231 C283 D287 T129 E165 K220 N224 C276 D280 1.1.1.22 0002009,0003979,0005634,0005737,0006024,0006065,0009792,0016491,0016616,0018991,0022414,0040025,0042802,0051287 remove_due_to_license_issue Q19905 31616809 500 KVSKVVCVGAGYVGGPTCAMIAHKCPHITVTVVDMNTAKIAEWNSDKLPIYEPGLDEIVFAARGRNLFFSSDIPKAIAEADLIFISVNTPTKMYGRGKGMAPDLKYVESVSRTIAQYAGGPKIVVEKSTVPVKAAESIGCILREAQKNNENLKFQVLSNPEFLAEGTAMKDLANPDRVLIGGESSPEGLQAVAELVRIYENWVPRNRIITTNTWSSELSKLVANAFLAQRISSINSISAVCEATGAEISEVAHAVGYDTRIGSKFLQASVGFGGSCFQKDVLSLVYLCESLNLPQVADYWQGVININNWQRRRFADKIIAELFNTVTDKKIAIFGFAFKKNTGDTRESSAIHVIKHLMEEHAKLSVYDPKVQKSQMLNDLASVTSAQDVERLITVESDPYAAARGAHAIVVLTEWDEFVELNYSQIHNDMQHPAAIFDGRLILDQKALREIGFRTFAIGTSPD 6om8 A 2.449 BS02 UDX A 2 F169 L170 A171 E172 K227 I238 F272 Q274 S276 F279 G280 C283 F284 F345 K346 R447 F162 L163 A164 E165 K220 I231 F265 Q267 S269 F272 G273 C276 F277 F338 K339 R440 T136 E172 K227 N231 C283 D287 T129 E165 K220 N224 C276 D280 1.1.1.22 0002009,0003979,0005634,0005737,0006024,0006065,0009792,0016491,0016616,0018991,0022414,0040025,0042802,0051287 remove_due_to_license_issue Q19905 31616809 501 KVSKVVCVGAGYVGGPTCAMIAHKCPHITVTVVDMNTAKIAEWNSDKLPIYEPGLDEIVFAARGRNLFFSSDIPKAIAEADLIFISVNTPTKMYGRGKGMAPDLKYVESVSRTIAQYAGGPKIVVEKSTVPVKAAESIGCILREAQKNNENLKFQVLSNPEFLAEGTAMKDLANPDRVLIGGESSPEGLQAVAELVRIYENWVPRNRIITTNTWSSELSKLVANAFLAQRISSINSISAVCEATGAEISEVAHAVGYDTRIGSKFLQASVGFGGSCFQKDVLSLVYLCESLNLPQVADYWQGVININNWQRRRFADKIIAELFNTVTDKKIAIFGFAFKKNTGDTRESSAIHVIKHLMEEHAKLSVYDPKVQKSQMLNDLASVTSAQDVERLITVESDPYAAARGAHAIVVLTEWDEFVELNYSQIHNDMQHPAAIFDGRLILDQKALREIGFRTFAIGTSPD 6omu A 1.41 BS01 MZJ A 1 L408 A428 K430 M449 T474 M477 C481 L528 S538 D539 F540 L20 A40 K42 M61 T86 M89 C93 L140 S150 D151 F152 D521 A523 R525 N526 D539 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=8.9nM remove_due_to_license_issue Q06187 31368705 702 GLGYGSWEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMDEES 6on0 A 1.6 BS01 dna C 0 T23 A26 Q29 W30 R40 T23 A26 Q29 W30 R40 ? 0003677 remove_due_to_license_issue Q37964 31180482 1 ~ 17 MKPEELVRHFGDVEKAAVGVGVTPGAVYQWLQAGEIPPLRQSDIEVRTAYKLKSDFTSQRMG 6on0 A 1.6 BS02 dna N 0 Y28 Q32 Y28 Q32 ? 0003677 remove_due_to_license_issue Q37964 31180482 1 ~ 17 MKPEELVRHFGDVEKAAVGVGVTPGAVYQWLQAGEIPPLRQSDIEVRTAYKLKSDFTSQRMG 6on0 B 1.6 BS01 dna C 0 Y28 Q32 Y28 Q32 ? 0003677 remove_due_to_license_issue Q37964 31180482 1 ~ 17 MKPEELVRHFGDVEKAAVGVGVTPGAVYQWLQAGEIPPLRQSDIEVRTAYKLKSDFTSQRMGK 6on0 B 1.6 BS02 dna N 0 V22 T23 A26 Q29 P37 R40 V22 T23 A26 Q29 P37 R40 ? 0003677 remove_due_to_license_issue Q37964 31180482 1 ~ 17 MKPEELVRHFGDVEKAAVGVGVTPGAVYQWLQAGEIPPLRQSDIEVRTAYKLKSDFTSQRMGK 6ooy A 2.5 BS01 A7M C 1 L57 Y59 L51 Y53 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 201 TPSDKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSHVLLTHTISRIAVSYQTKVNLLSAIKSPCKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6ooy B 2.5 BS01 A7M C 1 Y119 G121 Y102 G104 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 201 PSDKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSHVLLTHTISRIAVSYQTKVNLLSAIKSPCAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6ooy C 2.5 BS01 A7M C 1 Y59 S60 Y119 Y151 Y49 S50 Y96 Y128 ? 0005164,0006955,0016020 Kd=22uM remove_due_to_license_issue P01375 31857588 201 KPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCHVLLTHTISRIAVSYQTKVNLLSAIKSPCKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6ooz A 2.8 BS01 A6Y C 1 L57 Y59 Y119 L51 Y53 Y109 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 202 TPSDKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCQRETPAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6ooz B 2.8 BS01 A6Y C 1 Y119 G122 Y104 G107 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 202 RTPSDKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPHVLLTHTISRIAVSYQTKVNLLSAIKSPCEAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6ooz C 2.8 BS01 A6Y C 1 Y59 S60 Y119 L120 Y151 Y41 S42 Y91 L92 Y120 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 202 DKPVAHVVANPEGQLQWLNANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCTHVLLTHTISRIAVQTKVNLLSAIKSPCQREAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFGQVYFGIIAL 6op0 A 2.55 BS01 A7A C 1 L57 Y59 Y119 L51 Y53 Y109 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 201 TPSDKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCQRETPAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6op0 B 2.55 BS01 A7A C 1 Y119 G121 Y103 G105 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 201 TPSDKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPHVLLTHTISRIAVSYQTKVNLLSAIKSPCEAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 6op0 C 2.55 BS01 A7A C 1 L57 Y59 S60 Y119 Y151 I155 L35 Y37 S38 Y85 Y113 I117 ? 0005164,0006955,0016020 remove_due_to_license_issue P01375 31857588 201 KPVAHVVANEGQLQWLNGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVQTKVNLLSAIKSPCKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDGQVYFGIIAL 6op9 A 2.501 BS01 DB8 A 1 L696 C721 I722 K723 L766 T768 L771 P772 G774 L822 D833 L17 C42 I43 K44 L87 T89 L92 P93 G95 L143 D154 N815 R819 N820 D833 N136 R140 N141 D154 2.7.10.1 0004672,0005524,0006468 remove_due_to_license_issue Kd=0.770000nM P21860 35108525 1101 VLARIFKETELRKLKVLGSGVFGTVHKGVWIPEGESIKIPVCIKVIEDKSGRQSFQAVTDHMLAIGSLDHAHIVRLLGLCPGSSLQLVTQYLPLGSLLDHVRQHRGALGPQLLLNWGVQIAKGMYYLEEHGMVHRNLAARNVLLKSPSQVQVADFGVADLLPPDDKQAKTPIKWMALESIHFGKYTHQSDVWSYGVTVWELMTFGAEPYAGLRLAEVPDLLEKGERLAQPQICTIDVYMVMVKCWMIDENIRPTFKELANEFTRMARDPPRYLVIK 6oqb A 1.6 BS01 N0J A 1 H224 A227 V249 M250 V253 F254 R263 T266 L267 F270 I294 H53 A56 V78 M79 V82 F83 R92 T95 L96 F99 I123 ? 0042981 Ki=0.00004uM remove_due_to_license_issue Ki=0.050000nM Q07820 30254093 401 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6oqc A 1.8 BS01 N0S A 1 H224 A227 F228 V249 M250 V253 R263 T266 L267 F270 H54 A57 F58 V79 M80 V83 R93 T96 L97 F100 ? 0042981 Ki=0.00005uM remove_due_to_license_issue Ki=0.040000nM Q07820 30254093 501 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 6oqd A 1.48 BS01 N0M A 1 H224 A227 V249 M250 V253 R263 T266 L267 F270 I294 H54 A57 V79 M80 V83 R93 T96 L97 F100 I124 ? 0042981 Ki=0.00014uM remove_due_to_license_issue Ki=0.140000nM Q07820 30254093 401 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6oqn A 1.7 BS01 N0P A 1 M250 V253 R263 T266 L267 F270 M80 V83 R93 T96 L97 F100 ? 0042981 ic50=0.01uM remove_due_to_license_issue Q07820 30254093 401 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6orr A 2.25 BS01 N37 A 1 Y11 Y20 Y25 G63 S64 T67 Y69 D85 Y86 S87 C141 D142 V143 T163 L164 A169 S201 Y204 S213 Y22 Y31 Y36 G74 S75 T78 Y80 D96 Y97 S98 C152 D153 V154 T174 L175 A180 S212 Y215 S224 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0030760,0031100,0032259,0034356,0045722,0090312 Ki=500pM remove_due_to_license_issue Ki=500nM P40261 31589440 301 HHSSGLVPRGSMESGFTSKDTYLSHFNPRDYLEKYYKFGSRHSAESQILKHLLKNLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIVVTDYSDQNLQELEKWLKAAPAAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPPADCVLSTLCLDAACPDLPTYCRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVARKL 6os5 A 1.66 BS01 TRP A 1 D55 V56 E64 Y326 D50 V51 E59 Y321 ? 0009820,0016740,0016765,0046872 Kd=4.4uM remove_due_to_license_issue A8M6W6 31251043 401 TTVRDACARTLENTARTLHLGASGTEFVAAFRAMTDHWGAARPHDLPLSDVSPDGSPVEYAVDLGGLAPALQFAMEPLTAGVPARDPLAARAIMPLLAGRYGADATRWSALADRLLPDDAHGPHVSMYGAEVRAGAPIRFKAWFYLNVTGPDGAFNLLYSALERMGTTHLWPVVQAHVHRAGEDVPFLLSLDLSDDPAARVKVYFRHFAADVEEVAAVLKAYPGFEPGEVRAFCKVMMGGRRRFSDQPAVTCVSLLDAQTFDRTAATLYVPLWTYAEHDGEVRQRVHRTLAAWPEALYRYDSVLAGIAHRGLDAGTGIHNYISWQPGRTRPRMKVYLSPEMHDVTPPPLGVSQ 6os6 A 1.33 BS02 TRP A 1 D55 V56 E64 Y326 D54 V55 E63 Y325 ? 0009820,0016740,0016765,0046872 Kd=1.1uM remove_due_to_license_issue A8M6W6 31251043 402 TEELTTVRDACARTLENTARTLHLGASGTEFVAAFRAMTDHWGAARPHDLPLSDVSPDGSPVEYAVDLGGLAPALQFAMEPLTAGVPARDPLAARAIMPLLAGRYGADATRWSALADRLLPDDAHGPHVSMYGAEVRAGAPIRFKAWFYLNVTGPDGAFNLLYSALERMGTTHLWPVVQAHVHRAGEDVPFLLSLDLSDDPAARVKVYFRHFAADVEEVAAVLKAYPGFEPGEVRAFCKVMMGGRRRFSDQPAVTCVSLLDAQTFDRTAATLYVPLWTYAEHDGEVRQRVHRTLAAWPEALYRYDSVLAGIAHRGLDAGTGIHNYISWQPGRTRPRMKVYLSPEMHDVTPPPLGVSQQHHLS 6ott A 2.55 BS01 N7Y A 1 R58 H59 R62 R58 H59 R62 C1 G27 N101 G102 Y258 R321 K326 M336 D444 C1 G27 N101 G102 Y258 R321 K326 M336 D444 2.4.2.14 0000287,0004044,0005737,0005829,0006164,0006189,0006541,0009113,0016757,0042802,0046872,0097216 remove_due_to_license_issue P0AG16 31695193 602 CGIVGIAGVMPVNQSIYDALTVLQHRGQDAAGIITIDANNCFRLRKANGLVSDVFEARHMQRLQGNMGIGHVRYPTAGSSSASEAQPFYVNSPYGITLAHNGNLTNAHELRKKLFEEKRRHINTTSDSEILLNIFASELDNFRHYPLEADNIFAAIAATNRLIRGAYACVAMIIGHGMVAFRDPNGIRPLVLGKRDIDENRTEYMVASESVALDTLGFDFLRDVAPGEAIYITEEGQLFTRQCADNPVSNPCLFEYVYFARPDSFIDKISVYSARVNMGTKLGEKIAREWEDLDIDVVIPIPETSCDIALEIARILGKPYRQGFVKNRYVGRTFIMPGQQLRRKSVRRKLNANRAEFRDKNVLLVDDSIVRGTTSEQIIEMAREAGAKKVYLASAAPEIRFPNVYGIDMPSATELIAHGREVDEIRQIIGADGLIFQDLNDLIDAVRAENPDIQQFECSVFNGVYVTKDVDQGYLDFLDTLRNDDAKAVQRQNEVE 6ouv A 1.937 BS01 TDK A 1 H51 S54 H82 H124 A125 G153 D154 G155 S156 N183 M185 S186 I187 K289 H304 M349 I371 E373 F398 D430 H434 H44 S47 H75 H117 A118 G146 D147 G148 S149 N176 M178 S179 I180 K255 H270 M315 I337 E339 F364 D396 H400 K289 H304 E373 R401 K255 H270 E339 R367 2.2.1.7 0000287,0003824,0005829,0008299,0008661,0009228,0016114,0016740,0019288,0030976,0046872,0052865 remove_due_to_license_issue Q9RUB5 31239351 701 SDTPLLDQIHGPKDLKRLSREQLPALTEELRGEIVRVCSRGGLHLASSLGAVDIITALHYVLDSPRDRILFDVGHQAYAHKILTGRRDQMADIKKEGGISGFTKVSESEHDAITVGHASTSLANALGMALARDAQGKDFHVAAVIGDGSLTGGMALAALNTIGDMGRKMLIVLNDNEMSISENVGAMNKFMRGLQVQKWFQAVEAVSKPSVNPFAAMGVRYVGPVDGHNVQELVWLLERLVDLDGPTILHIVTTKGKGLSYAEADPIYWHGPAKFDPATGEYVPSSAYSWSAAFGEAVTEWAKTDPRTFVVTPAMREGSGLVEFSRVHPHRYLDVGIAEEVAVTTAAGMALQGMRPVVAIYSTFLQRAYDQVLHDVAIEHLNVTFCIDRAGIVGADGATHNGVFDLSFLRSIPGVRIGLPKDAAELRGMLKYAQTHDGPFAIRYPRGNTAQVPAGTWPDLKWGEWERLKGGDDVVILAGGKALDYALKAAEDLPGVGVVNARFVKPLDEEMLREVGGRARALITVEDNTVVGGFGGAVLEALNSMNLHPTVRVLGIPDEFQEHATAESVHARAGIDAPAIRTVLAELGVDVPIEV 6ouv B 1.937 BS01 TDK B 1 H51 S54 H82 H124 A125 G153 D154 G155 S156 N183 M185 S186 I187 K289 H304 M349 I371 E373 F398 D430 H434 H44 S47 H75 H117 A118 G146 D147 G148 S149 N176 M178 S179 I180 K239 H254 M299 I321 E323 F348 D380 H384 K289 H304 E373 R401 K239 H254 E323 R351 2.2.1.7 0000287,0003824,0005829,0008299,0008661,0009228,0016114,0016740,0019288,0030976,0046872,0052865 remove_due_to_license_issue Q9RUB5 31239351 701 SDTPLLDQIHGPKDLKRLSREQLPALTEELRGEIVRVCSRGGLHLASSLGAVDIITALHYVLDSPRDRILFDVGHQAYAHKILTGRRDQMADIKKEGGISGFTKVSESEHDAITVGHASTSLANALGMALARDAQGKDFHVAAVIGDGSLTGGMALAALNTIGDMGRKMLIVLNDNEMSISENVGAMNKFMRGSVNPFAAMGVRYVGPVDGHNVQELVWLLERLVDLDGPTILHIVTTKGKGLSYAEADPIYWHGPAKFDPATGEYVPSSAYSWSAAFGEAVTEWAKTDPRTFVVTPAMREGSGLVEFSRVHPHRYLDVGIAEEVAVTTAAGMALQGMRPVVAIYSTFLQRAYDQVLHDVAIEHLNVTFCIDRAGIVGADGATHNGVFDLSFLRSIPGVRIGLPKDAAELRGMLKYAQTHDGPFAIRYPRGNTAQVPAGTWPDLKWGEWERLKGGDDVVILAGGKALDYALKAAEDLPGVGVVNARFVKPLDEEMLREVGGRARALITVEDNTVVGGFGGAVLEALNSMNLHPTVRVLGIPDEFQEHATAESVHARAGIDAPAIRTVLAELGVDVP 6ovc A -1.00 BS01 N8J A 1 H55 M62 V84 R94 T97 L98 F101 H55 M62 V84 R94 T97 L98 F101 ? 0042981 remove_due_to_license_issue Q07820 30254093 201 MEDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESSIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEGGHHHHHH 6ovz A 2.017 BS05 N9M A 1 F70 V73 K211 H250 F28 V31 K169 H208 H120 H122 D124 H189 C208 K211 N220 H250 H78 H80 D82 H147 C166 K169 N178 H208 3.5.2.6 remove_due_to_license_issue E5KIY2 31145588 1005 DQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKL 6ow2 P 1.7 BS01 NB4 P 1 Q57 G69 G70 V71 G72 Q77 E128 C130 L131 V170 H173 E174 H177 Q56 G68 G69 V70 G71 Q76 E117 C119 L120 V159 H162 E163 H166 G72 Q77 C130 L131 H173 E174 H177 G71 Q76 C119 L120 H162 E163 H166 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=3nM remove_due_to_license_issue Q8DP79 31160176 302 SAIERITKAAHLIDMNDIIREGNPTLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLIL 6ow7 P 1.45 BS01 N9Y P 1 R68 G69 G70 V71 G72 Q77 E128 G129 C130 L131 H173 E174 H177 R67 G68 G69 V70 G71 Q76 E122 G123 C124 L125 H167 E168 H171 G72 Q77 C130 L131 H173 E174 H177 G71 Q76 C124 L125 H167 E168 H171 3.5.1.88 0006412,0016787,0042586,0043686,0046872 ic50=1nM remove_due_to_license_issue Q8DP79 31160176 303 SAIERITKAAHLIDMNDIIREGNPTLRTVAEEVTFPLSDQEIILGEKMMQFLKHSQDPVMAEKMGLRGGVGLAAPQLDISKRIIAVLVPNITPQEAYDLEAIMYNPKIVSHSVQDAALGEGEGCLSVDRNVPGYVVRHARVTVDYFDKDGEKHRIKLKGYNSIVVQHEIDHINGIMFYDRINEKDPFAVKDGLLIL 6ox0 A 1.755 BS02 SFG A 1 R74 E103 F105 R253 D274 M275 N277 H278 Y312 S324 F326 R55 E84 F86 R234 D255 M256 N258 H259 Y293 S305 F307 2.1.1.85 0000785,0003713,0003779,0005515,0005634,0005654,0005737,0006338,0008168,0008170,0008276,0008757,0016279,0018021,0018023,0018064,0030047,0032259,0042800,0045893,0045944,0046975,0051149,0061629,0070472 remove_due_to_license_issue Q86TU7 31388018 1001 SPKEILNLTSELLQKCSSPAPGPGKEWEEYVQIRTLVEKIRKKQKGLSVTFDGKREDYFPDLMKWASENGASVEGFEMVNFKEEGFGLRATRDIKAEELFLWVPRKLLMTVESAKNSVLGPLYSQDRILQAMGNIALAFHLLCERASPNSFWQPYIQTLPSEYDTPLYFEEDEVRYLQSTQAIHDVFSQYKNTARQYAYFYKVIQTHPHANKLPLKDSFTYEDYRWAVSSVMTRQNQIPTEDGSRVTLALIPLWDMCNHTNGLITTGYNLEDDRCECVALQDFRAGEQIYIFYGTRSNAEFVIHSGFFFDNNSHDRVKIKLGVSKSDRLYAMKAEVLARAGIPTSSVFALHFTEPPISAQLLAFLRVFCMTEEELKEHLLGDSAIDRIFTLGNSEFPVSWDNEVKLWTFLEDRASLLLKTYKTTIEEDKSVLKNHDLSVRAKMAIKLRLGEKEILEKAVKSAAVNREYYRQQMEEKAPLPK 6oxp A 1.97 BS01 K2A A 1 D25 G27 A28 D29 D30 G48 I50 V82 D25 G27 A28 D29 D30 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxp B 1.97 BS01 K2A A 1 D25 A28 D30 P81 I84 D25 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxq A 1.89 BS01 F53 A 1 D25 G27 A28 D29 G48 I50 D25 G27 A28 D29 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxq B 1.89 BS01 F53 A 1 D25 A28 D30 P81 I84 D25 A28 D30 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxr A 2.035 BS01 NJA A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxr B 2.035 BS01 NJA A 1 D25 A28 D30 I47 P81 V82 I84 D25 A28 D30 I47 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxs A 1.989 BS01 NJ4 A 1 D25 G27 A28 D29 D30 G48 G49 I50 D25 G27 A28 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxs B 1.989 BS01 NJ4 A 1 D25 A28 D30 V32 G48 P81 V82 D25 A28 D30 V32 G48 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxt A 1.861 BS01 NEJ A 1 D25 G27 A28 D29 D30 G48 I50 V82 D25 G27 A28 D29 D30 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxt B 1.861 BS01 NEJ A 1 D25 A28 D30 I47 G48 I84 D25 A28 D30 I47 G48 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxu A 1.861 BS01 NE7 A 1 D25 G27 A28 D29 G48 I50 V82 D25 G27 A28 D29 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxu B 1.861 BS01 NE7 A 1 D25 A28 D30 V32 G48 P81 V82 I84 D25 A28 D30 V32 G48 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxv A 1.991 BS01 NF4 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxv B 1.991 BS01 NF4 A 1 D25 A28 D30 I47 P81 V82 D25 A28 D30 I47 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxw A 1.982 BS01 NFJ A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxw B 1.982 BS01 NFJ A 1 D25 A28 D30 V32 G48 I50 P81 V82 D25 A28 D30 V32 G48 I50 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxx A 1.962 BS01 NF7 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxx B 1.962 BS01 NF7 A 1 D25 A28 D29 D30 G48 P81 I84 D25 A28 D29 D30 G48 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxy A 1.96 BS01 NG4 A 1 D25 G27 A28 D29 D30 I47 G48 I50 D25 G27 A28 D29 D30 I47 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxy B 1.96 BS01 NG4 A 1 D25 A28 D30 I47 G48 L76 P81 D25 A28 D30 I47 G48 L76 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxz A 1.961 BS01 NJG A 1 D25 G27 A28 D29 D30 G48 G49 I50 V82 D25 G27 A28 D29 D30 G48 G49 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oxz B 1.961 BS01 NJG A 1 D25 A28 D29 D30 G48 P81 I84 D25 A28 D29 D30 G48 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 102 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oy0 A 2.0 BS01 NJ7 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oy0 B 2.0 BS01 NJ7 A 1 D25 A28 D29 D30 I47 G48 L76 P81 V82 I84 D25 A28 D29 D30 I47 G48 L76 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oy1 A 2.0 BS01 NJ1 A 1 D25 G27 A28 D29 D30 G48 I50 D25 G27 A28 D29 D30 G48 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oy1 B 2.0 BS01 NJ1 A 1 D25 G27 A28 D29 D30 G48 P81 I84 D25 G27 A28 D29 D30 G48 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 103 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oy2 A 1.99 BS01 NJJ A 1 D25 G27 A28 D29 I47 G48 I50 V82 D25 G27 A28 D29 I47 G48 I50 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oy2 B 1.99 BS01 NJJ A 1 D25 A28 D29 D30 I47 G48 L76 P81 I84 D25 A28 D29 D30 I47 G48 L76 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 31386368 101 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 6oyh A 2.95 BS01 NK4 A 1 K70 T75 N190 L191 D193 G194 L195 D196 F262 G264 H324 H325 K41 T46 N161 L162 D164 G165 L166 D167 F233 G235 H292 H293 2.7.8.13 0005886,0008360,0008963,0009252,0016020,0016740,0016780,0042802,0044038,0046872,0051301,0051992,0071555 remove_due_to_license_issue O66465 31266949 401 FAFNVLKYITFRSFTAVLIAFFLTLVLSPSFINRLRKIQVKKYTPTMGGIVILIVVTLSTLLLMRWDIKYTWVVLLSFLSFGTIGFWDDYVKLKNKKGISIKTKFLLQVLSASLISVLIYYWADIDTILYFPFFKELYVDLGVLYLPFAVFVIVGSANAVNLTDGLDGLAIGPAMTTATALGVVAYAVGHSKIAQYLNIPYVPYAGELTVFCFALVGAGLGFLWFNSFPAQMFMGDVGSLSIGASLATVALLTKSEFIFAVAAGVFVFETISVILQIIYFRWTGGKRRAPFHHHLELNGLPEPKIVVRMWIISILLAIIAISMLKL 6oyt A 2.824 BS01 NJV A 1 L686 G687 V694 A707 K709 M754 E755 Q756 V757 G759 G760 L810 D822 L21 G22 V29 A42 K44 M84 E85 Q86 V87 G89 G90 L140 D152 D803 K805 D807 N808 D822 D133 K135 D137 N138 D152 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=20nM Q99683 31710475 1001 MESDLLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLGKAADIWSLGCTIIEMATGKPPVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6oyt C 2.824 BS01 NJV C 1 L686 G687 V694 A707 K709 M754 E755 Q756 V757 P758 G759 L810 D822 L16 G17 V24 A37 K39 M84 E85 Q86 V87 P88 G89 L140 D152 D803 K805 D807 N808 D822 D133 K135 D137 N138 D152 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=20nM Q99683 31710475 1001 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLLQYMAPEIIDKGPRGGKAADIWSLGCTIIEMATGKPPFHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFL 6oyw C 2.603 BS01 NKJ C 1 L686 G689 A707 K709 M754 E755 Q756 V757 G760 L810 S821 D822 L16 G19 A37 K39 M80 E81 Q82 V83 G86 L136 S147 D148 D803 K805 D807 N808 D822 T842 D129 K131 D133 N134 D148 T163 2.7.11.25 0004672,0005524,0006468 remove_due_to_license_issue IC50=4.0nM Q99683 31710475 1001 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPEYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLATEEFTGTLQYMAPEIIDKGPRGYGKAADIWSLGCTIIEMATGKPPFYELGEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6oyz A 3.62 BS01 NKM A 1 K70 T75 K121 D193 G194 L195 D196 F262 M263 G264 K34 T39 K85 D157 G158 L159 D160 F226 M227 G228 2.7.8.13 0005886,0008360,0008963,0009252,0016020,0016740,0016780,0042802,0044038,0046872,0051301,0051992,0071555 remove_due_to_license_issue O66465 31266949 401 YITFRSFTAVLIAFFLTLVLSPSFINRLRKIQRKKYTPTMGGIVILIVVTLSTLLLMRWDIKYTWVVLLSFLSFGTIGFWDDYVKLKNKKGISIKTKFLLQVLSASLISVLIYYWADIDTILYFPFFKELYVDLGVLYLPFAVFVIVGSANAVNLTDGLDGLAIGPAMTTATALGVVAYAVGHSKIAQYLNIPYVPYAGELTVFCFALVGAGLGFLWFNSFPAQMFMGDVGSLSIGASLATVALLTKSEFIFAVAAGVFVFETISVILQIIYFRWTPFHHHLELNGLPEPKIVVRMWIISILLAIIAISMLKL 6oz6 A 3.7 BS01 NKD A 1 T75 N190 L191 D193 G194 L195 D196 F262 G264 V302 A321 T48 N163 L164 D166 G167 L168 D169 F235 G237 V275 A294 2.7.8.13 0005886,0008360,0008963,0009252,0016020,0016740,0016780,0042802,0044038,0046872,0051301,0051992,0071555 remove_due_to_license_issue O66465 31266949 401 AFNVLKYITFRSFTAVLIAFFLTLVLSPSFINRLRKIQRLFGKKYTPTMGGIVILIVVTLSTLLLMRWDIKYTWVVLLSFLSFGTIGFWDDYVKLKNKKGISIKTKFLLQVLSASLISVLIYYWADIDTILYFPFFKELYVDLGVLYLPFAVFVIVGSANAVNLTDGLDGLAIGPAMTTATALGVVAYAVGHSKIAQYLNIPYVPYAGELTVFCFALVGAGLGFLWFNSFPAQMFMGDVGSLSIGASLATVALLTKSEFIFAVAAGVFVFETISVILQIIYFRWTGGKRLFKRAPFHHHLELNGLPEPKIVVRMWIISILLAIIAISMLKL 6p0g A 2.27 BS01 dna B 0 N19 W53 G54 R55 R81 F121 I154 N17 W51 G52 R53 R79 F119 I152 ? remove_due_to_license_issue C5A3Z3 31822563 2 ~ 7 NQLFIIGIGTGTDEYENFEETILKGVKRNELEGQIGPDILDNCCSDVCYFWGRSKETIYEKKIDKGDMVLFYVGKRISRNKVDLNQETAVYLGIICETVEISENDVSFLNDFWRKGENFRFLMFFKKKPEKLHHSINEINSKLGYNPDYFPIAGYVKPERMSGVYDILKNILK 6p0g A 2.27 BS02 dna C 0 Y61 N82 K83 Y147 N148 Y151 Y157 K159 R162 Y59 N80 K81 Y145 N146 Y149 Y155 K157 R160 ? remove_due_to_license_issue C5A3Z3 31822563 2 ~ 7 NQLFIIGIGTGTDEYENFEETILKGVKRNELEGQIGPDILDNCCSDVCYFWGRSKETIYEKKIDKGDMVLFYVGKRISRNKVDLNQETAVYLGIICETVEISENDVSFLNDFWRKGENFRFLMFFKKKPEKLHHSINEINSKLGYNPDYFPIAGYVKPERMSGVYDILKNILK 6p10 B 2.301 BS01 SKE B 1 D484 I485 A486 G526 C527 G528 L531 L659 G688 T692 D25 I26 A27 G67 C68 G69 L72 L185 G214 T218 5.6.1.1 0005524,0016887 ic50=6uM remove_due_to_license_issue Q8I0P1 31257183 802 GVEQKLVQLILDEIVEGGAKVEWTDIAGQDVAKQALQEMVILPSVRPELFTGLRAPAKGLLLFGPPGCGKTLLARAVATECSATFLNISAASLTSKYGEKLVRALFAVARHMQPSIIFIDEVDSLLSRRLKTEFLVEFDGLPPDGDRIVVLAATNRPQELDEAALRRFTKRVYVSLPDEQTRELLLNRLLQKQGSPLDTEALRRLAKITDGYSGSDLTALAKDAALEPIRELNVEQVKCLDISAMRAITEQDFHSSLKRIRRSVAPQSLNSYEKWSQDYGD 6p11 B 2.15 BS01 SKE B 1 D484 I485 A486 G526 N527 G528 L659 G688 S689 D25 I26 A27 G67 N68 G69 L184 G213 S214 5.6.1.1 0005524,0016887 ic50=0.9uM remove_due_to_license_issue Q8I0P1 31257183 802 GVEQKLVQLILDEIVEGGAKVEWTDIAGQDVAKQALQEMVILPSVRPELFTGLRAPAKGLLLFGPPGNGKTLLARAVATECSATFLNISAASLTSKYGEKLVRALFAVARHMQPSIIFIDEVDSLLSRRLKTEFLVEFDGLPGGDRIVVLAATNRPQELDEAALRRFTKRVYVSLPDEQTRELLLNRLLQKQGSPLDTEALRRLAKITDGYSGSDLAALAKDAALEPIRELNVEQVKCLDISAMRAITEQDFHSSLKRIRRSVAPQSLNSYEKWSQDYGD 6p12 B 1.94132 BS01 NKY B 1 D484 I485 A486 Q488 N527 L531 S649 L650 P651 L659 G688 S689 T692 D25 I26 A27 Q29 N68 L72 S174 L175 P176 L184 G213 S214 T217 5.6.1.1 0005524,0016887 ic50=0.23uM remove_due_to_license_issue Q8I0P1 31257183 801 GVEQKLVQLILDEIVEGGAKVEWTDIAGQDVAKQALQEMVILPSVRPELFTGLRAPAKGLLLFGPPGNGKTLLARAVATECSATFLNISAASLTSKYDGELVRALFAVARHMQPSIIFIDEVDSLLSRRLKTEFLVEFDGLPGNDRIVVLAATNRPQELDEAALRRFTKRVYVSLPDEQTRELLLNRLLQKQGSPLDTEALRRLAKITDGYSGSDLTALAKDAALEPIRELNVEQVKCLDISAMRAITEQDFHSSLKRIRRSVAPQSLNSYEKWSQDYGDI 6p14 A 1.93001 BS01 NKY A 1 A486 Q488 N527 L531 S649 L650 P651 L659 G688 S689 A30 Q32 N71 L75 S160 L161 P162 L170 G199 S200 5.6.1.1 0005524,0016887 ic50=0.22uM remove_due_to_license_issue Q8I0P1 31257183 804 VVSVKEQKLVQLILDEIVEGGAKVEWTDIAGQDVAKQALQEMVILPSVRPELFTGLRAPAKGLLLFGPPGNGKTLLARAVATECSATFLNISKLVRALFAVARHMQPSIIFIDEVDSLRLKTEFLVEFDGDRIVVLAATNRPQELDEAALRRFTKRVYVSLPDEQTRELLLNRLLQKQGSPLDTEALRRLAKITDGYSGSDLAALAKDAALEPIRELNVEQVKCLDISAMRAITEQDFHSSLKRIRRSVAPQSLNSYEKWSQDYG 6p1d B 2.4 BS02 NQ1 B 1 A743 K745 M766 C775 R776 L788 M790 D855 F856 L858 L861 A42 K44 M65 C74 R75 L87 M89 D154 F155 L157 L160 D837 R841 N842 D855 D136 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=>10000nM P00533 31749909 1102 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDA 6p3p A 1.61 BS01 NQJ A 1 H224 A227 F228 M231 M250 V253 N260 G262 R263 T266 L267 H54 A57 F58 M61 M80 V83 N90 G92 R93 T96 L97 ? 0042981 ic50=0.145uM remove_due_to_license_issue IC50=145nM Q07820 31235261 501 SDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6p3t A 2.5 BS01 NRS A 1 F24 D26 F27 I28 A33 W36 L63 S83 F84 F22 D24 F25 I26 A31 W34 L57 S77 F78 2.3.1.- 0005576,0005829,0008080,0016746,0016747,0030649,0033661,0034054,0034069,0042802,0043655,0044161,0046677,0051701,0052032,0052040,0052167,0061733,0097691 remove_due_to_license_issue IC50=0.240nM P9WFK7 31433614 501 VTLCSPTEDDWPGMFLLAAASFTDFIGPESATAWRTLVPTDGAVVVRDGSEVVGMALYMDLRLTVPGEVVLPTAGLSFVAVAPTHRRRGLLRAMCAELHRRIADSGYPVAALHASEGGIYGRFGYGPATTLHELTVDRRFARFHADAPGGGLGGSSVRLVRPTEHRGEFEAIYERWRQQVPGGLLRPQVLWDELLAEAKAAPGGDRESFALLHPDGYALYRVDRTDLKLARVSELRAVTADAHCALWRALIGLDSMERISIITHPQDPLPHLLTDTRLARTTWRQDGLWLRIMNVPAALEARGYAHEVGEFSTVLEVSDGGRFALKIGDGRARCTPTDAAAEIEMDRDVLGSLYLGAHRASTLAAANRLRTKDSQLLRRLDAAFASDVPVQTAFEF 6p3u A 2.55 BS01 NRY A 1 D26 F27 I28 S32 W36 R37 L63 F84 E401 F402 D24 F25 I26 S30 W34 R35 L57 F78 E395 F396 2.3.1.- 0005576,0005829,0008080,0016746,0016747,0030649,0033661,0034054,0034069,0042802,0043655,0044161,0046677,0051701,0052032,0052040,0052167,0061733,0097691 remove_due_to_license_issue P9WFK7 31433614 501 VTLCSPTEDDWPGMFLLAAASFTDFIGPESATAWRTLVPTDGAVVVRDGSEVVGMALYMDLRLTVPGEVVLPTAGLSFVAVAPTHRRRGLLRAMCAELHRRIADSGYPVAALHASEGGIYGRFGYGPATTLHELTVDRRFARFHADAPGGGLGGSSVRLVRPTEHRGEFEAIYERWRQQVPGGLLRPQVLWDELLAEAKAAPGGDRESFALLHPDGYALYRVDRTDLKLARVSELRAVTADAHCALWRALIGLDSMERISIITHPQDPLPHLLTDTRLARTTWRQDGLWLRIMNVPAALEARGYAHEVGEFSTVLEVSDGGRFALKIGDGRARCTPTDAAAEIEMDRDVLGSLYLGAHRASTLAAANRLRTKDSQLLRRLDAAFASDVPVQTAFEF 6p3v A 2.5 BS01 NRV A 1 D26 F27 A33 W36 R37 L63 F84 D24 F25 A31 W34 R35 L57 F78 2.3.1.- 0005576,0005829,0008080,0016746,0016747,0030649,0033661,0034054,0034069,0042802,0043655,0044161,0046677,0051701,0052032,0052040,0052167,0061733,0097691 remove_due_to_license_issue P9WFK7 31433614 501 VTLCSPTEDDWPGMFLLAAASFTDFIGPESATAWRTLVPTDGAVVVRDGSEVVGMALYMDLRLTVPGEVVLPTAGLSFVAVAPTHRRRGLLRAMCAELHRRIADSGYPVAALHASEGGIYGRFGYGPATTLHELTVDRRFARFHADAPGGGGSSVRLVRPTEHRGEFEAIYERWRQQVPGGLLRPQVLWDELLAEAKAAPGGDRESFALLHPDGYALYRVDRTDLKLARVSELRAVTADAHCALWRALIGLDSMERISIITHPQDPLPHLLTDTRLARTTWRQDGLWLRIMNVPAALEARGYAHEVGEFSTVLEVSDGGRFALKIGDGRARCTPTDAAAEIEMDRDVLGSLYLGAHRASTLAAANRLRTKDSQLLRRLDAAFASDVPVQTAFEF 6p5o A 1.49 BS02 O2Y A 1 A86 R87 Y235 G236 K243 K244 H264 D311 F333 N403 R405 A84 R85 Y233 G234 K241 K242 H262 D309 F331 N401 R403 R87 Y235 K244 H264 S286 C288 D311 R405 R85 Y233 K242 H262 S284 C286 D309 R403 2.7.11.-,4.1.1.32 0000287,0004550,0004611,0004613,0005525,0005737,0005783,0005829,0006006,0006094,0006107,0006629,0009617,0014823,0016301,0016831,0017076,0018105,0019003,0019543,0030145,0031406,0031667,0032496,0032868,0032869,0033993,0042593,0042594,0043382,0043648,0045944,0046166,0046327,0046872,0046889,0046890,0051365,0070365,0070741,0071300,0071320,0071332,0071333,0071347,0071356,0071377,0071456,0071474,0071475,0071476,0071477,0071549,0072350,0097403,0106264,1904628,1904640 ic50=97uM remove_due_to_license_issue P07379 31461616 703 PQLHNGLDFSAKVIQGSLDSLPQEVRKFVEGNAQLCQPEYIHICDGSEEEYGRLLAHMQEEGVIRKLKKYDNCWLALTDPRDVARIESKTVIITQEQRDTVPIPKSGQSQLGRWMSEEDFEKAFNARFPGCMKGRTMYVIPFSMGPLGSPLAKIGIELTDSPYVVASMRIMTRMGTSVLEALGDGEFIKCLHSVGCPLPLKKPLVNNWACNPELTLIAHLPDRREIISFGSGYGGNSLLGKKCFALRIASRLAKEEGWLAEHMLILGITNPEGKKKYLAAAFPSACGKTNLAMMNPTLPGWKVECVGDDIAWMKFDAQGNLRAINPENGFFGVAPGTSVKTNPNAIKTIQKNTIFTNVAETSDGGVYWEGIDEPLAPGVTITSWKNKEWRPQDEEPCAHPNSRFCTPASQCPIIDPAWESPEGVPIEGIIFGGRRPAGVPLVYEALSWQHGVFVGAAMRSEATAAAHKGKVIMHDPFAMRPFFGYNFGKYLAHWLSMAHRPAAKLPKIFHVNWFRKDKNGKFLWPGFGENSRVLEWMFGRIEGEDSAKLTPIGYVPKEDALNLKGLGDVNVEELFGISKEFWEKEVEEIDKYLEDQVNADLPYEIERELRALKQRISQM 6p5v A 1.398 BS01 O37 A 1 I1086 P1097 A1106 Q1114 C1115 E1116 F1117 F1164 A1180 Y1181 I202 P213 A222 Q230 C231 E232 F233 F280 A296 Y297 E11 D20 E24 D33 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 ic50=0.2uM remove_due_to_license_issue D9IEF7,Q96GG9 31465221 1302 HSQDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRTKRVITTFRTGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQIAGTKSTTV 6p5w A 1.69 BS01 O0A A 1 I1086 Q1087 P1097 V1102 L1103 Q1114 C1115 E1116 F1117 F1164 A1180 Y1181 L1184 I202 Q203 P213 V218 L219 Q230 C231 E232 F233 F280 A296 Y297 L300 E11 D20 E24 D33 3.2.1.17 0003796,0009253,0016798,0016998,0030430,0031640,0042742,0044659 ic50=5.1uM remove_due_to_license_issue D9IEF7,Q96GG9 31465221 1301 HSQDLENLYFQGSMNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRTKRVITTFRTGTWDAYKNLRKKLEQLYNRYKDPQDENKIGIDGIQQFCDDLALDPASISVLIIAWKFRAATQCEFSKQEFMDGMTELGCDSIEKLKAQIPKMEQELKEPGRFKDFYQFTFNFAKNPGQKGLDLEMAIAYWNLVLNGRFKFLDLWNKFLLEHHSIPKDTWNLLLDFSTMIADDMSNYDEEGAWPVLIDDFVEFARPQIAGTKS 6p83 A 1.7 BS01 O3Y A 1 A250 M266 I267 G268 G269 V285 A248 M264 I265 G266 G267 V283 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 Kd=0.08uM remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p83 A 1.7 BS02 O3Y B 1 F183 I254 A256 F181 I252 A254 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 Kd=0.08uM remove_due_to_license_issue P21645 31402665 501 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p83 C 1.7 BS01 O3Y A 1 F183 I254 A256 F182 I253 A255 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 Kd=0.08uM remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p83 C 1.7 BS02 O3Y C 1 A250 M266 I267 G268 G269 A249 M265 I266 G267 G268 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 Kd=0.08uM remove_due_to_license_issue P21645 31402665 501 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p84 A 1.7 BS01 O3V A 1 A250 M266 I267 G268 G269 A248 M264 I265 G266 G267 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p84 A 1.7 BS02 O3V B 1 F183 I254 A256 F181 I252 A254 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 501 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p84 C 1.7 BS01 O3V A 1 I254 A256 I253 A255 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p84 C 1.7 BS02 O3V C 1 A250 M266 I267 G268 G269 A249 M265 I266 G267 G268 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 501 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p85 A 1.9 BS01 O4V A 1 A250 G268 G269 G287 A248 G266 G267 G285 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p85 C 1.9 BS01 O4V A 1 V272 N274 V291 V271 N273 V290 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p86 A 1.8 BS01 O4S A 1 A248 A250 G268 G269 T286 G287 A246 A248 G266 G267 T284 G285 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p86 C 1.8 BS01 O4S A 1 V272 N274 M290 V271 N273 M289 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p87 A 1.9 BS01 O4P A 1 A250 M266 G268 G269 T286 G287 A248 M264 G266 G267 T284 G285 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p87 C 1.9 BS01 O4P A 1 A256 N274 M290 M292 A255 N273 M289 M291 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p88 A 1.7 BS01 O4G A 1 A250 M266 G287 A248 M264 G285 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p88 C 1.7 BS01 O4G A 1 F183 I254 A256 V272 N274 V291 F182 I253 A255 V271 N273 V290 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p89 A 1.4 BS01 O4A A 1 M266 I267 G268 T286 G287 M264 I265 G266 T284 G285 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p89 C 1.4 BS01 O4A A 1 N274 M290 M292 N273 M289 M291 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p8a A 1.8 BS01 O4D A 1 A248 A250 M266 I267 G268 T286 G287 A246 A248 M264 I265 G266 T284 G285 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 SIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKV 6p8a C 1.8 BS01 O4D A 1 N274 M292 N273 M291 2.3.1.191 0005515,0005737,0005829,0009245,0016020,0016410,0016740,0016746,0016747,0042802,0046677,0103118 remove_due_to_license_issue P21645 31402665 403 GSIRLADLAQQLDAELHGDGDIVITGVASMQSAQTGHITFMVNPKYREHLGLCQASAVVMTQDDLPFAKSAALVVKNPYLTYARMAQILDTTPQPAQNIAPSAVIDATAKLGNNVSIGANAVIESGVELGDNVIIGAGCFVGKNSKIGAGSRLWANVTIYHEIQIGQNCLIQSGTVVGADGFGYANDRGNWVKIPQIGRVIIGDRVEIGACTTIDRGALDDTIIGNGVIIDNQCQIAHNVVIGDNTAVAGGVIMAGSLKIGRYCMIGGASVINGHMEICDKVTVTGMGMVMRPITEPGVYSSGIPLQPNKVWRKTAALVMNIDDMSKRLKSLERKVN 6p8x A 2.11 BS02 O5V A 1 C12 K16 G60 M72 D92 H95 Y96 Q99 C11 K15 G59 M71 D91 H94 Y95 Q98 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31531201 305 TEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6p8y A 2.31 BS02 O5Y A 1 C12 K16 P34 A59 R68 M72 H95 Y96 Q99 C12 K16 P34 A59 R68 M72 H95 Y96 Q99 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31531201 303 MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKH 6p8z A 1.65 BS02 O5S A 1 V9 C12 K16 T58 A59 G60 R68 M72 D92 H95 Y96 I100 V10 C13 K17 T59 A60 G61 R65 M69 D89 H92 Y93 I97 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31531201 304 GMTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKE 6p8z A 1.65 BS03 O5S B 1 I24 Q25 H27 Y32 Y40 I25 Q26 H28 Y33 Y41 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31531201 304 GMTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKE 6p9e A 2.0 BS01 O6D A 1 R121 K123 S128 F163 L165 I167 R101 K103 S108 F143 L145 I147 ? 0002437,0005125,0005149,0005576,0005615,0005654,0005737,0005829,0005886,0006954,0006955,0007267,0010628,0019221,0045087,0071222 Kd=67.6nM remove_due_to_license_issue Q9NZH8 31235749 4000 KPITGTINDLNQQVWTLQGQNLVAVPRSDSVTPVTVAVITCKYPEALEQGRGDPIYLGIQNPEMCLYCEKVGEQPTLQLKEQKIMDLYGQPEPVKPFLFYRAKTGRTSTLESVAFPDWFIASSKRDQPIILTSELGKSYNTAFELNIN 6pdj A 1.81 BS01 ODJ A 1 L251 A271 K273 M280 F285 N290 I314 T316 Y318 M319 G322 L371 D382 F383 G384 L25 A45 K47 M54 F59 N64 I88 T90 Y92 M93 G96 L145 D156 F157 G158 D364 A368 N369 D382 D138 A142 N143 D156 2.7.10.2 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=42nM P06239 31620238 601 GHMQKPWWEDEWEVPRETLKLVERLGAGQFGEVWMGYYNGHTKVAVKSLKQGSMSPDAFLAEANLMKQLQHQRLVRLYAVVTQEPIYIITEYMENGSLVDFLKTPSGIKLTINKLLDMAAQIAEGMAFIEERNYIHRDLRAANILVSDTLSCKIADFGLARLIEDNEYTAREGAKFPIKWTAPEAINYGTFTIKSDVWSFGILLTEIVTHGRIPYPGMTNPEVIQNLERGYRMVRPDNCPEELYQLMRLCWKERPEDRPTFDYLRSVLEDFFTA 6peb A 2.46 BS01 OE4 A 1 H191 F193 R196 D219 V242 A244 P273 S275 P307 R311 I351 H176 F178 R181 D204 V227 A229 P258 S260 P292 R296 I336 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=2.7nM remove_due_to_license_issue IC50=2.7nM P43490 31749905 601 EFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKVKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 6peb B 2.46 BS01 OE4 A 1 D16 Y18 D10 Y12 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=2.7nM remove_due_to_license_issue IC50=2.7nM P43490 31749905 601 AEFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 6peb B 2.46 BS02 OE4 B 1 H191 F193 R196 D219 A244 P273 S275 P307 R311 I351 H175 F177 R180 D203 A228 P257 S259 P291 R295 I335 2.4.2.12 0005125,0005515,0005576,0005615,0005634,0005737,0005829,0007165,0007267,0007623,0008284,0008286,0009435,0016607,0016757,0019363,0030054,0032922,0034356,0042802,0045944,0047280,0048511,0051770,0060612,0070062 ic50=2.7nM remove_due_to_license_issue IC50=2.7nM P43490 31749905 601 AEFNILLATDSYKVTHYKQYPPNTSKVYSYFECREKKYEETVFYGLQYILNKYLKGKVVTKEKIQEAKDVYKEHFQDDVFNEKGWNYILEKYDGHLPIEIKAVPEGFVIPRGNVLFTVENTDPECYWLTNWIETILVQSWYPITVATNSREQKKILAKYLLETSGNLDGLEYKLHDFGYRGVSSQETAGIGASAHLVNFKGTDTVAGLALIKKYYGTKDPVPGYSVPAAEHSTITAWGKDHEKDAFEHIVTQFSSVPVSVVSDSYDIYNACEKIWGEDLRHLIVSRSTQAPLIIRPDSGNPLDTVLKVLEILGKKFPVTENSKGYKLLPPYLRVIQGDGVDINTLQEIVEGMKQKMWSIENIAFGSGGGLLQKLTRDLLNCSFKCSYVVTNGLGINVFKDPVADPNKRSKKGRLSLHRTPAGNFVTLEEGKGDLEEYGQDLLHTVFKNGKVTKSYSFDEIRKNAQLNI 6pf3 A 2.391 BS02 OE7 A 1 F80 I108 D218 L221 G222 F225 Y258 M311 A312 F52 I80 D190 L193 G194 F197 Y230 M283 A284 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 31536894 601 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 6pf3 C 2.391 BS02 OE7 C 1 I108 D218 L221 G222 F225 Y258 M311 A312 I80 D190 L193 G194 F197 Y230 M283 A284 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 31536894 601 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 6pf4 B 2.854 BS02 OF7 B 1 I108 W109 D218 L221 G222 F225 M311 I80 W81 D190 L193 G194 F197 M283 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 31536894 601 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMA 6pf4 D 2.854 BS03 OF7 D 1 F80 I108 W109 N112 D218 L221 G222 F225 M309 M311 A312 F52 I80 W81 N84 D190 L193 G194 F197 M281 M283 A284 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 31536894 601 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMA 6pf5 A 2.39 BS02 OED A 1 R78 F80 D218 G222 F225 M311 A312 R50 F52 D190 G194 F197 M283 A284 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 31536894 601 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 6pf6 B 2.502 BS02 OEJ B 1 F80 I108 D218 L221 G222 F225 M311 A312 F52 I80 D190 L193 G194 F197 M283 A284 E87 W109 Y135 C195 R215 D218 E59 W81 Y107 C167 R187 D190 2.1.1.45 0000900,0003729,0004799,0005542,0005634,0005737,0005739,0005743,0005759,0005829,0006206,0006231,0006235,0006417,0007623,0008168,0009165,0009410,0009636,0014070,0016741,0017148,0019860,0032259,0032570,0033189,0034097,0035999,0042803,0045471,0046653,0046683,0048589,0051216,0051384,0051593,0060574,0071897,0097421,1901363,1990825 remove_due_to_license_issue P04818 31536894 601 SELQYLGQIQHILRCGVRKDDRTGTGTLSVFGMQARYSLRDEFPLLTTKRVFWKGVLEELLWFIKGSTNAKELSSKGVKIWDANGSRDFLDSLGFSTREEGDLGPVYGFQWRHFGAEYRDMESDYSGQGVDQLQRVIDTIKTNPDDRRIIMCAWNPRDLPLMALPPCHALCQFYVVNSELSCQLYQRSGDMGLGVPFNIASYALLTYMIAHITGLKPGDFIHTLGDAHIYLNHIEPLKIQLQREPRPFPKLRILRKVEKIDDFKAEDFQIEGYNPHPTIKMEMAV 6pfj A 2.08 BS01 C2E T 2 G61 R62 V65 G37 R38 V41 ? 0000166,0003677,0003700,0003899,0006352,0006355,0016987,2000142 remove_due_to_license_issue A0A3N1Q704 31810759 202 APTSLDELWRSYKETGDERLREQLILHYSPLVKYVAGRVSVGLPSNVEQADFVSSGVFGLIDAIEKFDVERAIKFETYAITRIRGAMIDELRALDWIPRSVRQKARNVERAYATLEAQLRRTPSETEVAAEMDISLEDLHAVFSQLSLANVVALEELLHRRLLARAINTLPEREKTVVTLYYYEGLTLAEIGHVLGVTESRVSQIHTKSVLQLRAKLAD 6pfj T 2.08 BS01 C2E T 1 R71 Q75 D79 S108 H110 E162 S166 R169 R22 Q26 D30 S59 H61 E113 S117 R120 ? Kd=0.39uM remove_due_to_license_issue F2RFR7 31810759 201 LPELRTLRREAQSDEADLSYVRRMLQGRIDILRAELARRTDGEAPVLDRLSEILADVPSRHRSSARHVTLSTPRGEEYRRLAAEMLSEVELSDLTARTDEELHAAMGRLAGYEQQISRRRHHLQRTADDCSAEIARRYREGEAQVDDLL 6pfj T 2.08 BS02 C2E T 2 E64 S68 R71 S108 S112 R115 R169 Q173 D177 E15 S19 R22 S59 S63 R66 R120 Q124 D128 ? Kd=0.39uM remove_due_to_license_issue F2RFR7 31810759 202 LPELRTLRREAQSDEADLSYVRRMLQGRIDILRAELARRTDGEAPVLDRLSEILADVPSRHRSSARHVTLSTPRGEEYRRLAAEMLSEVELSDLTARTDEELHAAMGRLAGYEQQISRRRHHLQRTADDCSAEIARRYREGEAQVDDLL 6pg3 A 2.04 BS01 OHJ A 1 S91 F133 S175 A176 F219 C261 F263 S61 F103 S145 A146 F185 C227 F229 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=480uM remove_due_to_license_issue P61964 31768400 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pg4 A 1.6 BS01 OHG A 1 S91 F133 S175 A176 F219 C261 F263 S62 F104 S146 A147 F190 C232 F234 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=260uM remove_due_to_license_issue P61964 31768400 401 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pg5 A 1.99 BS01 OHV A 1 S49 S91 F133 F149 S175 A176 Y191 F219 Y260 C261 F263 I305 S20 S62 F104 F120 S146 A147 Y162 F190 Y231 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=11uM remove_due_to_license_issue P61964 31768400 401 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pg6 A 1.68 BS01 OH7 A 1 S91 F133 S175 A176 Y260 C261 F263 I305 S61 F103 S145 A146 Y227 C228 F230 I272 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=200uM remove_due_to_license_issue P61964 31768400 402 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pg7 A 2.45 BS01 OH4 A 1 S49 S91 F133 S175 F219 C261 F263 S20 S62 F104 S146 F190 C232 F234 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=22uM remove_due_to_license_issue P61964 31768400 401 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pg8 A 1.67 BS01 OGY A 1 S49 S91 F133 S175 A176 C261 F263 I305 S19 S61 F103 S145 A146 C227 F229 I271 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=140uM remove_due_to_license_issue P61964 31768400 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pg9 A 1.75 BS01 OH1 A 1 S49 S91 F133 S175 A176 Y191 Y260 C261 F263 I305 S19 S61 F103 S145 A146 Y161 Y230 C231 F233 I275 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=12uM remove_due_to_license_issue P61964 31768400 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pga A 2.45 BS01 OGM A 1 S49 S91 F133 S175 A176 F219 Y260 C261 F263 I305 S20 S62 F104 S146 A147 F190 Y231 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=28.9uM remove_due_to_license_issue P61964 31768400 401 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pgb A 1.73 BS01 OJG A 1 S49 S91 F133 S175 A176 F219 K259 Y260 C261 F263 I305 S20 S62 F104 S146 A147 F190 K230 Y231 C232 F234 I276 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=25uM remove_due_to_license_issue P61964 31768400 401 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pgc A 1.81 BS01 OJJ A 1 S49 S91 F133 S175 A176 F219 Y260 C261 F263 I305 E322 S20 S62 F104 S146 A147 F190 Y231 C232 F234 I276 E293 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=4.5uM remove_due_to_license_issue P61964 31768400 403 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pge A 1.76 BS01 OJM A 1 S49 S91 F133 S175 A176 F219 C261 F263 S20 S62 F104 S146 A147 F190 C232 F234 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=240uM remove_due_to_license_issue P61964 31768400 401 GSKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6pgo A 1.6 BS02 OJ1 A 1 V9 C12 K16 T58 A59 G60 R68 M72 Y96 Q99 V9 C12 K16 T58 A59 G60 R61 M65 Y89 Q92 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31820981 303 MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6pgp A 1.5 BS02 OHY A 1 C12 K16 T58 A59 G60 E62 R68 M72 H95 Y96 Q99 C12 K16 T58 A59 G60 E62 R68 M72 H95 Y96 Q99 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31820981 504 MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETSLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEK 6pgx A 1.36 BS02 OJ4 A 1 E69 D72 I91 Q92 E68 D71 I90 Q91 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.62nM remove_due_to_license_issue Ki=0.620000nM P00918 31401537 302 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6pgx A 1.36 BS03 OJ4 A 2 W5 H15 W16 D19 W4 H14 W15 D18 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.62nM remove_due_to_license_issue Ki=0.620000nM P00918 31401537 303 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6pgx A 1.36 BS04 OJ4 A 3 H94 H119 F131 L198 T199 T200 P202 H93 H118 F129 L196 T197 T198 P200 H64 H94 H96 E106 H119 T199 H63 H93 H95 E105 H118 T197 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=0.62nM remove_due_to_license_issue Ki=0.620000nM P00918 31401537 304 SHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6phr A 1.65 BS01 SS9 A 1 E17 D19 D117 H159 Y168 H197 F225 Y323 E20 D22 D120 H162 Y171 H200 F228 Y326 ? 0004407,0040029,0046872 ic50=160uM remove_due_to_license_issue A0A0J7JFD7 31436969 502 LGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6phr B 1.65 BS01 SS9 B 1 E17 D19 D117 H159 Y168 D195 H197 F225 E21 D23 D121 H163 Y172 D199 H201 F229 ? 0004407,0040029,0046872 ic50=160uM remove_due_to_license_issue A0A0J7JFD7 31436969 502 PLGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pht A 1.8 BS01 OKP A 1 H158 H159 G167 Y168 D195 H197 F225 D284 Y323 H161 H162 G170 Y171 D198 H200 F228 D287 Y326 ? 0004407,0040029,0046872 ic50=390uM remove_due_to_license_issue A0A0J7JFD7 31436969 401 LGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6phz A 2.0 BS03 FKS A 1 E17 L18 D19 D117 P156 H158 H159 G167 Y168 D195 H197 F225 G321 E22 L23 D24 D122 P161 H163 H164 G172 Y173 D200 H202 F230 G326 ? 0004407,0040029,0046872 ic50=350uM remove_due_to_license_issue A0A0J7JFD7 31436969 406 GPLGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGK 6phz B 2.0 BS03 FKS B 1 E17 L18 D19 D117 P156 H158 H159 G167 Y168 D195 H197 F225 E320 G321 Y323 E19 L20 D21 D119 P158 H160 H161 G169 Y170 D197 H199 F227 E322 G323 Y325 ? 0004407,0040029,0046872 ic50=350uM remove_due_to_license_issue A0A0J7JFD7 31436969 406 GSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGK 6pi1 A 1.7 BS03 B3N A 1 D19 D117 H158 H159 Y168 D195 H197 F225 I291 Y323 D21 D119 H160 H161 Y170 D197 H199 F227 I293 Y325 ? 0004407,0040029,0046872 ic50=160uM remove_due_to_license_issue A0A0J7JFD7 31436969 405 GSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pi1 B 1.7 BS03 B3N B 1 D19 D117 H158 H159 Y168 D195 H197 F225 I291 Y323 D22 D120 H161 H162 Y171 D198 H200 F228 I294 Y326 ? 0004407,0040029,0046872 ic50=160uM remove_due_to_license_issue A0A0J7JFD7 31436969 406 LGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pi5 A 1.67 BS01 GUN A 1 Y45 S97 F98 E165 W194 N220 Y19 S71 F72 E139 W168 N194 ? 0005886,0046872 Kd=0.11uM remove_due_to_license_issue Q936X6 31692473 401 QEPLKVAFVYAGPVSDAGYTYAHDQGRLAMEKNLGAKVKSSYVENVPEGADAERVIRKLAADGNKLIFTTSFGFMNPTERVAKAFPNVVFEHATGVKLAKNLGVYESRQYEGTYLQGVLAAKMTKTGVIGFVGSFPVPEVIRNINAYTLGAQSVNPKIKTKVIWVSTWYDPAKERQAAETLIAQGADVLTQNTNSPATLQVAQEKGKYAFGCDADMSKFAPKAHLTASISNWGDFYTKTAQAVMAGTWKSEEVHWGMAEGMVKMAPLNAAVPPDAAKLFEEKKAAMVSGKIKPFQGPLKDQSGAVKVAAGSDLPLASLKGMNWYVQGVEGTIPK 6pi6 A 1.65 BS01 OKM A 1 A37 Y45 S97 F98 E165 W194 N218 N220 D239 A10 Y18 S70 F71 E138 W167 N191 N193 D212 ? 0005886,0046872 Kd=2.2uM remove_due_to_license_issue Q936X6 31692473 401 EPLKVAFVYAGPVSDAGYTYAHDQGRLAMEKNLGAKVKSSYVENVPEGADAERVIRKLAADGNKLIFTTSFGFMNPTERVAKAFPNVVFEHATGVKLAKNLGVYESRQYEGTYLQGVLAAKMTKTGVIGFVGSFPVPEVIRNINAYTLGAQSVNPKIKTKVIWVSTWYDPAKERQAAETLIAQGADVLTQNTNSPATLQVAQEKGKYAFGCDADMSKFAPKAHLTASISNWGDFYTKTAQAVMAGTWKSEEVHWGMAEGMVKMAPLNAAVPPDAAKLFEEKKAAMVSGKIKPFQGPLKDQSGAVKVAAGSDLPLASLKGMNWYVQGVEGTIPK 6pia A 1.75 BS03 XS6 A 1 E17 L18 D19 D117 H158 H159 G167 Y168 D195 H197 F225 Y323 E19 L20 D21 D119 H160 H161 G169 Y170 D197 H199 F227 Y325 ? 0004407,0040029,0046872 ic50=550uM remove_due_to_license_issue A0A0J7JFD7 31436969 407 GSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pia B 1.75 BS03 XS6 B 1 E17 L18 D19 D117 H158 H159 Y168 D195 H197 F225 Y323 E19 L20 D21 D119 H160 H161 Y170 D197 H199 F227 Y325 ? 0004407,0040029,0046872 ic50=550uM remove_due_to_license_issue A0A0J7JFD7 31436969 406 GSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pid A 1.546 BS04 OKS A 1 E17 D19 D117 H158 H159 Y168 D195 H197 Y323 E20 D22 D120 H161 H162 Y171 D198 H200 Y326 ? 0004407,0040029,0046872 ic50=380uM remove_due_to_license_issue A0A0J7JFD7 31436969 406 LGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pid B 1.546 BS03 OKS B 1 H158 H159 Y168 D195 H197 F225 D284 Y323 H161 H162 Y171 D198 H200 F228 D287 Y326 ? 0004407,0040029,0046872 ic50=380uM remove_due_to_license_issue A0A0J7JFD7 31436969 405 LGSMKTVFSPLHSRRHVKTELDGGLLIEPHEKPSRAETILARVKDQALGEILEPEEFGLGPVKRVHTADYVSFLETCWDEWVAAGKRGEAIPTFWVGRGMRARLPKDIDGRLGYYSLGADTSISDGTWEAARASANVALTAQKLVAEGERAAFALCRPPGHHAHADVFGGYCFFNNAAIAAQAFRDQGYGKVAVLDVDFHHGNGTQAIFYDRSDVLTISLHGDPDLVFPHFLGFEDETGEGDGEAYNLNIVFPPDTPFSIWSQGLEKACERIRTFAPDALVVALGVDTFEEDPISFFKLTSGDYLKLGKRLEQLGLPTVFTMEGGYDVDAIGVNAVNVMQGFEGKS 6pii A 1.87 BS01 GUN A 1 Y45 S97 F98 E165 W194 N220 Y21 S73 F74 E141 W170 N196 ? 0005886,0046872 remove_due_to_license_issue Q936X6 31692473 401 HMQEPLKVAFVYAGPVSDAGYTYAHDQGRLAMEKNLGAKVKSSYVENVPEGADAERVIRKLAADGNKLIFTTSFGFMNPTERVAKAFPNVVFEHATGVKLAKNLGVYESRQYEGTYLQGVLAAKMTKTGVIGFVGSFPVPEVIRNINAYTLGAQSVNPKIKTKVIWVSTWYDPAKERQAAETLIAQGADVLTQNTNSPATLQVAQEKGKYAFGCDADMSKFAPKAHLTASISNWGDFYTKTAQAVMAGTWKSEEVHWGMAEGMVKMAPLNAAVPPDAAKLFEEKKAAMVSGKIKPFQGPLKDQSGAVKVAAGSDLPLASLKGMNWYVQGVEGTIPK 6pk7 A 3.1 BS02 CTP A 1 D153 I154 E155 D153 I154 E155 6.3.4.2 0003883,0005515,0005524,0005737,0005739,0005829,0006220,0006221,0006241,0016874,0019856,0042802,0044210,0097268 remove_due_to_license_issue Q9NRF8 31873303 602 MKYILVTGGVISGIGKGIIASSIGTILKSCGLRVTAIKIDPYINIDAGTFSPYEHGEVFVLNDGGEVDLDLGNYERFLDINLYKDNNITTGKIYQHVINKERRGDYLGKTVQVVPHITDAVQEWVMNQAKVPVDGNKEEPQICVIELGGTIGDIEGMPFVEAFRQFQFKAKRENFCNIHVSLVPQLSATGEQKTKPTQNSVRALRGLGLSPDLIVCRSSTPIEMAVKEKISMFCHVNPEQVICIHDVSSTYRVPVLLEEQSIVKYFKERLHLPIGDSASNLLFKWRNMADRYERLQKICSIALVGKYTKLRDCYASVFKALEHSALAINHKLNLMYIDSIDLEKITETEDPVKFHEAWQKLCKADGILVPGGFGIRGTLGKLQAISWARTKKIPFLGVCLGMQLAVIEFARNCLNLKDADSTEFRPNAPVPLVIDMPEHNPGNLGGTMRLGIRRTVFKTENSILRKLYGDVPFIEERHRHRFEVNPNLIKQFEQNDLSFVGQDVDGDRMEIIELANHPYFVGVQFHPEFSSRPMKPSPPYLGLLLAATGNLNAYLQQ 6pk7 A 3.1 BS03 CTP D 1 K193 T194 K195 K229 K193 T194 K195 K229 6.3.4.2 0003883,0005515,0005524,0005737,0005739,0005829,0006220,0006221,0006241,0016874,0019856,0042802,0044210,0097268 remove_due_to_license_issue Q9NRF8 31873303 602 MKYILVTGGVISGIGKGIIASSIGTILKSCGLRVTAIKIDPYINIDAGTFSPYEHGEVFVLNDGGEVDLDLGNYERFLDINLYKDNNITTGKIYQHVINKERRGDYLGKTVQVVPHITDAVQEWVMNQAKVPVDGNKEEPQICVIELGGTIGDIEGMPFVEAFRQFQFKAKRENFCNIHVSLVPQLSATGEQKTKPTQNSVRALRGLGLSPDLIVCRSSTPIEMAVKEKISMFCHVNPEQVICIHDVSSTYRVPVLLEEQSIVKYFKERLHLPIGDSASNLLFKWRNMADRYERLQKICSIALVGKYTKLRDCYASVFKALEHSALAINHKLNLMYIDSIDLEKITETEDPVKFHEAWQKLCKADGILVPGGFGIRGTLGKLQAISWARTKKIPFLGVCLGMQLAVIEFARNCLNLKDADSTEFRPNAPVPLVIDMPEHNPGNLGGTMRLGIRRTVFKTENSILRKLYGDVPFIEERHRHRFEVNPNLIKQFEQNDLSFVGQDVDGDRMEIIELANHPYFVGVQFHPEFSSRPMKPSPPYLGLLLAATGNLNAYLQQ 6pk7 A 3.1 BS04 CTP E 1 Q112 V113 V114 Q112 V113 V114 6.3.4.2 0003883,0005515,0005524,0005737,0005739,0005829,0006220,0006221,0006241,0016874,0019856,0042802,0044210,0097268 remove_due_to_license_issue Q9NRF8 31873303 602 MKYILVTGGVISGIGKGIIASSIGTILKSCGLRVTAIKIDPYINIDAGTFSPYEHGEVFVLNDGGEVDLDLGNYERFLDINLYKDNNITTGKIYQHVINKERRGDYLGKTVQVVPHITDAVQEWVMNQAKVPVDGNKEEPQICVIELGGTIGDIEGMPFVEAFRQFQFKAKRENFCNIHVSLVPQLSATGEQKTKPTQNSVRALRGLGLSPDLIVCRSSTPIEMAVKEKISMFCHVNPEQVICIHDVSSTYRVPVLLEEQSIVKYFKERLHLPIGDSASNLLFKWRNMADRYERLQKICSIALVGKYTKLRDCYASVFKALEHSALAINHKLNLMYIDSIDLEKITETEDPVKFHEAWQKLCKADGILVPGGFGIRGTLGKLQAISWARTKKIPFLGVCLGMQLAVIEFARNCLNLKDADSTEFRPNAPVPLVIDMPEHNPGNLGGTMRLGIRRTVFKTENSILRKLYGDVPFIEERHRHRFEVNPNLIKQFEQNDLSFVGQDVDGDRMEIIELANHPYFVGVQFHPEFSSRPMKPSPPYLGLLLAATGNLNAYLQQ 6pk7 D 3.1 BS01 CTP A 1 K193 T194 K195 K229 K193 T194 K195 K229 6.3.4.2 0003883,0005515,0005524,0005737,0005739,0005829,0006220,0006221,0006241,0016874,0019856,0042802,0044210,0097268 remove_due_to_license_issue Q9NRF8 31873303 602 MKYILVTGGVISGIGKGIIASSIGTILKSCGLRVTAIKIDPYINIDAGTFSPYEHGEVFVLNDGGEVDLDLGNYERFLDINLYKDNNITTGKIYQHVINKERRGDYLGKTVQVVPHITDAVQEWVMNQAKVPVDGNKEEPQICVIELGGTIGDIEGMPFVEAFRQFQFKAKRENFCNIHVSLVPQLSATGEQKTKPTQNSVRALRGLGLSPDLIVCRSSTPIEMAVKEKISMFCHVNPEQVICIHDVSSTYRVPVLLEEQSIVKYFKERLHLPIGDSASNLLFKWRNMADRYERLQKICSIALVGKYTKLRDCYASVFKALEHSALAINHKLNLMYIDSIDLEKITETEDPVKFHEAWQKLCKADGILVPGGFGIRGTLGKLQAISWARTKKIPFLGVCLGMQLAVIEFARNCLNLKDADSTEFRPNAPVPLVIDMPEHNPGNLGGTMRLGIRRTVFKTENSILRKLYGDVPFIEERHRHRFEVNPNLIKQFEQNDLSFVGQDVDGDRMEIIELANHPYFVGVQFHPEFSSRPMKPSPPYLGLLLAATGNLNAYLQQ 6pk7 D 3.1 BS03 CTP D 1 D153 I154 E155 D153 I154 E155 6.3.4.2 0003883,0005515,0005524,0005737,0005739,0005829,0006220,0006221,0006241,0016874,0019856,0042802,0044210,0097268 remove_due_to_license_issue Q9NRF8 31873303 602 MKYILVTGGVISGIGKGIIASSIGTILKSCGLRVTAIKIDPYINIDAGTFSPYEHGEVFVLNDGGEVDLDLGNYERFLDINLYKDNNITTGKIYQHVINKERRGDYLGKTVQVVPHITDAVQEWVMNQAKVPVDGNKEEPQICVIELGGTIGDIEGMPFVEAFRQFQFKAKRENFCNIHVSLVPQLSATGEQKTKPTQNSVRALRGLGLSPDLIVCRSSTPIEMAVKEKISMFCHVNPEQVICIHDVSSTYRVPVLLEEQSIVKYFKERLHLPIGDSASNLLFKWRNMADRYERLQKICSIALVGKYTKLRDCYASVFKALEHSALAINHKLNLMYIDSIDLEKITETEDPVKFHEAWQKLCKADGILVPGGFGIRGTLGKLQAISWARTKKIPFLGVCLGMQLAVIEFARNCLNLKDADSTEFRPNAPVPLVIDMPEHNPGNLGGTMRLGIRRTVFKTENSILRKLYGDVPFIEERHRHRFEVNPNLIKQFEQNDLSFVGQDVDGDRMEIIELANHPYFVGVQFHPEFSSRPMKPSPPYLGLLLAATGNLNAYLQQ 6pk7 D 3.1 BS04 CTP F 1 Q112 V113 V114 Q112 V113 V114 6.3.4.2 0003883,0005515,0005524,0005737,0005739,0005829,0006220,0006221,0006241,0016874,0019856,0042802,0044210,0097268 remove_due_to_license_issue Q9NRF8 31873303 602 MKYILVTGGVISGIGKGIIASSIGTILKSCGLRVTAIKIDPYINIDAGTFSPYEHGEVFVLNDGGEVDLDLGNYERFLDINLYKDNNITTGKIYQHVINKERRGDYLGKTVQVVPHITDAVQEWVMNQAKVPVDGNKEEPQICVIELGGTIGDIEGMPFVEAFRQFQFKAKRENFCNIHVSLVPQLSATGEQKTKPTQNSVRALRGLGLSPDLIVCRSSTPIEMAVKEKISMFCHVNPEQVICIHDVSSTYRVPVLLEEQSIVKYFKERLHLPIGDSASNLLFKWRNMADRYERLQKICSIALVGKYTKLRDCYASVFKALEHSALAINHKLNLMYIDSIDLEKITETEDPVKFHEAWQKLCKADGILVPGGFGIRGTLGKLQAISWARTKKIPFLGVCLGMQLAVIEFARNCLNLKDADSTEFRPNAPVPLVIDMPEHNPGNLGGTMRLGIRRTVFKTENSILRKLYGDVPFIEERHRHRFEVNPNLIKQFEQNDLSFVGQDVDGDRMEIIELANHPYFVGVQFHPEFSSRPMKPSPPYLGLLLAATGNLNAYLQQ 6pl1 A 2.03 BS01 OOJ A 1 A542 E560 L564 F589 Y591 M592 F646 H648 L657 G667 D668 F669 M671 A43 E58 L62 F87 Y89 M90 F144 H146 L155 G165 D166 F167 M169 D650 R654 N655 D668 D148 R152 N153 D166 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Kd=0.000000064M remove_due_to_license_issue Ki=67nM, Kd=1.1nM, IC50=263nM P04629 31610943 801 ACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 6pl2 A 2.59 BS01 OOM A 1 V524 A542 K544 R559 E560 L564 F589 F646 H648 L657 G667 D668 F669 V26 A44 K46 R61 E62 L66 F91 F148 H150 L159 G169 D170 F171 D650 R654 N655 D668 D152 R156 N157 D170 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue P04629 31444087 801 DACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 6pl3 A 3.0 BS01 OOD A 1 A542 E560 L564 F589 H648 L657 G667 D668 F669 A43 E60 L64 F89 H144 L153 G163 D164 F165 D650 R654 N655 D668 D146 R150 N151 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 remove_due_to_license_issue IC50=3.0nM P04629 31444087 801 ACVHHIKRRDIVLKWELGEGAFGKVFLAECHNLLPEQDKMLVAVKALKESESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAPPVYLDVL 6plf A 1.7 BS01 ONV A 1 Y174 D175 P176 L193 H206 T207 P208 L216 Y170 D171 P172 L189 H202 T203 P204 L212 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 ic50=0.238uM remove_due_to_license_issue IC50=238nM, Ki=214nM O43175 31327531 401 NLRKVLISDSLDPCCRKILQDGGLQVVEKQNLSKEELIAELQDCEGLIVRSATKVTADVINAAEKLQVVGRAGTGVDNVDLEAATRKGILVMNTPNGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQFVDMVKG 6plg A 2.93 BS01 ONS A 1 G154 R155 D175 P176 I177 I178 H206 T207 L210 G149 R150 D170 P171 I172 I173 H201 T202 L205 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 remove_due_to_license_issue IC50=15nM O43175 31327531 401 LRKVLISDSLDPCCRKILQDGGLQVVEKQNLSKEELIAELQDCEGLIVRSATKVTADVINAAEKLQVVGRAGTGVDNVDLEAATRKGILVMNTPNGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQFVDMVK 6pm9 A 2.86 BS01 OQ1 A 1 G67 Y69 K98 D174 D175 Y219 T250 V254 W278 N280 D285 N313 G9 Y11 K40 D116 D117 Y161 T192 V196 W220 N222 D227 N255 3.2.1.169 remove_due_to_license_issue Ki=5.70nM, EC50=53nM, IC50=7.9nM O60502 31487175 501 RFLCGVVEGFYGRPWVMEQRKELFRRLQKWELNTYLYAPKDDYKHRMFWREMYSVEEAEQLMTLISAAREYEIEFIYAISPGLDITFSNPKEVSTLKRKLDQVSQFGCRSFALLFDDIDHNMCAADKEVFSSFAHAQVSITNEIYQYLGEPETFLFCPTEYCGTFCYPNVSQSPYLRTVGEKLLPGIEVLWTGPKVVSKEIPVESIEEVSKIIKRAPVIWDNIHANDYDQKRLFLGPYKGRSTELIPRLKGVLTNPNCEFEANYVAIHTLATWYKSNMNGVRDVLYSPQMALKLALTEWLQEFGVPHQY 6pml A 2.0 BS01 OR4 A 1 H32 F36 P151 P163 T168 M171 H32 F36 P151 P163 T168 M171 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=820uM remove_due_to_license_issue P0AEG4 31635355 202 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 6pnm A 1.82 BS01 XX0 A 1 C32 P33 F34 I131 W222 L226 Y229 C30 P31 F32 I129 W220 L224 Y227 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue Ki=6700nM, IC50=160nM P78417 32105470 1001 GESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 6pnn A 2.1 BS01 OR7 A 1 C32 P33 F34 I131 F225 Y229 C29 P30 F31 I128 F222 Y226 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue IC50=80nM, Ki=6900nM P78417 32105470 904 ESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 6pno A 1.82 BS01 ORM A 1 C32 F34 Y229 C30 F32 Y227 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 remove_due_to_license_issue Ki=4800nM, IC50=70nM P78417 32105470 1001 GESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL 6poh A 1.67 BS01 OVG A 1 H32 F36 P163 H32 F36 P163 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=1970uM remove_due_to_license_issue P0AEG4 31635355 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 6poi A 1.77 BS01 OVS A 1 H32 F36 P163 Q164 T168 M171 F174 H32 F36 P163 Q164 T168 M171 F174 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=326uM remove_due_to_license_issue P0AEG4 31635355 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 6poq A 1.8 BS01 OVJ A 1 H32 Q35 P151 P163 T168 H32 Q35 P151 P163 T168 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=2700uM remove_due_to_license_issue P0AEG4 31635355 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 6ppy A 2.0 BS01 OVY A 1 K53 Q55 N74 T110 K129 G131 Y186 D247 K52 Q54 N73 T109 K128 G130 Y185 D246 2.5.1.56 0016051,0016740,0046872,0047444,0050462,0070085 remove_due_to_license_issue H2VFG5 31549502 401 QNNNEFKIGNRSVGYNHEPLIICEIGINHEGSLKTAFEMVDAAYNAGAEVVKHQTHIVEDEMSDEAKQVIPGNADVSIYEIMERCALNEEDEIKLKEYVESKGMIFISTPFSRAAALRLQRMDIPAYKIGSGECNNYPLIKLVASFGKPIILSTGMNSIESIKKSVEIIREAGVPYALLHCTNIYPTPYEDVRLGGMNDLSEAFPDAIIGLSDHTLDNYACLGAVALGGSILERHFTDRMDRPGPDIVCSMNPDTFKELKQGAHALKLARGGKKDTIIAGEKPTKDFAFASVVADKDIKKGELLSGDNLWVKRPGNGDFSVNEYETLFGKVAACNIRKGAQIKKTDIE 6prc L 2.3 BS04 CEB L 1 F216 V220 Y222 S223 I224 G225 A226 I229 F216 V220 Y222 S223 I224 G225 A226 I229 ? 0009772,0015979,0016020,0019684,0030077,0042314,0042717,0045156,0046872 remove_due_to_license_issue P06009 10024457 502 ALLSFERKYRVRGGTLIGGDLFDFWVGPYFVGFFGVSAIFFIFLGVSLIGYAASQGPTWDPFAISINPPDLKYGLGAAPLLEGGFWQAITVCALGAFISWMLREVEISRKLGIGWHVPLAFCVPIFMFCVLQVFRPLLLGSWGHAFPYGILSHLDWVNNFGYQYLNWHYNPGHMSSVSFLFVNAMALGLHGGLILSVANPGDGDKVKTAEHENQYFRDVVGYSIGALSIHRLGLFLASNIFLTGAFGTIASGPFWTRGWPEWWGWWLDIPFWS 6prt A 1.3 BS01 OWA A 1 F83 L92 N140 F41 L50 N98 ? ic50=2120uM remove_due_to_license_issue IC50=2120000nM O60885 31727451 201 SNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6ps0 A 3.4 BS01 CAU A 1 T110 D113 V114 F193 S203 S207 W286 F289 F290 N293 N312 Y316 T80 D83 V84 F163 S173 S177 W384 F387 F388 N391 N410 Y414 ?,3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue D9IEF7,P07550 31709066 1201 VWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIWTLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6ps1 A 3.2 BS01 TIM A 1 D113 V114 V117 F193 S203 W286 F289 F290 N293 N312 D85 V86 V89 F165 S175 W386 F389 F390 N393 N412 ?,3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue D9IEF7,P07550 31709066 1201 DEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIWTLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6ps3 A 2.5 BS01 CVD A 1 D113 V117 F193 S203 F289 F290 N293 N312 Y316 D85 V89 F165 S175 F389 F390 N393 N412 Y416 ?,3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 Ki=0.166nM remove_due_to_license_issue D9IEF7,P07550 31709066 1201 DEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIWTLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6ps4 A 2.6 BS01 JRZ A 1 W109 D113 V114 S203 F289 F290 N312 W81 D85 V86 S175 F389 F390 N412 ?,3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue D9IEF7,P07550 31709066 1201 DEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIWTLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6ps5 A 2.9 BS01 SNP A 1 D113 F193 S203 F289 F290 N312 D85 F165 S175 F389 F390 N412 ?,3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue D9IEF7,P07550 31709066 1201 DEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIWTLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6ps6 A 2.7 BS01 TIM A 1 D113 V114 V117 F193 S203 W286 F289 F290 N293 N312 D86 V87 V90 F166 S176 W387 F390 F391 N394 N413 ?,3.2.1.17 0003796,0004930,0004941,0006940,0007186,0007189,0009253,0016020,0016798,0016998,0030430,0031640,0042742,0044659,0097746 remove_due_to_license_issue D9IEF7,P07550 31709066 1201 RDEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIWTLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYAEETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLNAAKSELDKAIGRNTNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRAALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVITTFRTGTWDAYKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCL 6ps9 A 1.21 BS01 Y17 A 1 W81 F83 N140 D144 D145 I146 W39 F41 N98 D102 D103 I104 ? ic50=79uM remove_due_to_license_issue IC50=79000nM O60885 31727451 201 SNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE 6psb A 1.59 BS01 Y18 A 1 W81 P82 N140 D144 I146 W39 P40 N98 D102 I104 ? ic50=24uM remove_due_to_license_issue IC50=24000nM O60885 31727451 201 SNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE 6pt3 A 3.3 BS01 OWY A 1 A98 D128 Y129 S131 M132 V217 W274 I277 H278 V281 W284 L300 G307 Y308 S311 A166 D196 Y197 S199 M200 V285 W342 I345 H346 V349 W352 L368 G375 Y376 S379 ? 0004930,0004985,0005506,0007186,0009055,0016020,0020037,0022900,0038046,0042597 remove_due_to_license_issue P41143 31807708 1201 TMADLEDNWETLNDNLKVIEKADNAAQVKDALTKMRAAALDAQKATPPKLEDKSPDSPEMKDFRHGFDILVGQIDDALKLANEGKVKEAQAAAEQLKTTRNAYIQKYLRSASSLALAIAITALYSAVCAVGLLGNVLVMFVIVRYTKMKTATNIYIFSLALAGALATSTLPFQSADYLMETWPFGELLCKAVLSIDYYSMFTSIFTLTMMCVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVVAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAALHLCIALGYINSSLNPVLYAFLDKNFKRCF 6pun A 2.099 BS01 rna B 0 N244 Y245 K284 R288 Q291 Q322 N323 H326 Q329 K360 Y361 R364 Q367 N415 Y416 Q419 K450 S453 H454 E457 N500 Y501 Q504 S553 S554 K557 N78 Y79 K118 R122 Q125 Q156 N157 H160 Q163 K194 Y195 R198 Q201 N243 Y244 Q247 K278 S281 H282 E285 N328 Y329 Q332 S381 S382 K385 ? 0003723 remove_due_to_license_issue Q09312 31397673 1 ~ 8 VLPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTALTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGGYDHAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLANLRST 6pun C 2.099 BS01 rna D 0 N244 Y245 F285 R288 Q291 Q322 N323 H326 Q329 K360 Y361 C363 R364 Q367 N415 Y416 Q419 K450 S453 H454 E457 F498 N500 Y501 Q504 S553 S554 K557 N78 Y79 F119 R122 Q125 Q156 N157 H160 Q163 K194 Y195 C197 R198 Q201 N243 Y244 Q247 K278 S281 H282 E285 F326 N328 Y329 Q332 S377 S378 K381 ? 0003723 remove_due_to_license_issue Q09312 31397673 2 ~ 8 VLPTWSLDSNGEMRSRLSLSEVLDSGDLMKFAVDKTGCQFLEKAVKGSLTSYQKFQLFEQVIGRKDDFLKLSTNIFGNYLVQSVIGISLATNDDGYTKRQEKLKNFISSQMTDMCLDKFACRVIQSSLQNMDLSLACKLVQALPRDARLIAICVDQNANHVIQKVVAVIPLKNWEFIVDFVATPEHLRQICSDKYGCRVVQTIIEKLTALTSAAQNLRERALQRLMTSVTNRCQELATNEYANYIIQHIVSNDDLAVYRECIIEKCLMRNLLSLSQEKFASHVVEKAFLHAPLELLAEMMDEIFDGYIPHPDTGKDALDIMMFHQFGNYVVQCMLTICCDAVSGRRQTKEGAISFQDWLKKLHSRVTKERHRLSRFSSGKKMIETLAN 6pve A 2.3 BS01 OZP A 1 Y11 Y20 Y25 G63 S64 G65 T67 Y69 D85 Y86 D142 T163 L164 C165 A169 A198 S201 Y204 S213 Y242 Y21 Y30 Y35 G73 S74 G75 T77 Y79 D95 Y96 D152 T173 L174 C175 A179 A208 S211 Y214 S223 Y252 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0030760,0031100,0032259,0034356,0045722,0090312 Ki=43nM remove_due_to_license_issue P40261 31724854 301 HSSGLVPRGSMESGFTSKDTYLSHFNPRDYLEKYYKFGSRHSAESQILKHLLKNLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIVVTDYSDQNLQELEKWLKAAPAAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPPADCVLSTLCLDAACPDLPTYCRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVARKL 6pvs A 2.575 BS01 P0V A 1 Y20 Y25 G63 S64 G65 T67 D85 Y86 D142 V143 T163 L164 S201 Y203 Y204 S213 Y242 Y30 Y35 G73 S74 G75 T77 D95 Y96 D152 V153 T173 L174 S211 Y213 Y214 S223 Y252 2.1.1.1 0005737,0005829,0006769,0008112,0008168,0008757,0009410,0030760,0031100,0032259,0034356,0045722,0090312 remove_due_to_license_issue P40261 31724854 301 HSSGLVPRGSMESGFTSKDTYLSHFNPRDYLEKYYKFGSRHSAESQILKHLLKNLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIVVTDYSDQNLQELEKWLKAAPAAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPPADCVLSTLCLDAACPDLPTYCRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVARKL 6pvu A 1.49 BS01 P0S A 1 K7 Q11 H12 R39 K41 H119 K7 Q11 H12 R39 K41 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue P61823 31651164 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 6pvw A 1.6 BS01 OZV A 1 K7 Q11 H12 K41 N67 Q69 N71 A109 E111 H119 K7 Q11 H12 K41 N67 Q69 N71 A109 E111 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=0.48uM remove_due_to_license_issue P61823 31651164 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 6pvx A 1.55 BS01 U5F A 1 H12 K41 V43 N44 T45 F120 H12 K41 V43 N44 T45 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676 Ki=0.068uM remove_due_to_license_issue P61823 31651164 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 6pvx A 1.55 BS02 U5F A 2 K7 R10 Q11 C65 N67 Q69 N71 A109 E111 V118 H119 K7 R10 Q11 C65 N67 Q69 N71 A109 E111 V118 H119 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676 Ki=0.068uM remove_due_to_license_issue P61823 31651164 202 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 6pvy A 1.74 BS01 OZG A 1 H32 Q35 F36 L40 V150 P151 T168 F174 H32 Q35 F36 L40 V150 P151 T168 F174 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=639uM remove_due_to_license_issue P0AEG4 31635355 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 6pvz A 1.99 BS01 OZM A 1 H32 Q35 F36 P163 Q164 T168 M171 F174 H32 Q35 F36 P163 Q164 T168 M171 F174 ? 0003756,0005515,0015035,0015036,0016491,0030288,0042597,0071236 Kd=341uM remove_due_to_license_issue P0AEG4 31635355 201 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEK 6pw2 A 3.01 BS01 dna E 0 K461 W464 F465 R469 G470 G472 G473 K514 Y518 R522 P535 L536 R538 P587 K1 W4 F5 R9 G10 G12 G13 K54 Y58 R62 P75 L76 R78 P127 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 3 ~ 59 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 A 3.01 BS02 dna F 0 K461 G462 G463 W464 H468 R469 K477 N480 I481 T515 N519 P589 T590 K1 G2 G3 W4 H8 R9 K17 N20 I21 T55 N59 P129 T130 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 5 ~ 57 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 B 3.01 BS01 dna E 0 K461 G462 G463 W464 R469 S513 T515 S516 N519 P589 T590 K1 G2 G3 W4 R9 S53 T55 S56 N59 P129 T130 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 3 ~ 59 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 B 3.01 BS02 dna F 0 W464 F465 K467 R469 G470 G472 Y518 R521 R522 P535 L536 W4 F5 K7 R9 G10 G12 Y58 R61 R62 P75 L76 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 5 ~ 57 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 C 3.01 BS01 dna E 0 G462 G463 W464 H468 R469 K477 N480 S513 T515 N519 K586 P589 T590 G2 G3 W4 H8 R9 K17 N20 S53 T55 N59 K126 P129 T130 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 3 ~ 59 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 C 3.01 BS02 dna F 0 K461 F465 K467 G470 Q471 G472 G473 K514 Y518 R521 R522 P535 L536 K1 F5 K7 G10 Q11 G12 G13 K54 Y58 R61 R62 P75 L76 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 5 ~ 57 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 D 3.01 BS01 dna E 0 K461 F465 K467 R469 G470 G472 K514 Y518 R522 P535 L536 R538 K1 F5 K7 R9 G10 G12 K54 Y58 R62 P75 L76 R78 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 3 ~ 59 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 D 3.01 BS02 dna F 0 K461 G462 G463 W464 H468 R469 N519 K586 P589 T590 K1 G2 G3 W4 H8 R9 N59 K126 P129 T130 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 5 ~ 57 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 I 3.01 BS01 dna G 0 K461 F465 G470 G472 G473 N475 K514 Y518 R521 R522 P535 L536 R538 K1 F5 G10 G12 G13 N15 K54 Y58 R61 R62 P75 L76 R78 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 8 ~ 56 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 I 3.01 BS02 dna H 0 K461 G462 G463 W464 R469 K477 N480 S513 T515 N519 P589 K1 G2 G3 W4 R9 K17 N20 S53 T55 N59 P129 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 7 ~ 55 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 J 3.01 BS01 dna G 0 K461 G462 G463 W464 H468 K477 S513 T515 P589 T590 K1 G2 G3 W4 H8 K17 S53 T55 P129 T130 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 8 ~ 56 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 J 3.01 BS02 dna H 0 K461 W464 F465 K467 G470 G472 G473 K514 Y518 R522 P535 L536 R538 K1 W4 F5 K7 G10 G12 G13 K54 Y58 R62 P75 L76 R78 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 7 ~ 55 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 K 3.01 BS01 dna G 0 K461 G462 G463 W464 K477 N480 S513 T515 N519 K586 P589 K1 G2 G3 W4 K17 N20 S53 T55 N59 K126 P129 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 8 ~ 56 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 K 3.01 BS02 dna H 0 K461 F465 K467 G470 G472 K514 Y518 R521 R522 P535 L536 R538 K1 F5 K7 G10 G12 K54 Y58 R61 R62 P75 L76 R78 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 7 ~ 55 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 L 3.01 BS01 dna G 0 K461 F465 R469 G470 G472 K514 Y518 R522 P535 L536 R538 K1 F5 R9 G10 G12 K54 Y58 R62 P75 L76 R78 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 8 ~ 56 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6pw2 L 3.01 BS02 dna H 0 K461 G462 G463 W464 H468 R469 T515 N519 K586 P589 T590 K1 G2 G3 W4 H8 R9 T55 N59 K126 P129 T130 3.1.21.- 0003677,0003700,0006275,0006355,0042025,0045893 remove_due_to_license_issue P03211 31142669 7 ~ 55 KGGWFGKHRGQGGSNPKFENIAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLPFGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSFDDGVDLP 6py0 A 2.204 BS01 RTL C 1 A79 A82 V83 A60 A63 V64 ? 0005576,0005615,0006953,0009617,0034364,0035634,0035662,0042056,0050918,0060326,0071347 remove_due_to_license_issue P04918 31484771 201 RWVQFMKEAGQGSRDMWRAYSDMKKANWKNSDKYFHARGNYDAARRGPGGAWAAKVISDAREAVQKFTGHGDSRADQFANEWGRSGKDPNHFRPAGLPKRY 6pya A 1.71 BS01 P57 A 1 S42 F67 V105 M107 M139 L171 S29 F54 V92 M94 M126 L158 ? ic50=150nM remove_due_to_license_issue P04278 31852737 301 PAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGPLTSKRHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAKISASAPTSLRSC 6pyb A 1.8 BS01 P5G A 1 D65 F67 L80 N82 M107 R135 M139 D52 F54 L67 N69 M94 R119 M123 ? ic50=4200nM remove_due_to_license_issue IC50=2600nM, Kd=309nM P04278 31852737 301 PAVHLSNGPGQEPIAVMTFDLTKITKTSSSFEVRTWDPEGVIFYGDTNPKDDWFMLGLRDGRPEIQLHNHWAQLTVGAGPRLDDGRWHQVEVKMEGDSVLLEVDGEEVLRLRQVSGPKRHPIMRIALGGLLFPASNLRLPLVPALDGCLRRDSWLDKQAKISASAPTSLRSC 6pyc H 3.6 BS01 P4S H 1 Y97 I100 Y96 I99 remove_due_to_license_issue 31879340 301 IVMTQSPDSLAVSLGERATINCKSSQSVLYSSNNKNYLAWFQQKPGQPPKLLIYWASLRESGVSDRFSGSGSGTDFTLTISGLQAEDVAVYYCQQYYSILWTFGQGTKVEIKSTKGPSVFPLAPCTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTKTYTCNVDHKPSNTKVDKRVES 6pyc H 3.6 BS02 P4S L 1 Q95 W102 Q94 W101 remove_due_to_license_issue 31879340 301 IVMTQSPDSLAVSLGERATINCKSSQSVLYSSNNKNYLAWFQQKPGQPPKLLIYWASLRESGVSDRFSGSGSGTDFTLTISGLQAEDVAVYYCQQYYSILWTFGQGTKVEIKSTKGPSVFPLAPCTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTKTYTCNVDHKPSNTKVDKRVES 6pyc L 3.6 BS01 P4S L 1 Q90 Y92 Y97 Q90 Y92 Y97 remove_due_to_license_issue 31879340 301 EIVLTQSPGTLSLSPGERATLSCRASQSVGNNYLAWFQQKPGQAPRLLIYGASSRATGIPDRFSGSGSGTDFTLTISRLEPEDFVVYYCQQYSRSPYIFGQGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRG 6pyd H 2.0 BS01 P4S H 1 Y50 Y100 G101 G103 Y49 Y99 G100 G102 remove_due_to_license_issue 31879340 301 VQLQESGPSLVKPSQTLSLTCSVTGDSITSGYWNWIRKFPGNKLEYMGYISYSGTTYYNPSLKSRISITRDTSKNQYYLQLNSVTTEDTATYYCARARYGYGFDYWGQGTTLTVSSASTKGPSVFPLAPTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTKTYTCNVDHKPSNTKVDKRVESKY 6pyd L 2.0 BS01 P4S H 1 Y36 E38 G95 Y29 E31 G88 remove_due_to_license_issue 31879340 301 VLMTQTPLSLPVSLGDQASISCRSSQSTYLEWYLQKPGQSPKLLIYKVSNRFSGVPDRFSGSGSGTDFTLKISRVEAEDLGVYYCFQGSHVPLTFGAGTKLELKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNR 6pyr A 2.21 BS01 P5J A 1 W760 I825 V828 N836 M900 D911 W684 I744 V747 N755 M809 D820 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 ic50=1nM remove_due_to_license_issue IC50=1.000000nM O00329 31416665 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPSNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKATVRQVEQPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDESSVSLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEKAADCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHTEEEQLQLREILEGELYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEESVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLNNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNFERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVN 6pys A 2.19 BS01 P5J A 1 M772 S774 W780 I800 K802 Y836 I848 V851 T856 M922 I932 M628 S630 W636 I656 K658 Y692 I704 V707 T712 M769 I779 2.7.11.1,2.7.1.137,2.7.1.153 0016301,0046854 remove_due_to_license_issue P42336 31416665 1101 NREEKILNREIGFAIGMPVCEFDMVKDPEVQDFRRNILNVCKEAVDLRDLNSPHSRAMYVYPPNVESSPELPKHIYNKLDKGQIIVVIWVIVSDKQKYTLKINHDCVPEQVIAEAIRKKTRSMYQGKYILKVCGCDEYFLEKYPLSQYKYIRSCIMLGRMPNLMLMAKESLYSQLPMDCFTMPSYSRTSTKSLWVINSALRIKILCATYVNVNIDKIYVRTGIYHGGEPLCDNVNTQRVPCSNPRWNEWLNYDIYIPDLPRAARLCLSICSVEEHCPLAWGNINLFDYTDTLVSGKMALNLWPVPHGLEDLLNPIGVTGSNPNKETPCLELEFDWFSSVVKFPDMSVIEEHANWSVSREAGFSYSHAGLSNRLARDNELRENDKEQLKAISTRDPLSEITEQEKDFLWSHRHYCVTIPEILPKLLLSVKWNSRDEVAQMYCLVKDWPPIKPEQAMELLDCNYPDPMVRGFAVRCLEKYLTDDKLSQYLIQLVQVLKYEQYLDNLLVRFLLKKALTNQRIGHFFFWHLKSEMHNKTVSQRFGLLLESYCRACGMYLKHLNRQVEAMEKLINLTDILKQEKKDETQKVQMKFLVEQMRRPDFMDALQGFLSPLNPAHQLGNLRLEECRIMSSAKRPLWLNWENPDIMSELLFQNNEIIFKNGDDLRQDMLTLQIIRIMENIWQNQGLDLRMLPYGCLSIGDCVGLIEVVRNSHTIMQIQCKNSHTLHQWLKDKNKGEIYDAAIDLFTRSCAGYCVATFILGIGDRHNSNIMVKDDGQLFHIDFGHFLDHRERVPFVLTQDFLIVISKGAQECTKTREFERFQEMCYKAYLAIRQHANLFINLFSMMLGSGMPELQSFDDIAYIRKTLALDKTEQEALEYFMKQMNDAHHGGW 6pyu A 2.54 BS01 P5V A 1 T750 W760 Y813 I825 E826 V828 N836 M900 T667 W677 Y730 I742 E743 V745 N753 M805 2.7.1.137,2.7.1.153 0001779,0001819,0001938,0002250,0002551,0002679,0005515,0005524,0005737,0005829,0005886,0005942,0005943,0006468,0006629,0006935,0006954,0006955,0007165,0010595,0010628,0010818,0016301,0016303,0030101,0030154,0030183,0030217,0030335,0030593,0033031,0035005,0035747,0035754,0036092,0038084,0042110,0042113,0043303,0043491,0045087,0045766,0046854,0046934,0048015,0050852,0050853,0060374,0072672,1905278 remove_due_to_license_issue IC50=10.0nM O00329 31416665 1101 NQSVVVDFLLPTGVYLNFPVSRNANLSTIKQLLWHRAQYEPLFHMLSGPEAYVFTCINQTAEQQELEDEQRRLCDVQPFLPVLRLVAREGDRVKKLINSQISLLIGKGLHEFDSLCDPEVNDFRAKMCQFCEEAAARRQQLGWEAWLQYSFPLQLEPSAPNRALLVNVKFEGSEESFTFQVSTKDVPLALMACALRKKATQPEDYTLQVNGRHEYLYGSYPLCQFQYICSCLHSGLTPHLTMVHSSSILAMRDEVSLWSLEQPFRIELIQGSKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVSVCSEPVWKQRLEFDINICDLPRMARLCFALYAVIEDCPIAWANLMLFDYKDQLKTGERCLYMWPSVPDEKGELLNPTGTVRSNPNTDSAAALLICLPEVAPHPVYYPALEKILELGRHSEEEQLQLREILERGELYEHEKDLVWKLRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCHVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLDRALANRKIGHFLFWHLRSEMHVPSVALRFGLILEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKLSSQKTPKPQTKELMHLCMRQEAYLEALSHLQSPLDPSTLLAEVCVEQCTFMDSKMKPLWIMYSNEEAGSGGSVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLRSDTIANIQLKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVNWL 6pz4 A 1.85 BS01 P6J A 1 G72 G74 Y75 D93 Y132 F169 D289 G291 T292 T293 A396 G13 G15 Y16 D34 Y73 F110 D222 G224 T225 T226 A329 3.4.23.46 0004190,0006508,0016020 ic50=0.4nM remove_due_to_license_issue IC50=1.2nM P56817 31589043 506 FVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNI 6q2y A 1.0 BS05 HCQ A 1 M67 W93 H122 Q123 D124 H189 N220 M28 W54 H83 Q84 D85 H150 N181 H120 H122 D124 H189 C208 K211 N220 H250 H81 H83 D85 H150 C169 K172 N181 H211 3.5.2.6 remove_due_to_license_issue C7C422 30996812 305 ETGDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6q30 A 1.5 BS05 HCH A 1 L65 W93 H122 Q123 D124 H189 N220 L24 W52 H81 Q82 D83 H148 N179 H120 H122 D124 H189 C208 K211 N220 H250 H79 H81 D83 H148 C167 K170 N179 H209 3.5.2.6 remove_due_to_license_issue C7C422 30996812 305 GDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6q35 A 1.4 BS01 HD5 A 1 C63 S64 W99 N127 E161 S165 T232 C45 S46 W81 N109 E143 S147 T214 S64 K67 S125 E161 K229 T232 S46 K49 S107 E143 K211 T214 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue Q09HD0 30996812 404 SEKLTFKTDLEKLEREKAAQIGVAIVDPQGEIVAGHRMAQRFAMCSTFKFPLAALVFERIDSGTERGDRKLSYGPDMIVEWSPATERFLASGHMTVLEAAQAAVQLSDNGATNLLLREIGGPAAMTQYFRKIGDSVSRLDRKEPEMSDNTPGDLRDTTTPIAMARTVAKVLYGGALTSTSTHTIERWLIGNQTGDATLRAGFPKDWVVGEKTGTCANGGRNDIGFFKAQERDYAVAVYTTAPKLSAVERDELVASVGQVITQLILST 6q37 A 2.211 BS03 HE8 A 1 H120 D143 H145 D147 N149 S156 H160 G161 D202 D251 H97 D120 H122 D124 N126 S133 H137 G138 D179 D228 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=440nM remove_due_to_license_issue P78540 31408339 405 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 6q39 A 2.213 BS03 HDQ A 1 H120 D143 H145 D147 N149 S156 H160 D200 D202 D251 T265 E296 H97 D120 H122 D124 N126 S133 H137 D177 D179 D228 T242 E273 H120 D143 H145 D147 H160 D251 D253 E296 H97 D120 H122 D124 H137 D228 D230 E273 3.5.3.1 0004053,0006525,0016813,0046872 ic50=16nM remove_due_to_license_issue P78540 31408339 405 HSVAVIGAPFSQGQKRKGVEHGPAAIREAGLMKRLSSLGCHLKDFGDLSFTPVPKDDLYNNLIVNPRSVGLANQELAEVVSRAVSDGYSCVTLGGDHSLAIGTISGHARHCPDLCVVWVDAHADINTPLTTSSGNLHGQPVSFLLRELQDKVPQLPGFSWIKPCISSASIVYIGLRDVDPPEHFILKNYDIQYFSMRDIDRLGIQKVMERTFDLLIGKRQRPIHLSFDIDAFDPTLAPATGTPVVGGLTYREGMYIAEEIHNTGLLSALDLVEVNPQLATSEEEAKTTANLAVDVIASSFGQTREG 6q3y A 1.2 BS01 HG5 A 1 W81 P82 Q85 V87 L92 L94 Y97 Y139 W39 P40 Q43 V45 L50 L52 Y55 Y97 ? Kd=54nM remove_due_to_license_issue IC50=540nM, Kd=54nM O60885 30789735 202 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6q3y A 1.2 BS02 HG5 B 1 H77 Q78 F79 L148 M149 H35 Q36 F37 L106 M107 ? Kd=54nM remove_due_to_license_issue IC50=540nM, Kd=54nM O60885 30789735 204 MNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT 6q3z A 2.0 BS01 HG8 A 1 W81 P82 Q85 V87 L92 Y97 D145 I146 W40 P41 Q44 V46 L51 Y56 D104 I105 ? Kd=44nM remove_due_to_license_issue Kd=44nM, IC50=260nM O60885 30789735 201 SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELP 6q4e A 1.06 BS01 HH5 A 1 A31 K33 V64 F80 F82 L83 L134 A32 K34 V58 F74 F76 L77 L128 D127 K129 Q131 N132 D145 T165 D121 K123 Q125 N126 D139 T151 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=350uM remove_due_to_license_issue P24941 30860382 303 FMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 6q4g A 0.98 BS01 HJK A 1 G13 T14 V18 A31 K33 F82 L83 Q131 L134 G13 T14 V18 A31 K33 F76 L77 Q125 L128 D127 K129 Q131 N132 D145 T165 D121 K123 Q125 N126 D139 T149 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 Kd=50uM remove_due_to_license_issue Kd=50000nM P24941 30860382 301 MENFEKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 6q54 A 1.4 BS01 HJ8 A 1 Y61 T91 R96 G141 S142 T143 L192 E193 Y61 T91 R96 G141 S142 T143 L192 E193 ? 0015276,0016020 remove_due_to_license_issue EC50=65000nM, Ki=710nM P19491 30943028 307 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECGSG 6q5b A 2.22 BS01 NXL A 1 A69 S70 S118 T209 G210 Y211 R250 A46 S47 S95 T177 G178 Y179 R218 S70 K73 S118 Y123 Y211 S47 K50 S95 Y100 Y179 3.5.2.6 0008658,0008800,0017001 remove_due_to_license_issue Q6XEC0 30918055 301 EWQENKSWNAHFTEHKSQGVVVLWNENKQQGFTNNLKRANQAFLAASTFKIPNSLIALDLGVVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDYGNEDIDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYIIRAKTGYSTRIEPKIGWWVGWVELDDNVWFFAMNMDMPTSDGLGLRQAITKEVLKQEKIIP 6q60 A 1.55 BS01 HJH A 1 Y61 T91 R96 G141 S142 T143 L192 E193 Y61 T91 R96 G141 S142 T143 L192 E193 ? 0015276,0016020 remove_due_to_license_issue Ki=1970nM P19491 30943028 301 GANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECGSG 6q6f A 3.3 BS01 HJQ A 1 L288 H309 G310 V312 T313 R314 N328 D375 L276 H297 G298 V300 T301 R302 N316 D363 1.1.1.42 0000287,0004450,0005515,0005576,0005737,0005739,0005777,0005782,0005829,0006097,0006099,0006102,0006103,0006739,0006749,0006979,0008585,0014070,0016491,0016616,0034774,0042802,0042803,0045296,0046872,0048545,0050661,0051287,0060696,0070062,0071071,1904724,1904813 remove_due_to_license_issue O75874 31586149 501 MSKKISGGSVVEMQGDEMTRIIWELIKEKLIFPYVELDLHSYDLGIENRDATNDQVTKDAAEAIKKHNVGVKCATITPDEKRVEEFKLKQMWKSPNGTIRNILGGTVFREAIICKNIPRLVSGWVKPIIIGHHAYGDQYRATDFVVPGPGKVEITYTPSDGTQKVTYLVHNFEEGGGVAMGMYNQDKSIEDFAHSSFQMALSKGWPLYLSTKNTILKKYDGRFKDIFQEIYDKQYKSQFEAQKIWYEHRLIDDMVAQAMKSEGGFIWACKNGYGSLGMMTSVLVCPDGKTVEAEAAHGTVTRHYRMYQKGQETSTNPIASIFAWTRGLAHRAKLDNNKELAFFANALEEVSIETIEAGFMTKDLAACIKGLPNVQRSDYLNTFEFMDKLGENLKIKLAQAKL 6q6m A 2.35 BS01 HJW A 1 C320 H323 L324 V361 V376 F388 L391 I397 H479 C56 H59 L60 V97 V112 F124 L127 I133 H215 ? 0003677,0004879,0005634,0006355 ic50=128nM remove_due_to_license_issue IC50=128nM P51449 31729873 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLH 6q6o A 2.3 BS01 HKE A 1 W317 C320 H323 L324 V361 M365 F388 I397 I400 H479 L483 W53 C56 H59 L60 V97 M101 F124 I133 I136 H215 L219 ? 0003677,0004879,0005634,0006355 ic50=29nM remove_due_to_license_issue IC50=452nM P51449 31729873 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLH 6q6y A 2.03 BS01 HKQ A 1 W760 I777 K779 Y813 I825 E826 V828 D897 M900 I910 D911 W598 I615 K617 Y651 I663 E664 V666 D735 M738 I748 D749 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 30532965 4001 DRVKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSARNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLVEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNPASLWSLEQPFSIELIEGRKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPHPVYFPALEKILELGRHGERGRITEEEQLQLREILERGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVN 6q73 A 2.21 BS01 HKK A 1 M752 W760 I777 K779 Y813 I825 E826 V827 V828 M900 I910 D911 M591 W599 I616 K618 Y652 I664 E665 V666 V667 M739 I749 D750 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 30532965 4001 DRVKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSARGNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLVEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNPASLWSLEQPFSIELIEGRKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPHPVYFPALEKILELGRHGERGRITEEEQLQLREILERGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNRERVPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTKVN 6q74 A 2.48 BS01 HKN A 1 M752 W760 I777 K779 D787 Y813 I825 E826 V827 V828 T833 D897 M900 I910 D911 M588 W596 I613 K615 D623 Y649 I661 E662 V663 V664 T669 D733 M736 I746 D747 2.7.1.137,2.7.1.153 0016301,0016303,0043491,0046854 remove_due_to_license_issue O35904 30532965 4001 DRVKKLINSQISLLIGKGLHEFDSLRDPEVNDFRTKMRQFCEEAAAHRQQLGWVEWLQYSFPLQLEPSARGNRALLVNVKFEGSEESFTFQVSTKDMPLALMACALRKKATVFRQPLVEQPEEYALQVNGRHEYLYGNYPLCHFQYICSCLHSGLTPHLTMVHSSSILAMRDEQSNPASLWSLEQPFSIELIEGRKVNADERMKLVVQAGLFHGNEMLCKTVSSSEVNVCSEPVWKQRLEFDISVCDLPRMARLCFALYAVVDCPIAWANLMLFDYKDQLKTGERCLYMWPSVLLNPAGTVRGNPNTESAAALVIYLPEVAPHPVYFPALEKILELGRHGERITEEEQLQLREILEGELYEHEKDLVWKMRHEVQEHFPEALARLLLVTKWNKHEDVAQMLYLLCSWPELPVLSALELLDFSFPDCYVGSFAIKSLRKLTDDELFQYLLQLVQVLKYESYLDCELTKFLLGRALANRKIGHFLFWHLRSEMHVPSVALRFGLIMEAYCRGSTHHMKVLMKQGEALSKLKALNDFVKVSSQKTTKPQTKEMMHMCMRQETYMEALSHLQSPLDPSTLLEEVCVEQCTFMDSKMKPLWIMYSSEEAGSAGNVGIIFKNGDDLRQDMLTLQMIQLMDVLWKQEGLDLRMTPYGCLPTGDRTGLIEVVLHSDTIANIQLNKSNMAATAAFNKDALLNWLKSKNPGEALDRAIEEFTLSCAGYCVATYVLGIGDRHSDNIMIRESGQLFHIDFGHFLGNPFILTYDFVHVIQQGKTNNSEKFERFRGYCERAYTILRRHGLLFLHLFALMRAAGLPELSCSKDIQYLKDSLALGKTEEEALKHFRVKFNEALRESWKTK 6q7a A 2.2 BS01 HKZ A 1 W317 C320 H323 L324 V361 M365 V376 F388 I397 I400 H479 L483 F486 W53 C56 H59 L60 V97 M101 V112 F124 I133 I136 H215 L219 F222 ? 0003677,0004879,0005634,0006355 ic50=29nM remove_due_to_license_issue IC50=160nM P51449 31729873 501 ASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPI 6q7h A 2.3 BS01 HL8 A 1 L324 M358 L362 M365 V376 F378 F388 I400 H479 L58 M92 L96 M99 V110 F112 F122 I134 H213 ? 0003677,0004879,0005634,0006355 ic50=21nM remove_due_to_license_issue IC50=21nM P51449 31729873 501 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHP 6q7h A 2.3 BS02 HL8 A 2 T325 I328 V332 L353 T59 I62 V66 L87 ? 0003677,0004879,0005634,0006355 ic50=21nM remove_due_to_license_issue IC50=21nM P51449 31729873 502 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHP 6q7v A 2.56 BS01 HLK A 1 I149 A168 F221 I236 I263 I57 A76 F129 I144 I171 ? remove_due_to_license_issue Q9I4X0 31709767 400 RNLRVLLDTAIPPSFCDTVSSVLLDDFNMVSLIRTSPADSLATIKQDNAEIDIAITIDEELKISRFNQCVLGYTKAFVVAHPQHPLCNASLHSIASLANYRQISLGSRSGQHSNLLRPVSDKVLFVENFDDMLRLVEAGVGWGIAPHYFVEERLRNGTLAVLSELYEPGGIDTKVYCYYNTALESERSFLRFLESARQRLRELGRQ 6q7v B 2.56 BS01 HLK B 1 F221 I236 I263 F128 I143 I170 ? remove_due_to_license_issue Q9I4X0 31709767 400 NLRVLLDTAIPPSFCDTVSSVLLDDFNMVSLIRTSPADSLATIKQDNAEIDIAITIDEELKISRFNQCVLGYTKAFVVAHPQHPLCNASLHSIASLANYRQISLGSRSGQHSNLLRPVSDKVLFVENFDDMLRLVEAGVGWGIAPHYFVEERLRNGTLAVLSELYEPGGIDTKVYCYYNTALESERSFLRFLESARQRLREL 6q7w A 2.82 BS01 HLQ A 1 I149 L207 L208 I236 A237 Y258 I263 I57 L115 L116 I144 A145 Y166 I171 ? remove_due_to_license_issue Q9I4X0 31709767 400 RNLRVLLDTAIPPSFCDTVSSVLLDDFNMVSLIRTSPADSLATIKQDNAEIDIAITIDEELKISRFNQCVLGYTKAFVVAHPQHPLCNASLHSIASLANYRQISLGSRSGQHSNLLRPVSDKVLFVENFDDMLRLVEAGVGWGIAPHYFVEERLRNGTLAVLSELYEPGGIDTKVYCYYNTALESERSFLRFLESARQRLRELGR 6q89 A 2.21 BS01 LSS A 1 F41 P42 Y43 G51 H52 N55 D80 G543 G544 E546 H547 H551 Q580 M582 V583 F41 P42 Y43 G51 H52 N55 D80 G543 G544 E546 H547 H551 Q580 M582 V583 0000166,0002161,0004812,0004823,0005524,0006418,0006429 remove_due_to_license_issue 30995568 901 MQEHYQPAAIEPAAQKKWDDARISNVSEDASKPKYYCLSMFPYPSGKLHMGHVRNYTIGDVLSRFKLLNGFNVMQPMGWDAFGMPAENAAMKNNVAPAAWTYDNIEYMKTQLKSLGFAVDWEREVATCKPEYYRWEQWLFTKLFEKGIVYRKNGTVNWDPVDQTVLANEQVIDGRGWRSGALIEKREIPMYYFKITDYAEELLNDLDKLEHWPEQVKTMQRNWIGKSRGMTVRFAVSDDSKQGLEGDYAKFLQVYTTRPDTLMGATYVAVAAEHPLATAAAADKPELQAFIAECKAGSVAEADMATMEKKGVPTGRYVVNPLNGDKLEVWIANYVLWGYGDGAVMAVPAHDERDFEFAAKYNLPKKQVIAVGDNAFDANRWQEWYGDKENGVLVNSGDLDGLDFQTAFDAVAAKLQSQGAGEPKTQYRLRDWGISRQRYWGCPIPIVHCEKCGNVPVPADQLPVVLPENVVPDGMGSPLAKMPEFYETSCPCCGGAAKRETDTMDTFIESSWYFFRYMSPKFSDGMVSAESAKYWGAVDQYIGGIEHAILHLLYARFFTKLMRDEGLVNVDEPFERLLTQGMVVCETYYDWINPADVELDGLPVVISGTEKMSKSKNNGVDPQELINAYGADTARLFMMFAAPPEQSLEWSDSGVEGAHRFLRRLWRTVYEYLKQGGAVKAFAGNQDGLSKELKDLRHKLHSTTAKVSDDYGRRQQFNTAIAAVMELLNQYDKTDTGSEQGRAVAQEVLEAAVRLLWPIVPHICETLWSELNGAKLWEAGWPTVDEAALVKSEIEVMVQVNGKLRGKITVAADASKADLEAAALANEGAVKFMEGKPAKKIIVVPGRLVNIV 6q8a A 2.11 BS01 HQ5 A 1 M40 F41 P42 Y43 H49 G51 H52 N55 D80 S510 G543 G544 E546 H547 H551 Q580 M40 F41 P42 Y43 H49 G51 H52 N55 D80 S510 G543 G544 E546 H547 H551 Q580 F41 D80 F507 H547 F557 K634 K637 F41 D80 F507 H547 F557 K619 K622 6.1.1.4 0000166,0002161,0004812,0004823,0005524,0005737,0005829,0006412,0006418,0006429,0106074 remove_due_to_license_issue B4RNT1 30995568 901 MQEHYQPAAIEPAAQKKWDDARISNVSEDASKPKYYCLSMFPYPSGKLHMGHVRNYTIGDVLSRFKLLNGFNVMQPMGWDAFGMPAENAAMKNNVAPAAWTYDNIEYMKTQLKSLGFAVDWEREVATCKPEYYRWEQWLFTKLFEKGIVYRKNGTVNWDPVDQTVLANEQVIDGRGWRSGALIEKREIPMYYFKITDYAEELLNDLDKLEHWPEQVKTMQRNWIGKSRGMTVRFAVSDDSKQGLEGDYAKFLQVYTTRPDTLMGATYVAVAAEHPLATAAAADKPELQAFIAECKAGSVAEADMATMEKKGVPTGRYVVNPLNGDKLEVWIANYVLWGYGDGAVMAVPAHDERDFEFAAKYNLPKKQVIAVGDNAFDANRWQEWYGDKENGVLVNSGDLDGLDFQTAFDAVAAKLQSQGAGEPKTQYRLRDWGISRQRYWGCPIPIVHCEKCGNVPVPADQLPVVLPENVVPDGMGSPLAKMPEFYETSCPCCGGAAKRETDTMDTFIESSWYFFRYMSPKFSDGMVSAESAKYWGAVDQYIGGIEHAILHLLYARFFTKLMRDEGLVNVDEPFERLLTQGMVVCETYYRENDKGGKDWINPADVELTGLPVVISGTEKMSKSKNNGVDPQELINAYGADTARLFMMFAAPPEQSLEWSDSGVEGAHRFLRRLWRTVYEYLKQGGAVKAFAGNQDGLSKELKDLRHKLHSTTAKVSDDYGRRQQFNTAIAAVMELLNQYDKTDTGSEQGRAVAQEVLEAAVRLLWPIVPHICETLWSELNGAKLWEAGWPTVDEAALVKSEIITVAADIIVVPGRLVNIV 6q8b A 2.2 BS01 L3U A 1 M40 F41 P42 Y43 H49 G51 H52 N55 D80 G544 E546 H547 H551 Q580 M40 F41 P42 Y43 H49 G51 H52 N55 D80 G540 E542 H543 H547 Q576 0000166,0002161,0004812,0004823,0005524,0006418,0006429 remove_due_to_license_issue 30995568 901 MQEHYQPAAIEPAAQKKWDDARISNVSEDASKPKYYCLSMFPYPSGKLHMGHVRNYTIGDVLSRFKLLNGFNVMQPMGWDAFGMPAENAAMKNNVAPAAWTYDNIEYMKTQLKSLGFAVDWEREVATCKPEYYRWEQWLFTKLFEKGIVYRKNGTVNWDPVDQTVLANEQVIDGRGWRSGALIEKREIPMYYFKITDYAEELLNDLDKLEHWPEQVKTMQRNWIGKSRGMTVRFAVSDDSKQGLEGDYAKFLQVYTTRPDTLMGATYVAVAAEHPLATAAAADKPELQAFIAECKAGADMATMEKKGVPTGRYVVNPLNGDKLEVWIANYVLWGYGDGAVMAVPAHDERDFEFAAKYNLPKKQVIAVGDNAFDANRWQEWYGDKENGVLVNSGDLDGLDFQTAFDAVAAKLQSQGAGEPKTQYRLRDWGISRQRYWGCPIPIVHCEKCGNVPVPADQLPVVLPENVVPDGMGSPLAKMPEFYETSCPCCGGAAKRETDTMDTFIESSWYFFRYMSPKFSDGMVSAESAKYWGAVDQYIGGIEHAILHLLYARFFTKLMRDEGLVNVDEPFERLLTQGMVVCETYYWINPADVELTPVVISGTEKMSKSKNNGVDPQELINAYGADTARLFMMFAAPPEQSLEWSDSGVEGAHRFLRRLWRTVYEYLKQGGAVKAFAGNQDGLSKELKDLRHKLHSTTAKVSDDYGRRQQFNTAIAAVMELLNQYDKTDTGSEQGRAVAQEVLEAAVRLLWPIVPHICETLWSELNGAKLWEAGWPTVDEAALVKSEIGKLRGKITVAADASKADLEAAALANEGAVKFMEGKIIVVPGRLVNIV 6q8c A 2.31 BS01 LSU A 1 M40 F41 P42 Y43 G51 H52 N55 D80 S510 G543 G544 E546 H547 H551 Q580 M40 F41 P42 Y43 G51 H52 N55 D80 S507 G540 G541 E543 H544 H548 Q577 0000166,0002161,0004812,0004823,0005524,0006418,0006429 remove_due_to_license_issue 30995568 901 MQEHYQPAAIEPAAQKKWDDARISNVSEDASKPKYYCLSMFPYPSGKLHMGHVRNYTIGDVLSRFKLLNGFNVMQPMGWDAFGMPAENAAMKNNVAPAAWTYDNIEYMKTQLKSLGFAVDWEREVATCKPEYYRWEQWLFTKLFEKGIVYRKNGTVNWDPVDQTVLANEQVIDGRGWRSGALIEKREIPMYYFKITDYAEELLNDLDKLEHWPEQVKTMQRNWIGKSRGMTVRFAVSDDSKQGLEGDYAKFLQVYTTRPDTLMGATYVAVAAEHPLATAAAADKPELQAFIAECKAGEADMATMEKKGVPTGRYVVNPLNGDKLEVWIANYVLWGYGDGAVMAVPAHDERDFEFAAKYNLPKKQVIAVGDNAFDANRWQEWYGDKENGVLVNSGDLDGLDFQTAFDAVAAKLQSQGAGEPKTQYRLRDWGISRQRYWGCPIPIVHCEKCGNVPVPADQLPVVLPENVVPDGMGSPLAKMPEFYETSCPCCGGAAKRETDTMDTFIESSWYFFRYMSPKFSDGMVSAESAKYWGAVDQYIGGIEHAILHLLYARFFTKLMRDEGLVNVDEPFERLLTQGMVVCETYYDWINPADVELTDGLPVVISGTEKMSKSKNNGVDPQELINAYGADTARLFMMFAAPPEQSLEWSDSGVEGAHRFLRRLWRTVYEYLKQGGAVKAFAGNQDGLSKELKDLRHKLHSTTAKVSDDYGRRQQFNTAIAAVMELLNQYDKTDTGSEQGRAVAQEVLEAAVRLLWPIVPHICETLWSELNGAKLWEAGWPTVDEAALVKSEIVNGKLRGKITVAADASKADLEAAALANEIIVVPGRLVNIV 6q8k A 2.29 BS01 FG9 A 1 L167 F172 V175 A189 K191 F241 L243 L244 K290 N293 L295 V324 D325 L21 F26 V29 A43 K45 F95 L97 L98 K144 N147 L149 V178 D179 D288 K290 N293 D325 T342 D142 K144 N147 D179 T196 2.7.12.1 0004672,0005524,0006468 ic50=290nM remove_due_to_license_issue P49759 30731399 502 MHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVSTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKKSI 6q8p A 3.0 BS01 HQB A 1 L167 V175 K191 F241 E242 L243 L244 L295 V324 L22 V30 K46 F96 E97 L98 L99 L150 V179 D288 K290 N293 D325 T342 D143 K145 N148 D180 T196 2.7.12.1 0004672,0005524,0006468 remove_due_to_license_issue P49759 30731399 501 SMHLICQSGDVLSARYEIVDTLGEGAFGKVVECIDHKAGGRHVAVKIVKNVDRYCEAARSEIQVLEHLNTTDPNSTFRCVQMLEWFEHHGHICIVFELLGLSTYDFIKENGFLPFRLDHIRKMAYQICKSVNFLHSNKLTHTDLKPENILFVQSDYTEAYNPKIKRDERTLINPDIKVVDFGSATYDDEHHSTLVTRHYRAPEVILALGWSQPCDVWSIGCILIEYYLGFTVFPTHDSKEHLAMMERILGPLPKHMIQKTRKRKYFHHDRLDWDEHSSAGRYVSRACKPLKEFMLSQDVEHERLFDLIQKMLEYDPAKRITLREALKHPFFDLLKK 6q92 A 1.5 BS03 ABH A 1 D124 H126 D128 S137 H141 D183 D232 D234 D123 H125 D127 S136 H140 D182 D231 D233 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue P05089 32647818 403 SAKSRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 6q96 A 1.8 BS01 HRE A 1 L54 L57 G58 I61 M62 Y67 Q72 F86 V93 H96 I99 Y100 L30 L33 G34 I37 M38 Y43 Q48 F62 V69 H72 I75 Y76 2.3.2.27 0005634,0043066,0051726 ic50=0.1nM remove_due_to_license_issue IC50=0.166nM Q00987 31066983 201 ETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 6q9h A 2.0 BS01 HRH A 1 L54 I61 M62 H96 I99 Y100 L36 I43 M44 H78 I81 Y82 2.3.2.27 0005634,0043066,0051726 ic50=7.8nM remove_due_to_license_issue Q00987 31066983 201 IPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 6q9l A 1.13 BS01 HTZ A 1 L54 L57 G58 I61 M62 Y67 Q72 V93 H96 I99 Y100 L37 L40 G41 I44 M45 Y50 Q55 V76 H79 I82 Y83 2.3.2.27 0005634,0043066,0051726 ic50=3.9nM remove_due_to_license_issue Q00987 31066983 201 QIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVN 6q9o A 1.21 BS01 HU8 A 1 L54 F55 G58 I61 M62 F91 V93 H96 I99 L38 F39 G42 I45 M46 F75 V77 H80 I83 2.3.2.27 0005634,0043066,0051726 ic50=3.4nM remove_due_to_license_issue Q00987 31066983 201 SQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 6q9o A 1.21 BS02 HU8 B 1 K51 F55 K35 F39 2.3.2.27 0005634,0043066,0051726 ic50=3.4nM remove_due_to_license_issue Q00987 31066983 201 SQIPASEQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVV 6q9q A 2.1 BS01 HUE A 1 M54 L57 G58 I61 M62 Y67 Q72 V93 L99 M29 L32 G33 I36 M37 Y42 Q47 V68 L74 ? 0005634,0043066,0051726 ic50=145nM remove_due_to_license_issue O15151 31066983 201 NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT 6q9s A 2.4 BS01 HRN A 1 M54 H55 L57 G58 I61 M62 Y67 V93 L99 M32 H33 L35 G36 I39 M40 Y45 V71 L77 ? 0005634,0043066,0051726 ic50=17nM remove_due_to_license_issue O15151 31066983 201 GQINQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT 6q9u A 2.4 BS01 HRE A 1 M54 G58 I61 M62 Y67 Q72 V93 P96 L99 Y100 M30 G34 I37 M38 Y43 Q48 V69 P72 L75 Y76 ? 0005634,0043066,0051726 ic50=1300nM remove_due_to_license_issue O15151 31066983 201 INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTL 6q9w A 1.55 BS01 HRT A 1 M54 G58 I61 M62 Y67 Q72 M74 V93 P96 L99 Y100 M29 G33 I36 M37 Y42 Q47 M49 V68 P71 L74 Y75 ? 0005634,0043066,0051726 ic50=580nM remove_due_to_license_issue O15151 31066983 201 NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLA 6q9y A 1.2 BS01 HRQ A 1 G58 I61 Y67 Q72 V75 V93 P96 L99 Y100 G32 I35 Y41 Q46 V49 V67 P70 L73 Y74 ? 0005634,0043066,0051726 ic50=3700nM remove_due_to_license_issue O15151 31066983 201 QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLA 6q9y A 1.2 BS02 HRQ B 1 H73 V93 K94 P96 H47 V67 K68 P70 ? 0005634,0043066,0051726 ic50=3700nM remove_due_to_license_issue O15151 31066983 201 QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDQQEQHMVYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVTLA 6qaa A 1.897 BS02 HUN A 1 D70 W82 G117 P285 L286 F329 W430 D67 W79 G114 P282 L283 F326 W427 G116 G117 S198 A199 E325 H438 G113 G114 S195 A196 E322 H435 3.1.1.8 0004104 ic50=22nM remove_due_to_license_issue P06276 30864579 613 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6qab A 2.49 BS02 HUQ A 1 W82 G117 Q119 P285 L286 V288 F329 Y332 H438 W79 G114 Q116 P282 L283 V285 F326 Y329 H435 G116 G117 S198 A199 E325 H438 G113 G114 S195 A196 E322 H435 3.1.1.8 0004104 ic50=6.2nM remove_due_to_license_issue P06276 30864579 618 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6qac A 2.771 BS01 HUT A 1 W82 G117 W231 P285 L286 S287 V288 Y332 W79 G114 W228 P282 L283 S284 V285 Y329 G116 G117 S198 A199 E325 H438 G113 G114 S195 A196 E322 H435 3.1.1.8 0004104 remove_due_to_license_issue P06276 30864579 611 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6qad A 2.497 BS01 HUZ A 1 G116 G117 P285 S287 N289 F329 Y332 G113 G114 P282 S284 N286 F326 Y329 G116 G117 S198 A199 E325 H438 G113 G114 S195 A196 E322 H435 3.1.1.8 0004104 ic50=14nM remove_due_to_license_issue P06276 30864579 618 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6qae A 2.487 BS02 HUK A 1 N68 W82 G117 T120 L286 S287 A328 F329 Y332 H438 N65 W79 G114 T117 L283 S284 A325 F326 Y329 H435 G116 G117 S198 A199 E325 H438 G113 G114 S195 A196 E322 H435 3.1.1.8 0004104 ic50=3nM remove_due_to_license_issue P06276 30864579 612 IIIATKNGKVRGMQLTVFGGTVTAFLGIPYAQPPLGRLRFKKPQSLTKWSDIWNATKYANSCCQNIDQSFPGFHGSEMWNPNTDLSEDCLYLNVWIPAPKPKNATVLIWIYGGGFQTGTSSLHVYDGKFLARVERVIVVSMNYRVGALGFLALPGNPEAPGNMGLFDQQLALQWVQKNIAAFGGNPKSVTLFGESAGAASVSLHLLSPGSHSLFTRAILQSGSFNAPWAVTSLYEARNRTLNLAKLTGCSRENETEIIKCLRNKDPQEILLNEAFVVPYGTPLSVNFGPTVDGDFLTDMPDILLELGQFKKTQILVGVNKDEGTAFLVYGAPGFSKDNNSIITRKEFQEGLKIFFPGVSEFGKESILFHYTDWVDDQRPENYREALGDVVGDYNFICPALEFTKKFSEWGNNAFFYYFEHRSSKLPWPEWMGVMHGYEIEFVFGLPLERRDQYTKAEEILSRSIVKRWANFAKYGNPQETQNQSTSWPVFKSTEQKYLTLNTESTRIMTKLRAQQCRFWTSFFPKV 6qaf A 1.61 BS03 XC3 A 1 D124 H126 D128 N130 S137 H141 D183 D232 D123 H125 D127 N129 S136 H140 D182 D231 3.5.3.1 0000050,0002250,0004053,0005515,0005576,0005615,0005634,0005737,0005829,0006525,0006527,0009624,0016787,0016813,0019547,0030145,0035578,0035580,0042130,0042832,0045087,0046007,0046872,0060336,0070965,2000552 remove_due_to_license_issue P05089 32647818 403 SAKSRTIGIIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKEQECDVKDYGDLPFADIPNDSPFQIVKNPRSVGKASEQLAGKVAEVKKNGRISLVLGGDHSLAIGSISGHARVHPDLGVIWVDAHTDINTPLTTTSGNLHGQPVSFLLKELKGKIPDVPGFSWVTPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDRLGIGKVMEETLSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVVGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTAVAITLACFGLAREGNHKPIDYLN 6qat A 2.77 BS01 FE7 A 1 V15 A37 K39 E86 Y87 C88 G90 L138 V15 A37 K39 E86 Y87 C88 G90 L138 D131 K133 Q135 N136 D158 D131 K133 Q135 N136 D153 2.7.11.1 0004672,0004674,0005524,0006468,0010506 remove_due_to_license_issue Q8IYT8 30782972 301 MEVVGDFEYSKRDLVGHGAFAVVFRGRHRQKTDWEVAIKSINKKNLSKSQILLGKEIKILKELQHENIVALYDVQELPNSVFLVMEYCNGGDLADYLQAKGTLSEDTIRVFLHQIAAAMRILHSKGIIHRDLKPQNILLSYANVSGIRIKIADFGFARYLHSPMYMAPEVIMSQHYDAKADLWSIGTVIYQCLVGKPPFQANSPQDLRMFYEKNRSLMPSIPRETSPYLANLLLGLLQRNQKDRMDFEAFFSHPFLEQG 6qav A 2.05 BS01 HVH A 1 V15 H17 V23 A37 M85 E86 Y87 C88 G91 D95 L138 D158 V16 H18 V24 A38 M86 E87 Y88 C89 G92 D96 L139 D159 D131 K133 Q135 N136 D158 S177 D132 K134 Q136 N137 D159 S178 2.7.11.1 0004672,0004674,0005524,0006468,0010506 remove_due_to_license_issue IC50=1.1nM Q8IYT8 30782972 301 SMEVVGDFEYSKRDLVGHGAFAVVFRGRHRQKTDWEVAIKSINKKNLSKSQILLGKEIKILKELQHENIVALYDVQELPNSVFLVMEYCNGGDLADYLQAKGTLSEDTIRVFLHQIAAAMRILHSKGIIHRDLKPQNILLSYANRRKSSVSGIRIKIADFGFARYLHSNMMAADLCGSPMYMAPEVIMSQHYDAKADLWSIGTVIYQCLVGKPPFQANSPQDLRMFYEKNRSLMPSIPRETSPYLANLLLGLLQRNQKDRMDFEAFFSHPFLE 6qcj A 2.01 BS03 XEG A 1 I61 P62 F64 W71 F86 M136 V154 G155 T156 M157 I52 P53 F55 W62 F77 M127 V145 G146 T147 M148 P62 D63 F64 R65 N114 D116 H133 P53 D54 F55 R56 N105 D107 H124 2.3.1.-,2.3.1.286,2.4.2.- 0070403 remove_due_to_license_issue Q8N6T7 31844103 407 PFTADKGKCGLPEIFDPPEELERKVWELARLVWQSSSVVFHTGAGISTASGIPDFRGPHGVWTMEERGLAPKFDTTFESARPTQTHMALVQLERVGLLRFLVSQNVDGLHVRSGFPRDKLAELHGNMFVEECAKCKTQYVRDTVVGTMGLKATGRLCTVACRGELRDTILDWEDSLPDRDLALADEASRNADLSITLGTSLQIRPSGNLPLATKRRGGRLVIVNLQPTKHDRHADLRIHGYVDEVMTRLMKHLGLEIPAWDGPRVLERALPPLPRPPTPKLE 6qdx A 2.1 BS01 HY8 A 1 H9 D15 K18 H42 A43 G44 S100 D164 P166 E168 M235 H7 D13 K16 H40 A41 G42 S93 D157 P159 E161 M228 2.1.1.266 0003676,0003723,0005515,0005829,0006364,0008168,0008649,0008988,0015976,0032259,0036307,0070475 Kd=30uM remove_due_to_license_issue P37634 30879411 301 SYRHSFHAGNHADVLKHTVQSLIIESLKEKDKPFLYLDTHAGAGRYQLGRTGKYLEGIARIWQQDDLPAELEAYINVVKHFNRSGQLRYYPGSPLIARQLLREQDSLQLTELHPSDYPLLRSEFQKDSRARVEKADGFQQLKAKLPPVSRRGLILIDPPYEMKTDYQAVVSGIAEGYKRFATGTYALWYPVVLRQQIKRMIHDLEATGIRKILQIELAVLPDSDRRGMTASGMIVINPPWKLEQQMNNVLPWLHSKLVPAGTGHATVSWIVPE 6qe0 A 1.394 BS01 HZ2 A 1 H9 D15 K18 H19 H42 A43 S100 D164 P166 P197 M235 H12 D18 K21 H22 H45 A46 S98 D162 P164 P195 M233 2.1.1.266 0003676,0003723,0005515,0005829,0006364,0008168,0008649,0008988,0015976,0032259,0036307,0070475 Kd=25uM remove_due_to_license_issue P37634 30879411 301 GSHMLSYRHSFHAGNHADVLKHTVQSLIIESLKEKDKPFLYLDTHAGAGRYQLGRTGKYLEGIARIWQQDDLPAELEAYINVVKHFNRSGQLRYYPGSPLIARQLLREQDSLQLTELHPSDYPLLRSEFQKDSRARVEKADGFQQLKAKLPPVSRRGLILIDPPYEMKTDYQAVVSGIAEGYKRFATGTYALWYPVVLRQQIKRMIHDLEATGIRKILQIELAVLPDSDRRGMTASGMIVINPPWKLEQQMNNVLPWLHSKLVPAGTGHATVSWIVPE 6qe5 A 1.61 BS01 SAH A 1 Y4 H6 K18 H19 H42 A43 G99 S100 E118 L119 D143 G144 D164 P166 Y4 H6 K18 H19 H42 A43 G92 S93 E111 L112 D136 G137 D157 P159 2.1.1.266 0003676,0003723,0005515,0005829,0006364,0008168,0008649,0008988,0015976,0032259,0036307,0070475 Kd=7.5uM remove_due_to_license_issue P37634 30879411 301 MLSYRHSFHAGNHADVLKHTVQSLIIESLKEKDKPFLYLDTHAGAGRYQLGGKYLEGIARIWQQDDLPAELEAYINVVKHFNRSGQLRYYPGSPLIARQLLREQDSLQLTELHPSDYPLLRSEFQKDSRARVEKADGFQQLKAKLPPVSRRGLILIDPPYEMKTDYQAVVSGIAEGYKRFATGTYALWYPVVLRQQIKRMIHDLEATGIRKILQIELAVLPDSGMTASGMIVINPPWKLEQQMNNVLPWLHSKLVPAGTGHATVSWIVPE 6qed A 1.8 BS01 HZK A 1 F219 A230 H231 D251 L328 N329 H331 I338 H339 E364 H382 A414 Y444 E459 F109 A120 H121 D141 L218 N219 H221 I228 H229 E254 H272 A304 Y334 E349 D251 D262 H331 H339 E364 E459 D141 D152 H221 H229 E254 E349 3.4.11.18 0006508,0070006 ic50=0.015uM remove_due_to_license_issue IC50=15nM, Ki=0.160000nM P50579 30939017 506 VQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRG 6qef A 1.79 BS01 HZW A 1 F219 H231 D251 D262 L328 N329 H331 I338 H339 E364 H382 A414 Y444 E459 F109 H121 D141 D152 L218 N219 H221 I228 H229 E254 H272 A304 Y334 E349 D251 D262 H331 H339 E364 E459 D141 D152 H221 H229 E254 E349 3.4.11.18 0006508,0070006 ic50=0.06uM remove_due_to_license_issue IC50=60nM P50579 30939017 507 VQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRG 6qeg A 2.08 BS01 K4K A 1 F219 A230 H231 D251 D262 L328 N329 H331 I338 H339 E364 Y444 E459 F109 A120 H121 D141 D152 L218 N219 H221 I228 H229 E254 Y334 E349 D251 D262 H331 H339 E364 E459 D141 D152 H221 H229 E254 E349 3.4.11.18 0006508,0070006 ic50=0.05uM remove_due_to_license_issue IC50=50nM P50579 30939017 502 VQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSR 6qfd A 2.133 BS01 dna E 0 N49 G51 R52 N56 K73 R74 N43 G45 R46 N50 K67 R68 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd A 2.133 BS02 dna F 0 Y32 G33 L34 H50 Y54 K68 R74 T75 N76 Y26 G27 L28 H44 Y48 K62 R68 T69 N70 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd B 2.133 BS01 dna E 0 Y32 G33 L34 H50 G51 Y54 K68 R74 T75 N76 Y27 G28 L29 H45 G46 Y49 K63 R69 T70 N71 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd B 2.133 BS02 dna F 0 H50 G51 R52 N56 D72 K73 R74 H45 G46 R47 N51 D67 K68 R69 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd C 2.133 BS01 dna G 0 Y32 G33 L34 H50 Y54 R74 T75 N76 Y23 G24 L25 H41 Y45 R65 T66 N67 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 SDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd C 2.133 BS02 dna H 0 H50 G51 R52 N56 D72 K73 R74 H41 G42 R43 N47 D63 K64 R65 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 SDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd D 2.133 BS01 dna G 0 N49 H50 G51 R52 N56 K73 R74 N43 H44 G45 R46 N50 K67 R68 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfd D 2.133 BS02 dna H 0 Y32 G33 L34 H50 G51 Y54 R74 T75 N76 Y26 G27 L28 H44 G45 Y48 R68 T69 N70 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qfe A 1.67 BS01 J08 A 1 H57 H96 D189 S190 C191 Q192 S195 V213 S214 W215 G216 D217 Y218 C220 H42 H81 D173 S174 C175 Q176 S179 V193 S194 W195 G196 D197 Y198 C200 H57 D102 Q192 G193 D194 S195 G196 H42 D87 Q176 G177 D178 S179 G180 3.4.21.- 0004252,0006508 ic50=0.08uM remove_due_to_license_issue Q9Y337 31045568 305 IINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS 6qff A 1.64 BS01 J08 A 1 H57 H99 D189 S190 C191 Q192 S195 V213 S214 W215 G216 N217 I218 C220 H41 H82 D170 S171 C172 Q173 S176 V190 S191 W192 G193 N194 I195 C197 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 ic50=2.04uM remove_due_to_license_issue Q92876 31045568 301 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNIPCGSKEKPGVYTNVCRYTNWIQKTIQA 6qfg A 1.68 BS01 J08 A 1 H57 H99 D189 S190 C191 S195 V213 S214 W215 G216 N217 Y218 C220 H41 H82 D170 S171 C172 S176 V190 S191 W192 G193 N194 Y195 C197 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 ic50=3.01uM remove_due_to_license_issue Q92876 31045568 302 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNYPCGSKEKPGVYTNVCRYTNWIQKTIQAK 6qfg A 1.68 BS02 J08 B 1 G38 H39 G22 H23 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 ic50=3.01uM remove_due_to_license_issue Q92876 31045568 302 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNYPCGSKEKPGVYTNVCRYTNWIQKTIQAK 6qfh A 1.65 BS01 J08 A 1 H57 H99 D189 S190 C191 Q192 S195 V213 S214 W215 G216 D217 Y218 C220 H41 H82 D170 S171 C172 Q173 S176 V190 S191 W192 G193 D194 Y195 C197 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 ic50=1.38uM remove_due_to_license_issue Q92876 31045568 301 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGDYPCGSKERPGVYTNVCRYTNWIQKTIQA 6qfh A 1.65 BS02 J08 B 1 G38 H39 G22 H23 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 ic50=1.38uM remove_due_to_license_issue Q92876 31045568 303 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGDYPCGSKERPGVYTNVCRYTNWIQKTIQA 6qfq A 1.6 BS01 J3E A 1 A227 F228 M250 V253 R263 L267 F270 G271 I294 A56 F57 M79 V82 R92 L96 F99 G100 I123 ? 0003824,0042981 remove_due_to_license_issue IC50=100nM Q07820 31459977 401 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6qfq A 1.6 BS02 J3E A 2 H224 N260 G262 F318 F319 H53 N89 G91 F147 F148 ? 0003824,0042981 remove_due_to_license_issue IC50=100nM Q07820 31459977 402 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6qft A 2.7 BS01 J0B A 1 M212 E213 M215 C218 M94 E95 M97 C100 D259 K261 N264 D277 C296 D141 K143 N146 D159 C166 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue O14733 31083997 501 QTGYLTIGQRYQAEINDLENLGEMGSGTCGQVWKMRFRKTGHVIAVKQMRRSGNKEENKRILMDLDVVLKSHDCPYIVQCFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGKMTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCDFGISGRCAAYMAPERIDPRADVWSLGISLVELATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQSFVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFKDVMAK 6qfu A 1.8 BS01 J0K A 1 Q92 H94 H119 F130 L197 T198 T199 Q89 H91 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=35nM remove_due_to_license_issue P00918 31080690 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6qfv A 1.45 BS01 J0N A 1 I91 Q92 H94 H119 F130 L197 T198 T199 I87 Q88 H90 H115 F126 L193 T194 T195 H64 H94 H96 E106 H119 T198 H60 H90 H92 E102 H115 T194 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=49nM remove_due_to_license_issue P00918 31080690 301 WGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6qfw A 1.2 BS01 JR8 A 1 H94 H96 H119 F130 L197 T198 T199 P201 H91 H93 H116 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=149nM remove_due_to_license_issue P00918 31080690 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6qfx A 1.32 BS01 JR3 A 1 H94 H96 H119 F130 L197 T198 T199 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T198 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=20nM remove_due_to_license_issue P00918 31080690 301 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6qg4 A 2.3 BS01 J0E A 1 M142 A163 K165 D182 M212 M215 C218 K221 C276 M24 A40 K42 D59 M89 M92 C95 K98 C153 D259 K261 N264 D277 D136 K138 N141 D154 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue O14733 31083997 501 QTGYLTIGQRYQAEINDLENLGEMGQVWKMRFRKTGHVIAVKQMRRSGNKEENKRILMDLDVVLKSHDCPYIVQCFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGKMTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCDFGISGRAAYMAPERIDPIRADVWSLGISLVELATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQSFVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFKDVMAKT 6qge A 1.16 BS01 J1E A 1 R144 I145 A146 H158 R162 W181 E184 R186 S237 R32 I33 A34 H46 R50 W69 E72 R74 S125 ? 0030246 Kd=0.000000064M remove_due_to_license_issue P17931 30618244 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qgf A 1.34 BS01 J0T A 1 R144 I145 A146 H158 R162 W181 E184 R186 S237 R32 I33 A34 H46 R50 W69 E72 R74 S125 ? 0030246 Kd=0.000000064M remove_due_to_license_issue P17931 30618244 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qgg A 1.5 BS01 J1H A 1 A100 D103 F104 R107 Y108 D111 M115 L137 W144 G145 V148 Y202 A37 D40 F41 R44 Y45 D48 M52 L74 W81 G82 V85 Y139 ? 0042981 remove_due_to_license_issue P10415,Q07817 31459977 401 SQDNREIVMKYISYKLSQRGYEWDTESEVVHQTLRQAGDDFSLRYRRDFAEMSSQLHLTPGTAYASFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSVLVDNIAAWMATYLNDHLHTWIQDNGGWDAFVELYG 6qgj A 1.9 BS01 J1T A 1 F104 Y108 N143 W144 G145 F153 F198 L201 Y202 N204 E209 F36 Y40 N75 W76 G77 F85 F130 L133 Y134 N136 E141 ? 0042981 remove_due_to_license_issue P10415,Q07817 31459977 301 NREIVMKYISYKLSQRGYEWESEVVHQTLRQAGDDFSLRYRRDFAEMSSQLHLTPGTAYASFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSVLVDNIAAWMATYLNDHLHTWIQDNGGWDAFVELYGNNAAAESRKGQ 6qgk A 1.8 BS01 J1Q A 1 F104 Y108 D111 M115 L137 F41 Y45 D48 M52 L74 ? 0042981 remove_due_to_license_issue P10415,Q07817 31459977 401 DNREIVMKYISYKLSQRGYEWDAGDESEVVHQTLRQAGDDFSLRYRRDFAQMSSQLHLTPGTAYASFATVVAELFRDGVNWGRIVAFFEFGGVMCVESVNRAMSVLVDNIAAWMATYLNDHLHTWIQDNGGWDAFVELYGNNAAAESR 6qh0 A 2.436 BS01 dna G 0 N49 G51 R52 N56 K73 R74 N43 G45 R46 N50 K67 R68 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 A 2.436 BS02 dna H 0 Y32 G33 L34 H50 Y54 K68 R74 T75 N76 Y26 G27 L28 H44 Y48 K62 R68 T69 N70 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 B 2.436 BS01 dna G 0 G33 L34 H50 Y54 R74 T75 N76 G28 L29 H45 Y49 R69 T70 N71 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 B 2.436 BS02 dna H 0 N49 H50 G51 R52 N56 D72 R74 N44 H45 G46 R47 N51 D67 R69 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 C 2.436 BS01 dna E 0 Y32 G33 L34 H50 Y54 R74 T75 N76 Y21 G22 L23 H39 Y43 R63 T64 N65 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 ARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 C 2.436 BS02 dna F 0 N49 G51 R52 N56 D72 K73 R74 N38 G40 R41 N45 D61 K62 R63 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 ARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 D 2.436 BS01 dna E 0 N49 H50 G51 R52 N56 K73 R74 N42 H43 G44 R45 N49 K66 R67 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 ARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh0 D 2.436 BS02 dna F 0 Y32 G33 L34 H50 G51 Y54 R74 T75 N76 Y25 G26 L27 H43 G44 Y47 R67 T68 N69 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 ARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qh9 A 2.27 BS01 J2N A 1 D189 S190 Q192 G193 S195 V213 G216 N217 D170 S171 Q173 G174 S176 V190 G193 N194 H57 D102 Q192 G193 D194 S195 G196 H41 D85 Q173 G174 D175 S176 G177 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 remove_due_to_license_issue Q92876 30691925 302 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNIPCGSKEKPGVYTNVCRYTNWIQKTIQA 6qha A 1.82 BS01 J2Q A 1 H57 D189 S190 C191 Q192 S195 W215 G216 N217 H41 D170 S171 C172 Q173 S176 W192 G193 N194 H57 D102 Q192 G193 D194 S195 G196 H41 D85 Q173 G174 D175 S176 G177 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 remove_due_to_license_issue Q92876 30691925 303 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNIPCGSKEKPGVYTNVCRYTNWIQKTIQA 6qhb A 1.84 BS01 J2W A 1 H57 D189 S190 C191 Q192 S195 W215 G216 N217 C220 H41 D170 S171 C172 Q173 S176 W192 G193 N194 C197 H57 D102 Q192 G193 D194 S195 G196 H41 D85 Q173 G174 D175 S176 G177 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 remove_due_to_license_issue Q92876 30691925 301 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNIPCGSKEKPGVYTNVCRYTNWIQKTIQAK 6qhd A 2.85 BS01 dna C 0 M331 H332 K340 V343 Q344 N466 M187 H188 K196 V199 Q200 N313 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P40763 31170499 1001 ~ 1018 VVTEKQQMLEQHLQDVRKRVQDLEQKMKVVENLQDDFDFNYKTLKSQGDSVTRQKMQQLEQMLTALDQMRRSIVSELAGLLSAMEYVQKTLTDEELADWKRRQQIACIGGPPNICLDRLENWITSLAESQLQTRQQIKKLEELQQKVSYKGDPIVQHRPMLEERIVELFRNLMKSAFVVERQPCMPMHPDRPLVIKTGVQFTTKVRLLVKFPELNYQLKIKVCIDKDSGDVAALRGSRKFNILGTNTKVMNMEESNNGSLSAEFKHLTLREQRCASLIVTEELHLITFETEVYHQGLKIDLETHSLPVVVISNICQMPNAWASILWYNMLTNNPKNVNFFTKPPIGTWDQVAEVLSWQFSSTTKRGLSIEQLTTLAEKLLGPYSGCQITWAKFCKENMAGKGFSFWVWLDNIIDLVKKYILALWNEGYIMGFISKERERAILSTKPPGTFLLRFSESSKEGGVTFTWVEQIQSVEPYTKQQLNNMSFAEIIMGYLVSPLVYLYPDIPKEEAFGKYCRAPYLKTKFICVTP 6qhd A 2.85 BS02 dna D 0 R382 I431 V432 S465 N466 Q469 R238 I278 V279 S312 N313 Q316 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P40763 31170499 1001 ~ 1018 VVTEKQQMLEQHLQDVRKRVQDLEQKMKVVENLQDDFDFNYKTLKSQGDSVTRQKMQQLEQMLTALDQMRRSIVSELAGLLSAMEYVQKTLTDEELADWKRRQQIACIGGPPNICLDRLENWITSLAESQLQTRQQIKKLEELQQKVSYKGDPIVQHRPMLEERIVELFRNLMKSAFVVERQPCMPMHPDRPLVIKTGVQFTTKVRLLVKFPELNYQLKIKVCIDKDSGDVAALRGSRKFNILGTNTKVMNMEESNNGSLSAEFKHLTLREQRCASLIVTEELHLITFETEVYHQGLKIDLETHSLPVVVISNICQMPNAWASILWYNMLTNNPKNVNFFTKPPIGTWDQVAEVLSWQFSSTTKRGLSIEQLTTLAEKLLGPYSGCQITWAKFCKENMAGKGFSFWVWLDNIIDLVKKYILALWNEGYIMGFISKERERAILSTKPPGTFLLRFSESSKEGGVTFTWVEQIQSVEPYTKQQLNNMSFAEIIMGYLVSPLVYLYPDIPKEEAFGKYCRAPYLKTKFICVTP 6qhd B 2.85 BS01 dna C 0 R382 I431 V432 S465 N466 R237 I276 V277 S310 N311 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P40763 31170499 1001 ~ 1018 VVTEKQQMLEQHLQDVRKRVQDLEQKMKVVENLQDDFDFNYKTLKSQGSVTRQKMQQLEQMLTALDQMRRSIVSELAGLLSAMEYVQKTLTDEELADWKRRQQIACIGGPPNICLDRLENWITSLAESQLQTRQQIKKLEELQQKVSYKGDPIVQHRPMLEERIVELFRNLMKSAFVVERQPCMPMHPDRPLVIKTGVQFTTKVRLLVKFPELNYQLKIKVCIDKDSGDVAALRGSRKFNILGTNTKVMNMEESNNGSLSAEFKHLTLREQRASLIVTEELHLITFETEVYHQGLKIDLETHSLPVVVISNICQMPNAWASILWYNMLTNNPKNVNFFTKPPIGTWDQVAEVLSWQFSSTTKRGLSIEQLTTLAEKLLGPYSGCQITWAKFCKENMAGKGFSFWVWLDNIIDLVKKYILALWNEGYIMGFISKERERAILSTKPPGTFLLRFSESSKEGGVTFTWVETQIQSVEPYTKQQLNNMSFAEIIMGYKIILVSPLVYLYPDIPKEEAFGKYCRAPYLKTKFICVTP 6qhd B 2.85 BS02 dna D 0 M331 H332 K340 V343 Q344 N466 I467 M186 H187 K195 V198 Q199 N311 I312 ? 0003677,0003700,0006355,0007165 remove_due_to_license_issue P40763 31170499 1001 ~ 1018 VVTEKQQMLEQHLQDVRKRVQDLEQKMKVVENLQDDFDFNYKTLKSQGSVTRQKMQQLEQMLTALDQMRRSIVSELAGLLSAMEYVQKTLTDEELADWKRRQQIACIGGPPNICLDRLENWITSLAESQLQTRQQIKKLEELQQKVSYKGDPIVQHRPMLEERIVELFRNLMKSAFVVERQPCMPMHPDRPLVIKTGVQFTTKVRLLVKFPELNYQLKIKVCIDKDSGDVAALRGSRKFNILGTNTKVMNMEESNNGSLSAEFKHLTLREQRASLIVTEELHLITFETEVYHQGLKIDLETHSLPVVVISNICQMPNAWASILWYNMLTNNPKNVNFFTKPPIGTWDQVAEVLSWQFSSTTKRGLSIEQLTTLAEKLLGPYSGCQITWAKFCKENMAGKGFSFWVWLDNIIDLVKKYILALWNEGYIMGFISKERERAILSTKPPGTFLLRFSESSKEGGVTFTWVETQIQSVEPYTKQQLNNMSFAEIIMGYKIILVSPLVYLYPDIPKEEAFGKYCRAPYLKTKFICVTP 6qhg A 1.483 BS01 MGT A 1 F1713 R1716 Q1717 Y1728 M1782 F10 R13 Q14 Y25 M79 2.7.7.48,3.1.-.- Kd=737uM remove_due_to_license_issue A2SZS3 31136637 2001 GPGAGTVGGFIKRQQSKVVQNKVVYYGVGIWRGFMDGYQVHLEIENDIGQPPRLRNVTTNCQSSPWDLSIPIRQWAEDMGVTNNQDYSSKSSRGARYWMHSFRMQGPSKPFGCPVYIIK 6qho A 2.7 BS01 J3H A 1 M215 C218 K221 S263 L266 M98 C101 K104 S146 L149 D259 K261 N264 D277 D142 K144 N147 D160 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue O14733 31083997 501 QTGYLTIGGQRYQAEINDLENLGEMGSGTCGQVWKMRFRKTGHVIAVKQMRRSGNKEENKRILMDLDVVLKSHDCPYIVQCFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGKMTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCDFGISGRYMAPERIDPRADVWSLGISLVELATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQSFVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFKDVMAKT 6qhr A 2.52 BS01 J3N A 1 S144 K165 M212 E213 M215 C218 K221 S28 K49 M96 E97 M99 C102 K105 D259 K261 N264 D277 C296 D143 K145 N148 D161 C171 2.7.12.2 0004672,0005524,0006468 remove_due_to_license_issue O14733 31083997 501 KQTGYLTIGGQRYQAEINDLENLGEMGSGTCGQVWKMRFRKTGHVIAVKQMRRSGNKEENKRILMDLDVVLKSHDCPYIVQCFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGKMTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCDFGISGRLAGCAAYMAPERIDPPYDIRADVWSLGISLVELATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQSFVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFKDVMAKT 6qi4 B 1.78 BS04 FKW B 1 W30 Y52 V68 F72 F85 W103 W28 Y50 V66 F70 F83 W101 ? 0005245,0005509,0005515,0005737,0005794,0005886,0008048,0009966,0010975,0014069,0030424,0030425,0043231,0045202,0046872,0048471,0070588 Kd=43uM remove_due_to_license_issue P62166 31243268 212 KSNSKLKPEVVEELTRKTYFTEKEVQQWYKGFIKDCPSGQLDAAGFQKIYKQFFPFGDPTKFATFVFNVFDENKDGRIEFSEFIQALSVTSRGTLDEKLRWAFKLYDLDNDGYITRNEMLDIVDAIYQMVGNTVELPEEENTPEKRVDRIFAMMDKNADGKLTLQEFQEGSKADPSIVQALSLYDGL 6qil A 2.0 BS01 dna E 0 Y32 G33 L34 H50 G51 Y54 K68 R74 T75 N76 Y26 G27 L28 H44 G45 Y48 K62 R68 T69 N70 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil A 2.0 BS02 dna F 0 N49 H50 G51 R52 N56 K73 R74 N43 H44 G45 R46 N50 K67 R68 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil B 2.0 BS01 dna E 0 H50 G51 R52 N56 D72 K73 R74 H45 G46 R47 N51 D67 K68 R69 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil B 2.0 BS02 dna F 0 Y32 G33 L34 H50 G51 Y54 K68 R74 T75 N76 Y27 G28 L29 H45 G46 Y49 K63 R69 T70 N71 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil C 2.0 BS01 dna G 0 H50 G51 R52 D72 K73 R74 H41 G42 R43 D63 K64 R65 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 SDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil C 2.0 BS02 dna H 0 Y32 G33 L34 H50 G51 Y54 P55 R74 T75 N76 Y23 G24 L25 H41 G42 Y45 P46 R65 T66 N67 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 SDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil D 2.0 BS01 dna G 0 Y32 G33 H50 Y54 K68 R74 T75 N76 Y25 G26 H43 Y47 K61 R67 T68 N69 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 ARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qil D 2.0 BS02 dna H 0 N49 H50 G51 R52 D72 K73 R74 N42 H43 G44 R45 D65 K66 R67 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 ARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6ql1 A 1.42 BS02 V50 A 1 Q92 H94 H96 H119 Q135 L198 T199 T200 Q89 H91 H93 H116 Q131 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=15nM remove_due_to_license_issue Kd=10.0nM P00918 31481705 305 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHTFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDYGKAQQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLTECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ql1 A 1.42 BS03 V50 A 2 H4 W5 H10 N11 H15 D19 H1 W2 H7 N8 H12 D16 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=15nM remove_due_to_license_issue Kd=10.0nM P00918 31481705 306 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHTFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDYGKAQQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLTECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ql2 A 1.3 BS02 EZL A 1 H94 H96 H119 Y131 Q135 L198 T199 T200 P201 H91 H93 H116 Y127 Q131 L194 T195 T196 P197 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=1.1nM remove_due_to_license_issue Ki=8nM, IC50=3nM, Kd=0.71nM P00918 31481705 306 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHTFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDYGKAQQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLTECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ql3 A 1.35 BS02 V14 A 1 N62 Q67 Q92 H94 H96 H119 V121 Q135 L198 T199 T200 N59 Q64 Q89 H91 H93 H116 V118 Q131 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Kd=4.5nM remove_due_to_license_issue Kd=60nM P00918 31481705 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHTFQVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDYGKAQQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLTECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6qln A 1.0 BS01 J5Q A 1 R144 I145 A146 H158 R162 W181 E184 R32 I33 A34 H46 R50 W69 E72 ? 0030246 Kd=88uM remove_due_to_license_issue Kd=22000nM P17931 31246331 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qlo A 1.18 BS01 J5E A 1 R144 I145 A146 H158 R162 W181 E184 S237 G238 R32 I33 A34 H46 R50 W69 E72 S125 G126 ? 0030246 Kd=92uM remove_due_to_license_issue Kd=8800nM P17931 31246331 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qlp A 1.081 BS01 J3Q A 1 R144 I145 A146 H158 R162 N174 W181 E184 S237 G238 R32 I33 A34 H46 R50 N62 W69 E72 S125 G126 ? 0030246 Kd=22uM remove_due_to_license_issue Kd=5200nM P17931 31246331 302 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qlq B 1.079 BS01 J4E B 1 R144 A146 H158 N160 R162 N174 W181 E184 S237 G238 R32 A34 H46 N48 R50 N62 W69 E72 S125 G126 ? 0030246 Kd=31uM remove_due_to_license_issue Kd=31000nM P17931 31246331 302 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qlr A 0.97 BS01 J4N A 1 R144 I145 A146 H158 R162 W181 E184 S237 R32 I33 A34 H46 R50 W69 E72 S125 ? 0030246 Kd=8.8uM remove_due_to_license_issue Kd=15000nM P17931 31246331 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qls A 1.047 BS01 HRK A 1 R144 A146 H158 N160 R162 W181 E184 S237 R32 A34 H46 N48 R50 W69 E72 S125 ? 0030246 Kd=15uM remove_due_to_license_issue P17931 31246331 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qlt A 1.15 BS01 J5W A 1 R144 A146 H158 N160 R162 N174 W181 E184 S237 R32 A34 H46 N48 R50 N62 W69 E72 S125 ? 0030246 Kd=23uM remove_due_to_license_issue Kd=92000nM P17931 31246331 302 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qlu A 1.1 BS01 J62 A 1 R144 I145 A146 H158 N160 R162 W181 E184 S237 G238 R32 I33 A34 H46 N48 R50 W69 E72 S125 G126 ? 0030246 Kd=5.2uM remove_due_to_license_issue Kd=23000nM P17931 31246331 301 PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI 6qm7 L 2.8 BS01 J6E L 1 T100 S120 G122 G146 S195 M196 G197 Y212 S226 V227 G228 S229 T1 S21 G23 G47 S96 M97 G98 Y113 S127 V128 G129 S130 T100 D116 R118 K132 G146 S229 D266 S269 T1 D17 R19 K33 G47 S130 D167 S170 3.4.25.1 0000502,0004298,0005634,0005737,0005839,0006508,0051603 remove_due_to_license_issue A4IDD6 30962368 4000 TTTLAFRFNGGIIVAVDSRASTGQYIASQTVMKVLEINDYLLGTLAGGAADCQYWERVLGMECRLWELRNGSRITVAAASKILANITYAYRNHGLSMGTMVAGWDQFGPSLYYVDDKGSRVKQDLFSVGSGSIYAYGVLDTGYRKDLSVEDACDLARRSIFHATYRDGASGGIVTVYHVHEKGWTKISRDDQTKLYHRYFPS 6qmd A 1.94 BS01 J6N A 1 R415 G462 R483 S508 G509 Y525 S555 A556 R91 G138 R159 S184 G185 Y201 S231 A232 ? ic50=170uM remove_due_to_license_issue Q9Z2X8 30973731 702 GRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 6qmd A 1.94 BS02 J6N A 2 Y334 Y572 F577 Y10 Y248 F253 ? ic50=170uM remove_due_to_license_issue Q9Z2X8 30973731 703 GRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 6qme A 1.81 BS01 J6Q A 1 R415 R483 S508 G509 Y525 S555 A556 R92 R160 S185 G186 Y202 S232 A233 ? ic50=44uM remove_due_to_license_issue Q9Z2X8 30973731 702 VGRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 6qmj A 1.86 BS01 J6K A 1 Y334 R415 G462 F478 R483 S508 G509 Y525 S555 A556 S602 G603 Y10 R91 G138 F154 R159 S184 G185 Y201 S231 A232 S278 G279 ? ic50=0.069uM remove_due_to_license_issue Q9Z2X8 30973731 703 GRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 6qmk A 1.72 BS01 J8H A 1 Y334 S363 R415 G462 F478 R483 S508 G509 Y525 S555 A556 S602 G603 Y11 S40 R92 G139 F155 R160 S185 G186 Y202 S232 A233 S279 G280 ? ic50=0.047uM remove_due_to_license_issue Q9Z2X8 30973731 702 VGRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC 6qmr A 2.0 BS01 J6T A 1 C42 H57 D189 S190 C191 K192 G193 S195 V213 T214 S215 R218 C220 G226 C26 H41 D177 S178 C179 K180 G181 S183 V197 T198 S199 R202 C204 G211 H57 D102 K192 G193 D194 S195 H41 D89 K180 G181 D182 S183 3.4.21.46 0004252,0006508 ic50=0.012uM remove_due_to_license_issue IC50=12nM P00746 30995036 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 6qmt A 1.8 BS01 J7B A 1 L41 C42 H57 D61 D189 S190 C191 K192 G193 S195 S215 R218 C220 L25 C26 H41 D45 D177 S178 C179 K180 G181 S183 S199 R202 C204 H57 D102 K192 G193 D194 S195 H41 D89 K180 G181 D182 S183 3.4.21.46 0004252,0006508 ic50=0.12uM remove_due_to_license_issue IC50=120nM P00746 30995036 301 ILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLASA 6qmu A 1.98 BS01 ZCQ A 1 X36 F52 S68 W79 R81 X32 F48 S64 W75 R77 ? 0005506,0005515,0005576,0005615,0006826,0006915,0015891,0031410,0035580,0036094,0042742,0042802,0045087,0060205,0070062,0120162,0140315,1903981 remove_due_to_license_issue P80188 31390134 201 SDLIPAPPLSKVPLQQNFQDNQFHGKWYVVGFAGNAILREDKDPQKMFATIYELKEDKSYNVTSVLFRKKKCDYWIRTFVPGSQPGEFTLGNIKSYPGLTSYLVRVVSTNYNQHAMVFFKWVSQNREYFNITLYGRTKELTSELKENFIRFSKSLGLPENHIVFPVPIDQCIDGSAWSHPQFEK 6qpl B 1.6 BS01 JC5 B 1 D95 H139 F141 W151 Y170 Y177 Y179 D184 D44 H79 F81 W91 Y110 Y117 Y119 D124 ? 0007276 ic50=77nM remove_due_to_license_issue IC50=77nM, Kd=91nM Q9Y657 31260300 305 NIVGCRIQHGWKEGNGPVTQWKGTVLDQVPVNPSLYLIKYDGFDCVYGLELNKDERVSALEVLPDRVLADTMIGKAVEHMFETEDGSKDEWRGMVLARAPVMNTWFYITYEKDPVLYMYQLLDDYKEGDLRIMPSLVGKQVEYADGSKRTGMVIHQVEAKPSVYFIKFDDDFHIYVYDLVKTSAENLYFQ 6qqq A 1.85 BS01 JDE A 1 P83 T84 P85 Y111 E112 S132 I133 V137 L138 G140 G141 P84 T85 P86 Y112 E113 S133 I134 V138 L139 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=6.7uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qqq B 1.85 BS01 JDE B 1 P83 T84 P85 E112 S132 I133 V137 L138 G140 G141 P73 T74 P75 E102 S122 I123 V127 L128 G130 G131 P85 E112 R154 P75 E102 R144 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=6.7uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qqt A 1.673 BS01 JCH A 1 P83 T84 P85 G109 R110 Y111 E112 I133 G134 Y136 V137 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 E113 I134 G135 Y137 V138 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=59uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qqt B 1.673 BS01 JCH B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 L138 N139 G140 G141 P74 T75 P76 G100 R101 Y102 E103 S123 I124 G125 Y127 L129 N130 G131 G132 P85 E112 R154 P76 E103 R145 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=59uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQAGLVDVAVHDLRRWTHDVSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qqu A 1.59 BS01 JF8 A 1 P83 T84 P85 G109 R110 S132 I133 G134 Y136 L138 G140 G141 A144 P85 T86 P87 G111 R112 S134 I135 G136 Y138 L140 G142 G143 A146 P85 E112 R154 P87 E114 R156 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=5uM remove_due_to_license_issue B1MDI3 31282680 301 GSMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qqu B 1.59 BS01 JF8 B 1 P83 T84 P85 G109 R110 S132 G134 Y136 L138 N139 G140 G141 P72 T73 P74 G98 R99 S121 G123 Y125 L127 N128 G129 G130 P85 E112 R154 P74 E101 R143 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=5uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qqv A 1.712 BS01 JEW A 1 P83 T84 P85 G109 R110 Y111 E112 I133 G134 Y136 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 E113 I134 G135 Y137 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=12uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qqv B 1.712 BS01 JEW B 1 P83 T84 P85 G109 R110 Y111 E112 G113 S132 I133 G134 Y136 L138 N139 G140 G141 P71 T72 P73 G97 R98 Y99 E100 G101 S120 I121 G122 Y124 L126 N127 G128 G129 P85 E112 R154 P73 E100 R142 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=12uM remove_due_to_license_issue B1MDI3 31282680 303 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qqw A 1.8 BS01 JDQ A 1 P83 T84 P85 G109 R110 Y111 E112 I133 G134 Y136 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 E113 I134 G135 Y137 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=19uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qqw B 1.8 BS01 JDQ B 1 P83 T84 P85 G109 R110 Y111 E112 I133 G134 Y136 L138 G140 G141 P68 T69 P70 G94 R95 Y96 E97 I118 G119 Y121 L123 G125 G126 P85 E112 R154 P70 E97 R139 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=19uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qqz A 1.702 BS01 JEB A 1 P83 T84 P85 G109 R110 Y111 E112 S132 G134 Y136 V137 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 E113 S133 G135 Y137 V138 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.18uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qqz B 1.702 BS01 JEB B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 G141 P68 T69 P70 G94 R95 Y96 E97 S117 I118 G119 Y121 V122 L123 N124 G125 G126 P85 E112 R154 P70 E97 R139 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.18uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qr0 A 1.59 BS01 JFB A 1 P83 T84 P85 G109 R110 Y111 E112 S132 G134 Y136 V137 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 E113 S133 G135 Y137 V138 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.12uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr0 B 1.59 BS01 JFB B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 G141 P68 T69 P70 G94 R95 Y96 E97 S117 I118 G119 Y121 V122 L123 N124 G125 G126 P85 E112 R154 P70 E97 R139 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.12uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSPT 6qr1 A 1.67 BS01 JFT A 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 A144 P84 T85 P86 G110 R111 Y112 E113 S133 I134 G135 Y137 V138 L139 N140 G141 A145 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=8.5uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr1 B 1.67 BS01 JFT B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 A144 P69 T70 P71 G95 R96 Y97 E98 S118 I119 G120 Y122 V123 L124 N125 G126 A130 P85 E112 R154 P71 E98 R140 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=8.5uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRGLVDVAVHDLRRWTSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qr2 A 1.55 BS01 JQB A 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 L138 N139 G140 G141 A144 P84 T85 P86 G110 R111 Y112 E113 S133 I134 G135 Y137 L139 N140 G141 G142 A145 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=3.2uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr2 B 1.55 BS01 JQB B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 L138 G140 G141 P68 T69 P70 G94 R95 Y96 E97 S117 I118 G119 Y121 L123 G125 G126 P85 E112 R154 P70 E97 R139 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=3.2uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qr3 A 1.614 BS01 JE8 A 1 P83 T84 P85 G109 R110 Y111 E112 S132 G134 Y136 V137 L138 N139 G140 G141 A144 P84 T85 P86 G110 R111 Y112 E113 S133 G135 Y137 V138 L139 N140 G141 G142 A145 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.36uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr3 B 1.614 BS01 JE8 B 1 P83 T84 P85 G109 R110 Y111 E112 S132 G134 Y136 L138 N139 G140 G141 A144 P67 T68 P69 G93 R94 Y95 E96 S116 G118 Y120 L122 N123 G124 G125 A128 P85 E112 R154 P69 E96 R138 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.36uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPGLVDVAVHDLRRWTSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qr4 A 1.52 BS01 JD8 A 1 P83 T84 P85 G109 R110 Y111 S132 G134 Y136 V137 L138 N139 G140 G141 A144 P85 T86 P87 G111 R112 Y113 S134 G136 Y138 V139 L140 N141 G142 G143 A146 P85 E112 R154 P87 E114 R156 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.59uM remove_due_to_license_issue B1MDI3 31282680 301 GSMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr4 B 1.52 BS01 JD8 B 1 P83 T84 P85 G109 R110 Y111 S132 I133 G134 Y136 L138 N139 G140 G141 P73 T74 P75 G99 R100 Y101 S122 I123 G124 Y126 L128 N129 G130 G131 P85 E112 R154 P75 E102 R144 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=0.59uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qr7 A 2.03 BS01 JEK A 1 P83 T84 P85 G109 R110 Y111 E112 S132 G134 Y136 V137 L138 N139 G140 G141 P85 T86 P87 G111 R112 Y113 E114 S134 G136 Y138 V139 L140 N141 G142 G143 P85 E112 R154 P87 E114 R156 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=70nM remove_due_to_license_issue B1MDI3 31282680 301 GSMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr7 B 2.03 BS01 JEK B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 G141 P70 T71 P72 G96 R97 Y98 E99 S119 I120 G121 Y123 V124 L125 N126 G127 G128 P85 E112 R154 P72 E99 R141 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=70nM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPGLVDVAVHDLRRWTHDVSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDS 6qr9 A 2.42 BS01 JEE A 1 P83 T84 P85 G109 R110 Y111 E112 S132 G134 Y136 V137 L138 N139 G140 G141 P85 T86 P87 G111 R112 Y113 E114 S134 G136 Y138 V139 L140 N141 G142 G143 P85 E112 R154 P87 E114 R156 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=190nM remove_due_to_license_issue B1MDI3 31282680 301 GSMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qr9 B 2.42 BS01 JEE B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 G141 P73 T74 P75 G99 R100 Y101 E102 S122 I123 G124 Y126 V127 L128 N129 G130 G131 P85 E112 R154 P75 E102 R144 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=190nM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDS 6qra A 1.71 BS01 JDK A 1 P83 T84 P85 G109 R110 Y111 S132 I133 G134 Y136 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 S133 I134 G135 Y137 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=710nM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qra B 1.71 BS01 JDK B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 L138 N139 G140 G141 P73 T74 P75 G99 R100 Y101 E102 S122 I123 G124 Y126 L128 N129 G130 G131 P85 E112 R154 P75 E102 R144 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=710nM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qrc A 1.73 BS01 JFE A 1 P83 T84 P85 G109 R110 Y111 E112 I133 G134 Y136 L138 N139 G140 G141 P84 T85 P86 G110 R111 Y112 E113 I134 G135 Y137 L139 N140 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=13uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGNASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qrc B 1.73 BS01 JFE B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 L138 G140 G141 P73 T74 P75 G99 R100 Y101 E102 S122 I123 G124 Y126 L128 G130 G131 P85 E112 R154 P75 E102 R144 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=13uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSPT 6qrd A 1.75 BS01 JEH A 1 P83 T84 P85 G109 R110 Y111 S132 I133 G134 Y136 V137 L138 N139 G140 G141 A144 P84 T85 P86 G110 R111 Y112 S133 I134 G135 Y137 V138 L139 N140 G141 G142 A145 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=100nM remove_due_to_license_issue B1MDI3 31282680 303 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qrd B 1.75 BS01 JEH B 1 P83 T84 P85 G109 R110 Y111 E112 S132 I133 G134 Y136 V137 L138 N139 G140 G141 A144 P71 T72 P73 G97 R98 Y99 E100 S120 I121 G122 Y124 V125 L126 N127 G128 G129 A132 P85 E112 R154 P73 E100 R142 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=100nM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVGLVDVAVHDLRRWTHDVSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qre A 1.93 BS01 JCQ A 1 P83 T84 P85 G113 S132 I133 L138 G140 G141 P84 T85 P86 G114 S133 I134 L139 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=14uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qre A 1.93 BS02 JCQ B 2 P85 A86 Y111 D135 Y136 V137 P86 A87 Y112 D136 Y137 V138 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=14uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qre A 1.93 BS03 JCQ B 3 L179 E180 L163 E164 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=14uM remove_due_to_license_issue B1MDI3 31282680 303 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qre B 1.93 BS01 JCQ B 1 P83 T84 P85 S132 I133 G134 L138 G140 G141 P80 T81 P82 S129 I130 G131 L135 G137 G138 P85 E112 R154 P82 E109 R151 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=14uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVMASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qre B 1.93 BS02 JCQ B 2 M175 L178 E180 L226 M157 L160 E162 L208 P85 E112 R154 P82 E109 R151 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=14uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVRGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVMASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qre B 1.93 BS03 JCQ B 3 P85 A86 D135 P82 A83 D132 P85 E112 R154 P82 E109 R151 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=14uM remove_due_to_license_issue B1MDI3 31282680 303 SMKIDVVTIFPEYLQPVRGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVMASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qrf A 1.86 BS01 JF5 A 1 T84 P85 E112 G113 S132 I133 L138 G140 G141 T85 P86 E113 G114 S133 I134 L139 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=33uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qrf A 1.86 BS02 JF5 A 2 P85 D135 P86 D136 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=33uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qrf A 1.86 BS03 JF5 A 3 L179 E180 L165 E166 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=33uM remove_due_to_license_issue B1MDI3 31282680 303 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLGSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qrf B 1.86 BS01 JF5 A 2 A176 E180 A148 E152 P85 E112 R154 P73 E100 R142 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=33uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVDAGLVDVAVHDLRRWTKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qrf B 1.86 BS02 JF5 A 3 P85 D135 P73 D123 P85 E112 R154 P73 E100 R142 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=33uM remove_due_to_license_issue B1MDI3 31282680 303 SMKIDVVTIFPEYLQPVDAGLVDVAVHDLRRWTKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qrf B 1.86 BS03 JF5 B 1 T84 P85 E112 S132 I133 L138 G140 G141 T72 P73 E100 S120 I121 L126 G128 G129 P85 E112 R154 P73 E100 R142 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=33uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVDAGLVDVAVHDLRRWTKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVASLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qrg A 1.84 BS01 JET A 1 P83 T84 P85 Y111 G113 I114 S132 I133 L138 G140 G141 P84 T85 P86 Y112 G114 I115 S133 I134 L139 G141 G142 P85 E112 R154 P86 E113 R155 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=10uM remove_due_to_license_issue B1MDI3 31282680 301 SMKIDVVTIFPEYLQPVRQSLPGKAIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVLSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLL 6qrg B 1.84 BS01 JET B 1 V82 P83 P85 Y111 G113 S132 I133 L138 G140 G141 V80 P81 P83 Y109 G111 S130 I131 L136 G138 G139 P85 E112 R154 P83 E110 R152 2.1.1.228 0002939,0005737,0005829,0006400,0008033,0008168,0032259,0052906 Kd=10uM remove_due_to_license_issue B1MDI3 31282680 302 SMKIDVVTIFPEYLQPVRQSLPIDAGLVDVAVHDLRRWTHDVHKSVDDSPYGGGPGMVMKPTVWGDALDEICTSETLLVVPTPAGYPFTQETAWQWSTEDHLVIACGRYEGIDQRVADDAATRMRVREVSIGDYVLNGGEAAALVIIEAVLRLVPGVSLLEGPSYTRPPSWRGMDVPPVLLSGDHAKIAAWRAEQSRQRTIERRPDLLGFDSP 6qri B 2.4 BS02 CV9 B 1 D24 D25 Y143 A144 G146 I341 I345 L349 D20 D21 Y128 A129 G131 I326 I330 L334 3.6.4.- 0000287,0001725,0003785,0005509,0005515,0005523,0005524,0005737,0005856,0005865,0005884,0010628,0016787,0019904,0030027,0030041,0030175,0030240,0031013,0031432,0031941,0032036,0032432,0042802,0044297,0048306,0048741,0051017,0090131,0098723,0140660 remove_due_to_license_issue P68135 31260301 403 TTALVCDNGSGLVKAGFAGDDAPRAVFPSIVGRPRDSYVGDEAQSKRGILTLKYPIEHGIITNWDDMEKIWHHTFYNELRVAPEEHPTLLTEAPLNPKANREKMTQIMFETFNVPAMYVAIQAVLSLYASGRTTGIVLDSGDGVTHNVPIYEGYALPHAIMRLDLAGRDLTDYLMKILTERGYSFVTTAEREIVRDIKEKLCYVALDFENEMATAASSSSLEKSYELPDGQVITIGNERFRCPETLFQPSFIGMESAGIHETTYNSIMKCDIDIRKDLYANNVMSGGTTMYPGIADRMQKEITALAPSTMKIKIIAPPERKYSVWIGGSILASLSTFQQMWITKQEYDEAGPSIVHRKC 6qri B 2.4 BS03 CV9 A 1 R147 I330 R132 I315 3.6.4.- 0000287,0001725,0003785,0005509,0005515,0005523,0005524,0005737,0005856,0005865,0005884,0010628,0016787,0019904,0030027,0030041,0030175,0030240,0031013,0031432,0031941,0032036,0032432,0042802,0044297,0048306,0048741,0051017,0090131,0098723,0140660 remove_due_to_license_issue P68135 31260301 403 TTALVCDNGSGLVKAGFAGDDAPRAVFPSIVGRPRDSYVGDEAQSKRGILTLKYPIEHGIITNWDDMEKIWHHTFYNELRVAPEEHPTLLTEAPLNPKANREKMTQIMFETFNVPAMYVAIQAVLSLYASGRTTGIVLDSGDGVTHNVPIYEGYALPHAIMRLDLAGRDLTDYLMKILTERGYSFVTTAEREIVRDIKEKLCYVALDFENEMATAASSSSLEKSYELPDGQVITIGNERFRCPETLFQPSFIGMESAGIHETTYNSIMKCDIDIRKDLYANNVMSGGTTMYPGIADRMQKEITALAPSTMKIKIIAPPERKYSVWIGGSILASLSTFQQMWITKQEYDEAGPSIVHRKC 6qs5 A 1.961 BS01 JGB A 1 I66 K68 F113 V116 M163 I174 D175 I60 K62 F107 V110 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0004676,0004677,0004679,0004694,0004711,0005524,0005634,0005829,0005956,0006338,0006468,0006974,0035175,0035402,0035403,0035979,0044022,0044023,0044024,0044025,0051726,0072354,0072371,0072518,0106310,0140823,0140855,0140857,1990244 ic50=0.57uM remove_due_to_license_issue P28523 22794353 401 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAE 6qua A 2.681 BS01 dna E 0 N49 R52 N56 K73 R74 N40 R43 N47 K64 R65 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 SDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qua A 2.681 BS02 dna F 0 Y32 L34 H50 Y54 K68 R74 T75 N76 Y23 L25 H41 Y45 K59 R65 T66 N67 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 SDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qua B 2.681 BS01 dna E 0 Y32 G33 L34 H50 Y54 K68 R74 T75 N76 Y27 G28 L29 H45 Y49 K63 R69 T70 N71 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qua B 2.681 BS02 dna F 0 G51 R52 N56 G46 R47 N51 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 PDARSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALE 6qua C 2.681 BS01 dna G 0 Y32 G33 L34 H50 Y54 K68 R74 T75 N76 Y22 G23 L24 H40 Y44 K58 R64 T65 N66 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALEH 6qua C 2.681 BS02 dna H 0 N49 G51 R52 N56 K73 R74 N39 G41 R42 N46 K63 R64 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 DARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALEH 6qua D 2.681 BS01 dna G 0 N49 R52 N56 K73 R74 N41 R44 N48 K65 R66 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 RSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALEH 6qua D 2.681 BS02 dna H 0 Y32 G33 L34 H50 Y54 R74 T75 N76 Y24 G25 L26 H42 Y46 R66 T67 N68 ? 0046872 remove_due_to_license_issue Q9HSF4 31310308 1 ~ 28 RSDARDLTAFQKNILTVLGEEARYGLAIKRELEEYYGEEVNHGRLYPNLDDLVNKGLVEKSELDKRTNEYALTNEGFDAVVDDLEWTLSKFVADADRRERVETIVADDAAALEH 6quv B 1.475 BS01 JJN B 1 K5 V7 S39 D54 L56 T74 K5 V7 S39 D54 L56 T74 3.6.5.2 0003924,0005525,0007165,0016020 Kd=1mM remove_due_to_license_issue P01116 31231840 201 MTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6quw B 1.242 BS02 JJQ B 1 K5 V7 S39 D54 L56 T74 K5 V7 S39 D54 L56 T74 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 31231840 203 MTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHK 6qw7 B 1.78 BS01 MK7 B 1 S70 H105 S130 N132 N170 T216 T235 G236 S237 S50 H85 S110 N112 N150 T196 T215 G216 S217 S70 K73 S130 E166 K234 S237 S50 K53 S110 E146 K214 S217 3.5.2.6 0008800,0016787,0017001,0030655,0046677 ic50=470nM remove_due_to_license_issue Q9RBQ1 31383664 301 NAPTDAAITAASDFAALEKACAGRLGVTLLDTASGRRIGHRQDERFPMCSTFKSMLAATVLSQAERMPALLDRRVPVGEADLLSHAPVTRRHAGKDMTVRDLCRATIITSDNTAANLLFGVVGGPPAVTAFLRASGDTVSRSDRLEPELNSFAKGDPRDTTTPAAMAATLQRVVLGEVLQPASRQQLADWLIDNETGDACLRAGLGKRWRVGDKTGSNGEDARNDIAVLWPVAGGAPWVLTAYLQAGAISYEQRASVLAQVGRIADRLIG 6qw8 A 1.1 BS01 MK7 A 1 S70 N104 S130 N132 T216 T235 G236 S237 S43 N77 S103 N105 T189 T208 G209 S210 S70 K73 S130 E166 K234 S237 S43 K46 S103 E139 K207 S210 3.5.2.6 0008800,0017001,0030655,0046677 remove_due_to_license_issue G3G192 31383664 301 ADVQQKLAELERQSGGRLGVALINTADNSQILYRADERFAMCSTSKVMAAAAVLKKSESEPNLLNQRVEIKKSDLVNYNPIAEKHVNGTMSLAELSAAALQYSDNVAMNKLIAHVGGPASVTAFARQLGDETFRLDRTEPTLNTAIPGDPRDTTSPRAMAQTLRNLTLGKALGDSQRAQLVTWMKGNTTGAASIQAGLPASWVVGDKTGSGGYGTTNDIAVIWPKDRAPLILVTYFTQPQPKAESRRDVLASAAKIVTDGL 6qw9 A 1.04 BS01 MK7 A 1 S70 W105 S130 N170 T235 G236 T237 S45 W80 S105 N145 T210 G211 T212 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31383664 305 LTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6qwa A 1.06 BS01 MK7 A 1 S70 W105 S130 T235 G236 T237 S45 W80 S105 T210 G211 T212 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31383664 305 LTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKYSEAVIAAAARLALEGLGVNG 6qwb A 1.04 BS02 MK7 A 1 S70 W105 S130 T235 G236 T237 S45 W80 S105 T210 G211 T212 S70 K73 S130 E166 K234 T237 S45 K48 S105 E141 K209 T212 3.5.2.6 0008800,0016787,0017001,0030655,0046677 remove_due_to_license_issue Q9F663 31383664 307 LTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVRWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGGYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNG 6qwi A 2.85 BS01 JJW A 1 Q20 H121 W122 E166 L173 W326 E352 W398 E405 W406 Q20 H121 W122 E166 L173 W326 E352 W398 E405 W406 3.2.1.21 0004553,0005829,0005975,0008422,0016052,0016798,0030245 remove_due_to_license_issue P22073 31226649 501 MTIFQFPQDFMWGTATAAYQIEGAYQEDGRGLSIWDTFAHTPGKVFNGDNGNVACDSYHRYEEDIRLMKELGIRTYRFSVSWPRIFPNGDGEVNQKGLDYYHRVVDLLNDNGIEPFCTLYHWDLPQALQDAGGWGNRRTIQAFVQFAETMFREFHGKIQHWLTFNEPWCIAFLSNMLGVHAPGLTNLQTAIDVGHHLLVAHGLSVRRFRELGTSGQIGIAPNVSWAVPYSTSEEDKAACARTISLHSDWFLQPIYQGSYPQFLVDWFAEQGATVPIQDGDMDIIGEPIDMIGINYYSMSVNRFNPEAGFLQSEEINMGLPVTDIGWPVESRGLYEVLHYLQKYGNIDIYITENGACINDEVVNGKVQDDRRISYMQQHLVQVHRAIHDGLHVKGYMAWSLLDNFEWAEGYSMRFGIIHVDFRTQVRTPKESYYWYRKVVGNNWLETRR 6qxa A 3.41 BS08 GQB A 1 Q268 G528 P530 Q267 G527 P529 7.2.3.1 0000287,0004427,0005509,0005515,0005886,0006814,0009678,0015081,0016020,0030955,0035725,0042803,0046872,1902600 remove_due_to_license_issue Q9S5X0 31131322 809 YVAALFFLIPLVALGFAAANFAAVVRKPEGTERMKEISSYIRSGADSFLAHETKAIFKVAIVIAILLMIFTTWQTGVAFLLGAVMSASAGIVGMKMATRANVRVAEAARTTKKIGPALKVAYQGGSVMGLSVGGFALLGLVLVYLIFGKWMGQVDNLNIYTNWLGINFVPFAMTVSGYALGCSIIAMFDRVGGGVYTKAADMAADLVGKTELNLPEDDPRNPATIADNVGDNVGDVAGLGADLLESFVGAIVSSIILASYMFPIYVQKIGENLVHQVPKETIQALISYPIFFALVGLGCSMLGILYVIVKKPSDNPQRELNISLWTSALLTVVLTAFLTYFYLKDLQGLDVLGFRFGAISPWFSAIIGIFSGILIGFWAEYYTSYRYKPTQFLGKSSIEGTGMVISNGLSLGMKSVFPPTLTLVLGILFADYFAGLYGVAIAALGMLSFVATSVSVDSYGPIADNAGGISEMCELDPEVRKITDHLDAVGNTTAAIGKGFAIGSAIFAALSLFASYMFSQISPSDIGKPPSLVLLLNMLDARVIAGALLGAAITYYFSGYLISAVTKAAMKMVDEIRRQAREIPGLLEGKAKPDYNRCIEITSDNALKQMGYPAFIAILTPLVTGFLLGAEFVGGVLIGTVLSGAMLAILTANSGGAWDNAKKYLEAGNLEGYGKGSEPHKALVIGDTVGDPLKDTVGPSLDILIKIMSVVSVIAVSIFKHVHLF 6qxa A 3.41 BS09 GQB A 2 Q268 D351 V352 Q267 D350 V351 7.2.3.1 0000287,0004427,0005509,0005515,0005886,0006814,0009678,0015081,0016020,0030955,0035725,0042803,0046872,1902600 remove_due_to_license_issue Q9S5X0 31131322 810 YVAALFFLIPLVALGFAAANFAAVVRKPEGTERMKEISSYIRSGADSFLAHETKAIFKVAIVIAILLMIFTTWQTGVAFLLGAVMSASAGIVGMKMATRANVRVAEAARTTKKIGPALKVAYQGGSVMGLSVGGFALLGLVLVYLIFGKWMGQVDNLNIYTNWLGINFVPFAMTVSGYALGCSIIAMFDRVGGGVYTKAADMAADLVGKTELNLPEDDPRNPATIADNVGDNVGDVAGLGADLLESFVGAIVSSIILASYMFPIYVQKIGENLVHQVPKETIQALISYPIFFALVGLGCSMLGILYVIVKKPSDNPQRELNISLWTSALLTVVLTAFLTYFYLKDLQGLDVLGFRFGAISPWFSAIIGIFSGILIGFWAEYYTSYRYKPTQFLGKSSIEGTGMVISNGLSLGMKSVFPPTLTLVLGILFADYFAGLYGVAIAALGMLSFVATSVSVDSYGPIADNAGGISEMCELDPEVRKITDHLDAVGNTTAAIGKGFAIGSAIFAALSLFASYMFSQISPSDIGKPPSLVLLLNMLDARVIAGALLGAAITYYFSGYLISAVTKAAMKMVDEIRRQAREIPGLLEGKAKPDYNRCIEITSDNALKQMGYPAFIAILTPLVTGFLLGAEFVGGVLIGTVLSGAMLAILTANSGGAWDNAKKYLEAGNLEGYGKGSEPHKALVIGDTVGDPLKDTVGPSLDILIKIMSVVSVIAVSIFKHVHLF 6qxd A 2.317 BS03 JKB A 1 H42 H60 H69 F197 H204 N205 H208 R209 G216 V218 A221 F227 H231 H39 H57 H66 F194 H201 N202 H205 R206 G213 V215 A218 F224 H228 ? 0016491,0046872 ic50=0.96uM remove_due_to_license_issue B2ZB02 31202126 303 KYRVRKNVLHLTDTEKRDFVRTVLILKEKGIYDRYIAWHGAAGKFHTPPGSDRNAAHMSSAFLPWHREYLLRFERDLQSINPEVTLPYWEWETDAQMQDPSQSQIWSADFMGGNGNPIKDFIVDTGPFAAGRWTTIDEQGNPSGGLKRNFGATKEAPTLPTRDDVLNALKITQYDTPPWDMTSQNSFRNQLEGFINGPQLHNRVHRWVGGQMGVVPTAPNDPVFFLHHANVDRIWAVWQIIHRNQNYQPMKNGPFGQNFRDPMYPWNTTPEDVMNHRKLGYVYDIEL 6qxj A 1.7 BS03 JKQ A 1 F228 V253 R263 T266 F270 F421 V446 R456 T459 F463 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q07820 31339316 401 MKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6qxs A 2.88 BS01 UFP B 1 R177 R178 R156 R157 E59 W81 Y145 C197 R217 D220 E59 W81 Y124 C176 R196 D199 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue Q834R3 30935102 401 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPI 6qxs B 2.88 BS01 UFP B 1 R22 Y145 C197 H198 R217 S218 D220 N228 H258 Y260 R22 Y145 C197 H198 R217 S218 D220 N228 H258 Y260 E59 W81 Y145 C197 R217 D220 E59 W81 Y145 C197 R217 D220 2.1.1.45 0004799,0005737,0005829,0006231,0006235,0008168,0009165,0016741,0032259 remove_due_to_license_issue Q834R3 30935102 401 MEEAYLALGKKILEEGHFKEDRTGTGTYSLFGYQMRFDLAKGFPLLTTKRVPFGLIKSELLWFLKGDTNIRYLLERNNHIWDEWAFERYVKSADYQGPDMTDFGHRVLQDPAFAEQYKEEHQKFCDAILNDAEFAEKYGELGNIYGAQWRHWETKDGSFIDQLANVIEMIKTNPDSRRLIVSAWNPEDVPSMALPPCHTMFQFYVNEGKLSCQLYQRSADVFLGVPFNIASYALLTHLIAHETGLEVGEFVHTLGDAHLYQNHVEQMQEQLSREVRSFPTLVLNPDKASVFDFDMEDIKVEGYDPHPTIKAPIAV 6qxu A 1.2 BS01 JKN A 1 H1184 G1185 Y1203 Y1213 F1214 A1215 K1220 S1221 Y1224 H80 G81 Y99 Y109 F110 A111 K116 S117 Y120 2.4.2.-,2.4.2.30 0003950 ic50=7nM remove_due_to_license_issue IC50=10.0nM O95271 31381853 1402 GTILLDLAPEDKEYQSVEEEMQSTIREHRDGGNAGGIFNRYNVIRIQKVVNKKLRERFCHRQKEVSEENHNHHNERMLFHGSPFINAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPTHKDRSCYICHRQMLFCRVTLGKSFLQFSTMKMAHAPPGHHSVIGRPSVNGLAYAEYVIYRGEQAYPEYLITYQIMKP 6qyk A 2.3 BS03 JLB A 1 F228 M231 V253 R263 T266 L267 F270 F422 M425 V447 R457 T460 L461 F464 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q07820 31339316 401 MKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6qyl A 2.2 BS03 JLE A 1 H224 A227 M231 V253 R263 T266 L267 F270 H416 A419 M423 V445 R455 T458 L459 F462 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q07820 31339316 401 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6qyn A 2.5 BS03 JL8 A 1 H224 A227 M231 V253 R263 T266 L267 F270 H418 A421 M425 V447 R457 T460 L461 F464 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q07820 31339316 401 MKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6qyo A 2.1 BS03 JLH A 1 H224 A227 F228 M231 V253 R263 T266 L267 F270 H416 A419 F420 M423 V445 R455 T458 L459 F462 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q07820 31339316 401 MKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6qyp A 2.2 BS01 JL5 A 1 H224 A227 F228 M231 V253 R263 T266 L267 H55 A58 F59 M62 V84 R94 T97 L98 ? 0003824,0042981 remove_due_to_license_issue Ki=46nM Q07820 31339316 401 SEDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6qz5 A 2.0 BS01 JLE A 1 H224 A227 F228 M231 V253 R263 T266 L267 H55 A58 F59 M62 V84 R94 T97 L98 ? 0003824,0042981 remove_due_to_license_issue Ki=1600nM Q07820 31339316 401 SEDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6qz6 A 1.9 BS01 JLE A 1 H224 F228 M231 V253 R263 T266 L267 F270 H55 F59 M62 V84 R94 T97 L98 F101 ? 0003824,0042981 remove_due_to_license_issue Ki=1600nM Q07820 31339316 401 SEDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6qz7 A 2.2 BS03 JLE A 1 H224 M231 V253 R263 T266 F270 H416 M423 V445 R455 T458 F462 ? 0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0042981,0043190,0055052,0055085,0060326,1901982,1990060 remove_due_to_license_issue P0AEX9,Q07820 31339316 401 KIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPDKAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTGSELYRQSLEIISRYLREQATGAADTAPMGASGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6qz8 A 2.15 BS01 JL8 A 1 H224 A227 F228 M231 V253 R263 T266 L267 F270 H55 A58 F59 M62 V84 R94 T97 L98 F101 ? 0003824,0042981 remove_due_to_license_issue Ki=51nM Q07820 31339316 401 SEDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVE 6qzb A 2.0 BS01 JLK A 1 H224 F228 M231 V253 R263 T266 F270 H54 F58 M61 V83 R93 T96 F100 ? 0003824,0042981 remove_due_to_license_issue Ki=2400nM Q07820 31339316 401 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFH 6qzh A 2.1 BS01 JLW A 1 V79 T82 F86 T91 T93 D94 L97 R154 I262 Y326 V331 K332 F333 V28 T31 F35 T40 T42 D43 L46 R103 I673 Y729 V734 K735 F736 3.2.1.18 0004930,0004950,0006935,0006954,0006955,0007186,0016020,0016493 Kd=3nM remove_due_to_license_issue P32248,P62576 31442409 1502 DVRNFKAWFLPIMYSIICFVGLLGNGLVVLTYIYFKRLKTMTDTYLLNLAVADILFLLTLPFWAYSAAKSWVFGVHFCKLIFAIYKMSFFSGMWLLLCISIDRYVAIVHRHRARVLLISKLSCVGIWILATVLSIPELLYSDLQRSSSEQAMRCSLITEHVEAFITIQVAQMVIGFLVPLLAMSFCYLVIISKLHALTEKTDIFESGRNGNPNKDGIKSYRIPALLKTDKGTLIAGADERRLHSSDWGDIGMVIRRSEDNGKTWGDRVTITNLRDNPKASDPSIGSPVNIDMVLVQDPETKRIFSIYDMFPEGKGIFGMSSQKEEAYKKIDGKTYQILYREGEKGAYTIRENGTVYTPDGKATDYRVVVDPVKPAYSDKGDLYKGDQLLGNIYFTTNKTSPFRIAKDSYLWMSYSDDDGKTWSAPQDITPMVKADWMKFLGVGPGTGIVLRNGPHKGRILIPVYTTNNVSHLDGSQSSRVIYSDDHGKTWHAGEAVNDNRQVDGQKIHSSTMNNRRAQNTESTVVQLNNGDVKLFMRGLTGDLQVATSKDGGVTWEKDIKRYPQVKDVYVQMSAIHTMHEGKEYIILSNAGGPKRENGMVHLARVEENGELTWLKHNPIQKGEFAYNSLQELGNGEYGILYEHTEKGQNAYTLSFRKFNWEFLSKSKGHERNIKVIIAVVVVFIVFQLPYNGVVLAQTVTCELSKQLNIAYDVTYSLACVRCCVNPFLYAFIGVKFRNDLFKLF 6r0k A 1.15 BS02 JNN A 1 P464 S531 H573 H574 F583 D612 H614 F643 L712 Y745 P23 S90 H132 H133 F142 D171 H173 F202 L271 Y304 ? ic50=12nM remove_due_to_license_issue F8W4B7 31414801 2004 PITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLTPLKTSATVSINNVLRAHAPFWSSLR 6r0s C 1.55 BS02 JOH C 1 N50 F77 W79 W85 W99 N34 F61 W63 W69 W83 ? 0046872 remove_due_to_license_issue Ki=>40000nM A4TVL0 31251063 202 PGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r0u C 1.7 BS02 JO5 C 1 N50 P51 F77 W79 W99 Y101 N33 P34 F60 W62 W82 Y84 ? 0046872 remove_due_to_license_issue Ki=>40000nM A4TVL0 31251063 202 GASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r0v A 1.6 BS02 JO2 A 1 N50 F77 W79 W85 H96 W99 Y101 N37 F64 W66 W72 H83 W86 Y88 ? 0046872 remove_due_to_license_issue A4TVL0 31251063 202 VLAPGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r0x E 3.13 BS03 SGN H 2 R111 H112 R81 H82 ? 0016020 remove_due_to_license_issue O95866 31436532 7 GASLDGRPGDRVDLSCGGVRWVWAPSFPACKGLSKGRRPILWAAAAGAPTVPPLQPFVGRIRRLELLLSAGDSGTFFCKGRHEDESRTVLHVLGDRTYC 6r0x F 3.13 BS01 SGN H 1 R60 P62 K109 R38 P40 K80 ? 0016020 remove_due_to_license_issue O95866 31436532 5 PGASLDGRPGDRVDLSCGGVRWVWAPSFPACKGLSKGRRPILWAAAAGAPTVPPLQPFVGRIRRLELLLSAGDSGTFFCKGRHEDESRTVLHVLGDRT 6r11 A 1.75 BS02 JOB A 1 N50 F77 W79 W85 W99 Y101 N35 F62 W64 W70 W84 Y86 ? 0046872 Ki=12uM remove_due_to_license_issue Ki=12000nM A4TVL0 31251063 202 APGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPAD 6r12 B 1.74 BS02 JOT B 1 N50 P51 F77 W79 W85 W99 Y101 N32 P33 F59 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue Ki=>40000nM A4TVL0 31251063 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r13 B 1.65 BS02 JOK B 1 N50 P51 S78 W79 W85 W99 Y101 N32 P33 S60 W61 W67 W81 Y83 ? 0046872 remove_due_to_license_issue A4TVL0 31251063 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r18 B 1.35 BS02 JOQ B 1 N50 F77 S78 W79 W85 I87 H96 W99 Y101 N36 F63 S64 W65 W71 I73 H82 W85 Y87 ? 0046872 remove_due_to_license_issue A4TVL0 31251063 202 MVLAPSIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r1a C 1.54 BS02 JP8 C 1 N50 F77 S78 W79 W85 W99 Y101 N35 F62 S63 W64 W70 W84 Y86 ? 0046872 remove_due_to_license_issue A4TVL0 31251063 202 APGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r1b A 2.27 BS01 CH5 A 1 Y78 D102 S153 W208 S272 G305 G306 Y345 Y43 D67 S118 W173 S237 G270 G271 Y310 ? 0005886,0046872 Kd=3.6uM remove_due_to_license_issue P71619 31433162 501 SGPIDFWSSHPGQSSAAERELIGRFQDRFPTLSVKLIDAGKDYDEVAQKFNAALIGTDVPDVVLLDDRWWFHFALSGVLTALDDLFGQVGVDTTDYVDSLLADYEFNGRHYAVPYARSTPLFYYNKAAWQQAGLPDRGPQSWSEFDEWGPELQRVVGAGRSAHGWANADLISWTFQGPNWAFGGAYSDKWTLTLTEPATIAAGNFYRNSIHGKGYAAVANDIANEFATGILASAVASTGSLAGITASARFDFGAAPLPTGPDAAPACPTGGAGLAIPAKLSEERKVNALKFIAFVTNPTNTAYFSQQTGYLPVRKSAVDDASERHYLADNPRARVALDQLPHTRTQDYARVFLPGGDRIISAGLESIGLRGADVTKTFTNIQKRLQVILDRQIM 6r1c B 1.5 BS02 JOW B 1 N50 M54 F77 W79 W85 I87 H96 W99 Y101 N37 M41 F64 W66 W72 I74 H83 W86 Y88 ? 0046872 remove_due_to_license_issue Ki=12000nM A4TVL0 31251063 202 VLAPGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r1d A 1.1 BS02 JP5 A 1 N50 F77 W79 W85 I87 H96 W99 Y101 N32 F59 W61 W67 I69 H78 W81 Y83 ? 0046872 Ki=4uM remove_due_to_license_issue Ki=4000nM A4TVL0 31251063 202 ASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPAD 6r1k A 1.94 BS02 JPB A 1 N50 P51 F77 W79 W85 I87 W99 Y101 N31 P32 F58 W60 W66 I68 W80 Y82 ? 0046872 Ki=9uM remove_due_to_license_issue Ki=9000nM A4TVL0 31251063 202 SIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r1w B 1.35 BS02 JPW B 1 N50 F77 S78 W79 W85 W99 Y101 N38 F65 S66 W67 W73 W87 Y89 ? 0046872 remove_due_to_license_issue A4TVL0 31251063 204 MVLAPGASIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r1x A 1.8 BS02 JPQ A 1 N50 F77 W79 W85 W99 Y101 N31 F58 W60 W66 W80 Y82 ? 0046872 remove_due_to_license_issue Ki=>40000nM A4TVL0 31251063 202 SIFRCRQCGQTISRRDWLLPMGGDHEHVVFNPAGMIFRVWCFSLAQGLRLIGAPSGEFSWFKGYDWTIALCGQCGSHLGWHYEGGSQPQTFFGLIKDRLAEGPA 6r49 A 2.209 BS03 JSB A 1 K166 L178 Y199 H201 K40 L52 Y73 H75 D256 K258 E260 N261 D274 T292 D130 K132 E134 N135 D148 T161 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 remove_due_to_license_issue O14965 31026091 504 QWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS 6r4k A 2.13 BS01 JSK A 1 Q20 H121 E166 L173 E352 W398 E405 W406 Q20 H121 E166 L173 E352 W398 E405 W406 3.2.1.21 0004553,0005829,0005975,0008422,0016052,0016798,0030245 Ki=51uM remove_due_to_license_issue P22073 31226649 501 MTIFQFPQDFMWGTATAAYQIEGAYQEDGRGLSIWDTFAHTPGKVFNGDNGNVACDSYHRYEEDIRLMKELGIRTYRFSVSWPRIFPNGDGEVNQKGLDYYHRVVDLLNDNGIEPFCTLYHWDLPQALQDAGGWGNRRTIQAFVQFAETMFREFHGKIQHWLTFNEPWCIAFLSNMLGVHAPGLTNLQTAIDVGHHLLVAHGLSVRRFRELGTSGQIGIAPNVSWAVPYSTSEEDKAACARTISLHSDWFLQPIYQGSYPQFLVDWFAEQGATVPIQDGDMDIIGEPIDMIGINYYSMSVNRFNPEAGFLQSEEINMGLPVTDIGWPVESRGLYEVLHYLQKYGNIDIYITENGACINDEVVNGKVQDDRRISYMQQHLVQVHRAIHDGLHVKGYMAWSLLDNFEWAEGYSMRFGIIHVDFRTQVRTPKESYYWYRKVVGNNWLETRR 6r4s A 2.75 BS04 ATP A 1 D79 D109 D111 S160 R162 R163 H166 L316 L317 K318 H324 D77 D107 D109 S158 R160 R161 H164 L314 L315 K316 H322 2.7.7.102 0000287,0000428,0003896,0005515,0005654,0005658,0006260,0006269,0006270,0008270,0016020,0016779,0032553,0046872 remove_due_to_license_issue P49642 31479243 504 TFDPTELPELLKLYYRRLFPYSQYYRWLNYGGVIKNYFQHREFSFTLKDDIYIRYQSFNNQSDLEKEMQKMNPYKIDIGAVYSHRPNQHNTVKLGAFQAQEKELVFDIDMTDYDDVRRCCSSADICPKCWTLMTMAIRIIDRALKEDFGFKHRLWVYSGRRGVHCWVCDESVRKLSSAVRSGIVEYLSLVKGGQDVKKKVHLSEKIHPFIRKSINIIKKYFEEYALVNQDILENKESWDKILALVPETIHDELQQSFQKSHNSLQRWEHLKKVASRYQNNIKNDKYGPWLEWEIMLQYCFPRLDINVSKGINHLLKSPFSVHPKTGRISVPIDLQKVDQFDPFTVPTISFICRELDADYKKTSLAPYVKVFEHFLENLDKSR 6r4v A 2.202 BS03 BFQ A 1 S60 D64 R73 Q126 K151 K202 S56 D60 R69 Q122 K147 K194 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 Kd=1.74uM remove_due_to_license_issue IC50=79430nM O95749 31427399 1304 QETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRDDYANLHSENKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFK 6r4v B 2.202 BS03 BFQ B 1 S60 D64 R73 L122 Q126 K151 D188 K212 S57 D61 R70 L119 Q123 K148 D185 K204 2.5.1.-,2.5.1.1,2.5.1.10,2.5.1.29 0004161,0004311,0004337,0004659,0005515,0005654,0005737,0005829,0006720,0008299,0016740,0030018,0033384,0033386,0042802,0045337,0046872,0048471 Kd=1.74uM remove_due_to_license_issue IC50=79430nM O95749 31427399 1304 TQETVQRILLEPYKYLLQLPGKQVRTKLSQAFNHWLKVPEDKLQIIIEVTEMLHNASLLIDDIEDNSKLRRGFPVAHSIYGIPSVINSANYVYFLGLEKVLTLDHQDAVKLFTRQLLELHQGQGLDIYWRDNYTCPTEEEYKAMVLQKTGGLFGLAVGLMQLFSDYKEDLKPLLNTLGLFFQIRDDYANLHSNKSFCEDLTEGKFSFPTIHAIWSRPESTQVQNILRQRTENIDIKKYCVHYLEDVGSFEYTRNTLKELEAKAYKQIDARGGNPELVALVKHLSKMFKEE 6r5f A 3.25 BS01 JSW A 1 K45 M67 L70 V76 L78 M92 L129 H136 I154 A155 D156 L157 S161 F162 K22 M41 L44 V50 L52 M66 L103 H110 I128 A129 D130 L131 S135 F136 D138 K140 E142 N143 D156 T189 D112 K114 E116 N117 D130 T147 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13546 31013427 301 VIKMKSSDSLAFHRTQGLMIMKTGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEETLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 6r64 A 2.64 BS01 dna C 0 S30 G32 P33 S65 S66 S108 R109 K113 G118 N119 K122 S32 G34 P35 S67 S68 S110 R111 K115 G120 N121 K124 3.1.21.- remove_due_to_license_issue P24200 31724709 1 ~ 10 EFMHVFDNNGIELKAECSIGEEDGVYGLILESWGPGDRNKDYNIALDYIIERLVDSGVSQVVVYLASSSVRKHMHSLDERKIHPGEYFTLIGNSPRDIRLKMCGYQAYFSRTGRKEIPSGNRTKRILINVPGIYSDSFWASIIRG 6r64 A 2.64 BS02 dna D 0 W31 P33 R97 L98 R120 W33 P35 R99 L100 R122 3.1.21.- remove_due_to_license_issue P24200 31724709 1 ~ 10 EFMHVFDNNGIELKAECSIGEEDGVYGLILESWGPGDRNKDYNIALDYIIERLVDSGVSQVVVYLASSSVRKHMHSLDERKIHPGEYFTLIGNSPRDIRLKMCGYQAYFSRTGRKEIPSGNRTKRILINVPGIYSDSFWASIIRG 6r64 B 2.64 BS01 dna E 0 S30 G32 P33 R36 S65 S66 S108 R109 K113 G118 N119 K122 S32 G34 P35 R38 S67 S68 S110 R111 K115 G120 N121 K124 3.1.21.- remove_due_to_license_issue P24200 31724709 1 ~ 10 EFMHVFDNNGIELKAECSIGEEDGVYGLILESWGPGDRNKDYNIALDYIIERLVDSGVSQVVVYLASSSVRKHMHSLDERKIHPGEYFTLIGNSPRDIRLKMCGYQAYFSRTGRKEIPSGNRTKRILINVPGIYSDSFWASIIRG 6r64 B 2.64 BS02 dna F 0 W31 P33 L98 N119 R120 W33 P35 L100 N121 R122 3.1.21.- remove_due_to_license_issue P24200 31724709 1 ~ 10 EFMHVFDNNGIELKAECSIGEEDGVYGLILESWGPGDRNKDYNIALDYIIERLVDSGVSQVVVYLASSSVRKHMHSLDERKIHPGEYFTLIGNSPRDIRLKMCGYQAYFSRTGRKEIPSGNRTKRILINVPGIYSDSFWASIIRG 6r7b A 3.12 BS01 rna D 0 G9 D10 Y14 S15 Y19 F29 S51 L52 H155 V180 M181 G9 D10 Y14 S15 Y19 F29 S51 L52 H155 V180 M181 ? remove_due_to_license_issue F0NE21 31541109 1 ~ 4 MKCLFYIAGDVSNYSIVNYELNGQTQNTFFAAHALYNLFKPDKVIALIPDSLVKDNVSDEECYKNLVINRAKELNFAGMEEFMNKVEIRKIPNVGIASAIQCENGAPKKEKNKEGREVLKRLPYNEKRSPIFIFNAIYAIFKDEACDEYLVDLTHGTNVLVSIGMNVGALFNAKFYSAPVMGMPGKDSIVNIVELTDVVQATNDSLMIRSSIENLDERYFKDYSAKLSRLNPTIFEEEEKKVLTRVKGTDVNVVINFLWNIRNGFTVNAVKSMNELKNIINQLEEDLEKLKSFYKNWEEHKNFQGETLLVLSDLDSTLKVKDLLIEGNDLEKLNYLLDLYIKASIYDKALSLARELPVAICLNKVGGGMFDDKNEKYKHCNEIVTSYLRLRYSGLMEFRNTLMHGGLSTDMKPNVDKDGNITPGKIVTKNKIEDFVKRELRNYFDKIVNFLSSA 6r7b B 3.12 BS01 rna D 0 G9 D10 S15 F29 S51 S98 H155 V180 M181 G182 G9 D10 S15 F29 S51 S98 H155 V180 M181 G182 ? remove_due_to_license_issue F0NE21 31541109 1 ~ 4 MKCLFYIAGDVSNYSIVNYELNGQTQNTFFAAHALYNLFKPDKVIALIPDSLVKDNVSDEECYKNLVINRAKELNFAGMEEFMNKVEIRKIPNVGIASAIQCENGAPKKEKNKEGREVLKRLPYNEKRSPIFIFNAIYAIFKDEACDEYLVDLTHGTNVLVSIGMNVGALFNAKFYSAPVMGMPGKDSIVNIVELTDVVQATNDSLMIRSSIENLDERYFKDYSAKLSRLNPTIFEEEEKKVLTRVKGTDVNVVINFLWNIRNGFTVNAVKSMNELKNIINQLEEDLEKLKSFYKNWEEHKNFQGETLLVLSDLDSTLKVKDLLIEGNDLEKLNYLLDLYIKASIYDKALSLARELPVAICLNKVGGGMFDDKNEKYKHCNEIVTSYLRLRYSGLMEFRNTLMHGGLSTDMKPNVDKDGNITPGKIVTKNKIEDFVKRELRNYFDKIVNFLSSA 6r7b C 3.12 BS01 rna E 0 D10 Y14 S15 V17 Y19 F29 S51 L52 A97 S98 H155 V180 M181 D10 Y14 S15 V17 Y19 F29 S51 L52 A97 S98 H155 V180 M181 ? remove_due_to_license_issue F0NE21 31541109 1 ~ 2 MKCLFYIAGDVSNYSIVNYELNGQTQNTFFAAHALYNLFKPDKVIALIPDSLVKDNVSDEECYKNLVINRAKELNFAGMEEFMNKVEIRKIPNVGIASAIQCENGAPKKEKNKEGREVLKRLPYNEKRSPIFIFNAIYAIFKDEACDEYLVDLTHGTNVLVSIGMNVGALFNAKFYSAPVMGMPGKDSIVNIVELTDVVQATNDSLMIRSSIENLDERYFKDYSAKLSRLNPTIFEEEEKKVLTRVKGTDVNVVINFLWNIRNGFTVNAVKSMNELKNIINQLEEDLEKLKSFYKNWEEHKNFQGETLLVLSDLDSTLKVKDLLIEGNDLEKLNYLLDLYIKASIYDKALSLARELPVAICLNKVGGGMFDDKNEKYKHCNEIVTSYLRLRYSGLMEFRNTLMHGGLSTDMKPNVDKDGNITPGKIVTKNKIEDFVKRELRNYFDKIVNFLSSA 6r7d A 2.35 BS01 JUQ A 1 N55 Y59 R90 Y93 R104 L108 A112 L115 W116 N60 Y64 R95 Y98 R109 L113 A117 L120 W121 2.5.1.-,4.4.1.20 0004364,0004464,0004602,0005515,0005634,0005635,0005640,0005783,0005789,0006629,0006691,0008047,0008289,0016020,0016740,0016829,0019370,0031965,0042759,0042802,0043231,0098869 ic50=2.4nM remove_due_to_license_issue IC50=50.0nM Q16873 31415176 201 HHHHHHKDEVALLAAVTLLGVLLQAYFSLQVISARRAFRVSPPLTTGPPEFERVYRAQVNCSEYFPLFLATLWVAGIFFHEGAAALCGLVYLFARLRYFQGYARSAQLRLAPLYASARALWLLVALAALGLLAHFLPAALRAALLGRLR 6r7d C 2.35 BS01 JUQ C 1 N55 Y59 R90 Y93 R104 L108 A112 L115 W116 N60 Y64 R95 Y98 R109 L113 A117 L120 W121 2.5.1.-,4.4.1.20 0004364,0004464,0004602,0005515,0005634,0005635,0005640,0005783,0005789,0006629,0006691,0008047,0008289,0016020,0016740,0016829,0019370,0031965,0042759,0042802,0043231,0098869 ic50=2.4nM remove_due_to_license_issue IC50=50.0nM Q16873 31415176 201 HHHHHHKDEVALLAAVTLLGVLLQAYFSLQVISARRAFRVSPPLTTGPPEFERVYRAQVNCSEYFPLFLATLWVAGIFFHEGAAALCGLVYLFARLRYFQGYARSAQLRLAPLYASARALWLLVALAALGLLAHFLPAALRAALLGRL 6r7j A 1.84 BS02 JUN A 1 Q286 L287 H323 R364 M365 R367 A368 F377 F378 E379 F388 Q29 L30 H66 R107 M108 R110 A111 F120 F121 E122 F131 ? 0003677,0004879,0005634,0006355 ic50=0.00000001M remove_due_to_license_issue IC50=32nM P51449 31223457 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 6r7k A 1.54 BS02 JUH A 1 Q286 L287 H323 L324 R364 M365 R367 A368 F377 F378 E379 G380 F388 I400 Q29 L30 H66 L67 R107 M108 R110 A111 F120 F121 E122 G123 F131 I143 ? 0003677,0004879,0005634,0006355 ic50=0.00000001M remove_due_to_license_issue IC50=50nM P51449 31223457 601 ENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG 6r7r A 2.8 BS01 DAS A 1 R278 S280 M314 T317 T355 G357 V358 G362 D398 R401 T402 N405 R263 S265 M299 T302 T340 G342 V343 G347 D383 R386 T387 N390 ? 0005886,0015293,0016020,0046942,0055085 remove_due_to_license_issue Q5JID0 30969168 504 YPVLWKILWGLVLGAVFGLIAGHFGYAGAVKTYIKPFGDLFVRLLKMLVMPIVLASLVVGAASISPARLGRVGVKIVVYYLATSAMAVFFGLIVGRLFNVGANVNLGSGTGAQPPSLVQTLLNIVPTNPFASLAKGEVLPVIFFAIILGIAITYLMNRNEERVRKSAETLLRVFDGLAEAMYLIVGGVMQYAPIGVFALIAYVMAEQGVRVVGPLAKVVGAVYTGLFLQIVITYFILLKVFGIDPIKFIRKAKDAMITAFVTRSSSGTLPVTMRVAEEEMGVDKGIFSFTLPLGATINMDGTALYQGVTVLFVANAIGHPLTLGQQLVVVLTAVLASIGTAGVPGAGAIMLAMVLQSVGLDLTPGSPVALAYAMILGIDAILDMGRTMVNVTGDLAGTVIVAKTEKELDESKWISH 6r8l A 1.64 BS01 JUZ A 1 R97 F102 M103 Q105 G114 G116 G117 S123 A143 N144 T149 Q153 F155 H168 R54 F59 M60 Q62 G71 G73 G74 S80 A100 N101 T106 Q110 F112 H125 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=0.006uM remove_due_to_license_issue P30405 31635932 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6r8o A 1.36 BS01 JV2 A 1 R97 F102 M103 Q105 S123 A143 N144 T149 Q153 F155 R54 F59 M60 Q62 S80 A100 N101 T106 Q110 F112 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=0.67uM remove_due_to_license_issue P30405 31635932 304 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6r8p A 1.45 BS01 JVB A 1 W128 F268 F319 F320 W41 F181 F232 F233 3.1.1.98 0016787 ic50=33uM remove_due_to_license_issue Q6P988 31534655 517 DLRLHLLLNTSVTCNDGSPAGYYLKESRGSRRWLLFLEGGWYCFNRENCDSRYDTMRRLMSSRDWPRTRTGTGILSSQPEENPYWWNANMVFIPYCSSDVWSGASSKSEKNEYAFMGALIIQEVVRELLGRGLSGAKVLLLAGSSAGGTGVLLNVDRVAEQLEKLGYPAIQVRGLADSGWFLDNKQYRHTDCVDTITCAPTEAIRRGIRYWNGVVPERCRRQFQEGEEWNCFFGYKVYPTLRSPVFVVQWLFDEAQLTVDNVHPVQEGLRLYIQNLGRELRHTLKDVPASFAPACLSHEIIIRSHWTDVQVKGTSLPRALHCWDRSLHTPLKGCPVHLVDSCPWPHCNPSCPT 6r8q A 1.5 BS01 JV5 A 1 W128 A233 T236 F268 P287 I291 F319 F320 A342 V346 W42 A147 T150 F182 P201 I205 F233 F234 A256 V260 3.1.1.98 0016787 ic50=0.12uM remove_due_to_license_issue Q6P988 31534655 515 EDLRLHLLLNTSVTCNDGSPAGYYLKESRGSRRWLLFLEGGWYCFNRENCDSRYDTMRRLMSSRDWPRTRTGTGILSSQPEENPYWWNANMVFIPYCSSDVWSGASSKSEKNEYAFMGALIIQEVVRELLGRGLSGAKVLLLAGSSAGGTGVLLNVDRVAEQLEKLGYPAIQVRGLADSGWFLDNKQYRHTDCVDTITCAPTEAIRRGIRYWNGVVPERCRRQFQEGEEWNCFFGYKVYPTLRSPVFVVQWLFDEAQLTVDNVHLTGQPVQEGLRLYIQNLGRELRHTLKDVPASFAPACLSHEIIIRSHWTDVQVKGTSLPRALHCWDRSLHDTPLKGCPVHLVDSCPWPHCNPSCPTG 6r8r A 1.27 BS01 JV8 A 1 W128 F268 P287 F320 T345 W43 F183 P202 F235 T260 3.1.1.98 0016787 ic50=0.085uM remove_due_to_license_issue IC50=85nM Q6P988 31534655 502 NEDLRLHLLLNTSVTCNDGSPAGYYLKESRGSRRWLLFLEGGWYCFNRENCDSRYDTMRRLMSSRDWPRTRTGTGILSSQPEENPYWWNANMVFIPYCSSDVWSGASSKSEKNEYAFMGALIIQEVVRELLGRGLSGAKVLLLAGSSAGGTGVLLNVDRVAEQLEKLGYPAIQVRGLADSGWFLDNKQYRHTDCVDTITCAPTEAIRRGIRYWNGVVPERCRRQFQEGEEWNCFFGYKVYPTLRSPVFVVQWLFDEAQLTVDNVHLTGQPVQEGLRLYIQNLGRELRHTLKDVPASFAPACLSHEIIIRSHWTDVQVKGTSLPRALHCWDRSLHDTPLKGCPVHLVDSCPWPHCNPSCPTGT 6r8w A 1.4 BS02 JVH A 1 R97 F102 Q105 G114 A143 N144 T149 Q153 F155 H168 R54 F59 Q62 G71 A100 N101 T106 Q110 F112 H125 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=1.2uM remove_due_to_license_issue P30405 31635932 303 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6r9s A 2.0 BS01 JVN A 1 G114 S123 R124 N144 T149 G151 Q153 G71 S80 R81 N101 T106 G108 Q110 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=7.1mM remove_due_to_license_issue P30405 31635932 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6r9s A 2.0 BS02 JVN A 2 T115 R124 A145 T72 R81 A102 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=7.1mM remove_due_to_license_issue P30405 31635932 302 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6r9u A 1.26 BS01 JVQ A 1 T115 G116 G117 S123 R124 A143 N144 T149 Q153 T72 G73 G74 S80 R81 A100 N101 T106 Q110 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=7.5mM remove_due_to_license_issue P30405 31635932 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6r9x A 1.66 BS01 JW2 A 1 R97 F102 M103 Q105 G114 A143 N144 Q153 F155 H168 R54 F59 M60 Q62 G71 A100 N101 Q110 F112 H125 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 Kd=1.1mM remove_due_to_license_issue P30405 31635932 301 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6ra1 A 2.0 BS02 JVQ A 1 T115 G116 G117 S123 R124 A143 N144 T149 Q153 T72 G73 G74 S80 R81 A100 N101 T106 Q110 R97 F102 Q105 N144 F155 L164 H168 R54 F59 Q62 N101 F112 L121 H125 5.2.1.8 0000413,0003755,0006457 remove_due_to_license_issue P30405 31635932 302 GNPLVYLDVDANGKPLGRVVLELKADVVPKTAENFRALCTGEKGFGYKGSTFHRVIPSFMCQAGDFTNHNGTGGKSIYGSRFPDENFTLKHVGPGVLSMANAGPNTNGSQFFICTIKTDWLDGKHVVFGHVIEGMDVVKKIESFGSKSGRTSKKIVITDCGQLS 6rfi A 2.31 BS01 K1H A 1 M192 G193 E194 V200 A211 K213 Y262 Y264 M265 D272 L277 L318 M24 G25 E26 V30 A41 K43 Y84 Y86 M87 D94 L99 L140 D311 K313 A315 N316 D329 T351 D133 K135 A137 N138 D151 T168 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=0.037uM remove_due_to_license_issue IC50=160nM Q9NWZ3 31622099 502 FHSFSFYELKNVTNNFDERPGNKMGEGGVVYKGYVNNTTVAVKKLEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6rfj A 2.61 BS01 K1E A 1 G193 A211 K213 Y262 Y264 M265 G268 D272 L277 L318 G24 A42 K44 Y79 Y81 M82 G85 D89 L94 L135 D311 K313 A315 N316 D329 T351 D128 K130 A132 N133 D146 T161 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 remove_due_to_license_issue IC50=4.0nM Q9NWZ3 31622099 501 FHSFSFYELKNVTNNFDERPNKMGEGGFGVVYKGYVNNTTVAVKKLEELKQQFDQEIKVMAKCQHENLVELLGFSCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 6rfn A 2.29 BS02 K3W A 1 M785 D822 N825 M861 G873 Q874 F877 M200 D237 N240 M276 G288 Q289 F292 3.1.4.- 0004114,0007165,0008081 Ki=0.00000079M remove_due_to_license_issue Ki=200nM Q8WQX9 31378593 1009 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLETR 6rfw A 2.183 BS02 K1Q A 1 M785 N825 M861 G873 Q874 G876 F877 M200 N240 M276 G288 Q289 G291 F292 3.1.4.- 0004114,0007165,0008081 Ki=0.00000079M remove_due_to_license_issue Ki=316nM Q8WQX9 31378593 1007 VTAITKVEREAVLVCELPSFDVTDVEFDLFRARESTDKPLDVAAAIAYRLLLGSGLPQKFGCSDEVLLNFILQCRKKYRNVPYHNFYHVVDVCQTIHTFLYRGNVYEKLTELECFVLLITALVHDLDHMGLNNSFYLKTESPLGILSSASGNTSVLEVHHCNLAVEILSDPESDVFDGLEGAERTLAFRSMIDCVLATDMAKHGSALEAFLASAADQSSDEAAFHRMTMEIILKAGDISNVTKPFDISRQWAMAVTEEFYRQGDMEKERGVEVLPMFDRSKNMELAKGQIGFIDFVAAPFFQKIVDACLQGMQWTVDRIKSNRAQWERVLET 6rih A 2.15 BS01 K4T A 1 G153 Y173 D174 P175 I176 I177 T206 P207 L215 G149 Y169 D170 P171 I172 I173 T202 P203 L211 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 Kd=105uM remove_due_to_license_issue Kd=105000nM O43175 31365252 401 LRKVLISDSLDPCCRKILQDGGLQVVEKQNLSKEELIAELQDCEGLIVRSATKVTADVINAAEKLQVVGRAGTGVDNVDLEAATRKGILVMNTPNGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQFVDMV 6rj2 A 2.0 BS01 K52 A 1 G153 I155 Y173 D174 P175 I176 I177 H205 T206 L215 R235 G146 I148 Y166 D167 P168 I169 I170 H198 T199 L208 R228 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 ic50=0.1uM remove_due_to_license_issue IC50=70nM O43175 31365252 402 VLISDSLDPCCRKILQDGGLQVVEKQNLSKEELIAELQDCEGLIVRSATKVTADVINAAEKLQVVGRAGTGVDNVDLEAATRKGILVMNTPNGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQFVDMV 6rj3 A 1.42 BS01 K58 A 1 L150 Y173 D174 P175 I176 I177 H205 T206 P207 L215 L145 Y168 D169 P170 I171 I172 H200 T201 P202 L210 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 ic50=0.4uM remove_due_to_license_issue IC50=900nM O43175 31365252 402 RKVLISDSLDPCCRKILQDGGLQVVEKQNLSKEELIAELQDCEGLIVRSATKVTADVINAAEKLQVVGRAGTGVDNVDLEAATRKGILVMNTPNGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQF 6rj5 A 1.89 BS01 K5N A 1 L150 Y173 D174 P175 I177 H205 T206 P207 L215 L146 Y169 D170 P171 I173 H201 T202 P203 L211 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 ic50=0.3uM remove_due_to_license_issue IC50=300nM O43175 31365252 402 LRKVLISDSLDPCCRKILQDGGLQVVEKQNLSKEELIAELQDCEGLIVRSATKVTADVINAAEKLQVVGRAGTGVDNVDLEAATRKGILVMNTPNGNSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQFVDM 6rj6 A 1.984 BS01 K5K A 1 G151 R154 I155 Y173 D174 P175 I176 I177 H205 T206 P207 T212 G52 R55 I56 Y74 D75 P76 I77 I78 H106 T107 P108 T113 1.1.1.37,1.1.1.399,1.1.1.95 0016616,0051287 ic50=2nM remove_due_to_license_issue IC50=3.0nM O43175 31365252 401 NGSLSAAELTCGMIMCLARQIPQATASMKDGKWERKKFMGTELNGKTLGILGLGRIGREVATRMQSFGMKTIGYDPIISPEVSASFGVQQLPLEEIWPLCDFITVHTPLLPSTTGLLNDNTFAQCKKGVRVVNCARGGIVDEGALLRALQSGQCAGAALDVFTEEPPRDRALVDHENVISCPHLGASTKEAQSRCGEEIAVQFV 6rk4 A 1.43 BS01 K5T A 1 N405 Y407 Y411 T429 P431 F432 M435 E451 M453 Y472 N5 Y7 Y11 T29 P31 F32 M35 E51 M53 Y72 3.4.24.75 Kd=890uM remove_due_to_license_issue P10547 31686030 501 GWKTNKYGTLYKSESASFTPNTDIITRTTGPFRSMPQSGVLKAGQTIHYDEVMKQDGHVWVGYTGNSGQRIYLPVRTWNKSTNTLGVLWGTIK 6rln A 2.87 BS01 K8K A 1 V31 M44 K45 V76 L90 M92 H136 A155 D156 L157 S161 F162 V14 M27 K28 V59 L73 M75 H119 A138 D139 L140 S144 F145 D138 K140 E142 N143 D156 T189 D121 K123 E125 N126 D139 T161 2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue Q13546 31223438 301 NVIKMKSSDFLEKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE 6rmf A 1.51 BS04 K9B A 1 W93 H122 D124 H189 C208 K211 G219 N220 H250 W57 H86 D88 H153 C172 K175 G183 N184 H214 H120 H122 D124 H189 C208 K211 N220 H250 H84 H86 D88 H153 C172 K175 N184 H214 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 remove_due_to_license_issue C7C422 31454231 307 PTIGQQMETGDQRFGDLVFRQLAPNVWQHTSYLDGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR 6rn6 E 2.4 BS01 K9Q E 1 G232 C234 E275 G276 G277 F278 G27 C29 E70 G71 G72 F73 Q228 C234 Q23 C29 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 HLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6rn6 F 2.4 BS01 K9Q E 1 T379 N380 H381 T8 N9 H10 H381 N403 H10 N31 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 PFNPFELTNHAVLLVGYGTDSAGMDYWIVKNSWGTGWGENGYFRIRRGTDECAIESIAVAATPIPKL 6rn7 A 1.66 BS01 K9W B 1 D1 P3 D1 P3 3.4.14.1 remove_due_to_license_issue P53634 31413809 401 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKV 6rn7 B 1.66 BS01 K9W B 1 G232 C234 E275 G276 G277 F278 G27 C29 E70 G71 G72 F73 Q228 C234 Q23 C29 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 HLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6rn7 C 1.66 BS01 K9W B 1 N380 H381 A382 N9 H10 A11 H381 N403 H10 N32 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 PFNPFELTNHAVLLVGYGTDSASGMDYWIVKNSWGTGWGENGYFRIRRGTDECAIESIAVAATPIPKL 6rn9 A 1.9 BS01 K9Z B 1 D1 P3 D1 P3 3.4.14.1 remove_due_to_license_issue P53634 31413809 401 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKV 6rn9 B 1.9 BS01 K9Z B 1 G232 C234 E275 G276 G277 F278 G26 C28 E69 G70 G71 F72 Q228 C234 Q22 C28 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 LPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6rn9 C 1.9 BS01 K9Z B 1 N380 H381 A382 N9 H10 A11 H381 N403 H10 N32 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 PFNPFELTNHAVLLVGYGTDSASGMDYWIVKNSWGTGWGENGYFRIRRGTDECAIESIAVAATPIPKL 6rna A 2.62 BS01 KA2 A 1 L24 S25 V32 A45 K47 E66 L79 T95 Y97 M98 G101 E105 L153 D164 L20 S21 V27 A40 K42 E55 L68 T84 Y86 M87 G90 E94 L142 D153 D146 Q150 N151 D164 D135 Q139 N140 D153 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=0.002000nM O43353 31265286 401 AICSALPTIPYHKLADLRYLSRGSGTVSSARHADWRVQVAVKHLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSKWRMGGTIIYMPPENYSIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 6rne B 1.65 BS01 KA8 B 1 G232 C234 E275 G276 G277 F278 G26 C28 E69 G70 G71 F72 Q228 C234 Q22 C28 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 LPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6rne C 1.65 BS01 KA8 B 1 N380 H381 N9 H10 H381 N403 H10 N32 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 401 PFNPFELTNHAVLLVGYGTDSASGMDYWIVKNSWGTGWGENGYFRIRRGTDECAIESIAVAATPIPKL 6rni A 1.54 BS01 KAQ B 1 D1 P3 D1 P3 3.4.14.1 remove_due_to_license_issue P53634 31413809 402 DTPANCTYLDLLGTWVFQVGSSGSQRDVNCSVMGPQEKKVVVYLQKLDTAYDDLGNSGHFTIIYNQGFEIVLNDYKWFAFFKYKEEGSKVTTYCNETMTGWVHDVLGRNWACFTGKKV 6rni B 1.54 BS01 KAQ B 1 G232 C234 E275 G276 G277 F278 A349 G28 C30 E71 G72 G73 F74 A145 Q228 C234 Q24 C30 3.4.14.1 0006508,0008234 remove_due_to_license_issue P53634 31413809 402 LHLPTSWDWRNVHGINFVSPVRNQASCGSCYSFASMGMLEARIRILTNNSQTPILSPQEVVSCSQYAQGCEGGFPYLIAGKYAQDFGLVEEACFPYTGTDSPCKMKEDCFRYYSSEYHYVGGFYGGCNEALMKLELVHHGPMAVAFEVYDDFLHYKKGIYHHT 6rnt A 1.8 BS01 2AM A 1 N36 Y38 H40 E58 G74 R77 H92 N36 Y38 H40 E58 G74 R77 H92 Y38 H40 E58 D76 R77 T91 H92 F100 Y38 H40 E58 D76 R77 T91 H92 F100 4.6.1.24 0001411,0003723,0004519,0004521,0004540,0008150,0016829,0030428,0046589 Kd=4.3mM remove_due_to_license_issue P00651 1651320 105 ACDYTCGSNCYSSSDVSTAQAAGYKLHEDGETVGSNSYPHKYNNYEGFDFSVSSPYYEWPILSSGDVYSGGSPGADRVVFNENNQLAGVITHTGASGNNFVECT 6rnu A 2.4 BS01 KBH A 2 F97 A104 F105 L130 R132 D133 R139 F43 A50 F51 L76 R78 D79 R85 ? 0042981 remove_due_to_license_issue EC50=>31500nM, IC50=>99200nM Q07817 31606346 302 SQSNRELVVDFLSYKLSQKGYSWSQFSESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 6rnu B 2.4 BS01 KBH A 1 F97 A104 F105 L130 R132 D133 R139 F43 A50 F51 L76 R78 D79 R85 ? 0042981 remove_due_to_license_issue EC50=>31500nM, IC50=>99200nM Q07817 31606346 301 SQSNRELVVDFLSYKLSQKGYSWSQFSESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 6rnu B 2.4 BS02 KBH A 2 R100 Y101 R46 Y47 ? 0042981 remove_due_to_license_issue EC50=>31500nM, IC50=>99200nM Q07817 31606346 302 SQSNRELVVDFLSYKLSQKGYSWSQFSESEAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAYQSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEPWIQENGGWDTFVELYG 6rot H 1.339 BS03 KDQ H 1 H57 Y60A W60D E97A A190 S195 V213 S214 W215 G216 E217 F227 H43 Y47 W50 E94 A192 S197 V217 S218 W219 G220 E221 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 Ki=483.63nM remove_due_to_license_issue Ki=484nM P00734 31633354 301 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG 6rpg A 2.7 BS01 KDW B 1 Y56 Q66 M115 I116 S117 A121 D122 Y123 Y39 Q49 M98 I99 S100 A104 D105 Y106 ? remove_due_to_license_issue IC50=3.0nM, EC50=763nM Q9NZQ7 31298541 201 AFTVTVPKDLYVVEYGSNMTIECKFPVEKQLDLAALIVYWEMEDKNIIQFVHGEEDLKVQHSSYRQRARLLKDQLSLGNAALQITDVKLQDAGVYRCMISYGGADYKRITVKVNAPY 6rpg B 2.7 BS01 KDW B 1 Y56 Q66 M115 I116 S117 A121 D122 Y123 Y39 Q49 M98 I99 S100 A104 D105 Y106 ? remove_due_to_license_issue IC50=3.0nM, EC50=763nM Q9NZQ7 31298541 201 AFTVTVPKDLYVVEYGSNMTIECKFPVEKQLDLAALIVYWEMEDKNIIQFVHGEEDLKVQHSSYRQRARLLKDQLSLGNAALQITDVKLQDAGVYRCMISYGGADYKRITVKVNAPY 6rqk A 1.85 BS01 MVL A 1 T55 I58 W62 R64 D65 S219 D220 N302 H350 W357 E393 R405 T54 I57 W61 R63 D64 S218 D219 N301 H349 W356 E392 R404 ? 0005975,0046872 Kd=1.6mM remove_due_to_license_issue Q8XNB2 31407758 501 SLSTNELKEIVRKIGKDLSGKIEDKKLQELFYNCFINTMDTTVEVSEGDAFVITGDIPAMWLRDSTSQVEHYLPFVKEYPELKAIFTGLINRQVKCIFIDPYANAFNKEPNGQKWDNDITKDSPWVWERKYEIDSLCYPVRLIHKYWKESGDETFFNDDIKKAFNMIIDLWRVEQYHREKSDYSFQRLNCSVTDTLSHEGLGTPVTYTGMTWSGFRPSDDACEYGYLIPANMFAVVALRYISEIAEKVYKDEELKEKADSLREEIDNAIEKHGKVYKEGFGEVYAYETDGMGNYNFMDDANVPSLLSIPYLEYKGIEDEVYQNTRKFILSKNNRFFFEGKAAKGIGSPHTPDQYIWHIALSMQGLTTNNQEEIDQLIKLLKETDAGTGYMHEGFHVDDPTKFTRDWFAWSNSLFSHFIYEKVINK 6rqk A 1.85 BS02 MVL A 2 W116 E129 K131 D195 D220 H350 W115 E128 K130 D194 D219 H349 ? 0005975,0046872 Kd=1.6mM remove_due_to_license_issue Q8XNB2 31407758 502 SLSTNELKEIVRKIGKDLSGKIEDKKLQELFYNCFINTMDTTVEVSEGDAFVITGDIPAMWLRDSTSQVEHYLPFVKEYPELKAIFTGLINRQVKCIFIDPYANAFNKEPNGQKWDNDITKDSPWVWERKYEIDSLCYPVRLIHKYWKESGDETFFNDDIKKAFNMIIDLWRVEQYHREKSDYSFQRLNCSVTDTLSHEGLGTPVTYTGMTWSGFRPSDDACEYGYLIPANMFAVVALRYISEIAEKVYKDEELKEKADSLREEIDNAIEKHGKVYKEGFGEVYAYETDGMGNYNFMDDANVPSLLSIPYLEYKGIEDEVYQNTRKFILSKNNRFFFEGKAAKGIGSPHTPDQYIWHIALSMQGLTTNNQEEIDQLIKLLKETDAGTGYMHEGFHVDDPTKFTRDWFAWSNSLFSHFIYEKVINK 6rrm A 1.64 BS01 9JT A 1 M303 N316 Y318 V322 H336 H352 C354 M247 N260 Y262 V266 H280 H296 C298 2.3.2.- 0005886,0008360,0009252,0016740,0016746,0018104,0046872,0071555,0071972 remove_due_to_license_issue I6Y9J2 31380528 504 LLVPKLTASVTDGAVGVTVDAPVSVTAADGVLAAVTMVNDNGRPVAGRLSPDGLRWSTTEQLGYNRRYTLNATALGLGGAATRQLTFQTSSPAHLTMPYVMPGDGEVVGVGEPVAIRFDENIADRGAAEKAIKITTNPPVEGAFYWLNNREVRWRPEHFWKPGTAVDVAVNTYGVDLGEGMFGEDNVQTHFTIGDEVIATADDNTKILTVRVNGEVVKSMPTSMGKDSTPTANGIYIVGSRYKHIIMDSSTYGVPVNSPNGYRTDVDWATQISYSGVFVHSAPWSVGAQGHTNTSHGCLNVSPSNAQWFYDHVKRGDIVEVVNTVGGTLPGIDGLGDWNIPWDQWRAGNAK 6rsa A 2.0 BS01 UVC A 1 Q11 H12 K41 V43 N44 T45 H119 F120 Q11 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0004519,0004522,0004540,0005515,0005576,0016829,0050830 remove_due_to_license_issue P61823 4016100 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 6rt6 B 1.461 BS01 rna E 0 K361 S362 N363 N367 W377 S378 R404 W428 L439 G474 D476 K18 S19 N20 N24 W34 S35 R61 W81 L92 G127 D129 ? 0003723 remove_due_to_license_issue Q96MU7 31670957 1 ~ 2 GTSKLKYVLQDARFFLIKSNNHENVSLAKAKGVWSTLPVNEKKLNLAFRSARSVILIFSVRESGKFQGFARLSSESHHIHWVLPAGMSAKMLGGVFKIDWICRRELPFTKSAHLTNPWNEHKPVKIGRDGQEIELECGTQLCLLFPPDESIDLYQVIHKM 6rt6 C 1.461 BS01 rna A 0 K361 S362 N363 N367 W377 S378 W428 L439 D476 K18 S19 N20 N24 W34 S35 W85 L96 D133 ? 0003723 remove_due_to_license_issue Q96MU7 31670957 1 ~ 2 GTSKLKYVLQDARFFLIKSNNHENVSLAKAKGVWSTLPVNEKKLNLAFRSARSVILIFSVRESGKFQGFARLSSESHHGGSPIHWVLPAGMSAKMLGGVFKIDWICRRELPFTKSAHLTNPWNEHKPVKIGRDGQEIELECGTQLCLLFPPDESIDLYQVIHKM 6rt7 B 1.73 BS01 rna E 0 K361 S362 N363 N367 W377 S378 R404 E405 W428 P431 M434 K472 I473 G474 R475 D476 K18 S19 N20 N24 W34 S35 R61 E62 W81 P84 M87 K125 I126 G127 R128 D129 ? 0003723 remove_due_to_license_issue Q96MU7 31670957 1 ~ 3 GTSKLKYVLQDARFFLIKSNNHENVSLAKAKGVWSTLPVNEKKLNLAFRSARSVILIFSVRESGKFQGFARLSSESHHIHWVLPAGMSAKMLGGVFKIDWICRRELPFTKSAHLTNPWNEHKPVKIGRDGQEIELECGTQLCLLFPPDESIDLYQVIHKM 6rt7 C 1.73 BS01 rna A 0 K361 S362 N363 N367 W377 S378 W428 R475 D476 K18 S19 N20 N24 W34 S35 W85 R132 D133 ? 0003723 remove_due_to_license_issue Q96MU7 31670957 1 ~ 2 GTSKLKYVLQDARFFLIKSNNHENVSLAKAKGVWSTLPVNEKKLNLAFRSARSVILIFSVRESGKFQGFARLSSESHHGGSPIHWVLPAGMSAKMLGGVFKIDWICRRELPFTKSAHLTNPWNEHKPVKIGRDGQEIELECGTQLCLLFPPDESIDLYQVIHKM 6rtn A 2.17 BS01 KJK A 1 S67 K70 S115 V117 T206 G207 F208 R250 S48 K51 S96 V98 T187 G188 F189 R231 S67 K70 S115 F120 W154 F208 S48 K51 S96 F101 W135 F189 3.5.2.6 0005886,0008658,0008800,0016787,0017001,0042597,0046677,0071555 remove_due_to_license_issue P14489 31454231 506 GSITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNDLARASKEYLPASTFKIPNAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLTLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLYLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKETEVYFFAFNMDIDNESKLPLRKSIPTKIMESEGII 6rtw A 1.9 BS01 Y01 A 1 Y215 L223 Y224 L248 W278 L282 A285 Y67 L75 Y76 L100 W130 L134 A137 ? remove_due_to_license_issue Q13635 31548691 504 EEAMFNPQLMIQTPKEEGANVLTTEALLQHLDSALQASRVHVYMYNRQWKLEHLCYKSGELITETGYMDQIIEYLYPCLIITPLDCFWEGAKLQSGTAYLLGKPPLRWTNFDPLEFLEELKKINYQVDSWEEMLNKAEVGHGYMDRPCLNPADPDCPATAPNKNSTKPLDMALVLNGGCHGLSRKYMHWQEELIVGGTVKNSTGKLVSAHALQTMFQLMTPKQMYEHFKGYEYVSHINWNEDKAAAILEAWQRTYVEVVHQSVAQNSTQKVLSFTGT 6rvf A 2.07 BS02 KKH A 1 H94 V121 F131 L198 T199 P202 H91 V118 F127 L194 T195 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=730nM remove_due_to_license_issue P00918 31423863 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6rvk A 1.58 BS02 R29 A 1 H94 H96 H119 F131 V135 L198 T199 P202 H91 H93 H116 F127 V131 L194 T195 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=439nM remove_due_to_license_issue P00918 31423863 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6rvl A 1.72 BS02 KKE A 1 Q92 H94 H96 H119 V121 F131 L198 T199 T200 P202 Q89 H91 H93 H116 V118 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1148nM remove_due_to_license_issue P00918 31423863 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6rw1 A 1.7 BS02 KL5 A 1 Q92 H94 H96 H119 V121 F131 L198 T199 T200 P202 Q89 H91 H93 H116 V118 F127 L194 T195 T196 P198 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=1305nM remove_due_to_license_issue P00918 31423863 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASF 6rz6 A 2.43 BS01 KNW A 1 K37 Y119 Y123 S170 M201 N202 R267 L271 H284 K9 Y91 Y95 S139 M168 N169 R310 L314 H327 ? 0004930,0004974,0005506,0007186,0009055,0016020,0020037,0022900,0042597,0046872 remove_due_to_license_issue P0ABE7,Q9NS75 31811124 2001 RNCTIENFKREFFPIVYLIIFFVGVLGNGLSIYVFLQPYKKSTSVNVFMLNLAISNLLFISTLPFRADYYLRGSNWIFGDLACRIMSYSLYVNMYSSIYFLTVLSVVRYLAMVHPFRVTSIRSAWILCGIIWILIMASSIMLLDSEQNGSVTSCLELNLYKIAKLQTMNYIALVVGCLLPFFTLSICYLLIIRVLLKVEADLEDNWETLNDNLKVIEKAAAQVKDALTKMRAAALDAQMKDFRHGFDILVGQIDDALKLVKEAQAAAEQLKTTRNAYIQKYLVSHRKALTTIIITLIIFFLCFLPYHTLRTVHLTTWKVGLCKDRLHKALVITLALAAANACFNPLLYYFAGENFKDRLKSALRK 6s0e A 1.9 BS01 DAN A 1 N15 S16 C53 W95 R129 H134 R202 N346 Q351 T352 N10 S11 C48 W90 R124 H129 R197 N341 Q346 T347 remove_due_to_license_issue 31645552 609 IPGISLNEDNSHYFYTRAGRRLSAEEVDSWVDQYAGTQVKELMLCPNCMRTSYASQVWDPIWRGYDPAGPDDQPLLASLPPEERVAARGWIHTAWQLHQDGIDIYARWIRRCRQRGISPWISMRMNDVHYVNDERCFLHSEFWRENPQLRRVPYRFAEWTDRAFDYGRAEVREHHLKLIRELAARYDFDGLELDWMRFGFHFRPGYEAEGAEILTAFTAEVRRLLDDWEKRRGHKIHLGARIPSRPATALGLGMDAVTWARRGLVDMLVITPFWASAETDMPVEIWRQLLEGTGVTLAAGLEVLLRPYPDSPLFQTNSLETVRGAAASLLDRGAQRIYLFNYMDSQTAMEDLENYPTLLREIGSLETLAGKPRRHVLTFADTWAPGEPRAIPLPATCRPGEWRAFRLHTGPKPEPGEVIAALGIEGGAIGPETLEVRVNGELCAFLGLVDLSKPRPDFPVYGFSVPLAAMRRGYNLIEVTARQELRFGWAEFLIRP 6s1s A 1.78 BS01 KRT A 1 S64 Q120 Y151 Y223 S319 T320 S62 Q118 Y149 Y221 S317 T318 S64 K67 Y151 E273 K316 S319 S62 K65 Y149 E271 K314 S317 3.5.2.6 0008800,0017001,0030288 remove_due_to_license_issue Q541D8 31574990 401 APADRLKALVDAAVQPVMKANDIPGLAVAISLKGEPHYFSYGLASKEDGRRVTPETLFEIGSVSKTFTATLAGYALTQDKMRLDDRASQHWPALQGSRFDGISLLDLATYTAGGLPLQFPDSVQKDQAQIRDYYRQWQPTYAPGSQRLYSNPSIGLFGYLAARSLGQPFERLMEQQVFPALGLEQTHLDVPEAALAQYAQGYGKDDRPLRVGPGPLDAEGYGVKTSAADLLRFVDANLHPERLDRPWAQALDATHRGYYKVGDMTQGLGWEAYDWPISLKRLQAGNSTPMALQPHRIARLPAPQALEGQRLLNKTGSTNGFGAYVAFVPGRDLGLVILANRNYPNAERVKIAYAILSGLEQQGKVPL 6s43 A 1.42 BS01 KUE A 1 L303 T304 L429 R432 L294 T295 L412 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=4uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s43 A 1.42 BS02 KUE C 1 A307 H397 R400 L401 R432 A298 H380 R383 L384 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=4uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s43 C 1.42 BS01 KUE A 1 A307 H397 R400 L401 R432 A298 H379 R382 L383 R414 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=4uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s43 C 1.42 BS02 KUE C 1 L303 T304 L429 R432 L294 T295 L411 R414 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=4uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s4n D 1.9 BS01 KUW D 1 F271 T272 L274 A275 I309 M312 L313 T316 R319 F329 L330 L345 H435 L442 W457 F47 T48 L50 A51 I85 M88 L89 T92 R95 F105 L106 L121 H211 L218 W233 ? 0003677,0004879,0006629 Kd=1.6uM remove_due_to_license_issue P55055 31799433 501 QLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s4n D 1.9 BS02 KUW D 2 L226 Q229 L8 Q11 ? 0003677,0004879,0006629 Kd=1.6uM remove_due_to_license_issue P55055 31799433 502 QLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s4n D 1.9 BS03 KUW D 3 V279 V283 K287 Q300 L304 E455 I456 V55 V59 K63 Q76 L80 E231 I232 ? 0003677,0004879,0006629 Kd=1.6uM remove_due_to_license_issue P55055 31799433 503 QLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s4t A 2.0 BS01 KVB A 1 F271 L274 S278 T316 R319 F329 L330 F340 I353 H435 L449 W457 F50 L53 S57 T95 R98 F108 L109 F119 I132 H214 L228 W236 ? 0003677,0004879,0006629 Ki=0.00000079M remove_due_to_license_issue EC50=90nM, IC50=2000nM P55055 31799433 501 QLTAAQELMIQQLVAAQLQCNKRSFSKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s4t A 2.0 BS02 KVB A 2 V279 V283 K287 Q300 I301 L304 K305 T308 V58 V62 K66 Q79 I80 L83 K84 T87 ? 0003677,0004879,0006629 Ki=0.00000079M remove_due_to_license_issue EC50=90nM, IC50=2000nM P55055 31799433 502 QLTAAQELMIQQLVAAQLQCNKRSFSKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s4u A 2.81 BS01 KVK A 1 F271 L274 A275 S278 M312 E315 T316 R319 F329 L330 H435 F48 L51 A52 S55 M89 E92 T93 R96 F106 L107 H212 ? 0003677,0004879,0006629 remove_due_to_license_issue P55055 31799433 501 QLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s55 A 2.09 BS01 KW5 A 1 V1008 F1009 K1011 V1013 D1014 E1017 V1018 Y1021 I1056 A1060 I1074 V30 F31 K33 V35 D36 E39 V40 Y43 I78 A82 I96 3.6.1.- remove_due_to_license_issue IC50=631nM Q6PL18 31398032 1205 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 6s56 A 2.01 BS01 KVZ A 1 V1008 K1011 P1012 V1013 D1014 E1017 Y1021 I1056 A1060 V30 K33 P34 V35 D36 E39 Y43 I78 A82 3.6.1.- remove_due_to_license_issue IC50=5012nM, Kd=7943nM Q6PL18 31398032 1205 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 6s57 A 1.82 BS01 KVT A 1 V1008 F1009 K1011 V1013 D1014 Y1021 Y1063 I1074 V30 F31 K33 V35 D36 Y43 Y85 I96 3.6.1.- remove_due_to_license_issue IC50=10000nM, Kd=7943nM Q6PL18 31398032 1202 SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEVPDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICSNALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFEQLCEEIQESR 6s5k A 1.6 BS01 KWE A 1 F243 F268 F271 T272 A275 L313 R319 F329 L345 I353 H435 L442 W457 F25 F32 F35 T36 A39 L77 R83 F93 L109 I117 H199 L206 W221 ? 0003677,0004879,0006629 Ki=0.00000079M remove_due_to_license_issue P55055 31799433 501 QLTAAQELMIQQLVAAQLQCNKRSFSARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWDV 6s7k A 1.55 BS01 KYZ A 1 L303 L429 R432 L294 L412 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=57uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7k A 1.55 BS02 KYZ C 1 A307 H397 R400 L401 A298 H380 R383 L384 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=57uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7k C 1.55 BS01 KYZ A 1 A307 H397 R400 R432 A298 H380 R383 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=57uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7k C 1.55 BS02 KYZ C 1 L303 T304 L429 R432 L294 T295 L412 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=57uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLQKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7s A 1.7 BS01 KZ8 A 1 L303 T304 L429 R432 L294 T295 L412 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=17uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7s A 1.7 BS02 KZ8 C 1 A307 N394 H397 R400 L401 R432 A298 N377 H380 R383 L384 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=17uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7s C 1.7 BS01 KZ8 A 1 A307 N394 H397 R400 L401 R432 A298 N378 H381 R384 L385 R416 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=17uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLPGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7s C 1.7 BS02 KZ8 C 1 L303 T304 L429 R432 L294 T295 L413 R416 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=17uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLPGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7z A 1.85 BS01 KZN A 1 L303 T304 L429 R432 L294 T295 L411 R414 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=2.2uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7z A 1.85 BS02 KZN C 1 A307 N394 H397 R400 L401 R432 A298 N376 H379 R382 L383 R414 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=2.2uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7z C 1.85 BS01 KZN A 1 A307 N394 H397 R400 R432 A298 N376 H379 R382 R414 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=2.2uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s7z C 1.85 BS02 KZN C 1 L303 T304 L429 R432 L294 T295 L411 R414 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=2.2uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s88 A 1.59 BS01 L0K A 1 L303 L429 R432 L294 L412 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=0.67uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s88 A 1.59 BS02 L0K C 1 A307 H397 L401 R432 A298 H380 L384 R415 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=0.67uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s88 C 1.59 BS01 L0K A 1 A307 H397 R400 R432 A298 H381 R384 R416 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=0.67uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLPGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s88 C 1.59 BS02 L0K C 1 L303 T304 L429 R432 L294 T295 L413 R416 4.2.1.2 0003824,0004333,0005576,0005737,0005829,0005886,0006099,0006106,0009274,0016829 ic50=0.67uM remove_due_to_license_issue P9WN93 31517489 501 YRIEHDTMGEVRVPAKALWRAQTQRAVENFPISGRGLERTQIRALGLLKGACAQVNSDLGLLAPEKADAIIAAAAEIADGQHDDQFPIDVFQTGSGTSSNMNTNEVIASIAAKGGVTLHPNDDVNMSQSSNDTFPTATHIAATEAAVAHLIPALQQLHDALAAKALDWHTVVKSGRTHLMDAVPVTLGQEFSGYARQIEAGIERVRACLPRLGELAIGGTAVGTGLNAPDDFGVRVVAVLVAQTGLSELRTAANSFEAQAARDGLVEASGALRTIAVSLTKIANDIRWMGSGPLTGLAEIQLPDLPGKVNPVLPEAVTQVAAQVIGNDAAIAWGGANGAFELNVYIPMMARNILESFKLLTNVSRLFAQRCIAGLTANVEHLRRLAESSPSIVTPLNSAIGYEEAAAVAKQALKERKTIRQTVIDRGLIGDRLSIEDLDRRLDVLAMAKAE 6s89 A 2.701 BS01 L0Q A 1 L718 G719 V726 A743 Q791 M793 P794 G796 L844 L22 G23 V30 A47 Q95 M97 P98 G100 L148 D837 R841 N842 D855 D141 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 31857889 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGSLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAAAAEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDEFYRALMDEEDMDDVVDADEYL 6s8a A 2.6 BS01 L0N A 1 L718 V726 A743 M790 Q791 M793 G796 L844 L22 V30 A47 M94 Q95 M97 G100 L148 D837 R841 N842 D855 D141 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 31857889 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGSLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAAAAEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDESNFYRALMDEEDMDDVVDADEYLI 6s90 A 1.82 BS01 L0Z A 1 L408 Q412 F413 V416 A428 K430 Y476 M477 A478 N479 G480 L528 D539 Y551 L14 Q18 F19 V22 A34 K36 Y82 M83 A84 N85 G86 L134 D145 Y157 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 ic50=13nM remove_due_to_license_issue IC50=13nM Q06187 31620235 701 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVMD 6s9b A 3.25 BS01 L1H A 1 L718 A743 K745 E762 M790 Q791 M793 P794 G796 L844 T854 L22 A47 K49 E63 M91 Q92 M94 P95 G97 L145 T155 D837 R841 N842 D855 D138 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 31689114 1101 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKEATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPDDVVDADEYLIP 6s9c A 2.73 BS01 L1K A 1 L718 F723 A743 M790 Q791 M793 P794 G796 L844 T854 D855 L25 F30 A50 M95 Q96 M98 P99 G101 L149 T159 D160 D837 R841 N842 D855 D142 R146 N147 D160 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 31689114 1101 SMGEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPEEDMDDVVDADEYLIP 6s9d A 2.67 BS01 L3Z A 1 L718 F723 A743 M790 M793 P794 G796 L844 T854 D855 L25 F30 A50 M95 M98 P99 G101 L149 T159 D160 D837 R841 N842 D855 D142 R146 N147 D160 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue P00533 31689114 1101 SMGEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRTSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLLGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDDMDDVVDADEYL 6s9w A 2.3 BS01 L1Z A 1 E17 W80 I84 L210 Y272 R273 D274 D292 C296 C310 E15 W78 I82 L179 Y241 R242 D243 D261 C265 C277 D274 K276 N279 D292 T312 D243 K245 N248 D261 T279 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue P31749 31584233 501 DVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDVDQREAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKKKHRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTA 6s9x A 2.6 BS01 L1W A 1 Q79 W80 I84 L210 L264 V270 Y272 R273 D292 C296 C310 Q73 W74 I78 L156 L210 V216 Y218 R219 D238 C242 C249 D274 K276 N279 D292 T312 D220 K222 N225 D238 T251 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004676,0004677,0004679,0004694,0004711,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035175,0035402,0035403,0035556,0035655,0035924,0035979,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043161,0043276,0043325,0043488,0043491,0043536,0044022,0044023,0044024,0044025,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072354,0072371,0072518,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0140823,0140855,0140857,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1903898,1904263,1905552,1990090,1990244,1990418,2000010,2000074,2000117,2000402,2001240,2001243 remove_due_to_license_issue P31749 31584233 501 DVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDEAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFT 6saf A 2.05 BS01 L2Q A 1 Y57 D68 F77 G84 Q85 V86 I87 W90 Y113 K121 F130 Y45 D56 F65 G72 Q73 V74 I75 W78 Y101 K109 F118 Y57 F67 D68 I87 Y113 F130 Y45 F55 D56 I75 Y101 F118 5.2.1.8 0003755 Ki=0.23uM remove_due_to_license_issue Ki=230nM Q13451 31800244 201 GAPATVTEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 6sal A 1.61 BS01 L3E A 1 L324 T325 I328 Q329 L353 K354 M358 L483 Q484 A496 A497 F498 Y502 L505 F506 L59 T60 I63 Q64 L88 K89 M93 L218 Q219 A231 A232 F233 Y237 L240 F241 ? 0003677,0004879,0005634,0006355 ic50=0.264uM remove_due_to_license_issue P51449 31821760 601 SLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLHKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFS 6sbt A 2.3 BS01 L5H A 1 E13 Y61 P88 L89 T90 R95 D139 Y216 E10 Y58 P85 L86 T87 R92 D136 Y213 ? 0015276,0016020 Ki=43nM remove_due_to_license_issue P22756 31622082 303 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWR 6sde A 2.49 BS01 V0L A 1 I1084 V1092 A1108 Y1159 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I17 V25 A36 Y81 M82 D86 R130 M133 A143 D144 Y152 D1204 R1208 N1209 D1222 D126 R130 N131 D144 2.7.10.1 0004672,0004713,0005524,0006468 remove_due_to_license_issue IC50=2.0nM P08581 31531204 1401 HVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRIEVSQFLTEGIIMKDFSHPNVLSLLGICLRSSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG 6sfc B 2.0 BS01 L9T B 1 F97 Y148 N194 L240 Y365 R367 F17 Y68 N114 L160 Y278 R280 ? Kd=5.2uM remove_due_to_license_issue O75530 31525019 501 SFKCVNSLKEDHNQPLFGVQFNWHSKEGDPLVFATVGSNRVTLYECHSQGEIRLLQSYVDADADENFYTCAWTYDSNTSHPLLAVAGSRGIIRIINPITMQCIKHYVGHGNAINELKFHPRDPNLLLSVSKDHALRLWNIQTDTLVAIFGGVEGHRDEVLSADYDLLGEKIMSCGMDHSLKLWRINSKRMMNAIKESYDRPFISQKIHFPDFSTRDIHRNYVDCVRWLGDLILSKSCENAIVCWKPGKMEDDIDKIKPSESNVTILGRFDYSQCDIWYMRFSMDFWQKMLALGNQVGKLYVWDLECTTLTHHKCGAAIRQTSFSRDSSILIAVCDDASIWRWDR 6sfi A 1.6 BS01 LB5 A 1 Y35 A51 K53 E71 T106 M109 A111 D168 F169 Y32 A48 K50 E68 T103 M106 A108 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T172 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=26nM Q16539 31702918 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 6sfj A 1.95 BS01 LBB A 1 Y35 K53 E71 L75 T106 M109 L167 D168 Y32 K50 E68 L72 T103 M106 L164 D165 D150 K152 N155 D168 T185 D147 K149 N152 D165 T173 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=18nM Q16539 31702918 401 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 6sfk A 1.8 BS01 LB8 A 1 A51 K53 E71 T106 M109 A111 H148 L167 D168 F169 A48 K50 E68 T103 M106 A108 H145 L164 D165 F166 D150 K152 N155 D168 T185 D147 K149 N152 D165 T171 2.7.11.24 0000077,0000165,0000902,0000922,0001502,0001525,0001649,0001890,0002021,0002062,0002862,0004672,0004674,0004705,0004707,0004708,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005829,0006006,0006355,0006357,0006366,0006468,0006915,0006935,0006974,0007165,0007166,0007178,0007254,0007519,0010628,0010831,0016301,0016607,0018105,0019395,0019899,0019903,0030168,0030278,0030316,0031098,0031281,0031663,0032495,0032496,0032735,0032868,0033554,0034774,0035331,0035556,0035924,0035994,0038066,0042307,0042770,0043536,0045648,0045663,0045944,0046323,0046326,0048010,0048273,0048863,0051146,0051149,0051403,0051525,0060045,0060348,0070935,0071222,0071223,0071356,0071479,0071493,0090090,0090336,0090398,0090400,0098586,0098978,0099179,0106310,1900015,1901741,1904813,2000379 remove_due_to_license_issue IC50=71nM Q16539 31702918 405 ERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQSIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPL 6sge A 1.5 BS01 GTP A 1 A15 G17 K18 T19 C20 F30 Y34 P36 T37 G62 K118 D120 L121 A161 K162 A13 G15 K16 T17 C18 F28 Y32 P34 T35 G60 K116 D118 L119 A159 K160 ? 0000281,0001525,0003924,0005515,0005525,0005634,0005768,0005769,0005770,0005829,0005886,0005925,0006886,0006915,0007015,0007155,0007165,0007264,0007266,0008333,0010008,0010595,0015031,0016020,0019003,0030154,0030334,0030336,0031902,0032154,0043065,0045766,0045786,0061154,0070062,0070301,0071479,0098685,0099159 remove_due_to_license_issue P62745 31522999 201 AIRKKLVVVGDGACGKTCLLIVFSKDEFPEVYVPTVFENYVADIEVDGKQVELALWDTAGLEDYDRLRPLSYPDTDVILMCFSVDSPDSLENIPEKWVPEVKHFCPNVPIILVANKKDLRSDEHVRTELARMKQEPVRTDDGRAMAVRIQAYDYLECSAKTKEGVREVFETATRAALQ 6skb A 1.84 BS01 LH5 A 1 L41 C42 H57 D189 S190 C191 Q192 G193 S195 V213 G216 D217 Y218 C220 L25 C26 H41 D170 S171 C172 Q173 G174 S176 V190 G193 D194 Y195 C197 H57 L63 V65 A97 D102 Q192 G193 D194 S195 H41 L47 V49 A80 D85 Q173 G174 D175 S176 3.4.21.- 0004252,0006508 remove_due_to_license_issue Q92876 31521475 301 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGDYPCGSKERPGVYTNVCRYTNWIQKTIQAK 6skc A 2.18 BS01 LH8 A 1 H57 D189 S190 C191 Q192 G193 S195 V213 W215 G216 H41 D170 S171 C172 Q173 G174 S176 V190 W192 G193 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 remove_due_to_license_issue Q92876 31521475 301 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNYPCGSKEKPGVYTNVCRYTNWIQKTIQA 6skd A 2.26 BS01 LH2 A 1 L41 C42 H57 D189 S190 Q192 G193 S195 V213 W215 G216 N217 L25 C26 H41 D170 S171 Q173 G174 S176 V190 W192 G193 N194 H57 D102 Q192 G193 D194 S195 H41 D85 Q173 G174 D175 S176 3.4.21.- 0001533,0004252,0005515,0005576,0005615,0005634,0005654,0005730,0005737,0005739,0005783,0006508,0007417,0008233,0008236,0009611,0010975,0016540,0016787,0030141,0030574,0031965,0042246,0042445,0042552,0042982,0045171,0045595,0045745,0051604 remove_due_to_license_issue Q92876 31521475 302 LVHGGPCDKTSHPYQAALYTSGHLLCGGVLIHPLWVLTAAHCKKPNLQVFLGKHNLGQQESSQEQSSVVRAVIHPDYDAASHDQDIMLLRLARPAKLSELIQPLPLERDCSAQTTSCHILGWGKTADGDFPDTIQCAYIHLVSREECEHAYPGQITQNMLCAGDEKYGKDSCQGDSGGPLVCGDHLRGLVSWGNYPCGSKEKPGVYTNVCRYTNWIQKTIQA 6slg A 1.33 BS02 LHZ A 1 E33 G34 Y36 G37 V39 A52 K54 Q105 M108 E109 T110 K114 L156 D167 E16 G17 Y19 G20 V22 A35 K37 Q88 M91 E92 T93 K97 L139 D150 D149 K151 N154 D167 T190 D132 K134 N137 D150 T173 2.7.11.24 0000165,0001784,0003677,0004672,0004674,0004705,0004707,0005515,0005524,0005576,0005634,0005654,0005737,0005739,0005769,0005770,0005788,0005794,0005813,0005819,0005829,0005856,0005886,0005901,0005925,0006357,0006468,0006915,0006935,0006974,0007165,0007166,0007254,0007268,0007507,0007611,0008286,0008353,0009887,0010759,0010800,0014032,0014044,0016020,0016301,0018105,0018107,0019858,0019902,0030278,0030521,0030641,0030878,0031143,0031647,0031663,0032206,0032496,0032872,0033554,0033598,0034198,0035094,0035556,0035578,0038127,0038133,0042473,0042552,0042802,0043330,0043401,0045202,0045542,0045596,0048009,0048538,0050847,0050852,0050853,0051403,0051493,0060020,0060291,0060324,0060425,0060440,0060716,0061308,0070161,0070371,0070849,0071356,0072584,0072686,0090170,0106310,0120041,1904813,2000641 Kd=0.000000064M remove_due_to_license_issue Kd=0.100000nM, IC50=0.660000nM P28482 31710489 401 VFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKLPKEKLKELIFEETARFQP 6so9 A -1.00 BS01 rna B 0 H523 C525 N526 I551 L552 M553 K554 S555 Q558 F560 L589 R591 S593 T594 R595 Y596 L599 Q600 L601 K602 K603 H14 C16 N17 I42 L43 M44 K45 S46 Q49 F51 L80 R82 S84 T85 R86 Y87 L90 Q91 L92 K93 K94 ? 0003676,0003723 remove_due_to_license_issue Q3UQS8 32187365 1 ~ 6 GAMAQRKGAGRVVHICNLPEGSCTENDVINLGLPFGKVTNYILMKSTNQAFLEMAYTEAAQAMVQYYQEKPAIINGEKLLIRMSTRYKELQLKKPGKNVAAIIQDIHSQRER 6sq0 A 1.77 BS01 LRQ A 1 L346 L384 F404 G521 H524 L525 L36 L74 F94 G204 H207 L208 ? ic50=0.00000001M remove_due_to_license_issue IC50=16nM P03372 31620239 601 GSHMALSLTADQMVSALLDAEPPILYSEEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMPSYDLLLEMLDAHRLHAP 6ssy A 1.62 BS01 P7I A 1 Q30 G61 G79 P82 S131 T132 W176 D205 Q9 G40 G58 P61 S110 T111 W155 D184 ? 0022857,0042597,0043190,0055085 remove_due_to_license_issue Q47537 31802112 401 MVNVTVAYQTSAEPAKVAQADNTFAKESGATVDWRKFDSGASIVRALASGDVQIGNLGSSPLAVAASQQVPIEVFLLASKLGNSEALVVKKTISKPEDLIGKRIAVPFISTTHYSLLAALKHWGIKPGQVEIVNLQPPAIIAAWQRGDIDGAYVWAPAVNALEKDGKVLTDSEQVGQWGAPTLDVWVVRKDFAEKHPEVVKAFAKSAIDAQQPYIANPDVWLKQPENISKLARLSGVPEGDVPGLVKGNTYLTPQQQTAELTGPVNKAIIDTAQFLKEQGKVPAVANDYSQYVTSRFV 6st0 A 1.5 BS01 LUQ A 1 Q30 S32 G61 G79 P82 E106 S131 T132 W176 D205 Q9 S11 G40 G58 P61 E85 S110 T111 W155 D184 ? 0022857,0042597,0043190,0055085 remove_due_to_license_issue Q47537 31802112 405 MVNVTVAYQTSAEPAKVAQADNTFAKESGATVDWRKFDSGASIVRALASGDVQIGNLGSSPLAVAASQQVPIEVFLLASKLGNSEALVVKKTISKPEDLIGKRIAVPFISTTHYSLLAALKHWGIKPGQVEIVNLQPPAIIAAWQRGDIDGAYVWAPAVNALEKDGKVLTDSEQVGQWGAPTLDVWVVRKDFAEKHPEVVKAFAKSAIDAQQPYIANPDVWLKQPENISKLARLSGVPEGDVPGLVKGNTYLTPQQQTAELTGPVNKAIIDTAQFLKEQGKVPAVANDYSQYVTSRFV 6st3 A 2.426 BS01 LUW A 1 R252 T296 Y303 Y310 H313 D315 R322 H374 V376 W389 F391 R57 T101 Y108 Y115 H118 D120 R127 H179 V181 W194 F196 1.14.11.29 0005506,0016705,0031418 ic50=0.256uM remove_due_to_license_issue Q9GZT9 31751494 601 PALKLALEYIVPCMNKHGICVVDDFLGKETGQQIGDEVRALHDTGKFTDGQLVSQIRGDKITWIEGKEPGCETIGLLMSSMDDLIRHCNGKLGSYKINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVTCIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYAITVWYFDADERARAKVKYLT 6std A 1.8 BS02 MS2 A 1 W26 Y50 F53 V75 L76 V108 N131 F162 G165 W18 Y42 F45 V67 L68 V100 N123 F154 G157 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=2.3nM remove_due_to_license_issue P56221 10382670 601 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFGDK 6suo A 1.74 BS01 LVH A 1 L346 T347 L349 E353 L384 R394 F404 G521 L525 L37 T38 L40 E44 L75 R85 F95 G203 L207 ? ic50=0.00000001M remove_due_to_license_issue IC50=1.3nM P03372 31620239 601 GSHMALSLTADQMVSALLDAEPPILYSEYEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMPSYDLLLEMLDAHRLHAP 6sy7 A 2.75 BS01 AMP A 1 A288 Q289 A290 R312 I450 A269 Q270 A271 R293 I418 G107 R173 G174 D199 G200 K226 T227 D229 D231 R274 G88 R154 G155 D180 G181 K207 T208 D210 D212 R255 2.7.1.11 0003872,0005524,0005737,0006002,0006096,0016301,0020015,0042301,0046872,0061615 remove_due_to_license_issue O15648 31838765 503 MLNSVTQEDLKVDRLPGADYPNPSKKYSSRTEFRDKTDYIMYNPRPRDEPSSENPVSVSPLLCELAAARSRIHFNPTETTIGIVTCGGICPGLNDVIRSITLTGINVYNVKRVIGFRFGYWGLSKKGSQTAIELHRGRVTNIHHYGGTILGSSRGPQDPKEMVDTLERLGVNILFTVGGDGTQRGALVISQEAKRRGVDISVFGVPKTIDNDLSFSHRTFGFQTAVEKAVQAIRAAYAEAVSANYGVGVVKLMGRDSGFIAAQAAVASAQANICLVPENPISEQEVMSLLERRFCHSRSCVIIVAEGFGQDWGLIDIGVILTEKVKAFLKANKSRYPDSTVKYIDPSYMIRACPPSANDALFCATLATLAVHEAMAGATGCIIAMRHNNYILVPIKVATSVRRVLDLRGQLWRQVREITVDLGSDVRLARKLEIRRELEAINRNRDRLHEELAKL 6sy7 A 2.75 BS02 AMP B 1 R117 S118 L121 R155 R98 S99 L102 R136 G107 R173 G174 D199 G200 K226 T227 D229 D231 R274 G88 R154 G155 D180 G181 K207 T208 D210 D212 R255 2.7.1.11 0003872,0005524,0005737,0006002,0006096,0016301,0020015,0042301,0046872,0061615 remove_due_to_license_issue O15648 31838765 1001 MLNSVTQEDLKVDRLPGADYPNPSKKYSSRTEFRDKTDYIMYNPRPRDEPSSENPVSVSPLLCELAAARSRIHFNPTETTIGIVTCGGICPGLNDVIRSITLTGINVYNVKRVIGFRFGYWGLSKKGSQTAIELHRGRVTNIHHYGGTILGSSRGPQDPKEMVDTLERLGVNILFTVGGDGTQRGALVISQEAKRRGVDISVFGVPKTIDNDLSFSHRTFGFQTAVEKAVQAIRAAYAEAVSANYGVGVVKLMGRDSGFIAAQAAVASAQANICLVPENPISEQEVMSLLERRFCHSRSCVIIVAEGFGQDWGLIDIGVILTEKVKAFLKANKSRYPDSTVKYIDPSYMIRACPPSANDALFCATLATLAVHEAMAGATGCIIAMRHNNYILVPIKVATSVRRVLDLRGQLWRQVREITVDLGSDVRLARKLEIRRELEAINRNRDRLHEELAKL 6sze A 2.94 BS01 M2B A 1 V32 A45 K47 E66 L79 T95 Y97 M98 L153 V28 A41 K43 E57 L70 T86 Y88 M89 L144 D146 Q150 N151 D164 D137 Q141 N142 D155 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43353 31749904 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLSTIIYMPPENYESIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 6szj A 2.53 BS01 M5W A 1 V32 A45 V46 K47 L79 I93 T95 Y97 M98 L153 V28 A41 V42 K43 L72 I86 T88 Y90 M91 L146 D146 Q150 N151 D164 D139 Q143 N144 D157 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue O43353 31749904 401 AICSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLTPLLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLGTIIYMPPENYEPGQSIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 6szp A 1.76 BS01 M3B A 1 L30 D73 F76 D79 H173 V268 D269 C274 L23 D66 F69 D72 H166 V261 D262 C267 3.5.3.18 0000052,0003073,0003824,0005829,0006525,0006527,0007263,0008285,0016403,0016597,0016787,0043116,0045429,0045766,0046209,0046872,0070062,1900038 Ki=18uM remove_due_to_license_issue O94760 31841335 300 AAFGRATHAVVRALPESLGQHALRSAKGEEVDVARAERQHQLYVGVLGSKLGLQVVELPADESLPDCVFVEDVAVVCEETALITRPGAPSRRKEVDMMKEALEKLQLNIVEMKDENATLDGGDVLFTGREFFVGLSKRTNQRGAEILADTFKDYAVSTVPVADGLHLKSFCSMAGPNLIAIGSSESAQKALKIMQQMSDHRYDKLTVPDDIAANCIYLNIPNKGHVLLHRTPEEYPESAKVYEKLKDHMLIPVSMSELEKVDGLLTCCSVLINKK 6t1i A 1.8 BS01 M7W A 1 F28 H56 S58 F59 P60 G77 Y78 A79 F27 H55 S57 F58 P59 G76 Y77 A78 ? remove_due_to_license_issue Q03111 31857843 201 DNQCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6t1j A 1.97 BS01 M7T A 1 F28 H56 S58 F59 P60 G77 Y78 F27 H55 S57 F58 P59 G76 Y77 ? remove_due_to_license_issue Q03111 31857843 208 DNQCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6t1l A 2.0 BS01 M7N A 1 F28 H56 S58 F59 P60 G77 Y78 A79 G80 F26 H54 S56 F57 P58 G75 Y76 A77 G78 ? remove_due_to_license_issue Q03111 31857843 211 NQCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6t1m A 1.85 BS01 M8K A 1 F28 H56 S58 F59 P60 E75 S76 G77 Y78 A79 F81 F26 H54 S56 F57 P58 E73 S74 G75 Y76 A77 F79 ? remove_due_to_license_issue Q03111 31857843 201 NQCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6t1n A 1.95 BS01 M7Z A 1 F28 H56 S58 F59 P60 E75 S76 G77 Y78 A79 F81 F25 H53 S55 F56 P57 E72 S73 G74 Y75 A76 F78 ? remove_due_to_license_issue Q03111 31857843 201 QCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6t1o A 1.9 BS01 M82 A 1 F28 H56 S58 F59 P60 E75 S76 G77 Y78 A79 F81 F25 H53 S55 F56 P57 E72 S73 G74 Y75 A76 F78 ? remove_due_to_license_issue Q03111 31857843 201 QCTVQVRLELGHRAQLRKKPTTEGFTHDWMVFVRGPEQCDIQHFVEKVVFWLHDSFPKPRRVCKEPPYKVEESGYAGFIMPIEVHFKNKEEPRKVCFTYDLFLNLEGNPPVNHLRCEKLTFNNPTTEFRYKLLRAGGVMVM 6t6a A 2.8 BS01 MLW A 1 F170 A186 F36 A52 D287 K289 N292 D307 S324 D153 K155 N158 D173 S190 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 remove_due_to_license_issue Q13627 31766108 507 VYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKDGKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFFKK 6te6 A 1.98 BS01 N4W A 1 P130 F131 S140 L143 M147 V169 F239 N241 F243 S268 S269 V310 S311 Y312 P120 F121 S130 L133 M137 V159 F229 N231 F233 S258 S259 V297 S298 Y299 2.1.1.360 0031151,0051726 ic50=0.27uM remove_due_to_license_issue IC50=270nM Q8TEK3 31857842 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKNP 6tel A 2.19 BS01 N4Z A 1 P130 F131 S140 L143 V169 F239 V240 N241 F243 V267 S268 S269 V310 S311 Y312 P113 F114 S123 L126 V152 F222 V223 N224 F226 V250 S251 S252 V290 S291 Y292 2.1.1.360 0031151,0051726 ic50=0.00011uM remove_due_to_license_issue IC50=0.110000nM Q8TEK3 31857842 401 LELRLKSPVGAEPAVYPWPLPVYHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKNP 6ten A 2.21 BS01 N5K A 1 P130 F131 S140 L143 V169 F239 V240 N241 F243 V267 S268 S269 V310 S311 Y312 P119 F120 S129 L132 V158 F228 V229 N230 F232 V256 S257 S258 V296 S297 Y298 2.1.1.360 0031151,0051726 ic50=0.00017uM remove_due_to_license_issue IC50=0.170000nM Q8TEK3 31857842 401 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKSWTGKPVSYYLHTIDRTILENYFSSLKNP 6tim B 2.2 BS01 G3P B 1 N11 K13 H95 E167 I172 G173 S213 L232 G234 N10 K12 H94 E166 I171 G172 S212 L231 G233 N11 K13 H95 E97 E167 G173 S213 N10 K12 H94 E96 E166 G172 S212 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0020015,0046166 Ki=0.61mM remove_due_to_license_issue P04789 2062828 300 SKPQPIAAANWKCNGSQQSLSELIDLFNSTSINHDVQCVVASTFVHLAMTKERLSHPKFVIAAQNAIAKSGAFTGEVSLPILKDFGVNWIVLGHSERRAYYGETNEIVADKVAAAVASGFMVIACIGETLQERESGRTAVVVLTQIAAIAKKLKKADWAKVVIAYEPVWAIGTGKVATPQQAQEAHALIRSWVSSKIGADVAGELRILYGGSVNGKNARTLYQQRDVNGFLVGGASLKPEFVDIIKATQ 6tl2 A 3.8 BS01 NJZ A 1 D51 N54 A231 L410 S459 D39 N42 A219 L398 S447 ? 0005384,0005886,0006811,0006828,0012505,0015086,0015293,0016020,0030001,0034755,0046872,0046873,0070574,0071421 remove_due_to_license_issue E4KPW4 31804182 601 DLSLSDINSTVEVPEGHSFWKTLLAYSGPGALVAVGYMDPGNWSTSITGGQNFQYLLLSIIVISSLLAMLLQNMAAKLGIVCQLDLAQAIRARTSRRLGFIFWILTELAIMATDIAEVIGAAIALYLLFKIPIFLAVVITVLDVFLLLLLNRIGFRKIEALVVCLIFVILFVFLYQIILSQPAWHQVAKGLIPSWASVQTSPKIGGQTPLSASLGIIGATIMPHNLFLHSAISQSRKIDRTDSSKVAEAVRFSNWDSNIQLSLAMVVNALLLIMGVAVFKSGAVQDPSFFGLYQALSNPDMVSNPVLAEAARSGVLSTLFAVALLASGQNSTITGTITGQVIMEGFIHLRLPLWLRRLVTRLIAIIPVVVCVAITSHQGSLDEHQALNNLMNNSQVFLALALPFSIVPLLMLTDSAAQMGNQFKNTRWVKVMGWLTVIILTLLNLISISSQIAGFFGDNPSSQDLLLSQVISIGIILAMIGLLIWTIIDIRRFT 6tld A 1.61 BS02 NK5 A 1 D100 H142 G150 D186 H188 F216 Y341 D99 H141 G149 D176 H178 F206 Y314 3.5.1.98 0004407,0005634,0006325,0031507,0046872 Kd=4.4uM remove_due_to_license_issue A5H660 31816172 504 SVGIVYGDQYRQLCCSSPKFGDRYALVMDLINAYKLIPELSRVPPLQWDSPSRMYEAVTAFHSTEYVDALKKLQMLHCEEKELTADDELLMDSFSLNYDCPGFPSVFDYSLAAVQGSLAAASALICRHCEVVINWGGGWHHAKRSEASGFCYLNDIVLAIHRLVSSQTRVLYVDLDLHHGDGVEEAFWYSPRVVTFSVHHASPGFFPGTGTWNKLPIFLNGAGRGRFSAFNLPLEEGINDLDWSNAIGPILDSLNIVIQPSYVVVQCGADCLATDPHRIFRLTNFYPSLSGYLYAIKKILSWKVPTLILGGGGYNFPDTARLWTRVTALTIEEVKGKKMTISPEIPEHSYFSRYGPDFELDIDYFPDSIQKHHRRILEQLRNYADLNKLIYDYDQVYQLY 6u5m A 1.8 BS01 Q0S A 1 S223 P224 N225 Y228 L240 K250 F266 K272 W273 L288 Q289 S191 P192 N193 Y196 L208 K218 F234 K240 W241 L256 Q257 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=0.511uM remove_due_to_license_issue Kd=511nM P61964 31724864 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u5y A 1.532 BS01 Q0M A 1 S223 P224 N225 Y228 L240 K250 F266 S267 K272 W273 L288 Q289 S193 P194 N195 Y198 L210 K220 F236 S237 K242 W243 L258 Q259 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=0.069uM remove_due_to_license_issue Kd=69nM P61964 31724864 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u6w A 1.2 BS01 Q0Y A 1 S223 P224 N225 Y228 K250 F266 K272 W273 L288 S198 P199 N200 Y203 K225 F241 K247 W248 L263 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=4.71uM remove_due_to_license_issue Kd=4710nM P61964 31724864 401 TQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u7o A 1.33 BS01 Q1D B 1 D25 A28 D30 G48 P81 V82 D25 A28 D30 G48 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q5RZ08 31549492 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6u7o B 1.33 BS01 Q1D B 1 D25 G27 D29 D30 I47 G48 G49 I50 D25 G27 D29 D30 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 Ki=15.5uM remove_due_to_license_issue Q5RZ08 31549492 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6u7p A 1.13 BS01 B4R A 1 D25 A28 D30 I47 G48 P81 V82 D25 A28 D30 I47 G48 P81 V82 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q5RZ08 31549492 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6u7p B 1.13 BS01 B4R A 1 D25 G27 D29 D30 G48 G49 I50 D25 G27 D29 D30 G48 G49 I50 D25 T26 G27 D25 T26 G27 ? 0004190,0006508 remove_due_to_license_issue Q5RZ08 31549492 201 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 6u7t A 2.0 BS01 dna B 0 Q48 R50 G85 L86 G87 Y88 Y89 G260 L261 L262 H305 F307 S308 H309 P345 V346 Q42 R44 G79 L80 G81 Y82 Y83 G254 L255 L256 H294 F296 S297 H298 P334 V335 E43 Y126 D144 E37 Y120 D138 3.2.2.31 0000701,0003677,0003824,0006281,0006284,0006298,0006950,0016798,0019104,0032357,0034039,0035485,0046872,0051539 remove_due_to_license_issue P83847 31829624 1 ~ 11 RFPAREFQRDLLDWFARERRDLPWRKDRDPYKVWVSEVMLQQTRVETVIPYFEQFIDRFPTLEALADADEDEVLKAWEGLGYYSRVRNLHAAVKEVKTRYGGKVPDDPDEFSRLKGVGPYTVGAVLSLAYGVPEPAVDGNVMRVLSRLFLVTDDIAKPSTRKRFEQIVREIMAYENPGAFNEALIELGALVCTPRRPSCLLCPVQAYCQAFAEGVAEELPVKMKKTAVKQVPLAVAVLADDEGRVLIRKRDSTGLLANLWEFPSCETDGADGKEKLEQMVGEQELTEPIVSFEHAFSHLVWQLTVFPGRLVHGGPVEEPYRLAPEDELKAYAFPVSHQRVWREYKEWAS 6u7t A 2.0 BS02 dna C 0 L46 Q47 Q48 R50 V51 G122 G124 P125 Y126 T127 D144 G145 R149 L40 Q41 Q42 R44 V45 G116 G118 P119 Y120 T121 D138 G139 R143 E43 Y126 D144 E37 Y120 D138 3.2.2.31 0000701,0003677,0003824,0006281,0006284,0006298,0006950,0016798,0019104,0032357,0034039,0035485,0046872,0051539 remove_due_to_license_issue P83847 31829624 13 ~ 22 RFPAREFQRDLLDWFARERRDLPWRKDRDPYKVWVSEVMLQQTRVETVIPYFEQFIDRFPTLEALADADEDEVLKAWEGLGYYSRVRNLHAAVKEVKTRYGGKVPDDPDEFSRLKGVGPYTVGAVLSLAYGVPEPAVDGNVMRVLSRLFLVTDDIAKPSTRKRFEQIVREIMAYENPGAFNEALIELGALVCTPRRPSCLLCPVQAYCQAFAEGVAEELPVKMKKTAVKQVPLAVAVLADDEGRVLIRKRDSTGLLANLWEFPSCETDGADGKEKLEQMVGEQELTEPIVSFEHAFSHLVWQLTVFPGRLVHGGPVEEPYRLAPEDELKAYAFPVSHQRVWREYKEWAS 6u80 A 1.55 BS01 Q1J A 1 P224 N225 Y228 F266 K272 W273 L288 P199 N200 Y203 F241 K247 W248 L263 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=37uM remove_due_to_license_issue Kd=37000nM P61964 31724864 401 TQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u8b A 1.261 BS01 Q1M A 1 S223 P224 N225 Y228 K250 F266 K272 W273 L288 Q289 S197 P198 N199 Y202 K224 F240 K246 W247 L262 Q263 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=0.431uM remove_due_to_license_issue Kd=431nM P61964 31724864 401 TQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLINPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u8d H 1.807 BS01 rna A 0 Y58 Y60 T61 R104 S105 Y106 Y107 R109 Y55 Y57 T58 R101 S102 Y103 Y104 R106 remove_due_to_license_issue 31765566 143 ~ 248 EVQLVESGGGLVQPGGSLRLSCAASGFYISSYSIHWVRQAPGKGLEWVASIYPSYGYTSYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRYRSYYSRYGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSC 6u8d L 1.807 BS01 rna A 0 Y94 Y95 Y94 Y95 remove_due_to_license_issue 31765566 143 ~ 248 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQSSYYPSTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 6u8k D 2.75 BS01 rna B 0 Y31 Y34 S35 S36 S55 S57 S58 S60 Y62 S102 R103 Y104 S105 R106 R108 R109 Y28 Y31 S32 S33 S52 S54 S55 S57 Y59 S99 R100 Y101 S102 R103 R105 R106 remove_due_to_license_issue 31765566 143 ~ 248 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPSSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARSRYSRYRRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6u8k E 2.75 BS01 rna B 0 Y92 S93 Y97 Y92 S93 Y97 remove_due_to_license_issue 31765566 143 ~ 248 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYSSSPYTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 6u8k F 2.75 BS01 rna B 0 R22 Q85 R19 Q82 remove_due_to_license_issue 31765566 143 ~ 248 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPSSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARSRYSRYRRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6u8k F 2.75 BS02 rna C 0 Y34 S35 S36 S55 S57 S58 S60 Y62 S102 R103 Y104 S105 R106 R109 Y31 S32 S33 S52 S54 S55 S57 Y59 S99 R100 Y101 S102 R103 R106 remove_due_to_license_issue 31765566 143 ~ 248 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPSSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARSRYSRYRRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6u8k G 2.75 BS01 rna C 0 Y92 S93 Y97 Y92 S93 Y97 remove_due_to_license_issue 31765566 143 ~ 248 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYSSSPYTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 6u8k H 2.75 BS01 rna A 0 Y34 S35 S36 S55 S57 S58 S60 Y62 S102 R103 Y104 S105 R106 R109 Y31 S32 S33 S52 S54 S55 S57 Y59 S99 R100 Y101 S102 R103 R106 remove_due_to_license_issue 31765566 143 ~ 248 EVQLVESGGGLVQPGGSLRLSCAASGFYISYSSIHWVRQAPGKGLEWVASISPSSGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARSRYSRYRRGFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPK 6u8k L 2.75 BS01 rna A 0 Y50 Y92 S93 Y97 Y50 Y92 S93 Y97 remove_due_to_license_issue 31765566 143 ~ 248 SDIQMTQSPSSLSASVGDRVTITCRASQSVSSAVAWYQQKPGKAPKLLIYSASSLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQYSSSPYTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC 6u8l A 1.57 BS01 Q1P A 1 S223 P224 N225 Y228 L240 F266 K272 W273 L288 Q289 S193 P194 N195 Y198 L210 F236 K242 W243 L258 Q259 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 remove_due_to_license_issue Kd=122nM P61964 31724864 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u8o A 1.6 BS01 Q1G A 1 S223 P224 N225 Y228 F266 K272 W273 L288 Q289 S193 P194 N195 Y198 F236 K242 W243 L258 Q259 ? 0000122,0000123,0001501,0005515,0005634,0005654,0006094,0006325,0006355,0006357,0035064,0035097,0042393,0042800,0044545,0044665,0044666,0045722,0045815,0045893,0045995,0048188,0051302,0051726,0071339,0072686,0090043,0140672 Kd=0.289uM remove_due_to_license_issue Kd=289nM P61964 31724864 401 VKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC 6u9v A 2.9 BS02 GDP A 1 R546 H547 Y550 A567 L569 R574 K583 S589 R511 H512 Y515 A532 L534 R539 K548 S554 ? 0000165,0000287,0000902,0001530,0001614,0001845,0001913,0001916,0002028,0004931,0005102,0005216,0005507,0005515,0005524,0005635,0005737,0005739,0005886,0005911,0006509,0006649,0006811,0006812,0006816,0006884,0006900,0006954,0007005,0007009,0007166,0008270,0009306,0009410,0009612,0009617,0009897,0010043,0010467,0010524,0010628,0012501,0014047,0014049,0014051,0014054,0014070,0015267,0016020,0016079,0016485,0017121,0019228,0019233,0030163,0030501,0031594,0032059,0032060,0032308,0032310,0032496,0032730,0032731,0032755,0032963,0032991,0033198,0034220,0034405,0034767,0035590,0038023,0042098,0042802,0043025,0043029,0043065,0043132,0043195,0043409,0043410,0043539,0045202,0045332,0045778,0045779,0045794,0045821,0046513,0046931,0048705,0048873,0050714,0050830,0051209,0051495,0051592,0051602,0051649,0051882,0051899,0051901,0060079,0060907,0070227,0070230,0070231,0070234,0070588,0071359,0071407,0072593,0097110,0097190,0097191,0098655,0098794,0099161,1900227,1904172,1904669 remove_due_to_license_issue Q64663 31587896 701 CCSWNDVFQYETNKVTRIQSVNYGTIKWILHMTVFSYVSFALMSDKLYQRKEPLISSVHTKVKGVAEVTENVTKLVHGIFDTADYTLPLQGNSFFVMTNYLKSEGQEQKLCPEYPSRGKQCHSDQGCIKGWMDPQSKGIQTGRCIPYDQKRKTCEIFAWCPAEEGKEAPRPALLRSAENFTVLIKNNIDFPGHNYTTRNILPGMNISCTFHKTWNPQCPIFRLGDIFQEIGENFTEVAVQGGIMGIEIYWDCNLDSWSHRCQPKYSFRRLDDKYTNESLFPGYNFRYAKYYKENGMEKRTLIKAFGVRFDILVFGTGGKFDIIQLVVYIGSTLSYFGLATVCIDLIINTYASTCCRSRVYPSCKCCEPCAVNEYYYRKKCEPIVEPKPTLKYVSFVDEPHIWMVDQQLLGKSLQDVKGQEVPRPQTDFLELSRLSRDSPDWCQCGNCLPSQLPENRRALEELCCRRKPGQCITTSELFSKIVLSREALQLLLLYQEPLLALEGEAINSKLRHCAYRSYATWRFVSQDMADFAILPSCCRWKIRKEFPKTQGQYSGFKYPY 6u9x A 2.6 BS01 rna K 0 S112 M115 Y197 R199 R219 N221 R222 I229 I232 S233 L234 K235 Q276 W283 R284 V285 V287 Y289 I326 Q352 L355 R356 Y360 R364 S38 M41 Y111 R113 R133 N135 R136 I143 I146 S147 L148 K149 Q190 W197 R198 V199 V201 Y203 I240 Q266 L269 R270 Y274 R278 ? remove_due_to_license_issue B6SBM0 31704716 30 ~ 33 VHLQQSTIQLEKLSHPPARFDSFVYKWQTKAALARKVSGPMREWAAELKYRTGVHIELEPTYPERLSENAQWGAYETADDVDITVYLFGSERGIFNCHKLMEAAIQQDPVYVRLGIFRRLANSSEVEWLMLRRINRELRPPDIPPISLKLPGKWTLLYERYKEAAIRTLWEETGITVDASNVYPTGHLYQTVPQYYWRVPVRYFVAEVPSDIRVEGPQVVPLQYMRNWDARLLRQSPDPIDRAWAQLADPATGCAWMKASMIDQLQKPLRGDNYMAIRYTPPPYSNLQEVVGLG 6u9x D 2.6 BS01 rna H 0 S112 M115 R116 Y197 R199 R219 N221 R222 L224 P226 I229 I232 S233 L234 K235 L274 Y275 Q276 W283 V285 V287 Y289 I326 Q352 L355 R356 Y360 R364 S37 M40 R41 Y111 R113 R133 N135 R136 L138 P140 I143 I146 S147 L148 K149 L188 Y189 Q190 W197 V199 V201 Y203 I240 Q266 L269 R270 Y274 R278 ? remove_due_to_license_issue B6SBM0 31704716 30 ~ 33 VHLSTIQLEKLSHPPARFDNSFVYKWQTKAALARKVSGPMREWAAELKYRTGVHIELEPTYPERLSENAVQWGAYETADDVDITVYLFGSERGIFNCHKLMEAAIQQDPVYVRLGIFRRLANSSEVEWLMLRRINRELRPPDIPPISLKLPGKWTLLYERYKEAAIRTLWEETGITVDASNVYPTGHLYQTVPQYYWRVPVRYFVAEVPSDIRVEGPQVVPLQYMRNWDARLLRQSPDPIDRAWAQLADPATGCAWMKASMIDQLQKPLRGDNYMAIRYTPPPYSNLQEVVGLG 6ud2 A 1.7 BS01 Q4D A 1 H224 A227 F228 G230 M231 V249 M250 V253 R263 T266 L267 F270 G271 I294 H53 A56 F57 G59 M60 V78 M79 V82 R92 T95 L96 F99 G100 I123 ? 0042981 ic50=0.3nM remove_due_to_license_issue IC50=0.300000nM, Ki=0.060000nM Q07820 31736296 401 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6udi A 1.94 BS01 Q4S A 1 H224 A227 F228 V249 M250 V253 R263 T266 L267 F270 I294 H53 A56 F57 V78 M79 V82 R92 T95 L96 F99 I123 ? 0042981 ic50=0.3nM remove_due_to_license_issue IC50=0.300000nM, Ki=0.100000nM Q07820 31736296 401 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6udt A 1.5 BS01 Q4V A 1 H224 A227 V249 M250 V253 R263 T266 L267 F270 I294 H53 A56 V78 M79 V82 R92 T95 L96 F99 I123 ? 0042981 ic50=0.6nM remove_due_to_license_issue IC50=0.600000nM, Ki=0.100000nM Q07820 31736296 401 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6udu A 1.75 BS01 Q4Y A 1 H224 A227 V249 M250 V253 R263 T266 L267 F270 I294 H54 A57 V79 M80 V83 R93 T96 L97 F100 I124 ? 0042981 ic50=1.7nM remove_due_to_license_issue IC50=1.7nM, Ki=0.500000nM Q07820 31736296 401 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6udv A 1.35 BS01 Q51 A 1 H224 A227 V249 M250 V253 R263 T266 L267 F270 H53 A56 V78 M79 V82 R92 T95 L96 F99 ? 0042981 Ki=0.051nM remove_due_to_license_issue Ki=0.051000nM Q07820 31736296 401 DELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEG 6udx A 1.7 BS01 Q57 A 1 F228 V249 M250 V253 R263 T266 L267 F270 F58 V79 M80 V83 R93 T96 L97 F100 ? 0042981 ic50=10nM remove_due_to_license_issue Q07820 31736296 401 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6udy A 1.7 BS01 Q54 A 1 F228 V249 M250 V253 R263 T266 L267 F270 F58 V79 M80 V83 R93 T96 L97 F100 ? 0042981 ic50=27nM remove_due_to_license_issue IC50=27nM Q07820 31736296 401 EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHV 6ueg A 2.0 BS01 Q5G A 1 H118 A138 H156 Q157 H117 A137 H155 Q156 H121 D122 G139 H120 D121 G138 2.3.1.129 0005737,0008610,0008780,0009245,0016020,0016740,0016746 Kd=19.5uM remove_due_to_license_issue A6V1E4 31664082 301 SLIDPRAIIDPSARLAADVQVGPWSIVGAEVEIGEGTVIGPHVVLKGPTKIGKHNRIYQFSSVGEDTPDLKYKGEPTRLVIGDHNVIREGVTIHRGTVQDRAETTIGDHNLIMAYAHIGHDSVIGNHCILVNNTALAGHVHVDDWAILSGYTLVHQYCRIGAHSFSGMGSAIGKDVPAYVTVFGNPAEARSMNFEGMRRRGFSSEAIHALRRAYKVVYRQGHTVEEALAELAESAAQFPEVAVFRDSIQSATRGITR 6ueg A 2.0 BS02 Q5G A 2 V132 N133 V131 N132 H121 D122 G139 H120 D121 G138 2.3.1.129 0005737,0008610,0008780,0009245,0016020,0016740,0016746 Kd=19.5uM remove_due_to_license_issue A6V1E4 31664082 302 SLIDPRAIIDPSARLAADVQVGPWSIVGAEVEIGEGTVIGPHVVLKGPTKIGKHNRIYQFSSVGEDTPDLKYKGEPTRLVIGDHNVIREGVTIHRGTVQDRAETTIGDHNLIMAYAHIGHDSVIGNHCILVNNTALAGHVHVDDWAILSGYTLVHQYCRIGAHSFSGMGSAIGKDVPAYVTVFGNPAEARSMNFEGMRRRGFSSEAIHALRRAYKVVYRQGHTVEEALAELAESAAQFPEVAVFRDSIQSATRGITR 6ueg C 2.0 BS01 Q5G A 1 V132 N133 M169 V130 N131 M167 H121 D122 G139 H119 D120 G137 2.3.1.129 0005737,0008610,0008780,0009245,0016020,0016740,0016746 Kd=19.5uM remove_due_to_license_issue A6V1E4 31664082 301 LIDPRAIIDPSARLAADVQVGPWSIVGAEVEIGEGTVIGPHVVLKGPTKIGKHNRIYQFSSVGEDTPDLKYKGEPTRLVIGDHNVIREGVTIHRGTVQDRAETTIGDHNLIMAYAHIGHDSVIGNHCILVNNTALAGHVHVDDWAILSGYTLVHQYCRIGAHSFSGMGSAIGKDVPAYVTVFGNPAEARSMNFEGMRRRGFSSEAIHALRRAYKVVYRQGHTVEEALAELAESAAQFPEVAVFRDSIQSATRGITR 6ueg C 2.0 BS02 Q5G C 1 D70 H118 A138 H156 Q157 D68 H116 A136 H154 Q155 H121 D122 G139 H119 D120 G137 2.3.1.129 0005737,0008610,0008780,0009245,0016020,0016740,0016746 Kd=19.5uM remove_due_to_license_issue A6V1E4 31664082 301 LIDPRAIIDPSARLAADVQVGPWSIVGAEVEIGEGTVIGPHVVLKGPTKIGKHNRIYQFSSVGEDTPDLKYKGEPTRLVIGDHNVIREGVTIHRGTVQDRAETTIGDHNLIMAYAHIGHDSVIGNHCILVNNTALAGHVHVDDWAILSGYTLVHQYCRIGAHSFSGMGSAIGKDVPAYVTVFGNPAEARSMNFEGMRRRGFSSEAIHALRRAYKVVYRQGHTVEEALAELAESAAQFPEVAVFRDSIQSATRGITR 6uf0 A 1.96 BS01 Q5V A 1 Y334 G364 R415 I461 S508 G509 Y525 S555 F577 S602 G603 Y11 G41 R92 I138 S185 G186 Y202 S232 F254 S279 G280 ? ic50=73nM remove_due_to_license_issue Q14145 31682434 701 VGRLIYTAGGYFRQSLSYLEAYNPSDGTWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVATATWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVT 6ufn A 2.7 BS01 Q6M A 1 A24 D94 P134 H136 H137 F146 D174 H176 W205 E274 G305 Y307 A24 D94 P134 H136 H137 F146 D174 H176 W205 E274 G305 Y307 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSETNIVWPEPLKRMPASVRTVVVPPPGVELTLPKNCQHSDISESTAKEVQRIRDKHFHDLTDQNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCLREGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETARLMRVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGPRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6ufo A 2.68 BS01 Q6P A 1 D94 P134 H136 H137 F146 D174 H176 W205 E274 E304 G305 Y307 D94 P134 H136 H137 F146 D174 H176 W205 E274 E304 G305 Y307 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSETDIVWPEPLKRMPASVRTVVVPPPGVELTLPKNCQHSDISESTAKEVQRIRDKHFHDLTDQNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEPERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCLRGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETARLMRVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGPLRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6ugn A 1.406 BS02 Q77 A 1 H94 H96 H119 F131 L198 T199 T200 H91 H93 H116 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=763.5nM remove_due_to_license_issue Ki=764nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugn A 1.406 BS03 Q77 A 2 Y128 K133 Y124 K129 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=763.5nM remove_due_to_license_issue Ki=764nM P00918 31794211 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugo A 1.457 BS02 Q77 A 1 H94 H96 H119 V121 L198 T199 T200 H91 H93 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=764nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugo A 1.457 BS03 Q77 A 2 Q67 Q92 Q64 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=764nM P00918 31794211 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugo A 1.457 BS04 Q77 A 3 G6 Y7 G8 F231 G3 Y4 G5 F227 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=764nM P00918 31794211 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugp A 1.306 BS02 Q7A A 1 H94 H96 H119 V121 L198 T199 T200 H91 H93 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=685.5nM remove_due_to_license_issue Ki=686nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugp A 1.306 BS03 Q7A A 2 K111 K112 K113 K108 K109 K110 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=685.5nM remove_due_to_license_issue Ki=686nM P00918 31794211 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugq A 1.305 BS02 Q7A A 1 H94 H96 H119 V121 L198 T199 T200 H91 H93 H116 V118 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=686nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugq A 1.305 BS03 Q7A A 2 Q67 Q92 Q64 Q89 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=686nM P00918 31794211 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugr A 1.307 BS02 Q71 A 1 H94 H96 H119 V121 F131 L198 T199 T200 H91 H93 H116 V118 F127 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=533.6nM remove_due_to_license_issue Ki=534nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6ugz A 1.306 BS02 Q71 A 1 H94 H96 H119 V121 V143 L198 T199 T200 H91 H93 H116 V118 V139 L194 T195 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 remove_due_to_license_issue Ki=534nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHSFQVTFDDSQDKAVLKGGPLDGTYRLLQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDVGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTEGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLAECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6uh0 A 1.306 BS02 PX7 A 1 H94 H96 H119 V121 V143 L198 T199 T200 W209 H91 H93 H116 V118 V139 L194 T195 T196 W205 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 Ki=853.1nM remove_due_to_license_issue Ki=853nM P00918 31794211 302 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 6uhu A 2.8 BS01 Q7V A 1 A24 I27 D94 P134 H136 H137 G145 F146 D174 H176 W205 E274 G305 Y307 A24 I27 D94 P134 H136 H137 G145 F146 D174 H176 W205 E274 G305 Y307 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAIVWPEPLKRMPASVRTVVVPPPGVELTLPKNCQHSDISESTAKEVQRIRDKHFHDLTDQNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCLREGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETTRLMRVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6uhv A 2.53 BS01 XS6 A 1 D94 H136 H137 F146 D174 H176 W205 E274 Y307 D94 H136 H137 F146 D174 H176 W205 E274 Y307 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFHDLTDQNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCLREGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETARVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGPLRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6uii A 2.65 BS01 SS9 A 1 A24 D94 H136 H137 F146 D174 H176 W205 E274 G305 A24 D94 H136 H137 F146 D174 H176 W205 E274 G305 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGFNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFDLTDNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETDKCVNRLTLCLGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETLMRVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGLRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6uil A 2.85 BS01 FKS A 1 D94 P134 H136 H137 F146 D174 H176 W205 E274 E304 G305 Y307 D93 P133 H135 H136 F145 D173 H175 W204 E273 E303 G304 Y306 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 ASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFDQNILRSLGNIISVLDRMMVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETRLMRVWGHMTCLIQGLARGRMLTLLQDKDLLELTVSALSGASISPLGPAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6uim A 2.75 BS01 Q7Y A 1 D94 H137 F146 D174 H176 W205 E274 Y307 D94 H137 F146 D174 H176 W205 E274 Y307 3.5.1.48,3.5.1.62 0005634,0005737,0008270,0016236,0016787,0019213,0033558,0035825,0036269,0040029,0046872,0047609,0047611,0090043,0106047,0106048 remove_due_to_license_issue F1QCV2 31746596 701 AASGSALIFDEEMSRYKLLWTDPACEIEVPERLTVSYEALRTHGLAQRCKAVPVRQATEQEILLAHSEEYLEAVKQTPGMNVEELMAFSKKYNDVYFHQNIYHCAKLAAGATLQLVDSVMKREVRNGMALVRPPGHHSQRSAANGFCVFNNVAFAALYAKKNYNLNRILIVDWDVHHGQGIQYCFEEDPSVLYFSWHRYEHQSFWPNLPESDYSSVGKGKGSGFNINLPWNKVGMTNSDYLAAFFHVLLPVAYEFDPELVIVSAGFDSAIGDPEGEMCALPEIFAHLTHLLMPLAAGKMCVVLEGGYNLTSLGQSVCQTVHSLLGDPTPRISGLGTACDSALESIQNVRNVQSSYWSSFKHLAQSVRTVVVPPPGVELTLPKNCQHSISESTAKEVQRIRDKHFTDQNILRSLGNIISVLDRMMRSDEVCNGCVVVSDLSVSVQCALQHALTEPAERVLVVYVGDGELPVKTNDGKVFLVQICTKETEDKCVNRLTLCLREGESLTAGFMQALLGLILPVAYEFNPALVLGIVEETTRLMRVWGHMTCLIQGLARGRMLTLLQGYDKDLLELTVSALSGASISPLGPRAPKPEDVEMMEKQRQRLQERWGLLRCTVSESW 6ul8 A 2.68 BS01 Q9J A 1 V32 A45 K47 L79 T95 Y97 M98 L153 V28 A41 K43 L72 T88 Y90 M91 L146 D146 Q150 N151 D164 D139 Q143 N144 D157 2.7.10.2,2.7.11.1 0004672,0005524,0006468 remove_due_to_license_issue IC50=50nM O43353 31749904 401 AISSALPTIPYHKLADLRYLSRGASGTVSSARHADWRVQVAVKHLHILLDSERKDVLREAEILHKARFSYILPILGICNEPEFLGIVTEYMPNGSLNELLHRKTEYPDVAWPLRFRILHEIALGVNYLHNMTPPLLHHDLKTQNILLDNEFHVKIADFGLCKWGTIIYMPPENYESIKHDIYSYAVITWEVLSRKQPFEDVTNPLQIMYSVSQGHRPVINEESLPYDIPHRARMISLIESGWAQNPDERPSFLKCLIELEPVLRTFEEITFLEAVIQLK 6un1 A 2.26 BS01 TJ7 A 1 S294 V333 S349 N351 Y409 S485 G486 T487 R489 F533 S245 V284 S300 N302 Y360 S436 G437 T438 R440 F474 3.4.16.4 0000917,0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0043093,0051301,0071555 remove_due_to_license_issue G3XD46 31685462 601 ARSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKNAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLP 6un3 A 1.9 BS01 XT8 A 1 S294 V333 S349 N351 Y409 S485 G486 T487 R489 F533 S245 V284 S300 N302 Y360 S436 G437 T438 R440 F474 3.4.16.4 0000917,0004180,0005886,0006508,0008360,0008658,0008955,0009002,0009252,0043093,0051301,0071555 remove_due_to_license_issue G3XD46 31685462 602 ARSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKNAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLP 6upj A 2.34 BS01 NIU A 1 D25 G27 A28 I50 D25 G27 A28 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=480nM remove_due_to_license_issue P04584 7783120 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTLEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 6upj B 2.34 BS01 NIU A 1 D25 G49 D25 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 remove_due_to_license_issue P04584 7783120 100 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTLEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 6uvp A 1.56 BS01 QJJ A 1 S10 G11 Q12 G13 D32 Y71 I118 D228 G230 T232 S16 G17 Q18 G19 D38 Y77 I124 D234 G236 T238 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D234 T237 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=>100000nM P56817 31786008 401 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6uvp A 1.56 BS03 QJJ B 2 S164 E165 S170 E171 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D234 T237 3.4.23.46 0004190,0006508,0016020 remove_due_to_license_issue IC50=>100000nM P56817 31786008 402 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6uvv A 1.63 BS01 QJV A 1 G13 L30 D32 Y71 D228 G230 G21 L38 D40 Y79 D236 G238 D32 S35 N37 A39 Y71 D228 T231 D40 S43 N45 A47 Y79 D236 T239 3.4.23.46 0004190,0006508,0016020 ic50=6.64uM remove_due_to_license_issue IC50=6640nM P56817 31786008 401 PGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6uvy A 1.71 BS01 QJP A 1 G11 Q12 G13 L30 D32 Y71 D228 G230 T231 G15 Q16 G17 L34 D36 Y75 D232 G234 T235 D32 S35 N37 A39 Y71 D228 T231 D36 S39 N41 A43 Y75 D232 T235 3.4.23.46 0004190,0006508,0016020 ic50=0.99uM remove_due_to_license_issue IC50=990nM P56817 31786008 401 GSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6uwp A 1.29 BS01 QKA A 1 G11 Q12 G13 L30 D32 S35 V69 Y71 D228 G230 T232 G19 Q20 G21 L38 D40 S43 V77 Y79 D236 G238 T240 D32 S35 N37 A39 Y71 D228 T231 D40 S43 N45 A47 Y79 D236 T239 3.4.23.46 0004190,0006508,0016020 ic50=0.028uM remove_due_to_license_issue IC50=18nM P56817 31786008 401 PGRRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6uwv A 1.47 BS01 QK7 A 1 Q12 G13 D32 S35 V69 Y71 R128 D228 G230 T231 Q18 G19 D38 S41 V75 Y77 R134 D234 G236 T237 D32 S35 N37 A39 Y71 D228 T231 D38 S41 N43 A45 Y77 D234 T237 3.4.23.46 0004190,0006508,0016020 ic50=0.01uM remove_due_to_license_issue IC50=10.0nM P56817 31786008 401 RRGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGAGFPLNQSEVLASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVEDVATSQDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYN 6v5l A -1.00 BS03 QPD A 1 K5 L6 V7 D54 L56 Q70 Y71 K5 L6 V7 D54 L56 Q70 Y71 3.6.5.2 0003924,0005525,0007165,0016020 remove_due_to_license_issue P01116 30903639 203 MTEYKLVVVGAGGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEK 7abp A 1.67 BS01 FCA A 1 K10 E14 W16 D90 R151 M204 N232 K9 E13 W15 D89 R150 M203 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.35uM remove_due_to_license_issue P02924 2069949 307 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMLAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 7abp A 1.67 BS02 FCB A 1 K10 E14 W16 D90 R151 N232 K9 E13 W15 D89 R150 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.35uM remove_due_to_license_issue P02924 2069949 308 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMLAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 7cpa A 2.0 BS02 FVF A 1 H69 R71 E72 R127 N144 R145 H196 S197 Y198 I243 Y248 A250 E270 H69 R71 E72 R127 N144 R145 H196 S197 Y198 I243 Y248 A250 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=11fM remove_due_to_license_issue P00730 1868092 309 ARSTNTFNYATYHTLDEIYDFMDLLVAQHPELVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 7gat A -1.00 BS01 dna C 0 P21 N34 F39 H43 R47 R61 N62 S63 P21 N34 F39 H43 R47 R61 N62 S63 ? 0003700,0006355,0006357,0008270,0043565 remove_due_to_license_issue P17429 9533884 114 ~ 126 MKNGEQNGPTTCTNCFTQTTPVWRRNPEGQPLCNACGLFLKLHGVVRPLSLKTDVIKKRNRNSANS 7gch F 1.8 BS02 LPF G 1 H57 I99 H42 I84 H57 D102 H42 D87 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 2271520 246 IVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGVTTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKYNSLTINNDITLLKLSTAASFSQTVSAVCLPSASDDFAAGTTCVTTGWGLTRY 7gch G 1.8 BS01 LPF G 1 S190 C191 M192 G193 D194 S195 S214 W215 G216 S40 C41 M42 G43 D44 S45 S64 W65 G66 G193 S195 G196 G43 S45 G46 3.4.21.1 0004252,0006508 remove_due_to_license_issue P00766 2271520 246 TPDRLQQASLPLLSNTNCKKYWGTKIKDAMICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQTLAAN 7gpb A 2.9 BS02 AMP A 1 Q71 Q72 Y75 R309 R310 Q62 Q63 Y66 R295 R296 H377 K568 R569 K574 T676 K680 H363 K554 R555 K560 T662 K666 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1900534 920 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 7gpb A 2.9 BS03 AMP B 1 D42 N44 V45 D33 N35 V36 H377 K568 R569 K574 T676 K680 H363 K554 R555 K560 T662 K666 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1900534 920 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 7gpb B 2.9 BS02 AMP B 1 Q71 Y75 R309 R310 Q62 Y66 R295 R296 H377 K568 R569 K574 T676 K680 H363 K554 R555 K560 T662 K666 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 remove_due_to_license_issue P00489 1900534 920 RKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAP 7prc L 2.65 BS05 CET L 1 L189 F216 V220 Y222 S223 I224 G225 I229 L189 F216 V220 Y222 S223 I224 G225 I229 ? 0009772,0015979,0016020,0019684,0030077,0042314,0042717,0045156,0046872 remove_due_to_license_issue P06009 10024457 502 ALLSFERKYRVRGGTLIGGDLFDFWVGPYFVGFFGVSAIFFIFLGVSLIGYAASQGPTWDPFAISINPPDLKYGLGAAPLLEGGFWQAITVCALGAFISWMLREVEISRKLGIGWHVPLAFCVPIFMFCVLQVFRPLLLGSWGHAFPYGILSHLDWVNNFGYQYLNWHYNPGHMSSVSFLFVNAMALGLHGGLILSVANPGDGDKVKTAEHENQYFRDVVGYSIGALSIHRLGLFLASNIFLTGAFGTIASGPFWTRGWPEWWGWWLDIPFWS 7std A 1.8 BS02 CRP A 1 W26 Y50 F53 V75 L76 L106 V108 N131 I151 G165 W18 Y42 F45 V67 L68 L98 V100 N123 I143 G157 Y30 D31 Y50 H85 H110 Y22 D23 Y42 H77 H102 4.2.1.94 0005575,0005768,0006582,0016829,0030411,0042438,0046872 Ki=19pM remove_due_to_license_issue Ki=30nM P56221 10382670 600 GEITFSDYLGLMTCVYEWADSYDSKDWDRLRKVIAPTLRIDYRSFLDKLWEAMPAEEFVGMVSSKQVLGDPTLRTQHFIGGTRWEKVSEDEVIGYHQLRVPHQRYKDTTMKEVTMKGHAHSANLHWYKKIDGVWKFAGLKPDIRWGEFDFDRIFEDGRETFGDK 7upj A 2.0 BS01 INU A 1 L23 D25 G27 A28 D29 G48 G49 I50 L23 D25 G27 A28 D29 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.2nM remove_due_to_license_issue P03367 9089336 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 7upj B 2.0 BS01 INU A 1 R8 D25 G27 G49 R8 D25 G27 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P03367 9089336 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 830c A 1.6 BS04 RS1 A 1 L185 A186 H222 E223 H226 H232 L239 F241 I243 Y244 L82 A83 H119 E120 H123 H129 L136 F138 I140 Y141 H222 E223 H226 H232 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=0.52nM remove_due_to_license_issue IC50=0.010000nM, Ki=0.52nM P45452 10074939 1 YNVFPRTLKWSKMNLTYRIVNYTPDMTHSEVEKAFKKAFKVWSDVTPLNFTRLHDGIADIMISFGIKEHGDFYPFDGPSGLLAHAFPPGPNYGGDAHFDDDETWTSSSKGYNLFLVAAHEFGHSLGLDHSKDPGALMFPIYTYTFMLPDDDVQGIQSLYGPGDE 8a3h A 0.97 BS01 IDC A 1 H35 Y66 H101 L103 E139 Y202 E228 A234 T235 G236 W262 K267 E269 H32 Y63 H98 L100 E136 Y199 E225 A231 T232 G233 W259 K264 E266 3.2.1.4 0000272,0004553,0005975 Ki=88uM remove_due_to_license_issue O85465 500 SVVEEHGQLSISNGELVNERGEQVQLKGMSSHGLQWYGQFVNYESMKWLRDDWGINVFRAAMYTSSGGYIDDPSVKEKVKEAVEAAIDLDIYVIIDWHILSDNDPNIYKEEAKDFFDEMSELYGDYPNVIYEIANEPNGSDVTWGNQIKPYAEEVIPIIRNNDPNNIIIVGTGTWSQDVHHAADNQLADPNVMYAFHFYAGTHGQNLRDQVDYALDQGAAIFVSEWGTSAATGDGGVFLDEAQVWIDFMDERNLSWANWSLTHKDESSAALMPGANPTGGWTEAELSPSGTFVREKIRES 8abp A 1.49 BS01 GLA A 1 K10 E14 W16 D89 D90 L108 R151 M204 N232 K9 E13 W15 D88 D89 L107 R150 M203 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.01uM remove_due_to_license_issue P02924 2069949 307 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMLAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLPSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 8cpa A 2.0 BS02 AGF A 1 H69 E72 R127 N144 R145 H196 S197 Y198 I243 Y248 A250 E270 H69 E72 R127 N144 R145 H196 S197 Y198 I243 Y248 A250 E270 H69 E72 R127 H196 E270 H69 E72 R127 H196 E270 3.4.17.1 0004181,0006508,0008270 Ki=710pM remove_due_to_license_issue P00730 1868092 309 ARSTNTFNYATYHTLDEIYDFMDLLVAQHPELVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTENYGQNPSFTAILDSMDIFLEIVTNPNGFAFTHSENRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKNHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVAALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTVNN 8gpb A 2.2 BS02 AMP A 1 Q72 Y75 R309 R310 Q62 Y65 R299 R300 H377 K568 R569 K574 T676 K680 H367 K558 R559 K564 T666 K670 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Kd=250uM remove_due_to_license_issue P00489 1900534 930 KQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 8gpb A 2.2 BS03 AMP A 2 N282 F285 P611 G612 Y613 N272 F275 P601 G602 Y603 H377 K568 R569 K574 T676 K680 H367 K558 R559 K564 T666 K670 2.4.1.1 0000166,0004645,0005737,0005975,0005977,0005980,0008184,0016757,0030170,0031220,0098723 Kd=250uM remove_due_to_license_issue P00489 1900534 940 KQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPKRIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIRYEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNTMRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRDPVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHLQIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQNKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPNSLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRLRVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDRLDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRMVIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP 966c A 1.9 BS06 RS2 A 1 N180 L181 H218 E219 H222 H228 L235 Y237 S239 T241 N73 L74 H111 E112 H115 H121 L128 Y130 S132 T134 H218 E219 H222 H228 H111 E112 H115 H121 3.4.24.7 0004222,0006508,0008237,0008270,0031012 Ki=23nM remove_due_to_license_issue Ki=23nM P03956 10074939 1 RWEQTHLTYRIENYTPDLPRADVDHAIEKAFQLWSNVTPLTFTKVSEGQADIMISFVRGDHRDNSPFDGPGGNLAHAFQPGPGIGGDAHFDEDERWTNNFREYNLHRVAAHELGHSLGLSHSTDIGALMYPSYTFSGDVQLAQDDIDGIQAIYGRSQ 9abp A 1.97 BS01 GLA A 1 K10 E14 W16 D89 D90 R151 M204 N205 N232 K9 E13 W15 D88 D89 R150 M203 N204 N231 ? 0015407,0016020,0030246,0030288,0042597,0042882,0048029,0055052 Kd=0.01uM remove_due_to_license_issue P02924 2204627 307 NLKLGFLVKQPEEPWFQTEWKFADKAGKDLGFEVIKIAVPDGEKTLNAIDSLAASGAKGFVICTPDPKLGSAIVAKARGYDMKVIAVDDQFVNAKGKPMDTVPLVMMAATKIGERQGQELYKEMQKRGWDVKESAVMAITANELDTARRRTTGSMDALKAAGFPEKQIYQVPTKSNDIPGAFDAANSMLVQHPEVKHWLIVGMNDSTVLGGVRATEGQGFKAADIIGIGINGVDAVSELSKAQATGFYGSLLGSPDVHGYKSSEMLYNWVAKDVEPPKFTEVTDVVLITRDNFKEELEKKGLGGK 9hvp A 2.8 BS01 0E9 A 1 L23 D25 G27 A28 D29 I47 G48 G49 L23 D25 G27 A28 D29 I47 G48 G49 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 2200122 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 9hvp B 2.8 BS01 0E9 A 1 D25 G27 A28 D29 G48 P81 I84 D25 G27 A28 D29 G48 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 remove_due_to_license_issue P12497 2200122 100 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 9icd A 2.5 BS01 NAP A 1 I37 H339 G340 A342 Y345 N352 Y391 R395 I35 H337 G338 A340 Y343 N350 Y389 R393 Y160 K230 D283 D307 D311 Y158 K228 D281 D305 D309 1.1.1.42 0000287,0004450,0005515,0005737,0005829,0006097,0006099,0006979,0016491,0016616,0022900,0046872,0051287,0097216 Kd=125uM remove_due_to_license_issue P08200 1888729 417 SKVVVPAQGKKITLQNGKLNVPENPIIPYIEGDGIGVDVTPAMLKVVDAAVEKAYKGERKISWMEIYTGEKSTQVYGQDVWLPAETLDLIREYRVAIKGPLTTPVGGGIRSLNVALRQELDLYICLRPVRYYQGTPSPVKHPELTDMVIFRENSEDIYAGIEWKADSADAEKVIKFLREEMGVKKIRFPEHCGIGIKPCSEEGTKRLVRAAIEYAIANDRDSVTLVHKGNIMKFTEGAFKDWGYQLAREEFGGELIDGGPWLKVKNPNTGKEIVIKDVIADAFLQQILLRPAEYDVIACMNLNGDYISDALAAQVGGIGIAPGANIGDECALFEATHGTAPKYAGQDKVNPGSIILSAEMMLRHMGWTEAADLIVKGMEGAINAKTVTYDFERLMDGAKLLKCSEFGDAIIENM